PATENT CLAIM ANALYSIS

Application Number: 16135512
Application Type: Utility
Filing Date: 2018-09
Publication Date: 2019-01
Patent Classification: ["514", "219000"]

Abstract:
Provided are certain fused term or penta-cyclic compounds and salts thereof, compositions thereof, and methods of use thereof.

Claim (Index 3):
The at least one compound according to  claim 1 , which is selected from the compounds of Formula (III): stereoisomers thereof, and pharmaceutically acceptable salts thereof, wherein:\n R N  is selected from hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, heterocyclyl, aryl, and heteroaryl, wherein each of the alkyl, alkenyl, alkynyl, cycloalkyl, heterocyclyl, aryl or heteroaryl is independently optionally substituted with at least one substituent R 12 ; \n m and n, which may be the same or different are each an integer of (0, 1, 2, or 3; \n t is an integer of 0, 1, 2, or 3; \n R 1  at each occurrence, is independently selected from halogen, CN, NO 2 , OR 9 , NR 9 R 10 , NR 9 COR 10 , NR 9 SO 2 R 10 , CONR 9 R 10 , COOR 9 , SO 2 R 9 , alkyl, alkenyl, alkynyl, cycloalkyl, heterocyclyl, aryl, and heteroaryl wherein each of the alkyl, alkenyl, alkynyl, cycloalkyl, heterocyclyl, aryl, and heteroaryl is independently optionally substituted with at least one substituent R 12 . R 2  is selected from hydrogen COR 9 , CONR 9 R 10 , CO 2 R 9 , SO 2 R 9 , alkyl, alkenyl, alkynyl, cycloalkyl, heterocyclyl, aryl, and heteroaryl, wherein each of the alkyl, alkenyl, alkynyl, cycloalkyl, heterocyclyl, aryl, and heteroaryl is independently optionally substituted with at least one substituent R 12 , R 3 , R 4 , R 5 , R 6 , R 7  and R 8 , which may be the same or different, are each independently selected from hydrogen, halogen, \u2014NR 9 R 10 , \u2014OR 9 , oxo, \u2014COR 9 , \u2014CO 1 R 9 , \u2014CONR 9 R 10 , \u2014NR 9 CONR 10 R 11 , \u2014NR 9 CO 2 R 10 , \u2014NR 9 SO 2 R 10 , \u2014SO 2 R 9 , alkyl, alkenyl, cycloalkyl, aryl, heterocyclyl, alkynyl, and heteroaryl, wherein each of the alkyl, alkenyl, alkynyl, cycloalkyl, aryl, heterocyclyl, and heteroaryl is independently optionally substituted with at least one substituent R 12 , or (R 3  and R 4 ), and/or (R 4  and R 5 ), and/or (R 5  and R 7 ), and/or (R 7  and R 8 ), together with the atom(s) they are attached, form a 3- to 8-membered saturated, partially or fully unsaturated ring having 0, 1 or 2 heteroatoms independently selected from \u2014NR 13 \u2014, \u2014O\u2014, \u2014S\u2014, \u2014SO\u2014 or \u2014SO 2 \u2014, and said ring is optionally substituted with at least one substituent R 12 ,\n provided that\n when one of R 3  and R 4  is oxo, the other is absent; and \n \n when one of R 7  and R 8  is oxo, the other is absent;\n R 9 , R 10 , and R 11 , which may be the same or different, are each selected from hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, heterocyclyl, aryl, and heteroaryl, wherein each of the alkyl, alkenyl, alkynyl, cycloalkyl, heterocyclyl, aryl, and heteroaryl is independently optionally substituted with at least one substituent R 12 , \n R 12  is selected from CN, halogen, haloalkyl, NO 2 , \u2014NR\u2032R\u2033, \u2014OR\u2032, oxo, \u2014COR\u2032, \u2014CO 2 R\u2032, \u2014CONR\u2032R\u2033, \u2014NR\u2032CONR\u2033R\u2032\u2033, \u2014NR\u2032CO 2 R\u2033, NR\u2032SO 2 R\u2033, \u2014SO\u2014R\u2032, alkyl, alkenyl, alkynyl, cycloalkyl, heterocyclyl, aryl, and heteroaryl, wherein R\u2032R\u2033, and R\u2032\u2033 are independently selected from hydrogen, haloalkyl, alkyl, arylalkyl, alkenyl, alkynyl, cycloalkyl, heterocyclyl, aryl, and heteroaryl, or (R\u2032 and R\u2033), and/or (R\u2033 and R\u2032\u2033)together with the atoms to which they are attached form a 3- to 8-membered saturated, partially or fully unsaturated ring having 0, 1 or 2 additional heteroatoms independently selected from \u2014NR 11 \u2014, \u2014O\u2014, \u2014S\u2014, \u2014SO\u2014 or \u2014SO 2 \u2014, and \n R 11  is selected from hydrogen, alkyl, cycloalkyl, aryl, heteroaryl, and heterocyclyl.

Metadata:
- Claim Count in Document: 50.0
- Percentile: 97.0
- Lexical Diversity: 1.23529
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15479958', '14369374', '14988484', '14369388', '14723417']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8154923764992288
- 35 USC 102 Novelty (BERT): 0.6418937844891834
- Combined Prediction Score: 0.7981325172982243
- Mean Citation Score: 501.35223800000006
- Max Citation Score: 585.71405
- Similarity Product: 576.9504464676112

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test