PATENT CLAIM ANALYSIS

Application Number: 16228835
Application Type: Utility
Filing Date: 2018-12
Publication Date: 2019-06
Patent Classification: ["514", "253120"]

Abstract:
Disclosed are compounds, compositions and methods for the prevention and/or treatment of diseases which are pathophysiologically mediated by the neurokinin (NK 1 ) receptor. The compounds have the general formula (I):

Claim (Index 10):
A compound selected from the group consisting of: GA2 1-(acetoxymethyl)-4-(5-(2-(3,5- bis(trifluoromethyl)phenyl)-N,2- dimethylpropanamido)-4-(o- tolyl)pyridin-2-yl)-1- methylpiperazin-1-ium,    GA3 4-(5-(2-(3,5- bis(trifluoromethyl)phenyl)-N,2- dimethylpropanamido)-4-(o- tolyl)pyridin-2-yl)-1- ((butyryloxy)methyl)-1- methylpiperazin-1-ium,   GA4 1-(5-(2-(3,5- bis(trifluoromethyl)phenyl)-N,2- dimethylpropanamido)-4-(o- tolyl)pyridin-2-yl)-4- methylpiperazine 1,4-dioxide,   GA5 1-(5-(2-(3,5- bis(trifluoromethyl)phenyl)-N,2- dimethylpropanamido)-1-oxido-4- (o-tolyl)pyridin-2-yl)-4- methylpiperazine 1-oxide,   GA6 4-(5-(2-(3,5- bis(trifluoromethyl)phenyl)-N,2- dimethylpropanamido)-1-oxido-4- (o-tolyl)pyridin-2-yl)-1- methylpiperazine 1-oxide,   GA7 5-(2-(3,5- bis(trifluoromethyl)phenyl)-N,2- dimethylpropanamido)-2-(4- methylpiperazin-1-yl)-4-(o- tolyl)pyridine 1-oxide, and   GA8 4-(5-(2-(3,5- bis(trifluoromethyl)phenyl)-N,2- dimethylpropanamido)-4-(o- tolyl)pyridin-2-yl)-1- methylpiperazine 1-oxide. or a pharmaceutically acceptable salt thereof.

Metadata:
- Claim Count in Document: 17.0
- Percentile: 98.0
- Lexical Diversity: 1.19355
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['15194984', '15874325', '14360991', '12637719', '11582293']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8275319678326823
- 35 USC 102 Novelty (BERT): 0.5386428247861524
- Combined Prediction Score: 0.7986430535280293
- Mean Citation Score: 329.305366
- Max Citation Score: 397.34216
- Similarity Product: 262.2948133711194

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test