PATENT CLAIM ANALYSIS

Application Number: 15772587
Application Type: Utility
Filing Date: 2018-05
Publication Date: 2019-03
Patent Classification: ["544", "262000"]

Abstract:
Compounds of the formula I in which Z, W, Q, R and Y have the meanings indicated in claim  1 , are inhibitors of Tankyrase, and can be employed, inter alia, for the treatment of diseases such as cancer, cardiovascular diseases, central nervous system injury and different forms of inflammation.

Claim (Index 1):
Compounds of the formula I in which Z denotes W denotes CH 2  or C(CH 3 ) 2 , Q denotes C(CH 3 ) 2 , CH(CH 3 ), CH(CH 2 CH 3 ), CH[CH(CH 3 ) 2 ], CH[CH 2 CH(CH 3 ) 2 ], or \u2014O\u2014,\n R denotes CH 2 , C(CH 3 ) 2 , NH or N(CH 3 ), \n Y denotes Ar or Het, \n R 1  denotes H, F or CH 3 , \n R 2  denotes H or CH 3 , \n Ar denotes phenyl, which is unsubstituted, or mono-, di- or trisubstituted by Hal, CN, A, OR 3 , (CH 2 ) m N(R 3 ) 2 , COOR 3  and/or CON(R 3 ) 2 , \n Het denotes pyrazolyl, pyridyl, pyrimidyl or pyridazinyl, each of which is unsubstituted or mono- or disubstituted by Hal, CN, A, OR 3 , N(R 3 ) 2  and/or (CH 2 ) m CON(R 3 ) 2  \n A denotes unbranched or branched alkyl with 1-8 C-Atoms, wherein one or two non-adjacent CH- and/or CH 2 -groups may be replaced by N- or O-atoms and wherein 1-7 H-atoms may be replaced by F, Cl and/or OH, \n R 3  denotes H or unbranched or branched alkyl with 1, 2, 3 or 4 C-Atoms, \n Hal denotes F, Cl, Br or I, \n m denotes 0, 1 or 2, \n n denotes 0, 1 or 2,\n and pharmaceutically acceptable salts, tautomers and stereoisomers thereof, including mixtures thereof in all ratios.

Metadata:
- Claim Count in Document: 15.0
- Percentile: 93.0
- Lexical Diversity: 1.40476
- Patent Class: 544.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['14909365', '15308974', '13383605', '16069326', '14378009']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7927667965793757
- 35 USC 102 Novelty (BERT): 0.5536758597306763
- Combined Prediction Score: 0.7688577028945058
- Mean Citation Score: 375.466308
- Max Citation Score: 428.29956
- Similarity Product: 301.94385593140123

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test