PATENT CLAIM ANALYSIS

Application Number: 16015925
Application Type: Utility
Filing Date: 2018-06
Publication Date: 2018-10
Patent Classification: ["546", "245000"]

Abstract:
Compounds and methods in the fields of chemistry and medicine are disclosed. Some of the disclosed embodiments include compounds, compositions and methods of using heterocycle amines. Some of the disclosed embodiments include heterocycle amines useful to treat inflammatory disorders.

Claim (Index 1):
A method of treating a disorder selected from the group consisting of an inflammatory disorder, a skin disorder, a respiratory disorder, diabetes, obesity, allergic disease, cancer, and sepsis, the method comprising administering to a subject in need thereof an effective amount of a compound of Formula (I): or a salt thereof, wherein:  is a single or double bond; W is selected from CH, CH\u2014CH, O, S, NR 6 , and CO; Y is N or CR 9 ; Z is N or C, and Z is N if W is CH and Y is CR 9 ; R 4  is selected from hydrogen, halogen, OR 6 , CN, NR 7 R 8 , CH 2 OR 6 , an optionally substituted aryl, an optionally substituted heteroaryl, an optionally substituted non-aromatic ring, an optionally substituted carbocycle, an optionally substituted C 1 -C 6  alkyl, an optionally substituted C 1 -C 6  haloalkyl, an optionally substituted C 1 -C 6  heteroalkyl, an optionally substituted C 1 -C 6  alkenyl, an optionally substituted C 1 -C 6  alkynyl, CO 2 R 6 , SO 3 R 6 , SO 2 R 6  and SO 2 NR 7 R 8 ; R 5  is selected from hydrogen, halogen, OR 6 , an optionally substituted C 1 -C 6  alkyl, an optionally substituted C 1 -C 6  haloalkyl, an optionally substituted C 1 -C 6  heteroalkyl, an optionally substituted C 1 -C 6  haloheteroalkyl, an optionally substituted C 1 -C 6  alkenyl, and an optionally substituted C 1 -C 6  alkynyl; or R 4  and R 5  are linked to form an optionally substituted non-aromatic ring; each R 6  is independently selected from an optionally substituted aryl, an optionally substituted heteroaryl, and an optionally substituted non-aromatic ring, each optionally fused with a substituted aryl or a substituted heteroaryl, hydrogen, an optionally substituted C 1 -C 10  alkyl, an optionally substituted C 1 -C 10  haloalkyl, and an optionally substituted C 1 -C 10  heteroalkyl; each R 7  and R 8  is independently selected from an optionally substituted aryl, an optionally substituted heteroaryl, an optionally substituted non-aromatic ring, each optionally fused with a substituted aryl or a substituted heteroaryl, hydrogen, an optionally substituted C 1 -C 10  alkyl, an optionally substituted C 1 -C 10  haloalkyl, an optionally substituted C 1 -C 10  alkenyl, an optionally substituted C 1 -C 10  alkynyl, and an optionally substituted C 1 -C 10  heteroalkyl, or R 7  and R 8  are linked to form an optionally substituted non-aromatic ring; R 9  is selected from hydrogen, halogen, OR 6 , CN, NR 7 R 8 , CH 2 OR 6 , an optionally substituted aryl, an optionally substituted heteroaryl, an optionally substituted non-aromatic ring, an optionally substituted C 1 -C 6  alkyl, an optionally substituted C 1 -C 6  haloalkyl, an optionally substituted C 1 -C 6  heteroalkyl, an optionally substituted C 1 -C 6  alkenyl, an optionally substituted C 1 -C 6  alkynyl, CO 2 R 6 , SO 3 R 6 , and SO 2 NR 7 R 8 ; A is an optionally substituted aryl or an optionally substituted heteroaryl group; and each optionally substituted group is either unsubstituted or substituted with one or more groups independently selected from alkyl, heteroalkyl, alkenyl, alkynyl, haloalkyl, heterohaloalkyl, aryl, arylalkyl, heteroaryl, non-aromatic ring, hydroxy, alkoxy, aryloxy, mercapto, alkylthio, arylthio, cyano, halo, carbonyl, thiocarbonyl, O-carbamyl, N-carbamyl, O-thiocarbamyl, N-thiocarbamyl, C-amido, N-amido, S-sulfonamido, N-sulfonamido, C-carboxy, O-carboxy, isocymato, thiocyanato, isothiocymato, nitro, silyl, trihalomethanesulfonyl, \u2550O, \u2550S, amino, and protected derivatives of amino groups.

Metadata:
- Claim Count in Document: 2.0
- Percentile: 94.0
- Lexical Diversity: 1.65385
- Patent Class: 546.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['12784916', '15006940', '15513125', '14137318', '15894025']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7282608424074477
- 35 USC 102 Novelty (BERT): 0.5395158088830564
- Combined Prediction Score: 0.7093863390550086
- Mean Citation Score: 378.900244
- Max Citation Score: 383.6451
- Similarity Product: 239.9206490963101

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test