Patent ID: 7816324

Claim:
A tris-benzamide peptidomimetic that binds to a glucagon-like peptide 1 receptor consisting of the formula: wherein i) R1 is acetyl, R2 is benzyl, R3 and R4 are 4-fluorobenzyl, and R5 is GLP-1 (22-36) amide; ii) R1 is t-butoxycarbonyl, R2 is methyl, R3 is benzyl, R4 is 2-naphthylmethyl and R5 is GLP-1 (22-36) amide; iii) R1 is the dipeptide His-Gly, R2 is benzyl, R3 is isopropyl, R4 is 4-fluorobenzyl group and R5 is GLP-1 (22-36) amide; or iv) R1 is histidine, R2 is benzyl, R3 is isopropyl, R4 is 4-fluorobenzyl and R5 is GLP-1 (22-36) amide.