Patent ID: 8357698

Claim:
A compound of the formulae I or II: wherein X is identically or differently ═C(—R)— or ═N—, where only one X is ═N—; R is identically or differently hydrogen, halogen, (C 1 -C 6 )-alkyl, (C 1 -C 3 )-alkyloxy-(C 1 -C 3 )-alkylene, (C 1 -C 3 )-haloalkyl, hydroxy, (C 1 -C 6 )-alkylmercapto, amino, (C 1 -C 6 )-alkylamino, di-(C 2 -C 12 )-alkylamino, mono-(C 1 -C 6 )-alkylaminocarbonyl, di-(C 2 -C 8 )-alkylaminocarbonyl, COOR3, cyano, (C 1 -C 6 )-alkylsulfonyl, alkylsulfinyl, aminosulfonyl, nitro, pentafluorosulfanyl, phenyl, heterocycle, phenoxy, O-heterocycle, CO—NR6R7, O—CO—NR6R7, O—CO—(C 1 -C 6 )-alkylene-CO—O—(C 1 -C 6 )-alkyl, O—CO—(C 1 -C 6 )-alkylene-CO—OH, O—CO—(C 1 -C 6 )-alkylene-CO—NR6R7 or unsubstituted or mono- or poly-F-substituted (C 1 -C 6 )-alkyloxy; R1 is identically or differently (C 5 -C 16 )-alkyl, (C 3 -C 12 )-cycloalkyl, Y-aryl, Y-heterocycle or bicycle, where cycloalkyl, aryl, heterocycle or bicycle are optionally substituted one or more times by halogen, (C 1 -C 6 )-alkyl, (C 1 -C 3 )-alkyloxy, hydroxy, (C 1 -C 6 )-alkylmercapto, amino, (C 1 -C 6 )-alkylamino, di-(C 2 -C 12 )-alkylamino, mono-(C 1 -C 6 )-alkylaminocarbonyl, di-(C 2 -C 8 )-alkylaminocarbonyl, (C 1 -C 6 )-alkyloxycarbonyl, (C 1 -C 6 )-alkylcarbonyl, cyano, trifluoromethyl, trifluoromethyloxy, (C 1 -C 6 )-alkylsulfonyl, aminosulfonyl, and nitro; Y is (C 1 -C 3 )-alkyl, which is optionally substituted one or more times by halogen, (C 1 -C 3 )-alkyl, hydroxy or trifluoromethyl; R2 is hydrogen; or R1 and R2 together with the nitrogen atom carrying them form a monocyclic, saturated or partly unsaturated 4- to 7-membered ring system or a bicyclic saturated or partly unsaturated 8- to 14-membered ring system whose individual members of the ring systems are optionally replaced by one to three atoms or atomic groups from the series —CHR4-, —CR4R5-, —(C═R4)-, —NR4-, —C(═O)—, —O—, —S—, —SO—, —SO 2 —, with the proviso that two units from the series —O—, —S—, —SO—, —SO 2 — are not adjacent to each other; R3 is hydrogen, (C 1 -C 6 )-alkyl or benzyl; R4, R5 are identically or differently (C 1 -C 6 )-alkyl, halogen, trifluoromethyl, phenyl, heterocycle, COOR3 or (C 3 -C 12 )-cycloalkyl; and R6, R7 are identically or differently hydrogen, (C 1 -C 6 )-alkyl, phenyl, benzyl or (C 3 -C 12 )-cycloalkyl; or a tautomer thereof or a physiologically tolerated salt thereof, with the proviso that not more than one R is phenyl or heterocycle.