PATENT CLAIM ANALYSIS

Application Number: 15909801
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2018-07
Patent Classification: ["435", "060000"]

Abstract:
The present invention provides compounds of the formula: which are useful as inhibitors of PHD, pharmaceutical compositions thereof, methods for treatment of conditions associated with HIF, processes for making the compounds and intermediates thereof.

Claim (Index 12):
A compound of the formula: or a pharmaceutically acceptable salt thereof, wherein: R 1  is selected from the group consisting of optionally substituted C 1-6  alkyl, optionally substituted C 3-8  cycloalkyl, and optionally substituted C 3-6  heterocyclyl; R 2  is selected from the group consisting of hydrogen and C 1-4  alkyl; R 3 , each time taken, is independently selected from the group consisting of hydrogen, hydroxyl, amino, C 1-8  alkylamino, cyano, halo, optionally substituted C 1-6  alkyl, and C 1-4  alkoxy; R 4  is selected from the group consisting of hydrogen, cyano, halo, methyl, ethyl, methoxy, and trifluoromethyl; R 5  is selected from the group consisting of G is C; A is selected from the group consisting of N, O, S, CR 6 , and NR 6 ; E is selected from the group consisting of N, O, S, and CR 6 ; provided that only one of A and E can be O or S; or G is N and A and E are CR 6 ; or G and A are N and E is CR 6 ; or G, A, and E are N; R 6 , each time taken, is independently selected from the group consisting of hydrogen, cyano, halo, C 3-8  cycloalkyl, C 1-6  alkyl, C 1-4  alkoxy, and trifluoromethyl; and R 7  is selected from the group consisting of cyano and cyanomethyl.

Metadata:
- Claim Count in Document: 14.0
- Percentile: 90.0
- Lexical Diversity: 1.25806
- Patent Class: 435.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['14693110', '14226722', '15150976', '16080506', '15620620']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.6743299038781926
- 35 USC 102 Novelty (BERT): 0.5342262186711595
- Combined Prediction Score: 0.6603195353574893
- Mean Citation Score: 359.5609760000001
- Max Citation Score: 367.1524
- Similarity Product: 287.6281746243477

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test