PATENT CLAIM ANALYSIS

Application Number: 15978041
Application Type: Utility
Filing Date: 2018-05
Publication Date: 2018-11
Patent Classification: ["514", "262100"]

Abstract:
The present disclosure provides compounds of Formula (IA) and/or pharmaceutically acceptable salts thereof that are tyrosine kinase inhibitors, in particular BTK, and are potentially useful for the treatment of diseases treatable by inhibition of tyrosine kinases such as cancer, inflammatory diseases such as arthritis, and the like. Also provided are pharmaceutical compositions containing such compounds and/or pharmaceutically acceptable salts thereof and processes for preparing such compounds and pharmaceutically acceptable salts thereof.

Claim (Index 56):
A method of treating a disease treatable by inhibition of a tyrosine kinase in a patient in recognized need thereof, wherein the disease is chosen from allergy, urticaria, antiphospholipid antibody syndrome, and vasculitis, and wherein the method comprises the step of administering to the patient a pharmaceutical composition comprising a pharmaceutically acceptable excipient and a therapeutically effective amount of a mixture of (E) and (Z) stereoisomers of (R)-2-(3-(4-amino-3-(2-fluoro-4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidine-1-carbonyl)-4-methyl-4-(4-(oxetan-3-yl)piperazin-1-yl)pent-2-enenitrile, and/or a pharmaceutically acceptable salt thereof.

Metadata:
- Claim Count in Document: 5.0
- Percentile: 93.0
- Lexical Diversity: 1.61224
- Patent Class: 514.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['14464602', '14997330', '14374788', '14418484', '13859569']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8403389497774194
- 35 USC 102 Novelty (BERT): 0.6460444906318845
- Combined Prediction Score: 0.8209095038628659
- Mean Citation Score: 647.798482
- Max Citation Score: 684.86005
- Similarity Product: 562.5501182966053

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test