PATENT CLAIM ANALYSIS

Application Number: 16141397
Application Type: Utility
Filing Date: 2018-09
Publication Date: 2019-03
Patent Classification: ["549", "483000"]

Abstract:
The present invention relates to fungicidal N-cycloalkyl-N-[(heterocyclylphenyl)methylene] carboxamide derivatives and their thiocarbonyl derivatives, their process of preparation and intermediate compounds for their preparation, their use as fungicides; particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions.

Claim (Index 20):
A compound of formula (Xa) wherein\n Z 2  and Z 3 , which can be the same or different, are a hydrogen atom; non-substituted C 1 -C 8 -alkyl; non-substituted C 2 -C 8 -alkenyl; non-substituted C 2 -C 8 -alkynyl; a halogen atom; non-substituted C 1 -C 8 -alkoxy; non-substituted C 2 -C 8 -alkenyloxy; or non-substituted C 2 -C 8 -alkynyloxy; \n A is A 13 \n wherein: R 34  is a hydrogen atom; a halogen atom; substituted or non-substituted C 1 -C 5 -alkyl; substituted or non-substituted C 3 -C 5 -cycloalkyl; C 1 -C 5 -halogenoalkyl comprising up to 9 halogen atoms that can be the same or different substituted or non-substituted C 1 -C 5 -alkoxy; substituted or non-substituted C 2 -C 5 -alkynyloxy or C 1 -C 5 -halogenoalkoxy comprising up to 9 halogen atoms that can be the same or different; R 35  is a hydrogen atom; a halogen atom; substituted or non-substituted C 1 -C 5 -alkyl; a cyano; substituted or non-substituted C 1 -C 5 -alkoxy; substituted or non-substituted C 1 -C 5 -alkylsulfanyl; C 1 -C 5 -halogenoalkyl comprising up to 9 halogen atoms that can be the same or different C 1 -C 5 -halogenoalkoxy comprising up to 9 halogen atoms that can be the same or different amino; substituted or non-substituted C 1 -C 5 -alkylamino or substituted or non-substituted di(C 1 -C 5 -alkyl)amino; R 36  is a hydrogen atom or substituted or non-substituted C 1 -C 5 -alkyl; X a1  is a halogen atom; substituted or non-substituted C 1 -C 8 -alkyl; C 1 -C 8 -halogenoalkyl comprising up to 9 halogen atoms which can be the same or different; substituted or non-substituted C 3 -C 7 -cycloalkyl; tri(C 1 -C 8 -alkyl)silyl; substituted or non-substituted C 1 -C 8 -alkoxy; or substituted or non-substituted C 1 -C 8 -alkylsulfanyl; X a2  is hydrogen, a halogen atom; substituted or non-substituted C 1 -C 8 -alkyl; C 1 -C 8 -halogenoalkyl comprising up to 9 halogen atoms which can be the same or different; substituted or non-substituted C 3 -C 7 -cycloalkyl; tri(C 1 -C 8 -alkyl)silyl; substituted or non-substituted C 1 -C 8 -alkoxy; or substituted or non-substituted C 1 -C 8 -alkylsulfanyl, and U 2  is a halogen atom or a triflate group, providing that (Xa) does not represent:\n N-(2,5-dichlorobenzyl)-3-(difluoromethyl)-5-fluoro-1-methyl-1H-pyrazole-4-carboxamide; \n N-[1-(2,5-dichlorophenyl)ethyl]-3-(difluoromethyl)-5-fluoro-1-methyl-1H-pyrazole-4-carboxamide; \n N-[2-(2,5-dichlorophenyl)propan-2-yl]-3-(difluoromethyl)-5-fluoro-1-methyl-1H-pyrazole-4-carboxamide; \n N-[1-(2,5-dichlorophenyl)cyclopropyl]-3-(difluoromethyl)-5-fluoro-1-methyl-1H-pyrazole-4-carboxamide; \n 5-chloro-N-[1-(2,5-dichlorophenyl)ethyl]-3-(difluoromethyl)-1-methyl-1H-pyrazole-4-carboxamide; \n 5-chloro-N-[2-(2,5-dichlorophenyl)propan-2-yl]-3-(difluoromethyl)-1-methyl-1H-pyrazole-4-carboxamide; \n 5-chloro-N-[1-(2,5-dichlorophenyl)cyclopropyl]-3-(difluoromethyl)-1-methyl-1H-pyrazole-4-carboxamide; \n 5-chloro-N-(2,5-dichlorobenzyl)-3-(difluoromethyl)-1-methyl-1H-pyrazole-4-carboxamide; \n N-(5-bromo-2-fluorobenzyl)-1,3,5-trimethyl-1H-pyrazole-4-carboxamide; \n N-(5-bromo-2-fluorobenzyl)-3,5-dimethyl-1H-pyrazole-4-carboxamide; \n 1-methyl-N-[1-(2,4,5-trichlorophenyl)ethyl]-3-(trifluoromethyl)-1H-pyrazole-4-carboxamide; \n 3-(difluoromethyl)-1-methyl-N-[1-(2,4,5-trichlorophenyl)ethyl]-1H-pyrazole-4-carboxamide; \n N-(5-chloro-2-fluorobenzyl)-1-methyl-5-propoxy-3-(trifluoromethyl)-1H-pyrazole-4-carboxamide; or \n N-(2,5-dichlorobenzyl)-1-methyl-5-propoxy-3-(trifluoromethyl)-1H-pyrazole-4-carboxamide, \n a salt thereof.

Metadata:
- Claim Count in Document: 35.0
- Percentile: 97.0
- Lexical Diversity: 1.39535
- Patent Class: 549.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['14395038', '14388179', '14361534', '15176653', '15566159']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7680889934532928
- 35 USC 102 Novelty (BERT): 0.575176965792262
- Combined Prediction Score: 0.7487977906871898
- Mean Citation Score: 414.81178
- Max Citation Score: 496.60413
- Similarity Product: 396.0992542096514

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 0
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test