PATENT CLAIM ANALYSIS

Application Number: 16122975
Application Type: Utility
Filing Date: 2018-09
Publication Date: 2019-01
Patent Classification: ["514", "269000"]

Abstract:
The present invention provides compounds of Formula (I): wherein all variables are as defined in the specification, and compositions comprising any of such novel compounds. These compounds are APJ agonists which may be used as medicaments.

Claim (Index 10):
A compound according to  claim 5 , having Formula (V): or a stereoisomer, an enantiomer, a diastereoisomer, a tautomer, or a pharmaceutically acceptable salt thereof, wherein: ring B is independently selected from R 1 , at each occurrence, is independently selected from H, F, Cl, OH, CN, and OC 1-4  alkyl; R 2  is independently selected from \u2014CH 2 CH 2 CH 2 CH 3 , \u2014CH 2 CH 2 CH(CH 3 ) 2 , CH 2 CH 2 CH 2 CF 3 , \u2014CH 2 -cyclopropyl, \u2014CH 2 CH 2 -cyclopropyl, cyclobutyl, cyclopentyl, CH 2 O(CH 2 ) 1-3 CH 3 , and CH 2 OCH(CH 3 ) 2 , phenyl substituted with 0-2 R e , and 5- to 6-membered heteroaryl substituted with 0-2 R e ; R 5 , at each occurrence, is independently selected from R 8 , at each occurrence, is independently selected from F, Cl, Br, \u2014OCH 3 , \u2014OCF 3 , \u2550O, CN, CH 3 , CF 3 , \u2014C(\u2550O)NH 2 , \u2014(CH 2 ) n -aryl substituted with 0-3 R e , \u2014(CH 2 ) n \u2014C 3-6  cycloalkyl substituted with 0-3 R e , and \u2014(CH 2 ) n -heterocyclyl substituted with 0-3 R e ; R e , at each occurrence, is independently selected from F, Cl, Br, CN, NO 2 , \u2550O, CO 2 H, C 1-6  alkyl (optionally substituted with F and CO, OH, OCH 3 , OCF 3 , \u2014(CH 2 ) n \u2014C 3-6  cycloalkyl, \u2014(CH 2 ) n \u2014C 4-6  heterocyclyl, \u2014(CH 2 ) n -aryl, and \u2014(CH 2 ) n -heteroaryl; R e ' is independently selected from C 1-2  alkyl, \u2014CH 2 OC 1-2  alkyl, and cyclopropyl; and n is independently selected from zero, 1, 2, 3, and 4.

Metadata:
- Claim Count in Document: 27.0
- Percentile: 97.0
- Lexical Diversity: 1.16667
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15468230', '15767364', '16309161', '16061365', '15171276']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8143293695435995
- 35 USC 102 Novelty (BERT): 0.554194987935945
- Combined Prediction Score: 0.7883159313828341
- Mean Citation Score: 382.398828
- Max Citation Score: 411.5391
- Similarity Product: 400.9856631204128

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test