PATENT CLAIM ANALYSIS

Application Number: 15987277
Application Type: Utility
Filing Date: 2018-05
Publication Date: 2018-12
Patent Classification: ["514", "210180"]

Abstract:
Compounds of formula (I) defined herein are p38 MAPK inhibitors and are useful as anti-inflammatory agents in the treatment of, inter alia, diseases of the respiratory tract.

Claim (Index 2):
A compound or pharmaceutically acceptable salt according to  claim 1 , wherein B is a group of formula (IIa), (IIb), (IIc), (IId), (IIe), (IIg), (IIh), or (IIi): R 1  is H, \u2014CN, linear or branched (C 1 -C 4 )alkyl, (R 8 )(R 9 )NC(O)\u2014, R 12 O\u2014(C 1 -C 4 )alkylene-, (R 8 )(R 9 )N\u2014(C 1 -C 4 )alkylene-, (C 1 -C 4 )alkyl-S(O) 2 NH\u2014, (C 1 -C 4 )alkyl-S\u2014, (C 1 -C 4 )alkyl-OC(O)\u2014, or (R 8 )(R 9 )N\u2014(C 1 -C 4 )alkylene-O\u2014(C 1 -C 4 )alkylene-; R 6  and R 7  form, together with the nitrogen atom to which they are attached, an optionally substituted 4-7 membered saturated heterocyclic monocyclic ring system, optionally containing a further oxygen or nitrogen heteroatom; R 8  is H, linear or branched \u2014(C 1 -C 4 )alkyl-; R 9  is linear or branched (C 1 -C 4 )alkyl-, optionally substituted (C 3 -C 7 )cycloalkyl-, R 12 O\u2014(C 1 -C 4 )alkylene-, or (R 10 )(R 11 )N\u2014(C 1 -C 4 )alkylene-, wherein said (C 1 -C 4 )alkylene- in (R 10 )(R 11 )N\u2014(C 1 -C 4 )alkylene- may be optionally substituted with one or more groups selected from the group consisting of linear or branched (C 1 -C 4 )alkyl-, spiro-(C 1 -C 6 )cycloalkyl, and spiro-(C 1 -C 6 )heterocycloalkyl; or R 8  and R 9  may form, together with the nitrogen atom to which they are attached, an optionally substituted 4-7 membered saturated heterocyclic monocyclic ring system, optionally containing a further oxygen or nitrogen heteroatom; R 10  is linear or branched (C 1 -C 4 )alkyl- or (C 3 -C 7 )cycloalkyl-; R 11  is linear or branched (C 1 -C 4 )alkyl- or R 12 O\u2014(C 1 -C 4 )alkylene-; or R 10  and R 11  may form, together with the nitrogen atom to which they are attached, an optionally substituted 4-7 membered saturated heterocyclic monocyclic ring system, optionally containing a further oxygen or nitrogen heteroatom; n is 3; m is 1; and z is 1.

Metadata:
- Claim Count in Document: 2.0
- Percentile: 93.0
- Lexical Diversity: 1.18519
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15388350', '14296730', '14895718', '14868516', '14296794']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.850144249168643
- 35 USC 102 Novelty (BERT): 0.5933747726519641
- Combined Prediction Score: 0.8244673015169751
- Mean Citation Score: 514.875808
- Max Citation Score: 525.1804
- Similarity Product: 436.1901229397296

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test