PATENT CLAIM ANALYSIS

Application Number: 15867010
Application Type: Utility
Filing Date: 2018-01
Publication Date: 2018-05
Patent Classification: ["546", "071000"]

Abstract:
The invention provides novel compounds having the general formula: wherein R 1  to R 6 , V, W, X and Y are as described herein, compositions including the compounds and methods of using the compounds.

Claim (Index 1):
A compound of formula I, wherein R 1 , R 2 , R 3  and R 4  are independently selected from hydrogen, C 1-6  alkyl, haloC 1-6  alkyl, halogen, cyano, amino, C 1-6  alkylamino, diC 1-6  alkylamino, pyrrolidinyl and OR 7 ; R 5  is hydrogen or C 1-6  alkyl; R 6  is hydrogen or C 1-6  alkyl; R 7  is hydrogen; C 1-6  alkyl; haloC 1-6  alkyl; C 3-7  cycloalkylC 1-6  alkyl; phenylC 1-6  alkyl; cyanoC 1-6 alkyl; hydroxyC 1-6 alkyl; C 1-6 alkoxyC 1-6  alkyl; carboxyC 1-6  alkyl; C 1-6 alkoxycarbonylC 1-6  alkyl; C 1-6 alkylsulfanylC 1-6  alkyl; C 1-6  alkylsulfonylC 1-6 alkyl; aminoC 1-6  alkyl; C 1-6  alkylaminoC 1-6 alkyl; diC 1-6  alkylaminoC 1-6  alkyl; C 1-6  alkylcarbonylaminoC 1-6  alkyl; C 1-6  alkylsulfonylaminoC 1-6 alkyl; C 1-6  alkoxycarbonylaminoC 1-6  alkyl; or heterocycloalkylC 1-6  alkyl, wherein heterocycloalkyl is N-containing monocyclic heterocycloalkyl; One of V, W, X and Y is selected from CR 8 R 9 , O, S, SO 2  and NR 10 , the others of V, W, X and Y are independently selected from a bond and CR 8 R 9 , wherein\n R 8  is hydrogen or C 1-6  alkyl; \n R 9  is hydrogen or C 1-6  alkyl; \n R 10  is phenylC 1-6  alkoxycarbonyl, phenylC 1-6  alkylcarbonyl, phenylC 1-6  alkylsulfonyl, C 1-6  alkoxycarbonyl, C 1-6  alkylcarbonyl, or C 1-6  alkylsulfonyl; \n or a pharmaceutically acceptable salt, or an enantiomer, or a diastereomer thereof.

Metadata:
- Claim Count in Document: 53.0
- Percentile: 86.0
- Lexical Diversity: 1.29032
- Patent Class: 546.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15866429', '15866954', '14926393', '15674810', '15639966']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8372120713502811
- 35 USC 102 Novelty (BERT): 0.584840886446973
- Combined Prediction Score: 0.8119749528599504
- Mean Citation Score: 442.209188
- Max Citation Score: 484.67615
- Similarity Product: 473.8524716412217

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test