PATENT CLAIM ANALYSIS

Application Number: 15861399
Application Type: Utility
Filing Date: 2018-01
Publication Date: 2018-05
Patent Classification: ["514", "233200"]

Abstract:
The present invention relates to novel fused Imidazobenzothiazole derivatives, their pharmaceutically acceptable salts, and their isomers, steroisomers, atropisomers, conformers, tautomers, polymorphs, hydrates, solvates and N-oxide. The present invention also encompasses pharmaceutically acceptable compositions of said compounds and process for preparing novel compounds. The invention further relates to the use of the above-mentioned compounds for the preparation of medicament for use as pharmaceuticals.

Claim (Index 2):
The method according to  claim 1 , wherein in the compound of formula (I):\n X is O, NH or S(O); R 1  and R 2  are independently selected from hydrogen, A, CHO, CH 2 OH, CH 2 R 3 , CH 2 -halogen, N(R 5 )CO 2 R 4 , C(O)NR 5 R 6 , CO 2 R 7  and C(O)-A; R is independently selected from CN, CHO, C(O)-A, NR 5 R 6 , N(R 5 )C(O)-A, N(R 5 )C(O)O-A, N(R 5 )C(O)N(R 5 )-A, C(O)N(R 5 )-A, (C 1 -C 6 )alkyl-OR 7 , (C 1 -C 6 )alkyl-halogen, (C 1 -C 6 )alkyl-N 3 , (C 1 -C 6 )alkyl-NR 5 R 6 , (C 1 -C 6 )alkyl-N(R 5 )C(O)-A, (C 1 -C 6 )alkyl-N(R 5 )C(O)O-A, (C 1 -C 6 )alkyl-N(R 5 )C(O)N(R 5 )-A and (C 1 -C 6 )alkyl-OC(O)N(R 5 )-A; A is independently selected from (C 1 -C 6 )alkyl, (C 3 -C 10 )carbocycle, aryl, heteroaryl and heterocyclic, the said (C 1 -C 6 )alkyl, aryl or heteroaryl may be further substituted with 1-3 substituents independently selected from halogen, (C 1 -C 6 )alkyl, (C 3 -C 10 )carbocycle, aryl, heterocyclic, hydroxyl, CF 3 , O(C 1 -C 6 )alkyl, N(R 5 )S(O) m \u2014(C 1 -C 6 )alkyl and (C 1 -C 6 )alkyl-OH, each aryl may be further substituted with 1-3 substituents independently selected from halogen, (C 1 -C 6 )alkyl, hydroxyl, OSO 3 H, O(C 1 -C 6 )alkyl and R 3  is independently selected from O-A, NR 5 R 6 , S(O) n -A, S(O) n \u2014(C 1 -C 6 )alkyl-CO 2 (C 1 -C 6 )alkyl and S(O) n \u2014(C 1 -C 6 )alkyl-OH; R 4  is hydrogen or A; R 5  is hydrogen or (C 1 -C 6 )alkyl; R 6  is independently selected from hydrogen, (C 1 -C 6 )alkyl-OH, CH(CH 2 OH)-aryl, CH(CH 2 OH) 2 , (C 1 -C 6 )alkyl-aryl, (C 1 -C 6 )alkyl-heterocyclic and (C 1 -C 6 )alkyl-heteroaryl; or R 5  and R 6  together with the nitrogen to which they are attached may form a 3 to 8 membered monocyclic heterocycle ring, which ring contains an additional heteroatom selected from O, S and N and the said ring is substituted by R 9 ; the nitrogen of said ring may also form N-oxide; R 7  is hydrogen or A, which is (C 1 -C 6 )alkyl; R 8  is hydrogen or A, which is (C 1 -C 6 )alkyl; R 8  is hydrogen, hydroxyl or A, which is (C 1 -C 6 )alkyl; n is O; and m is 2.

Metadata:
- Claim Count in Document: 38.0
- Percentile: 86.0
- Lexical Diversity: 1.7619
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15128886', '15505902', '13639959', '15689075', '14424361']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7730387187634201
- 35 USC 102 Novelty (BERT): 0.6380129299462344
- Combined Prediction Score: 0.7595361398817015
- Mean Citation Score: 399.13778
- Max Citation Score: 583.3345
- Similarity Product: 556.3100179014207

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test