PATENT CLAIM ANALYSIS

Application Number: 15566418
Application Type: Utility
Filing Date: 2018-02
Publication Date: 2018-07
Patent Classification: ["514", "210000"]

Abstract:
Compounds of formula I are provided. Also provided are methods of preparing the compounds of formula (I), and methods of using the compounds of formula (I) as a negative allosteric modulator of a metabotropic glutamate receptor (mGluR) subtype 5.

Claim (Index 2):
The compound of  claim 1 , wherein R 2  and R 3  are each independently selected from the group consisting of hydrogen, substituted or unsubstituted phenyl, substituted or unsubstituted 3-7 membered heteroaryl, substituted or unsubstituted 5-7 membered aryl-methylene, 3-7 membered heterocyclyl-methylene, while each heterocyclyl independently contains 1 to 4 heteroatoms selected from oxygen, sulfur and nitrogen; R 2  and R 3  are not simultaneously hydrogen;\n or R 2  and R 3  together with the attached N atom form a group selected from the group consisting of substituted or unsubstituted hetero spirocyclic ring, substituted or unsubstituted fused heterocyclic ring; wherein the substituted means one or more hydrogen atoms of the group are substituted by substituents selected from the group consisting of halogen, C1-C6 alkyl, C1-C6 alkoxy, halogen-substituted C1-C6 alkoxy, cyano, nitro, amino, hydroxy, hydroxymethyl, carboxy, mercapto, sulfonyl, or trifluoromethyl.

Metadata:
- Claim Count in Document: 22.0
- Percentile: 88.0
- Lexical Diversity: 1.71429
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['14344957', '12908588', '15771920', '12912124', '13542234']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8374117394948496
- 35 USC 102 Novelty (BERT): 0.5287261288085555
- Combined Prediction Score: 0.8065431784262201
- Mean Citation Score: 333.88199999999995
- Max Citation Score: 349.1565
- Similarity Product: 258.77081273674963

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 0
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test