PATENT CLAIM ANALYSIS

Application Number: 15744510
Application Type: Utility
Filing Date: 2018-01
Publication Date: 2018-07
Patent Classification: ["514", "222800"]

Abstract:
The invention provides a compound which is a diazine of formula (I) or a tautomer thereof, or a pharmaceutically acceptable salt thereof, for use as an antifungal agent: (I) wherein X, N′, C′, A and E are as defined herein. The invention also provides a compound of Formula (I) as defined herein.

Claim (Index 12):
A compound for use according to  claim 1  wherein the compound is selected from:\n 5-[4-(4-ethylphenoxy)butyl]-6\u02dc{H}-1,3,4-thiadiazin-2-amine; 5-[5-(2-pyridyloxy)pentyl]-6\u02dc{H}-1,3,4-thiadiazin-2-amine; 5-[2-(2-phenoxyethoxy)ethyl]-6\u02dc{H}-1,3,4-thiadiazin-2-amine; 5-[4-[(3-bromophenyl)methoxy]butyl]-6\u02dc{H}-1,3,4-thiadiazin-2-amine; 5-[4-[(2,4-difluorophenyl)methoxy]butyl]-6\u02dc{H}-1,3,4-thiadiazin-2-amine; 5-(4-benzyloxybutyl)-6\u02dc{H}-1,3,4-thiadiazin-2-amine; 5-(5-benzyloxypentyl)-6\u02dc{H}-1,3,4-thiadiazin-2-amine; 5-(5-methoxypentyl)-4-methyl-3\u02dc{H}-1,3,4-thiadiazin-2-imine; 5-[5-(4-fluorophenoxy)pentyl]-6\u02dc{H}-1,3,4-thiadiazin-2-amine; 5-(2-hexoxyethyl)-6\u02dc{H}-1,3,4-thiadiazin-2-amine; 5-(5-methoxypentyl)-6\u02dc{H}-1,3,4-thiadiazin-2-amine; ethyl 4-(2-amino-4\u02dc{H}-1,3,4-thiadiazin-5-yl)benzoate; 5-(5-phenoxypentyl)-6\u02dc{H}-1,3,4-thiadiazin-2-amine and 5-(2-butoxyethyl)-6\u02dc{H}-1,3,4-thiadiazin-2-amine, \n and tautomers thereof and salts thereof

Metadata:
- Claim Count in Document: 5.0
- Percentile: 86.0
- Lexical Diversity: 1.65
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['12989410', '14625532', '12601284', '11914516', '12515354']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7416153066415038
- 35 USC 102 Novelty (BERT): 0.5173280593157539
- Combined Prediction Score: 0.7191865819089288
- Mean Citation Score: 288.72395399999994
- Max Citation Score: 300.37643
- Similarity Product: 226.2690742091644

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test