PATENT CLAIM ANALYSIS

Application Number: 15773975
Application Type: Utility
Filing Date: 2018-05
Publication Date: 2018-11
Patent Classification: ["514", "269000"]

Abstract:
The present teachings relate to hydroxypyridinone and hydroxypyrimidinone derivatives, pharmaceutical compositions thereof, and methods of using such compounds to treat bacterial infections.

Claim (Index 12):
The compound of either of  claim 10  or  11 , wherein\n L 2  \u2014(C(R 4 )(R 5 )) n (C 0-3  alkylene)-, \u2014(C(R 4 )(R 5 )) n \u2014(C 0-3  alkylene)-N(R 5 )\u2014, \u2014(C(R 4 )(R 5 )) n \u2014(C 0-3  alkylene)-S(\u2550O) 2 \u2014; \n wherein each R 4  is H or optionally substituted C 1-6  alkyl; and \n each R 5  is independently H, an optionally substituted C 1-6  alkyl, an optionally substituted C 1-6  heteroalkyl, an optionally substituted C 1-6  alkenyl, an optionally substituted C 1-6  alkynyl, an optionally substituted C 6-14  aryl, an optionally substituted 5- to 14-membered heteroaryl, an optionally substituted C 3 -C 8  cycloalkyl, on optionally substituted \u2014(C 0-4  alkylene)-OR f , \u2014(C 0-4  alkylene)-(C 1-4  alkene), \u2014(C 0-4  alkylene)-(C 1-4  alkyne), C 2 -C 7  heterocycle, \u2014(C 0-4  alkylene)-C(\u2550O)\u2014(C 1 -C 6  alkyl), \u2014(C 0-4  alkylene)-C(\u2550O)H, \u2014(C 0-4  alkylene)-C(\u2550O)OR f , alkylene)-CN, \u2014(C 0-4  alkylene)-halo, alkylene)-NO 2 , \u2014(C 0-4  alkylene)-NR f ) 2 , \u2014(C 0-4  alkylene)-S(\u2550O) 2 -(R f ), \u2014(C 0-4  alkylene)-(C 6-14  aryl), \u2014(C 1-4  alkylene)-(5- to 14-membered heteroaryl), \u2014(C 0-4  alkylene)- C(\u2550O)NR b R f  or \u2014(C 0-4  alkylene)-NR b C(\u2550O)R f ; \n wherein each R f  is independently H, an optionally substituted alkyl, an optionally substituted cycloalkyl, an optionally substituted heterocyclyl, or an optionally substituted alkoxy; \n L 3  is \u2014(C 2-6  alkynylene)-; \n L 4  is \u2014C(\u2550O)\u2014, \u2014(C(\u2550O)O)\u2014, \u2014(C(\u2550O)NR e )\u2014, or \u2014(C 1-4  alkylene)-; \n G 1  and G 2  are each independently, at each occurrence, \u2014(C 6-14  arylene)-; \n G 3  is H, C 3-7  cycloalkyl, C 3-10  heterocycloalkyl, C 6-14  aryl, 5- to 14-membered heteroarylene, (C 1-4  alkylene)-(C 1-4  heteroalkyl), (C 1-4  alkylene)-(C 1-4  heterocycloalkyl), (C 3-10  heterocycloalkylene)-(C 1-4  alkyl), (C 3-10  heterocycloalkylene)-(C 1-4  heteroalkyl), (C 3-10  heterocycloalkylene)-(C 3-10  heterocycloalkyl), C 1-6  alkyl, or (C 3-10  heterocycloalkylene)-hydroxy; and \n R a , R b , R c , R d , and R e  are each independently, at each occurrence, H or C 1-6  alkyl; and \n n is 1 or 2.

Metadata:
- Claim Count in Document: 1.0
- Percentile: 93.0
- Lexical Diversity: 1.13636
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15773976', '15123232', '13460524', '14222500', '13121157']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7876976316578548
- 35 USC 102 Novelty (BERT): 0.5782416218170121
- Combined Prediction Score: 0.7667520306737705
- Mean Citation Score: 375.364822
- Max Citation Score: 519.7719999999998
- Similarity Product: 378.1395008358954

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test