PATENT CLAIM ANALYSIS

Application Number: 15975128
Application Type: Utility
Filing Date: 2018-05
Publication Date: 2018-09
Patent Classification: ["514", "255000"]

Abstract:
The present invention provides a pyrrolidine compound of General Formula (1) or a salt thereof, wherein R 101  and R 102  are each independently a phenyl group or a pyridyl group, the phenyl group or the pyridyl group may have one or more substituents selected from halogen atoms and lower alkyl groups optionally substituted with one or more halogen atoms, etc. The pyrrolidine compound or a salt thereof of the present invention is usable to produce a pharmaceutical preparation having a wider therapeutic spectrum and being capable of exhibiting sufficient therapeutic effects after short-term administration.

Claim (Index 6):
A pharmaceutical composition selected from the group consisting of:\n (3-chloro-4-fluorophenyl)-3-thienyl-(S)-pyrrolidin-3-ylamine, (4-chlorophenyl)phenyl-(S)-pyrrolidin-3-ylamine, (4-fluorophenyl)phenyl-(S)-pyrrolidin-3-ylamine, (3,4-difluorophenyl)phenyl-(S)-pyrrolidin-3-ylamine, bis-(4-fluorophenyl)-(S)-pyrrolidin-3-ylamine, (3,4-difluorophenyl)-(4-fluorophenyl)-(S)-pyrrolidin-3-ylamine, (3-chloro-4-fluorophenyl)-(S)-pyrrolidin-3-yl-p-tolylamine, 4-[(S)-(4-fluoro-3-methylphenyl)pyrrolidin-3-ylamino]-benzonitrile, bis-(3-fluorophenyl)-(S)-pyrrolidin-3-ylamine, (3-chloro-4-fluorophenyl)-(S)-pyrrolidin-3-ylthiazol-2-ylamine, (4-fluorophenyl)-(S)-pyrrolidin-3-ylthiazol-2-ylamine, (3,4-dichlorophenyl)-(S)-pyrrolidin-3-ylthiazol-2-ylamine, (3,4-dichlorophenyl)pyrimidin-5-yl-(S)-pyrrolidin-3-ylamine, (3-chloro-4-fluorophenyl)pyrazin-2-yl-(S)-pyrrolidin-3-ylamine, (3-chloro-4-fluorophenyl)-(5-chloropyridin-2-yl)-(S)-pyrrolidin-3-ylamine, (3-chloro-4-fluorophenyl)pyridin-2-yl-(S)-pyrrolidin-3-ylamine, (3-chloro-4-fluorophenyl)pyridin-3-yl-(S)-pyrrolidin-3-ylamine, (3-chloro-4-fluorophenyl)-(6-fluoropyridin-3-yl)-(S)-pyrrolidin-3-ylamine, (3,4-dichlorophenyl)pyridin-3-yl-(S)-pyrrolidin-3-ylamine, (3-chloro-4-fluorophenyl)-(S)-pyrrolidin-3-ylthiophen-3-ylamine, (3-chloro-4-fluorophenyl)-(5-fluoropyridin-3-yl)-(S)-pyrrolidin-3-ylamine, (4-fluoro-3-methylphenyl)-(5-fluoropyridin-3-yl)-(S)-pyrrolidin-3-ylamine, (3-chloro-4-fluorophenyl)-(1-methyl-1H-indazol-5-yl)-(S)-pyrrolidin-3-ylamine benzo[b]thiophen-6-yl-(S)-pyrrolidin-3-ylthiophen-3-ylamine, and benzo[b]thiophen-5-yl-(S)-pyrrolidin-3-ylthiophen-3-ylamine, and the salts thereof, as an active ingredient, and pharmaceutically acceptable carrier or excipient.

Metadata:
- Claim Count in Document: 13.0
- Percentile: 93.0
- Lexical Diversity: 1.59375
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15435084', '14300619', '13792971', '13298336', '11914183']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8456979239537821
- 35 USC 102 Novelty (BERT): 0.5866475319335432
- Combined Prediction Score: 0.8197928847517582
- Mean Citation Score: 493.381876
- Max Citation Score: 502.38043
- Similarity Product: 423.7621239412362

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test