PATENT CLAIM ANALYSIS

Application Number: 15923948
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2018-07
Patent Classification: ["544", "006000"]

Abstract:
The invention relates to 3-((hetero-)aryl)-8-amino-2-oxo-1,3 -diaza-spiro-[4.5]-decane derivatives, their preparation and their use in medicine, particularly in the treatment of pain.

Claim (Index 24):
The compound according to  claim 1 , which has a structure according to general formula (IX) or (X) wherein R 2  means \u2014H or \u2014CH 3 ; R 3  means -phenyl or -3-fluorophenyl; R C  means \u2014H or \u2014OH; R E  means \u2014H, \u2014CH 3 , \u2014F, \u2014CF 3 , -cyclopropyl, -aziridinyl, \u2014OH; \u2014O\u2014C 1 -C 4 -alkyl; \u2014OCF 3 ; \u2014O\u2014C 1 -C 4 -alkyl-CO 2 H; \u2014O\u2014C 1 -C 4 -alkyl-C(\u2550O)O\u2014C 1 -C 4 -alkyl; or \u2014O\u2014C 1 -C 4 -alkyl-CONH 2 ; R F  means \u2014CF 3 , -cyclopropyl, \u2014S(\u2550O) 2 CH 3 , \u2014NH 2 ; \u2014NHC 1 -C 4 -alkyl; \u2014N(C 1 -C 4 -alkyl) 2 ; \u2014NHC 1 -C 4 -alkyl-OH; \u2014NCH 3 C 1 -C 4 -alkyl-OH; \u2014NH\u2014C 1 -C 4 -alkyl-C(\u2550O)NH 2 ; \u2014NCH 3 \u2014C 1 -C 4 -alkyl-C(\u2550O)NH 2 ; \u2014NHC(\u2550O)\u2014C 1 -C 4 -alkyl; \u2014NCH 3 C(\u2550O)\u2014C 1 -C 4 -alkyl; -6-14-membered aryl, unsubstituted, mono- or polysubstituted; or -5-14-membered heteroaryl, unsubstituted, mono- or polysubstituted; U means \u2550CH\u2014 or \u2550N\u2014; and V means \u2550CH\u2014 or \u2550N\u2014; or a physiologically acceptable salt thereof.

Metadata:
- Claim Count in Document: 65.0
- Percentile: 90.0
- Lexical Diversity: 1.17241
- Patent Class: 544.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15125615', '12604691', '12699451', '15326138', '12700857']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8471407581446906
- 35 USC 102 Novelty (BERT): 0.5515324367776466
- Combined Prediction Score: 0.8175799260079862
- Mean Citation Score: 423.427142
- Max Citation Score: 437.00952
- Similarity Product: 335.8095820751524

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test