PATENT CLAIM ANALYSIS

Application Number: 15762670
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2018-10
Patent Classification: ["514", "218000"]

Abstract:
A series of substituted pyrazolo[1,5-a]pyrimidine and pyrazolo[1,5-a][1,3,5]-triazine derivatives of formula (I), as defined herein, being selective inhibitors of phosphatidylinositol-4-kinase IIIβ (PI4KIIIβ) activity, are beneficial in the treatment and/or prevention of various human ailments, including inflammatory, autoimmune and oncological disorders; viral diseases and malaria; and organ and cell transplant rejection.

Claim (Index 13):
The compound as claimed in  claim 2  wherein M represents the residue of an azetidin-1-yl, pyrrolidin-1-yl, piperidin-1-yl, morpholin-4-yl, piperazin-1-yl, azepan-1-yl or [1,4]diazepan-1-yl ring, or M represents the residue of a 1,2,3,3a,4,5,6,6a-octahydrocyclopenta[c]pyrrol-2-yl, 2,3,4,4a,5,6,7,7a-octahydropyrrolo-[3,4-b][1,4]oxazin-6-yl, 1,2,3,4,6,7,8,8a-octahydropyrrolo[1,2-a]-pyrazin-2-yl, 3-aza-bicyclo[3.1.0]hexan-3-yl, 2-oxa-5-azabicyclo[2.2.1]heptan-5-yl, 8-azabicyclo[3.2.1]-octan-8-yl or 2-oxa-6-azaspiro[3.3]heptan-6-yl ring system, any of which may be optionally substituted by one, two or three substituents independently selected from halogen, C 1-6  alkyl, benzyl, heteroaryl, (C 1-6 )alkylheteroaryl, C 1-6  alkoxy, C 1-6  alkoxy-(C 1-6 )alkyl, C 1-6  alkylsulfonyl, oxo, C 2-6  alkylcarbonyl, C 2-6  alkoxycarbonyl, di(C 1-6 )alkyl-amino, di(C 1-6 )alkylamino(C 1-6 )alkyl, morpholinyl, dioxothiomorpholinyl, N\u2014[(C 1-6 )-alkyl]-N\u2014[(C 2-6 )alkylcarbonyl]amino, C 2-6  alkoxycarbonylamino, C 3-6  alkenyloxy-carbonylamino, aminocarbonyl, di(C 1-6 )alkylaminocarbonyl, (C 1-6  alkoxy)(C 1-6  alkyl)-phenylaminocarbonyl, morpholinylcarbonyl and pyrrolidinylcarbonyl(C 1-6 )alkyl.

Metadata:
- Claim Count in Document: 40.0
- Percentile: 90.0
- Lexical Diversity: 1.38462
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15318422', '15318507', '16060486', '14357340', '13508956']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7924848196956081
- 35 USC 102 Novelty (BERT): 0.5497330343324666
- Combined Prediction Score: 0.768209641159294
- Mean Citation Score: 379.267696
- Max Citation Score: 396.2881
- Similarity Product: 297.4921527063847

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test