PATENT CLAIM ANALYSIS

Application Number: 15906934
Application Type: Utility
Filing Date: 2018-02
Publication Date: 2018-09
Patent Classification: ["514", "210180"]

Abstract:
The present disclosure provides a compound of formula (I) and the use thereof for the therapeutic treatment of human cancers including B-cell lymphoma and autoimmune diseases such as rheumatoid arthritis, systemic lupus erythematosus, and multiple sclerosis.

Claim (Index 40):
A compound of formula (I), including tautomers, rotamers, geometric isomers, diastereomers, racemates, and enantiomers, a pharmaceutically acceptable salt, a solvate, or a hydrate thereof, wherein A is selected from the group consisting of CR 0  and N; and wherein R 0  is selected from the group consisting of hydrogen, halogen, and alkyl; R a , R b , R c  and R d  are independently selected from the group consisting of hydrogen, halogen, and alkoxyl; B is selected from the group consisting of hydrogen, alkyl, cycloalkyl, heterocycloalkyl, aryl, heteroaryl, and B is either unsubstituted or substituted with at least one member selected from the group consisting of halogen, cyano, nitro, hydroxyl, alkyl, and alkoxyl; L is alkylene, or absent; and Y is selected from the group consisting of cycloalkyl, heterocycloalkyl, aryl, and heteroaryl, wherein Y is either unsubstituted or substituted with at least one member selected from the group consisting of halogen, \u2014CN, \u2014C(O)R 11 , and \u2014NHC(O)R 12  and wherein R 11 , and R 12  are independently selected from the group consisting of alkyl, cycloalkyl, alkenyl, cycloalkenyl, and alkynyl, or wherein Y is substituted with at least one member selected from the group consisting of F, \u2014C(O)CH\u2550CH 2 , \u2014C(O)CH\u2550CHCH 2 N(CH 3 ) 2 , \u2014NHC(O)CH\u2550CH 2 , \u2014C(O)CH\u2550CHCH 2 N(CH 3 )(COOC(CH 3 ) 3 , \u2014C(O)CH\u2550CHCH 2 NH(CH 3 ), \u2014C(O)CH 2 CH 3 , \u2014C(O)CH 2 CH 2 CH 3 , \u2014C(O)CH 2 CH 2 Cl, \u2014C(O)CH 2 CN,

Metadata:
- Claim Count in Document: 11.0
- Percentile: 88.0
- Lexical Diversity: 1.13889
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['15323929', '14708099', '14081053', '13828285', '15309396']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7162282006289751
- 35 USC 102 Novelty (BERT): 0.5204157265609543
- Combined Prediction Score: 0.6966469532221731
- Mean Citation Score: 266.72180799999995
- Max Citation Score: 289.41644
- Similarity Product: 200.5829178685308

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test