PATENT CLAIM ANALYSIS

Application Number: 16205637
Application Type: Utility
Filing Date: 2018-11
Publication Date: 2019-03
Patent Classification: ["514", "751000"]

Abstract:
The present invention is directed to novel compounds of Formula (I), pharmaceutically acceptable salts or solvates thereof, and their use.

Claim (Index 40):
A diagnostic imaging composition comprising a compound of Formula I: or a pharmaceutically acceptable salt or solvate thereof and at least one pharmaceutically acceptable carrier, diluent, excipient and/or adjuvant, wherein X 1  and X 5  are independently selected from the group consisting of hydrogen, halogen, C1-C4-alkyl, C1-C4-haloalkyl, cyano, nitro, di(C1-C4-alkyl)amino, \u2014NHCOOR\u2032, and \u2014COOR\u2032, wherein R\u2032 is methyl, ethyl, n-propyl, n-butyl iso-propyl, iso-butyl or tert-butyl; X 2 , X 3 , X 4  are independently selected from the group consisting of hydrogen, chloro, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy, cyano, nitro, di(C1-C4-alkyl)amino, \u2014NHCOOR\u2032, and \u2014COOR\u2032, wherein R\u2032 is methyl, ethyl, n-propyl, n-butyl, iso-propyl, iso-butyl or tert-butyl; with the proviso that at least one of X 1 , X 2 , X 3 , X 4 , X 5  is not hydrogen and that at least one of X 2 , X 3 , X 4  is not C1-C4-alkoxy; L is \u2014C(O)NH\u2014, \u2014NHC(O)\u2014, \u2014SO 2 NH\u2014, \u2014NHSO 2 \u2014, or \u2014NH\u2014; n is 0, 1 or 2; n is 1, 2, 3, 4 or 5; R 1  is H or alkyl, and R 2  is 5- or 6-membered arylalkyl, 5- or 6-membered cycloalkylalkyl, wherein the cyclic moiety of said arylalkyl or cycloalkylalkyl is optionally substituted by one or more substituents independently selected from halogen; or R 1  and R 2  together with the nitrogen atom to which they are attached, form a 5-membered heterocyclyl group, which is fused to a 5- or 6-membered aryl group and which is optionally substituted by one or more substituents independently selected from C1-C3 alkyl, and wherein the resulting heterocyclic moiety is optionally substituted by one or more substituents independently selected from halogen.

Metadata:
- Claim Count in Document: 35.0
- Percentile: 98.0
- Lexical Diversity: 1.04167
- Patent Class: 514.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15317742', '11829531', '11463825', '15109101', '11909144']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7707772711769191
- 35 USC 102 Novelty (BERT): 0.5833654860190854
- Combined Prediction Score: 0.7520360926611357
- Mean Citation Score: 334.06991000000005
- Max Citation Score: 502.98242
- Similarity Product: 422.9217329779077

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test