Patent ID: 7205299

Claim:
An indole derivative of the general formula (I) wherein R: is a saturated, unsaturated or aromatic, substituted or unsubstituted (C 2 –C 14 )-heterocycle which contains one or more heteroatoms selected from the group N, O and S and is linked directly to the amide nitrogen, R1: is unsubstituted or substituted alkyl-aryl, R2: is (i) hydrogen, (ii) unsubstituted or substituted (C 1 –C 6 )-alkyl, R3–R6: are (i) hydrogen (ii) unsubstituted or substituted (C 1 –C 6 )-alkyl, (iii) unsubstituted or substituted (C 3 –C 7 )-cycloalkyl, (iv) amino, mono-(C 1 –C 4 )-alkylamino, di-(C 1 –C 4 )-alkylamino, (v) halogen, (vi) (C 1 –C 4 )-alkyl which is substituted by one or more fluorine atoms, (vii) cyano, straight-chain or branched cyano-(C 1 –C 6 )-alkyl, (viii) (C 1 –C 6 )-alkylcarbonyl, (ix) carboxyl, (C 1 –C 4 )-alkoxycarbonyl, carboxy-(C 1 –C 6 )-alkyl or (C 1 –C 6 )-alkoxycarbonyl-(C 1 –C 6 )-alkyl, (x) hydroxyl, (xi) —(C 1 –C 6 )-alkoxy, (xii) aryl-(C 1 –C 4 )-alkoxy, preferably benzyloxy, (xiii) (C 1 –C 6 )-alkoxycarbonylamino, (C 1 –C 6 )-alkoxycarbonylamino-(C 1 –C 6 )-alkyl, R7: is (C 1 –C 6 )-alkylcarbonyl or (C 1 –C 6 )-alkoxy-carbonyl and X, Y: are oxygen or sulfur, with the proviso that, when R is an unsubstituted or substituted 2-, 3-, 4-, 5- or 6-pyridyl group and R1–R6 have the abovementioned meaning, R7 is not an acetyl radical or a tert-butyloxycarbonyl group; the tautomers, stereoisomers, including the diastereomers and enantiomers, thereof, and also the physiologically tolerated salts thereof.