Patent ID: 6958338

Claim:
A 4-, 5-, 6- or 7-methylene substituted indolyl derivative of formula I wherein R is phenyl substituted one or more times with a substituent selected from halogen, cyano, nitro, C 1-6 -alkyl, C 2-6 -alkenyl, C 2-6 -alkynyl, C 3-8 -cycloalkyl, C 3-8 -cycloalkyl-C 1-6 -alkyl, C 1-6 -alkoxy, C 1-6 -alkylthio, hydroxy, hydroxy-C 1-6 -alkyl, trifluoromethyl, trifluoromethylsulfonyl, C 1-6 -alkylsulfonyl, amino, C 1-6 -alkylamino, di-(C 1-6 -alkyl)amino, acyl, aminocarbonyl and a methylene dioxy group; X is N; R 1 is hydrogen, C 1-6 -alkyl, C 2-6 -alkenyl, C 2-6 -alkynyl, C 3-8 -cycloalkyl, C 3-8 -cycloalkyl-C 1-6 -alkyl, aryl, aryl-C 1-6 -alkyl, acyl, thioacyl, C 1-6 -alkylsulfonyl, trifluoromethylsulfonyl or arylsulfonyl; and R 2 and R 3 are independently selected from hydrogen, halogen, cyano, nitro, C 1-6 -alkyl, C 2-6 -alkenyl, C 2-6 -alkynyl, C 3-8 -cycloalkyl, C 3-8 -cycloalkyl-C 1-6 -alkyl, C 1-6 -alkoxy, C 1-6 -alkylthio, hydroxy, hydroxy-C 1-6 -alkyl, trifluoromethyl, trifluoromethylsulfonyl, C 1-6 -alkylsulfonyl, amino, C 1-6 -alkylamino, di-(C 1-6 -alkyl)amino, acyl and aminocarbonyl; or a pharmaceutically acceptable salt thereof.