PATENT CLAIM ANALYSIS

Application Number: 16141397
Application Type: Utility
Filing Date: 2018-09
Publication Date: 2019-03
Patent Classification: ["549", "483000"]

Abstract:
The present invention relates to fungicidal N-cycloalkyl-N-[(heterocyclylphenyl)methylene] carboxamide derivatives and their thiocarbonyl derivatives, their process of preparation and intermediate compounds for their preparation, their use as fungicides; particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions.

Claim (Index 16):
A compound of formula (IIa) wherein\n Z 2  and Z 3 , which can be the same or different, are a hydrogen atom; non-substituted C 1 -C 8 -alkyl; non-substituted C 2 -C 8 -alkenyl; non-substituted C 2 -C 8 -alkynyl; a halogen atom; non-substituted C 1 -C 8 -alkoxy; non-substituted C 2 -C 8 -alkenyloxy; or non-substituted C 2 -C 8 -alkynyloxy; \n n is 0, 1, 2, 3 or 4; \n each X is independently a halogen atom; nitro; cyano; isonitrile; hydroxy; amino; sulfanyl; pentafluoro-\u03bb 6 -sulfanyl; formyl; formyloxy; formylamino; substituted or non-substituted (hydroxyimino)-C 1 -C 8 -alkyl; substituted or non-substituted (C 1 -C 8 -alkoxyimino)-C 1 -C 8 -alkyl; substituted or non-substituted (C 2 -C 8 -alkenyloxyimino)-C 1 -C 8 -alkyl; substituted or non-substituted (C 2 -C 8 -alkynyloxyimino)-C 1 -C 8 -alkyl substituted or non-substituted (benzyloxyimino)-C 1 -C 8 -alkyl; carboxy; carbamoyl; N-hydroxycarbamoyl; carbamate; substituted or non-substituted C 1 -C 8 -alkyl; C 1 -C 8 -halogenoalkyl having 1 to 9 halogen atoms; substituted or non-substituted C 2 -C 8 -alkenyl; C 2 -C 8 -halogenoalkenyl having 1 to 9 halogen atoms; substituted or non-substituted C 2 -C 8 -alkynyl; C 2 -C 8 -halogenoalkynyl having 1 to 9 halogen atoms; substituted or non-substituted C 1 -C 8 -alkoxy; C 1 -C 8 -halogenoalkoxy having 1 to 9 halogen atoms; substituted or non-substituted C 1 -C 8 -alkylsulfanyl; C 1 -C 8 -halogenoalkylsulfanyl having 1 to 9 halogen atoms; substituted or non-substituted C 1 -C 8 -alkylsulfinyl; C 1 -C 8 -halogenoalkylsulfinyl having 1 to 9 halogen atoms; substituted or non-substituted C 1 -C 8 -alkylsulfonyl; C 1 -C 8 -halogenoalkylsulfonyl having 1 to 9 halogen atoms; substituted or non-substituted C 1 -C 8 -alkylamino; substituted or non-substituted di-C 1 -C 8 -alkylamino; substituted or non-substituted C 2 -C 8 -alkenyloxy; C 2 -C 8 -halogenoalkenyloxy having 1 to 9 halogen atoms; substituted or non-substituted C 3 -C 8 -alkynyloxy; C 2 -C 8 -halogenoalkynyloxy having 1 to 9 halogen atoms; substituted or non-substituted C 3 -C 7 -cycloalkyl; C 3 -C 7 -halogenocycloalkyl having 1 to 9 halogen atoms; substituted or non-substituted (C 3 -C 7 -cycloalkyl)-C 1 -C 8 -alkyl; substituted or non-substituted C 4 -C 7 -cycloalkenyl; C 4 -C 7 -halogenocycloalkenyl having 1 to 9 halogen atoms; substituted or non-substituted (C 3 -C 7 -cycloalkyl)-C 2 -C 8 -alkenyl; substituted or non-substituted (C 3 -C 7 -cycloalkyl)-C 2 -C 8 -alkynyl; substituted or non-substituted tri(C 1 -C 8 )alkylsilyl; substituted or non-substituted tri(C 1 -C 8 )alkylsilyl-C 1 -C 8 -alkyl; substituted or non-substituted C 1 -C 8 -alkylcarbonyl; C 1 -C 8 -halogenoalkylcarbonyl having 1 to 9 halogen atoms; substituted or non-substituted C 1 -C 8 -alkylcarbonyloxy; C 1 -C 8 -halogenoalkylcarbonyloxy having 1 to 9 halogen atoms; substituted or non-substituted C 1 -C 8 -alkylcarbonylamino; C 1 -C 8 -halogenoalkylcarbonylamino having 1 to 9 halogen atoms; substituted or non-substituted C 1 -C 8 -alkoxycarbonyl; C 1 -C 8 -halogenoalkoxycarbonyl having 1 to 9 halogen atoms; substituted or non-substituted C 1 -C 8 -alkyloxycarbonyloxy; C 1 -C 8 -halogenoalkoxycarbonyloxy having 1 to 9 halogen atoms; substituted or non-substituted C 1 -C 8 -alkylcarbamoyl; substituted or non-substituted di-C 1 -C 8 -alkylcarbamoyl; substituted or non-substituted C 1 -C 8 -alkylaminocarbonyloxy; substituted or non-substituted di-C 1 -C 8 -alkylaminocarbonyloxy; substituted or non-substituted N\u2014(C 1 -C 8 -alkyl)hydroxy carbamoyl; substituted or non-substituted C 1 -C 8 -alkoxycarbamoyl; substituted or non-substituted N\u2014(C 1 -C 8 -alkyl)-C 1 -C 8 -alkoxycarbamoyl; aryl that can be substituted by up to 6 groups Q which can be the same or different aryl-C 1 -C 8 -alkyl that can be substituted by up to 6 groups Q which can be the same or different aryl-C 2 -C 8 -alkenyl that can be substituted by up to 6 groups Q which can be the same or different aryl-C 2 -C 8 -alkynyl that can be substituted by up to 6 groups Q which can be the same or different aryloxy that can be substituted by up to 6 groups Q which can be the same or different arylsulfanyl that can be substituted by up to 6 groups Q which can be the same or different arylamino that can be substituted by up to 6 groups Q which can be the same or different aryl-C 1 -C 8 -alkyloxy that can be substituted by up to 6 groups Q which can be the same or different aryl-C 1 -C 8 -alkylsulfanyl that can be substituted by up to 6 groups Q which can be the same or different aryl-C 1 -C 8 -alkylamino that can be substituted by up to 6 groups Q which can be the same or different pyridinyl which can be substituted by up to 4 groups Q, or pyridinyloxy which can be substituted by up to 4 groups Q; \n each Q is independently a halogen atom, cyano, nitro, substituted or non-substituted C 1 -C 8 -alkyl, C 1 -C 8 -halogenoalkyl comprising up to 9 halogen atoms that can be the same or different, substituted or non-substituted C 1 -C 8 -alkoxy, C 1 -C 8 -halogenoalkoxy comprising up to 9 halogen atoms that can be the same or different, substituted or non-substituted C 1 -C 8 -alkylsulfanyl, C 1 -C 8 -halogenoalkylsulfanyl comprising up to 9 halogen atoms that can be the same or different, substituted or non-substituted tri(C 1 -C 8 )alkylsilyl, substituted or non-substituted tri(C 1 -C 8 )alkylsilyl-C 1 -C 8 -alkyl, substituted or non-substituted (C 1 -C 8 -alkoxyimino)-C 1 -C 8 -alkyl, or substituted or non-substituted (benzyloxyimino)-C 1 -C 8 -alkyl; \n L is a direct bond; and \n B is a substituted or non-substituted oxiranyl ring, a substituted or non-substituted thienyl ring, a substituted or non-substituted benzothienyl ring, a substituted or non-substituted furan ring, or a substituted or non-substituted benzofuran ring, \n providing that (IIa) does not represent:\n N-[2-(2-furyl)benzyl]cyclopropanamine; \n N-[2-(2-furyl)-4,5-dimethoxybenzyl]cyclopropanamine; \n N-[2-(3-bromo-2-furyl)-4,5-dimethoxybenzyl]cyclopropanamine; \n N-[2-(3-bromo-2-furyl)benzyl]cyclopropanamine; \n N-[2-(3-furyl)benzyl]cyclopropanamine; \n N-[2-(2-thienyl)benzyl]cyclopropanamine; or \n N-[4,5-dimethoxy-2-(2-thienyl)benzyl]cyclopropanamine, \n or a salt thereof.

Metadata:
- Claim Count in Document: 35.0
- Percentile: 97.0
- Lexical Diversity: 1.39535
- Patent Class: 549.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['14395038', '14388179', '14361534', '15176653', '15566159']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7681304269835985
- 35 USC 102 Novelty (BERT): 0.5750436538062451
- Combined Prediction Score: 0.7488217496658631
- Mean Citation Score: 414.81178
- Max Citation Score: 496.60413
- Similarity Product: 395.4001338701105

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test