PATENT CLAIM ANALYSIS

Application Number: 15896970
Application Type: Utility
Filing Date: 2018-02
Publication Date: 2018-08
Patent Classification: ["514", "317000"]

Abstract:
The invention provides compounds having the general formula I: and pharmaceutically acceptable salts thereof, wherein the variables R AA , n, ring A, X 1 , L, m, X 2 , R 2 , R 3 , R 4 , R 5 , X, and R 6  have the meaning as described herein, and compositions containing such compounds and methods for using such compounds and compositions.

Claim (Index 1):
A compound of Formula I: or a salt thereof; wherein each RA is independently selected from the group consisting of F, Cl, Br, I, \u2014CN, \u2014OR A1 , (X RA )-(6-12 membered aryl), \u2014(X RA )-(5-12 membered heteroaryl), and \u2014R 2 , wherein said 6-12 membered aryl and 5-12 membered heteroaryl of R AA  is optionally substituted with from 1 to 5 substitutents independently selected from the group consisting of F, Cl, Br, I, C 1-4  alkyl, C 1-4  haloalkyl, and C 1-4 (halo)alkoxy; R A1  is selected from the group consisting of hydrogen, C 1-8  alkyl, C 2-8  alkenyl, C 1-8  haloalkyl, C 3-8  cycloalkyl, phenyl and benzyl; R A2  is selected from the group consisting of C 1-8  alkyl that is optionally substituted with one or more substituents selected from oxo (\u2550O), fluoro, amino, C 1-4  alkylamino and di(C 1-4 alkyl)amino; X RA  is selected from the group consisting of absent, \u2014C(\u2550O)\u2014, and C 1-4  alkylene; wherein any C 1-4  alkylene of X RA  is optionally substituted with 1 to 3 substituents selected from the group consisting of C 1-4  alkyl, C 1-4  haloalkyl, and phenyl that is optionally substituted with 1 to 5 substitutents selected from, F, Cl, Br, I, \u2014NH 2 , \u2014OH, \u2014CN, \u2014NO 2 , C 1-4  alkyl, C 1-4  haloalkyl, C 1-4  alkoxy, C 1-4 (halo)alkoxy, C 1-4  alkylamino and C 1-4  dialkylamino; n is 0, 1, 2, 3, 4, 5, 6, 7, or 8; ring \u201cA\u201d is a 3-15 membered carbocyclyl, a 6-12 membered aryl, a 5-12 membered heteroaryl, or a 3-15 membered heterocyclyl; X 1  and X 2  are each independently selected from the group consisting of absent, \u2014S\u2014, \u2014O\u2014 and \u2014N(R X )\u2014 wherein R x  is H, C 1-8  alkyl, or C 1-8  haloalkyl, and wherein if the subscript m is 0 then one of X 1  or X 2  is absent; L is C 1-6  alkylene, wherein L is optionally substituted with from 1 to 3 substituents independently selected from the group consisting of C 1-4  alkyl, C 1-4  alkoxy, halo, oxo (\u2550O), and C 1-4  haloalkyl; wherein any two substituents attached to the same atom on L are optionally combined to form a 3- to 5-membered carbocyclic ring; m is 0 or 1; R 2 , R 3 , R 4 , and R 5  are each independently selected from the group consisting of H, F, Cl, Br, I, \u2014CN, C 1-8  alkyl, C 3-8  cycloalkyl, C 1-8  haloalkyl and C 1-8  alkoxy; X is selected from the group consisting of O, S, S\u2550O, SO 2 , N(R N ), C\u2550O, CH 2 , and C\u2550S, wherein R N  is selected from the group consisting of H, C 1-6  alkyl and acyl; ring \u201cB\u201d is selected from the group consisting of cyclobutyl, cyclopentyl, cyclohexyl, cycloheptyl, and cyclooctyl, wherein ring B is optionally substituted with one or more groups independently selected from C 1-4  alkyl; and R 6  is hydrogen or C 1-6  alkyl.

Metadata:
- Claim Count in Document: 46.0
- Percentile: 88.0
- Lexical Diversity: 1.70455
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['15321335', '14772735', '14772726', '13899469', '15799771']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8232861958288424
- 35 USC 102 Novelty (BERT): 0.5286989954918054
- Combined Prediction Score: 0.7938274757951388
- Mean Citation Score: 340.7303780000001
- Max Citation Score: 357.13367
- Similarity Product: 259.83016424994645

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test