PATENT CLAIM ANALYSIS

Application Number: 15978988
Application Type: Utility
Filing Date: 2018-05
Publication Date: 2019-05
Patent Classification: ["552", "500000"]

Abstract:
The subject matter of the instant invention is pertinent to the field of treatment of hormone-dependent conditions. New compounds and methods for treating these conditions are disclosed. Embodiments of the instant invention disclose methods for treating endometriosis, dysmenorrhea, breast cancer, uterine fibroids and endometrial hyperproliferation.

Claim (Index 1):
A compound having the general formula: or a pharmaceutically acceptable salt thereof wherein: R 1  is selected from the group consisting of: alkyl; alkenyl; cycloalkyl; cycloalkenyl; aryl; H; CH 3 SO; CH 3 SO 2 ; acyl; alkoxy; thioalkoxy; thioalkyl, acyloxy; Si(CH 3 ) 3 ; wherein X and Y are acyl; aziridinyl, azirinyl, azetidinyl, pyrrolidinyl, ethoxypyrrolidinyl methoxypyrrolidinyl, piperidinyl, ethoxypiperidinyl, morpholinyl, ethoxymorpholinyl, oxazinyl, piperazinyl, methylpiperazinyl, ethylpiperazinyl, and diazinyl; R 2  is selected from the group consisting of: hydrogen, halogen, alkyl, acyl, hydroxyl, alkoxy, acyloxy, alkyl carbonate, cypionyloxy, S-alkyl, S\u2014CN, S-acyl and \u2014OC(O)R 6  wherein R 6  is alkyl, alkoxyalkyl or alkoxy; R 3  is selected from the group consisting of: alkyl, hydroxy, alkoxy, and acyloxy with the proviso that R 3  is other than acetoxy or propynyl; R 4  is hydrogen or alkyl; and X is selected from the group consisting of: \u2550O, \u2550N\u2014OR5 wherein R5 is hydrogen or alkyl, OH, CH 2 , OAlk 1 , and OCOAlk 2 , wherein Alk 1  and Alk 2  are C1-C8 alkyl or C7-C15 aralalkyl, with the proviso that if R 1  is at the para position and is \u2014OCH 3 , \u2014SCH 3 , \u2014NC 4 H 8 , \u2014NC 5 H 10 , \u2014NC 4 H 8 O, \u2014CHO, \u2014CH(OH)CH 3 , \u2014COCH 3 , \u2014O(CH 2 ) 2 NC 4 H 8 , or \u2014O(CH 2 ) 2 NC 5 H 10 , X is other than \u2550O or \u2550N\u2014OR5 wherein R5 is hydrogen or alkyl.

Metadata:
- Claim Count in Document: 20.0
- Percentile: 93.0
- Lexical Diversity: 1.45714
- Patent Class: 552.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['14440023', '14403141', '12990203', '15308804', '13855559']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7395202305241387
- 35 USC 102 Novelty (BERT): 0.6122980935401896
- Combined Prediction Score: 0.7267980168257439
- Mean Citation Score: 370.2074280000001
- Max Citation Score: 390.39532
- Similarity Product: 295.00256630657674

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test