PATENT CLAIM ANALYSIS

Application Number: 15766667
Application Type: Utility
Filing Date: 2018-04
Publication Date: 2018-10
Patent Classification: ["514", "300000"]

Abstract:
The present disclosure is directed to disclosed compounds that modulate, e.g., address underlying defects in cellular processing of CFTR activity.

Claim (Index 2):
The compound of  claim 1 , wherein A is selected from the group consisting of: wherein: X 4  is independently for each occurrence selected from the group consisting of O, S, and N(R 4 ); X 5  is selected from the group consisting of N and C(R X5 ); R A1  is independently for each occurrence selected from the group consisting of hydrogen, halogen, C 1-6 alkyl, C 2-6 alkenyl, C 2-6 alkynyl, C 1-6 alkoxy, C 3-6 cycloalkyl, phenyl, \u2014NR a R b , \u2014OC(O)NR a R b , \u2014NR a \u2014C(O)-phenyl, and \u2014O\u2014C(O)\u2014NR a -phenyl; wherein C 1-6 alkyl, C 2-6 alkenyl, C 2-6 alkynyl, C 1-6 alkoxy, C 3-6 cycloalkyl, phenyl, \u2014OC(O)NR a R b , \u2014NR a \u2014C(O)-phenyl, and \u2014O\u2014C(O)\u2014NR a -phenyl may optionally be substituted by one or more substituents selected from the group consisting of halogen, hydroxyl, phenyl, and NR a R b ; R A2  is selected from the group consisting of hydrogen and C 1-6 alkyl; R A3  and R A4  are each independently selected from the group consisting of hydrogen, halogen, C 1-6 alkyl, C 1-6 alkoxy, and NR a R b , wherein C 1-6 alkyl and C 1-6 alkoxy may optionally be substituted by one or more substituents selected from the group consisting of halogen, hydroxyl, phenyl, and NR a R b ; R 4  is selected from the group consisting of hydrogen, C 1-6 alkyl, C 3-6 cycloalkyl, phenyl, heterocycle, C 1-6 alkyl-S(O) 2 \u2014, and phenyl-S(O) 2 \u2014; wherein C 1-6 alkyl, C 3-6 cycloalkyl, phenyl, and heterocycle may optionally be substituted by one or more substituents selected from the group consisting of halogen, hydroxyl, phenyl, and NR a R b ; and R X5  is selected from the group consisting of hydrogen, halogen, and C 1-6 alkyl.

Metadata:
- Claim Count in Document: 140.0
- Percentile: 91.0
- Lexical Diversity: 1.04545
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['15747290', '15539392', '16091401', '15539397', '15320172']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8353129726919531
- 35 USC 102 Novelty (BERT): 0.5325125740568805
- Combined Prediction Score: 0.8050329328284459
- Mean Citation Score: 357.125496
- Max Citation Score: 371.4623
- Similarity Product: 255.7673538051129

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test