PATENT CLAIM ANALYSIS

Application Number: 15772521
Application Type: Utility
Filing Date: 2018-04
Publication Date: 2018-11
Patent Classification: ["546", "022000"]

Abstract:
The present invention relates to a preparation method for a tedizolid compound in Formula I. In Formula I, R is selected from hydrogen, formula A, formula B, benzyl or benzyl substituted by a substituent, the substituent is selected from a group consisting of halogen, nitryl, C 1 -C 6  alkyl, and C 1 -C 6  alkoxy, and R 1  is C 1 -C 6  alkyl or C 1 -C 6  alkyl substituted by halogen. The method comprises: generating a compound having a structure as shown in Formula C and a compound having a structure as shown in Formula D by a coupled reaction under the catalysis of a metal catalyst, a substituent of R being defined as above, where X is a leaving group, the leaving group comprising chlorine, bromine, iodine, and sulfonyl oxy such as trifluoromethane sulfonic oxy, methylsulfonyl oxy and benzenesulfonyl oxy, or benzenesulfonyl oxy substituted by one or more substituents, the substituent being selected from a group consisting of halogen, C 1 -C 6  alkyl, and C 1 -C 6  alkoxy.

Claim (Index 9):
The preparation method according to  claim 7 , wherein the reaction solvent for the coupled reaction is any one of water, toluene, tetrahydrofuran, N,N-dimethylformamide, dimethyl sulfoxide, dioxane, isopropanol, ethanol, or acetonitrile or any combination thereof; and the reaction temperature is 50-120\u00b0 C.

Metadata:
- Claim Count in Document: 24.0
- Percentile: 91.0
- Lexical Diversity: 2.57143
- Patent Class: 546.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['14236801', '14925544', '12809011', '10561051', '10546373']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7660410986415337
- 35 USC 102 Novelty (BERT): 0.5122981726725715
- Combined Prediction Score: 0.7406668060446375
- Mean Citation Score: 264.664574
- Max Citation Score: 272.6859
- Similarity Product: 194.28411380503167

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test