PATENT CLAIM ANALYSIS

Application Number: 16242902
Application Type: Utility
Filing Date: 2019-01
Publication Date: 2019-07
Patent Classification: ["514", "338000"]

Abstract:
The present invention is directed to indazole derivatives, pharmaceutical compositions containing them and their use in the treatment and/or prevention of disorders and conditions ameliorated by antagonizing one or more glucagon receptors, including for example metabolic diseases such as Type II diabetes mellitus and obesity.

Claim (Index 5):
A compound of  claim 4 , wherein\n R 1  is selected from the group consisting of 4-t-butyl-phenyl, 2,4-dimethyl-phenyl, 4-trifluoromethyl-phenyl, 2,4-dichloro-phenyl, 2-chloro-4-methyl-phenyl, 2-methyl-4-chloro-phenyl, 2-chloro-4-trifluoromethyl-phenyl, 2-methyl-4-trifluoromethyl-phenyl, 3-chloro-4-trifluoromethyl-phenyl, benzofuran-2-yl, benzothien-2-yl, 5-fluoro-benzothien-2-yl and 6-fluoro-benzothien-2-yl; a is an integer from 0 to 1; R 2  is selected from the group consisting of 4-chloro, 4-methyl, 4-methoxy, 4-ethoxy, 6-chloro and 6-methyl; R 4  is selected from the group consisting of n-propyl, isobutyl, n-pentyl, isopentyl, 2,2-dimethyl-n-propyl, n-hexyl, 3,3,3-trifluoro-n-propyl, 3,3,4,4,4-pentafluoro-n-butyl, 2-fluoro-2-methyl-propyl, cyclopropyl-methyl, cyclobutyl-methyl-, cyclobutyl-ethyl, cyclopentyl-methyl-, cyclopentyl-ethyl, cyclohexyl, cyclohexyl-methyl-, cyclohexyl-ethyl, phenylethyl- and 4-chloro-phenylethyl-; Z is selected from the group consisting of C and N; or a stereoisomer or pharmaceutically acceptable salt thereof.

Metadata:
- Claim Count in Document: 44.0
- Percentile: 99.0
- Lexical Diversity: 1.06667
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['15695118', '15695129', '15695107', '13478534', '13478568']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8262436474417808
- 35 USC 102 Novelty (BERT): 0.596790352036835
- Combined Prediction Score: 0.8032983179012861
- Mean Citation Score: 455.527282
- Max Citation Score: 492.78116
- Similarity Product: 485.2933149427533

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test