PATENT CLAIM ANALYSIS

Application Number: 15995586
Application Type: Utility
Filing Date: 2018-06
Publication Date: 2018-10
Patent Classification: ["424", "722000"]

Abstract:
The present invention provides compounds of formula (I) and pharmaceutically acceptable salts thereof, wherein L, X, R a , R b , R 1 , R 2  and R 3  are as defined in the specification, processes for their preparation, pharmaceutical compositions containing them and their use in therapy.

Claim (Index 10):
The method according to  claim 1 , wherein R 3  represents a group selected from:\n (i) 2-fluorophenyl, (ii) 2-chlorophenyl, (iii) 2-methylphenyl, (iv) 2-cyclopropylphenyl, (v) 2-methoxyphenyl, (vi) 2-ethoxyphenyl, (vii) 2-(difluoromethoxy)phenyl, (viii) 3-methylphenyl, (ix) 3-methoxyphenyl, (x) 2,6-difluorophenyl, (xi) 2,6-dichlorophenyl, (xii) 2,6-dimethoxyphenyl, (xiii) 2,6-diethoxyphenyl, (xiv) 2-ethoxy-5-methylphenyl, (xv) 2,5-dimethoxyphenyl, (xvi) 2-fluoro-6-methoxyphenyl, (xvii) 5-fluoro-2-methoxyphenyl, (xviii) 3-fluoro-2-methoxyphenyl, (xix) 2-(1H-1,2,4-triazol-1-yl)phenyl, (xx) 2-(2H-1,2,3-triazol-2-yl)phenyl, (xxi) 5-methyl-2-(1H-1,2,3-triazol-1-yl)phenyl, (xxii) 5-methyl-2-(2H-1,2,3-triazol-2-yl)phenyl, (xxiii) 5-fluoro-2-(1H-1,2,3-triazol-1-yl)phenyl, (xxiv) 5-fluoro-2-(2H-1,2,3-triazol-2-yl)phenyl, (xxv) 2-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl, (xxvi) 2-(pyrimidin-2-yl)phenyl, (xxvii) 5-fluoro-2-(pyrimidin-2-yl)phenyl, (xxviii) 2-(1H-pyrazol-1-yl)phenyl, (xxix) 2-(1H-imidazol-1-yl)phenyl, (xxx) 2-(1H-1,2,3-triazol-1-yl)phenyl, (xxxi) 2-(pyrimidin-2-yl)-5-fluorophenyl, (xxxii) 2-fluoro-6-(2H-1,2,3-triazol-2-yl)phenyl, (xxxiii) 2-methoxy-5-methylphenyl, (xxxiv) 2-chloro-6-(2H-1,2,3-triazol-2-yl)phenyl, (xxxv) 2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl, (xxxvi) 5-trifluoromethyl-2-(2H-1,2,3-triazol-2-yl)phenyl, (xxxvii) 2-fluoro-6-(pyrazol-1-yl)phenyl, (xxxviii) 5-fluoro-2-(pyrazol-1-yl)phenyl, (xxxix) 5-methyl-2-(pyrazol-1-yl)phenyl, (xl) 2-bromo-6-methoxyphenyl, (xli) 2-methoxy-6-(pyrazol-1-yl)phenyl, (xlii) 5-chloro-2-(2H-1,2,3-triazol-2-yl)phenyl, (xliii) 3-fluoro-2-(2H-1,2,3-triazol-2-yl)phenyl, (xliv) 5-trifluoromethyl-2-(1H-1,2,3-triazol-1-yl)phenyl, (xlv) 5-chloro-2-(1H-1,2,3-triazol-1-yl)phenyl, (xlvi) 2,3-difluoro-6-(2H-1,2,3-triazol-2-yl)phenyl, (xlvii) 5-cyclopropyl-2-(2H-1,2,3-triazol-2-yl)phenyl, (xlviii) 5-chloro-2-(pyrazol-1-yl)phenyl, (xlix) 3,5-difluoro-2-(2H-1,2,3-triazol-2-yl)phenyl, (l) 2-(difluoromethyl)phenyl, (li) 2-(trifluoromethyl)phenyl, (lii) 3,6-difluoro-2-(2H-1,2,3-triazol-2-yl)phenyl, (liii) 2-cyclopropyl-6-fluorophenyl, (liv) 2-(5-ethoxypyrimidin-2-yl)phenyl, (lv) 3-(pyrimidin-2-yl)pyridin-2-yl, (lvi) 3-ethoxy-6-methylpyridin-2-yl, (lvii) 3-(pyrazol-1-yl)pyridin-2-yl, (lviii) 3-(piperidin-1-yl)pyridin-2-yl, (lix) 3-(trifluoromethoxy)pyridin-2-yl, (lx) 3-(ethoxy)pyridin-2-yl, (lxi) 3-(cyclopropyl)pyridin-2-yl, (lxii) 3-chloropyridin-2-yl, (lxiii) 3-bromopyridin-2-yl, (lxiv) 3-methoxypyridin-2-yl, (lxv) 3-(propan-2-yloxy)pyridin-2-yl, (lxvi) 6-bromo-3-methoxypyridin-2-yl, (lxvii) 3-methoxy-6-methylpyridin-2-yl, and (lxviii) 3-(2H-1,2,3-triazol-2-yl)pyridin-2-yl.

Metadata:
- Claim Count in Document: 50.0
- Percentile: 94.0
- Lexical Diversity: 1.35714
- Patent Class: 424.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['14625812', '15120048', '15029356', '15320887', '15120002']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8572461540612194
- 35 USC 102 Novelty (BERT): 0.7213193602391377
- Combined Prediction Score: 0.8436534746790112
- Mean Citation Score: 675.908338
- Max Citation Score: 867.8966
- Similarity Product: 771.6574850073337

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test