PATENT CLAIM ANALYSIS

Application Number: 16148774
Application Type: Utility
Filing Date: 2018-10
Publication Date: 2019-01
Patent Classification: ["514", "300000"]

Abstract:
A process for producing a compound of the following Formula (VII-CR): The process involving providing a compound represented by the following Formula (VI): in a case where the R 3 ONHC(═O) side chain in the compound of the Formula (VI) has a protecting group, removing the protecting group from the compound of the Formula (VI) with an acid, and adding an ester-based poor solvent to the resultant reaction solution to precipitate the compound of Formula (VII-CR), wherein in the compounds of the Formulas (VII-CR) and (VI), R 3  is a C 1-6  alkyl or a heterocycle.

Claim (Index 2):
The process according to  claim 1 , wherein R 3  in the Formulas (VI) and (VII-CR) is each independently selected from the group consisting of:\n 2-(tert-butoxycarbonylamino)ethyl, 2-aminoethyl, 2-((tert-butoxycarbonyl)(methyl)amino)ethyl, 2-(methylamino)ethyl, 2-((tert-butoxycarbonyl)(isopropyl)amino)ethyl, 2-(isopropylamino)ethyl, 2-(dimethylamino)ethyl, (2S)-2-((tert-butoxycarbonyl)amino)propyl, (2S)-2-(amino)propyl, (2R)-2-((tert-butoxycarbonyl)amino)propyl, (2R)-2-(amino)propyl, 3-((tert-butoxycarbonyl)amino)propyl, 3-(amino)propyl, (2S)-tert-butoxycarbonylazetidin-2-ylmethyl, (2S)-azetidin-2-ylmethyl, (2R)-tert-butoxycarbonylpyrrolidin-2-ylmethyl, (2R)-pyrrolidin-2-ylmethyl, (3R)-tert-butoxycarbonylpiperidin-3-ylmethyl, (3R)-piperidin-3-ylmethyl, (3S)-tert-butoxycarbonylpyrrolidin-3-yl, (3S)-pyrrolidin-3-yl, 1-(tert-butoxycarbonyl)azetidin-3-yl and azetidin-3-yl.

Metadata:
- Claim Count in Document: 5.0
- Percentile: 97.0
- Lexical Diversity: 2.06897
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15027956', '15023976', '15613620', '15973861', '14872988']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8169352418022628
- 35 USC 102 Novelty (BERT): 0.6586588541419526
- Combined Prediction Score: 0.8011076030362319
- Mean Citation Score: 370.669024
- Max Citation Score: 464.994
- Similarity Product: 422.5498819431065

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 0
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test