PATENT CLAIM ANALYSIS

Application Number: 16179709
Application Type: Utility
Filing Date: 2018-11
Publication Date: 2019-03
Patent Classification: ["514", "243000"]

Abstract:
The present invention provides a method for treating a disease, disorder or condition associated with GPR139 using compounds of formula 1: which are agonists of GPR139, certain compounds encompassed by formula 1, pharmaceutical compositions thereof, processes for making the compounds, and intermediates thereof.

Claim (Index 19):
A method of treating a disease, disorder or condition associated with GPR 139  in a subject, the method comprising administering to the subject a compound of formula 1, or a pharmaceutically acceptable salt thereof, wherein: m is selected from 0, 1, and 2; n is selected from 0, 1, and 2; each R 1  is independently selected from the group consisting of cyano, halo, hydroxy, amino, C 1-4  alkyl, C 1-4  alkoxy, trifluoromethyl, and trifluoromethoxy; R 2  is selected from the group consisting of hydrogen and C 1-4  alkyl; R 3  is selected from the group consisting of hydrogen and methyl; each R 4  is independently selected from the group consisting of cyano, halo, hydroxy, amino, C 1-4  alkyl, C 1-4  alkoxy, trifluoromethyl, fluoromethoxy, difluoromethoxy, and trifluoromethoxy; G is selected from the group consisting of \u2014CHR 5 \u2014, \u2014CHR 5 \u2014CH 2 \u2014, and \u2014CH 2 \u2014CHR 5 \u2014; and R 5  is selected from the group consisting of hydrogen, trifluoromethyl, and C 1-4  alkyl.

Metadata:
- Claim Count in Document: 44.0
- Percentile: 98.0
- Lexical Diversity: 1.35135
- Patent Class: 514.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['14946194', '15683589', '15382490', '13509442', '13824174']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8322198505181447
- 35 USC 102 Novelty (BERT): 0.6526601207533409
- Combined Prediction Score: 0.8142638775416644
- Mean Citation Score: 524.891476
- Max Citation Score: 645.68604
- Similarity Product: 612.6221601747253

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 0

Dataset: test