PATENT CLAIM ANALYSIS

Application Number: 16247132
Application Type: Utility
Filing Date: 2019-01
Publication Date: 2019-08
Patent Classification: ["546", "113000"]

Abstract:
The present invention relates to compounds of the formula (I), or pharmaceutically acceptable salts, enantiomer or diastereomer thereof, wherein R 1  to R 5  are as described above. The compounds may be useful for the treatment or prophylaxis of hepatitis B virus infection.

Claim (Index 4):
A compound selected from:\n 3-(2-oxopyrrolidin-1-yl)-N-(3,4,5-trifluorophenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carboxamide; 3-(5,5-dimethyl-2-oxo-oxazolidin-3-yl)-N-(3,4,5-trifluorophenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carboxamide; 3-(2,4-difluorophenyl)-N-(3,4,5-trifluorophenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carboxamide; 3-cyclopentyl-N-(3,4,5-trifluorophenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carboxamide; 3-(1,1-dioxo-1,2-thiazolidin-2-yl)-N-(3,4,5-trifluorophenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carboxamide; 3-(5-benzyl-1,1-dioxo-1,2,5-thiadiazolidin-2-yl)-N-(3,4,5-trifluorophenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carboxamide; 3-(1,1-dioxo-1,2,5-thiadiazolidin-2-yl)-N-(3,4,5-trifluorophenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carboxamide; 3-(4-cyano-2-oxo-pyrrolidin-1-yl)-N-(3,4,5-trifluorophenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carboxamide; 3-(3-oxomorpholin-4-yl)-N-(3,4,5-trifluorophenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carboxamide; 3-[4-(3-methyl-1,2,4-oxadiazol-5-yl)-2-oxo-pyrrolidin-1-yl]-N-(3,4,5-trifluorophenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carboxamide; 3-(2,4-difluorophenyl)-N-(3-thienyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carboxamide; 3-(2,4-difluorophenyl)-N-[4-fluoro-3-(trifluoromethyl)phenyl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carboxamide; N-(3-cyano-4-fluoro-phenyl)-3-(2,4-difluorophenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carboxamide; 3-(2,4-difluorophenyl)-N-(4-fluoro-3-methyl-phenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carboxamide; 3-(2,4-difluorophenyl)-N-(2,6-difluoro-4-pyridyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carboxamide; 3-(2,4-difluorophenyl)-N-(2-fluoro-4-pyridyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carboxamide; 3-(6-fluoro-3-pyridyl)-N-(3,4,5-trifluorophenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carboxamide; and 3-[4-(5-methyl-1,2,4-oxadiazol-3-yl)-2-oxo-pyrrolidin-1-yl]-N-(3,4,5-trifluorophenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-5-carboxamide.

Metadata:
- Claim Count in Document: 4.0
- Percentile: 99.0
- Lexical Diversity: 1.28205
- Patent Class: 546.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['14997346', '16247170', '16196324', '16247084', '14632078']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8041323357955437
- 35 USC 102 Novelty (BERT): 0.580757124662433
- Combined Prediction Score: 0.7817948146822327
- Mean Citation Score: 415.54647000000006
- Max Citation Score: 473.76462
- Similarity Product: 425.1012020296097

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test