PATENT CLAIM ANALYSIS

Application Number: 16000968
Application Type: Utility
Filing Date: 2018-06
Publication Date: 2018-10
Patent Classification: ["514", "263100"]

Abstract:
Provided herein are Purine Compounds of Formula (I) or pharmaceutically acceptable salts, tautomers, isotopologues, or stereoisomers thereof, wherein R 1 , R 2 , and R 3  are as defined herein, compositions comprising an effective amount of a Purine Compound, and methods for treating or preventing malaria comprising the administration of an effective amount of a Purine Compound.

Claim (Index 1):
A method of treating or preventing malaria, comprising administering to a subject having malaria an effective amount of a compound of formula (I), or a pharmaceutically acceptable salt, tautomer, isotopologue, or stereoisomer thereof, wherein R 1  is CR 1a R 1b R 1c , wherein R 1a  and R 1b  are (C 1-4 )alkyl and R 1c  is H or (C 1-4 )alkyl; or R 1a  and R 1b  form a 3-6 membered cycloalkyl or 3-6 membered heterocyclyl, and R 1c  is H or (C 1-4 )alkyl; R 2  is L-R 2a  or L-R 2b , L is a bond or (C 1-2  alkyl); R 2a  is 3-6 membered N-containing heterocyclyl or heteroaryl, each optionally substituted with one or more (C 1-4 )alkyl, or (C 1-4 )alkyl-NR 2 ; R 2b  is (C 1-4  branched or unbranched alkyl)-NR 2 ,\n R 3  is phenyl or pyridyl, substituted with at least one halogen, CN, (C 1-4 )alkyl, or O(C 1-4 )alkyl, wherein the alkyl is optionally fluorinated; and \n R is H or (C 1-4 ) alkyl.

Metadata:
- Claim Count in Document: 56.0
- Percentile: 94.0
- Lexical Diversity: 1.59524
- Patent Class: 514.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['15611108', '15611061', '16000969', '15864499', '15091887']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7710046712049548
- 35 USC 102 Novelty (BERT): 0.6140159113077054
- Combined Prediction Score: 0.7553057952152298
- Mean Citation Score: 428.277916
- Max Citation Score: 563.66614
- Similarity Product: 486.5460003573168

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test