PATENT CLAIM ANALYSIS

Application Number: 15886014
Application Type: Utility
Filing Date: 2018-02
Publication Date: 2018-06
Patent Classification: ["514", "252000"]

Abstract:
The disclosed compounds relate to treatments and therapies for protein kinase-associated disorders. There is also a need for compounds useful in the treatment or prevention or amelioration of one or more symptoms of cancer, transplant rejections, and autoimmune diseases. Furthermore, there is a need for methods for modulating the activity of protein kinases, such as CDK1, CDK2, CDK4, CDK5, CDK6, CDK7, CDK8 and CDK9, using the compounds provided herein.

Claim (Index 21):
A compound of formula I(a): or a pharmaceutically acceptable salt thereof, wherein: R 50  is CONR 54 R 55 , or CN; R 51  is C 3-14 cycloalkyl which may be unsubstituted or substituted by C 1-3 alkyl, or OH; Z is CH or N; and V is NR 56  or CHR 57 ; R 54  and R 55  are independently H, C 1-3 alkyl, R 52 , R 53  R 56 , and R 57  are independently H, C 1-8 alkyl, C 3-14 cycloalkyl, C 1-8 haloalkyl, NR 58 R 59 , C(O)OR 60 , C(O)C 1-8 alkyl, C 0-8 alkylC(O)C 0-8 alkyl-NR 61 R 62 , C 1-8 alkoxy, C 1-8 alkylOR 63 , C(O)-5-14cycloheteroalkyl group, C 3-14 cycloalkyl group, each of which when not H may be substituted by one or more of C 1-8 alky, OH, or CN; R 58 , R 59 , R 60 , R 61 , R 62 , and R 63  are H or C 1-8 alkyl.

Metadata:
- Claim Count in Document: 8.0
- Percentile: 88.0
- Lexical Diversity: 1.53704
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['13060154', '14158358', '12545322', '13579359', '13786955']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8137250796779071
- 35 USC 102 Novelty (BERT): 0.6190700961384676
- Combined Prediction Score: 0.7942595813239631
- Mean Citation Score: 489.78964
- Max Citation Score: 549.5182
- Similarity Product: 513.7363361583709

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test