PATENT CLAIM ANALYSIS

Application Number: 16152735
Application Type: Utility
Filing Date: 2018-10
Publication Date: 2019-01
Patent Classification: ["544", "331000"]

Abstract:
Disclosed are inhibitors of human galactokinase of formula (I) that are useful in treating or preventing a galactokinase mediated disease or disorder, e.g., galactosemia. Also disclosed are a composition comprising a pharmaceutically acceptable carrier and at least one inhibitor of the invention, and a method of treating or preventing such disease or disorder in a mammal. Formula (I).

Claim (Index 15):
The method of claim  37 , wherein R 3  is selected from the group consisting of \u2014NH-alkyl, \u2014NH-cycloalkyl, \u2014NH-aryl, \u2014NH-alkylaryl, \u2014NH-heteroaryl, and \u2014NR 12  R 13  wherein R 12  and R 13  are each independently selected from the group consisting of hydrogen, alkyl, cycloalkyl, aryl, arylalkyl, and heteroaryl, or wherein R 12  and R 13  together form a heteroaryl or a heterocycloalkyl,\n wherein R 4  is selected from the group consisting of hydrogen and alkyl, wherein R 5  is heteroaryl, and wherein alkyl, aryl, heterocycloalkyl, carbocyclic ring, heterocyclic ring, arylalkyl, and heteroaryl groups are unsubstituted or optionally substituted with one or more substituents selected from the group consisting of alkyl, aryl, halo, trifluoromethyl, alkoxy, aryloxy, amino, alkylamino, and dialkylamino.

Metadata:
- Claim Count in Document: 48.0
- Percentile: 97.0
- Lexical Diversity: 1.61905
- Patent Class: 544.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['14346400', '14409374', '10715662', '10559405', '16119962']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.822409237029422
- 35 USC 102 Novelty (BERT): 0.5038544215097555
- Combined Prediction Score: 0.7905537554774553
- Mean Citation Score: 260.10813
- Max Citation Score: 287.9479
- Similarity Product: 212.9031591666221

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test