PATENT CLAIM ANALYSIS

Application Number: 16029228
Application Type: Utility
Filing Date: 2018-07
Publication Date: 2018-11
Patent Classification: ["514", "211000"]

Abstract:
The present invention provides a compound of formula I having BACE1 inhibitory activity, their manufacture, pharmaceutical compositions containing them and their use as therapeutically active substances. The active compounds of the present invention are useful in the therapeutic and/or prophylactic treatment of e.g. Alzheimer's disease.

Claim (Index 9):
A compound of formula I according to any one of  claims 1 - 8  that is selected from the group consisting of\n 5-Cyano-pyridine-2-carboxylic acid [6-((3R,4aR)-1-amino-3-methyl-4a-oxo-3,4,6,7,8,9-hexahydro-4a\u03bb 6 -thia-2,5,9a-triaza-benzocyclohepten-3-yl)-5-fluoro-pyridin-2-yl]-amid, \n 5-Cyano-pyridine-2-carboxylic acid [6-((3R,4aS)-1-amino-3-methyl-4a-oxo-3,4,6,7,8,9-hexahydro-4a\u03bb 6 -thia-2,5,9a-triaza-benzocyclohepten-3-yl)-5-fluoro-pyridin-2-yl]-amide, \n 5-Cyano-3-methyl-pyridine-2-carboxylic acid [6-((3R,4aS)-1-amino-3-methyl-4a-oxo-3,4,6,7,8,9-hexahydro-4a\u03bb 6 -thia-2,5,9a-triaza-benzocyclohepten-3-yl)-5-fluoro-pyridin-2-yl]-amide, \n N-[6-[(1S,10S)-8-Amino-10-(fluoromethyl)-1-oxo-1\u03bb 6 -thia-2,7,9-triazabicyclo[5.4.0]undeca-1,8-dien-10-yl]-5-fluoropyridin-2-yl]-5-cyanopyridine-2-carboxamide, and \n N-[6-[(1R,10S)-8-Amino-10-(fluoromethyl)-1-oxo-1\u03bb 6 -thia-2,7,9-triazabicyclo[5.4.0]undeca-1,8-dien-10-yl]-5-fluoropyridin-2-yl]-5-cyanopyridine-2-carboxamide.

Metadata:
- Claim Count in Document: 14.0
- Percentile: 95.0
- Lexical Diversity: 1.275
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15314718', '15105725', '15502044', '14400448', '13467085']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8419689303952044
- 35 USC 102 Novelty (BERT): 0.5904020393977386
- Combined Prediction Score: 0.8168122412954578
- Mean Citation Score: 422.914858
- Max Citation Score: 521.9717
- Similarity Product: 448.21634030584704

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test