PATENT CLAIM ANALYSIS

Application Number: 16227132
Application Type: Utility
Filing Date: 2018-12
Publication Date: 2019-06
Patent Classification: ["544", "283000"]

Abstract:
The present invention relates to quinazolinones and related compounds which are inhibitors of PARP14 and are useful, for example, in the treatment of cancer and inflammatory diseases.

Claim (Index 33):
The compound of  claim 1 , or a pharmaceutically acceptable salt thereof, wherein each R W , R X , R Y , and R Z  is independently selected from H, halo, C 1-6  alkyl, C 1-6  haloalkyl, 5-10 membered heteroaryl, 4-10 membered heterocycloalkyl, C 6-10  aryl-C 1-4  alkyl, CN, OR a2 , C(O)NR c2 R d2 , NR c2 R d2 , NR c2 C(O)R b2 , NR c2 C(O)OR a2 , NR c2 C(O)NR c2 R d2 , C(\u2550NR e2 )R b2 , C(\u2550NR e2 )NR c2 R d2 , NR c2 C(\u2550NR e2 )NR c2 R d2 , NR c2  S(O)R b2 , NR c2 S(O) 2 R b2 , and NR c2 S(O) 2 NR c2 R d2 ; wherein said C 1-6  alkyl, C 1-6  haloalkyl, 5-10 membered heteroaryl, 4-10 membered heterocycloalkyl, and C 6-10  aryl-C 1-4  alkyl of R W , R X , R Y , and R Z  are each optionally substituted with 1, 2, 3, 4, or 5 substituents independently selected from Cy 2 , Cy 2 -C 1-4  alkyl, halo, C 1-6  alkyl, C 2-6  alkenyl, C 2-6  alkynyl, C 1-6  haloalkyl, CN, NO 2 , OR a2 , SR a2 , C(O)R b2 , C(O)NR c2 R d2 , C(O)OR a2 , OC(O)R b2 , OC(O)NR c2 R d2 , C(\u2550NR e2 )NR c2 R d2 , NR c2 C(\u2550NR e2 )NR c2 R d2 , NR c2 R d2 , NR c2 C(O)R b2 , NR c2 C(O)OR a2 , NR c2 C(O)NR c2 R d2 , NR c2 S(O)R b2 , NR c2 S(O) 2 R b2 , NR c2 S(O) 2 NR c2 R d2 , S(O)R b2 , S(O)NR c2 R d2 , S(O) 2 R b2 , and S(O) 2 NR c2 R d2 .

Metadata:
- Claim Count in Document: 87.0
- Percentile: 98.0
- Lexical Diversity: 1.2
- Patent Class: 544.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15166380', '12270135', '14465910', '16308739', '15521202']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.816822439770544
- 35 USC 102 Novelty (BERT): 0.5170419882001346
- Combined Prediction Score: 0.7868443946135031
- Mean Citation Score: 326.669524
- Max Citation Score: 338.04504
- Similarity Product: 300.7667100455475

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test