PATENT CLAIM ANALYSIS

Application Number: 15768960
Application Type: Utility
Filing Date: 2018-04
Publication Date: 2018-11
Patent Classification: ["514", "220000"]

Abstract:
The present invention relates to a benzodiazepine derivative of Formula I as a short-acting anesthetic, a pharmaceutical composition comprising the same, a kit comprising the same, a preparation method thereof, an method of anesthesia using the same and use thereof in the manufacture of an anesthetic medicament.

Claim (Index 5):
A compound of  claim 1 , wherein,\n K is CR 4 ; J is N; R 2  is phenyl optionally substituted with one or more (e.g., 1, 2, 3 or 4) halogen, preferably, R 2  is 2-fluorophenyl; and R 5  is independently selected from the group consisting of 3-10 membered cycloalkyl and C 1-6  alkyl, wherein the 3-10 membered cycloalkyl is optionally substituted with one or more (e.g., 1, 2, 3 or 4) substituents independently selected from the group consisting of halogen, hydroxy, C 1-6  alkyl, R 6 R 7 N\u2014, C 1-6  alkoxy, 3-10 membered cycloalkyl, 3-10 membered heterocyclyl, 6-14 membered aryl and 5-14 membered heteroaryl, and the C 1 -C 6  alkyl is substituted with one or more (e.g., 1, 2, 3 or 4) substituents independently selected from the group consisting of halogen, R 6 R 7 N\u2014, C 1-6  alkoxy, 3-10 membered cycloalkyl, 3-10 membered heterocyclyl, 6-14 membered aryl and 5-14 membered heteroaryl, preferably, R 5  is independently selected from the group consisting of 3-10 membered cycloalkyl, and C 1-6  alkyl substituted with one or more (e.g., 1, 2, 3 or 4) C 1-6  alkoxy, more preferably, R 5  is independently selected from the group consisting of cyclopropyl and methoxymethyl, or a pharmaceutically acceptable salt, stereoisomer, tautomer, polymorph, solvate, metabolite or prodrug thereof.

Metadata:
- Claim Count in Document: 29.0
- Percentile: 91.0
- Lexical Diversity: 1.57576
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['12598882', '14858159', '14448160', '09927324', '15150038']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8355831440601479
- 35 USC 102 Novelty (BERT): 0.532843632225451
- Combined Prediction Score: 0.8053091928766782
- Mean Citation Score: 356.00754
- Max Citation Score: 373.12048
- Similarity Product: 298.5352634674358

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test