PATENT CLAIM ANALYSIS

Application Number: 16101250
Application Type: Utility
Filing Date: 2018-08
Publication Date: 2018-12
Patent Classification: ["544", "250000"]

Abstract:
The present application relates to novel substituted (aza)pyridopyrazolopyrimidinones and indazolopyrimidinones, to processes for their preparation, the compounds for use alone or in combinations in a method for the treatment and/or prophylaxis of diseases, in particular for the treatment and/or prophylaxis of acute and recurrent bleeding in patients with or without underlying hereditary or acquired bleeding disorders, wherein the bleeding is associated with a disease or medical intervention selected from the group consisting of menorrhagia, postpartum hemorrhage, hemorrhagic shock, trauma, surgery, transplantation, stroke, liver diseases, hereditary angioedema, nosebleed, and synovitis and cartilage damage following hemarthrosis.

Claim (Index 23):
The method of  claim 21 , wherein in the compound of the formula (I-B):\n R 1  is selected from hydrogen and methyl; X 1  is C\u2014R 2  X 2  is C\u2014R 3  X 3  is C\u2014R 4  X 4  is C\u2014R 5 ; and R 2 , R 3 , and R 4 , are independently from each other selected from hydrogen and fluorine; R 5  is selected from hydrogen, halogen, C 1 -C 4  alkyl, C 1 -C 4  haloalkyl, C 1 -C 4  alkoxy, C 1 -C 4  haloalkoxy, cyano, amino, nitro, dialkylamino, hydroxy, carboxyl, C 3 -C 7  cycloalkyl, triazolyl (bonded via N), thiazolyl, thienyl, pyridyl, imidazolyl, pyrrolyl, pyrazolyl (bonded via N or C), the pyrazolyl being optionally substituted with one or two substituents selected from C 1 -C 4  alkyl, and phenyl, the phenyl being optionally substituted with one or two substituents selected from halogen, C 1 -C 4  alkyl, C 1 -C 4  haloalkyl, C 1 -C 4  alkoxy, and C 1 -C 4  haloalkoxy; with a proviso that zero, one, or two of R 2  to R 5  are different from hydrogen, and salts thereof.

Metadata:
- Claim Count in Document: 53.0
- Percentile: 96.0
- Lexical Diversity: 1.57746
- Patent Class: 544.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15416651', '14533915', '15523954', '12678288', '12996465']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7855917081087401
- 35 USC 102 Novelty (BERT): 0.6057191919503018
- Combined Prediction Score: 0.7676044564928962
- Mean Citation Score: 405.642188
- Max Citation Score: 524.56165
- Similarity Product: 489.4831004443884

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test