PATENT CLAIM ANALYSIS

Application Number: 15764264
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2018-11
Patent Classification: ["546", "209000"]

Abstract:
Problem to be Solved There is a need for a new antibiotic having a novel mechanism of action which exhibit strong antibacterial activity not only against sensitive bacteria but also against resistant bacteria thereof, and at the same time possesses excellent solubility an a safety profile amenable to human use. Solution to the Problem As a result of intensive research, the present inventors have found that a compound represented by general formula (I), a stereoisomer, or a pharmaceutically acceptable salt thereof inhibits DNA gyrase GyrB subunit and/or topoisomerase IV ParE subunit possesses excellent solubility and a safety profile for use in humans for the treatment of bacterial infectious diseases.

Claim (Index 13):
The method according to  claim 15 , wherein said bacterial infectious disease is selected from pimples, impetigo, boils, cellulitis folliculitis, furuncles, carbuncles, scalded skin syndrome, pneumonia, meningitis, osteomyelitis, endocarditis, toxic shock syndrome, bronchitis, rhinitis, acute sinusitis, otitis media, conjunctivitis, bacteremia, sepsis, osteomyelitis, septic arthritis, peritonitis, pericarditis, cellulitis, brain abscess, urinary tract infections,  Clostridium difficile  infections, acne vulgaris, gonorrhea, gas gangrene, food poisoning, tetanus, botulism, diarrhea, pseudomembranous colitis, toxic mega colon, or perforation of colon.

Metadata:
- Claim Count in Document: 36.0
- Percentile: 90.0
- Lexical Diversity: 1.39286
- Patent Class: 546.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15547776', '15262112', '12187115', '11884923', '15314562']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.818997889661547
- 35 USC 102 Novelty (BERT): 0.5186419458360614
- Combined Prediction Score: 0.7889622952789984
- Mean Citation Score: 296.5449680000001
- Max Citation Score: 311.3937
- Similarity Product: 197.87241855282784

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 0
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test