PATENT CLAIM ANALYSIS

Application Number: 15751316
Application Type: Utility
Filing Date: 2018-02
Publication Date: 2018-08
Patent Classification: ["564", "134000"]

Abstract:
The present invention relates to processes, process steps and intermediates useful in the asymmetric bisamidation of malonic ester derivatives wherein the new processes, process steps and intermediates are, for example, useful in the preparation of asymmetric malonic acid bisanilides such as cabozantinib.

Claim (Index 5):
The process of  claim 1 , wherein the compound of formula (I) is the compound H 2 N\u2014X 1  is 4-fluoroaniline and the M a  salt of formula (II) is

Metadata:
- Claim Count in Document: 11.0
- Percentile: 88.0
- Lexical Diversity: 1.46875
- Patent Class: 564.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['14494631', '10994983', '12067612', '15750339', '15453953']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7340368224959095
- 35 USC 102 Novelty (BERT): 0.5175722388479397
- Combined Prediction Score: 0.7123903641311126
- Mean Citation Score: 227.855124
- Max Citation Score: 238.50386
- Similarity Product: 173.49022514502047

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 0
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test