PATENT CLAIM ANALYSIS

Application Number: 15934176
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2018-09
Patent Classification: ["514", "378000"]

Abstract:
A compound of Formula (I)) or or a pharmaceutically acceptable salt thereof, is provided that has been shown to be useful for treating hearing loss or balance disorder: wherein R 1  through R 3 , and L are as defined herein.

Claim (Index 1):
A compound of Formula (I) or a pharmaceutically acceptable salt thereof, wherein:\n R 1  is selected from phenyl, thienyl, and furanyl, which are each independently optionally substituted by 1-2 F; \n L is C 5 -C 6  alkylene optionally substituted with 1-4 substituents independently selected from C 1-6  alkyl and halogen, wherein optionally a C 1-6  alkyl substituent is taken together with the carbon atoms to which it is attached to form a 3-membered cycloalkyl ring; \n R 2  and R 3  are taken together with the nitrogen atom to which they are attached to form a 4- to 10-membered heterocyclyl comprising carbon atoms and 1-3 heteroatoms independently selected from N and O, which is optionally substituted with 1-4 R 4 ; \n each R 4  is independently selected from C 1-6  alkyl, C 3-8  cycloalkyl, halogen, (C 0 -C 3  alkylene)-CN, C 1-6  haloalkyl, C 1 -C 6  haloalkoxy, (C 0 -C 6  alkylene)-OR 5 , (\u2550O), NH(C\u2550O)R 5 , NH(C\u2550O)OR 7 , NH(C\u2550O)N(R 5 ) 2 , (C\u2550O)N(R 7 ) 2 , (C\u2550O)R 5 , (C\u2550O)O(C 1-6 alkyl), (C\u2550O)O(C 3-8  cycloalkyl), S(\u2550O) 2 R 5 , S(\u2550O) 2 N(R 7 ) 2 , NHS(\u2550O) 2 R 5 , phenyl optionally substituted with 1-3 R 6  and 5- to 6-membered heteroaryl comprising carbon atoms and 1-3 heteroatoms independently selected from N, O and S optionally substituted with 1-3 R 6 ; \n each R 5  is independently selected from H, C 1-6  alkyl and C 3-8  cycloalkyl; \n each R 6  is independently selected from C 1-6  alkyl, C 3-8  cycloalkyl, halogen, CN, C 1-6  haloalkyl, C 1 -C 6  haloalkoxy, OR 5 , N(R 5 ) 2 , NH(C\u2550O)R 5 , (C\u2550O)N(R 5 ) 2 , (C\u2550O)R 5 , (C\u2550O)OR 5 , S(\u2550O) 2 R 5  and S(\u2550O) 2 N(R 5 ) 2 ; and \n each R 7  is independently selected from H, C 1-6  alkyl, C 3-8  cycloalkyl optionally substituted with 1-2 OR 5 , (C 0 -C 3  alkylene)-CN and (C 0 -C 3  alkylene)-OR 5 .

Metadata:
- Claim Count in Document: 5.0
- Percentile: 90.0
- Lexical Diversity: 1.11905
- Patent Class: 514.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['14381187', '13993198', '14977508', '13360050', '15124264']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7454942131364747
- 35 USC 102 Novelty (BERT): 0.5074615394087123
- Combined Prediction Score: 0.7216909457636984
- Mean Citation Score: 282.68990799999995
- Max Citation Score: 290.67834
- Similarity Product: 228.0968285452008

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test