PATENT CLAIM ANALYSIS

Application Number: 15750440
Application Type: Utility
Filing Date: 2018-02
Publication Date: 2018-09
Patent Classification: ["544", "236000"]

Abstract:
The invention relates to novel compounds of the formula (I) in welcher R 1 , R 2 , R 3 , A 1 , X and n have the meanings given above,to their use as acaricides and/or insecticides for controlling animal pests and to processes and intermediates for their preparation.

Claim (Index 3):
Compound of formula (I) according to  claim 1  wherein\n A 1  represents nitrogen or \u2550C\u2014R 4 , \n R 1  represents (C 1 -C 4 )-alkyl, (C 1 -C 4 )-hydroxyalkyl, (C 1 -C 4 )-haloalkyl, (C 2 -C 4 )-alkenyl, (C 2 -C 4 )-haloalkenyl, (C 2 -C 4 )-alkynyl, (C 2 -C 4 )-haloalkynyl, (C 3 -C 6 )-cycloalkyl, (C 1 -C 4 )-alkylthio-(C 1 -C 4 )-alkyl, (C 1 -C 4 )-alkylsulphinyl-(C 1 -C 4 )-alkyl or (C 1 -C 4 )-alkylsulphonyl-(C 1 -C 4 )-alkyl, \n R 2  represents a 5- or 6-membered saturated, partially saturated or heteroaromatic ring from the group consisting of Q1 to Q101 which is optionally mono- or disubstituted by identical or different substituents, which may in each case contain at least one carbonyl group and/or where possible substituents are in each case as follows: hydrogen, cyano, (C 1 -C 4 )cyanoalkyl, (C 1 -C 4 )alkoxy-(C 1 -C 4 )alkyl, halogen, amino, (C 1 -C 4 )alkyl, (C 1 -C 4 )haloalkyl, (C 2 -C 4 )alkenyl, (C 2 -C 4 )haloalkenyl, (C 2 -C 4 )alkynyl, (C 2 -C 4 )haloalkynyl, (C 3 -C 6 )cycloalkyl, (C 3 -C 6 )cycloalkyl-(C 3 -C 6 )cycloalkyl, (C 1 -C 4 )alkyl-(C 3 -C 6 )cycloalkyl, (C 1 -C 4 )alkoxy, (C 1 -C 4 )haloalkoxy, (C 1 -C 4 )alkoxyimino, \u2014C(H)\u2550N\u2014O(C 1 -C 4 )alkyl, (C 1 -C 4 )alkylthio, (C 1 -C 4 )haloalkylthio, (C 1 -C 4 )alkylsulphinyl, (C 1 -C 4 )haloalkylsulphinyl, (C 1 -C 4 )alkylsulphonyl, (C 1 -C 4 )alkylsulphonyl-(C 1 -C 4 )alkyl, (C 1 -C 4 )haloalkylsulphonyl, (C 1 -C 4 )alkylsulphonyloxy, (C 1 -C 4 )alkylcarbonyl, (C 1 -C 4 )haloalkylcarbonyl, aminocarbonyl, (C 1 -C 4 )alkylaminocarbonyl, di-(C 1 -C 4 )alkylaminocarbonyl, (C 1 -C 4 )alkylsulphonylamino, (C 1 -C 4 )alkylamino, di-(C 1 -C 4 )alkylamino, aminosulphonyl, (C 1 -C 4 )alkylaminosulphonyl, di-(C 1 -C 4 )alkylaminosulphonyl, (C 1 -C 4 )alkylcarbonylamino, \n where the bond to the remainder of the molecule is identified by an asterisk *, R 2  furthermore represents a group selected from G1, G2, G3, G4, G6, G7, G8, G9, G10, G11, G12, G13, G14, G15, G16, G18 or G19, where if R 2  represents G6, G7, G8, G9, then n represents 2, R 3  represents hydrogen, cyano, halogen, nitro, hydroxy, amino, SCN, tri-(C 1 -C 4 )alkylsilyl, (C 3 -C 6 )cycloalkyl, (C 3 -C 6 )cycloalkyl-(C 3 -C 6 )cycloalkyl, (C 1 -C 4 )alkyl-(C 3 -C 6 )cycloalkyl, halo(C 3 -C 6 )cycloalkyl, (C 1 -C 4 )alkyl, (C 1 -C 4 )haloalkyl, (C 1 -C 4 )cyanoalkyl, (C 1 -C 4 )alkoxy-(C 1 -C 4 )alkyl, (C 2 -C 4 )alkenyl, (C 2 -C 4 )haloalkenyl, (C 2 -C 4 )cyanoalkenyl, (C 2 -C 4 )alkynyl, (C 2 -C 4 )haloalkynyl, (C 2 -C 4 )cyanoalkynyl, (C 1 -C 4 )alkoxy, (C 1 -C 4 )haloalkoxy, (C 1 -C 4 )cyanoalkoxy, (C 1 -C 4 )alkylhydroxyimino, (C 1 -C 4 )alkoxyimino, (C 1 -C 4 )alkyl-(C 1 -C 4 )alkoxyimino, (C 1 -C 4 )alkylthio, (C 1 -C 4 )haloalkylthio, (C 1 -C 4 )alkylsulphinyl, (C 1 -C 4 )haloalkylsulphinyl, (C 1 -C 4 )alkylsulphonyl, (C 1 -C 4 )haloalkylsulphonyl, (C 1 -C 4 )alkylsulphonyloxy, (C 1 -C 4 )alkylcarbonyl, (C 1 -C 4 )haloalkylcarbonyl, aminocarbonyl, (C 1 -C 4 )alkylaminocarbonyl, di-(C 1 -C 4 )alkylaminocarbonyl, (C 1 -C 4 )alkylsulphonylamino, (C 1 -C 4 )alkylamino, di-(C 1 -C 4 )alkylamino, aminosulphonyl, (C 1 -C 4 )alkylaminosulphonyl, di-(C 1 -C 4 )alkylaminosulphonyl, NHCO\u2014(C 1 -C 4 )alkyl ((C 1 -C 4 )alkylcarbonylamino), furthermore represents phenyl or hetaryl, each of which is optionally mono- or disubstituted by identical or different substituents, where (in the case of hetaryl) at least one carbonyl group may optionally be present and/or where possible substituents are in each case as follows: cyano, halogen, (C 3 -C 6 )cycloalkyl, (C 3 -C 6 )cycloalkyl-(C 3 -C 6 )cycloalkyl, (C 1 -C 4 )alkyl-(C 3 -C 6 )cycloalkyl, halogen(C 3 -C 6 )cycloalkyl, (C 1 -C 4 )alkyl, (C 1 -C 4 )haloalkyl, (C 1 -C 4 )cyanoalkyl, (C 2 -C 4 )alkenyl, (C 2 -C 4 )haloalkenyl, (C 2 -C 4 )cyanoalkenyl, (C 2 -C 4 )alkynyl, (C 2 -C 4 )haloalkynyl, (C 2 -C 4 )cyanoalkynyl, (C 1 -C 4 )alkoxy, (C 1 -C 4 )haloalkoxy, (C 1 -C 4 )alkylhydroxyimino, (C 1 -C 4 )alkoxyimino, (C 1 -C 4 )alkyl-(C 1 -C 4 )alkoxyimino, (C 1 -C 4 )alkylthio, (C 1 -C 4 )haloalkylthio, (C 1 -C 4 )alkylsulphinyl, (C 1 -C 4 )haloalkylsulphinyl, (C 1 -C 4 )alkylsulphonyl, (C 1 -C 4 )haloalkylsulphonyl, (C 1 -C 4 )alkylsulphonyloxy, (C 1 -C 4 )alkylcarbonyl, (C 1 -C 4 )haloalkylcarbonyl, aminocarbonyl, (C 1 -C 4 )alkylaminocarbonyl, di-(C 1 -C 4 )alkylaminocarbonyl, (C 1 -C 4 )alkylsulphonylamino, (C 1 -C 4 )alkylamino, di-(C 1 -C 4 )alkylamino, aminosulphonyl, (C 1 -C 4 )alkylaminosulphonyl, di-(C 1 -C 4 )alkylaminosulphonyl, NHCO\u2014(C 1 -C 4 )alkyl ((C 1 -C 4 )alkylcarbonylamino), R 4  represents hydrogen, halogen, cyano or (C 1 -C 4 )-alkyl, X represents a heteroaromatic 9-membered or 12-membered fused bicyclic or tricyclic ring system from the series H1 to H20, where the bond to the remainder of the molecule is identified by a diamond #, R 5 , R 6  independently of one another represent hydrogen, cyano, halogen, (C 1 -C 4 )alkyl, (C 1 -C 4 )haloalkyl, (C 2 -C 4 )alkenyl, (C 2 -C 4 )haloalkenyl, (C 2 -C 4 )alkynyl, (C 2 -C 4 )haloalkynyl, (C 3 -C 6 )cycloalkyl, (C 3 -C 6 )cycloalkyl-(C 3 -C 6 )cycloalkyl, (C 1 -C 4 )alkyl-(C 3 -C 6 )cycloalkyl, (C 1 -C 4 )alkoxy, (C 1 -C 4 )haloalkoxy, (C 1 -C 4 )alkoxyimino, (C 1 -C 4 )alkylthio, (C 1 -C 4 )haloalkylthio, (C 1 -C 4 )alkylsulphinyl, (C 1 -C 4 )haloalkylsulphinyl, (C 1 -C 4 )alkylsulphonyl, (C 1 -C 4 )haloalkylsulphonyl, (C 1 -C 4 )alkylsulphonyloxy, (C 1 -C 4 )alkylcarbonyl, (C 1 -C 4 )haloalkylcarbonyl, aminocarbonyl, (C 1 -C 4 )alkylaminocarbonyl, di-(C 1 -C 4 )alkylaminocarbonyl, (C 1 -C 4 )alkylsulphonylamino, (C 1 -C 4 )alkylamino, di-(C 1 -C 4 )alkylamino, aminosulphonyl, (C 1 -C 4 )alkylaminosulphonyl or di-(C 1 -C 4 )alkylaminosulphonyl, R 7  represents (C 1 -C 4 )alkyl, (C 1 -C 4 )haloalkyl, (C 1 -C 4 )cyanoalkyl, (C 1 -C 4 )hydroxyalkyl, (C 1 -C 4 )alkoxy-(C 1 -C 4 )alkyl, (C 1 -C 4 )haloalkoxy-(C 1 -C 4 )alkyl, (C 2 -C 4 )alkenyl, (C 2 -C 4 )alkenyloxy-(C 1 -C 4 )alkyl, (C 2 -C 4 )haloalkenyloxy-(C 1 -C 4 )alkyl, (C 2 -C 4 )haloalkenyl, (C 2 -C 4 )cyanoalkenyl, (C 2 -C 4 )alkynyl, (C 2 -C 4 )alkynyloxy-(C 1 -C 4 )alkyl, (C 2 -C 4 )haloalkynyl, (C 3 -C 6 )cycloalkyl, (C 3 -C 6 )cycloalkyl-(C 3 -C 6 )cycloalkyl, (C 1 -C 4 )alkyl-(C 3 -C 6 )cycloalkyl, halo(C 3 -C 6 )cycloalkyl, (C 1 -C 4 )alkylthio-(C 1 -C 4 )alkyl, (C 1 -C 4 )alkylsulphinyl-(C 1 -C 4 )alkyl, (C 1 -C 4 )alkylsulphonyl-(C 1 -C 4 )alkyl or (C 1 -C 4 )alkylcarbonyl-(C 1 -C 4 )alkyl, R 8  represents hydrogen, amino, (C 1 -C 4 )alkylthio-(C 1 -C 4 )alkyl, (C 1 -C 4 )alkylsulphinyl-(C 1 -C 4 )alkyl, (C 1 -C 4 )alkylsulphonyl-(C 1 -C 4 )alkyl, (C 1 -C 4 )alkylamino, (C 1 -C 4 )alkoxy-(C 1 -C 4 )alkyl, (C 3 -C 6 )cycloalkyl or (C 3 -C 6 )cycloalkyl-(C 1 -C 4 )alkyl, represents (C 1 -C 4 )alkyl or (C 1 -C 4 )alkoxy in each case optionally monosubstituted by halogen, cyano, phenyl or pyridyl, where phenyl or pyridyl can in each case be optionally mono- or disubstituted by identical or different substituents selected from the group consisting of trifluoromethyl, cyano, fluorine, chlorine, bromine or trifluoromethoxy, or R 8  represents phenyl, thiazolyl, pyrazolyl, pyridyl or a 3- to 6-membered saturated heterocycle comprising 1-2 heteroatoms from the group consisting of N, S and O, where phenyl, pyridyl and the heterocycle may each optionally be mono- or disubstituted by identical or different substituents, and where the substituents independently of one another may be selected from C 1 -C 4 -alkyl, C 1 -C 4 -haloalkyl, halogen or cyano, R 13 , R 14 , R 15  independently of one another represent (C 1 -C 4 )alkyl or (C 3 -C 6 )cycloalkyl, optionally monosubstituted by halogen, cyano, phenyl or pyridyl, where phenyl or pyridyl can in each case be optionally mono- or disubstituted by identical or different substituents from the group consisting of trifluoromethyl, cyano, fluorine, chlorine or trifluoromethoxy, or R 13 , R 14 , R 15  independently of one another represent phenyl, pyridyl or a 3- to 6-membered saturated heterocycle comprising 1-2 heteroatoms from the group consisting of N, S and O, where phenyl, pyridyl and the heterocycle may each be mono- or disubstituted by identical or different substituents, and where the substituents independently of one another may be selected from the group consisting of C 1 -C 4 -alkyl, C 1 -C 4 -haloalkyl, halogen and cyano, R 11 , R 12  independently of one another represent hydrogen or represent R 13 , n represents 0, 1 or 2, p represents 0 or 1, where if R 2  represents optionally substituted Q45, then X is not H1, H2 or H4 and if R 2  represents G10, G11, G12, G13, G14, G15 or G16 and A 1  represents N, then X does not represent H1, H2, H4, H5, H7, H8 or H14.

Metadata:
- Claim Count in Document: 10.0
- Percentile: 88.0
- Lexical Diversity: 1.34146
- Patent Class: 544.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15770738', '16068846', '15119124', '15742369', '15101767']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8115818240407011
- 35 USC 102 Novelty (BERT): 0.5577103864538914
- Combined Prediction Score: 0.7861946802820201
- Mean Citation Score: 406.019578
- Max Citation Score: 434.26294
- Similarity Product: 417.26936305931815

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test