PATENT CLAIM ANALYSIS

Application Number: 16250212
Application Type: Utility
Filing Date: 2019-01
Publication Date: 2019-05
Patent Classification: ["514", "303000"]

Abstract:
The purpose of the present invention is to provide novel compounds having ACC2 selective inhibitory activity. In addition, the present invention provides a pharmaceutical composition comprising the compound. A compound of Formula: or its pharmaceutically acceptable salt, wherein, R 1  is substituted or unsubstituted fused aromatic heterocyclyl represented by Formula: wherein,         ring B is 5-membered ring, ring C is 6-membered ring;           ring A is substituted or unsubstituted non-aromatic carbocycle or the like; -L 1 - is —O—(CR 6 R 7 )m- or the like; -L 2 - is —O—(CR 6 R 7 )n- or the like; each R 6  is independently hydrogen or the like; each R 7  is independently hydrogen or the like; each m is independently an integer of 0, 1, 2 or 3; each n is independently an integer of 1, 2 or 3; R 2  is substituted or unsubstituted alkyl; R 3  is hydrogen or substituted or unsubstituted alkyl; R 4  is substituted or unsubstituted alkylcarbonyl or the like.

Claim (Index 1):
A compound of Formula (I): or its pharmaceutically acceptable salt, wherein\n R 1  is substituted or unsubstituted fused aromatic heterocyclyl represented by Formula: \n wherein\n ring B is 5-membered ring, ring C is 6-membered ring; \n ring A is substituted or unsubstituted non-aromatic carbocycle; \n -L 1 - is \u2014O\u2014(CR 6 R 7 )m-, wherein the bond of left side is attached to R 1 , the bond of right side is attached to ring A; \n L 2 - is \u2014O\u2014(CR 6 R 7 )n-, \u2014O\u2014CR 6 \u2550CR 7 \u2014, \u2014CR 6 \u2550CR 7 \u2014 or \u2014(CR 6 R 7 )n-, wherein the bond of left side is attached to ring A, the bond of right side is attached to the group represented by Formula: \n each R 6  is independently hydrogen, halogen, cyano, substituted or unsubstituted alkyl, substituted or unsubstituted alkenyl or substituted or unsubstituted alkynyl; each R 7  is independently hydrogen, halogen, cyano, substituted or unsubstituted alkyl, substituted or unsubstituted alkenyl or substituted or unsubstituted alkynyl; R 6  and R 7  on the same carbon atom may be taken together with the carbon atom to form ring; each m is independently an integer of 0, 1, 2 or 3; each n is independently an integer of 1, 2 or 3; R 2  is substituted or unsubstituted alkyl; R 3  is hydrogen, or substituted or unsubstituted alkyl; R 4  is substituted or unsubstituted alkylcarbonyl, substituted or unsubstituted alkenylcarbonyl, substituted or unsubstituted alkynylcarbonyl, substituted or unsubstituted non-aromatic carbocyclylcarbonyl, substituted or unsubstituted aromatic carbocyclylcarbonyl, substituted or unsubstituted non-aromatic heterocyclylcarbonyl, substituted or unsubstituted aromatic heterocyclylcarbonyl, substituted or unsubstituted alkyloxycarbonyl, substituted or unsubstituted alkenyloxycarbonyl, substituted or unsubstituted alkynyloxycarbonyl, substituted or unsubstituted non-aromatic carbocyclyloxycarbonyl, substituted or unsubstituted aromatic carbocyclyloxycarbonyl, substituted or unsubstituted non-aromatic heterocyclyloxycarbonyl, substituted or unsubstituted aromatic heterocyclyloxycarbonyl, substituted or unsubstituted carbamoyl, substituted or unsubstituted alkylsulfonyl, substituted or unsubstituted alkenylsulfonyl, substituted or unsubstituted alkynylsulfonyl, substituted or unsubstituted non-aromatic carbocyclylsulfonyl, substituted or unsubstituted aromatic carbocyclylsulfonyl, substituted or unsubstituted non-aromatic heterocyclylsulfonyl, substituted or unsubstituted aromatic heterocyclylsulfonyl or substituted or unsubstituted sulfamoyl

Metadata:
- Claim Count in Document: 5.0
- Percentile: 99.0
- Lexical Diversity: 2.52632
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15557992', '15029031', '16176097', '15501749', '15741875']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8221036945417507
- 35 USC 102 Novelty (BERT): 0.5840820405055243
- Combined Prediction Score: 0.7983015291381281
- Mean Citation Score: 405.67489000000006
- Max Citation Score: 503.35162
- Similarity Product: 424.23633680122384

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test