PATENT CLAIM ANALYSIS

Application Number: 15751778
Application Type: Utility
Filing Date: 2018-02
Publication Date: 2018-11
Patent Classification: ["424", "001890"]

Abstract:
The present application provides compounds useful in methods of treating neurological disorders such as Alzheimer's disease, and cancer such as prostate cancer. Also provided herein are radiolabeled compounds useful for imaging techniques, and techniques for diagnosis and monitoring of treatment of neurological disorders and cancer. An exemplary radiolabeled compound provided herein is useful as a radiotracer for positron emission tomography or single-photon emission computed tomography. Methods for preparing radiolabeled compounds and methods for preparing unlabeled compounds are also provided.

Claim (Index 198):
The compound of  claim 196 , wherein:\n Hal is selected from the group consisting of: Cl, F, and I; X is selected from the group consisting of O and NR N ; L 1  is \u2014C 1-6  alkylene-, wherein said alkylene group is optionally substituted with 1, 2, or 3 substituents independently selected from halo, CN, OH, C 1-3  alkoxy, and amino; L 2  is \u2014C 1-6  alkylene-, wherein said alkylene group is optionally substituted with 1, 2, or 3 substituents independently selected from halo, CN, OH, C 1-3  alkoxy, and amino; R N  is selected from the group consisting of H and C 1-6  alkyl; group A is 5 or 6 membered heteroaryl, which is optionally substituted by 1, 2, or 3 independently selected R A  groups; alternatively, group A is H; with the proviso that when X is NR N , L 1  is \u2014C 1-6  alkylene-, L 2  is \u2014C 1-6  alkylene-, and R N  is C 1-6  alkyl, group A is not H; and each R A  is independently selected from the group consisting of OH, NO 2 , CN, halo, C 1-6  alkyl, C 2-6  alkenyl, C 2-6  alkynyl, C 1-6  haloalkyl, C 1-6  alkoxy, C 1-6  haloalkoxy, cyano-C 1-3  alkyl, HO\u2014C 1-3  alkyl, amino, C 1-6  alkylamino, and di(C 1-6  alkyl)amino.

Metadata:
- Claim Count in Document: 27.0
- Percentile: 88.0
- Lexical Diversity: 1.7551
- Patent Class: 424.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['15543826', '15326890', '12956146', '15884833', '13515638']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.761174152053198
- 35 USC 102 Novelty (BERT): 0.5091294358031779
- Combined Prediction Score: 0.7359696804281961
- Mean Citation Score: 279.745556
- Max Citation Score: 289.80746
- Similarity Product: 212.04581443125247

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 0
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test