PATENT CLAIM ANALYSIS

Application Number: 15890470
Application Type: Utility
Filing Date: 2018-02
Publication Date: 2018-06
Patent Classification: ["544", "280000"]

Abstract:
A pyrrolopyrimidine compound or a salt thereof and compositions, NAE inhibitors and anti-tumor agents containing the pyrrolopyrimidine compound or a salt thereof. The pyrrolopyrimidine compound or a salt thereof has an NAE inhibitory action and a cell growth inhibitory effect and is represented by Formula (A):

Claim (Index 1):
A compound or a salt thereof, represented by Formula (A) below: wherein: is a single bond or a double bond;\n X is \u2014O\u2014, \u2014CH 2 \u2014, or \u2014CH\u2550; \n Y is \u2014NH\u2014 or \u2014O\u2014; \n R 1  is hydrogen, fluorine, a hydroxy group, a cyano group, or an amino group; \n R 2  is hydrogen, fluorine, a hydroxy group, a cyano group, or an amino group; \n R 3  is a vinylene group, an ethynylene group, a C6-C14 arylene group, or a monocyclic or bicyclic heteroarylene group having at least one heteroatom selected from the group consisting of N, S, and O; \n R 4  is a bond, a methylene group, or a C3-C7 cycloalkylidene group; \n R 5  is a C3-C7 saturated cycloalkyl group that may have one or more R 6 , a C6-C10 unsaturated cycloalkyl group that may have one or more R 6 , or a monocyclic or bicyclic unsaturated heterocycloalkyl group that has at least one heteroatom selected from the group consisting of N, S, and O, and that may have one or more R 6 ; \n R 6  is selected from the group consisting of halogen, \n a hydroxy group, a cyano group, a C1-C6 alkyl group that may have one or more phenoxy group as a substituent, a carbamoyl group, a C1-C6 alkoxycarbonyl group, a monocyclic or bicyclic unsaturated heterocycloalkyl group having at least one heteroatom selected from the group consisting of N, S, and O, a monocyclic or bicyclic saturated heterocycloalkyl group that has at least one heteroatom selected from the group consisting of N, S, and O, and that may have one or more of either halogen, hydroxy group, carboxyl group, or C1-C6 alkyl group as a substituent, an amino group, a mono- or di-(C1-C4 alkyl) amino group that may have one or more hydroxy group or phenyl group as a substituent, a C1-C6 alkoxy group that may have one or more of either halogen, C3-C7 saturated cycloalkyl group, or monocyclic or bicyclic unsaturated heterocycloalkyl group having at least one heteroatom selected from the group consisting of N, S, and O as a substituent, a benzyloxy group that may have one or more carbamoyl group as a substituent, a C1-C6 alkylthio group, a C1-C6 alkylsulfonyl group, and an aminosulfonyl group,\n wherein when two or more R 6  are present, the plurality of R 6  may be the same or different.

Metadata:
- Claim Count in Document: 15.0
- Percentile: 88.0
- Lexical Diversity: 1.59375
- Patent Class: 544.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15122863', '15708917', '15700800', '11377363', '15545149']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8221911173281538
- 35 USC 102 Novelty (BERT): 0.5741292660641882
- Combined Prediction Score: 0.7973849322017572
- Mean Citation Score: 339.3252080000001
- Max Citation Score: 493.12094
- Similarity Product: 403.1294522899544

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test