PATENT CLAIM ANALYSIS

Application Number: 15758662
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2018-10
Patent Classification: ["424", "078170"]

Abstract:
The present invention relates in general to polymer-bioactive agent conjugates for delivering a bioactive agent to a subject. The polymer-bioactive agent conjugates contain triazole moieties in the polymer backbone and a bioactive moiety selected from quinolones, NSAIDs and mixtures thereof. The present invention also relates to methods for preparing the polymer conjugates using click cycloaddition chemical reactions, to monomer-bioactive agent conjugates suitable for preparing the polymer conjugates, and to pharmaceutical products comprising the polymer conjugates for the post-surgical care to treat or prevent infections, provide analgesia and treat inflammation.

Claim (Index 55):
A polymer-bioactive agent conjugate which is a copolymer of at least one monomer of formula (IV): where:\n X may be the same or different at each occurrence and represents a terminal functional group comprising an alkyne or an azide; \n Q is independently selected at each occurrence and may be present or absent and when present, represents a linking group; \n R is an optionally substituted linear or branched hydrocarbon and may comprise optionally substituted aromatic hydrocarbon or heteroaromatic hydrocarbon; \n Z is a cleavable linking group; and \n D is a bioactive agent selected from the group consisting of quinolones and NSAIDs; \n and a monomer of formula (V):\n A-L\ue8a0A] n  \u2003\u2003(V) \n where:\n A may be the same or different at each occurrence and represents a group comprising a terminal functional group comprising an alkyne or an azide functionality, wherein said terminal functional group is complementary to the terminal functional group of X; \n L is an optionally substituted linker group; and \n n is an integer and is at least 1.

Metadata:
- Claim Count in Document: 53.0
- Percentile: 90.0
- Lexical Diversity: 1.81132
- Patent Class: 424.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['14772981', '15435784', '15458546', '14409612', '13082841']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7937424180303664
- 35 USC 102 Novelty (BERT): 0.5901961393106278
- Combined Prediction Score: 0.7733877901583925
- Mean Citation Score: 466.697574
- Max Citation Score: 501.03647
- Similarity Product: 477.180578308372

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 0
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test