PATENT CLAIM ANALYSIS

Application Number: 15760812
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2018-09
Patent Classification: ["546", "268400"]

Abstract:
The present invention relates to a process for preparing a compound of 5 or 5*, or a mixture thereof, and/or a compound of 14 or 14*, or a mixture thereof, that is useful as an antifungal agent. In particular, the invention seeks to provide new methodology for preparing compounds 7, 7* and 11, 11* and substituted derivatives thereof.

Claim (Index 7):
The process of  claim 5 , further comprising:\n a. forming the tetrazole of a compound of Formula 11 or 11*, or mixture thereof; to afford a compound of Formula 13 or 13*, or mixture thereof; and b. alkynylating a compound of Formula 13 or 13*, or mixture thereof, to afford a compound of Formula 18 or 18*, or mixture thereof; wherein each R 2  is independently ethynyl, substituted ethynyl, or and\n each R 3  is independently halo, \u2014O(C\u2550O)-alkyl, \u2014O(C\u2550O)-substituted alkyl, \u2014O(C\u2550O)-aryl, \u2014O(C\u2550O)-substituted aryl, \u2014O(C\u2550O)\u2014O-alkyl, \u2014O(C\u2550O)\u2014O-substituted alkyl, \u2014O(C\u2550O)\u2014O-aryl, \u2014O(C\u2550O)\u2014O-substituted aryl, \u2014O(SO 2 )-alkyl, \u2014O(SO 2 )-substituted alkyl, \u2014O(SO 2 )-aryl, or \u2014O(SO 2 )-substituted aryl.

Metadata:
- Claim Count in Document: 11.0
- Percentile: 90.0
- Lexical Diversity: 1.775
- Patent Class: 546.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['15760738', '15126420', '15126392', '15126402', '15126412']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7550616474005167
- 35 USC 102 Novelty (BERT): 0.5304462738602217
- Combined Prediction Score: 0.7326001100464872
- Mean Citation Score: 316.704922
- Max Citation Score: 349.4831
- Similarity Product: 259.097210195297

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test