PATENT CLAIM ANALYSIS

Application Number: 15910083
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2018-09
Patent Classification: ["544", "106000"]

Abstract:
Compounds of formula (I) or salts thereof are disclosed. Also disclosed are pharmaceutical compositions comprising a compound of formula I, processes for preparing compounds of formula I, intermediates useful for preparing compounds of formula I and therapeutic methods for treating a Retroviridae viral infection including an infection caused by the HIV virus.

Claim (Index 55):
A process for preparing a compound of formula I: or a pharmaceutically acceptable salt thereof, the process comprising:\n reacting a compound of formula (4) \n or a salt thereof, with a compound of formula (5) or a salt thereof, wherein R 1  is an amine protecting group and X 1  is a halogen, with a palladium catalyst and a weak base to produce a compound of formula (6) or a salt thereof;\n treating the compound of formula (6), or a salt thereof, with a deprotecting agent to produce a compound of formula (7) \n or a salt thereof; and\n reacting the compound of formula (7), or a salt thereof, with a compound of formula (8) \n or a salt thereof, a peptide coupling agent, and a non-nucleophilic base, to produce the compound of formula (I).

Metadata:
- Claim Count in Document: 32.0
- Percentile: 90.0
- Lexical Diversity: 1.48718
- Patent Class: 544.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['14771779', '14836774', '14151758', '15680041', '15121643']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.809990163450461
- 35 USC 102 Novelty (BERT): 0.5739247307372226
- Combined Prediction Score: 0.7863836201791372
- Mean Citation Score: 451.968066
- Max Citation Score: 528.5361
- Similarity Product: 366.4511575051904

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test