PATENT CLAIM ANALYSIS

Application Number: 16250212
Application Type: Utility
Filing Date: 2019-01
Publication Date: 2019-05
Patent Classification: ["514", "303000"]

Abstract:
The purpose of the present invention is to provide novel compounds having ACC2 selective inhibitory activity. In addition, the present invention provides a pharmaceutical composition comprising the compound. A compound of Formula: or its pharmaceutically acceptable salt, wherein, R 1  is substituted or unsubstituted fused aromatic heterocyclyl represented by Formula: wherein,         ring B is 5-membered ring, ring C is 6-membered ring;           ring A is substituted or unsubstituted non-aromatic carbocycle or the like; -L 1 - is —O—(CR 6 R 7 )m- or the like; -L 2 - is —O—(CR 6 R 7 )n- or the like; each R 6  is independently hydrogen or the like; each R 7  is independently hydrogen or the like; each m is independently an integer of 0, 1, 2 or 3; each n is independently an integer of 1, 2 or 3; R 2  is substituted or unsubstituted alkyl; R 3  is hydrogen or substituted or unsubstituted alkyl; R 4  is substituted or unsubstituted alkylcarbonyl or the like.

Claim (Index 2):
The compound or its pharmaceutically acceptable salt according to  claim 1 , wherein R 1  is the group represented by Formula: wherein\n X 1  is N or C(R x1 ); \n X 2  is N or C(R x2 ); \n X 3  is N or C(R x3 ); \n X 4  is N or C(R x4 ); \n X 5  is N(R x5 ), O or S; \n X 6  is N or C(R x6 ); \n each R x1 , R x2 , R x3 , R x4 , R x5  and R x6  is independently hydrogen, halogen, hydroxy, carboxy, cyano, substituted or unsubstituted alkyl, substituted or unsubstituted alkenyl, substituted or unsubstituted alkynyl, substituted or unsubstituted alkyloxy, substituted or unsubstituted alkenyloxy, substituted or unsubstituted alkynyloxy, substituted or unsubstituted alkylsulfanyl, substituted or unsubstituted alkenylsulfanyl, substituted or unsubstituted alkynylsulfanyl, substituted or unsubstituted amino, substituted or unsubstituted carbamoyl, substituted or unsubstituted sulfamoyl, substituted or unsubstituted alkylcarbonyl, substituted or unsubstituted alkenylcarbonyl, substituted or unsubstituted alkynylcarbonyl, substituted or unsubstituted alkyloxycarbonyl, substituted or unsubstituted alkenyloxycarbonyl, substituted or unsubstituted alkynyloxycarbonyl, substituted or unsubstituted alkylsulfonyl, substituted or unsubstituted alkenylsulfonyl, substituted or unsubstituted alkynylsulfonyl, substituted or unsubstituted non-aromatic carbocyclyl, substituted or unsubstituted aromatic carbocyclyl, substituted or unsubstituted non-aromatic heterocyclyl, substituted or unsubstituted aromatic heterocyclyl, substituted or unsubstituted non-aromatic carbocyclylsulfonyl, substituted or unsubstituted aromatic carbocyclylsulfonyl, substituted or unsubstituted non-aromatic heterocyclylsulfonyl, substituted or unsubstituted aromatic heterocyclylsulfonyl, substituted or unsubstituted non-aromatic carbocyclyloxy, substituted or unsubstituted aromatic carbocyclyloxy, substituted or unsubstituted non-aromatic heterocyclyloxy, or substituted or unsubstituted aromatic heterocyclyloxy.

Metadata:
- Claim Count in Document: 5.0
- Percentile: 99.0
- Lexical Diversity: 2.52632
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15557992', '15029031', '16176097', '15501749', '15741875']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8226536105805403
- 35 USC 102 Novelty (BERT): 0.581906987547441
- Combined Prediction Score: 0.7985789482772304
- Mean Citation Score: 405.67489000000006
- Max Citation Score: 503.35162
- Similarity Product: 413.2109870991445

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test