PATENT CLAIM ANALYSIS

Application Number: 16054538
Application Type: Utility
Filing Date: 2018-08
Publication Date: 2018-12
Patent Classification: ["514", "340000"]

Abstract:
The present invention relates to novel derivatives of oxazolidinone, a method thereof and pharmaceutical compositions comprising the derivatives for use in an antibiotic. The oxazolidinone derivatives of the present invention show inhibitory activity against a broad spectrum of bacteria and lower toxicity. The prodrugs, prepared by reacting the compound having hydroxyl group with amino acid or phosphate, have an excellent efficiency on solubility thereof against water. Further, the derivatives of the present invention may exert potent antibacterial activity versus various human and animal pathogens, including Gram-positive bacteria such as Staphylococi, Enterococci and Streptococi, anaerobic microorganisms such as  Bacteroides  and Clostridia, and acid-resistant microorganisms such as  Mycobacterium tuberculosis  and  Mycobacterium avium . Accordingly, the compositions comprising the oxazolidinone are used in an antibiotic.

Claim (Index 5):
The method of  claim 4  wherein the bacterium is selected from the group consisting of  Staphylococcus, Enterococcus , and  Streptococcus.

Metadata:
- Claim Count in Document: 9.0
- Percentile: 96.0
- Lexical Diversity: 1.6875
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['10596412', '12211655', '13863216', '11792922', '12169164']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8416452976888784
- 35 USC 102 Novelty (BERT): 0.5586617556702201
- Combined Prediction Score: 0.8133469434870126
- Mean Citation Score: 362.199442
- Max Citation Score: 462.49002
- Similarity Product: 369.04287751477005

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test