PATENT CLAIM ANALYSIS

Application Number: 15766183
Application Type: Utility
Filing Date: 2018-04
Publication Date: 2018-10
Patent Classification: ["514", "192000"]

Abstract:
Compounds of Formula (I) or a stereoisomer or a pharmaceutically acceptable salt thereof, their preparation, and use in treating a bacterial infection are disclosed.

Claim (Index 1):
A compound of Formula (I): wherein: A is a four to six membered nitrogen containing ring optionally substituted with one or more substituents selected from C 1 -C 6  alkyl, oxo, NR 2 R 3 , aryl, heteroaryl, cycloalkyl or heterocycloalkyl; B is C\u2550O or CH\u2014Z; X is O or CONH; Z is H, C 1 -C 6  alkyl, OR 2  or NR 2 R 3 ; R 1  is selected from:\n (a) hydrogen, \n (b) C 1 -C 6  alkyl optionally substituted with one or more substituents independently selected from OR 2 , NR 2 R 3 , SR 2 , halogen, CN, COOR 2 , CONR 2 R 3 , SR 2 , CH 2 OR 2 , CH 2 NR 2 R 3 , OCOR 2 , aryl, heteroaryl, cycloalkyl or heterocycloalkyl, \n (c) CN, \n (d) CONR 2 R 3 , \n (e) COOR 2 , \n (f) NR 2 R 3 , \n (g) NHCOOR 2 , \n (h) aryl, \n (i) heteroaryl, \n (j) cycloalkyl, or \n (k) heterocycloalkyl; \n R 2  and R 3  are each independently selected from:\n (a) hydrogen, \n (b) C 1 -C 6  alkyl optionally substituted with one or more substituents selected from halogen, NR 4 R 5 , CONR 4 R 5 , CN, OR 4  or COOR 4 ; \n (c) aryl, \n (d) heteroaryl, \n (e) cycloalkyl, or \n (f) heterocycloalkyl; \n R 4  and R 5  are each independently selected from:\n (a) hydrogen or \n (b) C 1 -C 6  alkyl optionally substituted with one or more substituents selected from OH, halogen, NH 2 , CONH 2 , CN, OCH 3 , or COOH; \n n is 0, 1, 2, 3 or 4; or a stereoisomer or a pharmaceutically acceptable salt thereof.

Metadata:
- Claim Count in Document: 44.0
- Percentile: 91.0
- Lexical Diversity: 1.16
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15781121', '15171237', '15547487', '14113980', '14808804']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8047825296175504
- 35 USC 102 Novelty (BERT): 0.6257245195168899
- Combined Prediction Score: 0.7868767286074844
- Mean Citation Score: 462.09563800000006
- Max Citation Score: 588.6308
- Similarity Product: 510.9396921136856

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test