PATENT CLAIM ANALYSIS

Application Number: 16088695
Application Type: Utility
Filing Date: 2018-09
Publication Date: 2019-04
Patent Classification: ["514", "063000"]

Abstract:
The present invention discloses a silicon incorporated quinoline of formula (I) wherein, X, Y, A, R 1  and R 2  are as described. The present invention further discloses a process for the preparation of silicon incorporated quinolines of formula I; a pharmaceutical composition comprising silicon incorporated quinolines of formula (I) or pharmaceutically acceptable salt thereof. The present invention also discloses a method for treating diseases caused by  Plasmodium falciparum  or other  coccidian  parasites using the silicon incorporated quinolines of formula I or pharmaceutically acceptable salt thereof.

Claim (Index 14):
A pharmaceutical composition comprising the silicon incorporated quinolines of formula I or pharmaceutically acceptable salt thereof and at least one pharmaceutically acceptable carrier wherein, X is selected from the group consisting of hydrogen, halogen, C 1 -C 5  alkyl, C 1 -C 5 haloalkyl, C 1 -C 5 hydroxyalkyl, C 1 -C 5 thioalkyl, and C 1 -C 5  alkoxy; Y is CH 2  or absent; A is selected from the group consisting of R 1  and R 2  are independently selected from the group consisting of hydrogen, C 1  to C 12  alkyl, C 1 -C 5  aryl, C 1 -C 5  heteroaryl, C 1 -C 5  aralkyl, C 1 -C 5  hydroxyalkyl, C 1 -C 5  alkoxyalkyl, and C 1 -C 5  aminoalkyl which is optionally substituted or forms a 5 or 6 membered ring which optionally contains an additional hetero atoms selected from the group consisting of O, S, N and Si; and R 1  or R 2  essentially comprises at least one silicon atom.

Metadata:
- Claim Count in Document: 35.0
- Percentile: 97.0
- Lexical Diversity: 1.84906
- Patent Class: 514.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['14350766', '15752896', '14895710', '11477745', '12142846']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7851271667635001
- 35 USC 102 Novelty (BERT): 0.5314417214096537
- Combined Prediction Score: 0.7597586222281155
- Mean Citation Score: 315.892494
- Max Citation Score: 361.45117
- Similarity Product: 293.8135543253481

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test