PATENT CLAIM ANALYSIS

Application Number: 15981598
Application Type: Utility
Filing Date: 2018-05
Publication Date: 2018-09
Patent Classification: ["435", "060000"]

Abstract:
The present application relates to novel substituted 5-fluoro-1H-pyrazolopyridines, to processes for their preparation, to their use alone or in combinations for the treatment and/or prophylaxis of diseases, and to their use for producing medicaments for the treatment and/or prophylaxis of diseases, in particular for the treatment and/or prophylaxis of cardiovascular disorders.

Claim (Index 13):
A process for preparing the compound of  claim 12 , wherein a compound of the formula (II) [A] is reacted in an inert solvent in the presence of hexabutyltin and a suitable palladium catalyst with intermediate formation of a tin species with the compound of the formula (III) to give the compound of the formula (IV) this is then reduced in an inert solvent with a suitable reducing agent to give the compound of the formula (V) and this is then reacted in the presence of a suitable base in the presence or absence of a solvent with methyl chloroformate to give the compound of the formula (I-A) or [B] the compound of the formula (II) is reacted in an inert solvent with copper cyanide to give the compound of the formula (VI) this is then, under acidic conditions, converted into the compound of the formula (VII) this is subsequently reacted in an inert solvent in the presence of a suitable base with the compound of the formula (VIII) to give the compound of the formula (IX) and this is then reduced in an inert solvent in the presence of a suitable reducing agent to give the compound (V), and this is subsequently reacted further according to process [A] to give the compound of the formula (I-A).

Metadata:
- Claim Count in Document: 20.0
- Percentile: 93.0
- Lexical Diversity: 1.80645
- Patent Class: 435.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15348545', '13111856', '14552122', '14194224', '13882118']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.6369807207002859
- 35 USC 102 Novelty (BERT): 0.5609217780741291
- Combined Prediction Score: 0.6293748264376703
- Mean Citation Score: 380.31979400000006
- Max Citation Score: 433.06305
- Similarity Product: 357.81135708374967

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 0

Dataset: test