PATENT CLAIM ANALYSIS

Application Number: 16060771
Application Type: Utility
Filing Date: 2018-06
Publication Date: 2018-12
Patent Classification: ["564", "139000"]

Abstract:
Provided is a method of producing an aromatic amide derivative represented by Formula (I), which method includes a process a containing reacting an aniline derivative represented by Formula (II) with a carboxylic acid derivative represented by Formula (III) in the presence of a base to obtain an imide compound represented by Formula (IV) and a process b containing hydrolyzing the imide compound represented by Formula (IV) to obtain the aromatic amide derivative represented by Formula (I): wherein R 1  represents a C 1 -C 4  haloalkyl group, etc.; each of R 2  and R 3  independently represents a hydrogen atom, a halogen atom, etc.; R 4  represents a hydrogen atom, a C 1 -C 4  alkyl group, etc.; each of X 1  and X 2  independently represents a halogen atom, a C 1 -C 4  haloalkyl group, etc.; and Q represents a C 1 -C 4  alkyl group, a phenyl group, a pyridyl group, etc.

Claim (Index 1):
A method of producing an aromatic amide derivative represented by the following Formula (I), comprising the following process a and process b: in Formula (I), R 1  represents a halogen atom; a C 1 -C 4  haloalkyl group; or a C 1 -C 4  haloalkyl group substituted by 1 to 8 substituents, which may be the same or different, selected from the group consisting of a C 1 -C 4  alkyl group, a C 1 -C 4  haloalkyl group, a C 1 -C 4  alkoxy group, a C 1 -C 4  haloalkoxy group, a C 1 -C 4  alkylthio group, a C 1 -C 4  haloalkylthio group, a C 1 -C 4  alkylamino group, a di-C 1 -C 4  alkylamino group, a cyano group, and a nitro group; each of X 1  and X 2  independently represents a hydrogen atom, a halogen atom, a C 1 -C 4  alkyl group, a C 1 -C 4  haloalkyl group, a C 2 -C 4  alkenyl group, a C 2 -C 4  haloalkenyl group, a C 2 -C 4  alkynyl group, a C 2 -C 4  haloalkynyl group, a C 1 -C 4  alkoxy group, a C 1 -C 4  haloalkoxy group, a C 1 -C 4  alkylthio group, a C 1 -C 4  haloalkylthio group, a C 1 -C 4  alkylsulfinyl group, a C 1 -C 4  haloalkylsulfinyl group, a C 1 -C 4  alkylsulfonyl group, a C 1 -C 4  haloalkylsulfonyl group, a C 1 -C 4  alkylamino group, a di-C 1 -C 4  alkylamino group, a cyano group, a nitro group, a C 1 -C 4  alkylcarbonyl group, or a C 1 -C 4  haloalkylcarbonyl group; each of R 2  and R 3  independently represents a hydrogen atom, a halogen atom, a C 1 -C 4  alkyl group, a C 1 -C 4  haloalkyl group, a C 1 -C 4  alkoxy group, a C 1 -C 4  haloalkoxy group, a C 1 -C 4  alkylthio group, a C 1 -C 4  haloalkylthio group, a C 1 -C 4  alkylsulfinyl group, a C 1 -C 4  haloalkylsulfinyl group, a C 1 -C 4  alkylsulfonyl group, a C 1 -C 4  haloalkylsulfonyl group, a C 1 -C 4  alkylamino group, a di-C 1 -C 4  alkylamino group, a cyano group, or a nitro group; R 4  represents: a hydrogen atom; a C 1 -C 4  alkyl group; a C 1 -C 4  haloalkyl group; a C 1 -C 4  alkylcarbonyl group; a C 1 -C 4  haloalkylcarbonyl group; a C 1 -C 4  alkoxycarbonyl group; a C 1 -C 4  haloalkoxycarbonyl group; a C 1 -C 4  alkylsulfonyl group; a C 1 -C 4  haloalkylsulfonyl group; or a C 1 -C 4  alkyl group, a C 1 -C 4  haloalkyl group, a C 1 -C 4  alkylcarbonyl group, a C 1 -C 4  haloalkylcarbonyl group, a C 1 -C 4  alkoxycarbonyl group, a C 1 -C 4  haloalkoxycarbonyl group, a C 1 -C 4  alkylsulfonyl group, or a C 1 -C 4  haloalkylsulfonyl group, substituted by 1 to 9 substituents, which may be the same or different, selected from the group consisting of a C 1 -C 4  alkyl group, a C 1 -C 4  haloalkyl group, a C 1 -C 4  alkoxy group, a C 1 -C 4  haloalkoxy group, a C 1 -C 4  alkylthio group, a C 1 -C 4  haloalkylthio group, a C 1 -C 4  alkylsulfonyl group, a C 1 -C 4  haloalkylsulfonyl group, a C 1 -C 4  alkylamino group, a di-C 1 -C 4  alkylamino group, a C 1 -C 4  alkylcarbonyl group, a C 1 -C 4  alkoxycarbonyl group, a di-C 1 -C 4  alkylaminocarbonyl group, a cyano group, and a nitro group; and Q represents: a C 1 -C 4  alkyl group; a C 1 -C 4  haloalkyl group; a C 1 -C 4  alkylaminocarbonyl group; a C 1 -C 4  haloalkylaminocarbonyl group; a di-C 1 -C 4  alkylaminocarbonyl group; a di-C 1 -C 4  haloalkylaminocarbonyl group; a phenyl group; a heterocyclic group; a C 1 -C 4  alkyl group or a C 1 -C 4  haloalkyl group, substituted by 1 to 9 substituents, which may be the same or different, selected from the group consisting of a halogen atom, a C 1 -C 4  alkyl group, a C 1 -C 4  haloalkyl group, a C 1 -C 4  alkoxy group, a C 1 -C 4  haloalkoxy group, a C 1 -C 4  alkylthio group, a C 1 -C 4  haloalkylthio group, a C 1 -C 4  alkylamino group, a di-C 1 -C 4  alkylamino group, a cyano group, and a nitro group; a phenyl group substituted by 1 to 5 substituents, which may be the same or different, selected from the group consisting of a halogen atom, a C 1 -C 4  alkyl group, a C 1 -C 4  haloalkyl group, a C 1 -C 4  alkoxy group, a C 1 -C 4  haloalkoxy group, a C 1 -C 4  alkylthio group, a C 1 -C 4  haloalkylthio group, a C 1 -C 4  alkylamino group, a di-C 1 -C 4  alkylamino group, a cyano group, and a nitro group; or a heterocyclic group substituted by 1 to 4 substituents, which may be the same or different, selected from the group consisting of a halogen atom, a C 1 -C 4  alkyl group, a C 1 -C 4  haloalkyl group, a C 1 -C 4  alkoxy group, a C 1 -C 4  haloalkoxy group, a C 1 -C 4  alkylthio group, a C 1 -C 4  haloalkylthio group, a C 1 -C 4  alkylamino group, a di-C 1 -C 4  alkylamino group, a cyano group, and a nitro group; wherein the heterocyclic group is a pyridyl group, a pyridyl-N-oxide group, a pyrimidyl group, a pyridazyl group, a pyrazyl group, a furyl group, a thienyl group, an oxazolyl group, an isoxazolyl group, an oxadiazolyl group, a thiazolyl group, an isothiazolyl group, an imidazolyl group, a triazolyl group, a pyrrolyl group, a pyrazolyl group, or a tetrazolyl group; and wherein the process a comprises reacting an aniline derivative represented by the following Formula (II) with a carboxylic acid derivative represented by the following Formula (III), in the presence of a base, to thereby obtain an imide compound represented by the following Formula (IV): in Formula (II), R 1 , X 1 , and X 2  are the same as R 1 , X 1 , and X 2  in Formula (I), in Formula (III), X 3  represents a halogen atom or a C 1 -C 4  alkoxy group, and R 2 , R 3 , R 4 , and Q are the same as R 2 , R 3 , R 4 , and Q in Formula (I), in Formula (IV), R 1 , X 1 , X 2 , R 2 , R 3 , R 4 , and Q are the same as R 1 , X 1 , X 2 , R 2 , R 3 , R 4 , and Q in Formula (I), and two of R 2 , R 3 , R 4  and Q may be the same or different at each occurrence, respectively; and\n the process b comprises hydrolyzing the imide compound represented by Formula (IV), to thereby obtain the aromatic amide derivative represented by Formula (I).

Metadata:
- Claim Count in Document: 15.0
- Percentile: 94.0
- Lexical Diversity: 2.89231
- Patent Class: 564.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['13016604', '13845664', '14433787', '10587990', '14366715']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.761929884023736
- 35 USC 102 Novelty (BERT): 0.5529422244339787
- Combined Prediction Score: 0.7410311180647603
- Mean Citation Score: 368.154356
- Max Citation Score: 374.60898
- Similarity Product: 313.5261516359282

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test