PATENT CLAIM ANALYSIS

Application Number: 15973569
Application Type: Utility
Filing Date: 2018-05
Publication Date: 2018-11
Patent Classification: ["514", "210200"]

Abstract:
Series of 2-phenyl-4-methylthiazole analogues are disclosed as potential therapeutic agents for the treatment of bacterial infections, especially methicillin-resistant  Straphylococcus aureus  (MRSA) related infections. A method for the treatment of MRSA-related infections is also claimed.

Claim (Index 1):
A compound having formula (I) or a pharmaceutically acceptable salt, hydrate, or solvate thereof, wherein: R 1  is hydrogen, an amino, alkylamino, aminoalkylamino, aminoalcohol, cycloalkylamino, hydrazines, guanidino, thioguanidino, cyano amino, acyl, ester, alkyl, alkenyl, alkynyl, heteroalkyl, heteroalkenyl, heteroalkynyl, heterocyclyl, cycloalkyl, cycloalkenyl, cycloheteroalkyl, cycloheteroalkenyl, aryl, heteroaryl, arylalkyl, arylalkenyl, or arylalkynyl, each of which is optionally substituted; and R 2  is a halo, azido, cyano, nitro, hydroxy, amino, thio, carboxy, ester, amide, and derivatives thereof, and acyl, sulfoxyl, sulfonyl, phosphate, phosphoryl, alkyl, alkenyl, alkynyl, heteroalkyl, heteroalkenyl, heteroalkynyl, heterocyclyl, cycloalkyl, cycloalkenyl, cycloheteroalkyl, cycloheteroalkenyl, aryl, heteroaryl, arylalkyl, arylalkenyl, and arylalkynyl, each of which is optionally substituted; and R 3  is hydrogen, an alkyl, alkenyl, alkynyl, heteroalkyl, heteroalkenyl, heteroalkynyl, heterocyclyl, cycloalkyl, cycloalkenyl, cycloheteroalkyl, cycloheteroalkenyl, acyl, alkoxyl, aryl, heteroaryl, arylalkyl, arylalkenyl, or arylalkynyl, each of which is optionally substituted.

Metadata:
- Claim Count in Document: 8.0
- Percentile: 93.0
- Lexical Diversity: 1.25806
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15144311', '14111157', '14110391', '13388712', '14119673']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8148364077096022
- 35 USC 102 Novelty (BERT): 0.5529591980257987
- Combined Prediction Score: 0.7886486867412219
- Mean Citation Score: 379.947854
- Max Citation Score: 431.57492
- Similarity Product: 315.7688620596528

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test