PATENT CLAIM ANALYSIS

Application Number: 15767364
Application Type: Utility
Filing Date: 2018-04
Publication Date: 2018-10
Patent Classification: ["514", "210180"]

Abstract:
The present invention provides compounds of Formula (I): wherein all variables are as defined in the specification, O and compositions comprising any of such novel compounds. These compounds are APJ agonists which may be used as medicaments.

Claim (Index 7):
A compound according to  claim 3 , or a stereoisomer, an enantiomer, a diastereoisomer, a tautomer, or a pharmaceutically acceptable salt thereof, wherein:\n R 1  is independently selected from: \u2014CH 2 OH, \u2014OCH 3 , \u2014OCF 3 , OCH 2 Ph, \u2014C(\u2550O)NR a R a , \u2014NR a R a , CH 3 , CH 2 CH 3 , CH(CH 3 ) 2 , and cyclopropyl; R 2  is independently selected from: C 1-5  alkyl substituted with 0-3 R e ; C 1-5  alkenyl, phenyl substituted with 0-3 R e , 6-membered heteroaryl substituted with 0-3 R e , C 3-6  cycloalkyl and CH 2 O(CH 2 ) 1-3 CH 3 ; R 3  and R 4  are independently selected from: C 1-5  alkyl substituted with 0-3 R 6 ; \u2014(CH 2 ) n \u2014C 3-6  carbocyclyl substituted with 0-3 R 6 , and \u2014(CH 2 ) n -heterocyclyl substituted with 0-3 R 6 ; R 6  is independently selected from: H, halogen, \u2014(CH 2 ) n OR b , \u2014(CH 2 ) n NR a R a , \u2014(CH 2 ) n C(\u2550O)NR a R a , \u2014(CH 2 ) n NR a C(\u2550O)R b , \u2014(CH 2 ) n NR a C(\u2550O)OR b , \u2014(CH 2 ) n OC(\u2550O)NR a R a , \u2014(CH 2 ) n C(\u2550O)OR b , (CH 2 ) n S(O) p NR a R a , \u2014(CH 2 ) n NR a S(O) p NR a R a , C 1-5  alkyl substituted with 0-3 R e , phenyl substituted with 0-3 R e , and heterocyclyl substituted with 0-3 R e ; R a , at each occurrence, is independently selected from H, C 1-6  alkyl substituted with 0-5 R e , \u2014(CH 2 ) n -phenyl substituted with 0-5 R e , and \u2014(CH 2 ) n -heteroaryl substituted with 0-5 R e ; R b , at each occurrence, is independently selected from H, C 1-6  alkyl substituted with 0-5 R e , \u2014(CH 2 ) n \u2014C 3-10 carbocyclyl substituted with 0-5 R e , and \u2014(CH 2 ) n -heterocyclyl substituted with 0-5 R e ; R e , at each occurrence, is independently selected from C 1-6  alkyl (optionally substituted with F and Cl), OH, OCH 3 , OCF 3 , \u2014(CH 2 ) n \u2014C 3-6  cycloalkyl, \u2014(CH 2 ) n \u2014C 4-6  heterocyclyl, \u2014(CH 2 ) n -aryl, \u2014(CH 2 ) n -heteroaryl, F, Cl, Br, CN, NO 2 , \u2550O, CO 2 H; and n is independently selected from zero, 1, 2, 3, and 4.

Metadata:
- Claim Count in Document: 4.0
- Percentile: 91.0
- Lexical Diversity: 1.16216
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15468230', '15171276', '16309161', '16061365', '16340172']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7961332876686144
- 35 USC 102 Novelty (BERT): 0.5661953126233011
- Combined Prediction Score: 0.773139490164083
- Mean Citation Score: 401.784548
- Max Citation Score: 425.81107
- Similarity Product: 400.2194866677785

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test