PATENT CLAIM ANALYSIS

Application Number: 15988325
Application Type: Utility
Filing Date: 2018-05
Publication Date: 2018-09
Patent Classification: ["424", "441000"]

Abstract:
A process for the manufacture of semi-plastic pharmaceutical unit doses using a rotary moulding machine and semi-plastic pharmaceutical dosage units obtained by this process.

Claim (Index 7):
The process according to  claim 1 , wherein the active pharmaceutical ingredient is an isoxazoline compound of Formula (I) wherein R 1 =halogen, CF 3 , OCF 3 , CN, n=integer from 0 to 3, R 2 =C 1 -C 3 -haloalkyl, T=5- or 6-membered ring, which is optionally substituted by one or more radicals Y, Y=methyl, halomethyl, halogen, CN, NO 2 , NH 2 \u2014C\u2550S, or two adjacent radicals Y form together a chain; Q=X\u2014NR 3 R 4  or a 5-membered N-heteroaryl ring, which is optionally substituted by one or more radicals; X=CH 2 , CH(CH 3 ), CH(CN), CO, CS, R 3 =hydrogen, methyl, haloethyl, halopropyl, halobutyl, methoxymethyl, methoxyethyl, halomethoxymethyl, ethoxymethyl, haloethoxymethyl, propoxymethyl, ethylaminocarbonylmethyl, ethylaminocarbonylethyl, dimethoxyethyl, propynylaminocarbonylmethyl, N-phenyl-N-methyl-amino, haloethylaminocarbonylmethyl, haloethylaminocarbonylethyl, tetrahydrofuryl, methylaminocarbonylmethyl, (N,N-dimethylamino)-carbonylmethyl, propylaminocarbonylmethyl, cyclopropylaminocarbonylmethyl, propenylaminocarbonylmethyl, haloethylaminocarbonylcyclopropyl, wherein Z A =hydrogen, halogen, cyano, halomethyl (CF 3 ); R 4 =hydrogen, ethyl, methoxymethyl, halomethoxymethyl, ethoxymethyl, haloethoxymethyl, propoxymethyl, methylcarbonyl, ethylcarbonyl, propylcarbonyl, cyclopropylcarbonyl, methoxycarbonyl, methoxymethylcarbonyl, am inocarbonyl, ethylaminocarbonylmethyl, ethylaminocarbonylethyl, dimethoxyethyl, propynylaminocarbonylmethyl, haloethylaminocarbonylmethyl, cyanomethylaminocarbonylmethyl, or haloethylaminocarbonylethyl; Or R 3  and R 4  together form a substituent selected from the group consisting of: or a salt or solvate thereof.

Metadata:
- Claim Count in Document: 4.0
- Percentile: 93.0
- Lexical Diversity: 1.13636
- Patent Class: 424.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['14082813', '14390052', '13754969', '14977680', '15936778']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.764687917112426
- 35 USC 102 Novelty (BERT): 0.5289879217964654
- Combined Prediction Score: 0.74111791758083
- Mean Citation Score: 229.917072
- Max Citation Score: 359.86172
- Similarity Product: 315.47740119782924

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test