PATENT CLAIM ANALYSIS

Application Number: 16323863
Application Type: Utility
Filing Date: 2019-02
Publication Date: 2019-06
Patent Classification: ["544", "242000"]

Abstract:
Provided is a heterocyclic compound that may have a GCN2 inhibitory action, and is expected to be useful for the prophylaxis or treatment of GCN2 associated diseases including cancer and the like. A compound represented by the formula (I): wherein each symbol is as described in the DESCRIPTION, or a salt thereof.

Claim (Index 4):
The compound according to  claim 1 , wherein ring A is the formula wherein the combination of X 1 , X 2  and X 3  (X 1 , X 2 , X 3 ) is (carbon atom, carbon atom, carbon atom) or (carbon atom, carbon atom, nitrogen atom);\n R 1  is (1) a chlorine atom, a bromine atom, (2) methyl, trifluoromethyl, or (3) a hydroxy group substituted by methyl or trifluoromethyl; \n R 2  is (1) a halogen atom, (2) a C 1-6  alkyl group optionally substituted by 1 to 3 substituents selected from a halogen atom and a hydroxy group or (3) a C 1-6  alkoxy group optionally substituted by 1 to 3 halogen atoms; \n ring B is optionally further substituted by 1 to 3 substituents selected from (1) a halogen atom and (2) a C 1-6  alkyl group optionally substituted by 1 to 3 hydroxy groups; \n X 6  is a hydrogen atom, a fluorine atom or a chlorine atom; \n X 7  is a fluorine atom or a chlorine atom; \n the combination of X 8  and X 9  (X 8 , X 9 ) is (carbon atom, nitrogen atom); \n ring E is optionally further substituted by 1 to 3 C 1-6  alkyl groups; and \n X 10  is an amino group optionally substituted by 1-2 substituents selected from (1) a C 1-6  alkyl group optionally substituted by 1 to 3 hydroxy groups, (2) a C 3-10  cycloalkyl group optionally substituted by 1 to 3 hydroxy groups and (3) a 3- to 14-membered non-aromatic heterocyclic group, or a salt thereof.

Metadata:
- Claim Count in Document: 5.0
- Percentile: 99.0
- Lexical Diversity: 1.28261
- Patent Class: 544.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['14404126', '14902388', '15467548', '15563161', '13566091']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8064005938973378
- 35 USC 102 Novelty (BERT): 0.5126250662445133
- Combined Prediction Score: 0.7770230411320553
- Mean Citation Score: 316.363878
- Max Citation Score: 319.5668
- Similarity Product: 263.8294447422981

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 0
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 0

Dataset: test