PATENT CLAIM ANALYSIS

Application Number: 15744510
Application Type: Utility
Filing Date: 2018-01
Publication Date: 2018-07
Patent Classification: ["514", "222800"]

Abstract:
The invention provides a compound which is a diazine of formula (I) or a tautomer thereof, or a pharmaceutically acceptable salt thereof, for use as an antifungal agent: (I) wherein X, N′, C′, A and E are as defined herein. The invention also provides a compound of Formula (I) as defined herein.

Claim (Index 8):
A compound for use according to any one of the preceding claims wherein the compound is of Formula (Ia): wherein:\n X represents S; \n R 1  represents H or C 1 -C 2  alkyl; \n E represents either:\n (i) H or C 1 -C 6  alkyl which is unsubstituted or is substituted with 1 substituent selected from halogen, and C 1 -C 2  alkoxy; and wherein the alkyl group of E is uninterrupted or is interrupted by \u2014O\u2014; or \n (ii) a C 1 -C 6  alkylene group which is bonded to an atom of group A to form a C 5 -C 6  carbocyclyl moiety which is unsubstituted or is substituted by 1 or 2 substituents selected from halogen, C 1 -C 4  alkoxy and unsubstituted C 1 -C 4  alkyl; \n A represents the group -L-T or -T; \n L is selected from C 1 -C 10  alkylene and C 2 -C 10  alkenylene, wherein the alkylene or alkenylene group is unsubstituted or is substituted by 1 or 2 groups selected from halogen, and C 1 -C 4  alkoxy, and wherein the alkylene or alkenylene group is uninterrupted or is interrupted by a heteromoiety selected from \u2014O\u2014, \u2014S\u2014, \u2014C(O)O\u2014, \u2014NR 2 \u2014, and \u2014C(O)NR 2 \u2014 and wherein the alkylene or alkenylene group optionally terminates in a heteromoiety selected from \u2014O\u2014, \u2014S\u2014, \u2014C(O)\u2014, \u2014OC(O)\u2014, \u2014C(O)O\u2014, \u2014NR 2 \u2014, \u2014NR 2 C(O)\u2014, and \u2014C(O)NR 2 \u2014, wherein R 2  represents H or methyl; \n \n when A is -L-T, then T is H or represents a 5- to 10-membered heteroaryl group or a 6- to 10-membered aryl group, and when A is -T, then T represents a 5- to 10-membered heteroaryl group or a 6- to 10-membered aryl group; wherein the aryl or heteroaryl group of T is unsubstituted or is substituted by 1 or 2 groups V; \n each group V is independently selected from C 1 -C 4  alkoxy, unsubstituted C 1 -C 4  alkyl, C 1 -C 4  alkyl which is substituted with 1, 2 or 3 halogen atoms, C 2 -C 4  alkenyl, C 2 -C 4  alkynyl, C 3 -C 6  cycloalkyl, halogen, aryl, (C 1 -C 4  alkyl)-aryl, aryloxy, aryloxy-(C 1 -C 4  alkyl), \u2014CN, NO 2 , \u2014(C 1 -C 4  alkyl)-C(O)O(C 1 -C 4  alkyl), and \u2014C(O)O(C 1 -C 4  alkyl).

Metadata:
- Claim Count in Document: 5.0
- Percentile: 86.0
- Lexical Diversity: 1.65
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['12989410', '14625532', '12601284', '11914516', '12515354']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7418770609299107
- 35 USC 102 Novelty (BERT): 0.5150181283231802
- Combined Prediction Score: 0.7191911676692376
- Mean Citation Score: 288.72395399999994
- Max Citation Score: 300.37643
- Similarity Product: 238.7668430262017

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test