PATENT CLAIM ANALYSIS

Application Number: 15909088
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2018-07
Patent Classification: ["514", "156000"]

Abstract:
Disclosed are novel compounds of specific chemical structures having inhibitory activity on c-Myc/Max/DNA complex formation or pharmaceutically acceptable salts thereof.

Claim (Index 4):
The compound of  claim 1  having the structure of Formula 3a or 3b, or a pharmaceutically acceptable salt thereof: wherein, R 1a  to R 1d , R 3 , and n are the same as defined for Formula 1a or 1b in  claim 1 ; R 4a  and R 4b  are each independently hydrogen, a halogen, C 1-4  alkyl, C 1-4  haloalkyl, or C 1-4  alkyl in which one or more hydrogens are substituted with a substituent other than halogen; Ar is phenyl, a heteroaryl being 5-6-membered and having a heteroatom selected independently from N, S, and O, or a biheteroaryl being 8-12-membered and having a heteroatom selected independently from N, S, and or O, wherein Ar is unsubstituted or optionally substituted with one or more of a halogen, C 1-6  alkyl, C 1-6  alkylthio, C 1-6  haloalkyl, C 1-6  haloalkylthio, C 1-6  alkoxy, C 1-6  haloalkoxy, C 2-10  alkenyl, C 2-10  haloalkenyl, C 2-10  alkynyl, C 2-10  haloalkynyl, a hydroxyl group, COOH, nitro, cyano, C 1-6  alkoxycarbonyl, amino, C 1-6  alkylamino, alkyl)amino, amino(C 1-6 )alkyl, (C 1-6 )alkylamino(C 1-6 )alkyl, (C 1-6 )alkoxy(C 1-6 )alkylamino, (C 1-6 )alkylamino(C 1-6 ) alkylamino, C 1-6  alkanoyl, SF 5 , S(O)CF 3 , SCF 3 , NHC(\u2550O)CH 3 , C(\u2550O)NHCH 3 , NHSO 2 CH 3 , C 3-7  cycloalkyl, an aryl, benzoyl, a heterocycle, a heteroaryl, phenyl, oxazole, pyrazole, pyrrole, imidazole, thiazole, thiophene, pyridine, pyrimidine, furan, indole, benzopyrazole, benzothiazole, benzooxazole, isoxazole, benzoimidazole, and benzothiophene, wherein the substituent of Ar is unsubstituted or optionally substituted with one or more of CF3, a halogen, (C 1-3 )alkyl, (C 1-3 )haloalkyl, hydrogen, COOH, nitro, cyano, amino, di(C 1-3  alkyl)amino, NHC(\u2550O)CH 3 , and C(\u2550O)NHCH 3 .

Metadata:
- Claim Count in Document: 3.0
- Percentile: 90.0
- Lexical Diversity: 1.0
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['11208437', '15663179', '15586343', '14647521', '11015348']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8052870194020003
- 35 USC 102 Novelty (BERT): 0.5264085703588441
- Combined Prediction Score: 0.7773991744976847
- Mean Citation Score: 314.747628
- Max Citation Score: 325.22043
- Similarity Product: 246.02572914995315

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test