PATENT CLAIM ANALYSIS

Application Number: 15998528
Application Type: Utility
Filing Date: 2018-08
Publication Date: 2019-03
Patent Classification: ["546", "270100"]

Abstract:
Methods of synthesizing 2−(1′H-indole-3′-carbonyl)-thiazole-4-carboxylic acid methyl ester (ITE) and structural analogs thereof. The methods include condensation reactions or condensation and oxidation reactions to form the thiazoline or thiazole moiety of ITE or its structural analogs.

Claim (Index 52):
The method of  claim 51 , wherein the amino protecting group forms a group selected from the group consisting of an alkyl carbamate, allyl carbamate (Alloc), t-butyl carbamate (BOC), 9-fluorenylmethyl carbamate (FMOC), benzyl carbamate (Cbz), acetamide, chloroacetamide, trifluoroacetamide (TFA), phthalimide, benzylamine, triphenylmethylamine (tritylamine), benzylideneamine, p-toluenesulfonamide, and tosylamide.

Metadata:
- Claim Count in Document: 80.0
- Percentile: 96.0
- Lexical Diversity: 1.3871
- Patent Class: 546.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['15509722', '14380794', '14543341', '13867699', '12308399']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7925501140369313
- 35 USC 102 Novelty (BERT): 0.6264573129000496
- Combined Prediction Score: 0.7759408339232432
- Mean Citation Score: 286.88801
- Max Citation Score: 586.0267299999998
- Similarity Product: 551.0113763572035

Labels:
- Claim Label 101: 0
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 0
- Label 101 Adjusted: 0

Dataset: test