PATENT CLAIM ANALYSIS

Application Number: 15752260
Application Type: Utility
Filing Date: 2018-02
Publication Date: 2018-08
Patent Classification: ["514", "616000"]

Abstract:
Disclosed are a series of malonamide derivatives having a chemical structure(I), their synthesis, and evaluation of their bioactivities against bacterial cell, bacterial-infected  C.elegans  and mice.

Claim (Index 12):
A method of synthesizing the substituted malonamide of  claim 1 , comprising:\n (a) reacting a compound having chemical structure (II) with a first substituted amine R 1 \u2014NH 2  to obtain a compound having chemical structure (III), (b) the compound having chemical structure (III) further reacts with a second substituted amine R 2 \u2014NH 2  to obtain the substituted malonamide of  claim 1 , wherein R 1  is C 2-6  alkyl, C 2-6  alkenyl, or C 3-7  cycloalkyl;\n R 2  is \n C 2-6  alkyl, C 2-6  alkenyl, or C 3-7  cycloalkyl;\n R 3  is selected from C 3  cycloalkyl, C 2-6  alkenyl, or C 2-5  halogenoalkyl; \n R 4 , R 5 , R 6 , R 7 , R 8 , R 9 , R 10 , R 11 , R 12 , and R 13  are independently selected from hydrogen, C 1-5  alkyl, C 2-6  alkenyl, ethynyl, halogen, trihalogenomethyl, nitro, hydroxyl, trihalogenomethoxy, or pentafluorosulfanyl.

Metadata:
- Claim Count in Document: 9.0
- Percentile: 88.0
- Lexical Diversity: 1.23077
- Patent Class: 514.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['14234255', '13120568', '13821195', '13130440', '15302539']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7379344557636944
- 35 USC 102 Novelty (BERT): 0.5206842048802136
- Combined Prediction Score: 0.7162094306753464
- Mean Citation Score: 283.87426399999987
- Max Citation Score: 295.3933
- Similarity Product: 206.66165450255872

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test