Patent ID: 8884023

Claim:
A compound of formula (I) wherein R 1 denotes Y, COA, COOA, COO—(CH 2 ) n —Ar— or COO—(CH 2 ) n -Cyc; R 2 , R 3 denote independently from one another Y or SO 2 Y; R 4 denotes Cl, Br, I, COOY, SO 2 Y, CN, CAr 3 , (CH 2 ) m —Ar, R 5 denotes (CH 2 ) n —Ar, (CH 2 ) n -Cyc, (CH 2 ) n -Het, (CH 2 ) n —O—Ar, (CH 2 ) n —CY(OH)—Ar, (CH 2 ) n —CO—Ar or (CH 2 ) n —NY—Ar; X denotes CH 2 , CO or CH(OH); Y denotes H or A; A denotes unbranched or branched alkyl having 1-10 C atoms, in which 1-7H atoms can be replaced independently from one another by Hal or in which one CH 2 group can be replaced by a —CH═CH— group; Cyc denotes cycloalkyl having 3-7 C atoms, in which 1-4H atoms can be replaced independently from one another by Hal or which can be substituted by Ar; Ar denotes an unsaturated or aromatic mono- or bicyclic carbocycle having 3-12 C atoms, which can be substituted by at least one substituent selected from the group of Hal, A, (CY 2 ) n —OY, (CY 2 ) n —NYY, COOY, CONYY, NHCOY, SO 2 Y, CN and phenoxy; Het denotes an unsaturated or aromatic mono-, bi- or tricyclic heterocycle having 1-12 C atoms and 1-4 N atoms, which can be substituted by at least one substituent selected from the group of Hal, A, (CY 2 ) n —OY, (CY 2 ) n —NYY, COOY, CONYY, NHCOY, SO 2 Y, SO 2 Ar, CN and thiophenyl; Hal denotes F, Cl, Br or I; m denotes 1, 2 or 3; and n denotes 0, 1, 2, 3, 4, 5 or 6; or a physiologically acceptable salt thereof.