PATENT CLAIM ANALYSIS

Application Number: 15959663
Application Type: Utility
Filing Date: 2018-04
Publication Date: 2018-08
Patent Classification: ["514", "604000"]

Abstract:
The present invention provides fatty acid amide hydrolase inhibitors, solid forms thereof, compositions thereof, and methods of making and using the same.

Claim (Index 1):
A method of preparing Compound 1: or a pharmaceutically acceptable salt, hydrate or solvate thereof, or anhydride thereof; comprising the steps of: (a) coupling a compound of formula E-1: wherein: LG 1  and LG 2  are independently selected from a halogen or sulfonate; with a compound of formula E-2: wherein each R 1  and R 2  is independently selected from hydrogen or an C 1-6  alkyl, C 2-6  alkenyl, C 2-6  alkynyl, C 6-12  aryl or C 6-12  heteroaryl group, or R 1  and R 2  are joined to form a 5-8 membered ring; in order to provide a compound of formula E-3: wherein: LG 2  is selected from a halogen or sulfonate; and (b) reacting E-3 with a boronation reagent and a metal reagent in order to provide Compound 1 or a pharmaceutically acceptable salt, hydrate or solvate thereof, or anhydride thereof.

Metadata:
- Claim Count in Document: 5.0
- Percentile: 91.0
- Lexical Diversity: 1.18182
- Patent Class: 514.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['14631712', '13019262', '13347423', '14327499', '13992022']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7277871577565178
- 35 USC 102 Novelty (BERT): 0.58736682243076
- Combined Prediction Score: 0.7137451242239421
- Mean Citation Score: 269.21490800000004
- Max Citation Score: 375.56296
- Similarity Product: 268.1425242157316

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 0
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test