PATENT CLAIM ANALYSIS

Application Number: 15745315
Application Type: Utility
Filing Date: 2018-01
Publication Date: 2018-07
Patent Classification: ["504", "103000"]

Abstract:
The invention relates to substituted heteroaryl carboxylic acid hydrazides of general formula (I) or salts thereof, wherein the groups of formula (I) have the definitions stated in the description, for increasing the stress tolerance in plants with respect to abiotic stress, and also for strengthening plant growth and/or for increasing plant yield.

Claim (Index 1):
A substituted heteroarylcarbonyl hydrazide of formula (I) or salt thereof in which R 1 , R 2  and R 7  are independently hydrogen, halogen, cyano, nitro, NR 21 R 22 , OR 23 , S(O) n R 24 , thiocyanato, isothiocyanato, (C 1 -C 8 )-alkyl, (C 2 -C 8 )-alkenyl, (C 2 -C 8 )-alkynyl, (C 1 -C 10 )-haloalkyl, (C 2 -C 8 )-haloalkenyl, (C 2 -C 8 )-haloalkynyl, (C 3 -C 10 )-cycloalkyl, (C 3 -C 10 )-halocycloalkyl, (C 4 -C 10 )-cycloalkenyl, (C 4 -C 10 )-halocycloalkenyl, pentafluorothio, (C 1 -C 8 )-alkoxy-(C 1 -C 8 )-haloalkyl, (C 1 -C 8 )-haloalkoxy-(C 1 -C 8 )-haloalkyl, (C 1 -C 8 )-haloalkoxy-(C 1 -C 8 )-alkyl, aryl, aryl-(C 1 -C 8 )-alkyl, heteroaryl, heteroaryl-(C 1 -C 8 )-alkyl, (C 3 -C 8 )-cycloalkyl-(C 1 -C 8 )-alkyl, (C 4 -C 10 )-cycloalkenyl-(C 1 -C 8 )-alkyl, heterocyclyl, heterocyclyl-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkoxy-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkylthio-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-haloalkylthio-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkylcarbonyl-(C 1 -C 8 )-alkyl, COOR 23 , CONR 21 R 22 , COR 23 , \u2014C\u2550NOR 23 , R 21 R 22 N\u2014(C 1 -C 8 )-alkyl, R 23 OOC\u2014(C 1 -C 8 )-alkyl, aryl-(C 1 -C 8 )-alkynyl, heteroaryl-(C 1 -C 8 )-alkynyl, heterocyclyl-(C 1 -C 8 )-alkynyl, tris[(C 1 -C 8 )-alkyl]silyl-(C 2 -C 8 )-alkynyl, bis[(C 1 -C 8 )-alkyl](aryl)silyl-(C 2 -C 8 )-alkynyl, bisaryl[(C 1 -C 8 )-alkyl]silyl-(C 2 -C 8 )-alkynyl, (C 3 -C 8 )-cycloalkyl-(C 2 -C 8 )-alkynyl, aryl-(C 2 -C 8 )-alkenyl, heteroaryl-(C 2 -C 8 )-alkenyl, heterocyclyl-(C 2 -C 8 )-alkenyl, (C 3 -C 8 )-cycloalkyl-(C 2 -C 8 )-alkenyl, (C 1 -C 8 )-alkoxy-(C 1 -C 8 )-alkoxy-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkylaminosulfonylamino, (C 3 -C 8 )-cycloalkylaminosulfonylamino, diazo, aryldiazo, tris[(C 1 -C 8 )-alkyl]silyl, bis[(C 1 -C 8 )-alkyl](aryl)silyl, bisaryl[(C 1 -C 8 )-alkyl]silyl, X 1 , X 2  and X 3  are the same or different and are independently O (oxygen), S (sulfur), N (nitrogen), the C\u2014R 2  moiety or the N\u2014R 20  moiety, but no oxygen and sulfur atom are ever adjacent and there is never more than one oxygen or sulfur atom in the 5-membered ring formed, and where R 2  in the C\u2014R 2  moiety and R 20  in the N\u2014R 20  moiety are each the same or different as defined above or below, W is O (oxygen) or S (sulfur), A 1 , A 2 , A 3 , A 4  and A 5  are the same or different and are each independently N (nitrogen) or the C\u2014R 7  moiety, but there are never more than two adjacent nitrogen atoms, and where R 7  in each C\u2014R 7  moiety is the same or different as defined above, R 3  is (C 1 -C 8 )-alkyl, cyano-(C 1 -C 8 )-alkyl, (C 2 -C 8 )-alkenyl, (C 2 -C 8 )-alkynyl, (C 1 -C 10 )-haloalkyl, (C 2 -C 8 )-haloalkenyl, (C 2 -C 8 )-haloalkynyl, (C 3 -C 10 )-cycloalkyl, (C 3 -C 10 )-halocycloalkyl, (C 4 -C 10 )-cycloalkenyl, (C 4 -C 10 )-halocycloalkenyl, aryl, aryl-(C 1 -C 8 )-alkyl, heteroaryl, heteroaryl-(C 1 -C 8 )-alkyl, (C 3 -C 8 )-cycloalkyl-(C 1 -C 8 )-alkyl, heterocyclyl, heterocyclyl-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkoxy-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkylthio-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-haloalkoxy-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-haloalkylthio-(C 1 -C 8 )-alkyl, R 21 R 22 N\u2014(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkoxy-(C 1 -C 8 )-alkoxy-(C 1 -C 8 )-alkyl, R 4  is hydrogen, (C 1 -C 8 )-alkyl, (C 2 -C 8 )-alkenyl, (C 2 -C 8 )-alkynyl, (C 1 -C 10 )-haloalkyl, (C 2 -C 8 )-haloalkenyl, (C 2 -C 8 )-haloalkynyl, (C 3 -C 10 )-cycloalkyl, (C 3 -C 10 )-halocycloalkyl, (C 4 -C 10 )-cycloalkenyl, (C 4 -C 10 )-halocycloalkenyl, aryl, aryl-(C 1 -C 8 )-alkyl, heteroaryl, heteroaryl-(C 1 -C 8 )-alkyl, (C 3 -C 8 )-cycloalkyl-(C 1 -C 8 )-alkyl, heterocyclyl, heterocyclyl-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkoxy-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkylthio-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-haloalkoxy-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-haloalkylthio-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkylamino-(C 1 -C 8 )-alkyl, bis[(C 1 -C 8 )-alkyl]amino-(C 1 -C 8 )-alkyl, (C 3 -C 8 )-cycloalkylamino-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkoxy-(C 1 -C 8 )-alkoxy-(C 1 -C 8 )-alkyl, COR 23 , (C 1 -C 8 )-alkoxycarbonyl, (C 2 -C 8 )-alkenyloxycarbonyl, (C 2 -C 8 )-alkynyloxycarbonyl, aryl-(C 1 -C 8 )-alkoxycarbonyl, heteroaryl-(C 1 -C 8 )-alkoxycarbonyl, (C 3 -C 8 )-cycloalkyl-(C 1 -C 8 )-alkoxycarbonyl, CONR 21 R 22 , SO 2 R 24  hydroxycarbonyl-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkoxycarbonyl-(C 1 -C 8 )-alkyl, (C 2 -C 8 )-alkenyloxycarbonyl-(C 1 -C 8 )-alkyl, (C 2 -C 8 )-alkynyloxycarbonyl-(C 1 -C 8 )-alkyl, aryl-(C 1 -C 8 )-alkoxycarbonyl-(C 1 -C 8 )-alkyl, heteroaryl-(C 1 -C 8 )-alkoxycarbonyl-(C 1 -C 8 )-alkyl, heterocyclyl-(C 1 -C 8 )-alkoxycarbonyl-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkylcarbonyl-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkylsulfonyl-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkylsulfynyl-(C 1 -C 8 )-alkyl, R 5  and R 6  are independently hydrogen, (C 1 -C 8 )-alkyl, (C 2 -C 8 )-alkenyl, (C 2 -C 8 )-alkynyl, (C 1 -C 10 )-haloalkyl, (C 2 -C 8 )-haloalkenyl, (C 2 -C 8 )-haloalkynyl, (C 3 -C 10 )-cycloalkyl, (C 3 -C 10 )-halocycloalkyl, (C 4 -C 10 )-cycloalkenyl, (C 4 -C 10 )-halocycloalkenyl, aryl, aryl-(C 1 -C 8 )-alkyl, heteroaryl, heteroaryl-(C 1 -C 8 )-alkyl, (C 3 -C 8 )-cycloalkyl-(C 1 -C 8 )-alkyl, heterocyclyl, heterocyclyl-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkoxy-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkylthio-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-haloalkoxy-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-haloalkylthio-(C 1 -C 8 )-alkyl, COOR 23 , CONR 21 R 22 , hydroxycarbonyl-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkoxycarbonyl-(C 1 -C 8 )-alkyl, (C 2 -C 8 )-alkenyloxycarbonyl-(C 1 -C 8 )-alkyl, (C 2 -C 8 )-alkynyloxycarbonyl-(C 1 -C 8 )-alkyl, aryl-(C 1 -C 8 )-alkoxycarbonyl-(C 1 -C 8 )-alkyl, heteroaryl-(C 1 -C 8 )-alkoxycarbonyl-(C 1 -C 8 )-alkyl, heterocyclyl-(C 1 -C 8 )-alkoxycarbonyl-(C 1 -C 8 )-alkyl, R 3  and R 4  together with the nitrogen atom to which they are bonded form a fully saturated, partly saturated or fully unsaturated 3-7-membered ring optionally interrupted by heteroatoms and optionally having further substitution, R 1  and X 1 , when X 1  is a C\u2014R 2  group, together with the atoms to which they are bonded form a fully saturated, partly saturated or fully unsaturated 5-7-membered ring optionally interrupted by heteroatoms and optionally having further substitution, X 1  and X 2 , when each is a C\u2014R 2  group, together with the atoms to which they are bonded form a fully saturated, partly saturated or fully unsaturated 5-7-membered ring optionally interrupted by heteroatoms and optionally having further substitution, A 1  and A 2 , when each is a C\u2014R 7  group, together with the atoms to which they are bonded form a fully saturated, partly saturated or fully unsaturated 5-7-membered ring optionally interrupted by heteroatoms and optionally having further substitution, A 2  and A 3 , when each is a C\u2014R 7  group, together with the atoms to which they are bonded form a fully saturated, partly saturated or fully unsaturated 5-7-membered ring optionally interrupted by heteroatoms and optionally having further substitution and A 3  and A 4 , when each is a C\u2014R 7  group, together with the atoms to which they are bonded form a fully saturated, partly saturated or fully unsaturated 5-7-membered ring optionally interrupted by heteroatoms and optionally having further substitution, Y is a bond or the Y-1 to Y-7 moieties where R 8 , R 9 , R 10 , R 11 , R 12 , R 13 , R 14 , R 15 , R 16 , R 17 , R 18  and R 19  are each as per the definition below and where the arrow represents a bond to the 6-membered ring with the A 1 , A 2 , A 3 , A 4  and A 5  moieties,\n R 8 , R 9 , R 10 , R 11 , R 12 , R 13 , R 14 , R 15 , R 16 , R 17 , R 18  and R 19  are independently hydrogen, halogen, (C 1 -C 8 )-alkyl, (C 2 -C 8 )-alkenyl, (C 2 -C 8 )-alkynyl, (C 1 -C 10 )-haloalkyl, (C 2 -C 8 )-haloalkenyl, (C 2 -C 8 )-haloalkynyl, (C 3 -C 10 )-cycloalkyl, aryl, aryl-(C 1 -C 8 )-alkyl, heteroaryl, heteroaryl-(C 1 -C 8 )-alkyl, (C 3 -C 8 )-cycloalkyl-(C 1 -C 8 )-alkyl, heterocyclyl, heterocyclyl-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkoxy-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkylthio-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-haloalkoxy-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-haloalkylthio-(C 1 -C 8 )-alkyl, COOR 23 , \n R 5  and R 6  together with the atom to which they are bonded form a fully saturated or partly saturated 5-7-membered ring optionally interrupted by heteroatoms and optionally having further substitution, \n R 20  is hydrogen, (C 1 -C 8 )-alkyl, (C 2 -C 8 )-alkenyl, (C 2 -C 8 )-alkynyl, (C 1 -C 10 )-haloalkyl, (C 2 -C 8 )-haloalkenyl, (C 2 -C 8 )-haloalkynyl, (C 3 -C 10 )-cycloalkyl, (C 4 -C 10 )-cycloalkenyl, (C 1 -C 8 )-alkoxy, aryl, heteroaryl, heterocyclyl, (C 1 -C 8 )-alkylcarbonyl, aryl-(C 1 -C 8 )-alkylcarbonyl, (C 3 -C 8 )-cycloalkylcarbonyl, arylcarbonyl, heteroarylcarbonyl, (C 1 -C 8 )-alkoxycarbonyl, (C 2 -C 8 )-alkenyloxycarbonyl, aryl-(C 1 -C 8 )-alkoxycarbonyl, heteroaryl-(C 1 -C 8 )-alkoxycarbonyl, (C 3 -C 8 )-cycloalkyl-(C 1 -C 8 )-alkoxycarbonyl, (C 1 -C 8 )-alkylsulfonyl, (C 1 -C 8 )-haloalkylsulfonyl, arylsulfonyl, heteroarylsulfonyl, (C 3 -C 8 )-cycloalkylsulfonyl, (C 1 -C 8 )-alkylsulfinyl, arylsulfinyl, heteroarylsulfinyl, (C 3 -C 8 )-cycloalkylsulfinyl, \n n is 0, 1 or 2, \n R 21  and R 22  are the same or different and are independently hydrogen, (C 1 -C 8 )-alkyl, (C 2 -C 8 )-alkenyl, (C 2 -C 8 )-alkynyl, (C 1 -C 8 )-cyanoalkyl, (C 1 -C 10 )-haloalkyl, (C 2 -C 8 )-haloalkenyl, (C 2 -C 8 )-haloalkynyl, (C 3 -C 10 )-cycloalkyl, (C 3 -C 10 )-halocycloalkyl, (C 4 -C 10 )-cycloalkenyl, (C 4 -C 10 )-halocycloalkenyl, (C 1 -C 8 )-alkoxy-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-haloalkoxy-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkylthio-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-haloalkylthio-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkoxy-(C 1 -C 8 )-haloalkyl, aryl, aryl-(C 1 -C 8 )-alkyl, heteroaryl, heteroaryl-(C 1 -C 8 )-alkyl, (C 3 -C 8 )-cycloalkyl-(C 1 -C 8 )-alkyl, (C 4 -C 10 )-cycloalkenyl-(C 1 -C 8 )-alkyl, COR 23 , SO 2 R 24 , (C 1 -C 8 )-alkyl-HNO 2 S\u2014, (C 3 -C 8 )-cycloalkyl-HNO 2 S\u2014, heterocyclyl, (C 1 -C 8 )-alkoxycarbonyl-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkoxycarbonyl, aryl-(C 1 -C 8 )-alkoxycarbonyl-(C 1 -C 8 )-alkyl, aryl-(C 1 -C 8 )-alkoxycarbonyl, heteroaryl-(C 1 -C 8 )-alkoxycarbonyl, (C 2 -C 8 )-alkenyloxycarbonyl, (C 2 -C 8 )-alkynyloxycarbonyl, heterocyclyl-(C 1 -C 8 )-alkyl, \n R 23  is hydrogen, (C 1 -C 8 )-alkyl, (C 2 -C 8 )-alkenyl, (C 2 -C 8 )-alkynyl, (C 1 -C 8 )-cyanoalkyl, (C 1 -C 10 )-haloalkyl, (C 2 -C 8 )-haloalkenyl, (C 2 -C 8 )-haloalkynyl, (C 3 -C 10 )-cycloalkyl, (C 3 -C 10 )-halocycloalkyl, (C 4 -C 10 )-cycloalkenyl, (C 4 -C 10 )-halocycloalkenyl, (C 1 -C 8 )-alkoxy-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkoxy-(C 1 -C 8 )-haloalkyl, aryl, aryl-(C 1 -C 8 )-alkyl, heteroaryl, heteroaryl-(C 1 -C 8 )-alkyl, (C 3 -C 8 )-cycloalkyl-(C 1 -C 8 )-alkyl, (C 4 -C 10 )-cycloalkenyl-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkoxycarbonyl-(C 1 -C 8 )-alkyl, (C 2 -C 8 )-alkenyloxycarbonyl-(C 1 -C 8 )-alkyl, aryl-(C 1 -C 8 )-alkoxycarbonyl-(C 1 -C 8 )-alkyl, hydroxycarbonyl-(C 1 -C 8 )-alkyl, heterocyclyl, heterocyclyl-(C 1 -C 8 )-alkyl and \n R 24  is hydrogen, (C 1 -C 8 )-alkyl, (C 2 -C 8 )-alkenyl, (C 2 -C 8 )-alkynyl, (C 1 -C 8 )-cyanoalkyl, (C 1 -C 10 )-haloalkyl, (C 2 -C 8 )-haloalkenyl, (C 2 -C 8 )-haloalkynyl, (C 3 -C 10 )-cycloalkyl, (C 3 -C 10 )-halocycloalkyl, (C 4 -C 10 )-cycloalkenyl, (C 4 -C 10 )-halocycloalkenyl, (C 1 -C 8 )-alkoxy-(C 1 -C 8 )-alkyl, (C 1 -C 8 )-alkoxy-(C 1 -C 8 )-haloalkyl, aryl, aryl-(C 1 -C 8 )-alkyl, heteroaryl, heteroaryl-(C 1 -C 8 )-alkyl, heterocyclyl-(C 1 -C 8 )-alkyl, (C 3 -C 8 )-cycloalkyl-(C 1 -C 8 )-alkyl, (C 4 -C 10 )-cycloalkenyl-(C 1 -C 8 )-alkyl, NR 21 R 22 .

Metadata:
- Claim Count in Document: 3.0
- Percentile: 86.0
- Lexical Diversity: 1.39535
- Patent Class: 504.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['13364168', '14075248', '13583798', '10482216', '14223103']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7450960493349008
- 35 USC 102 Novelty (BERT): 0.5675930832907449
- Combined Prediction Score: 0.7273457527304853
- Mean Citation Score: 360.603976
- Max Citation Score: 384.6131
- Similarity Product: 305.9198474300861

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 0
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test