PATENT CLAIM ANALYSIS

Application Number: 15763807
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2018-11
Patent Classification: ["544", "238000"]

Abstract:
The present invention relates to a benzamide derivative of general formula I, a drug composition containing same and a use thereof as a drug, wherein the definitions of R 1 , Z and Q are as described in the description.

Claim (Index 9):
The compound of formula I, or the tautomer, the optical isomer and the pharmaceutically acceptable salt thereof according to  claim 1 , characterized in that:\n R 1  is: R 2  and R 3  are independently selected from the group consisting of H, C 1-6 alkyl, (CH 2 ) 0-3 -3\u02dc7-membered cycloalkyl and heterocycloalkyl containing 1 or 2 heteroatoms, and the R 2  and R 3  are not hydrogen at the same time; wherein the C 1-4 alkyl may be substituted by one or more substituents selected from the group consisting of halogen, hydroxyl, amino, cyano, C 1-6 alkoxy, (C 0-6  alkyl) (C 0-6  alkyl) amino, (C 0-6  alkyl) thio, (C 1-6  alkyl)carbonyl and (C 1-6  alkyl) sulfonyl; the 3\u02dc7-membered cycloalkyl or heterocycloalkyl is substituted by one R m , wherein the R m  is selected from the group consisting of hydrogen, C 1-6 alkyl, hydroxyl, halogen and amino, the heteroatom of the heterocycloalkyl is selected from O, N, and S; or R 2  and R 3 , together with the atoms attached thereto, form a 5, 6 or 7-membered ring, wherein, the 5-, 6- or 7-membered ring is substituted by one R n , wherein the R n  is selected from hydrogen, C 1-6 alkyl, hydroxyl, halogen and amino; the 5, 6 or 7-membered ring, in addition to the N atom attaching to R 2  and R 3 , further contain 0, 1 or 2 heteroatoms selected from O, N, and S.

Metadata:
- Claim Count in Document: 5.0
- Percentile: 90.0
- Lexical Diversity: 1.30303
- Patent Class: 544.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['10522955', '10581305', '12713448', '12875218', '12936784']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8425398306237307
- 35 USC 102 Novelty (BERT): 0.5289387370691947
- Combined Prediction Score: 0.8111797212682771
- Mean Citation Score: 363.297944
- Max Citation Score: 374.7806
- Similarity Product: 294.04958226765393

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test