PATENT CLAIM ANALYSIS

Application Number: 15757238
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2018-08
Patent Classification: ["514", "314000"]

Abstract:
Disclosed herein are compositions and methods for modulating the androgen receptor.

Claim (Index 1):
A compound, or a pharmaceutically acceptable salt thereof, having the formula: wherein R 1  is hydrogen or substituted or unsubstituted pyrid-2-yl; R 2  is independently a hydrogen, halogen, \u2014CX 2 3 , \u2014CHX 2 2 , \u2014CH 2 X 2 , \u2014CN, \u2014SO n2 R 10 , \u2014SO v2 NR 7 R 8 , \u2014NHNR 7 R 8 , \u2014ONR 7 R 8 , \u2014NHC\u2550(O)NHNR 7 R 8 , \u2014NHC\u2550(O)NR 7 R 8 , \u2014N(O) m2 , \u2014NR 7 R 8 , \u2014C(O)R 9 , \u2014C(O)\u2014OR 9 , \u2014C(O)NR 7 R 8 , \u2014OR 10 , \u2014NR 7 SO 2 R 10 , \u2014NR 7 C\u2550(O)R 9 , \u2014NR 7 C(O)\u2014OR 9 , \u2014NR 7 OR 9 , \u2014OCX 2 3 , \u2014OCHX 2 2 , \u2014OCH 2 X 2 , substituted or unsubstituted alkyl, substituted or unsubstituted heteroalkyl, substituted or unsubstituted cycloalkyl, substituted or unsubstituted heterocycloalkyl, substituted or unsubstituted aryl, or substituted or unsubstituted heteroaryl; R 3  is independently a hydrogen, halogen, \u2014CX 3 3 , \u2014CHX 3 2 , \u2014CH 2 X 3 , \u2014CN, \u2014SO n3 R 14 , \u2014SO v3 NR 11 R 12 , \u2014NHNH 2 , \u2014ONR 11 R 12 , \u2014NHC\u2550(O)NHNH 2 , \u2014NHC\u2550(O)NR 11 R 12 , \u2014N(O) m3 , \u2014NR 11 R 12 , \u2014C(O)R 13 , \u2014C(O)\u2014OR 13 , \u2014C(O)NR 11 R 12 , \u2014OR 14 , \u2014NR 11 SO 2 R 14 , \u2014NR 11 C\u2550(O)R 13 , \u2014NR 11 C(O)\u2014OR 13 , \u2014NR 11 OR 13 , \u2014OCX 3 3 , \u2014OCHX 3 2 , \u2014OCH 2 X 3 , substituted or unsubstituted alkyl, substituted or unsubstituted heteroalkyl, substituted or unsubstituted cycloalkyl, substituted or unsubstituted heterocycloalkyl, substituted or unsubstituted aryl, or substituted or unsubstituted heteroaryl; R 7 , R 8 , R 9 , R 10 , R 11 , R 12 , R 13 , and R 14  are independently hydrogen, halogen, \u2014CX 3 , \u2014CHX 2 , \u2014CH 2 X, \u2014OCX 3 , \u2014OCHX 2 , \u2014OCH 2 X, \u2014CN, \u2014OH, \u2014NH 2 , \u2014COOH, \u2014CONH 2 , \u2014NO 2 , \u2014SH, \u2014SO 3 H, \u2014SO 4 H, \u2014SO 2 NH 2 , \u2014NHNH 2 , \u2014ONH 2 , \u2014NHC\u2550(O)NHNH 2 , \u2014NHC\u2550(O)NH 2 , \u2014NHSO 2 H, \u2014NHC\u2550(O)H, \u2014NHC(O)\u2014OH, \u2014NHOH, substituted or unsubstituted alkyl, substituted or unsubstituted heteroalkyl, substituted or unsubstituted cycloalkyl, substituted or unsubstituted heterocycloalkyl, substituted or unsubstituted aryl, or substituted or unsubstituted heteroaryl; R 7  and R 8  substituents bonded to the same nitrogen atom may optionally be joined to form a substituted or unsubstituted heterocycloalkyl or substituted or unsubstituted heteroaryl; R 11  and R 12  substituents bonded to the same nitrogen atom may optionally be joined to form a substituted or unsubstituted heterocycloalkyl or substituted or unsubstituted heteroaryl; R 4  is independently hydrogen, a \u2014CX 4 3 , \u2014CHX 4 2 , \u2014CH 2 X 4 , \u2014CN, \u2014C(O)H, \u2014C(O)OH, \u2014C(O)NH 2 , substituted or unsubstituted alkyl, substituted or unsubstituted heteroalkyl, substituted or unsubstituted cycloalkyl, substituted or unsubstituted heterocycloalkyl, substituted or unsubstituted aryl, or substituted or unsubstituted heteroaryl; R 5  is independently a hydrogen, halogen, \u2014CX 5 3 , \u2014CHX 5 2 , \u2014CH 2 X 5 , \u2014CN, \u2014C(O)H, \u2014C(O)OH, \u2014C(O)NH 2 , substituted or unsubstituted alkyl, substituted or unsubstituted heteroalkyl, substituted or unsubstituted cycloalkyl, substituted or unsubstituted heterocycloalkyl, substituted or unsubstituted aryl, or substituted or unsubstituted heteroaryl; R 6  is independently a hydrogen, halogen, \u2014CX 6 3 , \u2014CHX 6 2 , \u2014CH 2 X 6 \u2014CN, \u2014C(O)H, \u2014C(O)OH, \u2014C(O)NH 2 , substituted or unsubstituted alkyl, substituted or unsubstituted heteroalkyl, substituted or unsubstituted cycloalkyl, substituted or unsubstituted heterocycloalkyl, substituted or unsubstituted aryl, or substituted or unsubstituted heteroaryl; L 1  is independently a bond, substituted or unsubstituted alkylene, substituted or unsubstituted alkenylene, substituted or unsubstituted alkynylene, substituted or unsubstituted heteroalkylene, substituted or unsubstituted heteroalkenylene, or substituted or unsubstituted heteroalkynylene; m2, m3, v2, and v3 are independently 1 or 2; n2 and n3 are independently an integer from 0 to 4; X, X 2 , X 3 , X 4 , X 5 , and X 6  are independently \u2014Cl, \u2014Br, \u2014I, or \u2014F.

Metadata:
- Claim Count in Document: 1.0
- Percentile: 90.0
- Lexical Diversity: 1.0
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15382942', '15760959', '15648245', '15518331', '15662861']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8405683345098737
- 35 USC 102 Novelty (BERT): 0.6393772532039294
- Combined Prediction Score: 0.8204492263792793
- Mean Citation Score: 587.369966
- Max Citation Score: 630.3422
- Similarity Product: 547.0988012297869

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test