PATENT CLAIM ANALYSIS

Application Number: 16157370
Application Type: Utility
Filing Date: 2018-10
Publication Date: 2019-08
Patent Classification: ["544", "131000"]

Abstract:
Disclosed is a compound represented by formula (1) or a pharmacologically acceptable salt thereof. (In the formula, R 1  is optionally substituted heteroaryl etc.; R 2  is hydrogen etc.; R 3  and R 4  are each independently hydrogen etc., R 5  is the following group: (wherein Y is optionally substituted five membered heteroaryl etc., R 9a  is optionally substituted aryl etc., R 9b  and R 9c  are each dependently hydrogen etc., and m is the integral 0 etc.) etc.; R 6  is hydrogen etc.; and R 7  is hydrogen etc.

Claim (Index 1):
A compound of formula 1: or pharmaceutically acceptable salt thereof, R 1  is optionally substituted heteroaryl, or optionally substituted heteroalicyclic: R 2  is hydrogen, optionally substituted alkyl, optionally substituted alkylcarbonyl, optionally substituted alkoxycarbonyl, or optionally substituted aminocarbonyl; R 3  and R 4  are each independently hydrogen, halogen, cyano, nitro, hydroxy, optionally substituted alkyl, optionally substituted alkoxy, optionally substituted amino, optionally substituted alkoxycarbonyl, optionally substituted alkylcarbonyl, optionally substituted aminocarbonyl, or the following group: (wherein X is optionally substituted five membered heteroaryl or optionally substituted heteroalicyclic, R 8a  is optionally substituted aryl, optionally substituted heteroaryl, or optionally substituted heteroalicyclic, R 8b  and R 8c  are each independently hydrogen, alkyl, halogen, cyano, amino, nitro, hydroxy, trifluoromethyl, optionally substituted aryl, optionally substituted heteroaryl, or optionally substituted heteroalicyclic, and n is the integral 0 to 2), R 5  is hydrogen, halogen, cyano, nitro, hydroxy, optionally substituted alkyl, optionally substituted alkoxy, optionally substituted amino, optionally substituted alkoxycarbonyl, optionally substituted alkylcarbonyl, optionally substituted aminocarbonyl, or the following group: (wherein Y is optionally substituted five membered heteroaryl (provided that the five membered heteroaryl is not the following group: wherein R 9a  is same as the above definition), R 9a  is optionally substituted aryl, optionally substituted heteroaryl, or optionally substituted heteroalicyclic, R 9b  and R 9c  are each dependently hydrogen, alkyl, halogen, cyano, amino, nitro, hydroxy, trifluoromethyl, and m is the integral 0 to 2), and at least one of R 3 , R 4  and R 5  is the following group: (X, R 8a , R 8b , R 8c  and n are same as the above definition), or the following group: (Y, R 9a , R 9b , R 9c  and m are same as the above definition); R 6  is hydrogen, halogen, cyano, nitro, hydroxy, amino, optionally substituted alkyl, optionally substituted alkoxy, optionally substituted amino, optionally substituted alkoxycarbonyl, optionally substituted alkyl carbonyl, or optionally substituted aminocarbonyl; and R 7  is hydrogen, optionally substituted alkyl, or optionally substituted cycloalkyl.

Metadata:
- Claim Count in Document: 1.0
- Percentile: 97.0
- Lexical Diversity: 2.15385
- Patent Class: 544.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['14208289', '13380376', '12809489', '11917239', '13935016']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7746972752794573
- 35 USC 102 Novelty (BERT): 0.5719899464312566
- Combined Prediction Score: 0.7544265423946372
- Mean Citation Score: 345.00844
- Max Citation Score: 441.44412
- Similarity Product: 429.5717231040143

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test