PATENT CLAIM ANALYSIS

Application Number: 16068627
Application Type: Utility
Filing Date: 2018-07
Publication Date: 2019-01
Patent Classification: ["544", "360000"]

Abstract:
The present invention discloses an N-sulfonyl benzamide derivative with a heterocyclic substituent, and a preparation method therefor and a pharmaceutical application thereof. More specifically, the invention discloses a compound represented by formula (II) or a pharmaceutically acceptable salt, stereoisomer, solvent compound, or prodrug thereof, and a preparation method therefor and an application thereof. Refer to the specification for definitions of each group in the

Claim (Index 8):
The compound of  claim 7 , or a pharmaceutically acceptable salt, solvate, stereoisomer or prodrug thereof, wherein the phenyl is wherein R 1 \u2032, R 2 \u2032, R 3 \u2032, R 4 \u2032, R 5 \u2032 are each independently a hydrogen, halogen, nitro, hydroxyl, cyano, C 6-20  aryl, C 1-20  alkyl, halogenated C 1-20  alkyl, halogenated C 1-20  alkoxy, C 1-20  alkoxy, C 3-20  cycloalkyl, halogenated C 3-20  cycloalkyl, C 3-20  cycloalkoxy, halogenated C 3-20  cycloalkoxy, C 2-20  alkenyl, halogenated C 2-20  alkenyl, C 2-20  alkynyl, halogenated C 2-20  alkynyl, \u2014NR a R b , \u2014C(O)NR a R b , \u2014N(R a )C(O)\u2014(C 1-20  alkyl), \u2014N(R a )SO 2 \u2014(C 1-20  alkyl), \u2014SO 2 N(R a R b ), \u2014C(O)O\u2014(C 1-20  alkyl), \u2014CHO, \u2014OC(O)\u2014(C 1-20  alkyl), \u2014SO 2 \u2014(C 1-20  alkyl), \u2014SO 2 \u2014(C 6-20  aryl), \u2014CO\u2014(C 1-20  alkyl), \u2014CO\u2014(C 6-20  aryl); and/or the pyridyl is wherein R 21 , R 31 , R 41 , R 51 , R 12 , R 32 , R 42 , R 52 , R 13 , R 23 , R 43 , R 53  are each independently a hydrogen, halogen, nitro, hydroxyl, cyano, C 6-20  aryl, C 1-20  alkyl, halogenated C 1-20  alkyl, halogenated C 1-20  alkoxy, C 1-20  alkoxy, C 3-20  cycloalkyl, halogenated C 3-20  cycloalkyl, C 3-20  cycloalkoxy, halogenated C 3-20  cycloalkoxy, C 2-20  alkenyl, halogenated C 2-20  alkenyl, C 2-20  alkynyl, halogenated C 2-20  alkynyl, \u2014NR a R b , \u2014C(O)NR a R b , \u2014N(R a )C(O)\u2014(C 1-20  alkyl), \u2014N(R a )SO 2 \u2014(C 1-20  alkyl), \u2014SO 2 N(R a R b ), \u2014C(O)O\u2014(C 1-20  alkyl), \u2014CHO, \u2014OC(O)\u2014(C 1-20  alkyl), \u2014SO 2 \u2014(C 1-20  alkyl), \u2014SO 2 \u2014(C 6-20  aryl), \u2014CO\u2014(C 1-20  alkyl), \u2014CO\u2014(C 6-20  aryl); and R a , R b  are defined as above.

Metadata:
- Claim Count in Document: 2.0
- Percentile: 95.0
- Lexical Diversity: 1.57447
- Patent Class: 544.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['16308790', '15537002', '15799771', '15296601', '12588882']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7691091365728138
- 35 USC 102 Novelty (BERT): 0.5337306948609642
- Combined Prediction Score: 0.7455712924016289
- Mean Citation Score: 330.6311199999999
- Max Citation Score: 357.7838
- Similarity Product: 294.4191364493728

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test