PATENT CLAIM ANALYSIS

Application Number: 16076836
Application Type: Utility
Filing Date: 2018-08
Publication Date: 2019-02
Patent Classification: ["514", "443000"]

Abstract:
This invention relates to novel 4,4,5,5,7,7-hexamethyl-5,7-dihydro-4H-thieno[2,3-c]pyranyl compounds, and pharmaceutically acceptable salts thereof. This invention also provides compositions comprising a compound of this invention and the use of such compositions in methods of treating diseases and conditions that are beneficially treated by administering cystic fibrosis transmembrane conductance regulator (CFTR) modulators.

Claim (Index 1):
A compound of Formula I: or a pharmaceutically acceptable salt thereof, wherein:\n each R 1  is independently CH 3 , CDH 2 , CD 2 H, or CD 3 ; \n each R 2  is independently CH 3 , CDH 2 , CD 2 H, or CD 3 ; \n each R 3  is independently H or D; \n Y is selected from\n (i) a C 1-5  hydroxyalkyl optionally substituted by 0-10 deuterium, \n (ii) a phenyl ring independently substituted by 0-5 deuterium and by 0-2 R 4  groups; \n (iii) a C 3-6  cycloalkyl independently substituted by 0-11 deuterium and by 0-2 R 5  groups and 0-2 oxo groups, and \n (iv) a 5- or 6-membered heteroaryl independently substituted by 0-4 deuterium and by 0-2 R 5  groups; \n \n R 4  is halo, \u2014OH, \u2014CN, C 1-4  alkyl, C 1-4  haloalkyl, C 1-4  alkoxy, or C 1-4  haloalkoxy, wherein each alkyl or alkoxy group is optionally substituted with deuterium; \n R 5  is halo, OH, \u2014OC(\u2550O)C 1-4 alkyl, \u2014COOH, \u2014C(\u2550O)C 1-4 alkoxy, C 1-4  haloalkyl, C 1-4  alkyl, C 1-4  alkoxy, or C 1-4  haloalkoxy, wherein each alkyl or alkoxy group is optionally substituted with deuterium; \n provided that when each R 1  is CH 3 , each R 2  is CH 3 , each R 3  is H, R 4 , if present, is not substituted by deuterium, and R 5 , if present, is not substituted by deuterium, then Y is substituted by at least one deuterium.

Metadata:
- Claim Count in Document: 19.0
- Percentile: 96.0
- Lexical Diversity: 1.18367
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['13808508', '13959716', '15562860', '13364724', '14915527']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7662188949534571
- 35 USC 102 Novelty (BERT): 0.5074871290707085
- Combined Prediction Score: 0.7403457183651823
- Mean Citation Score: 246.669346
- Max Citation Score: 253.55965
- Similarity Product: 195.0414598965466

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 0
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test