PATENT CLAIM ANALYSIS

Application Number: 15778168
Application Type: Utility
Filing Date: 2018-05
Publication Date: 2018-10
Patent Classification: ["514", "259310"]

Abstract:
The present invention relates to a novel azole derivative as an apelin receptor agonist and a method for treating cardiovascular disease, diabetic disease, renal disease, hypertension, and arteriosclerosis, etc., using the same. The present invention provides a compound represented by formula (I) or a pharmacologically acceptable salt thereof wherein X 1  represents —NH═ or —CH═, X 2  represents —CH═ or —N═, R 1  and R 2  each represent a C 1  to C 6  alkoxy group or the like, R 3  represents a heteroaryl group (the heteroaryl group is optionally substituted by a methyl group or the like) or the like, and R 4  represents a C 1  to C 6  alkylthio group or a C 2  to C 6  alkenyl group (the C 1  to C 6  alkylthio group and the C 2  to C 6  alkenyl group are each optionally substituted by one carboxy group or the like) or the like.

Claim (Index 34):
The method according to  claim 33 , wherein the disease is cardiovascular disease, coronary heart disease, stroke, heart failure, systolic heart failure, diastolic heart failure, diabetic heart failure, heart failure with preserved ejection fraction, cardiomyopathy, myocardial infarction, left ventricular dysfunction, left ventricular dysfunction after myocardial infarction, cardiac hypertrophy, myocardial remodeling, myocardial remodeling after infarction, myocardial remodeling after cardiac surgery, or valvular heart disease.

Metadata:
- Claim Count in Document: 43.0
- Percentile: 93.0
- Lexical Diversity: 2.40845
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['10718337', '13995300', '10344157', '14322505', '12397132']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8211976597503055
- 35 USC 102 Novelty (BERT): 0.5354766327992563
- Combined Prediction Score: 0.7926255570552005
- Mean Citation Score: 366.950764
- Max Citation Score: 379.27014
- Similarity Product: 173.37035054821553

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test