PATENT CLAIM ANALYSIS

Application Number: 16094030
Application Type: Utility
Filing Date: 2018-10
Publication Date: 2019-04
Patent Classification: ["544", "184000"]

Abstract:
Provided is a compound represented by the following formula, or a salt thereof: [wherein each symbol is as defined herein.].

Claim (Index 5):
The compound or salt thereof according to  claim 1 , wherein\n R 1  is (I) a C 1-6  alkyl group optionally having 1 to 5 substituents each selected from (a) a halogen atom, (b) a hydroxy group, (c) a cyano group, (d) a C 1-6  alkoxy group optionally having 1 to 3 substituents each selected from\n (i) a halogen atom, and \n (ii) a hydroxy group, and \n (e) a three- to eight-membered nonaromatic heterocyclic group optionally having 1 to 3 halogen atoms; (II) a three- to eight-membered nonaromatic heterocyclic group optionally having 1 to 5 substituents each selected from (a) a C 1-6  alkoxy group, (b) a halogen atom, and (c) a hydroxy group; (III) a five- to fourteen-membered aromatic heterocyclic group optionally having 1 to 3 optionally halogenated C 1-6  alkyl groups; (IV) a C 1-6  alkoxy group optionally having 1 to 5 substituents each selected from (a) a hydroxy group, (b) a three- to eight-membered nonaromatic heterocyclic group, and (c) a five- or six-membered monocyclic aromatic heterocyclic group optionally having 1 to 3 optionally halogenated C 1-6  alkyl groups; (V) an optionally halogenated C 3-10  cycloalkyl group; or (VI) an amino group optionally monosubstituted or disubstituted with a C 1-6  alkyl group optionally having 1 to 5 substituents each selected from (a) (i) a halogen atom,\n (ii) a hydroxy group, and \n (iii) a C 1-6  alkoxy group; \n R 2  is (I) a C 1-6  alkyl group optionally having 1 to 3 five- to fourteen-membered aromatic heterocyclic groups optionally having 1 to 3 substituents each selected from (a) a halogen atom, (b) a C 1-6  alkyl group optionally having 1 to 7 substituents each selected from\n (i) a halogen atom, \n (ii) a hydroxy group, and \n (iii) a C 1-6  alkoxy group, \n (c) an optionally halogenated C 3-10  cycloalkyl group, (d) a C 1-6  alkoxy group, (e) a C 1-6  alkyl group-C 3-10  cycloalkyl group (f) a C 1-6  alkyl group-three- to eight-membered monocyclic nonaromatic heterocyclic group, and (g) an oxo group; or (II) a C 7-16  aralkyl group optionally having 1 to 3 substituents each selected from (a) a C 1-6  alkyl group optionally having 1 to 3 substituents each selected from\n (i) a halogen atom, and \n (ii) a hydroxy group, \n (b) a C 1-6  alkoxy-carbonyl group, (c) a halogen atom, (d) a C 1-6  alkoxy group optionally having 1 to 3 substituents each selected from\n (i) a halogen atom, and \n (ii) a hydroxy group \n (e) a mono- or di-C 1-6  alkyl-carbamoyl group, (f) a cyano group, (g) an amino group optionally monosubstituted or disubstituted with a substituent selected from\n (i) a C 1-6  alkyl group, and \n (ii) a C 1-6  alkoxy-carbonyl group, \n (h) a nitro group, and (i) a carboxy group; each of R 6  and R 7  is a hydrogen atom; ring A is a bicyclic aromatic heterocycle selected from the formulae (1), (2), (3) and (4); Xs each independently represent C(R 5 ) or N; R 3  is a hydrogen atom; R 4  is (I) a hydrogen atom, (II) a halogen atom, (III) an optionally halogenated C 1-6  alkoxy group, or (IV) an amino group optionally monosubstituted or disubstituted with a C 1-6  alkyl group; and R 5  is (I) a hydrogen atom, (II) a halogen atom, (III) a cyano group, (IV) a C 1-6  alkyl group optionally having 1 to 5 substituents each selected from\n (a) a halogen atom, \n (b) a C 1-6  alkoxy group, \n (c) a C 1-6  alkoxy-C 1-6  alkoxy group, \n (d) a hydroxy group, and \n (e) a C 1-6  alkyl-carbonyloxy group, \n (V) a C 1-6  alkoxy group, \n (VI) a C 2-6  alkenyl group optionally having 1 to 3 C 1-6  alkoxy groups, \n (VII) a C 2-6  alkynyl group, \n (VIII) a cyano-C 6-14  aryl group, \n (IX) a five- to fourteen-membered aromatic heterocyclic group optionally having 1 or 2 C 1-6  alkyl groups optionally having 1 to 3 substituents each selected from\n (a) a halogen atom, \n (b) a five- or six-membered monocyclic aromatic heterocyclic group, and \n (c) a three- to eight-membered monocyclic nonaromatic heterocyclic group, \n \n (X) a C 1-6  alkyl-carbonyl group, \n (XI) a hydroxy group, \n (XII) a C 1-6  alkyl-five- to fourteen-membered aromatic heterocyclic oxy group, \n (XIII) a three- to eight-membered monocyclic nonaromatic heterocyclic group optionally having 1 to 3 substituents each selected from\n (a) a halogen atom, \n (b) a C 1-6  alkoxy group, and \n (c) an oxo group, or \n \n (XIV) an amino group optionally monosubstituted or disubstituted with an optionally halogenated C 1-6  alkyl.

Metadata:
- Claim Count in Document: 20.0
- Percentile: 97.0
- Lexical Diversity: 1.13043
- Patent Class: 544.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15304623', '16323863', '16049359', '15304727', '15565891']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7921482890291671
- 35 USC 102 Novelty (BERT): 0.5364702966987126
- Combined Prediction Score: 0.7665804897961217
- Mean Citation Score: 364.348058
- Max Citation Score: 367.53668
- Similarity Product: 317.4700089520502

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test