PATENT CLAIM ANALYSIS

Application Number: 15942345
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2018-08
Patent Classification: ["540", "360000"]

Abstract:
A compound is represented as Formula I, a tautomer thereof, a stereoisomer thereof, or a pharmaceutically acceptable salt thereof: Compounds of Formula I are inhibitors of N-acylethanolamine hydrolyzing acid amidase (NAAA).

Claim (Index 1):
A compound of Formula I, a tautomer thereof, a stereoisomer thereof, or a pharmaceutically acceptable salt thereof: wherein:\n M is N, C, or CR, wherein R is H or alkyl; \n Z is NCS, \u2014(CH 2 ) n NCS, CN, \u2014(CH 2 ) n CN, or \u2014CR 1 R 2 CN, wherein n is 1, 2, 3, 4, or 5, R 1  and R 2  are each independently H or C 1 -C 4  alkyl, or R 1  and R 2  together with the carbon to which they are joined form a C 3 -C 8  cycloalkyl; with the proviso that where Z is \u2014NCS, M is C or CR; \n W is (CH 2 ) n , and n is 0, 1, 2, or 3; \n D is a cycloalkyl, aryl, heterocyclyl, heteroaryl, or D is an a C 1 -C 3  alkylenyl linking Y and M; \n Y is (CH 2 ) n , O(CH 2 ) n , NR 3 (CH 2 ) n , (CH 2 ) n O, (CH 2 ) n NR 3 , where n is 0, 1, or 2, and R 3  is H or C 1 -C 4  alkyl; \n X is CR 4 R 5  or (CH 2 ) n , where n is 0, 1, or 2, and R 4  and R 5  are each independently H, C 1 -C 4  alkyl, cycloalkyl, aryl, heterocyclyl, heteroaryl, or together with the C to which they are attached form a saturated or unsaturated ring; with the proviso that one of R 4  and R 5  is H or that R 4  and R 5  together with the C to which they are attached form a saturated or unsaturated ring; \n V is absent, O, NR 5 , SO 2 , SO, CO, CONR 6 , CR 7 R 8 , or (CH 2 ) n , wherein R 6  is H or C 1 -C 4  alkyl; and R 7  and R 8  are each independently H, C 1 -C 4  alkyl, cycloalkyl, aryl, heterocyclyl, heteroaryl, or together with the C to which they are attached form a saturated or unsaturated ring; \n B is (CH 2 ) n\u2032  where n is 2, 3, or 4, cycloalkyl, heterocyclyl, aryl, heteroaryl; and \n A is absent, cycloalkyl, aryl, heterocyclyl, heteroaryl.

Metadata:
- Claim Count in Document: 9.0
- Percentile: 90.0
- Lexical Diversity: 1.31034
- Patent Class: 540.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15311817', '15253773', '14770331', '15763724', '14169770']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.73560832422082
- 35 USC 102 Novelty (BERT): 0.6138527599112398
- Combined Prediction Score: 0.723432767789862
- Mean Citation Score: 384.380926
- Max Citation Score: 623.34186
- Similarity Product: 463.7517161339701

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test