PATENT CLAIM ANALYSIS

Application Number: 16003990
Application Type: Utility
Filing Date: 2018-06
Publication Date: 2018-10
Patent Classification: ["546", "081000"]

Abstract:
The present invention relates to compounds of formulas III and V that are useful as pharmaceutical agents, particularly as autophagy inhibitors.

Claim (Index 2):
The compound of  claim 1 , wherein:\n Q is CH or N; R N  is \u2014H; R 1  is \u2014H, \u2014F, \u2014Cl, \u2014Br, or \u2014CF 3 ; R 2  is \u2014CH(R 2-1 )\u2014(CH 2 ) n2 \u2014X;\n R 2-1  is \u2014H, C 1 -C 3  alkyl, or C 3  cycloalkyl; \n n 2  is 3; \n X is \n where X 1-2  is selected from the group consisting of H, linear or branched C 1 -C 4  alkyl, cyclopropyl, cyclobutyl , and \u2014SO 2 \u2014X 1-4  where X 1-4  is selected from H and C 1 -C 3  alkyl; and X 1-3  is a linear or branched C 1 -C 4  alkyl substituted with one cyclopropyl; R 3  is \u2014H, \u2014F, \u2014Cl, \u2014Br, \u2014CF 3 , \u2014OR 4-1  where R 4-1  is H or C 1 -C 6  alkyl, \u2014N(R 4-1 ) 2  where the R 4-1  are the same or different and are as defined above, or \u2014SR 4-1  where R 4-1  is as defined above; R 4  is \u2014H, \u2014F, \u2014Cl, \u2014Br, \u2014CF 3 , \u2014OR 4-1  where R 4-1  is H or C 1 -C 6  alkyl, \u2014-N(R 4-1 ) 2  where the R 4-1  are the same or different and are as defined above, or \u2014SR 4-1  where R 4-1  is as defined above; and R 5  is \u2014H, \u2014F, \u2014Cl, \u2014Br, \u2014CF 3 , \u2014OR 4-1  where R 4-1  is H or C 1 -C 6  alkyl, \u2014N(R 4-1 ) 2  where the R 4-1  are the same or different and are as defined above, or \u2014SR 4-1  where R 4-1  is as defined above;\n with the proviso that one of R 1 , R 3 , R 4 , and R 5  must be other than \u2014H.

Metadata:
- Claim Count in Document: 11.0
- Percentile: 94.0
- Lexical Diversity: 1.04545
- Patent Class: 546.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['14116650', '15384823', '13995889', '14173072', '12316848']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7669097168537478
- 35 USC 102 Novelty (BERT): 0.5324030815463565
- Combined Prediction Score: 0.7434590533230087
- Mean Citation Score: 256.67405799999995
- Max Citation Score: 352.04474
- Similarity Product: 250.39761528948188

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test