PATENT CLAIM ANALYSIS

Application Number: 16162835
Application Type: Utility
Filing Date: 2018-10
Publication Date: 2019-06
Patent Classification: ["544", "360000"]

Abstract:
The invention relates to triazole compounds of formula I and I′ or pharmaceutically acceptable salts thereof, useful as modulators of demyelinating diseases: The invention also provides pharmaceutically acceptable compositions comprising the compounds of the invention, methods of using the compositions and kits thereof in the treatment of various demyelinating and neurodegenerative diseases, including multiple sclerosis.

Claim (Index 27):
The compound of  claim 10 , or a pharmaceutically acceptable salt thereof, wherein R 4  is\n a) phenyl,\n the phenyl being optionally substituted with one substituent selected from the group consisting of halogen, cyano, \u2014S(O) 2 C 1-4 alkyl, \u2014S(O)C 1-4 alkyl, \u2014SC 1-4 alkyl, C 1-4 alkyl, C 1-4 haloalkyl, \u2014OC 1-4 alkyl, \u2014OC 1-4 haloalkyl, \u2014C 1-4 alkylene-OC 1-4 alkyl, \u2014C 1-4 alkylene-N(C 1-4 alkyl)(C 1-4 alkyl), \u2014N(C 1-4 alkyl)(C 1-4 alkylene-OC 1-4 alkyl), or a 4- to 8-membered monocyclic heterocycle containing 1-2 nitrogen atoms, the 4- to 8-membered monocyclic heterocycle being independently optionally substituted with 1-2 substituents independently selected from the group consisting of halogen, \u2014OC 1-4 alkyl, C 1-4 alkyl, \u2014C 1-4 alkylene-OC 1-4 alkyl, and \u2014C 1-4 alkylene-OH, \n the phenyl being further optionally substituted with 1-2 substituents independently selected from the group consisting of halogen and C 1-4 alkyl; \n b) pyrazinyl,\n the pyrazinyl being optionally substituted with 1-3 C 1-4 alkyl groups; \n c) pyrimidinyl,\n the pyrimidinyl being optionally substituted with one substituent selected from halogen, \u2014S(O) 2 C 1-4 alkyl, \u2014S(O)C 1-4 alkyl, \u2014SC 1-4 alkyl, C 1-4 alkyl, \u2014OC 1-4 alkyl, or \u2014C 1-4 alkylene-OC 1-4 alkyl, the pyrimidinyl being further optionally substituted with C 1-4 alkyl; \n d) pyridazinyl; or e) pyridinyl,\n the pyridinyl being optionally substituted with one substituent selected from the group consisting of halogen, hydroxyl, C 1-4 alkyl, and a 4- to 8-membered monocyclic heterocycle containing 1-2 nitrogen atoms, \n the pyridinyl being further optionally substituted with 1-2 substituents selected from halogen and C 1-4 alkyl.

Metadata:
- Claim Count in Document: 2.0
- Percentile: 97.0
- Lexical Diversity: 1.53846
- Patent Class: 544.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['15173177', '15037090', '15287922', '14509793', '11703522']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8198326425762072
- 35 USC 102 Novelty (BERT): 0.6243890311590349
- Combined Prediction Score: 0.80028828143449
- Mean Citation Score: 421.580412
- Max Citation Score: 592.3917
- Similarity Product: 527.4438499993444

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test