Patent ID: 7659298

Claim:
A compound of the general formula (I) wherein: Ar represents phenyl group or a 5- or 6-membered heteroaromatic ring containing 1-3 heteroatoms, where any of these rings may optionally be mono- or polysubstituted with halogen atom, C 1-4 alkyl group, C 1-4 alkoxy group, hydroxyl group, cyano group, trihalogenomethyl group, amino group or an amino group substituted with one or two C 1-4 alkyl groups; Y stands —CH 2 - group; X stands for sulphur atom, oxygen atom, —NH-group, —N(C 1-4 alkyl)group, —CH 2 -group, —(S═O)— or —SO 2 -group; or X and Y together represent a —CH═CH— group with cis or trans geometry; A represents a moiety with a five- or six-membered aromatic ring which contains in ortho-, meta- or para-position two free valencies, and is optionally mono- or polysubstituted with halogen atom, C 1-4 alkyl group or C 1-4 alkoxy group; or with a partially or fully saturated five- or six-membered cycloalkyl ring optionally mono- or polysubstituted with halogen atom, C 1-4 alkyl group or C 1-4 alkoxy group; or with a heteroaromatic or partially or fully saturated heterocyclic ring which contains 1-3 heteroatoms and which is optionally mono- or polysubstituted with halogen atom, C 1-4 alkyl group or C 1-4 alkoxy group; R 1 represents benzyl group, C 1-4 -alkyl-, C 1-4 -hydroxyalkyl-, C 3-8 -alkoxycarbonylalkyl-, C 2-7 -alkylcarbonyl-, C 2-7 -carboxyalkyl-, aminocarbonyl-(C 1-4 )-alkyl, C 1-3 -alkylaminocarbonyl-(C 1-4 )-alkyl, amino-(C 1-4 )-alkyl, C 1-3 -alkylamino-(C 1-4 )-alkyl-, morpholino-(C 1-4 )-alkyl-, or morpholinocarbonyl-(C 1-4 )-alkyl group or a phenyl group, optionally substituted with one or more halogen atoms; R 2 represents one of the following groups which is optionally substituted with one or more halogen atom, hydroxyl group, C 1-4 alkyl group, trihalogenomethyl-group, thio-C 1-4 -alkyl group, amino group, —(C═O)—NH—C 1-4 -alkyl or cycloalkyl group: phenyl group, phenylethyl group, naphthyl group, indanyl- or indenyl group, five- or six-membered heteroaromatic or partially or fully saturated cyclic group containing 1-3 identical or different heteroatoms, a group containing a bicyclic heteroaromatic moiety or a partially or fully saturated bicyclic heteroring with 1 or 2 or 3 identical or different heteroatoms; R 3 stands for hydrogen atom or C 1-4 alkyl group; or R 3 and R 3 together with the nitrogen atom to which they are attached may represent a partly or fully saturated six-membered ring optionally substituted with a substituted phenyl or benzyl group; and R 5 stands for halogen atom, hydrogen atom, C 1-4 alkyl group, C 1-4 thioalkyl group, or C 1-4 alkoxy group; or a salt thereof.