PATENT CLAIM ANALYSIS

Application Number: 15767156
Application Type: Utility
Filing Date: 2018-04
Publication Date: 2018-10
Patent Classification: ["514", "373000"]

Abstract:
The invention relates to compounds of formula (I): wherein R 1 , R 2 , R 3 , R 4 , R 5  and R 6  are as defined in the description. The compounds of formula (I) are inhibitors of the YAP/TAZ-TEAD interaction.

Claim (Index 1):
A compound of formula (I) or a pharmaceutically acceptable salt thereof, wherein: R 1  is H, alkyl or alkyl-R 7  or -aryl-R 7 ; R 2 , R 3 , R 4 , R 5  are independently H, halo, \u2014B(O\u2014R 11 ) 2 , alkyl, alkoxyl, hydroxycarbonyl, \u2014COOR 11 , \u2014CO\u2014NR 8 R 9  or aryl; R 6  is H or alkyl; or R 1  and R 6  are bound together to form a 5 or 6-member heterocycle; R 7  is hydroxyl, alkylhydroxyl, \u2014NR 8 R 9 , \u2014CO\u2014X\u2014R 10 , \u2014CN, \u2014CF 3 , aryl; R 8  and R 9  are independently H, alkyl or form together with the nitrogen atom a 3 to 6-member cyclic group; X is \u2014O\u2014 or \u2014NR 11 \u2014; R 10  is H, alkyl or hydroxyalkyl; R 11  is H or alkyl.

Metadata:
- Claim Count in Document: 24.0
- Percentile: 91.0
- Lexical Diversity: 1.6129
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['10520621', '15569273', '13980182', '10788426', '11722075']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8355483562457454
- 35 USC 102 Novelty (BERT): 0.5041162790312582
- Combined Prediction Score: 0.8024051485242967
- Mean Citation Score: 262.577372
- Max Citation Score: 272.25116
- Similarity Product: 195.86976558159355

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test