PATENT CLAIM ANALYSIS

Application Number: 16037396
Application Type: Utility
Filing Date: 2018-07
Publication Date: 2018-11
Patent Classification: ["514", "063000"]

Abstract:
The present invention relates to a new compound of formula (I) wherein the variables have the meaning as indicated in the claims; or an enantiomer or salt thereof. The compounds of formula (I) are useful in the control of parasites, in particular endoparasites, in and on vertebrates.

Claim (Index 1):
A compound of formula or a salt or an enantiomer thereof, wherein n is 0 or 1; A is C 1 -C 6 -alkyl; C 1 -C 6 -haloalkyl; C 3 -C 6 -cycloalkyl; C 3 -C 6 -halocycloalkyl; 5- or 6-membered heterocycloalkyl having from 1 to 3 same or different heteroatoms selected from the group consisting of B, N, O and S, which is further unsubstituted or substituted by halogen, C 1 -C 4 -alkyl or C 1 -C 4 -alkoxy; or is cinnamyl, which is unsubstituted or substituted in the phenyl moiety by halogen, C 1 -C 4 -alkyl or C 1 -C 4 -alkoxy; or is a heteroaromatic radical, which is further unsubstituted or substituted by halogen, cyano, C 1 -C 4 -alkyl, C 1 -C 4 -haloalkyl, C 1 -C 4 -alkoxy, C 1 -C 4 -haloalkoxy, C 2 -C 4 -alkanoyl, 5- or 6-membered heterocycloalkyl-C 1 -C 2 -alkyl or unsubstituted or halogen-, C 1 -C 4 -alkyl- or C 1 -C 4 -alkoxy-substituted phenyl; or is a hetero-bicyclic ring radical comprising a total of 8 to 10 ring members, from which 1 to 5 members are same or different heteroatoms selected from the group consisting of B, N, O and S, and from which 0 to 2 members are a group \u2014C(O)\u2014, which bicyclic ring radical is further unsubstituted or substituted by halogen, cyano, hydroxyl, C 1 -C 4 -alkyl or C 1 -C 4 -haloalkyl; R 2  is H or \u2014S(O 2 )-T; T is C 1 -C 6 -alkyl which is unsubstituted or substituted by halogen, trimethylsilyl, C 3 -C 6 -cycloalkyl, carboxyl or C 1 -C 4 -alkoxycarbonyl; C 3 -C 6 -cycloalkyl; C 6 -C 12 -bicarbocyclyl; phenyl which is unsubstituted or substituted by halogen, cyano, nitro, C 1 -C 4 -alkyl, C 1 -C 4 -haloalkyl or C 1 -C 4 -alkoxy; a 5- or 6 membered heteroaromatic radical, which is further unsubstituted or substituted by halogen, cyano, nitro, C 1 -C 4 -alkyl, C 1 -C 4 -haloalkyl or C 1 -C 4 -alkoxy; 5- or 6-membered heterocycloalkyl having from 1 to 3 same or different heteroatoms selected from the group consisting of N, O, S and S(O 2 ), which is further unsubstituted or substituted by C 1 -C 4 -alkyl, C 1 -C 2 -alkoxycarbonyl or benzyloxycarbonyl ; a group amino; or N-mono- or N,N-di-C 1 -C 4 -alkylamino;\n R 3  is C 1 -C 4 -alkyl, unsubstituted or halogen-, C 1 -C 4 -alkyl- or C 1 -C 4 -haloalkyl-substituted phenyl, unsubstituted or halogen-, C 1 -C 4 -alkyl- or C 1 -C 4 -haloalkyl-substituted pyridyl, C 1 -C 4 -alkoxycarbonyl-methyl or morpholin-4-yl-carbonylmethyl; \n R 0  is H or hydroxy; and \n Y is \n (i) phenyl or a phenylamino, which is substituted by one or more same or different radicals selected from the group consisting of halogen; C 1 -C 6 -alkyl; C 1 -C 6 -haloalkyl; C 3 -C 6 -cycloalkyl; C 3 -C 6 -halocycloalkyl; hydroxyl; C 1 -C 6 -alkoxy; C 1 -C 6 -haloalkoxy; C 1 -C 6 -alkylthio; C 1 -C 6 -haloalkylthio; C 1 -C 6 -alkyl-sulfinyl; C 1 -C 6 -haloalkylsulfinyl; C 1 -C 6 -alkylsulfonyl; C 1 -C 6 -haloalkylsulfonyl; SF 5 ; amino; N-mono- or N,N-di-C 1 -C 6 -alkylamino; tri-C 1 -C 4 -alkylsilyl; C 1 -C 6 -alkoxycarbonyl; aminocarbonyl; N-mono- or N,N-di-C 1 -C 6 -alkylaminocarbonyl; aminosulfonyl; N-mono- or N,N-di-C 1 -C 6 -alkylaminosulfonyl; N\u2014C 1 -C 6 -alkylsulfonylamino; C 1 -C 6 -alkoxycarbonylamino; N\u2014C 1 -C 4 -alkyl-N\u2014C 1 -C 6 -alkoxycarbonylamino; cyano; nitro; and halogen-, C 1 -C 4 -alkyl-, C 1 -C 4 -haloalkyl-, C 1 -C 4 -alkoxy-, C 1 -C 4 -haloalkoxy-, amino-, cyano- or nitro-substituted C 3 -C 6 -heterocyclyl; or is \n (ii) 5- or 6 membered heteroaryl or heteroarylamino, which is each further unsubstituted or substituted by halogen, cyano, nitro, C 1 -C 4 -alkyl, C 1 -C 4 -haloalkyl, C 1 -C 4 -alkoxy, C 1 -C 4 -alkoxycarbonyl, C 2 -C 4 -alkanoyl, or phenyl or phenylsulfonyl which is each unsubstituted or substituted by halogen, cyano, nitro, methyl or methoxy; or is \n (iii) benzoyl or 5- or 6 membered heteroarylcarbonyl, which is each further unsubstituted or substituted by halogen, cyano, nitro, C 1 -C 4 -alkyl, C 1 -C 4 -haloalkyl, C 1 -C 4 -alkoxy, C 1 -C 4 -alkoxycarbonyl, C 2 -C 4 -alkanoyl or phenyl; or is \n (iv) a C 6 -C 12 -bicarbocyclic radical; or is a \n (v) a hetero-bicyclic ring radical comprising a total of 8 to 10 ring members, from which 1 to 5 members are same or different heteroatoms selected from the group consisting of B, N, O and S, and from which 0 to 2 members are a group \u2014C(O)\u2014, which bicyclic ring radical is further unsubstituted or substituted by halogen, cyano, hydroxyl, C 1 -C 4 -alkoxy, C 1 -C 4 -alkyl or C 1 -C 4 -haloalkyl; or is \n (vi) a radical H 2 C\u2014C(O)\u2014NH\u2014R 4 , wherein R 4  is C 1 -C 4 -haloalkyl, C 2 -C 3 -alkynyl or cyano-C 1 -C 4 -alkyl; or \n R 0  and Y together with the N-atom to which they are attached, form a piperidinyl or piperazinyl radical which is substituted by C 1 -C 4 -alkyl, C 1 -C 4 -alkoxy, unsubstituted or halogen-, C 1 -C 4 -alkyl-, C 1 -C 4 -haloalkyl-, amino- and/or C 1 -C 4 -alkoxy-substituted phenyl or benzoylamino, or unsubstituted or C 1 -C 4 -alkyl-, C 1 -C 4 -haloalkyl-, C 3 -C 6 -cycloalkyl- or halogen-substituted pyridyl or pyrimidinyl; subject to the proviso that \n T is C 1 -C 6 -alkyl which is unsubstituted or substituted as mentioned above if A is C 1 -C 6 -alkyl or C 1 -C 6 -haloalkyl.

Metadata:
- Claim Count in Document: 17.0
- Percentile: 95.0
- Lexical Diversity: 1.4
- Patent Class: 514.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15502512', '14649268', '13133678', '13740756', '14148205']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7812723566826154
- 35 USC 102 Novelty (BERT): 0.5655641407871628
- Combined Prediction Score: 0.7597015350930701
- Mean Citation Score: 414.029414
- Max Citation Score: 444.4163
- Similarity Product: 364.2799895569086

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test