PATENT CLAIM ANALYSIS

Application Number: 16046696
Application Type: Utility
Filing Date: 2018-07
Publication Date: 2019-01
Patent Classification: ["514", "241000"]

Abstract:
Disclosed herein are compounds of formula I: or a salt thereof and compositions comprising a compound of formula I or a pharmaceutically acceptable salt thereof. Also disclosed herein are methods for treating or preventing a bacterial infection in an animal comprising administering to the animal a compound of formula I or a pharmaceutically acceptable salt thereof, alone or in combination with a bacterial efflux pump inhibitor.

Claim (Index 33):
A compound of formula Ia or Ib: or a salt thereof, wherein: R 1  is hydrogen, (C 1 -C 4 )alkyl, or (C 1 -C 4 )haloalkyl; R 2  is hydrogen, (C 1 -C 4 )alkyl, or (C 1 -C 4 )haloalkyl; R 3  is hydrogen, (C 1 -C 4 )alkyl, or (C 1 -C 4 )haloalkyl; R 4  is hydrogen, (C 1 -C 6 )alkyl, aryl or heteroaryl, wherein the (C 1 -C 6 )alkyl is optionally substituted with one or more groups selected from halo, hydroxy, nitro, cyano, (C 1 -C 4 )alkoxy, \u2014NR X R Y , aryl, heteroaryl, aryloxy, or heteroaryloxy, wherein any ary, heteroaryl, aryloxy and heteroaryloxy is optionally substituted with one or more groups selected from halo, hydroxy, (C 1 -C 4 )alkyl, (C 1 -C 4 )haloalkyl, (C 1 -C 4 )alkoxy, nitro, cyano, or \u2014NR X R Y ; L is (C 1 -C 5 )alkylene that is optionally substituted with one or more R L  groups; each R L  is independently selected from hydrogen, halo, hydroxy, nitro, cyano, or (C 1 -C 4 )alkoxy; or any two R L  groups that are attached to the same carbon taken together form a (C 3 -C 6 )carbocycle; A is aryl or heteroaryl; each R A  is independently selected from the group consisting of halo, cyano, nitro, (C 1 -C 6 )alkyl, (C 1 -C 6 )alkoxy, \u2014NR X R Y , aryl or heteroaryl; wherein the (C 1 -C 6 )alkyl and (C 1 -C 6 )alkoxy is optionally substituted with one or more groups selected from oxo, halo, hydroxy, (C 1 -C 4 )alkoxy, nitro, cyano, or \u2014NR X R Y ; wherein the aryl and heteroaryl is optionally substituted with one or more groups selected from halo, hydroxy, (C 1 -C 4 )alkyl, (C 1 -C 4 )haloalkyl, (C 1 -C 4 )alkoxy, nitro, cyano, or \u2014NR X R Y ; each R X  and R Y  are independently hydrogen or (C 1 -C 4 )alkyl; or R X  and R Y  taken together with the nitrogen to which they are attached form pyrrolidinyl, piperidinyl, piperazinyl, or morpholinyl; and n is 0, 1, 2, 3, or 4; provided that when the compound is a compound of formula Ia and A is phenyl, then the A is substituted with at least one phenyl group; and provided that the compound of formula Ib is not or a salt thereof.

Metadata:
- Claim Count in Document: 25.0
- Percentile: 95.0
- Lexical Diversity: 1.75
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['15066911', '15323081', '15296601', '11791928', '13066616']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8302053252062873
- 35 USC 102 Novelty (BERT): 0.5510853030349799
- Combined Prediction Score: 0.8022933229891567
- Mean Citation Score: 388.26477400000016
- Max Citation Score: 418.62888
- Similarity Product: 346.9696560006093

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test