PATENT CLAIM ANALYSIS

Application Number: 15910307
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2018-07
Patent Classification: ["514", "259300"]

Abstract:
The invention provides novel compounds having the general formula (I) wherein R A , R B , R C , R C1  and W are as defined herein, compositions including the compounds and methods of using the compounds.

Claim (Index 38):
A compound according to any one of  claims 1  to  37 , selected from\n 3-[(2-tert-butyl-4-chloro-5-methylphenoxy)methyl ]-4-methyl-1H-1,2,4-triazol -5-one; \n 3-[(2-tert-butyl-4-chloro-5-fluorophenoxy)methyl ]-4-methyl-1H-1,2,4-triazol -5-one; \n 3-tert-butyl-4-[(4-methyl-5-oxo-1H-1,2,4-triazol -3-yl)methoxy]benzonitrile; \n 5-tert-butyl-2-methyl-4-[(4-methyl-5-oxo-1H-1,2,4-triazol -3-yl)methoxy]benzonitrile; \n 4-tert-butyl-2-methyl-5-[(4-methyl-5-oxo-1H-1,2,4-triazol -3-yl)methoxy]benzonitrile; \n 3-[(4-chloro-2-cyclohexyl-5-methylphenoxy)methyl]-4-methyl-1H-1,2,4-triazol-5-one; \n 5-tert-butyl-2-methyl-4-[(5-oxo-4-propan-2-yl-1H-1,2,4-triazol-3-yl)methoxy]benzonitrile; \n 3-[(4-chloro-5-methyl-2-propan-2-ylphenoxy)methyl]-4-methyl-1H-1,2,4-triazol-5-one; \n 3-[(4-chloro-2-cyclobutyl-5-methylphenoxy)methyl]-4-methyl-1H-1,2,4-triazol-5-one; \n 3-[[4-chloro-5-methyl-2-[3-(morpholine-4-carbonyl)phenyl ]phenoxy]methyl]-4-methyl-1H-1,2,4-triazol-5-one; \n 3-[[4-chloro-5-methyl-2-(1,2-oxazol-5-yl)phenoxy]methyl]-4-methyl-1H-1,2,4-triazol-5-one; \n 2-chloro-4-[(4-methyl-5-oxo-1H-1,2,4-triazol-3-yl)methoxy]-5-phenylbenzonitrile; \n 2-chloro-4-[(4-methyl-5-oxo-1H-1,2,4-triazol-3-yl)methoxy]-5-[3-(1H-pyrazol-3-yl)phenyl]b enzonitrile; \n 2-chloro-5-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-4-[(4-methyl-5-oxo-1H-1,2,4-triazol-3-yl)methoxy]benzonitrile; \n 3-[5-chloro-4-methyl-2-[(4-methyl-5-oxo-1H-1,2,4-triazol-3-yl)methoxy]phenyl]-4-fluoro-N,N-dimethylbenzamide; \n 3-[[4-chloro-2-(2-methoxypyridin-3-yl)-5-methylphenoxy]methyl]-4-methyl-1H-1,2,4-triazol-5-one; \n 3-[[4-chloro-2-(2-fluoro-5-propan-2-yloxyphenyl)-5-methylphenoxy]methyl]-4-methyl-1H-1,2,4-triazol-5-one; \n 3-[[4-chloro-2-[2-fluoro-5-(pyrrolidine-1-carbonyl)phenyl]-5-methylphenoxy]methyl]-4-methyl-1H-1,2,4-triazol-5-one; \n 4-[3-[5-chloro-4-methyl-2-[(4-methyl-5-oxo-1H-1,2,4-triazol-3-yl)methoxy]phenyl]-4-fluorobenzoyl]-1-methylpiperazin-2-one; \n 3-[5-chloro-4-methyl-2-[(4-methyl-5-oxo-1H-1,2,4-triazol-3-yl)methoxy]phenyl]-4-fluoro-N-(2-methoxyethyl)-N-methylbenzamide; \n 3-[[4-chloro-2-[2-fluoro-5-(oxolan-2-ylmethoxy)phenyl]-5-methylphenoxy]methyl]-4-methyl-1H-1,2,4-triazol -5-one; \n 2-[3-[5-chloro-4-methyl-2-[(4-methyl-5-oxo-1H-1,2,4-triazol-3-yl)methoxy]phenyl]-4-fluorophenoxy]-N,N-dimethylacetamide; \n N-[[3-[5-chloro-4-methyl-2-[(4-methyl-5-oxo-1H-1,2,4-triazol -3-yl)methoxy]phenyl]-4-fluorophenyl]methyl]-2-methoxy-N-methyl acetamide; \n 2-chloro-5-(2-fluorophenyl)-4-[(4-methyl-5-oxo-1H-1,2,4-triazol-3-yl)methoxy]benzonitrile; \n 2-chloro-5-(2-fluoro-3-methoxyphenyl)-4-[(4-methyl-5-oxo-1H-1,2,4-triazol-3-yl)methoxy]benzonitrile; \n 2-chloro-5-(2-fluoro-5-propan-2-yloxyphenyl)-4-[(4-methyl-5-oxazol-3-yl)methoxy]benzonitrile; \n 3-[[4-chloro-2-(5-cyclopropyloxy-2-fluorophenyl)-5-methylphenoxy]methyl]-4-methyl-1H-1,2,4-triazol-5-one; \n 2-chloro-5-(5-cyclopropyloxy-2-fluorophenyl)-4-[(4-methyl-5-oxo-1H-1,2,4-triazol -3-yl)methoxy]benzonitrile; \n -tert-butyl-2-methyl-4-(1H-pyrazolo[3,4-b]pyridin-3-yl methoxy)benzonitrile; \n 2-[[3-[(2-tert-butyl-4-chloro-5-methyl phenoxy)methyl]-1H-pyrazolo[3,4-d]pyrimidin-6-yl]-methylamino]ethanol; \n 2-[[3-[(2-tert-butyl-4-chloro-5-methyl phenoxy)methyl]-1H-pyrazolo[3,4-d]pyrimidin-6-yl]oxy]ethanol; \n 2-chloro-5-[2-fluoro-5-(pyrrolidine-1-carbonyl)phenyl]-4-(1H-pyrazolo[3,4-b]pyridin-3-ylmethoxy)benzonitrile; \n 3-[5-chloro-4-methyl-2-(1H-pyrazolo[3,4-c]pyridin-3-yl methoxy)phenyl]-4-fluoro-N-(2-methoxyethyl)-N-methylbenzamide; \n and pharmaceutically acceptable salts thereof.

Metadata:
- Claim Count in Document: 1.0
- Percentile: 90.0
- Lexical Diversity: 1.35484
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['12462417', '14844991', '15332398', '12466785', '14376307']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7852599768228714
- 35 USC 102 Novelty (BERT): 0.5412363437357082
- Combined Prediction Score: 0.7608576135141552
- Mean Citation Score: 361.796304
- Max Citation Score: 369.039
- Similarity Product: 308.1865787631869

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test