PATENT CLAIM ANALYSIS

Application Number: 15945429
Application Type: Utility
Filing Date: 2018-04
Publication Date: 2018-08
Patent Classification: ["514", "210180"]

Abstract:
The invention relates to a compound of formula (I) wherein R 1  and R 2  are defined as in the description and in the claims. The compound of formula (I) can be used as a medicament.

Claim (Index 1):
A compound of formula (I) wherein A is \u2014C(O)\u2014 or \u2014CHCF 3 \u2014; R 1  is propyl, pyridinyl or R 3 ; R 2  is (A), (B), (C), (D), (E), (F) or (G); R 3  is (H); R 4  is hydrogen, alkyl or haloalkyl; R 5  is alkyl, haloalkyl, cycloalkyl, phenyl, halophenyl or alkoxyphenyl; R 6  is halophenyl; R 7  is halophenyl; R 8  is alkyl; R 9  is alkyl, cycloalkyl, halocycloalkyl, phenyl, halophenyl, alkylsulphanylphenyl, pyridinyl, halopyridinyl, oxanyl, azaspiro[3.3]heptyl, alkoxycarbonylazaspiro[3.3]heptyl, oxetanyl, pyrrolidinyl, alkoxycarbonylpyrrolidinyl, azetidinyl or alkylcarbonylazetidinyl; R 10  is phenyl; R 11  is halophenyl; R 12  is phenyl or halophenyl; R 13  is hydrogen, halogen, haloalkyl, haloalkoxy, cycloalkylalkoxy, phenylalkoxy, alkoxyalkoxy or cyano; R 14  is hydrogen, halogen or haloalkyl; and R 15  is hydrogen, halogen, cyano or haloalkyl; or a pharmaceutically acceptable salt or ester thereof; provided that N-[(1S)-1-[(3-chlorophenyl)methyl]-2-[(1-cyanocyclopropyl)amino]-2-oxoethyl]-3-(1,1-dimethylethyl)-1-methyl-1H-pyrazole-5-carboxamide is excluded.

Metadata:
- Claim Count in Document: 14.0
- Percentile: 91.0
- Lexical Diversity: 1.5
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['12761427', '15567668', '13148296', '15320155', '13049941']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7887807945663552
- 35 USC 102 Novelty (BERT): 0.5192469040075015
- Combined Prediction Score: 0.7618274055104699
- Mean Citation Score: 279.468204
- Max Citation Score: 312.96332
- Similarity Product: 229.99424350663665

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test