PATENT CLAIM ANALYSIS

Application Number: 15767945
Application Type: Utility
Filing Date: 2018-04
Publication Date: 2018-10
Patent Classification: ["514", "064000"]

Abstract:
The present invention provides a urea peptidomimetic boronic compound and pharmaceutical compositions thereof, their preparative methods and uses. The compounds are represented by the following formula (1).

Claim (Index 1):
A compound of formula (1): or a pharmaceutically acceptable salt or solvate thereof, wherein:\n m and n represent the number of amino acid residues, m is 0, and n is 1 or 2; \n R 4  is a side chain of amino acids, and n of R 4  is of alkyl, cycloalkyl, alkenyl, acycloalkyl, alkynyl, aryl, andlkyl, heteroaryl, independently selected from hydrogen, aralkyl, heteroaralkyl, heterocycloalkyl, alkyl, heteroaralkyl, heterocyclyl, heterocycloalkyl, alkoxy, cycloalkoxy, aryloxy, alkylthio, cycloalkylthio, arylthio, alkoxycarbonyl, aryloxycarbonyl, acyl, thioacyl, acyloxy, amido, carbamido, sulfinyl, alkylsulfonyl, arylsulfonyl, haloalkyl, carbamoyl, halogen, cyano, isocyano, nitro, nitroso, thiocyano, isothiocyano, acylhydrazino, thioalkyl, sulpho and silyl; \n R 5  and R 6  are hydrogen at the same time, or together R 5  and R 6  form a diol ester group; \n R 1 , L and R 3  together with N atom to which L and R 3  are attached form a 5, 6 or 7 membered heterocyclic ring optionally having, in addition to the nitrogen atom, another ring heteroatom being N, and optionally having an oxo group; meanwhile, the 5, 6 or 7 membered heterocyclic ring above is fused to an aromatic ring or heteroaromatic ring each optionally substituted by one or more substituents independently selected from the group consisting of alkyl, cycloalkyl, alkenyl, cycloalkenyl, alkynyl, aryl, aralkyl, heteroaryl, heteroaralkyl, heterocyclyl, heterocycloalkyl, alkoxy, cycloalkoxy, aryloxy, alkylthio, cycloalkylthio, arylthio, alkoxycarbonyl, aryloxycarbonyl, acyl, thioacyl, acyloxy, amido, carbamido, sulfinyl, alkylsulfonyl, arylsulfonyl, haloalkyl, carbamoyl, halogen, cyano, isocyano, nitro, nitroso, thiocyano, isothiocyano, acylhydrazino, thioalkyl, sulpho and silyl.

Metadata:
- Claim Count in Document: 13.0
- Percentile: 91.0
- Lexical Diversity: 1.10345
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['13379142', '16300162', '14567480', '14734233', '13582678']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7640838928447566
- 35 USC 102 Novelty (BERT): 0.4966562038756405
- Combined Prediction Score: 0.737341123947845
- Mean Citation Score: 214.68997
- Max Citation Score: 237.31741
- Similarity Product: 186.15033033250927

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test