Patent ID: 7067501

Claim:
A compound represented by the general formula I wherein Y is N; X represent O or S; m is 1; p is 0, 1, 2, 3 or 4; q is 0, 1 or 2; s is 0, 1, 2 or 3; r is 0, 1 or 2; Q represents C, P—OR 5 , or S═O, wherein R 5 hydrogen or C 1-6 -alkyl; A is OR 6 , wherein R 6 represent hydrogen, C 1-6 -alkyl, aryl or aryl-C 1-6 -alkyl, wherein aryl may be substituted with halogen, CF 3 , OCF 3 , CN, NO 2 or C 1-6 alkyl; AR represents phenyl; each R 4 individually represents C 1-6 -alkyl, C 3-8 -cycloalkyl or C 3-8 -cycloalkyl-C 1-6 -alkyl; each R 1 is independently selected from the group consisting of C 1-6 -alkyl, or two R 1 attached to the same carbon atom may form a 3–6-membered spiro-attached cycloalkyl; each R 2 is independently selected from the groups consisting of halogen, cyano, nitro, C 1-6 -alk(en/yn)yl, C 1-6 -alk(en/yn)yloxy, C 1-6 -alk(en/yn)ylsulfanyl, hydroxy, hydroxy-C 1-6 -alk(en/yn)yl, halo-C 1-6 -alk(en/yn)yl, halo-C 1-6 -alk(en/yn)yloxy, C 3-8 -cycloalk(en)yl, C 3-8 -cycloalk(en)yl-C 1-6 -alk(en/yn)yl, acyl, C 1-6 -alk(en/yn)yloxycarbonyl, C 1-6 -alk(en/yn)ylsulfonyl or —NR 9 R 10 wherein R 9 and R 10 independently represent hydrogen, C 1-6 -alk(en/yn)yl, C 3-8 -cycloalk(en)yl, C 3-8 -cycloalk(en)yl-C 1-6 alk(en/yn)yl or aryl, or R 9 and R 10 together with the nitrogen atom to which they are attached form a 3–7-membered ring which optionally contains one further heteroatom selected from the group consisting of nitrogen and oxygen; each R 3 which is substituted on AR, is independently selected from the group consisting of halogen, cyano, nitro, C 1-6 -alk(en/yn)yl, C 1-6 -alk(en/yn)yloxy, C 1-6 -alk(en/yn)ylsulfanyl, hydroxy, hydroxy-C 1-6 -alk(en/yn)yl, halo-C 1-6 -alk(en/yn)yl, halo-C 1-6 -alk(en/yn)yloxy, C 3-8 -cycloalk(en)yl, C 3-8 -cycloalk(en)yl-C 1-6 -alk(en/yn)yl, C 1-6 -alk(en/yn)ylsulfonyl, aryl, aryl-C 1-6 -alk(en/yn)yloxy, aryl-C 1-6 -alk(en/yn)yl, C 1-6 -alk(en/yn)yloxycarbonyl, acyl, —NHCO—C 1-6 -alk(en/yn)yl, —CONR 11 R 12 wherein R 11 and R 12 independently represent hydrogen, C 1-6 -alk(en/yn)yl, C 3-8 -cycloalk(en)yl, C 3-8 -cycloalk(en)yl-C 1-6 -alk(en/yn)yl or aryl, or R 11 and R 12 together with the nitrogen to which they are attached form a 3–7-membered ring which optionally contains one further heteroatom selected from the group consisting of nitrogen and oxygen; or NR 13 R 14 wherein R 13 and R 14 independently represent hydrogen, C 1-6 -alk(en/yn)yl, C 3-8 -cycloalk(en)yl, C 3-8 -cycloalk(en)yl-C 1-6 -alk(en/yn)yl or aryl; or R 13 and R 14 together with the nitrogen to which they are attached form a 3–7-membered ring which optionally contains one further heteroatom selected from the group consisting of nitrogen and oxygen; or an acid addition salt thereof.