PATENT CLAIM ANALYSIS

Application Number: 16091859
Application Type: Utility
Filing Date: 2018-10
Publication Date: 2019-03
Patent Classification: ["514", "222500"]

Abstract:
Compounds of the formula (I) wherein the substituents are as defined in claim  1 , useful as a pesticides and especially as fungicides.

Claim (Index 1):
A compound of formula (I): wherein R 1  is hydrogen; R 2  is halogen, methyl or methoxy; R 3  represents hydrogen or C 1-4 alkyl; and R 4  represents R 4A , R 4B , R 4C , R 4D  or R 4E ; wherein R 4A  represents heterocyclylC 0-6 alkyl wherein the heterocyclyl moiety is a 5- or 6-membered non-aromatic ring which comprises 1, 2 or 3 heteroatoms individually selected from N, O and S, optionally substituted by 1, 2 or 3 substitutents, which may be the same or different, selected from R 5A ; R 5A  represents C 1-4 alkyl, C 1-4 alkoxy, C 1-4 alkoxycarbonyl, phenylC 0-2 alkyl; R 4B  represents C 3-8 cycloalkylC 0-6 alkyl optionally substituted by 1, 2, 3 or 4 substitutents, which may be the same or different, selected from R 5B ; R 5B  represents cyano, halogen, C 1-4 alkyl, C 2-4 alkynyl, C 1-4 alkoxycarbonyl, C 3-6 cycloalkylC 0-2 alkyl, phenylC 0-2 alkyl, and wherein any of said cycloalkyl or phenyl moieties are optionally substituted by 1, 2 or 3 substituents, which may be the same or different, selected from R 6B ; and R 6B  represents methyl, methoxy or halogen; R 4C  represents C 1-6 alkyl, C 2-6 alkenyl or C 2-6 alkynyl, wherein C 1-6 alkyl is optionally substituted by 1, 2 or 3 substituents, which may be the same or different, selected from R C ; R 5C  represents halogen, C 1-4 alkoxy, C 1-4 alkylcarbonyl, C 1-4 alkoxycarbonyl, hydroxyl, C 1-4 alkylaminocarbonyl; R 4D  represents a phenylC 0-6 alkyl optionally substituted by 1, 2, 3, 4 or 5 substitutents, which may be the same or different, selected from R 5D ; R 5D  represents cyano, halogen, hydroxy, C 1-4 alkyl, C 2-4 alkenyl, C 2-4 alkynyl, haloC 1-4 alkyl, C 1-4 alkoxy, C 1-4 alkylcarbonyl, C 1-4 alkoxycarbonyl, aminocarbonyl, C 1-4 alkylaminocarbonyl, diC 1-4 alkylaminocarbonyl, C 1-4 alkoxycarbonylamino, C 3-8 cycloalkylC 0-6 alkyl, phenylC 0-6 alkyl, heteroarylC 0-6 alkyl wherein the heteroaryl moiety is a 5- or 6-membered aromatic ring which comprises 1, 2, 3 or 4 heteroatoms individually selected from N, O and S, heterocyclylC 0-6 alkyl wherein the heterocyclyl moiety is a 5- or 6-membered non-aromatic ring which comprises 1, 2 or 3 heteroatoms individually selected from N, O and S, and wherein any of said cycloalkyl, phenyl, heteroaryl and heterocyclyl moieties are optionally substituted by 1, 2, 3, 4 or 5 substituents, which may be the same or different, selected from R 6D ; and R 6D  represents methyl, methoxy or halogen; and R 4E  represents heteroarylC 0-6 alkyl wherein the heteroaryl moiety is a 5- or 6-membered aromatic ring comprising 1, 2, 3 or 4 heteroatoms individually selected from N, O and S, and wherein the heteroarylC 0-6 alkyl moiety is optionally substituted by 1, 2, 3, 4 or 5 substitutents, which may be the same or different, selected from R 5E ; R 5E  represents cyano, amino, halogen, hydroxy, C 1-4 alkyl, C 2-4 alkenyl, C 2-4 alkynyl, haloC 1-4 alkyl, C 1-4 alkoxy, C 1-4 alkylamino, diC 1-4 alkylamino, C 1-4 alkylcarbonyl, C 1-4 alkoxycarbonyl, aminocarbonyl, C 1-4 alkylaminocarbonyl, diC 1-4 alkylaminocarbonyl, C 1-4 alkoxycarbonylamino, C 3-8 cycloalkylC 0-6 alkyl, phenylC 0-6 alkyl, heteroarylC 0-6 alkyl wherein the heteroaryl moiety is a 5- or 6-membered aromatic ring which comprises 1, 2, 3 or 4 heteroatoms individually selected from N, O and S, heterocyclylC 0-6 alkyl wherein the heterocyclyl moiety is a 5- or 6-membered non-aromatic ring which comprises 1, 2 or 3 heteroatoms individually selected from N, O and S, and wherein any of said cycloalkyl, phenyl, heteroaryl and heterocyclyl are optionally substituted by 1, 2, 3, 4 or 5 substitutents, which may be the same or different, selected from R 6E ; and R 6E  represents methyl, methoxy or halogen; or a salt or an N-oxide thereof; wherein when R 4  is R 4A , the compound according to Formula (I) is not: 2-fluoro-N-(pyrrolidin-3-yl)-4-[(5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl)]benzamide, 2-fluoro-N-(1-(pyrrolidin-1-yl)propan-2-yl)-4-[(5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl)]benzamide, 2-fluoro-N-(1-(piperidin-1-yl)propan-2-yl)-4-[(5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl)]benzamide, 2-fluoro-N-(1-morpholinopropan-2-yl)-4-[(5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl)]benzamide, or 2-fluoro-N-(4-methoxypyrrolidin-3-yl)-4-[(5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl)]benzamide; when R 4  is R 4C , the compound according to Formula (I) is not: 2-fluoro-N-(1-hydroxypropan-2-yl)-4-[(5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl)]benzamide; and when R 4  is R 4E , the compound according to Formula (I) is not: N-(2,6-dimethylpyridin-4-yl)-2-fluoro-4-(5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl)benzamide.

Metadata:
- Claim Count in Document: 4.0
- Percentile: 97.0
- Lexical Diversity: 1.13043
- Patent Class: 514.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['16339995', '14131558', '14908239', '14762007', '10415751']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7790151459774138
- 35 USC 102 Novelty (BERT): 0.5252114181326344
- Combined Prediction Score: 0.7536347731929358
- Mean Citation Score: 298.581178
- Max Citation Score: 345.29294
- Similarity Product: 271.05791004768133

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 0
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test