Patent ID: 8853207

Claim:
A compound of formula (I): wherein: R 1 and R 2 independently represent hydrogen, halo, cyano, alkyl, alkenyl, alkynyl, alkoxy, cycloalkyl, cycloalkenyl, —(CH 2 ) m OR a , —(CH 2 ) m NR a R b , —NR a R b , —OR a , SR b , —CO 2 R a , —NR a CO—(CH 2 ) nm NR a R b , —CONR a R b , —CONR a -(CH 2 ) m NR a R b ,aryl, heteroaryl or heterocyclyl, wherein the alkyl, alkenyl, alkynyl, alkoxy, cycloalkyl, cycloalkenyl, OR a , SR b , aryl, heteroaryl, and heterocyclyl groups are optionally substituted by one or more substituents selected from halo, hydroxyl, alkyl, haloalkyl, alkoxy, amino, cycloalkyl, aralkyl, aryl, heteroaryl, heterocyclyl, heterocyclyl-alkyl, and —CONH-heteroaryl; X represents alkylene, alkenylene, alkyl-carbonyl, alkenyl-carbonyl, carbonyl, oxygen, —C═NOR c ; Y represents a direct bond, alkylene, alkenylene, or —NH—; ring A represents aryl, heteroaryl, or heterocyclyl; R 3 and R 4 independently represent hydroxyl, hydrogen, halo, nitro, cyano, amino, oxo, alkyl, haloalkyl, alkoxy, haloalkoxy, alkenylene, aryl, alkylaryl, NR a R b , —NH-aryl, heteroaryl, alkenylene-aryl, S(O) n -heterocyclyl, —NH-heterocyclyl, or heterocyclyl, wherein the alkyl, haloalkyl, alkoxy, haloalkoxy, alkenylene, aryl, aralkyl, —NH-aryl, heteroaryl, alkenylene-aryl, S(O) n -heterocyclyl, —NH-heterocyclyl, and heterocyclyl groups are optionally substituted by one or more substituents selected from amino, cyano, halo, haloalkyl, hydroxyl, alkyl, alkoxy, and haloalkoxy; R a and R b are independently hydrogen, alkyl, alkenyl, alkynyl, alkoxy, cycloalkyl, cycloalkenyl, aryl, heteroaryl, or heterocyclyl, or R a and R b , together with the oxygen, nitrogen or sulfur atom to which they are bonded, form a heteroaryl or heterocyclyl group; R c represents hydrogen or alkyl, m is 0, 1, 2, or 3; and n is 0, 1 or 2, Y represents a direct bond, alkylene, alkenylene, or —NH—; ring A represents aryl, heteroaryl, or heterocyclyl; R 3 and R 4 independently represent hydroxyl, hydrogen, halo, nitro, cyano, amino, oxo, alkyl, haloalkyl, alkoxy, haloalkoxy, alkenylene, aryl, alkylaryl, NR a R b , —NH-aryl, heteroaryl, alkenylene-aryl, S(O) n -heterocyclyl, —NH-heterocyclyl, or heterocyclyl, wherein the alkyl, haloalkyl, alkoxy, haloalkoxy, alkenylene, aryl, aralkyl, —NH-aryl, heteroaryl, alkenylene-aryl, S(O) n -heterocyclyl, —NH-heterocyclyl, and heterocyclyl groups are optionally substituted by one or more substituents selected from amino, cyano, halo, haloalkyl, hydroxyl, alkyl, alkoxy, and haloalkoxy; R a and R b are independently hydrogen, alkyl, alkenyl, alkynyl, alkoxy, cycloalkyl, cycloalkenyl, aryl, heteroaryl, or heterocyclyl, or R a and R b , together with the oxygen, nitrogen or sulfur atom to which they are bonded, form a heteroaryl or heterocyclyl group; R c represents hydrogen or alkyl, m is 0, 1, 2, or 3; and n is 0, 1 or 2, or hydrates, solvates, or pharmaceutically acceptable salts thereof.