PATENT CLAIM ANALYSIS

Application Number: 15776094
Application Type: Utility
Filing Date: 2018-05
Publication Date: 2018-11
Patent Classification: ["514", "236200"]

Abstract:
Compounds of formula I or a stereoisomer or pharmaceutically-acceptable salt thereof, are useful in the modulation of IL-12, IL-23 and/or IFNα, by acting on Tyk-2 to cause signal transduction inhibition.

Claim (Index 4):
The compound according to  claim 3 wherein\n R 1  is \u2014NHR 2 ; \n R 2  is H, C 1 -C 6  alkyl, C 3 -C 8  cycloalkyl, hydroxy C 1 -C 6  alkyl, alkoxy C 1 -C 6  alkyl, C 3 -C 8  cycloalkyl C 1 -C 6  alkyl-, di (C 1 -C 4 ) alkyl aminoalkyl-, aryl, heteroaryl, or heterocyclyl C 1 -C 6  alkyl-, said heteroaryl group substituted with 0-2 R 8  \n R 3  is H, C 3 -C 10 -mono or bicyclic cycloalkyl, C 1 -C 6  alkyl, C 4 -C 10  mono or bicyclic aryl, or 4- to 10-membered mono or bicyclic heterocyclyl, each heterocyclyl containing 1-3 heteroatoms selected from N, O, and S, any of said groups other than H substituted with 0-4 R 6 ; \n R 4  is H, C 1 -C 6  alkyl, 3- to 10-membered mono or bicyclic cycloalkyl, 6- to 10-membered mono or bicyclic aryl, 4- to 10-membered mono or bicyclic heterocyclyl, or substituted 4- to 10-mono or bicyclic heteroaryl, each heterocyclyl or heteroaryl containing 1-3 heteroatoms selected from N, O, and S, any of said groups other than H substituted with 0-4 R 7 ; \n R 5  is H or C 1 -C 4  alkyl; \n R 6  is H, halo, CN, OH, C 1 -C 4  alkyl, (R 5 ) n N, \u2014NR 5 COR 5 , R 5 O, \u2014CON(R 5 ) n , \u2014SO n R 5 , \n n is 1 or 2; \n R 7  is H, halo, CN, CF 3 , C 1 -C 4  alkyl, C 1 -C 4  alkoxy, \u2014CONHC 1 -C 6  alkyl, \u2014CONH halo C 1 -C 6  alkyl, \u2014CONH halo C 1 -C 6  alkoxy, heteroaryl, alkynyl (\u2014CCR 5 ), alkenyl \u2014CR 5 \u2550C(R 5 ) n  or aryl, said aryl and heteroaryl groups substituted with 0-2 R 8 ; \n R 8  is H, halo, CF 3 , C 1 -C 4  alkyl or C 1 -C 4  alkoxy; \n or a pharmaceutically acceptable salt, tautomer or stereoisomer thereof.

Metadata:
- Claim Count in Document: 13.0
- Percentile: 93.0
- Lexical Diversity: 1.13333
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15034915', '15289437', '14441213', '14441193', '15480787']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8686738618627392
- 35 USC 102 Novelty (BERT): 0.6010195621175127
- Combined Prediction Score: 0.8419084318882166
- Mean Citation Score: 569.3277099999998
- Max Citation Score: 593.6887
- Similarity Product: 449.6393184382201

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test