PATENT CLAIM ANALYSIS

Application Number: 15971156
Application Type: Utility
Filing Date: 2018-05
Publication Date: 2018-11
Patent Classification: ["514", "230200"]

Abstract:
This invention is in the field of medicinal chemistry and relates to compounds, and pharmaceutical compositions thereof that are useful as antibacterial agents. The compounds are useful as inhibitors of bacterial gyrase activity and of bacterial infections, and have the structure of Formula (I): as further described herein. The invention further provides pharmaceutical compositions comprising a compound of Formula (I) and methods of using the compounds and compositions to treat bacterial infections.

Claim (Index 12):
The compound according to  claim 10 , wherein R 7A  and R 7B  together with the nitrogen atom to which they are attached form a 4- to 7-membered monocyclic heterocyclic group optionally including one additional heteroatom selected from N, O and S as a ring member,\n or a 6-10 membered bicyclic heterocyclic group optionally including one or two additional heteroatoms selected from N, O and S as ring members, wherein the monocyclic or bicyclic heterocyclic group formed by R 7A  and R 7B  together with the nitrogen atom to which they are attached is optionally substituted by up to three groups selected from halogen, \u2014CN, hydroxy, phenyl, oxo, \u2014OR 9 , \u2014N(R 9 ) 2 , \u2014COOR 9 , \u2014C(O)N(R 9 ) 2 , C 1 -C 4  alkyl, C 1 -C 4  haloalkyl, C 1 -C 4  alkoxy, oxo, C 3 -C 6  cycloalkyl, and a 4-6 membered heteroaryl or heterocyclyl group that contains up to two heteroatoms selected from N, O and S as ring members, wherein the C 1 -C 4  alkyl, C 3 -C 6  cycloalkyl, phenyl, and 4-6 membered heteroaryl or heterocyclyl are each optionally substituted by up to three groups independently selected from halogen, \u2014CN, hydroxy, oxo, -OR 10 , \u2550N\u2014OR 10 , \u2014N(R 10 ) 2, \u2014COOR 10 , \u2014C(O)N(R 10 ) 2 , C 1 -C 4  alkyl, C 1 -C 4  haloalkyl, and C 1 -C 4  alkoxy; or a pharmaceutically acceptable salt thereof.

Metadata:
- Claim Count in Document: 5.0
- Percentile: 93.0
- Lexical Diversity: 1.74468
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15500870', '14527328', '15965172', '12678120', '13902589']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.781767024731144
- 35 USC 102 Novelty (BERT): 0.5796950451081392
- Combined Prediction Score: 0.7615598267688436
- Mean Citation Score: 381.500244
- Max Citation Score: 455.14496
- Similarity Product: 427.1664795156861

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test