PATENT CLAIM ANALYSIS

Application Number: 16315710
Application Type: Utility
Filing Date: 2019-01
Publication Date: 2019-05
Patent Classification: ["514", "235200"]

Abstract:
The present invention relates to a compound of the formula: where n, R and R are those defined herein. The present invention also relates to use of a compound of Formula 1 in treating a clinical condition associated with fibrotic disorder.

Claim (Index 15):
The compound of  claim 1 , wherein the compound is:\n N-(N,N-diethylaminosulfonyl)-2-(indolin-1-yl)ethane-1-amine N-(2-(indolin-1-yl)ethyl)pyrrolidine-1-sulfonamide 1,1-diethyl-3-(2-(indolin-1-yl)propyl)urea N-(N,N-dimethylaminosulfonyl)-2-(indolin-1-yl)propane-1-amine N-(2-(indolin-1-yl)propyl)pyrrolidine-1-sulfonamide N-(2-(indolin-1-yl)ethyl)-4-methylpiperazine-1-carboxamide N-(2-(indolin-1-yl)ethyl)morpholine-4-sulfonamide N-(2-(indolin-1-yl)ethyl)piperidine-1-sulfonamide N-(2-(indolin-1-yl)propyl)-4-methylpiperazine-1-carboxamide N-(2-(indolin-1-yl)propyl)pyrrolidine-1-carboxamide N-(2-indolin-1-yl)ethyl)pyrrolidine-1-carboxamide 1-(indolin-1-yl)-2-(4-(pyrimidin-2-yl)piperazin-1-yl)ethan-1-one 1-(indolin-1-yl)-2-(4-(piperidin-1-ylsulfonyl)piperazin-1-yl)ethan-1-one 4-(2-(indolin-1-yl)-2-oxoethyl)-N,N-dimethylpiperazine-1-sulfonamide 1-(indolin-1-yl)-3-(4-(piperidin-1-ylsulfonyl)piperazin-1-yl)propan-1-one N-(2-(indolin-1-yl)propyl)-2-(pyridin-4-yl)thiazole-4-carboxamide N-(2-(indolin-1-yl)propyl)-4-methoxybenzenesulfonamide N-(2-(5-(3-methoxyphenyl)indolin-1-yl)propyl)-N,N-diethyl-1-sulfonamide N-(2-(indolin-1-yl)propyl)-4-methylpiperazine-1-sulfonamide N-(2-(5-(3-methoxyphenyl)indolin-1-yl)propyl)-4-methylpiperazine-1-sulfonamide N-(N,N-diethylaminosulfonyl)-4-(indolin-1-yl)-phenyl-1-amine N-(2-(indolin-1-yl)propyl)-4-(trifluoromethyl)benzenesulfonamide N-(2-(indolin-1-yl)propyl)-4-(trifluoromethoxy)benzenesulfonamide N-(2-(indolin-1-yl)propyl)-2-(4-methoxyphenyl)thiazole-4-carboxamide N-(2-(indolin-1-yl)propyl)-2-phenylthiazole-4-carboxamide N-(2-(indolin-1-yl)propyl)-2-(4-(trifluoromethyl)phenyl)thiazole-4-carboxamide 1-(2-(4-((4-(trifluoromethoxy)phenyl)sulfonyl)piperazin-1-yl)ethyl)indoline N,N-diethyl-4-(2-(indolin-1-yl)ethyl)piperazine-1-sulfonamide 1-(2-(4-((4-fluorophenyl)sulfonyl)piperazin-1-yl)ethyl)indoline N,N-diethyl-4-(2-(indolin-1-yl)ethyl)piperazine-1-carboxamide 1-(2-(4-(2-fluorobenzyl)piperazin-1-yl)ethyl)indoline N-(2-(indolin-1-yl)propyl)-4-((5-(trifluoromethyl)pyridin-2-yl)oxy)benzenesulfonamide N-(2-(indolin-1-yl)propyl)-4-phenoxybenzenesulfonamide 4-cyano-N-(2-(indolin-1-yl)propyl)benzenesulfonamide N-(2-(indolin-1-yl)ethyl)-4-(trifluoromethyl)benzenesulfonamide N-(2-(indolin-1-yl)ethyl)-4-(trifluoromethoxy)benzenesulfonamide N-(2-(indolin-1-yl)ethyl)-4-phenoxybenzenesulfonamide N-(2-(indolin-1-yl)ethyl)-4-((5-(trifluoromethyl)pyridin-2-yl)oxy)benzenesulfonamide 3,4-difluoro-N-(2-(indolin-1-yl)ethyl)benzenesulfonamide 4-cyano-N-(2-(indolin-1-yl)ethyl)benzenesulfonamide N-(N,N-diethylaminosulfonyl)-2-(indolin-1-yl)-2-methylpropane-1-amine N-(2-(indolin-1-yl)-2-methylpropyl)-4-(trifluoromethyl)benzenesulfonamide N-(2-(indolin-1-yl)-2-methylpropyl)-4-phenoxybenzenesulfonamide 4-fluoro-N-(2-(indolin-1-yl)-2-methylpropyl)benzenesulfonamide 3,4-difluoro-N-(2-(indolin-1-yl)-2-methylpropyl)benzenesulfonamide N-(2-(indolin-1-yl)-2-methylpropyl)-4-((5-(trifluoromethyl)pyridin-2-yl)oxy)benzenesulfonamide N-(2-(indolin-1-yl)-2-methylpropyl)-4-(methoxy)benzenesulfonamide N-(2-(indolin-1-yl)-2-methylpropyl)-4-(trifluoromethoxy)benzenesulfonamide or a pharmaceutically acceptable salt thereof.

Metadata:
- Claim Count in Document: 47.0
- Percentile: 99.0
- Lexical Diversity: 1.36364
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15736450', '14000829', '15315461', '15738900', '10516681']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7250936677421556
- 35 USC 102 Novelty (BERT): 0.5138300351699878
- Combined Prediction Score: 0.7039673044849388
- Mean Citation Score: 234.662008
- Max Citation Score: 248.7203
- Similarity Product: 167.82471184145808

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test