PATENT CLAIM ANALYSIS

Application Number: 15780436
Application Type: Utility
Filing Date: 2018-05
Publication Date: 2018-12
Patent Classification: ["544", "405000"]

Abstract:
Provided is a compound (chemotherapeutic agent) effective in the prevention and treatment of hyperlipidemia, obesity, or the like. A phenylimidazole compound or a pharmaceutically acceptable salt thereof represented by the following formula (1):

Claim (Index 1):
A phenylimidazole compound represented by the following formula (1) or a pharmaceutically acceptable salt thereof wherein R1 is (1-1) hydrogen, (1-2) pyrazolyl, (1-3) pyrimidinyl, (1-4) pyridyl having one or two substituents each independently selected from the group consisting of halogen, cyano, C1-C6 alkyl, C1-C6 alkylsulfonyl, and halogen-substituted C1-C6 alkyl, (1-5) oxazolyl having one or more C1-C6 alkyl groups, (1-6) pyrazinyl optionally substituted with at least one group selected from the group consisting of halogen and C1-C6 alkyl, (1-7) phenyl having one or two substituents each independently selected from the group consisting of halogen and halogen-substituted C1-C6 alkyl, (1-8) (pyridine 1-oxide)yl having one or two substituents each independently selected from the group consisting of halogen and halogen-substituted C1-C6 alkyl, (1-9) halogen-substituted thiazolyl, (1-10) C1-C6 alkyl-substituted isoxazolyl, (1-11) C3-C8 cycloalkyl-substituted 1,2,4-oxadiazolyl, or (1-12) phenyl; R2 represents hydrogen or C1-C6 alkoxy; R3 is (3-1) hydrogen, (3-2) C1-C6 alkoxy, (3-3) C1-C6 alkoxy C1-C6 alkoxy, (3-4) C1-C6 alkyl, (3-5) halogen, (3-6) benzyloxy, or (3-7) hydroxy; R4 is (4-1) pyridyl optionally having at least one substituent selected from the group consisting of halogen, cyano, hydroxy, pyrrolidinyl, C1-C6 alkyl, C1-C6 alkylthio, C1-C6 alkylsulfonyl, C1-C6 alkoxy, and halogen-substituted C1-C6 alkyl, (4-2) C3-C10 cycloalkyl optionally having one or two substituents each independently selected from the group consisting of halogen and C1-C6 alkyl, or (4-3) lower alkyl; R5 is (5-1) hydrogen, (5-2) C1-C6 alkyl, or (5-3) C1-C6 alkoxy; R6 is (6-1) hydrogen, (6-2) C1-C6 alkoxy C1-C6 alkyl, or (6-3) C1-C6 alkyl optionally substituted with one or more C3-C10 cycloalkyl groups, wherein R6 is attached to only one of N at the 1-position and N at the 3-position of the imidazole skeleton, R6 is attached to N at the 1-position when the bond between N at the 3-position and C at the 2-position of the imidazole skeleton is a double bond, and R6 is attached to N at the 3-position when the bond between N at the 3-position and C at the 2-position of the imidazole skeleton is a single bond; R7 is (7-1) hydrogen, (7-2) halogen, (7-3) C1-C6 alkyl, (7-4) hydroxymethyl, (7-5) halogen-substituted C1-C6 alkyl, or (7-6) cyano; A is a single bond when R1 is hydrogen, and A is C1-C6 alkylene when R1 is a group other than hydrogen; in the imidazole skeleton, the bond between C at the 2-position and N at the 1-position is a single bond when the bond between N at the 3-position and C at the 2-position is a double bond, and the bond between C at the 2-position and N at the 1-position is a double bond when the bond between N at the 3-position and C at the 2-position is a single bond; with the proviso that the compound represented by formula (1) wherein R1 is a group of (1-7) or (1-12) and R4 is a group of (4-3) is excluded.

Metadata:
- Claim Count in Document: 16.0
- Percentile: 93.0
- Lexical Diversity: 1.24242
- Patent Class: 544.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['14022540', '12862418', '12738885', '13133673', '13473230']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8353831027844825
- 35 USC 102 Novelty (BERT): 0.514138936564296
- Combined Prediction Score: 0.8032586861624638
- Mean Citation Score: 331.818016
- Max Citation Score: 334.57556
- Similarity Product: 287.34347998878

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test