PATENT CLAIM ANALYSIS

Application Number: 15742333
Application Type: Utility
Filing Date: 2018-01
Publication Date: 2018-07
Patent Classification: ["504", "343000"]

Abstract:
The present invention relates phenoxyhalogenphenylamidines of the general formula (I), to a process for their preparation, to the use of the amidines according to the invention for controlling unwanted microorganisms and also to an agrochemical formulation for this purpose, comprising the phenoxyhalogenphenylamidines according to the invention. Furthermore, the invention relates to a method for controlling unwanted microorganisms by applying the compounds according to the invention to the microorganisms and/or their habitat.

Claim (Index 5):
A process for preparing a compound as claimed in  claim 1  which comprises at least one of the following (a) to (j):\n (a) reaction of a nitrobenzene derivative of formula (III) with a phenol derivative of formula (II) according to the reaction scheme below: \n (b) reaction of a nitrophenol derivative of formula (V) with a phenyl derivative of formula (IV) according to the reaction scheme below: (c) reaction of an aniline of formula (VII) with a phenol derivative of formula (II) according to the reaction scheme below: (d) reaction of an aminophenol of formula (XII) with a phenyl derivative of formula (IV) according to the reaction scheme below: (e) reduction of a nitrophenyl ether of formula (VI) to an aminophenyl ether of the formula (VIII) according to the reaction scheme below: (f) reaction of a aminophenyl ether of formula (VIII) with (i) aminoacetal of formula (XIII) or (ii) with N-ethyl-N-methylformamide of formula (XIV) or (iii) with N-methylethanamine of formula (XV) in the presence of ortho ester of formula (XVI) according to the reaction scheme below: (g) reaction of an aminophenol of formula (XII) with (i) aminoacetal of formula (XIII) or (ii) with N-ethyl-N-methylformamide of formula (XIV) or (iii) with N-methylethanamine of formula (XV) in the presence of an ortho ester of formula (XVI) according to the reaction scheme below: (h) reaction of an aniline of formula (VII) with (i) aminoacetal of formula (XIII) or (ii) with N-ethyl-N-methylformamide of formula (XIV) or (iii) with N-methylethanamine of formula (XV) in the presence of an ortho ester of formula (XVI) according to the reaction scheme below: (i) reaction of an amidine of formula (XI) with a phenol derivative of the formula (II) according to the reaction scheme below: (j) reaction of an amidine of formula (XI) with a phenyl derivative of formula (IV) according to the reaction scheme below: where in the above schemes Z is a leaving group; R 6  and R 7  independently of one another are selected from the group consisting of C 1-12 -alkyl, C 2-12 -alkenyl, C 2-12 -alkynyl or C 5-18 -aryl or C 7-19 -arylalkyl groups and together with the atoms to which they are attached may form a five-, six- or seven-membered ring; R 8  to R 10  independently of one another are selected from the group consisting of C 1-12 -alkyl, C 2-12 -alkenyl, C 2-12 -alkynyl or C 5-18 -aryl or C 7-19 -arylalkyl, C 7-19 -alkylaryl groups and in each case R 8  with R 9 , R 9  with R 10  or R 8  with R 10  together with the atoms to which they are attached and if appropriate together with further carbon, nitrogen, oxygen or sulfur atoms may form a five-, six- or seven-membered ring.

Metadata:
- Claim Count in Document: 33.0
- Percentile: 86.0
- Lexical Diversity: 1.92683
- Patent Class: 504.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15736242', '15735718', '14783216', '15563414', '13000268']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7732932653054941
- 35 USC 102 Novelty (BERT): 0.5314690905196808
- Combined Prediction Score: 0.7491108478269128
- Mean Citation Score: 265.29646
- Max Citation Score: 322.6216
- Similarity Product: 312.26763178524965

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test