PATENT CLAIM ANALYSIS

Application Number: 15748786
Application Type: Utility
Filing Date: 2018-01
Publication Date: 2019-01
Patent Classification: ["544", "350000"]

Abstract:
Compounds of the formula Ia or of the formula Ib in which X, Y, R 1  and R 2  have the meanings indicated in claim  1 , are inhibitors of pyruvate dehydrogenase kinase (PDHK), and can be employed, inter alia, for the treatment of diseases such as cancer.

Claim (Index 4):
Compounds according to  claim 1  in which\n X denotes CH or N, \n Y denotes CH or N, \n R 1  denotes H, A, (CH 2 )\u2014Ar, (CH 2 ) n Het or Cyc, \n R 2  denotes H or CH 3 , \n Ar denotes phenyl, which is unsubstituted or mono-, di-, tri-, tetra- or pentasubstituted by Hal, A, CN and/or OA, \n Het denotes pyrimidyl, pyridyl, pyridazinyl, pyrazinyl, piperidinyl, pyrrolidinyl, pyrazolyl, thiazolyl, imidazolyl, furanyl, thiophenyl, pyrrolyl, oxazolyl, isoxazolyl, triazolyl, oxadiazolyl or thiadiazolyl, each of which is unsubstituted or mono- or disubstituted by Hal, A and/or OA, \n Cyc denotes cyclic alkyl with 3, 4, 5, 6 or 7 C-atoms, which is unsubstituted or monosubstituted by OH, \n A denotes unbranched or branched alkyl with 1-10 C-atoms, wherein one or two non-adjacent CH- and/or CH 2 -groups may be replaced by N-, O- and/or S-atoms and/or wherein 1-7 H-atoms may be replaced by R 4 , \n R 4  denotes F, Cl or OH, \n Hal denotes F, Cl, Br or I, \n n denotes 0, 1 or 2, \n with the proviso that, \n if X\u2550CH then Y\u2550N \n or \n if Y\u2550CH then X\u2550N, \n and pharmaceutically acceptable salts, tautomers and stereoisomers thereof, including mixtures thereof in all ratios.

Metadata:
- Claim Count in Document: 18.0
- Percentile: 86.0
- Lexical Diversity: 1.4
- Patent Class: 544.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15105154', '09927324', '12298369', '14342749', '14420003']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7923780740312975
- 35 USC 102 Novelty (BERT): 0.545627316884871
- Combined Prediction Score: 0.7677029983166549
- Mean Citation Score: 375.832478
- Max Citation Score: 391.2317
- Similarity Product: 335.07881602606767

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test