PATENT CLAIM ANALYSIS

Application Number: 16045427
Application Type: Utility
Filing Date: 2018-07
Publication Date: 2019-01
Patent Classification: ["544", "113000"]

Abstract:
The invention relates to a method of manufacturing triazine, pyrimidine and pyridine derivatives of formula (I) wherein U, V, W and Z are nitrogen or carbon atoms, whereby at least one of U, V and W is nitrogen, and the other substituents are defined as in the specification, by condensing a corresponding halo-triazine, pyrimidine or pyridine in a type of Suzuki coupling with a pyridyl- or pyrimidinyl-borane, wherein the amino function is protected as a formamidine. The invention further relates to suitable intermediates and methods of manufacturing of such intermediates. Furthermore the invention relates to pure 5-(4,6-dimorpholino-1,3,5-triazin-2-yl)-4-(trifluoromethyl)pyridin-2-amine in solid form.

Claim (Index 21):
The method of  claim 20 , wherein in said compound of formula (II)\n Y 2 B represents a cyclic boronic ester; R 4  is hydrogen; and R 5  and R 6  are methyl.

Metadata:
- Claim Count in Document: 8.0
- Percentile: 95.0
- Lexical Diversity: 1.76812
- Patent Class: 544.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15304595', '14620721', '12936451', '13617035', '12016897']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7577485229736046
- 35 USC 102 Novelty (BERT): 0.5306447080293275
- Combined Prediction Score: 0.7350381414791769
- Mean Citation Score: 282.585952
- Max Citation Score: 348.9181
- Similarity Product: 300.13031943551897

Labels:
- Claim Label 101: 0
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 0

Dataset: test