PATENT CLAIM ANALYSIS

Application Number: 15778168
Application Type: Utility
Filing Date: 2018-05
Publication Date: 2018-10
Patent Classification: ["514", "259310"]

Abstract:
The present invention relates to a novel azole derivative as an apelin receptor agonist and a method for treating cardiovascular disease, diabetic disease, renal disease, hypertension, and arteriosclerosis, etc., using the same. The present invention provides a compound represented by formula (I) or a pharmacologically acceptable salt thereof wherein X 1  represents —NH═ or —CH═, X 2  represents —CH═ or —N═, R 1  and R 2  each represent a C 1  to C 6  alkoxy group or the like, R 3  represents a heteroaryl group (the heteroaryl group is optionally substituted by a methyl group or the like) or the like, and R 4  represents a C 1  to C 6  alkylthio group or a C 2  to C 6  alkenyl group (the C 1  to C 6  alkylthio group and the C 2  to C 6  alkenyl group are each optionally substituted by one carboxy group or the like) or the like.

Claim (Index 25):
The compound according to any one of  claims 1  to  11  or a pharmacologically acceptable salt thereof, wherein R 4  is a heteroaryl-C 1  to C 6  alkylthio group, or a heteroaryl-C 2  to C 6  alkenyl group (the heteroaryl-C 1  to C 6  alkylthio group and the heteroaryl-C 2  to C 6  alkenyl group are each optionally substituted at the heteroaryl group moiety by 1 or 2 oxo groups).

Metadata:
- Claim Count in Document: 43.0
- Percentile: 93.0
- Lexical Diversity: 2.40845
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['10718337', '13995300', '10344157', '14322505', '12397132']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8190956863088621
- 35 USC 102 Novelty (BERT): 0.5372108627381956
- Combined Prediction Score: 0.7909072039517955
- Mean Citation Score: 366.950764
- Max Citation Score: 379.27014
- Similarity Product: 289.0386017280007

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test