PATENT CLAIM ANALYSIS

Application Number: 16307193
Application Type: Utility
Filing Date: 2018-12
Publication Date: 2019-08
Patent Classification: ["514", "230500"]

Abstract:
The present invention relates to novel antibacterial compounds, pharmaceutical compositions containing them and their use as antimicrobials.

Claim (Index 1):
A compound of formula (1):\n A-L 1 -Y-L 2 -R\u2014B\u2003\u2003(1) wherein\n A is a cyclic group having the formula (II): \n wherein G 3  is CH or N when the dashed line represents a double bond, or CH 2 , NH or O when the dashed line represents a single bond; C 1  represents the atoms necessary to form an aliphatic or aromatic six-membered cycle optionally comprising one or more heteroatom selected from nitrogen atom and oxygen atom, said cycle being optionally substituted by one or more substituent selected from the group consisting of halogen atom, (C 1-3 )alkyl group, cyano group, oxo group (\u2550O), and (C 1-3 )alkoxy group; L 1  is \u03c3 bond, or (C 1-3 )alkylenyl group, optionally substituted with hydroxy group; Y is a ring selected from the group consisting of piperidinyl, piperazinyl, pyrrolidinyl, 1-3 cyclobutyl, 1-3 cyclopentyl, 1-2 cyclopropyl, azetidinyl, azabicyclo-octyl, morpholinyl and cyclohexyl ring, said ring being optionally substituted by one or more substituent selected from the group consisting of hydroxy group, (C 1-3 )alkylenyl-OH group, (C 1-3 )alkylenyl-O\u2014(C 1-3 )alkyl group, (C 1-3 )alkylenyl-CONR\u2032R\u2033 group, and CONR\u2032R\u2033 group, wherein R\u2032 and R\u2033 are hydrogen atom or (C 1-3 )alkyl; L 2  is \u03c3 bond, \u2014(C 1-3 )alkylenyl- group, NR\u2032\u2033 group, NR\u2032\u2033\u2014(C 1-3 )alkylenyl group, (C 1-3 )alkylenyl-NR\u2032\u2033 group, NR\u2032\u2033\u2014(C 1-3 )alkylenyl-NR\u2032\u2033 group, or (C 1-3 )alkylenyl-NR\u2032\u2033\u2014(C 1-3 )alkylenyl group, said group being optionally substituted with a hydroxy group, wherein R\u2032\u2033 is hydrogen, (C 1-3 )alkyl, (C 1-3 )alkylenyl-OH, (C 1-3 )alkylenyl-O\u2014(C 1-3 )alkyl, or (C 1-3 )alkylenyl-CONR\u2032R\u2033, wherein R\u2032 and R\u2033 are hydrogen atom or (C 1-3 )alkyl; R is \u03c3 bond or heterocyclic ring, aliphatic or aromatic, having 5 members containing one or more nitrogen atoms, optionally substituted with CH 2 OH, CH 2 CN, CN or CONR\u2032R\u2033, wherein R\u2032 and R\u2033 are hydrogen atom or (C 1-3 )alkyl; and B is cyclic group having the following formula (VI): wherein G 6  is CH or N; and R 2  is hydrogen atom or halogen atom; or an addition salt with a pharmaceutically acceptable organic or inorganic acid or base, an enantiomer, an oxide thereof, or a quaternary ammonium salt thereof.

Metadata:
- Claim Count in Document: 14.0
- Percentile: 98.0
- Lexical Diversity: 1.0
- Patent Class: 514.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['16307410', '15533594', '15534874', '10518653', '15103215']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.769482843521308
- 35 USC 102 Novelty (BERT): 0.573402432484414
- Combined Prediction Score: 0.7498748024176187
- Mean Citation Score: 379.954476
- Max Citation Score: 479.58896
- Similarity Product: 362.6274744298172

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test