PATENT CLAIM ANALYSIS

Application Number: 15947343
Application Type: Utility
Filing Date: 2018-04
Publication Date: 2019-01
Patent Classification: ["514", "221000"]

Abstract:
Provided herein are heteroaryl compounds, methods of their synthesis, pharmaceutical compositions comprising the compounds, and methods of their use. In one embodiment, the compounds provided herein are useful for the treatment, prevention, and/or management of various disorders, such as CNS disorders and neurological disorders, including, but not limited to, e.g., psychosis, schizophrenia, depression, movement disorders, and Parkinson's disease.

Claim (Index 1):
A compound of formula (I): or a pharmaceutically acceptable salt or stereoisomer thereof, wherein\n n is 2, 3, or 4; \n W is O, NR 5 , or CH 2 ; \n X is CH; \n Y is N or CH; \n each R 10  and each R 11  are independently H, F, OH, or (C 1 -C 4 )alkyl; \n (i) R 1  is amido, sulfonamido, optionally substituted imidazolyl, or optionally substituted pyrazolyl; and R 2  is H, halogen, CN, (C 1 -C 4 )alkyl, or (C 1 -C 3 )alkoxyl; or (ii) R 1  and R 2  together with the carbon atoms to which they are attached form a 5-, 6-, or 7-membered aryl, heteroaryl, cycloalkyl, or heterocyclyl ring, each of which is optionally substituted with one to three R 6 ; \n R 3  and R 4  together with the nitrogen atom to which they are attached form an optionally substituted heterocyclyl Q; \n Q is \n R 5  is H or (C 1 -C 3 )alkyl; each R 6  is independently OH, keto, halogen, CN, (C 1 -C 3 )alkyl, or (C 1 -C 3 )alkoxyl; R 7  is 5- to 10-membered aryl or heteroaryl, each optionally substituted with one to three substituents; and Ring Ar is a benzo, pyrazolo, pyrido, thieno, pyrimido, pyrazino, furano, pyridazino, thiazolo, or imidazolo ring, each optionally substituted with one to three substituents; provided that: (i) when Q is \u2003then \u2003is not \u2003and (ii) when Ar is an optionally substituted benzo ring, then \u2003is not

Metadata:
- Claim Count in Document: 100.0
- Percentile: 91.0
- Lexical Diversity: 1.65217
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['14399334', '14950834', '15298469', '14884397', '14377673']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8018544108118503
- 35 USC 102 Novelty (BERT): 0.6217163529917805
- Combined Prediction Score: 0.7838406050298433
- Mean Citation Score: 390.945736
- Max Citation Score: 549.93964
- Similarity Product: 545.3638942918826

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test