PATENT CLAIM ANALYSIS

Application Number: 16080248
Application Type: Utility
Filing Date: 2018-08
Publication Date: 2019-02
Patent Classification: ["424", "490000"]

Abstract:
The present invention relates to a preparation containing esomeprazole as an active ingredient. The present invention is characterized in that a controlled-release system is introduced such that the efficacy of esomeprazole, which is an active ingredient, can be continuously exhibited.

Claim (Index 1):
A preparation comprising a plurality of unit sections including a first section pellet comprising an inert core, a drug layer coated on the inert core, and an outermost layer coated with an enteric layer; and a second section pellet comprising an inert core, a drug layer coated on the inert core, and an outermost layer coated with an enteric layer,\n wherein the drug layer of the first section pellet contains esomeprazole as an active ingredient, and the drug layer of the second section pellet contains esomeprazole as an active ingredient and meglumine as a solubilizer, wherein in the first section, when testing with 100 rotations per minute according to the first elution test method, the active ingredient in the unit section is released in the amount of 5% or less relative to the total amount until 10 minutes after elution initiation, and the active ingredient is released in the amount of 80% or more relative to the total amount until 30 minutes, and in the second section, when testing with 100 rotations per minute according to the first elution test method, the active ingredient in the unit section is released in the amount of 5% or less relative to the total amount until 3 hours after elution initiation, and the active ingredient is released in the amount of 70% or more relative to the total amount until 5 hours.

Metadata:
- Claim Count in Document: 11.0
- Percentile: 96.0
- Lexical Diversity: 1.41935
- Patent Class: 424.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['12630271', '14771207', '14484754', '15616494', '14463776']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7048087779616447
- 35 USC 102 Novelty (BERT): 0.4808968917583477
- Combined Prediction Score: 0.682417589341315
- Mean Citation Score: 188.329046
- Max Citation Score: 191.15828
- Similarity Product: 140.32231724189282

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test