PATENT CLAIM ANALYSIS

Application Number: 16009030
Application Type: Utility
Filing Date: 2018-06
Publication Date: 2018-11
Patent Classification: ["544", "134000"]

Abstract:
This invention relates to inhibitors of mitotic kinesins, particularly KSP, and methods for producing these inhibitors.

Claim (Index 36):
The compound of  claim 1 , which is wherein:\n R x  and R y  are independently H, alkyl, saturated or partially unsaturated cycloalkyl or aryl, wherein said alkyl, cycloalkyl and aryl are optionally substituted with one or more groups independently selected from oxo (with the proviso that it is not substituted on said aryl), halogen, cyano, nitro, trifluoromethyl, difluoromethyl, fluoromethyl, fluoromethoxy, difluoromethoxy, trifluoromethoxy, azido, \u2014O(C\u2550O)OR d , \u2014NR b SO 2 R d , \u2014SO 2 NR a R b , \u2014C(\u2550O)R a , \u2014C(\u2550O)OR a , \u2014OC(\u2550O)R a , \u2014OCH 2 C(\u2550O)OR a , \u2014NR b C(\u2550O)OR d , \u2014NR b C(\u2550O)R a , \u2014C(\u2550O)NR a R b , \u2014NR a R b , \u2014NR c C(\u2550O)NR a R b , \u2014NR c C(NCN)NR a R b , \u2014OR a , alkyl, alkenyl, alkynyl, cycloalkyl, aryl, heteroaryl, arylalkyl, heteroarylalkyl, heterocyclyl and heterocyclylalkyl, \n or R x  and R y  together with the atom to which they are attached form a saturated or partially unsaturated carbocyclic ring or heterocyclic ring having one or more heteroatoms independently selected from N, O and S, wherein said carbocyclic and heterocyclic rings are optionally substituted with one or more groups independently selected from oxo, halogen, cyano, nitro, trifluoromethyl, difluoromethyl, fluoromethyl, fluoromethoxy, difluoromethoxy, trifluoromethoxy, azido, \u2014O(C\u2550O)OR d , \u2014NR b SO 2 R d , \u2014SO 2 NR a R b , \u2014C(\u2550O)R a , \u2014C(\u2550O)OR a , \u2014OC(\u2550O)R a , \u2014NR b C(\u2550O)OR d , \u2014NR b C(\u2550O)R a , \u2014C(\u2550O)NR a R b , \u2014NR a R b , \u2014NR c C(\u2550O)NR a R b , \u2014NR c C(NCN)NR a R b , \u2014OR a , alkyl, alkenyl, alkynyl, cycloalkyl, aryl, heteroaryl, arylalkyl, heteroarylalkyl, heterocycloalkyl and heterocyclylalkyl; or R a  and R x  together with the atoms to which they are attached form a saturated or partially unsaturated heterocyclic ring which may include 1 to 3 additional heteroatoms, in addition to the oxygen atom to which said R a  is attached, selected from N, O and S, wherein said heterocyclic ring is optionally substituted with one or more groups independently selected from oxo, halogen, cyano, nitro, trifluoromethyl, difluoromethyl, fluoromethyl, fluoromethoxy, difluoromethoxy, trifluoromethoxy, azido, \u2014O(C\u2550O)OR h , \u2014NR f SO 2 R h , \u2014SO 2 NR e R f , \u2014C(\u2550O)R e , \u2014C(\u2550O)OR e , \u2014OC(\u2550O)R e , \u2014NR f C(\u2550O)OR h , \u2014NR f C(\u2550O)R e , \u2014C(\u2550O)NR e R f , \u2014NR e R f , \u2014NR g C(\u2550O)NR e R f , \u2014NR c C(NCN)NR e R f , \u2014OR e , alkyl, alkenyl, alkynyl, cycloalkyl, aryl, heteroaryl, arylalkyl, heteroarylalkyl, heterocycloalkyl and heterocyclylalkyl.

Metadata:
- Claim Count in Document: 12.0
- Percentile: 94.0
- Lexical Diversity: 1.11765
- Patent Class: 544.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15357613', '14679866', '12043456', '13093729', '14099276']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8669358181620117
- 35 USC 102 Novelty (BERT): 0.6215353735308465
- Combined Prediction Score: 0.8423957736988952
- Mean Citation Score: 575.379454
- Max Citation Score: 581.6764
- Similarity Product: 547.0970378629684

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test