PATENT CLAIM ANALYSIS

Application Number: 16020043
Application Type: Utility
Filing Date: 2018-06
Publication Date: 2018-10
Patent Classification: ["548", "126000"]

Abstract:
The present invention provides thiazole compounds of Formula I wherein W, Y, R 0 , R 2 , R 4 , R 5 , R 6 , R 7 , X 1 , X 2 , X 3  and X 4  are as defined herein, or a stereoisomer, tautomer, pharmaceutically acceptable salt, prodrug ester or solvate form thereof, wherein all of the variables are as defined herein. These compounds are inhibitors of platelet aggregation and thus can be used as medicaments for treating or preventing thromboembolic disorders.

Claim (Index 1):
A compound of Formula I: or a stereoisomer, tautomer, pharmaceutically acceptable salt, solvate or prodrug thereof, wherein: W is O or S; R 1  is \u2014CH 3 ; R 8  and R 9  are H; R 2  is\n H; \n X 1  is CH; X 2  and X 4  are each CH; X 3  is CR 3 ; R 3  is OCH 3 ; R 4  and R 5  are independently selected from H and C 1 -C 6  alkyl, or R 4  and R 5  can be taken together with the carbon to which they are attached to form a C 3 -C 7  cycloalkyl ring; R 6  is selected from the group consisting of:\n a) phenyl substituted by 0 to 3 groups independently selected from the group consisting of chloro, \u2014CF 3 , cyano, \u2014OCH 3 , \u2014OCF 3 , \u2014SO 2 CH 3  and (C\u2550O)N(CH 3 ) 2 ; \n b) pyridinyl or pyrimidinyl substituted by 0 to 3 groups independently selected from the group consisting of fluoro, chloro, \u2014CH 3  and \u2014OCH 3 ; and \n c) piperidinyl, morpholinyl or thiomorpholinyl substituted by 0 to 3 groups independently selected from the group consisting of fluoro, OH, \u2014CH 3  and \u2014NH 2 ; \n R 7  is selected from the group consisting of H, and \u2014CH 3 .

Metadata:
- Claim Count in Document: 2.0
- Percentile: 94.0
- Lexical Diversity: 1.65517
- Patent Class: 548.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['15593534', '14396831', '14746908', '15549257', '14396771']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8105780308056663
- 35 USC 102 Novelty (BERT): 0.6015386187074531
- Combined Prediction Score: 0.789674089595845
- Mean Citation Score: 473.259004
- Max Citation Score: 540.1893
- Similarity Product: 466.47155519356727

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 0
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test