PATENT CLAIM ANALYSIS

Application Number: 16093565
Application Type: Utility
Filing Date: 2018-10
Publication Date: 2019-03
Patent Classification: ["514", "259300"]

Abstract:
The present invention covers Pyrazolopyrimidine compounds of general formula (I), in which n, o, X, Y, R, Q, R 1 , R 2 , R 3  and R 4  are as defined herein, methods of preparing said compounds, intermediate compounds useful for preparing said compounds, pharmaceutical compositions and combinations comprising said compounds and the use of said compounds for manufacturing pharmaceutical compositions for the treatment, control and/or prevention of diseases, in particular of helminth infections, as a sole agent or in combination with other active ingredients.

Claim (Index 8):
A method of preparing a compound of formula (I) according to  claim 1 , said method comprising the step of allowing an intermediate compound of formula 1F: in which R 0 , R 1 , R 2 , R 3 , R 4 , X, Y, o and n are as defined for the compound of formula (I) according to  claim 1 , to react with a compound of formula 1H:\n Q-B(OR) 2 \u2003\u2003 1H, \n \n in which Q is as defined for the compound of general formula (I) according to  claim 1 , and each R may be individually H or Me or both R are pinacolate, thereby giving a compound of formula (I): in which Q, R 0 , R 1 , R 2 , R 3 , R 4 , X, Y, o and n are as defined for the compound of formula (I) according to  claim 1 , or the step of allowing an intermediate compound of formula 2E: in which Q, R 2 , R 3  and R 4  are as defined for the compound of formula (I) according to  claim 1 , to react with a compound of formula 1G: in which R, R 1 , X, Y, o and n are as defined for the compound of formula (I) according to  claim 1 , thereby giving a compound of formula (I): in which Q, R 0 , R 1 , R 2 , R 3 , R 4 , X, Y, o and n are as defined for the compound of formula (I) according to  claim 1 .

Metadata:
- Claim Count in Document: 11.0
- Percentile: 97.0
- Lexical Diversity: 1.67213
- Patent Class: 514.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15022583', '14914069', '15300057', '14767621', '14772471']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7489696122662309
- 35 USC 102 Novelty (BERT): 0.5235596747399979
- Combined Prediction Score: 0.7264286185136077
- Mean Citation Score: 295.60647
- Max Citation Score: 308.264
- Similarity Product: 217.06180535125733

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test