PATENT CLAIM ANALYSIS

Application Number: 16030382
Application Type: Utility
Filing Date: 2018-07
Publication Date: 2018-11
Patent Classification: ["564", "157000"]

Abstract:
Synthesis methods to produce a series of carboxamides built off of an (S)-2-amino acid backbone or an (R)-2-amino acid backbone, depending upon the desired diastereomer of the end product.

Claim (Index 1):
A method for preparing an N-menthanecarboxamide derivative of the following formula (I) comprising: and pharmaceutically acceptable salts thereof; A) a coupling reaction between an activated derivative of the p-menthane-3-carboxylic acid of Formula (II): wherein X=a suitable leaving group; and a primary amine of the general formula (III): to produce a compound of the general formula (IV):

Metadata:
- Claim Count in Document: 3.0
- Percentile: 95.0
- Lexical Diversity: 1.32143
- Patent Class: 564.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['13847641', '12541428', '15331329', '15262205', '14693915']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.730418292268249
- 35 USC 102 Novelty (BERT): 0.5284960912592117
- Combined Prediction Score: 0.7102260721673452
- Mean Citation Score: 277.256942
- Max Citation Score: 292.99277
- Similarity Product: 221.99394084857585

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test