PATENT CLAIM ANALYSIS

Application Number: 16118376
Application Type: Utility
Filing Date: 2018-08
Publication Date: 2019-05
Patent Classification: ["544", "353000"]

Abstract:
A heterocyclic compound represented by the general formula (1) or a salt thereof: wherein m, l, and n respectively represent an integer of 1 or 2; X represents —O— or —CH 2 —; R 1  represents hydrogen, a lower alkyl group, a hydroxy-lower alkyl group, a protecting group, or a tri-lower alkylsilyloxy-lower alkyl group; R 2  and R 3 , which are the same or different, each independently represent hydrogen or a lower alkyl group; or R 2  and R 3  are bonded to form a cyclo-C3-C8 alkyl group; and R 4  represents an aromatic group or a heterocyclic group, wherein the aromatic or heterocyclic group may have one or more arbitrary substituent(s).

Claim (Index 4):
The method according to  claim 1 , wherein in the compound represented by the formula (1) or a pharmaceutically acceptable salt thereof m represents 2; l and n respectively represent 1; X represents \u2014CH 2 \u2014;\n R 1  represents hydrogen, a C1-C6 alkyl group, a hydroxy C1-C6 alkyl group, a benzyl group, or a tri C1-C6 alkylsilyloxy C1-C6 alkyl group; and R 4  represents any of (1) a phenyl group, (2) an indolyl group, (4) a naphthyl group, (5) a benzofuryl group, and (31) a pyrrolopyridyl group, wherein these aromatic or heterocyclic groups may have 1 to 4 substituent(s) selected from (1-1) a halogen atom, (1-2) a C1-C6 alkyl group, (1-3) a C1-C6 alkanoyl group, (1-4) a halogen-substituted C1-C6 alkyl group, (1-5) a halogen-substituted C1-C6 alkoxy group, (1-6) a cyano group, (1-7) a C1-C6 alkoxy group, (1-8) a C1-C6 alkylthio group, (1-9) an imidazolyl group, (1-10) a tri C1-C6 alkylsilyl group, (1-11) an oxadiazolyl group which may have 1 C1-C6 alkyl group, (1-12) a pyrrolidinyl group which may have 1 oxo group, (1-13) a phenyl group which may have 1 C1-C6 alkoxy group, (1-14) a C1-C6 alkylamino C1-C6 alkyl group, (1-15) an oxo group, (1-16) a pyrazolyl group which may have 1 C1-C6 alkyl group, (1-17) a thienyl group, (1-18) a furyl group, (1-19) a thiazolyl group which may have 1 C1-C6 alkyl group, (1-20) a C1-C6 alkylamino group, (1-21) a pyrimidyl group which may have 1 C1-C6 alkyl group, (1-22) a phenyl C2-C6 alkenyl group, (1-23) a phenoxy group which may have 1 halogen atom, (1-24) a phenoxy C1-C6 alkyl group, (1-25) a pyrrolidinyl C1-C6 alkoxy group, (1-26) a C1-C6 alkylsulfamoyl group, (1-27) a pyridazinyloxy group which may have 1 C1-C6 alkyl group, (1-28) a phenyl C1-C6 alkyl group, (1-29) a C1-C6 alkylamino C1-C6 alkoxy group, (1-30) an imidazolyl C1-C6 alkyl group, (1-31) a phenyl C1-C6 alkoxy group, (1-32) a hydroxy group, (1-34) a hydroxy C1-C6 alkyl group, (1-35) an oxazolyl group, (1-36) a piperidyl group, (1-37) a pyrrolyl group, (1-38) a morpholinyl C1-C6 alkyl group, (1-39) a piperazinyl C1-C6 alkyl group which may have 1 C1-C6 alkyl group(s), (1-40) a piperidyl C1-C6 alkyl group, (1-41) a pyrrolidinyl C1-C6 alkyl group, (1-42) a morpholinyl group, and (1-43) a piperazinyl group which may have 1 C1-C6 alkyl group.

Metadata:
- Claim Count in Document: 13.0
- Percentile: 96.0
- Lexical Diversity: 2.07812
- Patent Class: 544.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['13822589', '15495862', '11991146', '13270544', '13388442']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7815909779964433
- 35 USC 102 Novelty (BERT): 0.6016447215165989
- Combined Prediction Score: 0.7635963523484588
- Mean Citation Score: 383.689886
- Max Citation Score: 503.9384
- Similarity Product: 494.5008429306507

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test