PATENT CLAIM ANALYSIS

Application Number: 15758466
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2019-01
Patent Classification: ["560", "024000"]

Abstract:
Disclosed herein are pharmaceutical compositions comprising fencamfamine or fencamfamine related prodrug derivatives for targeted therapeutic applications and methods of synthesizing the compositions.

Claim (Index 1):
A prodrug composition comprising at least one conjugate of N-ethyl-3-phenylbicyclo[2.2.1]heptan-2-amine or any of its stereoisomers wherein the conjugate is of the following formula (I): wherein Y is selected from the group consisting of-C(O)X and (A) n ; wherein: X is selected from the group consisting of \u2014OR 1 , \u2014NHR 1 , \u2014NR 1 R 5 \u2014O(CR 2 R 6 )OR 3 , \u2014O(CR 2 R 6 )SR 3 , O(CR 2 R 6 )NR 3  and R 4 ; wherein R 1  is independently selected from optionally substituted C 1-16  alkyl, optionally substituted aryl, and optionally substituted cycloalkyl; wherein R 2 , R 5 , and R 6  are independently selected from hydrogen, optionally substituted C 1-6  alkyl; wherein R 3  is independently selected from optionally substituted C 1-26  alkanoyl; optionally substituted C 1-26  alkenoyl, optionally substituted C 1-26  alkynoyl; optionally substituted cycloalkanoyl; wherein R 4  is independently selected from optionally substituted C 1-26  alkyl; optionally substituted C 1-26  alkenyl, optionally substituted C 1-26  alkynyl; optionally substituted cycloalkyl; wherein (A) n  is a peptide unit formed with amino acid units wherein n is independently 1, 2, 3, or 4.

Metadata:
- Claim Count in Document: 28.0
- Percentile: 90.0
- Lexical Diversity: 1.09524
- Patent Class: 560.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['15320353', '12915354', '11269913', '11404267', '10850231']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.702620338257361
- 35 USC 102 Novelty (BERT): 0.521220241218605
- Combined Prediction Score: 0.6844803285534855
- Mean Citation Score: 229.71749400000004
- Max Citation Score: 235.5983
- Similarity Product: 174.302792614609

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test