PATENT CLAIM ANALYSIS

Application Number: 15969670
Application Type: Utility
Filing Date: 2018-05
Publication Date: 2018-12
Patent Classification: ["514", "004900"]

Abstract:
The invention provides compounds having the general formula I: Y—X—Z   I and salts thereof, wherein the variables X, Y, and Z have the meaning as described herein, and compositions containing such compounds and methods for using such compounds and compositions.

Claim (Index 4):
The compound of  claim 1  which has the following formula II:\n CH 3 C(\u2550O)-A-X\u2014B\u2014NH 2  \u2003\u2003II \n or a salt thereof, wherein:\n A is -His-DPhe-Arg-Trp-(SEQ ID NO: 1), -His-DNal(2\u2032)-Arg-Trp-(SEQ ID NO: 2), -DTrp-DArg-Phe-DHis-, or \n -DTrp-DArg-Nal(2\u2032)-DHis-; \n B is -His-DPhe-Arg-Trp-(SEQ ID NO: 1), -His-DNal(2\u2032)-Arg-Trp-(SEQ ID NO: 2), -DTrp-DArg-Phe-DHis-, or \n -DTrp-DArg-Nal(2\u2032)-DHis-;\n X is a linking group; \n His is a residue of L-histidine; \n DHis is a residue of D-histidine; \n Phe is a residue of L-phenylalanine, wherein the phenyl ring is optionally substituted with one or more groups selected from halo, (C 1 -C 4 )alkyl, \u2014O(C 1 -C 4 )alkyl, (C 1 -C 4 )haloalkyl, or \u2014O(C 1 -C 4 )haloalkyl; \n DPhe is a residue of D-phenylalanine, wherein the phenyl ring is optionally substituted with one or more groups selected from halo, (C 1 -C 4 )alkyl, \u2014O(C 1 -C 4 )alkyl, (C 1 -C 4 )haloalkyl, or \u2014O(C 1 -C 4 )haloalkyl; \n Arg is a residue of L-arginine; \n DArg is a residue of D-arginine; \n Trp is a residue of L-tryptophan, wherein the indolyl ring is optionally substituted with one or more groups selected from halo, (C 1 -C 4 )alkyl, \u2014O(C 1 -C 4 )alkyl, (C 1 -C 4 )haloalkyl, or \u2014O(C 1 -C 4 )haloalkyl; \n DTrp is a residue of D-tryptophan, wherein the indolyl ring is optionally substituted with one or more groups selected from halo, (C 1 -C 4 )alkyl, \u2014O(C 1 -C 4 )alkyl, (C 1 -C 4 )haloalkyl, or \u2014O(C 1 -C 4 )haloalkyl; \n Nal(2\u2032) is a residue of L-2-naphthyl-alanine, wherein the phenyl ring is optionally substituted with one or more groups selected from halo, (C 1 -C 4 )alkyl, \u2014O(C 1 -C 4 )alkyl, (C 1 -C 4 )haloalkyl, or \u2014O(C 1 -C 4 )haloalkyl; and \n DNal(2\u2032) is a residue of D-2-naphthyl-alanine, wherein the phenyl ring is optionally substituted with one or more groups selected from halo, (C 1 -C 4 )alkyl, \u2014O(C 1 -C 4 )alkyl, (C 1 -C 4 )haloalkyl, or \u2014O(C 1 -C 4 )haloalkyl; \n provided if A is -His-DPhe-Arg-Trp-(SEQ ID NO: 1), B is not -His-DPhe-Arg-Trp-(SEQ ID NO: 1), wherein the phenyl ring and the indolyl ring are not substituted; \n and provided if A is -His-DNal(2\u2032)-Arg-Trp-(SEQ ID NO: 2), B is not -His-DNal(2\u2032)-Arg-Trp-(SEQ ID NO: 2), wherein the naphthyl ring and the indolyl ring are not substituted.

Metadata:
- Claim Count in Document: 29.0
- Percentile: 93.0
- Lexical Diversity: 1.4375
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['13320408', '12298826', '15050671', '13074565', '14117949']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8077760463958034
- 35 USC 102 Novelty (BERT): 0.5372979008621931
- Combined Prediction Score: 0.7807282318424424
- Mean Citation Score: 352.850674
- Max Citation Score: 377.4124
- Similarity Product: 263.7661644181967

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 0
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test