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323
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323
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267
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82
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683
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365
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62
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108 values
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float64
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float64
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2.16k
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1.83M
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90,205,160,000B
ord-89aff4b1c18042e4bbb1f88ebba96f86
S(Cl)([Cl:3])=O.[CH2:5]([O:13][C:14]1[CH:22]=[CH:21][C:17]([C:18](O)=[O:19])=[CH:16][CH:15]=1)[CH2:6][CH2:7][CH2:8][CH2:9][CH2:10][CH2:11][CH3:12]>>[CH2:5]([O:13][C:14]1[CH:22]=[CH:21][C:17]([C:18]([Cl:3])=[O:19])=[CH:16][CH:15]=1)[CH2:6][CH2:7][CH2:8][CH2:9][CH2:10][CH2:11][CH3:12]
S(=O)(Cl)Cl.C(CCCCCCC)OC1=CC=C(C(=O)O)C=C1.C(CCCCCCC)OC1=CC=C(C(=O)O)C=C1
thionyl chloride;p-octyloxybenzoic acid;( 1 )
0.0;10.0;0.0
mol;g;mol
null
null
null
null
null
null
null
null
null
null
null
null
null
null
C(CCCCCCC)OC1=CC=C(C(=O)Cl)C=C1
4-octyloxybenzoic acid chloride
null
null
null
ord-c218088b16c541088a933a7606f68c4c
[OH:1][C:2]1[CH:10]=[CH:9][C:5]([C:6]([OH:8])=[O:7])=[CH:4][CH:3]=1.[C:11](Cl)(=[O:21])[CH2:12][CH2:13][CH2:14][CH2:15][CH2:16][CH2:17][CH2:18][CH2:19][CH3:20].N1C=CC=CC=1>O>[C:11]([O:1][C:2]1[CH:10]=[CH:9][C:5]([C:6]([OH:8])=[O:7])=[CH:4][CH:3]=1)(=[O:21])[CH2:12][CH2:13][CH2:14][CH2:15][CH2:16][CH2:17][CH2:18][CH2:19...
OC1=CC=C(C(=O)O)C=C1.C(CCCCCCCCC)(=O)Cl.N1=CC=CC=C1
p-hydroxybenzoic acid;decanoic acid chloride;pyridine
0.0;15.0;7.2
mol;g;g
O
water
0.0
mol
null
null
null
null
null
null
null
null
null
24
C(CCCCCCCCC)(=O)OC1=CC=C(C(=O)O)C=C1
p-decanoyloxybenzoic acid
null
null
null
ord-d965967cbe69411f9fd760ac1f990dfb
F[C:2]1[CH:10]=[C:9]([OH:11])[CH:8]=[CH:7][C:3]=1[C:4]([OH:6])=[O:5].[OH:12][C:13]1C=CC(C(O)=O)=C[CH:14]=1.C(OC1C=CC(C(Cl)=O)=CC=1)(=O)CCCCCCCCC>>[C:13]([O:11][C:9]1[CH:8]=[CH:7][C:3]([C:4]([OH:6])=[O:5])=[CH:2][CH:10]=1)(=[O:12])[CH3:14]
OC1=CC=C(C(=O)O)C=C1.FC1=C(C(=O)O)C=CC(=C1)O.C(CCCCCCCCC)(=O)OC1=CC=C(C(=O)Cl)C=C1.OC1=CC=C(C(=O)O)C=C1
p-hydroxybenzoic acid;2-fluoro-4-hydroxybenzoic acid;( 2 );p-hydroxybenzoic acid
0.0;0.0;0.0;0.0
mol;mol;mol;mol
null
null
null
null
null
null
null
null
null
null
null
null
null
null
C(C)(=O)OC1=CC=C(C(=O)O)C=C1
p-Acetoxybenzoic acid
null
null
null
ord-e8642ae0ecb248809067cd131fde0eed
[NH2:1][C:2]1[CH:17]=[CH:16][C:5]([C:6]([NH:8][C:9]2[CH:14]=[CH:13][C:12]([NH2:15])=[CH:11][CH:10]=2)=[O:7])=[CH:4][CH:3]=1.[C:18]1([N:24]=[C:25]=[S:26])[CH:23]=[CH:22][CH:21]=[CH:20][CH:19]=1>CC(C)=O>[C:18]1([NH:24][C:25]([NH:1][C:2]2[CH:17]=[CH:16][C:5]([C:6]([NH:8][C:9]3[CH:14]=[CH:13][C:12]([NH:15][C:25](=[S:26])[N...
NC1=CC=C(C(=O)NC2=CC=C(C=C2)N)C=C1.C1(=CC=CC=C1)N=C=S
4,4'-Diaminobenzanilide;phenylisothiocyanate
0.658;0.676
g;g
CC(=O)C
acetone
20.0
mL
null
null
null
null
null
null
null
null
55.0
0.1667
C1(=CC=CC=C1)NC(=S)NC1=CC=C(C(=O)NC2=CC=C(C=C2)NC(NC2=CC=CC=C2)=S)C=C1
colorless crystal
0.9
g
72.3
ord-83e2d9b7b08846c09e3e4e23f2dc9784
[NH2:1][C:2]1[CH:17]=[CH:16][C:5]([C:6]([NH:8][C:9]2[CH:14]=[CH:13][C:12]([NH2:15])=[CH:11][CH:10]=2)=[O:7])=[CH:4][CH:3]=1.[CH2:18]([N:25]=[C:26]=[S:27])[C:19]1[CH:24]=[CH:23][CH:22]=[CH:21][CH:20]=1>CC(C)=O>[CH2:18]([NH:25][C:26]([NH:1][C:2]1[CH:17]=[CH:16][C:5]([C:6]([NH:8][C:9]2[CH:14]=[CH:13][C:12]([NH:15][C:26](=...
NC1=CC=C(C(=O)NC2=CC=C(C=C2)N)C=C1.C(C1=CC=CC=C1)N=C=S
4,4'-Diaminobenzanilide;benzylisothiocyanate
0.568;0.746
g;g
CC(=O)C
acetone
20.0
mL
null
null
null
null
null
null
null
null
55.0
0.1667
C(C1=CC=CC=C1)NC(=S)NC1=CC=C(C(=O)NC2=CC=C(C=C2)NC(NCC2=CC=CC=C2)=S)C=C1
colorless crystal
0.57
g
43.4
ord-96af32b871984951b1483d8522037b06
[CH:1]1[C:6]([NH2:7])=[CH:5][CH:4]=[C:3]([NH2:8])[CH:2]=1.[CH2:9]([N:16]=[C:17]=[S:18])[C:10]1[CH:15]=[CH:14][CH:13]=[CH:12][CH:11]=1>C(OCC)(=O)C>[CH2:9]([NH:16][C:17]([NH:7][C:6]1[CH:5]=[CH:4][C:3]([NH:8][C:17](=[S:18])[NH:16][CH2:9][C:10]2[CH:15]=[CH:14][CH:13]=[CH:12][CH:11]=2)=[CH:2][CH:1]=1)=[S:18])[C:10]1[CH:15]=...
C1=CC(=CC=C1N)N.C(C1=CC=CC=C1)N=C=S
p-Phenylenediamine;benzylisothiocyanate
2.707;7.461
g;g
C(C)(=O)OCC
ethyl acetate
20.0
mL
null
null
null
null
null
null
null
null
80.0
0.5
C(C1=CC=CC=C1)NC(=S)NC1=CC=C(C=C1)NC(NCC1=CC=CC=C1)=S
colorless crystal
6.26
g
61.6
ord-86468e176b4c448b95c93ea7f5a809d2
[CH3:1][C:2]1[CH:7]=[C:6]([NH2:8])[C:5]([CH3:9])=[CH:4][C:3]=1[NH2:10].[C:11]([N:19]=[C:20]=[S:21])(=[O:18])[C:12]1[CH:17]=[CH:16][CH:15]=[CH:14][CH:13]=1>C(OCC)(=O)C>[C:11]([NH:19][C:20]([NH:8][C:6]1[CH:7]=[C:2]([CH3:1])[C:3]([NH:10][C:20](=[S:21])[NH:19][C:11](=[O:18])[C:12]2[CH:17]=[CH:16][CH:15]=[CH:14][CH:13]=2)=[...
CC1=C(C=C(C(=C1)N)C)N.C(C1=CC=CC=C1)(=O)N=C=S
2,5-Dimethyl-p-phenylenediamine;benzoylisothiocyanate
0.34;0.816
g;g
C(C)(=O)OCC
ethyl acetate
30.0
mL
null
null
null
null
null
null
null
null
ambient
0.1667
C(C1=CC=CC=C1)(=O)NC(=S)NC1=C(C=C(C(=C1)C)NC(NC(C1=CC=CC=C1)=O)=S)C
colorless crystal
1.14
g
98.7
ord-d421bcbbd72f4cb18c2bcf8464545117
[C:1]1([NH2:12])[C:10]2[CH:9]=[CH:8][CH:7]=[C:6]([NH2:11])[C:5]=2[CH:4]=[CH:3][CH:2]=1.[CH2:13]([N:20]=[C:21]=[S:22])[C:14]1[CH:19]=[CH:18][CH:17]=[CH:16][CH:15]=1>C(OCC)(=O)C>[CH2:13]([NH:20][C:21]([NH:12][C:1]1[C:10]2[C:5](=[C:6]([NH:11][C:21](=[S:22])[NH:20][CH2:13][C:14]3[CH:19]=[CH:18][CH:17]=[CH:16][CH:15]=3)[CH:...
C1(=CC=CC=2C(=CC=CC12)N)N.C(C1=CC=CC=C1)N=C=S
1,5-Naphthalenediamine;benzylisothiocyanate
0.791;1.492
g;g
C(C)(=O)OCC
ethyl acetate
20.0
mL
null
null
null
null
null
null
null
null
80.0
0.5
C(C1=CC=CC=C1)NC(=S)NC1=CC=CC2=C(C=CC=C12)NC(NCC1=CC=CC=C1)=S
colorless crystal
0.7
g
30.7
ord-178874a666824f65bd0ae92352c272a1
[OH2:1].[OH:2][CH2:3][CH:4]([CH2:6][OH:7])[OH:5]>>[OH:2][CH2:3][C@@H:4]([C@H:6]([C@@H:6]([C@@H:4]([CH2:3][OH:2])[OH:5])[OH:1])[OH:7])[OH:5]
OCC(O)CO.O.O
glycerine;water;water
0.0;0.0;0.0
mol;mol;mol
null
null
null
null
null
null
null
null
null
null
null
null
null
null
OC[C@H](O)[C@@H](O)[C@H](O)[C@H](O)CO
sorbitol
null
null
null
ord-c078782347f44c58bb85cd3aadab3128
[Cl:1][C:2]1[CH:10]=[C:6]([C:7]([OH:9])=[O:8])[C:5]([OH:11])=[CH:4][CH:3]=1.S(=O)(=O)(O)O.[CH3:17]O>>[Cl:1][C:2]1[CH:10]=[C:6]([C:7]([O:9][CH3:17])=[O:8])[C:5]([OH:11])=[CH:4][CH:3]=1
ClC1=CC=C(C(C(=O)O)=C1)O.S(O)(O)(=O)=O.CO
5-Chlorosalicylic acid;sulfuric acid;methanol
0.0;0.0;0.0
mol;mol;mol
null
null
null
null
null
null
null
null
null
null
null
null
null
null
ClC1=CC=C(C(C(=O)OC)=C1)O
methyl 5-chlorosalicylate
null
null
null
ord-e00a6267a6b742de87d3f8d8a6c2a5b7
[C:1]([O-:13])(=[O:12])[CH2:2][C:3]([CH2:8][C:9]([O-:11])=[O:10])([C:5]([O-:7])=[O:6])[OH:4].[CH3:14][C:15]([CH3:17])=[O:16]>CO>[C:1]([O-:13])(=[O:12])[CH2:2][C:3]([CH2:8][C:9]([O-:11])=[O:10])([C:5]([O-:7])=[O:6])[OH:4].[CH3:14][C:15]([CH3:17])=[O:16].[CH3:3][OH:4] |f:3.4.5|
C(CC(O)(C(=O)[O-])CC(=O)[O-])(=O)[O-].CC(=O)C
Citrate;Acetone
18.0;27.0
mL;mL
CO
methanol
5.0
mL
null
null
null
null
null
null
null
null
null
null
C(CC(O)(C(=O)[O-])CC(=O)[O-])(=O)[O-].CC(=O)C.CO
Citrate Acetone MeOH
null
null
null
ord-e1ac06e7bdc449a283a63a6a8683ed03
[C:1]([O-:13])(=[O:12])[CH2:2][C:3]([CH2:8][C:9]([O-:11])=[O:10])([C:5]([O-:7])=[O:6])[OH:4].[CH3:14][C:15]([CH3:17])=[O:16]>CO>[C:1]([O-:13])(=[O:12])[CH2:2][C:3]([CH2:8][C:9]([O-:11])=[O:10])([C:5]([O-:7])=[O:6])[OH:4].[CH3:14][C:15]([CH3:17])=[O:16].[CH3:3][OH:4] |f:3.4.5|
C(CC(O)(C(=O)[O-])CC(=O)[O-])(=O)[O-].CC(=O)C
Citrate;Acetone
18.0;27.0
mL;mL
CO
methanol
5.0
mL
null
null
null
null
null
null
null
null
null
null
C(CC(O)(C(=O)[O-])CC(=O)[O-])(=O)[O-].CC(=O)C.CO
Citrate Acetone MeOH
null
null
null
ord-0b3cb71fbde54da5a7c439131d7d2319
[CH2:1]([NH:3][CH2:4][CH2:5][CH2:6][O:7][CH3:8])[CH3:2].C(O)(=O)C.[N:13]#[C:14][NH2:15].C([O-])(=O)C>>[CH3:8][O:7][CH2:6][CH2:5][CH2:4][N:3]([CH2:1][CH3:2])[C:14]([NH2:15])=[NH:13]
C(C)NCCCOC.C(C)(=O)O.C(C)(=O)[O-].N#CN
N-ethyl-3-methoxypropylamine;acetic acid;acetate;cyanamide
3.0;1.54;0.0;1.08
g;g;mol;g
null
two
50.0
mL
null
null
null
null
null
null
null
null
90.0
null
COCCCN(C(=N)N)CC
title compound
2.8
g
50
ord-b22e751eea1540b88d656fbdc64a0e99
[CH3:1][O:2][CH2:3][CH2:4][O:5][CH2:6][CH2:7][NH2:8].C(O)(=O)C.[N:13]#[C:14][NH2:15].C([O-])(=O)C>>[CH3:1][O:2][CH2:3][CH2:4][O:5][CH2:6][CH2:7][NH:8][C:14]([NH2:15])=[NH:13]
COCCOCCN.C(C)(=O)O.C(C)(=O)[O-].N#CN
2-(2-methoxyethoxy)ethylamine;acetic acid;acetate;cyanamide
5.96;3.0;0.0;3.1
g;g;mol;g
null
two
30.0
mL
null
null
null
null
null
null
null
null
90.0
null
COCCOCCNC(=N)N
title compound
3.15
g
28.4
ord-64d5f5dd2f664288acccc0452c5aa2a9
[C:1]([O:9][CH2:10][CH2:11][O:12][CH2:13][CH2:14][NH2:15])(=[O:8])[C:2]1[CH:7]=[CH:6][CH:5]=[CH:4][CH:3]=1.C(O)(=O)C.[N:20]#[C:21][NH2:22].C([O-])(=O)C>>[C:1]([O:9][CH2:10][CH2:11][O:12][CH2:13][CH2:14][NH:15][C:21]([NH2:22])=[NH:20])(=[O:8])[C:2]1[CH:7]=[CH:6][CH:5]=[CH:4][CH:3]=1
C(C1=CC=CC=C1)(=O)OCCOCCN.C(C)(=O)O.C(C)(=O)[O-].N#CN
2-(2-aminoethoxy)ethyl benzoate;acetic acid;acetate;cyanamide
2.14;0.624;0.0;0.68
g;g;mol;g
null
two
50.0
mL
null
null
null
null
null
null
null
null
90.0
null
C(C1=CC=CC=C1)(=O)OCCOCCNC(=N)N
title compound
1.97
g
62.1
ord-84fae49193d148f395e8e28f50d554ab
C(O)(=O)C[CH2:3][C:4]([OH:6])=[O:5].O[CH2:10][CH2:11][O:12][CH2:13][CH2:14][NH:15][C:16]([NH2:18])=[NH:17].C(OC(=O)C)(=O)C.C([O-])(=O)C>C(N(CC)CC)C>[C:4]([O:6][CH2:10][CH2:11][O:12][CH2:13][CH2:14][NH:15][C:16]([NH2:18])=[NH:17])(=[O:5])[CH3:3] |f:0.1|
.C(CCC(=O)O)(=O)O.OCCOCCNC(=N)N..C(C)(=O)[O-].C(C)(=O)OC(C)=O
two;2-(2-hydroxyethoxy)ethylguanidine succinate;4-N,N-dimethylaminopyridine;acetate;acetic anhydride
50.0;2.06;0.000122;0.0;1.02
mL;g;g;mol;g
C(C)N(CC)CC
triethylamine
8.0
mL
null
null
null
null
null
null
null
null
ambient
1
C(C)(=O)OCCOCCNC(=N)N
title compound
1
g
40
ord-a6fad661b27341e199b0050914752841
[CH3:1][CH2:2][CH2:3][CH2:4][CH2:5][CH3:6].[CH:7]1[CH:12]=[CH:11][CH:10]=[CH:9][CH:8]=1.C1(C)C=CC=CC=1>CC1C=CC(C)=CC=1>[CH3:1][CH2:2][CH2:3][CH2:4][CH2:5][CH2:6][CH2:11][CH2:12][CH2:7][CH2:8][CH2:9][CH3:10]
CCCCCC.C1=CC=CC=C1.C1(=CC=CC=C1)C
n-hexane;benzene;toluene
0.0;0.0;0.0
mol;mol;mol
CC=1C=CC(=CC1)C
p-xylene
0.0
mol
null
null
null
null
null
null
null
null
null
null
CCCCCCCCCCCC
dodecane
null
null
null
ord-ec57be9eb3044d5884323695460dbccf
[CH2:1]([C@H:3]([NH:10][C:11](=[O:49])[C@@H:12]([C@H:39]([CH3:48])[O:40]CC1C=CC=CC=1)[NH:13][C:14](=[O:38])[C@H:15]([CH:27](CC1C=CC=CC=1)[C:28](=[O:30])[OH:29])[NH:16]C(OCC1C=CC=CC=1)=O)[C:4]1[CH:9]=[CH:8][CH:7]=[CH:6][CH:5]=1)[CH3:2].C(O)(=O)C>CO.[Pd].[C]>[CH2:1]([C@H:3]([NH:10][C:11](=[O:49])[C@@H:12]([C@H:39]([CH3:4...
C(C)[C@@H](C1=CC=CC=C1)NC([C@H](NC([C@@H](NC(=O)OCC1=CC=CC=C1)C(C(O)=O)CC1=CC=CC=C1)=O)[C@@H](OCC1=CC=CC=C1)C)=O.C(C)(=O)O
N-benzyloxycarbonyl-β-benzyl-L-aspartyl-O-benzyl-D-threonine (S)-α-ethylbenzylamide;acetic acid
5.3;1.0
g;mL
CO
methanol
150.0
mL
[Pd].[C]
Pd carbon
3.0
g
null
null
null
null
null
8
C(C)[C@@H](C1=CC=CC=C1)NC([C@H](NC([C@@H](N)CC(O)=O)=O)[C@@H](O)C)=O
α-L-aspartyl-D-threonine (S)-α-ethylbenzylamide
1.6
g
57.5
ord-a473542e2c91474d920bd8a0505e632c
[CH2:1]([O:8][C:9]([NH:11][C@H:12]([C:24]([NH:26][C@@H:27]([C:32](O)=[O:33])[C@@H:28]([CH2:30][CH3:31])[CH3:29])=[O:25])[CH:13]([CH2:17][C:18]1[CH:23]=[CH:22][CH:21]=[CH:20][CH:19]=1)[C:14](=[O:16])[OH:15])=[O:10])[C:2]1[CH:7]=[CH:6][CH:5]=[CH:4][CH:3]=1.[CH2:35]([C@H:37]([NH2:44])[C:38]1[CH:43]=[CH:42][CH:41]=[CH:40][...
C(C1=CC=CC=C1)OC(=O)N[C@@H](C(C(O)=O)CC1=CC=CC=C1)C(=O)N[C@H]([C@H](C)CC)C(=O)O.C(C)[C@@H](C1=CC=CC=C1)N.O.C=1C=CC2=C(C1)N=NN2O
N-benzyloxycarbonyl-β-benzyl-L-aspartyl-D-isoleucine;(S)-α-ethylbenzylamine;water;HOBt
6.69;2.04;2.73;1.92
g;g;g;g
C(Cl)Cl
methylene chloride
200.0
mL
null
null
null
null
null
null
null
null
null
1
C(C)[C@@H](C1=CC=CC=C1)NC([C@H](NC([C@@H](NC(=O)OCC1=CC=CC=C1)C(C(O)=O)CC1=CC=CC=C1)=O)[C@H](C)CC)=O
N-benzyloxycarbonyl-β-benzyl-L-aspartyl-D-isoleucine (S)-α-ethylbenzylamide
2.81
g
33.1
ord-b4a1a9f06c874053b3ad0f85aaa15884
[CH2:1]([C@H:3]([NH:10][C:11](=[O:43])[C@@H:12]([C@@H:39]([CH2:41][CH3:42])[CH3:40])[NH:13][C:14](=[O:38])[C@H:15]([CH:27](CC1C=CC=CC=1)[C:28](=[O:30])[OH:29])[NH:16]C(OCC1C=CC=CC=1)=O)[C:4]1[CH:9]=[CH:8][CH:7]=[CH:6][CH:5]=1)[CH3:2]>CO.O.[Pd].[C]>[CH2:1]([C@H:3]([NH:10][C:11](=[O:43])[C@@H:12]([C@@H:39]([CH2:41][CH3:4...
C(C)[C@@H](C1=CC=CC=C1)NC([C@H](NC([C@@H](NC(=O)OCC1=CC=CC=C1)C(C(O)=O)CC1=CC=CC=C1)=O)[C@H](C)CC)=O
N-benzyloxycarbonyl-β-benzyl-L-aspartyl-D-isoleucine (S)-α-ethylbenzylamide
2.81
g
CO.O
methanol;water
150.0;50.0
mL;mL
[Pd].[C]
Pd carbon
2.0
g
null
null
null
null
null
5
C(C)[C@@H](C1=CC=CC=C1)NC([C@H](NC([C@@H](N)CC(O)=O)=O)[C@H](C)CC)=O
α-L-aspartyl-D-isoleucine (S)-α-ethylbenzylamide
1.22
g
72.3
ord-39d7a85f6c0943d29b102f7ee592196e
Cl.O1CCOCC1.[CH2:8]([C@H:10]([NH:17][C:18](=[O:32])[C:19]([CH2:30][CH3:31])([CH2:28][CH3:29])[NH:20][C:21]([O:23]C(C)(C)C)=O)[C:11]1[CH:16]=[CH:15][CH:14]=[CH:13][CH:12]=1)[CH3:9].C(N(CC)CC)C.C([CH:47]([C:63]([O-:65])=[O:64])[C@@H:48](C([O-])=O)[NH:49]C(OCC1C=CC=CC=1)=O)C1C=CC=CC=1.O.C1C=CC2N(O)N=NC=2C=1>>[CH2:8]([C@H:...
O.C=1C=CC2=C(C1)N=NN2O.Cl.O1CCOCC1.C(C)[C@@H](C1=CC=CC=C1)NC(C(NC(=O)OC(C)(C)C)(CC)CC)=O.C(C)N(CC)CC.C(C1=CC=CC=C1)C([C@H](NC(=O)OCC1=CC=CC=C1)C(=O)[O-])C(=O)[O-]
water;HOBt;HCl dioxane;N-t-butoxycarbonyl-α,α-diethylglycine (S)-α-ethylbenzylamide;triethylamine;β-benzyl-N-benzyloxycarbonyl-L-aspartate
0.79;0.51;0.0;1.31;0.55;1.48
g;g;mol;g;mL;g
null
null
null
null
null
null
null
null
null
null
null
null
ambient
1
C(C)[C@@H](C1=CC=CC=C1)NC(C(NC([C@@H](N)CC(O)=O)=O)(CC)CC)=O
α-L-aspartyl-α,α-diethylglycine (S)-α-ethylbenzylamide
0.4
g
29.3
ord-a2a351b69552484f9b0780b4d2a5b2e4
Cl.[O:2]1[CH2:7][CH2:6]OCC1.[CH2:8]([C@H:10]([NH:17][C:18](=[O:31])[C:19]([CH3:30])([CH2:28][CH3:29])[NH:20][C:21]([O:23]C(C)(C)C)=O)[C:11]1[CH:16]=[CH:15][CH:14]=[CH:13][CH:12]=1)[CH3:9].C([N:34]([CH2:37]C)CC)C.[OH2:39]>>[CH2:8]([C@H:10]([NH:17][C:18](=[O:31])[C:19]([CH3:30])([CH2:28][CH3:29])[NH:20][C:21](=[O:23])[C@...
Cl.O1CCOCC1..C(C)[C@@H](C1=CC=CC=C1)NC(C(NC(=O)OC(C)(C)C)(CC)C)=O.O.C(C)N(CC)CC.
HCl dioxane;0.66;N-t-butoxycarbonyl-DL-isovaline (S)-α-ethylbenzylamide;water;triethylamine;β-benzyl N-benzyloxycarbonyl-L-aspartate
0.0;0.00197;0.0;0.34;0.24;0.63
mol;mol;mol;g;mL;g
null
null
null
null
null
null
null
null
null
null
null
null
ambient
1
C(C)[C@@H](C1=CC=CC=C1)NC(C(NC([C@@H](N)CC(O)=O)=O)(CC)C)=O
α-L-aspartyl-DL-isovaline (S)-α-ethylbenzylamide
0.21
g
null
ord-3d062dc2d8ab4e1391656e4f536498a8
[ClH:1].O1CCOCC1.C(OC([NH:15][C@@H:16]([CH2:23][O:24][CH3:25])[C:17]1[CH:22]=[CH:21][CH:20]=[CH:19][CH:18]=1)=O)(C)(C)C>>[ClH:1].[CH3:25][O:24][CH2:23][C@H:16]([NH2:15])[C:17]1[CH:22]=[CH:21][CH:20]=[CH:19][CH:18]=1 |f:0.1,3.4|
Cl.O1CCOCC1.C(C)(C)(C)OC(=O)N[C@H](C1=CC=CC=C1)COC
HCl dioxane;N-t-butoxycarbonyl-(R)-α-methoxymethylbenzylamine
0.0;4.02
mol;g
null
null
null
null
null
null
null
null
null
null
null
null
ambient
1
Cl.COC[C@@H](C1=CC=CC=C1)N
(R)-α-methoxymethylbenzylamine hydrochloride
null
null
null
ord-1b033c485fa54b2cb55a6e97a581a99c
[CH3:1][O:2][CH2:3][C@H:4]([NH:11][C:12](=[O:43])[C@@H:13]([CH:40]([CH3:42])[CH3:41])[NH:14][C:15](=[O:39])[C@H:16]([CH:28](CC1C=CC=CC=1)[C:29](=[O:31])[OH:30])[NH:17]C(OCC1C=CC=CC=1)=O)[C:5]1[CH:10]=[CH:9][CH:8]=[CH:7][CH:6]=1>CO.O.[Pd].[C]>[CH3:1][O:2][CH2:3][C@H:4]([NH:11][C:12](=[O:43])[C@@H:13]([CH:40]([CH3:41])[C...
COC[C@@H](C1=CC=CC=C1)NC([C@H](NC([C@@H](NC(=O)OCC1=CC=CC=C1)C(C(O)=O)CC1=CC=CC=C1)=O)C(C)C)=O
N-benzyloxycarbonyl-β-benzyl-L-aspartyl-D-valine (R)-α-methoxymethylbenzylamide
6.2
g
CO.O
methanol;water
200.0;50.0
mL;mL
[Pd].[C]
Pd carbon
1.5
g
null
null
null
null
40.0
null
COC[C@@H](C1=CC=CC=C1)NC([C@H](NC([C@@H](N)CC(O)=O)=O)C(C)C)=O
α-L-aspartyl-D-valine (R)-α-methoxymethylbenzylamide
2.69
g
70.1
ord-ae03dc6af35144969588f144b56bba80
[ClH:1].O1CCOCC1.C(OC([NH:15][C@@H:16]([CH2:23][O:24][CH2:25][CH3:26])[C:17]1[CH:22]=[CH:21][CH:20]=[CH:19][CH:18]=1)=O)(C)(C)C>>[ClH:1].[CH2:25]([O:24][CH2:23][C@H:16]([NH2:15])[C:17]1[CH:22]=[CH:21][CH:20]=[CH:19][CH:18]=1)[CH3:26] |f:0.1,3.4|
Cl.O1CCOCC1.C(C)(C)(C)OC(=O)N[C@H](C1=CC=CC=C1)COCC
HCl dioxane;N-t-butoxycarbonyl-(R)-α-ethoxymethylbenzylamine
0.0;0.66
mol;g
null
null
null
null
null
null
null
null
null
null
null
null
ambient
1
Cl.C(C)OC[C@@H](C1=CC=CC=C1)N
(R)-α-ethoxymethylbenzylamine hydrochloride
null
null
null
ord-29bd294101a04d54b49813c6be393808
[CH2:1]([O:3][CH2:4][C@H:5]([NH:12][C:13](=[O:44])[C@@H:14]([CH:41]([CH3:43])[CH3:42])[NH:15][C:16](=[O:40])[C@H:17]([CH:29](CC1C=CC=CC=1)[C:30](=[O:32])[OH:31])[NH:18]C(OCC1C=CC=CC=1)=O)[C:6]1[CH:11]=[CH:10][CH:9]=[CH:8][CH:7]=1)[CH3:2]>CO.O.[Pd].[C]>[CH2:1]([O:3][CH2:4][C@H:5]([NH:12][C:13](=[O:44])[C@@H:14]([CH:41](...
C(C)OC[C@@H](C1=CC=CC=C1)NC([C@H](NC([C@@H](NC(=O)OCC1=CC=CC=C1)C(C(O)=O)CC1=CC=CC=C1)=O)C(C)C)=O
N-benzyloxycarbonyl-β-benzyl-L-aspartyl-D-valine (R)-α-ethoxymethylbenzylamide
1.2
g
CO.O.O
methanol;water;water
50.0;10.0;40.0
mL;mL;mL
[Pd].[C]
Pd carbon
0.3
g
null
null
null
null
40.0
null
C(C)OC[C@@H](C1=CC=CC=C1)NC([C@H](NC([C@@H](N)CC(O)=O)=O)C(C)C)=O
α-L-aspartyl-D-valine (R)-α-ethoxymethylbenzylamide
0.38
g
50.3
ord-f6a778234f084513ae50b4ca3b6875a0
C(OC([NH:11][C@H:12]([C:24]([NH:26][C@@H:27]([C:32](O)=[O:33])[C@@H:28]([CH2:30][CH3:31])[CH3:29])=[O:25])[CH:13](CC1C=CC=CC=1)[C:14](=[O:16])[OH:15])=O)C1C=CC=CC=1.Cl.[CH3:36][O:37][CH2:38][C@H:39]([NH2:46])[C:40]1[CH:45]=[CH:44][CH:43]=[CH:42][CH:41]=1>>[CH3:36][O:37][CH2:38][C@H:39]([NH:46][C:32](=[O:33])[C@@H:27]([...
C(C1=CC=CC=C1)OC(=O)N[C@@H](C(C(O)=O)CC1=CC=CC=C1)C(=O)N[C@H]([C@H](C)CC)C(=O)O.Cl.COC[C@@H](C1=CC=CC=C1)N
N-benzyloxycarbonyl-β-benzyl-L-aspartyl-D-isoleucine;(R)-α-methoxymethylbenzylamine hydrochloride
0.0;0.0
mol;mol
null
null
null
null
null
null
null
null
null
null
null
null
null
null
COC[C@@H](C1=CC=CC=C1)NC([C@H](NC([C@@H](N)CC(O)=O)=O)[C@H](C)CC)=O
α-L-aspartyl-D-isoleucine (R)-α-methoxymethylbenzylamide
null
null
22.1
ord-12a035e31d384b0d952ee7e106393c5e
C(OC([NH:11][C@H:12]([C:24]([NH:26][C@@H:27]([C:29](O)=[O:30])[CH3:28])=[O:25])[CH:13](CC1C=CC=CC=1)[C:14](=[O:16])[OH:15])=O)C1C=CC=CC=1.Cl.[CH3:33][O:34][CH2:35][C@H:36]([NH2:43])[C:37]1[CH:42]=[CH:41][CH:40]=[CH:39][CH:38]=1>>[CH3:33][O:34][CH2:35][C@H:36]([NH:43][C:29](=[O:30])[C@@H:27]([CH3:28])[NH:26][C:24](=[O:2...
C(C1=CC=CC=C1)OC(=O)N[C@@H](C(C(O)=O)CC1=CC=CC=C1)C(=O)N[C@H](C)C(=O)O.Cl.COC[C@@H](C1=CC=CC=C1)N
N-benzyloxycarbonyl-β-benzyl-L-aspartyl-D-alanine;(R)-α-methoxymethylbenzylamine hydrochloride
0.0;0.0
mol;mol
null
null
null
null
null
null
null
null
null
null
null
null
null
null
COC[C@@H](C1=CC=CC=C1)NC([C@H](NC([C@@H](N)CC(O)=O)=O)C)=O
α-L-aspartyl-D-alanine-(R)-α-methoxymethylbenzylamide
null
null
57.3
ord-d6db1ba811484e3384ed2f23fdfc613c
[P:1]([O-:5])([O-:4])([O-:3])=[O:2].[Na+].[Na+].[Na+].[Cl-].[Ca+2:10].[Cl-]>O>[P:1]([O-:5])([O-:4])([O-:3])=[O:2].[Ca+2:10].[Ca+2:10].[Ca+2:10].[P:1]([O-:5])([O-:4])([O-:3])=[O:2] |f:0.1.2.3,4.5.6,8.9.10.11.12|
P(=O)([O-])([O-])[O-].[Na+].[Na+].[Na+].[Cl-].[Ca+2].[Cl-]
sodium phosphate;calcium chloride
0.0;45.3
mol;g
O.O.O
water;water;water
300.0;300.0;200.0
g;g;g
null
null
null
null
null
null
null
null
null
null
P(=O)([O-])([O-])[O-].[Ca+2].[Ca+2].[Ca+2].P(=O)([O-])([O-])[O-]
tricalcium phosphate
null
null
null
ord-a5d5cdb2b6f74613b95722ef03582f33
[P:1]([O-:5])([O-:4])([O-:3])=[O:2].[Na+].[Na+].[Na+].[Cl-].[Ca+2:10].[Cl-]>O>[P:1]([O-:5])([O-:4])([O-:3])=[O:2].[Ca+2:10].[Ca+2:10].[Ca+2:10].[P:1]([O-:5])([O-:4])([O-:3])=[O:2] |f:0.1.2.3,4.5.6,8.9.10.11.12|
P(=O)([O-])([O-])[O-].[Na+].[Na+].[Na+].[Cl-].[Ca+2].[Cl-]
sodium phosphate;calcium chloride
0.0;45.3
mol;g
O.O.O
water;water;water
300.0;300.0;200.0
g;g;g
null
null
null
null
null
null
null
null
null
null
P(=O)([O-])([O-])[O-].[Ca+2].[Ca+2].[Ca+2].P(=O)([O-])([O-])[O-]
tricalcium phosphate
null
null
null
ord-1486324d16694ddca5c93306441d16d7
[P:1]([O-:5])([O-:4])([O-:3])=[O:2].[Na+].[Na+].[Na+].[Cl-].[Ca+2:10].[Cl-]>O>[P:1]([O-:5])([O-:4])([O-:3])=[O:2].[Ca+2:10].[Ca+2:10].[Ca+2:10].[P:1]([O-:5])([O-:4])([O-:3])=[O:2] |f:0.1.2.3,4.5.6,8.9.10.11.12|
P(=O)([O-])([O-])[O-].[Na+].[Na+].[Na+].[Cl-].[Ca+2].[Cl-]
sodium phosphate;calcium chloride
0.0;45.3
mol;g
O.O.O
water;water;water
300.0;300.0;200.0
g;g;g
null
null
null
null
null
null
null
null
null
null
P(=O)([O-])([O-])[O-].[Ca+2].[Ca+2].[Ca+2].P(=O)([O-])([O-])[O-]
tricalcium phosphate
null
null
null
ord-59691e7705044240a0b61a8537732528
[P:1]([O-:5])([O-:4])([O-:3])=[O:2].[Na+].[Na+].[Na+].[Cl-].[Ca+2:10].[Cl-]>O>[P:1]([O-:5])([O-:4])([O-:3])=[O:2].[Ca+2:10].[Ca+2:10].[Ca+2:10].[P:1]([O-:5])([O-:4])([O-:3])=[O:2] |f:0.1.2.3,4.5.6,8.9.10.11.12|
P(=O)([O-])([O-])[O-].[Na+].[Na+].[Na+].[Cl-].[Ca+2].[Cl-]
sodium phosphate;calcium chloride
0.0;22.65
mol;g
O.O.O.O.O
water;Solution A;water;Solution B;water
150.0;0.0;150.0;0.0;200.0
g;mol;g;mol;g
null
null
null
null
null
null
null
null
null
null
P(=O)([O-])([O-])[O-].[Ca+2].[Ca+2].[Ca+2].P(=O)([O-])([O-])[O-]
tricalcium phosphate
null
null
null
ord-d6f09b988e0848769dd846f380d71108
[OH:1][C:2]1[CH:9]=[CH:8][C:5]([CH:6]=[O:7])=[CH:4][CH:3]=1.Br[CH2:11][CH2:12][CH:13]1[O:18][CH2:17][CH2:16][CH2:15][O:14]1.[I-].[K+].C(=O)([O-])[O-].[K+].[K+]>C(OCC)(=O)C.C(#N)C>[O:14]1[CH2:15][CH2:16][CH2:17][O:18][CH:13]1[CH2:12][CH2:11][O:1][C:2]1[CH:9]=[CH:8][C:5]([CH:6]=[O:7])=[CH:4][CH:3]=1 |f:2.3,4.5.6|
OC1=CC=C(C=O)C=C1.BrCCC1OCCCO1.[I-].[K+].C([O-])([O-])=O.[K+].[K+]
4-hydroxybenzaldehyde;2-(2-bromoethyl)-1,3-dioxane;potassium iodide;potassium carbonate
13.8;21.1;1.8;35.8
g;g;g;g
C(C)(=O)OCC.C(C)#N
ethyl acetate;acetonitrile
200.0;120.0
mL;mL
null
null
null
null
null
null
null
null
null
null
O1C(OCCC1)CCOC1=CC=C(C=O)C=C1
4-(2-[1,3]-dioxane-2-yl-ethoxy)benzaldehyde
25.6
g
100.2
ord-7962a8e3cbfa49e3aabf54e37edc9672
[CH3:1]C(C)([O-])C.[K+].[O:7]1[CH2:12][CH2:11][CH2:10][O:9][CH:8]1[CH2:13][CH2:14][O:15][C:16]1[CH:23]=[CH:22][C:19]([CH:20]=O)=[CH:18][CH:17]=1>[Br-].C[P+](C1C=CC=CC=1)(C1C=CC=CC=1)C1C=CC=CC=1.CCOCC>[CH:20]([C:19]1[CH:22]=[CH:23][C:16]([O:15][CH2:14][CH2:13][CH:8]2[O:9][CH2:10][CH2:11][CH2:12][O:7]2)=[CH:17][CH:18]=1)...
CC(C)([O-])C.[K+].O1C(OCCC1)CCOC1=CC=C(C=O)C=C1
potassium tert-butoxide;4-(2-[1,3]-dioxane-2-yl-ethoxy)benzaldehyde
18.0;25.6
g;g
CCOCC.CCOCC
ether;ether
500.0;200.0
mL;mL
[Br-].C[P+](C1=CC=CC=C1)(C1=CC=CC=C1)C1=CC=CC=C1
methyl triphenylphosphonium bromide
57.2
g
null
null
null
null
null
null
C(=C)C1=CC=C(OCCC2OCCCO2)C=C1
2-[2-(4-vinylphenoxy)ethyl]-[1,3]-dioxane
19.7
g
77.6
ord-ab767623531e408bb0c0320b5128145a
[OH:1][C:2]1[CH:9]=[CH:8][C:5]([CH:6]=[O:7])=[CH:4][CH:3]=1.Br[CH2:11][CH2:12][CH:13]1[O:18][CH2:17][CH2:16]C[O:14]1.[I-].[K+].C(=O)([O-])[O-].[K+].[K+]>C(OCC)(=O)C.C(#N)C>[O:18]1[CH2:17][CH2:16][O:14][CH:13]1[CH2:12][CH2:11][O:1][C:2]1[CH:9]=[CH:8][C:5]([CH:6]=[O:7])=[CH:4][CH:3]=1 |f:2.3,4.5.6|
OC1=CC=C(C=O)C=C1.BrCCC1OCCCO1.[I-].[K+].C([O-])([O-])=O.[K+].[K+]
4-hydroxybenzaldehyde;2-(2-bromoethyl)-1,3-dioxane;potassium iodide;potassium carbonate
13.8;19.9;1.8;35.8
g;g;g;g
C(C)(=O)OCC.C(C)#N
ethyl acetate;acetonitrile
200.0;120.0
mL;mL
null
null
null
null
null
null
null
null
null
null
O1C(OCC1)CCOC1=CC=C(C=O)C=C1
4-(2-[1,3]-dioxolan-2-yl-ethoxy)benzaldehyde
23.7
g
104.5
ord-09284bc5f4434b24a76abcd1557a624c
[CH3:1]C(C)([O-])C.[K+].[O:7]1[CH2:11][CH2:10][O:9][CH:8]1[CH2:12][CH2:13][O:14][C:15]1[CH:22]=[CH:21][C:18]([CH:19]=O)=[CH:17][CH:16]=1>[Br-].C[P+](C1C=CC=CC=1)(C1C=CC=CC=1)C1C=CC=CC=1.CCOCC>[CH:19]([C:18]1[CH:21]=[CH:22][C:15]([O:14][CH2:13][CH2:12][CH:8]2[O:9][CH2:10][CH2:11][O:7]2)=[CH:16][CH:17]=1)=[CH2:1] |f:0.1,...
CC(C)([O-])C.[K+].O1C(OCC1)CCOC1=CC=C(C=O)C=C1
potassium tert-butoxide;4-(2-[1,3]-dioxolan-2-yl-ethoxy)benzaldehyde
18.0;23.7
g;g
CCOCC.CCOCC
ether;ether
500.0;200.0
mL;mL
[Br-].C[P+](C1=CC=CC=C1)(C1=CC=CC=C1)C1=CC=CC=C1
methyl triphenylphosphonium bromide
57.2
g
null
null
null
null
null
null
C(=C)C1=CC=C(OCCC2OCCO2)C=C1
2-[2-(4-vinylphenoxy)ethyl]-[1,3]-dioxolan
20.8
g
88.5
ord-ddf67391f0ff4ca08b0e3124c9c5cf53
[CH:1]1[C:6]([OH:7])=[CH:5][CH:4]=[CH:3][C:2]=1[CH3:8].[OH:9][CH2:10]C1C(O)=C(CO)C=C(C)C=1.O.O.C(O)(=O)C(O)=O.CCOCCOC(C)=O.C=O>O>[C:1]1([CH:10]=[O:9])[C:2]([CH3:8])=[CH:3][CH:4]=[CH:5][C:6]=1[OH:7] |f:2.3.4|
CCOCCOC(=O)C.C1=C(C=CC=C1O)C.OCC1=CC(=CC(=C1O)CO)C.O.O.C(C(=O)O)(=O)O.C=O
ethyl cellosolve acetate;m-cresol;2,6-bis(hydroxymethyl)-p-cresol;oxalic acid dihydrate;formaldehyde
200.0;519.0;538.2;20.0;32.6
mL;g;g;g;g
O
water
0.0
mol
null
null
null
null
null
null
null
null
70.0
null
C=1(C(=CC=CC1O)C)C=O
m-cresol formaldehyde
null
null
null
ord-3c799edf560b44e4b1b3a6fde9733781
[C:1]([O:9][CH2:10][CH:11](CC)[CH2:12][CH:13]([OH:16])[CH2:14][CH3:15])(=[O:8])[C:2]1[CH:7]=[CH:6][CH:5]=[CH:4][CH:3]=1.O.[CH2:20]1[CH2:24]OC(N2C(=O)NC(=O)C(F)=C2)[CH2:21]1.[CH3:34][CH2:35][C:36]1([OH:49])[N:41]=[C:40]([C:42]2[CH:47]=[CH:46][C:45]([CH3:48])=[CH:44][CH:43]=2)[Se:39][CH2:38][CH2:37]1>C(OCC)(=O)C>[C:1]([O...
.CCC1(CC[Se]C(=N1)C2=CC=C(C=C2)C)O.O.CCC1(CC[Se]C(=N1)C2=CC=C(C=C2)C)O.O.C1CC(OC1)N2C=C(C(=O)NC2=O)F.O.C1CC(OC1)N2C=C(C(=O)NC2=O)F.CCC1(CC[Se]C(=N1)C2=CC=C(C=C2)C)O.C(C1=CC=CC=C1)(=O)OCC(CC(CC)O)CC.CCC1(CC[Se]C(=N1)C2=CC=C(C=C2)C)O
zirconia;TS-2;water;TS-2;water;TS-1;water;TS-1;TS-2;4-hydroxy-(2'-ethylhexyl) benzoate;TS-2
0.0;12.0;66.0;0.0;74.9;15.0;35.9;0.0;18.0;0.0;0.0
mol;g;g;mol;g;g;g;mol;g;mol;mol
C(C)(=O)OCC
ethyl acetate
24.0
g
null
null
null
null
null
null
null
null
null
123
C(C1=CC=CC=C1)(=O)OCCCC(CCCCC)O
4-hydroxy-nonyl benzoate
null
null
null
ord-bfcf42b524d14d69860f018538be3094
OC1[CH:7]=[CH:6][C:5]([C:8]2([C:21]3[CH:26]=CC(O)=CC=3)[C:20]3[CH:19]=[CH:18][CH:17]=[CH:16][C:15]=3[C:14]3C2=[CH:10][CH:11]=[CH:12][CH:13]=3)=[CH:4]C=1.C1(=O)O[CH2:31][CH2:30][O:29]1.[C:34](=[O:37])([O-])[O-].[K+].[K+].C1OCCOCCOCCOCCOCCOC1>>[OH:29][CH2:30][CH2:31][O:37][C:34]1[CH:10]=[CH:11][CH:12]=[CH:13][C:14]=1[C:1...
OC1=CC=C(C=C1)C1(C2=CC=CC=C2C=2C=CC=CC12)C1=CC=C(C=C1)O.C1(OCCO1)=O.C([O-])([O-])=O.[K+].[K+].C1COCCOCCOCCOCCOCCO1
9,9-bis(4-hydroxyphenyl)fluorene;ethylene carbonate;potassium carbonate;18-crown-6
84.4;46.7;3.3;0.0
g;g;g;mol
null
xylenes
400.0
mL
null
null
null
null
null
null
null
null
ambient
6
OCCOC1=C(C=CC=C1)C1=CC=CC=2CC3=CC=CC=C3C12
white powder
70.4
g
970.1
ord-a9328cbc649c44739edcb5b4674d8842
[Br:1][C:2]1[CH:7]=[CH:6][CH:5]=[CH:4][CH:3]=1.[C:8](Cl)(=[O:14])/[CH:9]=[CH:10]/[C:11](Cl)=O.[CH2:16]=[CH2:17]>OS(O)(=O)=O.[Zn].CC(O)=O>[Br:1][C:2]1[CH:7]=[CH:6][C:5]([C:11]2[O:14][C:8]([C:16]3[CH:4]=[CH:3][C:2]([Br:1])=[CH:7][CH:17]=3)=[CH:9][CH:10]=2)=[CH:4][CH:3]=1 |f:4.5|
.C=C..BrC1=CC=CC=C1.C(\C=C\C(=O)Cl)(=O)Cl..
1,4-di-p-bromophenyl-1,4-butanedione;ethylene;trans-di-p-bromobenzoylethylene;bromobenzene;fumaryl chloride;1,4-diketone;water ice
0.0;0.0;0.0;0.0;0.0;7.9;1000.0
mol;mol;mol;mol;mol;g;mL
null
null
null
null
[Zn].CC(=O)O.OS(=O)(=O)O
Zn HOAc;H2SO4
0.0;0.0
mol;mol
null
null
null
null
null
0.0833
BrC1=CC=C(C=C1)C=1OC(=CC1)C1=CC=C(C=C1)Br
2,5-Bis(p-bromophenyl) furan
null
null
null
ord-523a53f4b10c44568fb08b813772adeb
Br[CH:2]([C:14](=[O:22])[C:15]1[CH:20]=[CH:19][C:18]([Br:21])=[CH:17][CH:16]=1)[CH:3](Br)[C:4](=[O:12])[C:5]1[CH:10]=[CH:9][C:8]([Br:11])=[CH:7][CH:6]=1.[CH3:23][C:24]1[CH:30]=[CH:29][C:27]([O-:28])=[CH:26][CH:25]=1.[Na+].CC1C=CC(O)=CC=1>C1COCC1>[C:24]1([CH3:23])[CH:30]=[CH:29][C:27]([O:28][C:2]([C:14](=[O:22])[C:15]2[...
BrC(C(C(C1=CC=C(C=C1)Br)=O)Br)C(C1=CC=C(C=C1)Br)=O.CC1=CC=C([O-])C=C1.[Na+]..CC1=CC=C(C=C1)O
1,2-dibromo-1,2-di(4-bromobenzoyl) ethane;sodium 4-methyl phenoxide;Na;4-methylphenol
11.1;30.0;0.04;0.04
g;mL;mol;mol
C1CCOC1.C1CCOC1
THF;THF
0.0;35.0
mol;mL
null
null
null
null
null
null
null
null
null
null
C1(=CC=C(C=C1)OC(=CC(C1=CC=C(C=C1)Br)=O)C(C1=CC=C(C=C1)Br)=O)C
1-(4-tolyloxyl)-1,2-bis(4-bromobenzoyl)ethylene
null
null
null
ord-67300f99f22241ef9811a9c1212c4492
[C:1]1([CH3:28])[CH:6]=[CH:5][C:4]([O:7][C:8]([C:19](=O)[C:20]2[CH:25]=[CH:24][C:23]([Br:26])=[CH:22][CH:21]=2)=[CH:9][C:10](=[O:18])[C:11]2[CH:16]=[CH:15][C:14]([Br:17])=[CH:13][CH:12]=2)=[CH:3][CH:2]=1.[K+].[Br-]>P(Cl)(Cl)Cl>[Br:26][C:23]1[CH:22]=[CH:21][C:20]([C:19]2[O:18][C:10]([C:11]3[CH:12]=[CH:13][C:14]([Br:17])...
C1(=CC=C(C=C1)OC(=CC(C1=CC=C(C=C1)Br)=O)C(C1=CC=C(C=C1)Br)=O)C.[K+].[Br-]
1-(4-tolyloxy)-1,2-bis-(4-bromobenzoyl)ethylene;KBr
5.0;0.0
g;mol
P(Cl)(Cl)Cl
phosphorus trichloride
10.0
mL
null
null
null
null
null
null
null
null
null
null
BrC1=CC=C(C=C1)C=1OC(=CC1OC1=CC=C(C=C1)C)C1=CC=C(C=C1)Br
2,5-bis(4-Bromophenyl)-3-(p-tolyloxy)furan
null
null
null
ord-68a4112e542d4a8cb9aa4b70a263e0cb
Br[CH:2]([C:14](=[O:22])[C:15]1[CH:20]=[CH:19][C:18]([Br:21])=[CH:17][CH:16]=1)[CH:3](Br)[C:4](=[O:12])[C:5]1[CH:10]=[CH:9][C:8]([Br:11])=[CH:7][CH:6]=1.[CH3:23][O-:24].[Na+].[K+].[Br-]>CO>[Br:11][C:8]1[CH:9]=[CH:10][C:5]([C:4]([CH:3]([O:24][CH3:23])[CH2:2][C:14](=[O:22])[C:15]2[CH:20]=[CH:19][C:18]([Br:21])=[CH:17][CH...
[K+].[Br-].BrC(C(C(C1=CC=C(C=C1)Br)=O)Br)C(C1=CC=C(C=C1)Br)=O.C[O-].[Na+].
KBr;1,2-dibromo-1,2-di(4-bromobenzoyl) ethane;sodium methoxide;methanol-ether
0.0;11.1;0.0;0.0
mol;g;mol;mol
CO.CO
methanol;methanol
150.0;50.0
mL;mL
null
null
null
null
null
null
null
null
null
null
BrC1=CC=C(C(=O)C(CC(C2=CC=C(C=C2)Br)=O)OC)C=C1
1,2-Bis(4-bromobenzoyl)-1-methoxyethane
null
null
null
ord-4d66dfcc15f145d887e1d654294844a8
N1CCCN=C1C1C=CC([C:13]2[O:14][C:15]([C:18]3[CH:23]=[CH:22][C:21]([C:24]4[NH:25][CH2:26][CH2:27][CH2:28][N:29]=4)=[CH:20][CH:19]=3)=[CH:16][CH:17]=2)=CC=1.[CH:30]1C(C2NC3C=C(C(N)=N)C=CC=3C=2)=CC=C(C(N)=N)C=1.CN1CCN(C2C=CC3NC(C4C=[CH:69][C:70]5[NH:75][C:74]([C:76]6[CH:77]=[CH:78][C:79](O)=[CH:80][CH:81]=6)=[N:73][C:71]=5...
N1C(=NCCC1)C1=CC=C(C=C1)C=1OC(=CC1)C1=CC=C(C=C1)C=1NCCCN1.C1=CC(=CC=C1C2=CC=3C=CC(=CC3N2)C(=N)N)C(=N)N.CN1CCN(CC1)C=2C=CC3=C(C2)N=C(N3)C=4C=CC5=C(C4)N=C(N5)C=6C=CC(=CC6)O
2,5-bis[4-(1,4,5,6-tetrahydropyrimidin-2-yl)phenyl] furan;DAPI;Hoechst 33258
0.0;0.0;0.0
mol;mol;mol
null
null
null
null
null
null
null
null
null
null
null
null
null
null
N1C(=NCCCC1)C1=CC=C(C=C1)C=1OC(=CC1)C1=CC=C(C=C1)C=1NCCCCN1
2,5-bis [4-(4,5,6,7-tetrahydro-1H-1,3-diazepin-2-yl) phenyl] furan
null
null
null
ord-a502aa411b624e959a294d1ade8139de
[ClH:1].[NH2:2][CH:3]([C:9]([OH:11])=[O:10])[CH2:4][CH2:5][CH2:6][CH2:7][NH2:8].S([O-])([O-])(=O)=O.[NH4+].[NH4+].P([O-])(O)(O)=O.[K+].S([O-])([O-])(=O)=O.[Mg+2].Cl>>[ClH:1].[NH2:2][C@@H:3]([C:9]([OH:11])=[O:10])[CH2:4][CH2:5][CH2:6][CH2:7][NH2:8] |f:0.1,2.3.4,5.6,7.8,10.11|
S(=O)(=O)([O-])[O-].[Mg+2].Cl.NC(CCCCN)C(=O)O.S(=O)(=O)([O-])[O-].[NH4+].[NH4+].Cl.P(=O)(O)(O)[O-].[K+]
magnesium sulfate;DL-lysine monohydrochloride;ammonium sulfate;hydrochloric acid;potassium dihydrogen phosphate
0.0;0.0;0.0;0.0;0.0
mol;mol;mol;mol;mol
null
null
null
null
null
null
null
null
null
null
null
null
null
0.1667
Cl.N[C@H](CCCCN)C(=O)O
D-lysine monohydrochloride
5.8
g
null
ord-bea45d3f17ff4aeeb2836945fd80d389
[ClH:1].[NH2:2][CH:3]([C:9]([OH:11])=[O:10])[CH2:4][CH2:5][CH2:6][CH2:7][NH2:8].N[C@H](C(O)=O)CCCCN>>[ClH:1].[NH2:2][C@@H:3]([C:9]([OH:11])=[O:10])[CH2:4][CH2:5][CH2:6][CH2:7][NH2:8] |f:0.1,3.4|
Cl.NC(CCCCN)C(=O)O.N[C@@H](CCCCN)C(=O)O
DL-lysine monohydrochloride;L-lysine
0.0;0.0
mol;mol
null
null
null
null
null
null
null
null
null
null
null
null
null
0.1667
Cl.N[C@H](CCCCN)C(=O)O
D-lysine monohydrochloride
14.2
g
null
ord-9053e57f398646fcad52b73dfd0e8b51
[Br:1][C:2]1[C:3](=[O:10])[N:4]([CH3:9])[N:5]=[CH:6][C:7]=1Br.[CH3:11][O-:12].[Na+]>CO>[Br:1][C:2]1[C:3](=[O:10])[N:4]([CH3:9])[N:5]=[CH:6][C:7]=1[O:12][CH3:11] |f:1.2|
BrC=1C(N(N=CC1Br)C)=O.C[O-].[Na+].
4,5-Dibromo-2-methyl-3(2H)-pyridazinone;sodium methoxide;solution
20.0;0.0;0.0
g;mol;mol
CO.CO
methanol;methanol
0.0;200.0
mol;mL
null
null
null
null
null
null
null
null
23.0
3
BrC=1C(N(N=CC1OC)C)=O
desired product
17
g
null
ord-415b27028875405d86f41fbc30253639
Br[C:2]1[CH:3]=[C:4]([CH3:15])[C:5]2[S:10][CH2:9][CH2:8][C:7]([CH3:12])([CH3:11])[C:6]=2[C:13]=1[CH3:14].C([Li])CCC.CN(C)[CH:23]=[O:24].Cl>C(OCC)C>[CH3:11][C:7]1([CH3:12])[C:6]2[C:13]([CH3:14])=[C:2]([CH:23]=[O:24])[CH:3]=[C:4]([CH3:15])[C:5]=2[S:10][CH2:9][CH2:8]1
Cl.C(CCC)[Li].BrC=1C=C(C2=C(C(CCS2)(C)C)C1C)C.CN(C=O)C
Hydrochloric acid;n-butyllithium;6-Bromo-3,4-dihydro-4,4,5,8-tetramethyl-2H-1-benzothiopyran;Dimethylformamide
100.0;42.0;19.8;16.0
mL;mL;g;mL
C(C)OCC
diethyl ether
350.0
mL
null
null
null
null
null
null
null
null
ambient
1
CC1(CCSC2=C1C(=C(C=C2C)C=O)C)C
desired compound
7.7
g
null
ord-bbaa547034cb4578bce2648d1c091a1f
[CH3:1][S-:2].[Na+].[Cl:4][C:5]1[CH:10]=[C:9](Cl)[N:8]=[C:7]([O:12][CH2:13][C:14]2[CH:19]=[CH:18][CH:17]=[CH:16][CH:15]=2)[N:6]=1>C1COCC1>[Cl:4][C:5]1[CH:10]=[C:9]([S:2][CH3:1])[N:8]=[C:7]([O:12][CH2:13][C:14]2[CH:19]=[CH:18][CH:17]=[CH:16][CH:15]=2)[N:6]=1 |f:0.1|
C[S-].[Na+].ClC1=NC(=NC(=C1)Cl)OCC1=CC=CC=C1
sodium thiomethoxide;4,6-dichloro-2-(phenylmethoxy)pyrimidine
2.75;0.0
g;mol
C1CCOC1
THF
0.0
mol
null
null
null
null
null
null
null
null
null
null
ClC1=NC(=NC(=C1)SC)OCC1=CC=CC=C1
4-chloro-6-methylthio-2-(phenylmethoxy)pyrimidine
null
null
null
ord-3d58caaef3e54ab9bff64df1e59b26f5
[F:1][C:2]([F:11])([F:10])[C:3]1[CH:4]=[C:5]([OH:9])[CH:6]=[CH:7][CH:8]=1.[H-].[Na+].Cl[C:15]1[CH:20]=[CH:19][N:18]=[C:17]([S:21][CH3:22])[N:16]=1>C1COCC1>[CH3:22][S:21][C:17]1[N:18]=[C:19]([O:9][C:5]2[CH:6]=[CH:7][CH:8]=[C:3]([C:2]([F:10])([F:11])[F:1])[CH:4]=2)[CH:20]=[CH:15][N:16]=1 |f:1.2|
[H-].[Na+].ClC1=NC(=NC=C1)SC.FC(C=1C=C(C=CC1)O)(F)F
NaH;4-chloro-2-(methylthio)pyrimidine;3-(trifluoromethyl)phenol
1.12;0.0;4.54
g;mol;g
C1CCOC1
THF
0.0
mol
null
null
null
null
null
null
null
null
null
null
CSC1=NC=CC(=N1)OC1=CC(=CC=C1)C(F)(F)F
phenoxide
null
null
null
ord-0c41a886f892437a80e1ebfc69bc8999
[CH2:1]([OH:3])[CH3:2].[H-].[Na+].Cl[C:7]1[CH:12]=[C:11](Cl)[N:10]=[C:9]([S:14][CH3:15])[N:8]=1.[F:16][C:17]([F:26])([F:25])[C:18]1[CH:19]=[C:20]([OH:24])[CH:21]=[CH:22][CH:23]=1>C1COCC1.CN(C=O)C>[CH2:1]([O:3][C:7]1[CH:12]=[C:11]([O:24][C:20]2[CH:21]=[CH:22][CH:23]=[C:18]([C:17]([F:16])([F:25])[F:26])[CH:19]=2)[N:10]=[...
C(C)O.[H-].[Na+].FC(C=1C=C(C=CC1)O)(F)F.[H-].[Na+].ClC1=NC(=NC(=C1)Cl)SC
Ethanol;NaH;m-trifluoromethyl-phenol;NaH;4,6-dichloro-2-methylthiopyrimidine
1.18;1.02;6.23;1.54;0.0
g;g;g;g;mol
C1CCOC1.CN(C)C=O
THF;DMF
0.0;0.0
mol;mol
null
null
null
null
null
null
null
null
ambient
0.5
C(C)OC1=NC(=NC(=C1)OC1=CC(=CC=C1)C(F)(F)F)SC
4-ethoxy-2-methylthio-6-[3-(trifluoromethyl)phenoxy]pyrimidine
null
null
null
ord-779700042b074f55b42f3a2202e7c555
[F:1][C:2]([F:11])([F:10])[C:3]1[CH:4]=[C:5]([OH:9])[CH:6]=[CH:7][CH:8]=1.[H-].[Na+].Cl[C:15]1[CH:20]=[C:19]([C:21]([F:24])([F:23])[F:22])[N:18]=[C:17]([S:25][CH3:26])[N:16]=1>C1COCC1>[CH3:26][S:25][C:17]1[N:18]=[C:19]([C:21]([F:24])([F:22])[F:23])[CH:20]=[C:15]([O:9][C:5]2[CH:6]=[CH:7][CH:8]=[C:3]([C:2]([F:10])([F:11]...
FC(C=1C=C(C=CC1)O)(F)F.[H-].[Na+].ClC1=NC(=NC(=C1)C(F)(F)F)SC
m-(Trifluoromethyl)phenol;NaH;4-chloro-2-methylthio-6-(trifluoromethyl)pyrimidine
1.06;0.26;0.0
g;g;mol
C1CCOC1
THF
0.0
mol
null
null
null
null
null
null
null
null
null
null
CSC1=NC(=CC(=N1)C(F)(F)F)OC1=CC(=CC=C1)C(F)(F)F
2-methylthio-4-trifluoromethyl-6-[3-(trifluoromethyl)phenoxy]pyrimidine
null
null
null
ord-3df2c010cc0541928156900e8959ed27
[F:1][C:2]([F:11])([F:10])[C:3]1[CH:4]=[C:5]([OH:9])[CH:6]=[CH:7][CH:8]=1.[H-].[Na+].[Br:14][C:15]1[CH:20]=[C:19](Br)[N:18]=[C:17]([S:22][CH3:23])[N:16]=1>C1COCC1>[Br:14][C:15]1[CH:20]=[C:19]([O:9][C:5]2[CH:6]=[CH:7][CH:8]=[C:3]([C:2]([F:10])([F:11])[F:1])[CH:4]=2)[N:18]=[C:17]([S:22][CH3:23])[N:16]=1 |f:1.2|
FC(C=1C=C(C=CC1)O)(F)F.[H-].[Na+].BrC1=NC(=NC(=C1)Br)SC
m-(trifluoromethyl)phenol;NaH;4,6-dibromo-2-(methylthio)pyrimidine
1.3;0.32;0.0
g;g;mol
C1CCOC1
THF
0.0
mol
null
null
null
null
null
null
null
null
null
null
BrC1=NC(=NC(=C1)OC1=CC(=CC=C1)C(F)(F)F)SC
phenoxide
null
null
null
ord-1754134a9e1b4ab5a610540df5e81abc
[CH3:1][C:2]1[CH:3]=[CH:4][CH:5]=[C:6]([NH2:11])[C:7]=1[C:8]([OH:10])=[O:9].[OH-].[Na+].[C:14](OC(=O)C)(=[O:16])[CH3:15].Cl>O>[CH3:1][C:2]1[CH:3]=[CH:4][CH:5]=[C:6]([NH:11][C:14](=[O:16])[CH3:15])[C:7]=1[C:8]([OH:10])=[O:9] |f:1.2|
Cl.CC=1C=CC=C(C1C(=O)O)N.[OH-].[Na+].C(C)(=O)OC(C)=O
HCl;6-methylanthranilic acid;NaOH;acetic anhydride
0.0;90.6;24.8;63.4
mol;g;g;g
O
water
500.0
mL
null
null
null
null
null
null
null
null
null
1
CC1=C(C(=O)O)C(=CC=C1)NC(C)=O
2-Methyl-6-acetamidobenzoic acid
null
null
null
ord-036dc1bd98f447088e22557193b51876
[N+:1]([O-:4])(O)=[O:2].[CH3:5][C:6]1[CH:14]=[CH:13][CH:12]=[C:11]([NH:15][C:16](=[O:18])[CH3:17])[C:7]=1[C:8]([OH:10])=[O:9]>O>[CH3:5][C:6]1[C:14]([N+:1]([O-:4])=[O:2])=[CH:13][CH:12]=[C:11]([NH:15][C:16](=[O:18])[CH3:17])[C:7]=1[C:8]([OH:10])=[O:9]
[N+](=O)(O)[O-].CC1=C(C(=O)O)C(=CC=C1)NC(C)=O.
nitric acid;2-methyl-6-acetamidobenzoic acid;ice
271.0;106.0;540.0
mL;g;g
O
water
270.0
mL
null
null
null
null
null
null
null
null
10.0
1
CC1=C(C(=O)O)C(=CC=C1[N+](=O)[O-])NC(C)=O
2-Methyl-3-nitro-6-acetamidobenzoic acid
null
null
null
ord-36a2a540166a44e2ae3ef4e91516ef3a
[CH3:1][C:2]1[C:10]([N+:11]([O-:13])=[O:12])=[CH:9][CH:8]=[C:7]([NH:14]C(=O)C)[C:3]=1[C:4]([OH:6])=[O:5].Cl>[OH-].[Na+]>[CH3:1][C:2]1[C:10]([N+:11]([O-:13])=[O:12])=[CH:9][CH:8]=[C:7]([NH2:14])[C:3]=1[C:4]([OH:6])=[O:5] |f:2.3|
CC1=C(C(=O)O)C(=CC=C1[N+](=O)[O-])NC(C)=O.Cl
2-methyl-3-nitro-6-acetamidobenzoic acid;HCl
75.6;425.0
g;mL
[OH-].[Na+]
NaOH
450.0
mL
null
null
null
null
null
null
null
null
95.0
1
CC1=C(C(=O)O)C(=CC=C1[N+](=O)[O-])N
2-Methyl-3-nitro-6-aminobenzoic acid
null
null
null
ord-24a3ddd0c4da4019a874af8b0e5c2e2d
[CH3:1][C:2]1[C:10]([N+:11]([O-:13])=[O:12])=[CH:9][CH:8]=[C:7]([NH2:14])[C:3]=1[C:4]([OH:6])=[O:5].[C:15](=O)([O-])O.[Na+].C(=O)=O.S(OC)(OC)(=O)=O.[Na]>CC(C)=O.O>[CH3:1][C:2]1[C:10]([N+:11]([O-:13])=[O:12])=[CH:9][CH:8]=[C:7]([NH2:14])[C:3]=1[C:4]([O:6][CH3:15])=[O:5] |f:1.2,^1:29|
C(=O)=O.S(=O)(=O)(OC)OC.[Na].CC1=C(C(=O)O)C(=CC=C1[N+](=O)[O-])N.C(O)([O-])=O.[Na+].CC1=C(C(=O)O)C(=CC=C1[N+](=O)[O-])N
CO2;dimethyl sulfate;sodium;2-methyl-3-nitro-6-aminobenzoic acid;sodium hydrogen carbonate;2-methyl-3-nitro-6-aminobenzoic acid
0.0;35.3;0.0;0.0;43.0;49.7
mol;g;mol;mol;g;g
CC(=O)C.O.CC(=O)C
acetone;water;acetone
0.0;1800.0;380.0
mol;mL;mL
null
null
null
null
null
null
null
null
null
null
CC1=C(C(=O)OC)C(=CC=C1[N+](=O)[O-])N
Methyl 2-methyl-3-nitro-6-aminobenzoate
null
null
null
ord-9750ebabdd9f4e72aa5a98408ce4247f
[NH3:1].O.C[O:4][C:5]([C:7]1[C:12]([CH3:13])=[C:11]([N+:14]([O-:16])=[O:15])[CH:10]=[CH:9][C:8]=1[S:17](Cl)(=[O:19])=[O:18])=O>O1CCCC1>[CH3:13][C:12]1[C:11]([N+:14]([O-:16])=[O:15])=[CH:10][CH:9]=[C:8]2[C:7]=1[C:5](=[O:4])[NH:1][S:17]2(=[O:19])=[O:18]
N.O.COC(=O)C1=C(C=CC(=C1C)[N+](=O)[O-])S(=O)(=O)Cl
ammonia;water;2-methoxycarbonyl-3-methyl-4-nitrobenzenesulfonyl chloride
104.0;100.0;48.7
mL;mL;g
O1CCCC1
tetrahydrofuran
70.0
mL
null
null
null
null
null
null
null
null
25.0
3
CC1=C2C(NS(=O)(=O)C2=CC=C1[N+](=O)[O-])=O
4-Methyl-5-nitrosaccharin
null
null
null
ord-67ec3bcdf85a4cd095b46cc07afa68ed
[CH3:1][C:2]1[C:12]([N+:13]([O-])=O)=[CH:11][CH:10]=[C:9]2[C:3]=1[C:4](=[O:16])[NH:5][S:6]2(=[O:8])=[O:7].[H][H]>O.[Pd]>[CH3:1][C:2]1[C:12]([NH2:13])=[CH:11][CH:10]=[C:9]2[C:3]=1[C:4](=[O:16])[NH:5][S:6]2(=[O:8])=[O:7]
CC1=C2C(NS(=O)(=O)C2=CC=C1[N+](=O)[O-])=O.[H][H]
4-methyl-5-nitrosaccharin;Hydrogen
33.6;0.0
g;mol
O
water
1200.0
mL
[Pd]
Pd/C
5.0
g
null
null
null
null
45.0
null
CC1=C2C(NS(=O)(=O)C2=CC=C1N)=O
4-Methyl-5-aminosaccharin
null
null
null
ord-64895c5b03224120a7cbd0bc650559fc
Cl.[CH3:2][C:3]1[C:13](N)=[CH:12][CH:11]=[C:10]2[C:4]=1[C:5](=[O:15])[NH:6][S:7]2(=[O:9])=[O:8].N([O-])=O.[Na+].[I-:20].[K+]>O.C(O)(=O)C>[CH3:2][C:3]1[C:13]([I:20])=[CH:12][CH:11]=[C:10]2[C:4]=1[C:5](=[O:15])[NH:6][S:7]2(=[O:9])=[O:8] |f:2.3,4.5|
.Cl.[I-].[K+].CC1=C2C(NS(=O)(=O)C2=CC=C1N)=O.N(=O)[O-].[Na+]
diazonium salt;HCl;potassium iodide;4-methyl-5-aminosaccharin;sodium nitrite
0.0;40.0;19.1;23.4;7.9
mol;mL;g;g;g
O.C(C)(=O)O.O
water;acetic acid;water
160.0;205.0;170.0
mL;mL;mL
null
null
null
null
null
null
null
null
50.0
null
CC1=C2C(NS(=O)(=O)C2=CC=C1I)=O
iodine
null
null
null
ord-5bfe10bbdded406ba8ad3cc28a98a377
[OH-].[Na+].[C:3]([CH:11]([CH2:17][C:18]#[CH:19])[C:12](OCC)=[O:13])(=[O:10])[C:4]1[CH:9]=[CH:8][CH:7]=[CH:6][CH:5]=1.[CH3:20][NH:21]O.Cl>O.CO.CCOCC>[CH3:20][N:21]1[C:12](=[O:13])[CH:11]([CH2:17][C:18]#[CH:19])[CH:3]([C:4]2[CH:9]=[CH:8][CH:7]=[CH:6][CH:5]=2)[O:10]1 |f:0.1|
[OH-].[Na+].CNO.C(C1=CC=CC=C1)(=O)C(C(=O)OCC)CC#C.[OH-].[Na+].Cl
NaOH;N-methylhydroxylamine;ethyl α-benzoyl-α-propargylacetate;NaOH;HCl
0.54;1.02;1.42;0.28;0.0
g;g;g;g;mol
O.CO.CCOCC.O.CO
water;methanol;ether;water;methanol
1.5;2.0;150.0;3.0;7.0
mL;mL;mL;mL;mL
null
null
null
null
null
null
null
null
-30.0
0.1667
CN1OC(C(C1=O)CC#C)C1=CC=CC=C1
2-methyl-5-phenyl-4-propargylisoxazolin-3-one
0.46
g
34.5
ord-c014829738084401b0a152f2e7cdf4bb
[CH3:1][C:2]([NH:5][S:6]([C:9]1[CH:13]=[CH:12][NH:11][CH:10]=1)(=[O:8])=[O:7])([CH3:4])[CH3:3].CI.[CH3:16]C(C)([O-])C.[K+]>CN(C)C=O.C(OCC)(=O)C>[CH3:4][C:2]([NH:5][S:6]([C:9]1[CH:13]=[CH:12][N:11]([CH3:16])[CH:10]=1)(=[O:8])=[O:7])([CH3:1])[CH3:3] |f:2.3|
CC(C)(C)NS(=O)(=O)C1=CNC=C1.CI.CC(C)([O-])C.[K+]
N-(1,1-dimethylethyl)-1H-pyrrole-3 -sulfonamide;methyl iodide;potassium t-butoxide
9.0;3.2;5.43
g;mL;g
CN(C=O)C.C(C)(=O)OCC
N,N-dimethylforamide;ethyl acetate
90.0;0.0
mL;mol
null
null
null
null
null
null
null
null
60.0
2
CC(C)(C)NS(=O)(=O)C1=CN(C=C1)C
N-(1,1-Dimethylethyl)-1-methyl-1H-pyrrole-3-sulfonamide
null
null
null
ord-a32d55e896f94ee09bb5a13e0797fb99
[CH3:1][C:2]([NH:5][S:6]([C:9]1[CH:13]=[CH:12][N:11]([CH3:14])[CH:10]=1)(=[O:8])=[O:7])([CH3:4])[CH3:3].C([Li])CCC.Cl[C:21]([O:23][CH3:24])=[O:22].Cl>C1COCC1.[Au]>[CH3:4][C:2]([NH:5][S:6]([C:9]1[CH:13]=[CH:12][N:11]([CH3:14])[C:10]=1[C:21]([O:23][CH3:24])=[O:22])(=[O:8])=[O:7])([CH3:1])[CH3:3]
CC(C)(C)NS(=O)(=O)C1=CN(C=C1)C.ClC(=O)OC.Cl.C(CCC)[Li]
N-(1,1-dimethylethyl)-1-methyl-1H-pyrrole-3-sulfonamide;Methyl chloroformate;HCl;n-butyllithium
4.62;0.37;0.0;4.1
mol;mL;mol;mL
C1CCOC1.
THF;hexanes
150.0;0.0
mL;mol
[Au].[Au]
gold;gold
0.0;0.0
mol;mol
null
null
null
null
-78.0
0.5
CC(C)(C)NS(=O)(=O)C1=C(N(C=C1)C)C(=O)OC
title compound
null
null
null
ord-476d1b77fb1f4defbab1a8181428d9b8
[CH3:1][C:2]([NH:5][S:6]([C:9]1[CH:13]=[CH:12][N:11]([CH3:14])[CH:10]=1)(=[O:8])=[O:7])([CH3:4])[CH3:3].C([Li])CCC.Cl[C:21]([O:23][CH3:24])=[O:22].Cl>C1COCC1.[Au]>[CH3:4][C:2]([NH:5][S:6]([C:9]1[CH:13]=[CH:12][N:11]([CH3:14])[C:10]=1[C:21]([O:23][CH3:24])=[O:22])(=[O:8])=[O:7])([CH3:1])[CH3:3]
Cl.CC(C)(C)NS(=O)(=O)C1=CN(C=C1)C.C(CCC)[Li].ClC(=O)OC
HCl;N-(1,1-dimethylethyl)-1-methyl-1H-pyrrole-3-sulfonamide;n-butyllithium;methyl chloroformate
0.0;5.0;20.0;1.87
mol;g;mL;mL
C1CCOC1.
THF;hexanes
150.0;0.0
mL;mol
[Au].[Au]
gold;gold
0.0;0.0
mol;mol
null
null
null
null
-78.0
0.5
CC(C)(C)NS(=O)(=O)C1=C(N(C=C1)C)C(=O)OC
title compound
3.53
g
55.9
ord-740719404b1e4815a4a77e34574adcd7
CC([NH:5][S:6]([C:9]1[CH:13]=[CH:12][N:11]([CH3:14])[C:10]=1[C:15]([O:17][CH3:18])=[O:16])(=[O:8])=[O:7])(C)C.FC(F)(F)C(O)=O>[Au].C(Cl)Cl>[NH2:5][S:6]([C:9]1[CH:13]=[CH:12][N:11]([CH3:14])[C:10]=1[C:15]([O:17][CH3:18])=[O:16])(=[O:8])=[O:7]
CC(C)(C)NS(=O)(=O)C1=C(N(C=C1)C)C(=O)OC.FC(C(=O)O)(F)F
methyl 3-[[(1,1-dimethylethyl)amino]-sulfonyl]-1-methyl-1H-pyrrole-2-carboxylate;trifluoroacetic acid
3.53;80.0
g;mL
C(Cl)Cl
methylene chloride
0.0
mol
[Au]
gold
0.0
mol
null
null
null
null
null
null
NS(=O)(=O)C1=C(N(C=C1)C)C(=O)OC
title compound
null
null
null
ord-ec291f168e3d4ab6bc17d0209ef33361
[CH3:1][C:2]([NH:5][S:6]([C:9]1[CH:13]=[CH:12][N:11]([CH3:14])[CH:10]=1)(=[O:8])=[O:7])([CH3:4])[CH3:3].C([Li])CCC.[CH3:20][S:21]SC.Cl>C1COCC1>[CH3:4][C:2]([NH:5][S:6]([C:9]1[CH:13]=[CH:12][N:11]([CH3:14])[C:10]=1[S:21][CH3:20])(=[O:8])=[O:7])([CH3:1])[CH3:3]
Cl.C(CCC)[Li].CC(C)(C)NS(=O)(=O)C1=CN(C=C1)C.CSSC
HCl;n-butyllithium;N-(1,1-dimethylethyl)-1-methyl-1H-pyrrole-3-sulfonamide;dimethyldisulfide
0.0;25.52;6.48;2.97
mol;mL;g;mL
.C1CCOC1
hexanes;THF
0.0;150.0
mol;mL
null
null
null
null
null
null
null
null
-78.0
0.5
CC(C)(C)NS(=O)(=O)C1=C(N(C=C1)C)SC
title compound
4.63
g
58.8
ord-ee7d05a9975a483f9332d56b8ce092a7
CC([NH:5][S:6]([C:9]1[CH:13]=[CH:12][N:11]([CH3:14])[C:10]=1[S:15][CH3:16])(=[O:8])=[O:7])(C)C.FC(F)(F)C(O)=O>C(Cl)Cl>[CH3:14][N:11]1[CH:12]=[CH:13][C:9]([S:6]([NH2:5])(=[O:7])=[O:8])=[C:10]1[S:15][CH3:16]
CC(C)(C)NS(=O)(=O)C1=C(N(C=C1)C)SC.FC(C(=O)O)(F)F
N-(1,1-dimethylethyl)-1-methyl-2-(methylthio)-1H-pyrrole-3-sulfonamide;trifluoroacetic acid
4.63;50.0
g;mL
C(Cl)Cl
methylene chloride
50.0
mL
null
null
null
null
null
null
null
null
ambient
16
CN1C(=C(C=C1)S(=O)(=O)N)SC
title compound
2.9
g
79.6
ord-0d425205828e434aa8465064fdc60f2d
[CH3:1][C:2]([NH:5][S:6]([C:9]1[CH:13]=[CH:12][N:11]([CH3:14])[CH:10]=1)(=[O:8])=[O:7])([CH3:4])[CH3:3].C([Li])CCC.[Br:20]Br.Cl>C(OCC)C>[Br:20][C:10]1[N:11]([CH3:14])[CH:12]=[CH:13][C:9]=1[S:6]([NH:5][C:2]([CH3:1])([CH3:3])[CH3:4])(=[O:8])=[O:7]
Cl.CC(C)(C)NS(=O)(=O)C1=CN(C=C1)C.C(CCC)[Li].BrBr
HCl;N-(1,1-dimethylethyl)-1-methyl-1H-pyrrole-3-sulfonamide;n-butyllithium;bromine
0.0;8.85;36.0;2.2
mol;g;mL;mL
C(C)OCC.
diethyl ether;hexanes
200.0;0.0
mL;mol
null
null
null
null
null
null
null
null
-78.0
0.25
BrC=1N(C=CC1S(=O)(=O)NC(C)(C)C)C
title compound
7.11
g
58.7
ord-952e75b6acac43568991fc07fe11133a
[Br:1][C:2]1[N:3]([CH3:15])[CH:4]=[CH:5][C:6]=1[S:7]([NH:10]C(C)(C)C)(=[O:9])=[O:8].C(O)(C(F)(F)F)=O>C(Cl)Cl>[Br:1][C:2]1[N:3]([CH3:15])[CH:4]=[CH:5][C:6]=1[S:7]([NH2:10])(=[O:8])=[O:9]
BrC=1N(C=CC1S(=O)(=O)NC(C)(C)C)C.C(=O)(C(F)(F)F)O
2-bromo-N-(1,1-dimethylethyl)-1-methyl-1H-pyrrole-3-sulfonamide;TFA
7.11;50.0
g;mL
C(Cl)Cl
methylene chloride
50.0
mL
null
null
null
null
null
null
null
null
ambient
16
BrC=1N(C=CC1S(=O)(=O)N)C
title compound
1.23
g
21.4
ord-1689ec83ac2b4e2e9bc10359a96a617b
[CH3:1][C:2]([NH:5][S:6]([C:9]1[CH:13]=[CH:12][N:11]([CH3:14])[CH:10]=1)(=[O:8])=[O:7])([CH3:4])[CH3:3].CN(C)[CH:17]=[O:18].Cl>C1COCC1>[CH3:4][C:2]([NH:5][S:6]([C:9]1[CH:13]=[CH:12][N:11]([CH3:14])[C:10]=1[CH:17]=[O:18])(=[O:8])=[O:7])([CH3:1])[CH3:3]
CC(C)(C)NS(=O)(=O)C1=CN(C=C1)C.CN(C=O)C.Cl
N-(1,1-dimethylethyl)-1-methyl-1H-pyrrole-3-sulfonamide;N,N-dimethylformamide;HCl
12.96;4.64;0.0
g;mL;mol
C1CCOC1.
THF;hexanes
300.0;0.0
mL;mol
null
null
null
null
null
null
null
null
-78.0
0.5
CC(C)(C)NS(=O)(=O)C1=C(N(C=C1)C)C=O
title compound
5.72
g
39
ord-3b75f1f1033143b794c5a9db7bc6a994
Cl.[CH3:2][O:3][NH2:4].C([O-])(=O)C.[Na+].[CH3:10][C:11]([NH:14][S:15]([C:18]1[CH:22]=[CH:21][N:20](C)[C:19]=1[CH:24]=O)(=[O:17])=[O:16])([CH3:13])[CH3:12].O>CO>[CH3:13][C:11]([NH:14][S:15]([C:18]1[CH:22]=[CH:21][NH:20][C:19]=1[CH:24]=[N:4][O:3][CH3:2])(=[O:17])=[O:16])([CH3:10])[CH3:12] |f:0.1,2.3|
O.C(C)(=O)[O-].[Na+].Cl.CON.CC(C)(C)NS(=O)(=O)C1=C(N(C=C1)C)C=O
water;sodium acetate;methoxyamine hydrochloride;N-(1,1-dimethylethyl)-2-formyl-1-methyl-1H-pyrrole-3-sulfonamide
500.0;3.84;3.91;5.72
mL;g;g;g
CO
methanol
60.0
mL
null
null
null
null
null
null
null
null
ambient
null
CC(C)(C)NS(=O)(=O)C1=C(NC=C1)C=NOC
title compound
5.74
g
96.2
ord-0d13730de7524a88a677102766469c81
CC([NH:5][S:6]([C:9]1[CH:13]=[CH:12][NH:11][C:10]=1[CH:14]=[N:15][O:16][CH3:17])(=[O:8])=[O:7])(C)C.[C:18](O)(C(F)(F)F)=O>C(Cl)Cl>[CH3:17][O:16][N:15]=[CH:14][C:10]1[N:11]([CH3:18])[CH:12]=[CH:13][C:9]=1[S:6]([NH2:5])(=[O:7])=[O:8]
CC(C)(C)NS(=O)(=O)C1=C(NC=C1)C=NOC.C(=O)(C(F)(F)F)O
N-(1,1-dimethylethyl)-2-[(methoxyimino)-methyl]-1H-pyrrole-3-sulfonamide;TFA
5.74;75.0
g;mL
C(Cl)Cl
methylene chloride
75.0
mL
null
null
null
null
null
null
null
null
ambient
16
CON=CC=1N(C=CC1S(=O)(=O)N)C
title compound
3.49
g
null
ord-00887c12283747658f3f8ff3622cc7d7
CC([NH:5][S:6]([C:9]1[CH:13]=[CH:12][N:11]([CH3:14])[CH:10]=1)(=[O:8])=[O:7])(C)C.C([Li])[CH2:16][CH2:17][CH3:18].[S:20](=[O:22])=[O:21].Cl[N:24]1[C:28](=O)CC[C:25]1=O.O1CCC[CH2:32]1>>[CH3:32][C:17]([C:13]1[C:9]([S:6]([NH2:5])(=[O:7])=[O:8])=[C:10]([S:20]([N:24]([CH3:28])[CH3:25])(=[O:22])=[O:21])[N:11]([CH3:14])[CH:12...
ClN1C(CCC1=O)=O.C(CCC)[Li].CC(C)(C)NS(=O)(=O)C1=CN(C=C1)C.O1CCCC1..S(=O)=O
N-chlorosuccinimide;n-butyllithium;N-(1,1-dimethylethyl)-1-methyl-1H-pyrrole-3-sulfonamide;tetrahydrofuran;dimethylimine;sulfur dioxide
0.031;0.0615;6.48;150.0;0.075;0.0
mol;mol;g;mL;mol;mol
null
hexanes
0.0
mol
null
null
null
null
null
null
null
null
ambient
1
CC(C)(C)C=1C(=C(N(C1)C)S(=O)(=O)N(C)C)S(=O)(=O)N
title compound
6.95
g
null
ord-bce13e6e0f2b4556bf712059577ecdcd
CC([C:5]1[C:6]([S:17]([NH2:20])(=[O:19])=[O:18])=[C:7]([S:11]([N:14]([CH3:16])[CH3:15])(=[O:13])=[O:12])[N:8]([CH3:10])[CH:9]=1)(C)C.C(O)(C(F)(F)F)=O>C(Cl)Cl>[CH3:15][N:14]([CH3:16])[S:11]([C:7]1[N:8]([CH3:10])[CH:9]=[CH:5][C:6]=1[S:17]([NH2:20])(=[O:19])=[O:18])(=[O:12])=[O:13]
CC(C)(C)C=1C(=C(N(C1)C)S(=O)(=O)N(C)C)S(=O)(=O)N.C(=O)(C(F)(F)F)O
(1,1-dimethylethyl)-N2,N2,1-trimethyl-1H-pyrrole-2,3-disulfonamide;TFA
0.0;75.0
mol;mL
C(Cl)Cl
methylene chloride
75.0
mL
null
null
null
null
null
null
null
null
ambient
16
CN(S(=O)(=O)C=1N(C=CC1S(=O)(=O)N)C)C
title compound
4.52
g
null
ord-acf44331951a4df6acd00502ec327265
[CH3:1][C:2]([NH:5][S:6]([C:9]1[CH:13]=[CH:12][N:11]([CH3:14])[CH:10]=1)(=[O:8])=[O:7])([CH3:4])[CH3:3].C([Li])CCC.[CH3:20][N:21]([CH3:25])[C:22](Cl)=[O:23].[Cl-].[NH4+].Cl>C1COCC1>[CH3:4][C:2]([NH:5][S:6]([C:9]1[CH:13]=[CH:12][N:11]([CH3:14])[C:10]=1[C:22]([N:21]([CH3:25])[CH3:20])=[O:23])(=[O:8])=[O:7])([CH3:1])[CH3:...
[Cl-].[NH4+].C(CCC)[Li].CC(C)(C)NS(=O)(=O)C1=CN(C=C1)C.CN(C(=O)Cl)C.Cl
ammonium chloride;n-butyllithium;N-(1,1-dimethylethyl)-1-methyl-1H-pyrrole-3-sulfonamide;N,N-dimethylcarbamyl chloride;HCl
60.0;25.0;6.48;3.1;30.0
mL;mL;g;mL;mL
.C1CCOC1.C1CCOC1
hexanes;THF;THF
0.0;150.0;10.0
mol;mL;mL
null
null
null
null
null
null
null
null
-78.0
0.5
CC(C)(C)NS(=O)(=O)C1=C(N(C=C1)C)C(=O)N(C)C
title compound
4.33
g
50.2
ord-4d0fbf7c4db24ef2820d2d87a9754e6c
CC([NH:5][S:6]([C:9]1[CH:13]=[CH:12][N:11]([CH3:14])[C:10]=1[C:15]([N:17]([CH3:19])[CH3:18])=[O:16])(=[O:8])=[O:7])(C)C.C(O)(C(F)(F)F)=O>C(Cl)Cl>[NH2:5][S:6]([C:9]1[CH:13]=[CH:12][N:11]([CH3:14])[C:10]=1[C:15]([N:17]([CH3:19])[CH3:18])=[O:16])(=[O:8])=[O:7]
CC(C)(C)NS(=O)(=O)C1=C(N(C=C1)C)C(=O)N(C)C.C(=O)(C(F)(F)F)O
3-[[(1,1-dimethylethyl)amino]sulfonyl]-N,N,1-trimethyl-1H-pyrrole-2-carboxamide;TFA
5.63;75.0
g;mL
C(Cl)Cl
methylene chloride
75.0
mL
null
null
null
null
null
null
null
null
ambient
16
NS(=O)(=O)C1=C(N(C=C1)C)C(=O)N(C)C
title compound
4.21
g
92.9
ord-66c80b7eb0654eda89cb0773db258c7f
[CH3:1][N:2]1[CH:6]=[CH:5][CH:4]=[CH:3]1.C([Li])CCC.[S:12](=[O:14])=[O:13].[C:15]([NH2:19])([CH3:18])([CH3:17])[CH3:16]>C1COCC1>[CH3:16][C:15]([NH:19][S:12]([C:3]1[N:2]([CH3:1])[CH:6]=[CH:5][CH:4]=1)(=[O:14])=[O:13])([CH3:18])[CH3:17]
S(=O)=O.C(CCC)[Li]..CN1C=CC=C1.C(C)(C)(C)N
sulfur dioxide;n-butyllithium;hexanes;N-methyl-pyrrole;t-butylamine
9.0;56.0;0.13;10.0;82.0
mL;mL;mol;g;mL
C1CCOC1
THF
120.0
mL
null
null
null
null
null
null
null
null
ambient
16
CC(C)(C)NS(=O)(=O)C=1N(C=CC1)C
title compound
7.4
g
28.5
ord-eaa9d1d720194b459594019c4118fe86
[CH3:1][C:2]([NH:5][S:6]([C:9]1[N:10]([CH3:14])[CH:11]=[CH:12][CH:13]=1)(=[O:8])=[O:7])([CH3:4])[CH3:3].C([Li])CCC.Cl[C:21]([O:23][CH3:24])=[O:22]>C1COCC1.C(OCC)(=O)C>[CH3:4][C:2]([NH:5][S:6]([C:9]1[N:10]([CH3:14])[CH:11]=[CH:12][C:13]=1[C:21]([O:23][CH3:24])=[O:22])(=[O:8])=[O:7])([CH3:1])[CH3:3]
ClC(=O)OC.CC(C)(C)NS(=O)(=O)C=1N(C=CC1)C.C(CCC)[Li]
methyl chloroformate;N-(1,1-dimethylethyl)-1-methyl-1H-pyrrole-2-sulfonamide;n-butyllithium
1.63;2.5;13.0
g;g;mL
C1CCOC1.C(C)(=O)OCC.C1CCOC1
THF;ethyl acetate;THF
6.0;200.0;50.0
mL;mL;mL
null
null
null
null
null
null
null
null
null
0.5
CC(C)(C)NS(=O)(=O)C=1N(C=CC1C(=O)OC)C
title compound
0.45
g
14.3
ord-a5a19d2e3ccc4cb7bff13f06f043ffc0
[NH2:1][S:2]([C:5]1[N:6]([CH3:14])[CH:7]=[CH:8][C:9]=1[C:10]([O:12][CH3:13])=[O:11])(=[O:4])=[O:3].C[O:16][C:17]1N=C(C)[N:20]=[C:19]([NH:24][C:25](=O)[O:26][C:27]2C=CC=CC=2)[N:18]=1.C1CCN2[C:37](=[N:38][CH2:39]CC2)CC1.Cl>C(#N)C.O>[CH3:27][O:26][C:25]1[N:24]=[C:19]([NH:18][C:17]([NH:1][S:2]([C:5]2[N:6]([CH3:14])[CH:7]=[...
Cl.NS(=O)(=O)C=1N(C=CC1C(=O)OC)C.COC1=NC(=NC(=N1)C)NC(OC1=CC=CC=C1)=O.C1CCC2=NCCCN2CC1
HCl;Methyl 2-(aminosulfonyl)-1-methyl-1H-pyrrole-3-carboxylate;phenyl (4-methoxy-6-methyl-1,3,5-triazin-2-yl)carbamate;DBU
0.5;0.1;0.13;0.075
mL;g;g;mL
O.C(C)#N
water;acetonitrile
15.0;2.0
mL;mL
null
null
null
null
null
null
null
null
ambient
0.5
COC=1N=C(NN(C1)C)NC(=O)NS(=O)(=O)C=1N(C=CC1C(=O)OC)C
oil
0.13
g
null
ord-819df65591774363bb9b76f5effae47b
[NH2:1][C:2]1[N:9]=[CH:8][CH:7]=[CH:6][C:3]=1[CH:4]=O.[CH3:10][C:11]([C:13]1[C:18]([F:19])=[CH:17][CH:16]=[CH:15][C:14]=1[F:20])=O.[OH-].[K+]>CO>[F:19][C:18]1[CH:17]=[CH:16][CH:15]=[C:14]([F:20])[C:13]=1[C:11]1[CH:10]=[CH:4][C:3]2[C:2](=[N:9][CH:8]=[CH:7][CH:6]=2)[N:1]=1 |f:2.3|
NC1=C(C=O)C=CC=N1.CC(=O)C1=C(C=CC=C1F)F.[OH-].[K+]
2-Aminonicotinaldehyde;2,6-difluoroacetophenone;KOH
2.44;3.28;3.0
g;g;mL
CO
MeOH
20.0
mL
null
null
null
null
null
null
null
null
null
null
FC1=C(C(=CC=C1)F)C1=NC2=NC=CC=C2C=C1
desired product
3.8
g
78.4
ord-6da8fccbc46d48d9b47085df7224e0c2
[NH2:1][C:2]1[N:9]=[CH:8][CH:7]=[CH:6][C:3]=1[CH:4]=O.[C:10]([C:13]1[S:14][CH:15]=[CH:16][N:17]=1)(=O)[CH3:11].[OH-].[K+]>CO>[S:14]1[CH:15]=[CH:16][N:17]=[C:13]1[C:10]1[CH:11]=[CH:4][C:3]2[C:2](=[N:9][CH:8]=[CH:7][CH:6]=2)[N:1]=1 |f:2.3|
NC1=C(C=O)C=CC=N1.C(C)(=O)C=1SC=CN1.[OH-].[K+]
2-Aminonicotinaldehyde;2-acetylthiazole;KOH
1.5;1.64;1.5
g;g;mL
CO
MeOH
12.0
mL
null
null
null
null
null
null
null
null
null
3
S1C(=NC=C1)C1=NC2=NC=CC=C2C=C1
desired product
1.22
g
46.5
ord-4fe7e7b0295444c08046dd75241f89c9
[OH:1][N:2]=[C:3]1[CH2:20][C@@:19]2([CH3:21])[C@@H:6]([CH2:7][CH2:8][C@@H:9]3[C@@H:18]2[CH2:17][CH2:16][C@@:14]2([CH3:15])[C@H:10]3[CH2:11][CH2:12][C@@H:13]2[OH:22])[CH2:5][C:4]1=O.[NH2:24][OH:25].Cl.[CH3:27][C:28]([O-:30])=O.[Na+].O>O>[C:28]([O:22][C@H:13]1[CH2:12][CH2:11][C@H:10]2[C@H:9]3[C@H:18]([CH2:17][CH2:16][C@:...
ON=C1C(C[C@@H]2CC[C@H]3[C@@H]4CC[C@@H]([C@@]4(C)CC[C@@H]3[C@]2(C1)C)O)=O.NO.Cl.CC(=O)[O-].[Na+].O
steroid;NH2OH.HCl;NaOAc H2O
0.0;0.0;0.0
mol;mol;mol
O
H2O
0.0
mol
null
null
null
null
null
null
null
null
ambient
null
C(C)(=O)O[C@@H]1[C@]2(C)[C@@H](CC1)[C@@H]1CC[C@H]3CC(C(C[C@]3(C)[C@H]1CC2)=NO)=NO
17β-Acetoxy-2,3-dihydroxyimino-5α-androstane
null
null
null
ord-9c0049ffd5bd4c2597bd8dc1da4f9125
[N+]([C:4]1[CH:11]=[CH:10][CH:9]=[C:8]([N+:12]([O-:14])=[O:13])[C:5]=1[C:6]#[N:7])([O-])=O.[C:15]1([SH:21])[CH:20]=[CH:19][CH:18]=[CH:17][CH:16]=1.C([O-])([O-])=O.[K+].[K+].N1C=CC=CC=1>CN(C=O)C.O>[N+:12]([C:8]1[CH:9]=[CH:10][CH:11]=[C:4]([S:21][C:15]2[CH:20]=[CH:19][CH:18]=[CH:17][CH:16]=2)[C:5]=1[C:6]#[N:7])([O-:14])=...
.[N+](=O)([O-])C1=C(C#N)C(=CC=C1)[N+](=O)[O-].C1(=CC=CC=C1)S.C(=O)([O-])[O-].[K+].[K+].N1=CC=CC=C1
ice water;2,6-dinitrobenzonitrile;thiophenol;K2CO3;Pyridine
0.0;2.0;1.06;1.44;0.0
mol;g;mL;g;mol
O.CN(C)C=O
H2O;DMF
100.0;50.0
mL;mL
null
null
null
null
null
null
null
null
null
0.5
[N+](=O)([O-])C1=C(C#N)C(=CC=C1)SC1=CC=CC=C1
2-nitro-6-(phenylthio)benzonitrile
1.94
g
75.7
ord-d850da0197e245649bff3ba3999f661f
O.[N+:2]([C:5]1[CH:12]=[CH:11][CH:10]=[C:9]([S:13][C:14]2[CH:19]=[CH:18][CH:17]=[CH:16][CH:15]=2)[C:6]=1[C:7]#[N:8])([O-])=O.Cl[Sn]Cl>COCCOCCOC.Cl>[NH2:2][C:5]1[CH:12]=[CH:11][CH:10]=[C:9]([S:13][C:14]2[CH:19]=[CH:18][CH:17]=[CH:16][CH:15]=2)[C:6]=1[C:7]#[N:8]
O.[N+](=O)([O-])C1=C(C#N)C(=CC=C1)SC1=CC=CC=C1.Cl[Sn]Cl
water;2-nitro-6-(phenylthio)benzonitrile;SnCl2
0.0;3.9;11.53
mol;g;g
COCCOCCOC.Cl
diglyme;HCl
85.0;35.0
mL;mL
null
null
null
null
null
null
null
null
null
null
NC1=C(C#N)C(=CC=C1)SC1=CC=CC=C1
2-Amino-6-(phenylthio)benzonitrile
null
null
null
ord-942c876021324f25bb9887685a674993
[N+]([C:4]1[CH:11]=[CH:10][CH:9]=[C:8]([N+:12]([O-:14])=[O:13])[C:5]=1[C:6]#[N:7])([O-])=O.C([O-])([O-])=O.[K+].[K+].[CH3:21][C:22]1[CH:23]=[C:24]([SH:29])[CH:25]=[C:26]([CH3:28])[CH:27]=1.O>CN(C=O)C>[CH3:21][C:22]1[CH:23]=[C:24]([S:29][C:4]2[CH:11]=[CH:10][CH:9]=[C:8]([N+:12]([O-:14])=[O:13])[C:5]=2[C:6]#[N:7])[CH:25]...
O.[N+](=O)([O-])C1=C(C#N)C(=CC=C1)[N+](=O)[O-].C(=O)([O-])[O-].[K+].[K+].CC=1C=C(C=C(C1)C)S
water;2,6-dinitrobenzonitrile;K2CO3;3,5-dimethylthiophenol
150.0;1.4;1.1;1.1
mL;g;g;g
CN(C)C=O.CN(C)C=O
DMF;DMF
10.0;10.0
mL;mL
null
null
null
null
null
null
null
null
0.0
null
CC=1C=C(C=C(C1)C)SC1=C(C#N)C(=CC=C1)[N+](=O)[O-]
2-[(3,5-dimethylphenyl)thio]-6-nitrobenzonitrile
1.64
g
73,011.2
ord-8c04216a28bb4609b9208e0d1a14c091
[CH3:1][C:2]1[CH:3]=[C:4]([S:9][C:10]2[CH:17]=[CH:16][CH:15]=[C:14]([N+:18]([O-])=O)[C:11]=2[C:12]#[N:13])[CH:5]=[C:6]([CH3:8])[CH:7]=1.[OH-].[Na+]>COCCOCCOC.Cl.O>[NH2:18][C:14]1[CH:15]=[CH:16][CH:17]=[C:10]([S:9][C:4]2[CH:3]=[C:2]([CH3:1])[CH:7]=[C:6]([CH3:8])[CH:5]=2)[C:11]=1[C:12]#[N:13] |f:1.2|
CC=1C=C(C=C(C1)C)SC1=C(C#N)C(=CC=C1)[N+](=O)[O-].[OH-].[Na+].
2-[(3,5-Dimethylphenyl)thio]-6-nitrobenzonitrile;NaOH;stannous chloride-2H2O
1.0;12.0;3.16
g;g;g
COCCOCCOC.O.Cl
diglyme;water;HCl
50.0;100.0;15.0
mL;mL;mL
null
null
null
null
null
null
null
null
null
null
NC1=C(C#N)C(=CC=C1)SC1=CC(=CC(=C1)C)C
2-amino-6-[(3,5-dimethylphenyl)thio]benzonitrile
0.57
g
64
ord-a610715a9a2049339b2b5008fb407eed
[F:1][C:2]1[CH:9]=[CH:8][CH:7]=[C:6]([S:10][C:11]2[CH:16]=[CH:15][CH:14]=[C:13]([O:17][CH3:18])[CH:12]=2)[C:3]=1[C:4]#[N:5].ClC1C=CC=C(C(OO)=[O:27])C=1.S(=O)(O)[O-].[Na+].[OH2:35]>>[F:1][C:2]1[CH:9]=[CH:8][CH:7]=[C:6]([S:10]([C:11]2[CH:16]=[CH:15][CH:14]=[C:13]([O:17][CH3:18])[CH:12]=2)(=[O:27])=[O:35])[C:3]=1[C:4]#[N:...
ClC1=CC(=CC=C1)C(=O)OO.S([O-])(O)=O.[Na+]..O.FC1=C(C#N)C(=CC=C1)SC1=CC(=CC=C1)OC.ClC1=CC(=CC=C1)C(=O)OO.
m-chloroperbenzoic acid;sodium bisulfite;resultant mixture;water;2-fluoro-6-[(3-methoxyphenyl)thio]benzonitrile;m-chloroperbenzoic acid;resultant mixture
0.29;0.0;0.0;0.0;2.0;2.93;0.0
g;mol;mol;mol;g;g;mol
null
null
null
null
null
null
null
null
null
null
null
null
null
null
FC1=C(C#N)C(=CC=C1)S(=O)(=O)C1=CC(=CC=C1)OC
2-Fluoro-6-[(3 -methoxyphenyl)sulfonyl]benzonitrile
null
null
null
ord-70d2fe8819214856a573963ea6b87bb1
F[C:2]1[CH:9]=[CH:8][CH:7]=[C:6]([S:10]([C:13]2[CH:18]=[CH:17][CH:16]=[C:15]([O:19][CH3:20])[CH:14]=2)(=[O:12])=[O:11])[C:3]=1[C:4]#[N:5].[NH4+:21].[OH-]>CO.CCO>[NH2:21][C:2]1[CH:9]=[CH:8][CH:7]=[C:6]([S:10]([C:13]2[CH:18]=[CH:17][CH:16]=[C:15]([O:19][CH3:20])[CH:14]=2)(=[O:12])=[O:11])[C:3]=1[C:4]#[N:5] |f:1.2,3.4|
FC1=C(C#N)C(=CC=C1)S(=O)(=O)C1=CC(=CC=C1)OC.[NH4+].[OH-]
2-fluoro-6-[(3-methoxyphenyl)sulfonyl]benzonitrile;NH4OH
0.7;20.0
g;mL
CO.CCO
MeOH EtOH
110.0
mL
null
null
null
null
null
null
null
null
130.0
null
NC1=C(C#N)C(=CC=C1)S(=O)(=O)C1=CC(=CC=C1)OC
2-Amino-6-[(3-methoxyphenyl)sulfonyl]benzonitrile
null
null
null
ord-f52f628e55bf48349560d5f7350120df
[F:1][C:2]1[CH:9]=[CH:8][CH:7]=[C:6]([S:10][C:11]2[CH:16]=[CH:15][CH:14]=[C:13]([O:17][CH3:18])[CH:12]=2)[C:3]=1[C:4]#[N:5].ClC1C=CC=C(C(OO)=[O:27])C=1.S(=O)(O)[O-].[Na+]>O>[F:1][C:2]1[CH:9]=[CH:8][CH:7]=[C:6]([S:10]([C:11]2[CH:16]=[CH:15][CH:14]=[C:13]([O:17][CH3:18])[CH:12]=2)=[O:27])[C:3]=1[C:4]#[N:5] |f:2.3|
ClC1=CC(=CC=C1)C(=O)OO.S([O-])(O)=O.[Na+]..FC1=C(C#N)C(=CC=C1)SC1=CC(=CC=C1)OC.ClC1=CC(=CC=C1)C(=O)OO.
m-chloroperbenzoic acid;sodium bisulfite;resultant mixture;2-fluoro-6-[(3-methoxyphenyl)thio]benzonitrile;m-chloroperbenzoic acid;resultant mixture
0.16;0.0;0.0;2.0;1.6;0.0
g;mol;mol;g;g;mol
O
water
0.0
mol
null
null
null
null
null
null
null
null
null
null
FC1=C(C#N)C(=CC=C1)S(=O)C1=CC(=CC=C1)OC
2-Fluoro-6-[(3-methoxyphenyl)sulfinyl]benzonitrile
null
null
null
ord-efbec65196ea4c25a91fe4f5f0f30b06
F[C:2]1[CH:9]=[CH:8][CH:7]=[C:6]([S:10]([C:12]2[CH:17]=[CH:16][CH:15]=[C:14]([O:18][CH3:19])[CH:13]=2)=[O:11])[C:3]=1[C:4]#[N:5].[NH4+:20].[OH-]>CO.CCO>[NH2:20][C:2]1[CH:9]=[CH:8][CH:7]=[C:6]([S:10]([C:12]2[CH:17]=[CH:16][CH:15]=[C:14]([O:18][CH3:19])[CH:13]=2)=[O:11])[C:3]=1[C:4]#[N:5] |f:1.2,3.4|
FC1=C(C#N)C(=CC=C1)S(=O)C1=CC(=CC=C1)OC.[NH4+].[OH-]
2-fluoro-6-[(3-methoxyphenyl)sulfinyl]benzonitrile;NH4OH
0.73;20.0
g;mL
CO.CCO
MeOH EtOH
65.0
mL
null
null
null
null
null
null
null
null
130.0
null
NC1=C(C#N)C(=CC=C1)S(=O)C1=CC(=CC=C1)OC
2-Amino-6-[(3-methoxyphenyl)sulfinyl]benzonitrile
null
null
null
ord-6ddfb59c25f34fe781aa3d4f78fc3efa
[CH3:1][C:2]1[CH:3]=[C:4]([S:9][C:10]2[CH:17]=[CH:16][CH:15]=[C:14]([F:18])[C:11]=2[C:12]#[N:13])[CH:5]=[C:6]([CH3:8])[CH:7]=1.[OH:19]OS([O-])=O.[K+]>CO.O>[CH3:8][C:6]1[CH:5]=[C:4]([S:9]([C:10]2[CH:17]=[CH:16][CH:15]=[C:14]([F:18])[C:11]=2[C:12]#[N:13])=[O:19])[CH:3]=[C:2]([CH3:1])[CH:7]=1 |f:1.2|
CC=1C=C(C=C(C1)C)SC1=C(C#N)C(=CC=C1)F.OOS(=O)[O-].[K+]
2-[(3,5-Dimethylphenyl)thio]-6-fluorobenzonitrile;OXONE
1.0;0.0
g;mol
O.CO
water;methanol
15.0;100.0
mL;mL
null
null
null
null
null
null
null
null
null
null
CC=1C=C(C=C(C1)C)S(=O)C1=C(C#N)C(=CC=C1)F
2-[(3,5-dimethylphenyl)sulfinyl]-6-fluorobenzonitrile
0.5
g
47
ord-3a63765ce57f4be88697886cd8f75569
[CH3:1][C:2]1[CH:3]=[C:4]([S:9][C:10]2[CH:17]=[CH:16][CH:15]=[C:14]([F:18])[C:11]=2[C:12]#[N:13])[CH:5]=[C:6]([CH3:8])[CH:7]=1.[OH:19]OS([O-])=O.[K+].[OH2:25]>CO>[CH3:8][C:6]1[CH:5]=[C:4]([S:9]([C:10]2[CH:17]=[CH:16][CH:15]=[C:14]([F:18])[C:11]=2[C:12]#[N:13])(=[O:19])=[O:25])[CH:3]=[C:2]([CH3:1])[CH:7]=1 |f:1.2|
O.OOS(=O)[O-].[K+].CC=1C=C(C=C(C1)C)SC1=C(C#N)C(=CC=C1)F.OOS(=O)[O-].[K+]
water;OXONE;2-[(3,5-Dimethylphenyl)thio]-6-fluorobenzonitrile;OXONE
30.0;0.0;1.0;0.0
mL;mol;g;mol
CO
methanol
100.0
mL
null
null
null
null
null
null
null
null
null
null
CC=1C=C(C=C(C1)C)S(=O)(=O)C1=C(C#N)C(=CC=C1)F
2-[(3,5-dimethylphenyl)sulfonyl]-6-fluorobenzonitrile
0.73
g
65
ord-ba9711ed922e47f3840d3a080575bd49
[CH3:1][C:2]1[CH:3]=[C:4]([S:9]([C:11]2[CH:18]=[CH:17][CH:16]=[C:15](F)[C:12]=2[C:13]#[N:14])=[O:10])[CH:5]=[C:6]([CH3:8])[CH:7]=1.[NH3:20].CCOC(C)=O>CO>[NH2:20][C:15]1[CH:16]=[CH:17][CH:18]=[C:11]([S:9]([C:4]2[CH:3]=[C:2]([CH3:1])[CH:7]=[C:6]([CH3:8])[CH:5]=2)=[O:10])[C:12]=1[C:13]#[N:14]
CCOC(=O)C.CC=1C=C(C=C(C1)C)S(=O)C1=C(C#N)C(=CC=C1)F.N
EtOAc;2-[(3,5-Dimethylphenyl)sulfinyl]-6-fluorobenzonitrile;ammonia
0.0;0.4;20.0
mol;g;mL
CO
methanol
40.0
mL
null
null
null
null
null
null
null
null
-78.0
null
NC1=C(C#N)C(=CC=C1)S(=O)C1=CC(=CC(=C1)C)C
2-amino-6-[(3,5-dimethylphenyl)sulfinyl]benzonitrile
0.24
g
59.2
ord-b5f73f3ea0a54afca47617c9e6b59c43
[CH3:1][C:2]1[CH:3]=[C:4]([S:9]([C:12]2[CH:19]=[CH:18][CH:17]=[C:16](F)[C:13]=2[C:14]#[N:15])(=[O:11])=[O:10])[CH:5]=[C:6]([CH3:8])[CH:7]=1.[NH3:21].CCOC(C)=O>CO>[NH2:21][C:16]1[CH:17]=[CH:18][CH:19]=[C:12]([S:9]([C:4]2[CH:3]=[C:2]([CH3:1])[CH:7]=[C:6]([CH3:8])[CH:5]=2)(=[O:11])=[O:10])[C:13]=1[C:14]#[N:15]
CCOC(=O)C.CC=1C=C(C=C(C1)C)S(=O)(=O)C1=C(C#N)C(=CC=C1)F.N
EtOAc;2-[(3,5-Dimethylphenyl)sulfonyl]-6-fluorobenzonitrile;ammonia
0.0;0.5;20.0
mol;g;mL
CO
methanol
80.0
mL
null
null
null
null
null
null
null
null
-78.0
24
NC1=C(C#N)C(=CC=C1)S(=O)(=O)C1=CC(=CC(=C1)C)C
2-amino-6-[(3,5-dimethylphenyl)sulfonyl]benzonitrile
0.28
g
57.5
ord-6c9f5721435e410ba7c84870a32cbc44
Br[C:2]1[CH:3]=[C:4]([CH3:10])[CH:5]=[C:6]([O:8][CH3:9])[CH:7]=1.[Li]C(CC)C.[S].[F:17][C:18]1[CH:25]=[CH:24][CH:23]=[C:22](F)[C:19]=1[C:20]#[N:21].C[S:28](C)=O>C(=O)=O.CC(C)=O.O.C1COCC1>[F:17][C:18]1[CH:25]=[CH:24][CH:23]=[C:22]([S:28][C:2]2[CH:7]=[C:6]([O:8][CH3:9])[CH:5]=[C:4]([CH3:10])[CH:3]=2)[C:19]=1[C:20]#[N:21] ...
FC1=C(C#N)C(=CC=C1)F.CS(=O)C.BrC=1C=C(C=C(C1)OC)C.[Li]C(C)CC..[S]
2,6-difluorobenzonitrile;DMSO;3-bromo-5-methoxytoluene;sec-BuLi;resultant mixture;sulfur
0.69;5.0;1.0;8.46;0.0;0.19
g;mL;g;mL;mol;g
.C(=O)=O.CC(=O)C.C1CCOC1.O
ice water;dry ice acetone;THF;water
0.0;0.0;0.0;100.0
mol;mol;mol;mL
null
null
null
null
null
null
null
null
null
0.3333
FC1=C(C#N)C(=CC=C1)SC1=CC(=CC(=C1)OC)C
2-Fluoro-6-[(3 -methyl-5-methoxyphenyl)thio]benzonitrile
null
null
null
ord-1a88c0d5212446d3b4c2d1662ded1557
F[C:2]1[CH:9]=[CH:8][CH:7]=[C:6]([S:10][C:11]2[CH:16]=[C:15]([O:17][CH3:18])[CH:14]=[C:13]([CH3:19])[CH:12]=2)[C:3]=1[C:4]#[N:5].[NH3:20]>C(O)C.C1COCC1>[NH2:20][C:2]1[CH:9]=[CH:8][CH:7]=[C:6]([S:10][C:11]2[CH:16]=[C:15]([O:17][CH3:18])[CH:14]=[C:13]([CH3:19])[CH:12]=2)[C:3]=1[C:4]#[N:5]
FC1=C(C#N)C(=CC=C1)SC1=CC(=CC(=C1)OC)C.N.
2-fluoro-6-[(3-methyl-5-methoxyphenyl)thio]benzonitrile;ammonia;resultant solution
0.1;0.0;0.0
g;mol;mol
C(C)O.C1CCOC1
ethanol;THF
10.0;2.0
mL;mL
null
null
null
null
null
null
null
null
145.0
null
NC1=C(C#N)C(=CC=C1)SC1=CC(=CC(=C1)OC)C
2-Amino-6-[(3 -methyl-5-methoxyphenyl)thio]benzonitrile
null
null
null
ord-b52dd58a1564476b8012385c8b071efd
F[C:2]1[CH:9]=[CH:8][CH:7]=[C:6]([S:10]([C:13]2[CH:18]=[C:17]([O:19][CH3:20])[CH:16]=[C:15]([CH3:21])[CH:14]=2)(=[O:12])=[O:11])[C:3]=1[C:4]#[N:5].[NH3:22]>C(O)C.C1COCC1>[NH2:22][C:2]1[CH:9]=[CH:8][CH:7]=[C:6]([S:10]([C:13]2[CH:18]=[C:17]([O:19][CH3:20])[CH:16]=[C:15]([CH3:21])[CH:14]=2)(=[O:12])=[O:11])[C:3]=1[C:4]#[N...
FC1=C(C#N)C(=CC=C1)S(=O)(=O)C1=CC(=CC(=C1)OC)C.N.
2-fluoro-6-[(3-methyl-5-methoxyphenyl)sulfonyl]benzonitrile;ammonia;resultant solution
0.3;0.0;0.0
g;mol;mol
C(C)O.C1CCOC1
ethanol;THF
10.0;2.0
mL;mL
null
null
null
null
null
null
null
null
130.0
null
NC1=C(C#N)C(=CC=C1)S(=O)(=O)C1=CC(=CC(=C1)OC)C
2-amino-6-[(3-methyl-5-methoxyphenyl)sulfonyl]benzonitrile
0.1
g
34
ord-57d496f8cfa74e14b0b60ed9b08a5969
[NH2:1][CH:2]([CH2:6][CH3:7])[C:3]([OH:5])=[O:4].S(Cl)([Cl:10])=O.[CH2:12](OCC)[CH3:13]>C(O)C>[ClH:10].[NH2:1][CH:2]([CH2:6][CH3:7])[C:3]([O:5][CH2:12][CH3:13])=[O:4] |f:4.5|
NC(C(=O)O)CC.S(=O)(Cl)Cl.C(C)OCC
2-aminobutyric acid;thionyl chloride;diethyl ether
100.0;120.8;600.0
g;g;mL
C(C)O
ethanol
300.0
mL
null
null
null
null
null
null
null
null
0.0
8
Cl.NC(C(=O)OCC)CC
desired product
150
g
null
ord-968da5d345074707bd8ae7f036b4987e
Cl.[NH2:2][CH:3]([CH2:9][CH3:10])[C:4]([O:6][CH2:7][CH3:8])=[O:5].S([O-])([O-])(=O)=O.[Mg+2].C(N(CC)CC)C.[CH:24](=O)[C:25]1[CH:30]=[CH:29][CH:28]=[CH:27][CH:26]=1>ClCCl>[CH:24](=[N:2][CH:3]([CH2:9][CH3:10])[C:4]([O:6][CH2:7][CH3:8])=[O:5])[C:25]1[CH:30]=[CH:29][CH:28]=[CH:27][CH:26]=1 |f:0.1,2.3|
C(C1=CC=CC=C1)=O.Cl.NC(C(=O)OCC)CC.S(=O)(=O)([O-])[O-].[Mg+2].C(C)N(CC)CC
benzaldehyde;product;magnesium sulphate;triethylamine
94.9;149.6;74.3;246.0
g;g;g;mL
ClCCl
dichloromethane
1500.0
mL
null
null
null
null
null
null
null
null
ambient
3
C(C1=CC=CC=C1)=NC(C(=O)OCC)CC
desired product
174
g
88.9
ord-8bc8a5b260b5493c8773ed6d142bea7c
[NH2:1][C:2]([CH2:12][CH3:13])([CH2:8][CH:9]=[CH:10][CH3:11])[C:3](OCC)=[O:4].[H-].[Al+3].[Li+].[H-].[H-].[H-].[OH-].[Na+]>C1COCC1>[NH2:1][C:2]([CH2:12][CH3:13])([CH2:8][CH:9]=[CH:10][CH3:11])[CH2:3][OH:4] |f:1.2.3.4.5.6,7.8|
[OH-].[Na+].NC(C(=O)OCC)(CC=CC)CC..[H-].[Al+3].[Li+].[H-].[H-].[H-]
NaOH;product;solution;lithium aluminium hydride
200.0;116.7;0.0;0.0
mL;g;mol;mol
C1CCOC1.C1CCOC1
THF;THF
100.0;800.0
mL;mL
null
null
null
null
null
null
null
null
ambient
8
NC(CO)(CC=CC)CC
desired product
29.3
g
32.5
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