PATENT CLAIM ANALYSIS

Application Number: 15753361
Application Type: Utility
Filing Date: 2018-02
Publication Date: 2018-08
Patent Classification: ["544", "115000"]

Abstract:
The invention relates to a compound of formula I: (I) or a pharmaceutically acceptable salt thereof, wherein each R 3  is independently selected from H, halo, fluorinated C 1 -C 10  alkyl, —I—C 1 -C 10  alkyl, —NH—C 1 -C 10  alkyl, —S—C 1 -C 10  alkyl, —O-fluorinated C 1 -C 10  alkyl, —NH-acyl, —NH—C(O)—NH-alkyl, —C—(O)—NH-alkyl, with the proviso that at least one of R 3  is not H.

Claim (Index 1):
A compound of formula I: or a pharmaceutically acceptable salt thereof, wherein: W is selected from the group consisting of O, N\u2014H, N\u2014(C 1 -C 10  alkyl) and S; each X is independently selected from CH or N; R 1  is a 5 to 7-membered saturated or unsaturated, optionally substituted heterocycle containing at least 1 heteroatom selected from N or O; R 2  is (LQ) v Y, with the proviso that R 2  is not H; each L is independently selected from the group consisting of a direct bond, C 1 -C 10  alkylene, C 2 -C 10  alkenylene, C 2 -C 10  alkynylene, arylene and C 3 -C 10  cycloalkylene; each Q is independently selected from the group consisting of a direct bond, heteroarylene, a heterocycle linker, \u2014O\u2014, \u2014NR 6 \u2014, \u2014C(O)\u2014, \u2014C(O)NR 6 \u2014, \u2014SO 2 \u2014, \u2014SO 2 \u2014NR 6 \u2014, \u2014NH\u2014C(O)\u2014NR 6 \u2014, \u2014NH\u2014SO 2 \u2014NR 6 , halogen, \u2014C(halogen) a (R 6 (2-a) \u2014, \u2014NR 4 R 5 \u2014, and \u2014C(O)NR 4 R 5 , where R 4  and R 5  together with the nitrogen to which they are attached form a 4 to 10-membered heterocycle linker; v is from 0 to 5; Y is selected from the group consisting of H, C 1 -C 10  alkyl, C 2 -C 10  alkenyl, C 2 -C 10  alkenyl, C 2 -C 10  alkynyl, aryl, C 3 -C 10  cycloalkyl, heterocycle, heteroaryl, \u2014OR 6 , \u2014N(R 6 ) 2 , \u2014C(O)R 6 , \u2014C(O)OR 6 , \u2014C(O)N(R 6 ) 2 , \u2014N(R 6 ) 2 , \u2014SO 2 \u2014R 6 , \u2014SO 2 \u2014N(R 6 ) 2 , \u2014NH\u2014C(O)\u2014N(R 6 ) 2 , \u2014NH\u2014SO 2 \u2014N(R 6 ) 2 , halogen, \u2014C(halogen) b R 6 (3-b) , \u2014CN, \u2014NR 4 R 5 -, and \u2014C(O)NR 4 R 5 , where R 4  and R 5  together with the nitrogen to which they are attached form a 4- to 10-membered heterocycle; b is from 1 to 3; a is 1 or 2; each R 6  is independently selected from the group consisting of H, C 1-10  alkyl, aryl and heteroaryl; and each R 3  is independently selected from the group consisting of H, halo, fluorinated C 1 -C 10  alkyl, \u2014O\u2014C 1 -C 10  alkyl, \u2014NH\u2014C 1 -C 10  alkyl, \u2014S\u2014C 1 -C 10  alkyl, \u2014O-fluorinated C 1 -C 10  alkyl, \u2014NH-acyl, \u2014NH\u2014C(O)\u2014NH-alkyl, and \u2014C\u2014(O)\u2014NH-alkyl, with the proviso that at least one of R 3  is not H.

Metadata:
- Claim Count in Document: 50.0
- Percentile: 88.0
- Lexical Diversity: 1.80392
- Patent Class: 544.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15117606', '15753358', '15753353', '14920410', '13388164']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8150130323654232
- 35 USC 102 Novelty (BERT): 0.5840614309796337
- Combined Prediction Score: 0.7919178722268443
- Mean Citation Score: 411.889446
- Max Citation Score: 488.13507
- Similarity Product: 440.3667643612182

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test