PATENT CLAIM ANALYSIS

Application Number: 15959419
Application Type: Utility
Filing Date: 2018-04
Publication Date: 2018-09
Patent Classification: ["514", "232800"]

Abstract:
Disclosed are a compound represented by Formula (1), or a pharmaceutically acceptable salt, hydrate, solvate, prodrug, tautomer, enantiomer, or pharmaceutically acceptable diastereomer thereof, a method of preparing the same, and a pharmaceutical composition, which have effects for treatment or prevention of metabolic syndromes, comprising the same: wherein R 1  to R 6 , X 1  to X 4 , and n are the same as defined in claim  1.

Claim (Index 10):
A method of preparing the compound of Formula (1) according to claim  1 , the method comprising:\n A) synthesizing a compound of Formula (7) below by reacting a compound of Formula (5) below and a compound of Formula (6) below under basic conditions; B) introducing \u2014NO 2  to a compound of Formula (7) below by reacting the compound generated in the synthesizing (A) and HNO 3  under acidic conditions; C) reducing \u2014NO 2  to \u2014NH 2  through reduction of the compound generated in the introducing (B); D) cyclizing the compound generated in the reducing (C) under acidic conditions; and E) generating a final product through selectively oxidation after selectively reacting the compound generated in the cyclizing (D) under basic conditions: wherein X 1 , X 2 , X 3 , X 4 , R 1 , R 2 , and R 4  are the same as defined in Formula (1); Z\u2032 is a halogen or R\u2032COO\u2014, where R\u2032 is substituted or unsubstituted C1-C9 alkyl, substituted or unsubstituted \u2014(CH 2 ) m \u2014C4-C10 aryl, substituted or unsubstituted \u2014(CH 2 ) m \u2014C4-C10 aryloxy, or substituted or unsubstituted C4-C10 aryl, wherein the substituted group is at least one selected from the group consisting of hydroxy, a halogen, C1-C10 alkyl, C2-C10 alkenyl, C2-C10 alkynyl, C1-C10 alkoxy, C1-C10 alkoxycarbonyl, C3-C8 cycloalkyl, C3-C8 heterocycloalkyl, C4-C10 aryl, and C5-C10 heteroaryl; and Y is \u2014NH 2 , \u2014NH 3 Z or \u2014NO 2 , where Z is a halogen.

Metadata:
- Claim Count in Document: 32.0
- Percentile: 91.0
- Lexical Diversity: 1.61538
- Patent Class: 514.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15102968', '11849230', '12946759', '13035640', '13138227']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7433933411025792
- 35 USC 102 Novelty (BERT): 0.5919972385188944
- Combined Prediction Score: 0.7282537308442106
- Mean Citation Score: 370.249616
- Max Citation Score: 649.2651
- Similarity Product: 383.6513306169033

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test