Patent ID: 8148395

Claim:
A compound of formula I wherein: X is identically or differently ═C(—R)— or ═N—, wherein one X is ═N—; Y is NR6 or O; R is identically or differently hydrogen, halogen, (C 1 -C 6 )-alkyl, (C 1 -C 3 )-haloalkyl, (C 1 -C 3 )-alkyloxy-(C 1 -C 3 )-alkylene, aryl, heterocycle, hydroxy, (C 1 -C 6 )-alkyloxy, (C 1 -C 3 )-haloalkyloxy, aryloxy, cyano, nitro, —S(O) p —(C 1 -C 6 )-alkyl, wherein p=0, 1 or 2, aminosulfonyl, pentafluorosulfanyl, amino, (C 1 -C 6 )-alkylamino, di-(C 2 -C 12 )-alkylamino, —CO—(C 1 -C 6 )-alkyl, —COOR3 , —CO—NR4R5, —O—CO—NR4R5, —O—CO—(C 1 -C 6 )-alkylene-CO—O—(C 1 -C 6 )-alkyl, —O—CO—(C 1 -C 6 )-alkylene-CO—OH or —O—CO—(C 1 -C 6 )-alkylene-CO—NR4R5; R1 is (C 8 -C 14 )-bicycle, where the bicycle moiety is optionally substituted one or more times by halogen, (C 1 -C 6 )-alkyl, (C 1 -C 3 )-alkyloxy, hydroxy, (C 1 -C 6 )-alkylmercapto, amino, (C 1 -C 6 )-alkylamino, di-(C 2 -C 12 )-alkylamino, mono-(C 1 -C 6 )-alkylaminocarbonyl, di-(C 2 -C 8 )-alkylaminocarbonyl, (C 1 -C 6 )-alkoxycarbonyl, (C 1 -C 6 )-alkylcarbonyl, cyano, nitro, trifluoromethyl, trifluoromethyloxy, pentafluorosulfanyl, (C 1 -C 6 )-alkylsulfonyl, or aminosulfonyl; R2 is hydrogen; R3 is hydrogen, (C 1 -C 6 )-alkyl, or benzyl; R4 and R5 are identically or differently hydrogen, (C 1 -C 6 )-alkyl, aryl, (C 3 -C 12 )-cycloalkyl, (C 1 -C 4 )-alkylene-aryl, or (C 1 -C 4 )-alkylene-(C 3 -C 12 )-cycloalkyl; and R6 is hydrogen, (C 1 -C 10 )-alkyl, (C 1 -C 4 )-alkylene-CN, (C 1 -C 4 )-alkylene-aryl, (C 1 -C 4 )-alkylene-heterocycle, (C 1 -C 4 )-alkylene-(C 3 -C 12 )-cycloalkyl, or (C 8 -C 14 )-bicycle, wherein the aryl, heterocycle, cycloalkyl or bicycle moiety is optionally substituted one or more times by halogen, (C 1 -C 6 )-alkyl, (C 1 -C 6 )-alkyloxy, hydroxy, (C 1 -C 6 )-alkylmercapto, amino, (C 1 -C 6 )-alkylamino, di-(C 2 -C 12 )-alkylamino, mono-(C 1 -C 6 )-alkylaminocarbonyl, di-(C 2 -C 8 )-alkylaminocarbonyl, (C 1 -C 6 )-alkoxycarbonyl, (C 1 -C 6 )-alkylcarbonyl, cyano, trifluoromethyl, trifluoromethyloxy, nitro (C 1 -C 6 )-alkylsulfonyl, or aminosulfonyl; or a tautomeric form thereof, or a physiologically tolerated salt thereof.