PATENT CLAIM ANALYSIS

Application Number: 16438135
Application Type: Utility
Filing Date: 2019-06
Publication Date: 2019-10
Patent Classification: ["544", "281000"]

Abstract:
Compounds of Formula (00A) and methods of use as Janus kinase inhibitors are described herein.

Claim (Index 2):
The compound of  claim 1 , further defined as a compound of Formula (II): wherein:\n w is 0 or 1; \n R 0b  is H or NH 2 ; \n R 1b  is selected from the group consisting of\n a. H, \n b. C 1 -C 6  alkyl optionally substituted by OH, halo, CN, \u2014O\u2014(C 1 -C 6  alkyl), naphthylenyl, 5-6 membered heteroaryl, or \u2014C(O)NR v R w , wherein R v  and R w  are independently H or C 1 -C 6  alkyl optionally substituted by halo, \n c. \u2014(C 1 -C 6  alkylene)-3-6 membered cycloalkyl wherein the cycloalkyl is optionally substituted by CN, \n d. \u2014(C 1 -C 6  alkylene)-phenyl wherein the alkyl is optionally substituted by halo and wherein the phenyl is optionally substituted by OH, halo, CF 3 , C 1 -C 6  alkyl, \u2014O\u2014(C 1 -C 6  alkyl) or \u2014O-phenyl, \n e. \u2014(C 1 -C 6  alkylene)-4-6 membered heterocycloalkyl wherein the heterocycloalkyl is optionally substituted by halo or C 1 -C 6  alkyl, \n f. \u2014(C 1 -C 6  alkylene)-O-phenyl wherein the phenyl is optionally substituted by halo or C 1 -C 6  alkyl, or \n g. 3-6 membered cycloalkyl; \n \n R 2b  is selected from the group consisting of H, C 1 -C 6  alkyl optionally substituted by halo, or C 2 -C 5  alkenyl; \n or R 1b  and R 2b  together form a 3-11 membered heterocycloalkyl optionally substituted by OH; \n R 3b  is absent or methyl, wherein when R 3b  is methyl, the nitrogen to which it is attached is N+ and w is 1; \n R 4b  is a bond or C 1 -C 6  alkylene; \n R 5b  is selected from the group consisting of H, OH, and phenyl; and \n Ring F is a 3-7 membered heterocycloalkyl wherein p 1b  is 0, 1 or 2 and p 2b  is 0, 1 or 2; \n wherein w is equal to 1 only when R 3b  is methyl.

Metadata:
- Claim Count in Document: 50.0
- Percentile: 100.0
- Lexical Diversity: 1.05882
- Patent Class: 544.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15139164', '15543826', '14904801', '14451600', '15257926']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8099969587729821
- 35 USC 102 Novelty (BERT): 0.5823799968744483
- Combined Prediction Score: 0.7872352625831287
- Mean Citation Score: 405.063252
- Max Citation Score: 495.0762
- Similarity Product: 421.0564001939535

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 0
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test