PATENT CLAIM ANALYSIS

Application Number: 15875187
Application Type: Utility
Filing Date: 2018-01
Publication Date: 2018-12
Patent Classification: ["514", "029000"]

Abstract:
Triazole-containing macrolide and ketolide antibiotics, therapeutic compositions containing them and methods of use for treating diseases caused by one or more resistant organisms are described.

Claim (Index 52):
A method for treating a disease in a host animal caused at least in part by  Legionella, Haemophilus, Mycobacterium leprae,  or a combination thereof; the method comprising administering to the host animal a therapeutically effective amount of a compound of the formula. or a pharmaceutically acceptable salt thereof, wherein:\n R 10  is hydrogen or acyl; \n X is H; and Y is OR 7 ; where R 7  is a monosaccharide; or X and Y are taken together with the attached carbon to form carbonyl; \n V is C(O), C(\u2550NR 11 ), CH(NR 12 , R 13 ), or N(R 14 )CH 2 , where N(R 14 ) is attached to the C-10 carbon; wherein R 11  is hydroxy or alkoxy, R 12  and R 13  are each independently selected from the group consisting of hydrogen, hydroxy, alkyl, aralkyl, alkylaryl, alkoxy, heteroalkyl, aryl, heteroaryl, dimethylaminoalkyl, acyl, sulfonyl, ureido, and carbamoyl; and R 14  is hydrogen, hydroxy, alkyl, aralkyl, alkylaryl, alkoxy, heteroalkyl, aryl, heteroaryl, dimethylaminoalkyl, acyl, sulfonyl, ureido, or carbamoyl; \n W is H, F, Cl, Br, I, or OH; \n A is CH 2 , C(O), C(O)O, C(O)NH, S(O) 2 , S(O) 2 NH, C(O)NHS(O) 2 ; \n B is (CH 2 )n where n is an integer ranging from 0-10, or B is an unsaturated carbon chain of 2-10 carbons; and \n C is alkyl, arylalkyl, heteroalkyl, aryl, heteroaryl, or heteroarylalkyl, each of which is optionally substituted.

Metadata:
- Claim Count in Document: 28.0
- Percentile: 86.0
- Lexical Diversity: 1.03846
- Patent Class: 514.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['13125555', '14309202', '14725247', '13125550', '14309178']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8188268071785668
- 35 USC 102 Novelty (BERT): 0.6110917830194933
- Combined Prediction Score: 0.7980533047626595
- Mean Citation Score: 492.58008000000007
- Max Citation Score: 565.2923599999998
- Similarity Product: 505.1060930777119

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 0
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test