PATENT CLAIM ANALYSIS

Application Number: 16044320
Application Type: Utility
Filing Date: 2018-07
Publication Date: 2018-11
Patent Classification: ["546", "268100"]

Abstract:
The invention relates to a compound of formula (I) wherein A and R 1  to R 4  are defined as in the description and in the claims. The compound of formula (I) can be used as a medicament.

Claim (Index 1):
A compound of formula (I): wherein A is \u2014CH\u2014 or nitrogen; R l  is halophenyl, halophenylalkyl, haloalkoxy, halogen, alkoxyalkoxy, oxopyrrolidinyl or cycloalkylalkoxy; R 2  is hydrogen, halophenylamino, cycloalkyl or haloazetidinyl; one of R 3  and R 4  is hydrogen and the other one is \u2014(CR 5 R 6 ) m \u2014(CH 2 ) n \u2014R 7 ;\n or R 3  and R 4  together with the nitrogen atom to which they are attached form aminocarbonylthiomorpholinyl; \n R 5  and R 6  are independently selected from hydrogen and alkyl; R 7  is 5-cycloalkyl-1,3,4-oxadiazolyl, 3-cycloalkyl-1,2,4-oxadiazolyl, 5-phenyl-1,3,4-oxadiazolyl, 3-phenyl-1,2,4-oxadiyzolyl, 5-alkyl-1,3,4-oxadiazolyl, 3-alkoxyalkoxyalkyl-1,2-oxazolyl, 1-hydroxyalkylpyrazolyl, 3-hydroxy-1-adamantyl, alkoxycarbonylmorpholinyl, 3-oxanyloxyalkyl-1,2-oxazol-5-yl, 3-azidoalkyl-1,2-oxazol-5-yl or 5-(4-fluorophenyl)-1,3,4-oxadiazolyl; m is 0 or 1; and n is 0 or 1; or a pharmaceutically acceptable salt or ester thereof; provided that the compound is other than 6-chloro-N-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-2-pyridinecarboxamide and pharmaceutically acceptable salts esters thereof is excluded.

Metadata:
- Claim Count in Document: 32.0
- Percentile: 95.0
- Lexical Diversity: 1.51724
- Patent Class: 546.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['14868305', '15050753', '14648418', '13486057', '15478435']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8241260072476638
- 35 USC 102 Novelty (BERT): 0.543602398622198
- Combined Prediction Score: 0.7960736463851172
- Mean Citation Score: 374.275046
- Max Citation Score: 408.03818
- Similarity Product: 317.25502486234313

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 0
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test