Patent ID: 7442696

Claim:
A compound selected from the group consisting of: 5-Chloro-6-(3-cyanophenyl)-1,4-dihydro-4,4-dimethyl-2H-3,1-benzoxazin-2-one (Compound 101); 5-Chloro-1,4-dihydro-4,4-dimethyl-6-[3-(trifluoromethyl)phenyl]-2H-3,1-benzoxazin-2-one (Compound 102); 6-(3-Acetylphenyl)-5-chloro-1,4-dihydro-4,4-dimethyl-2H-3,1-benzoxazin-2-one (Compound 103); 5-Chloro-1,4-dihydro-4,4-dimethyl-6-[3-(trifluoromethyl)phenyl]-2H-3,1-benzoxazin-2-thione (Compound 104); 5-Chloro-6-(3-chlorophenyl)-1,4-dihydro-4,4-dimethyl-2H-3,1-benzoxazin-2-one (Compound 105); 5-Chloro-6-(3-cyanophenyl)-1,4-dihydro-4,4-dimethyl-2H-3,1-benzoxazin-2-thione (Compound 106); 6-(3-Carboxymethylphenyl)-5-chloro-1,4-dihydro-4,4-dimethyl-2H-3,1-benzoxazin-2-one (Compound 107); 5-Chloro-6-(3-cyanophenyl)-1,4-dihydro-1,4,4-trimethyl-2H-3,1-benzoxazin-2-one (Compound 108); 5-Chloro-6-(3-cyano-2-methoxyphenyl)-1,4-dihydro-4,4-dimethyl-2H-3,1-benzoxazin-2-one (Compound 109); (±)-5-Chloro-1,4-dihydro-4-methyl-6-[3-(trifluoromethyl)phenyl]-2H-3,1-benzoxazin-2-one (Compound 110); (±)-5-Chloro-1,4-dihydro-4-methyl-6-[3-(trifluoromethyl)phenyl]-2H-3,1-benzoxazin-2-thione (Compound 111); (±)-5-Chloro-6-(3-cyanophenyl)-4-ethyl-1,4-dihydro-2H-3,1-benzoxazin-2-one (Compound 112); (±)-5-Chloro-6-(3-cyanophenyl)-4-ethyl-1,4-dihydro-2H-3,1-benzoxazin-2-thione (Compound 113); (±)-5-Chloro-6-(3-cyanophenyl)-4-(4-fluorophenyl)-1,4-dihydro-2H-3,1-benzoxazin-2-one (Compound 114); (±)-5-Chloro-4-ethyl-1,4-dihydro-6-[3-(trifluoromethyl)phenyl]-2H-3,1-benzoxazin-2-one (Compound 115); (±)-5-Chloro-6-(3-cyanophenyl)-4-(4-fluorophenyl)-1,4-dihydro-2H-3,1-benzoxazin-2-thione (Compound 116); (±)-5-Chloro-4-ethyl-1,4-dihydro-6-[3-(trifluoromethyl)phenyl]-2H-3,1-benzoxazin-2-thione (Compound 117); (±)-5-Chloro-4-(4-fluorophenyl)-1,4-dihydro-6-[3-(trifluoromethyl)phenyl]-2H-3,1-benzoxazin-2-one (Compound 118); (±)-5-Chloro-6-(3-cyanophenyl)-4-cyclopentyl-1,4-dihydro-2H-3,1-benzoxazin-2-one (Compound 119); (±)-5-Chloro-6-(3-cyanophenyl)-4-cyclopentyl-1,4-dihydro-2H-3,1-benzoxazin-2-thione (Compound 120); (±)-5-Chloro-6-(3-cyanophenyl)-4-(3,4-difluorobenzyl)-1,4-dihydro-2H-3,1-benzoxazin-2-one (Compound 121); (±)-5-Chloro-6-(3-cyanophenyl)-4-(3,4-difluorobenzyl)-1,4-dihydro-2H-3,1-benzoxazin-2-thione (Compound 122); 5-Chloro-1,4-dihydro-6-(2,6-dimethoxyphenyl)-4,4-dimethyl-2H-3,1-benzoxazin-2-one (Compound 123); 7-Chloro-6-(3-cyanophenyl)-1,4-dihydro-4,4-dimethyl-2H-3,1-benzoxazin-2-one (Compound 124); 7-Chloro-6-(3-cyanophenyl)-1,4-dihydro-4,4-dimethyl-2H-3,1-benzoxazin-2-thione (Compound 125); 7-Chloro-6-(3-cyano-2-methoxyphenyl)-1,4-dihydro-4,4-dimethyl-2H-3,1-benzoxazin-2-one (Compound 126); 7-Chloro-6-(3-cyano-2-methoxyphenyl)-1,4-dihydro-4,4-dimethyl-2H-3,1-benzoxazin-2-thione (Compound 127); 6-(3,5-Dimethylisoxazol-4-yl)-1,4-dihydro-4,4,8-trimethyl-2H-3,1-benzoxazin-2-one (Compound 128); 1,4-Dihydro-6-(indol-7-yl)-4,4,8-trimethyl-2H-3,1-benzoxazin-2-one (Compound 129); and a pharmaceutically acceptable salt, ester, or amide of any of those compounds.