PATENT CLAIM ANALYSIS

Application Number: 16090072
Application Type: Utility
Filing Date: 2018-09
Publication Date: 2019-05
Patent Classification: ["544", "238000"]

Abstract:
The present invention relates to a novel pyrimidine-4-carboxylic acid derivative having an anticancer activity, and the compound of the present invention is useful as a drug for treating and preventing tumor diseases.

Claim (Index 8):
The pharmaceutical composition according to  claim 5 , wherein the pyrimidine-4-carboxylic acid compound represented by Formula 1 is selected from the group consisting of:\n 5-(([1,1\u2032-biphenyl]-4-ylmethyl)amino)pyrimidine-4-carboxylic acid; 5-((2,4-dimethoxybenzyl)amino)pyrimidine-4-carboxylic acid; 5-((3,4-dichlorobenzyl)amino)pyrimidine-4-carboxylic acid; 5-((furan-2-ylmethyl)amino)pyrimidine-4-carboxylic acid; 5-(((3-methylthiophen-2-yl)methyl)amino)pyrimidine-4-carboxylic acid; 5-((4-fluorobenzyl)amino)pyrimidine-4-carboxylic acid; 5-((3,5-bis(trifluoromethyl)benzyl)amino)pyrimidine-4-carboxylic acid; 5-((4-methoxybenzyl)amino)pyrimidine-4-carboxylic acid; 5-((4-methylbenzyl)amino)pyrimidine-4-carboxylic acid; 5-((3-fluorobenzyl)amino)pyrimidine-4-carboxylic acid; 5-((2-fluorobenzyl)amino)pyrimidine-4-carboxylic acid; 5-((1-propyl-1H-indazol-3-yl)amino)pyrimidine-4-carboxylic acid; 5-((1-(2-(dimethylamino)ethyl)-1H-indazol-3-yl)amino)pyrimidine-4-carboxylic acid; 5-((1-(3-benzamidopropyl)-1H-pyrazol-4-yl)amino)pyrimidine-4-carboxylic acid; 5-((1-methyl-1H-pyrazol-3-yl)amino)pyrimidine-4-carboxylic acid; 5-((1-methyl-1H-pyrazol-4-yl)amino)pyrimidine-4-carboxylic acid; 5-(pyridazin-3-ylamino)pyrimidine-4-carboxylic acid; 5-(naphthalen-1-ylamino)pyrimidine-4-carboxylic acid; 5-((1-(3-(dimethylamino)propyl)-1H-pyrazol-4-yl)amino)pyrimidine-4-carboxylic acid; and 5-((4-(4-ethylpiperazin-1-yl)phenyl)amino)pyrimidine-4-carboxylic acid.

Metadata:
- Claim Count in Document: 8.0
- Percentile: 97.0
- Lexical Diversity: 1.17241
- Patent Class: 544.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15689115', '14475762', '14923525', '14775405', '14994824']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7807564315755074
- 35 USC 102 Novelty (BERT): 0.4965529000926902
- Combined Prediction Score: 0.7523360784272257
- Mean Citation Score: 255.124242
- Max Citation Score: 261.55322
- Similarity Product: 215.697265302856

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test