PATENT CLAIM ANALYSIS

Application Number: 16060641
Application Type: Utility
Filing Date: 2018-06
Publication Date: 2018-12
Patent Classification: ["514", "210210"]

Abstract:
The present invention relates to LpxC antibacterial compounds of Formula (IA): corresponding pharmaceutically acceptable salts thereof, corresponding pharmaceutical compositions, compound preparation, treatment methods and uses for bacterial infections, especially those caused by gram-negative bacteria.

Claim (Index 5):
The compound of Formula (II) according to  claim 4  which is: EX. Chemical Name Chemical Structures 1 (2R)-N-hydroxy-2- methanesulfonyl-2-methyl-4-(4- oxo-7-phenyl-3,4- dihydroquinazolin-3-yl)butanamide GSK3207527   2 (2R)-N-hydroxy-2- methanesulfonyl-2-methyl-4-[7-(4- methylphenyl)-4-oxo-3,4- dihydroquinazolin-3-yl]butanamide GSK3208383A   3 (2R)-N-hydroxy-2- methanesulfonyl-4-[7-(4- methoxyphenyl)-4-oxo-3,4- dihydroquinazolin-3-yl]-2- methylbutanamide GSK3208384A   4 (2R)-4-{7-[4- (dimethylamino)phenyl]-4-oxo-3,4- dihydroquinazolin-3-yl}-N-hydroxy- 2-methanesulfonyl-2- methylbutanamide GSK3212100A   5 (2R)-4-{7-[4- (difluoromethoxy)phenyl]-4-oxo- 3,4-dihydroquinazolin-3-yl}-N- hydroxy-2-methanesulfonyl-2- methylbutanamide GSK3228259A   6 (2R)-4-[7-(2,3-difluorophenyl)-4- oxo-3,4-dihydroquinazolin-3-yl]-N- hydroxy-2-methanesulfonyl-2- methylbutanamide GSK3235107A   7 (2R)-4-[7-(2,5-difluorophenyl)-4- oxo-3,4-dihydroquinazolin-3-yl]-N- hydroxy-2-methanesulfonyl-2- methylbutanamide GSK3235108A   8 (2R)-4-[7-(2-fluorophenyl)-4-oxo- 3,4-dihydroquinazolin-3-yl]-N- hydroxy-2-methanesulfonyl-2- methylbutanamide GSK3212098A   9 (2R)-4-[7-(3-fluoro-4- methylphenyl)-4-oxo-3,4- dihydroquinazolin-3-yl]-N-hydroxy- 2-methanesulfonyl-2- methylbutanamide GSK3230791A   10 (2R)-4-{7-[4- (difluoromethyl)phenyl]-4-oxo-3,4- dihydroquinazolin-3-yl}-N-hydroxy- 2-methanesulfonyl-2- methylbutanamide GSK3236458A  or a pharmaceutically acceptable salt thereof.

Metadata:
- Claim Count in Document: 56.0
- Percentile: 94.0
- Lexical Diversity: 1.10526
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['14004105', '14068956', '14154239', '13515607', '14110165']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7814575774283833
- 35 USC 102 Novelty (BERT): 0.5514300112328446
- Combined Prediction Score: 0.7584548208088295
- Mean Citation Score: 356.35282599999994
- Max Citation Score: 394.587
- Similarity Product: 337.21111515212056

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test