Patent ID: 7868172

Claim:
A compound of formula IA4 in which R 1 is A, CF 3 , OCF 3 , SA, SCN, CH 2 CN, —OCOA, Hal, or SCF 3 , R 2 is F or H, R 3 is H, R a is NHR, NR 2 , OR, NHR, NR 2 , NR(CH 2 ) n -aryl, NR(CH 2 ) n OR, COOR, OCOR, NR(CH 2 ) n NR 2 , N[(CH 2 ) n NR 2 ]CO(CH 2 ) n -aryl, N[(CH 2 ) n NHCOOR]CO-aryl, N[CH 2 (CH 2 ) n OR] 2 , NR(CH 2 ) n X(CH 2 ) n OH, O(CO)NR(CH 2 ) n OR, O(CO)(CH 2 ) n NR 2 , N[(CH 2 ) n NR 2 ]CO(CH 2 ) n -aryl, N(R)(CH 2 ) n N(R)COOR, OSO 2 A, OCH 2 (CH 2 ) n NR 2 , Hal, NCOOR, N(CH 2 ) n CONR 2 , XCONR(CH 2 ) n NR 2 , N[(CH 2 ) n XCOOR]CO(CH 2 ) n -aryl, N[(CH 2 ) n XR]CO(CH 2 ) n X-aryl, or N[(CH 2 ) n XR]SO 2 (CH 2 ) n -aryl, aryl is phenyl, naphthyl or biphenyl, each of which is un-substituted or mono-, di- or trisubstituted by Hal, A, OH, OA, NH 2 , NO 2 , CN, COOH, COOA, CONH 2 , NHCOA, NHCONH 2 , NHSO 2 A, CHO, COA, SO 2 NH 2 , SO 2 A, —CH 2 —COOH or —OCH 2 —COOH, R is H or A, in case of geminal radicals R is —(CH 2 ) 5 —, —(CH 2 ) 4 —, —(CH 2 ) 2 —X—(CH 2 ) 2 or —(CH 2 ) 2 —Z—(CH 2 ) n , A is alkyl or cycloalkyl, in which one or more H atoms are optionally replaced by Hal, Hal is F or Cl, X is O, S or NR, Z is X, CHCONH 2 , NCO, CH(CH 2 ) n COOR, NCOOR, N(CH 2 ) n OH, CHNH 2 , C(OH)R, CHNCOR, N(CH 2 ) n COOR, CH(CH 2 ) n X(CH 2 ) n -aryl, R 6 is phenyl, 2-, 3- or 4-pyridyl, pyrimidyl, furyl or thienyl, each of which is unsubstituted or mono- or polysubstituted by Hal, NO 2 , CN, OH, CF 3 , OCH(CF 3 ) 2 , OCOCH 3 or A, R 7 is H or A, m is 0, 1 or 2 and n is 0, 1, 2, 3, 4, 5, 6 or 7 or a tautomer, salt, stereoisomer thereof or mixture therefore in any ratio.