PATENT CLAIM ANALYSIS

Application Number: 16155846
Application Type: Utility
Filing Date: 2018-10
Publication Date: 2019-02
Patent Classification: ["544", "281000"]

Abstract:
The present teachings provide a compound represented by structural formula (I-0), or a pharmaceutically acceptable salt thereof. Also described are pharmaceutical compositions and methods of use thereof.

Claim (Index 30):
The compound of  claim 29 , wherein R 2  is\n azetidinyl optionally substituted with hydroxyl, hydroxymethyl, (C 3 -C 6 )cycloalkyl, or \u2014C(\u2550O)(C 1 -C 3 )alkyl; pyrrolidinyl optionally substituted with hydroxyl, hydroxymethyl, (C 3 -C 6 )cycloalkyl, or \u2014C(\u2550O)(C 1 -C 3 )alkyl; piperidinyl optionally substituted with hydroxyl, hydroxymethyl, (C 3 -C 6 )cycloalkyl, or \u2014C(\u2550O)(C 1 -C 3 )alkyl; piperazinyl optionally substituted with hydroxyl, hydroxymethyl, (C 3 -C 6 )cycloalkyl, or \u2014C(\u2550O)(C 1 -C 3 )alkyl; morpholinyl optionally substituted with hydroxyl, hydroxymethyl, (C 3 -C 6 )cycloalkyl, or \u2014C(\u2550O)(C 1 -C 3 )alkyl; pyridinyl, quinolinyl, OR c2 , wherein R c2  is phenyl optionally substituted with \u2014N(R a1 ) 2  or with 4-6 membered heterocycloalkyl with one ring heteroatom which is nitrogen; pyridinyl optionally substituted with halogen; piperidinyl optionally substituted with oxetanyl; or pyrrolidinyl optionally substituted with oxetanyl; wherein R a1  is H or (C 1 -C 3 )alkyl; \u2014NH-cyclopentyl, \u2014N\u2014((C 1 -C 3 )alkyl)-cyclopentyl or NHR b2 , wherein R b2  is phenyl or pyridinyl, each of which is optionally substituted with halo or (C 1 -C 3 )alkyl; cyclopropyl optionally substituted with hydroxyl, hydroxymethyl, or oxetanyl; cyclobutyl optionally substituted with hydroxyl, hydroxymethyl, or oxetanyl; cyclopentyl optionally substituted with hydroxyl, hydroxymethyl, or oxetanyl; cyclohexanyl optionally substituted with hydroxyl, hydroxymethyl, or oxetanyl; tetrahydropyranyl optionally substituted with hydroxyl or hydroxymethyl, tetrahydrofuranyl optionally substituted with hydroxyl or (C 1 -C 3 )alkoxy; oxetanyl; or (C 1 -C 4 )alkyl, wherein the (C 1 -C 4 )alkyl is optionally substituted with one or more groups selected from hydroxy, \u2014C(\u2550O)NH 2 , (C 1 -C 4 )alkoxy, hydroxy(C 1 -C 3 )alkyl, (C 3 -C 6 )cycloalkyl, 3-6 membered heterocycloalkyl containing one ring heteroatom which is oxygen.

Metadata:
- Claim Count in Document: 113.0
- Percentile: 97.0
- Lexical Diversity: 1.10345
- Patent Class: 544.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['14443072', '15434275', '14351381', '15543826', '14382123']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7944744632202814
- 35 USC 102 Novelty (BERT): 0.5925038414607147
- Combined Prediction Score: 0.7742774010443246
- Mean Citation Score: 421.832804
- Max Citation Score: 504.46133
- Similarity Product: 449.7227635348761

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test