PATENT CLAIM ANALYSIS

Application Number: 15747850
Application Type: Utility
Filing Date: 2018-01
Publication Date: 2018-08
Patent Classification: ["514", "254030"]

Abstract:
The present invention relates to novel compounds having histone deacetylase 6 (HDAC6) inhibitory activity, stereoisomers thereof or pharmaceutically acceptable salts thereof, the use thereof for the preparation of therapeutic medicaments, pharmaceutical compositions containing the same, a method for treating diseases using the composition, and methods for preparing the novel compounds. The novel compounds, stereoisomers thereof or pharmaceutically acceptable salts thereof according to the present invention have histone deacetylase (HDAC) inhibitory activity and are effective for the prevention or treatment of HDAC6-mediated diseases, including infectious diseases; neoplasms; endocrine, nutritional and metabolic diseases; mental and behavioral disorders; neurological diseases; diseases of the eye and adnexa; cardiovascular diseases; respiratory diseases; digestive diseases; diseases of the skin and subcutaneous tissue; diseases of the musculoskeletal system and connective tissue; or congenital malformations, deformations and chromosomal abnormalities.

Claim (Index 7):
The 1,3,4-oxadiazole sulfamide derivative compound represented by formula I, stereoisomer thereof or pharmaceutically acceptable salt thereof according to  claim 6 , wherein the compound represented by formula I is selected from the group consisting of compounds described in the following table: Ex. Comp. Structure 11 11301   12 11302   13 11303   15 11305   16 11306   23 11313   24 11314   25 11315   26 11316   33 11363   34 11379   35 11440   36 11498   39 11574   42 11641   49 11654   50 11659   54 11670   55 11671   56 11672   68 11825   72 11829   73 11830   74 11831   75 11832

Metadata:
- Claim Count in Document: 20.0
- Percentile: 86.0
- Lexical Diversity: 1.98734
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15747952', '15748081', '15763972', '11252232', '13522044']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8249050530208911
- 35 USC 102 Novelty (BERT): 0.5784409379161248
- Combined Prediction Score: 0.8002586415104145
- Mean Citation Score: 389.701144
- Max Citation Score: 467.68665
- Similarity Product: 424.1081372368991

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test