PATENT CLAIM ANALYSIS

Application Number: 15744510
Application Type: Utility
Filing Date: 2018-01
Publication Date: 2018-07
Patent Classification: ["514", "222800"]

Abstract:
The invention provides a compound which is a diazine of formula (I) or a tautomer thereof, or a pharmaceutically acceptable salt thereof, for use as an antifungal agent: (I) wherein X, N′, C′, A and E are as defined herein. The invention also provides a compound of Formula (I) as defined herein.

Claim (Index 9):
A compound for use according to any one of the preceding claims wherein:\n the compound is of Formula (Ia): wherein\n X represents S; \n R 1  represents H or methyl \n E represents either:\n (i) H or C 4 -C 6  alkyl which is unsubstituted and which is uninterrupted or is interrupted by \u2014O\u2014; or \n (ii) E is a C 1 -C 4  alkylene group which is bonded to an atom of group A to form a C 6  carbocyclylene group which is unsubstituted or is substituted by 1 substitutent selected from C 1 -C 4  alkoxy \n \n A represents the group -L-T or -T; \n L is selected from C 1 -C 10  alkylene and C 2 -C 10  alkenylene, wherein the alkylene or alkenylene group is unsubstituted or is substituted by 1 group selected from halogen and C 1 -C 4  alkoxy, and wherein the alkylene or alkenylene group is uninterrupted or is interrupted by a heteromoiety selected from \u2014O\u2014, \u2014S\u2014, and \u2014C(O)O\u2014, and wherein the alkylene or alkenylene group optionally terminates in a heteromoiety selected from \u2014O\u2014, and \u2014C(O)O\u2014 \n When A is L-T, then T is H or represents phenyl, napthyl, benzofuranyl, pyridyl, isoindoline-1,3-dione, benzothiazole, tetrahydrofuran, thienyl or cyclohexyl, and when A is T, then T represents phenyl, napthyl, benzofuranyl, pyridyl, isoindoline-1,3-dione, benzothiazole, tetrahydrofuran, thienyl or cyclohexyl; \n wherein T is unsubstituted or is substituted by 1 V group; \n Each V group is independently selected from C 1 -C 4  alkoxy, unsubstituted C 1 -C 4  alkyl, C 1 -C 4  alkyl which is substituted with 1, 2 or 3 halogen atoms, C 2 -C 4  alkenyl, C 2 -C 4  alkynyl, C 3 -C 6  cycloalkyl, halogen, aryl, (C 1 -C 4  alkyl)-aryl, aryloxy, aryloxy-(C 1 -C 4  alkyl), \u2014CN, NO 2 , \u2014(C 1 -C 4  alkyl)-C(O)O(C 1 -C 4  alkyl), and \u2014C(O)O(C 1 -C 4  alkyl).

Metadata:
- Claim Count in Document: 5.0
- Percentile: 86.0
- Lexical Diversity: 1.65
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['12989410', '14625532', '12601284', '11914516', '12515354']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7416854612582441
- 35 USC 102 Novelty (BERT): 0.5167091981851053
- Combined Prediction Score: 0.7191878349509303
- Mean Citation Score: 288.72395399999994
- Max Citation Score: 300.37643
- Similarity Product: 229.6178961680252

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test