PATENT CLAIM ANALYSIS

Application Number: 15956847
Application Type: Utility
Filing Date: 2018-04
Publication Date: 2018-08
Patent Classification: ["514", "252050"]

Abstract:
The present invention relates to azoline compounds of formula I wherein A, B 1 , B 2 , B 3 , G 1 , G 2 , X 1 , R 1 , R 3a , R 3b , R g1  and R g2  are as defined in the claims and the description. The compounds are useful for combating or controlling invertebrate pests, in particular arthropod pests and nematodes. The invention also relates to a method for controlling invertebrate pests by using these compounds and to plant propagation material and to an agricultural and a veterinary composition comprising said compounds.

Claim (Index 25):
A method for treating or protecting an animal from infestation or infection by invertebrate pests, which method comprises contacting the animal with a parasiticidally or pesticidally effective amount of at least one compound of the formula I: or an N-oxide, stereoisomer or veterinarily acceptable salt thereof; wherein X 1  is O or CH 2 ; A is a group of following formula: wherein # denotes the bond to the aromatic ring of formula (I); W is selected from O and S; Y is selected from hydrogen, \u2014N(R 5 )R 6  and \u2014OR 9 ; B 1 , B 2  and B 3  are each independently CR 2 ; G 1  and G 2  are each independently CR 4 ; R g1  and R g2  form together a bridging group selected from \u2014CH 2 CH 2 CH 2 CH 2 \u2014 and \u2014CH 2 CH 2 CH 2 \u2014; R 1  is CF 3 ; each R 2  is independently selected from the group consisting of hydrogen, halogen, C 1 -C 2 -haloalkoxy and C 1 -C 2 -haloalkyl; R 3a , R 3b  are each independently selected from the group consisting of hydrogen, halogen, hydroxyl, \u2014CO 2 R 3d , C 1 -C 3 -alkyl, C 1 -C 3 -haloalkyl, C 2 -C 3 -alkenyl, C 2 -C 3 -alkynyl, C 1 -C 3 -alkoxy, C 1 -C 3 -haloalkoxy, C 1 -C 3 -alkylthio, C 1 -C 3 -haloalkylthio, C 1 -C 3 -alkylsulfonyl and C 1 -C 3 -haloalkylsulfonyl; or\n R 3a  and R 3b  together form a group \u2550O, \u2550C(R 3c ) 2 , \u2550NOH or \u2550NOCH 3 ; \n each R 3c  is independently selected from the group consisting of hydrogen, halogen, CH 3  and CF 3 ; R 3d  is selected from the group consisting of hydrogen, C 1 -C 6 -alkyl and C 1 -C 3 -alkyloxy-C 1 -C 3 -alkyl-; each R 4  is independently selected from the group consisting of hydrogen, halogen and cyano; R 5  selected from hydrogen, C 1 -C 6 -alkyl, C 2 -C 3 -alkynyl and CH 2 \u2014CN; R 6  is selected from hydrogen, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, C 1 -C 4 -alkyl which carries one radical R 8 , C 2 -C 6 -alkenyl, C 2 -C 6 -haloalkenyl, C 2 -C 6 -alkynyl, C 3 -C 6 -cycloalkyl which may be substituted by 1 or 2 substituents selected from F, CN and pyridyl;\n \u2014N(R 101a )R 101b ,\n wherein \n R 101a  is selected from hydrogen and C 1 -C 6 -alkyl; and \n R 101b  is selected from hydrogen, \u2014C(\u2550O)N(R 14a )R 14b , wherein\n R 14a  is selected from the group consisting of hydrogen and C 1 -C 6 -alkyl; and \n R 14b  is selected from the group consisting of hydrogen, C 1 -C 6 -alkyl, C 2 -C 4 -alkynyl, CH 2 \u2014CN, C 1 -C 6 -haloalkyl, C 3 -C 6 -cycloalkyl, C 3 -C 6 -halocycloalkyl, C 1 -C 4 -alkoxy and C 1 -C 4 -haloalkoxy; \n phenyl, optionally substituted with 1, 2, 3, 4 or 5 substituents R 16 , and a heterocyclic ring selected from rings of formulae E-1 to E-42 \n \n \n where in these rings E-1 to E-42 as a meaning for R 101b  the zigzag line denotes the attachment point to the remainder of the molecule; \u2003k is 0, 1, 2 or 3, and each R 16  is independently selected from the group consisting of halogen, cyano, nitro, C 1 -C 4 -alkyl, C 1 -C 4 -haloalkyl, C 1 -C 4 -alkoxy, C 1 -C 4 -haloalkoxy, C 1 -C 4 -alkylthio, C 1 -C 4 -haloalkylthio, C 1 -C 4 -alkylsulfinyl, C 1 -C 4 -haloalkylsulfinyl, C 1 -C 4 -alkylsulfonyl, C 1 -C 4 -haloalkylsulfonyl, C 3 -C 6 -cycloalkyl, C 3 -C 6 -halocycloalkyl, C 2 -C 4 -alkenyl, C 2 -C 4 -haloalkenyl, C 2 -C 4 -alkynyl, C 2 -C 4 -haloalkynyl, C 1 -C 4 -alkylcarbonyl, C 1 -C 4 -haloalkylcarbonyl, aminocarbonyl, C 1 -C 4 -alkylaminocarbonyl and di-(C 1 -C 4 -alkyl)aminocarbonyl; CH\u2550NOR 9a , wherein R 9a  is selected from hydrogen, C 1 -C 6 -alkyl and C 1 -C 6 -haloalkyl; phenyl which may be substituted with 1, 2, 3, 4, or 5 substituents R 11 , and a 3-, 4-, 5- or 6-membered saturated, partially unsaturated or maximally unsaturated heteromonocyclic ring containing 1, 2 or 3 heteroatoms or heteroatom groups independently selected from N, O, S, NO, SO and SO 2 , as ring members, where the heteromonocyclic ring may be substituted with one or more substituents R 11 ; wherein each R 11  is independently selected from the group consisting of halogen, cyano, nitro, C 1 -C 4 -alkyl, C 1 -C 4 -haloalkyl, C 1 -C 4 -alkoxy, C 1 -C 4 -haloalkoxy, C 1 -C 4 -alkylthio, C 1 -C 4 -haloalkylthio, C 3 -C 6 -cycloalkyl, C 3 -C 6 -halocycloalkyl, C 2 -C 4 -alkenyl, C 2 -C 4 -haloalkenyl, C 2 -C 4 -alkynyl and C 2 -C 4 -haloalkynyl; or\n two R 11  present on the same carbon atom of a saturated heterocyclic ring may form together \u2550O or \u2550S; or \n two R 11  present on the same S or SO ring member of a heterocyclic ring may together form a group \u2550N(C 1 -C 6 -alkyl), \u2550NO(C 1 -C 6 -alkyl), \u2550NN(H)(C 1 -C 6 -alkyl) or \u2550NN(C 1 -C 6 -alkyl) 2 ; \n each R 8  is independently selected from OH, CN, C 3 -C 8 -cycloalkyl which optionally carries a CN or a C 1 -C 2 -haloalkyl substituent; C 3 -C 8 -halocycloalkyl, C 1 -C 6 -alkoxy, C 1 -C 6 -haloalkoxy, C 1 -C 6 -alkylthio, C 1 -C 6 -haloalkylthio, C 1 -C 6 -alkylsulfonyl, C 1 -C 6 -haloalkylsulfonyl, \u2014C(\u2550O)N(R 102a )R 102b , phenyl, optionally substituted with 1, 2, 3, 4 or 5 substituents R 16 , and a 3-, 4-, 5- or 6-membered saturated, partially unsaturated or maximally unsaturated heteromonocyclic ring containing 1, 2, 3 or 4 heteroatoms or heteroatom groups independently selected from N, O, S, NO, SO and SO 2 , as ring members, where the heteromonocyclic ring may be substituted with one or more substituents R 16 ;\n wherein \n R 102a  is selected from the group consisting of hydrogen, C 1 -C 6 -alkyl, C 2 -C 3 -alkynyl and CH 2 \u2014CN; \n R 102b  is selected from the group consisting of hydrogen, C 1 -C 6 -alkyl, C 2 -C 4 -alkenyl, C 2 -C 4 -alkynyl, CH 2 \u2014CN, C 1 -C 6 -haloalkyl, C 3 -C 6 -cycloalkyl, C 3 -C 6 -halocycloalkyl, C 3 -C 6 -cycloalkylmethyl, C 1 -C 6 -alkoxy, C 1 -C 6 -haloalkoxy, phenyl which is optionally substituted with 1, 2, 3, 4 or 5 substituents selected from the group consisting of halogen, cyano, nitro, C 1 -C 4 -alkyl, C 1 -C 4 -haloalkyl, C 2 -C 4 -alkenyl, C 2 -C 4 -haloalkenyl, C 2 -C 4 -alkynyl, C 2 -C 4 -haloalkynyl, C 3 -C 6 -cycloalkyl, C 3 -C 6 -halocycloalkyl, C 1 -C 4 -alkoxy, C 1 -C 4 -haloalkoxy, C 1 -C 4 -alkylthio and C 1 -C 4 -haloalkylthio; and a heterocyclic ring selected from rings of formulae E-1 to E-42 as defined above and E-43 to E-57: \n where in these rings E-43 to E-57 the zigzag line denotes the attachment point to the remainder of the molecule; \u2003k is 0, 1, 2 or 3, n is 0, 1 or 2; and each R 16  is independently selected from the group consisting of halogen, cyano, nitro, C 1 -C 4 -alkyl, C 1 -C 4 -haloalkyl, C 1 -C 4 -alkoxy, C 1 -C 4 -haloalkoxy, C 1 -C 4 -alkylthio, C 1 -C 4 -haloalkylthio, C 1 -C 4 -alkylsulfinyl, C 1 -C 4 -haloalkylsulfinyl, C 1 -C 4 -alkylsulfonyl, C 1 -C 4 -haloalkylsulfonyl, C 3 -C 6 -cycloalkyl, C 3 -C 6 -halocycloalkyl, C 2 -C 4 -alkenyl, C 2 -C 4 -haloalkenyl, C 2 -C 4 -alkynyl, C 2 -C 4 -haloalkynyl, C 1 -C 4 -alkylcarbonyl, C 1 -C 4 -haloalkylcarbonyl, aminocarbonyl, C 1 -C 4 -alkylaminocarbonyl and di-(C 1 -C 4 -alkyl)aminocarbonyl; or two R 16  present on the same carbon atom of a saturated ring may form together \u2550O or \u2550S; and each R 16  as a substituent on phenyl (as a meaning of R 8 ) or the heterocyclic rings (as a meaning of R 8 ) is independently selected from the group consisting of halogen, cyano, nitro, C 1 -C 4 -alkyl, C 1 -C 4 -haloalkyl, C 1 -C 4 -alkoxy, C 1 -C 4 -haloalkoxy, C 1 -C 4 -alkylthio, C 1 -C 4 -haloalkylthio, C 3 -C 6 -cycloalkyl, C 3 -C 6 -halocycloalkyl, C 2 -C 4 -alkenyl, C 2 -C 4 -haloalkenyl, C 2 -C 4 -alkynyl and C 2 -C 4 -haloalkynyl; or\n two R 16  present on the same carbon atom of a saturated heterocyclic ring may form together \u2550O or \u2550S; or \n two R 16  present on the same S or SO ring member of a heterocyclic ring may together form a group \u2550N(C 1 -C 6 -alkyl), \u2550NO(C 1 -C 6 -alkyl), \u2550NN(H)(C 1 -C 6 -alkyl) or \u2550NN(C 1 -C 6 -alkyl) 2 ; \n or R 5  and R 6 , together with the nitrogen atom to which they are bound, form a 5- or 6-membered saturated heterocyclic ring, where the ring may further contain 1 or 2 heteroatoms or heteroatom-containing groups selected from O, S, SO, SO 2 , NH and C\u2550O as ring members, wherein the heterocyclic ring may be substituted with 1, 2 or 3 substituents independently selected from the group consisting of halogen, cyano, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, C 1 -C 6 -alkoxy and C 1 -C 6 -haloalkoxy; or R 5  and R 6  together form a group \u2550S(R 9b ) 2 , where R 9b  is selected from C 1 -C 6 -alkyl and C 1 -C 6 -haloalkyl; R 9  is selected from the group consisting of hydrogen, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl and C 1 -C 6 -alkyl substituted by one radical R 13 ; where R 13  is selected from CN, C 1 -C 6 -alkoxy, C 1 -C 6 -haloalkoxy, C 1 -C 6 -alkylthio, C 1 -C 6 -haloalkylthio, C 1 -C 6 -alkylsulfinyl, C 1 -C 6 -haloalkylsulfinyl, C 1 -C 6 -alkylsulfonyl, C 1 -C 6 -haloalkylsulfonyl and a heterocyclic ring selected from rings of formulae E-1 to E-57 as defined above;\n where in these rings E-1 to E-57 as a meaning of R 13  \n the zigzag line denotes the attachment point to the remainder of the molecule; \n k is 0, 1, 2 or 3, \n n is 0, 1 or 2; and \n each R 16  is independently selected from the group consisting of halogen, cyano, nitro, C 1 -C 4 -alkyl, C 1 -C 4 -haloalkyl, C 1 -C 4 -alkoxy, C 1 -C 4 -haloalkoxy, C 1 -C 4 -alkylthio, C 1 -C 4 -haloalkylthio, C 1 -C 4 -alkylsulfinyl, C 1 -C 4 -haloalkylsulfinyl, C 1 -C 4 -alkylsulfonyl, C 1 -C 4 -haloalkylsulfonyl, C 3 -C 6 -cycloalkyl, C 3 -C 6 -halocycloalkyl, C 2 -C 4 -alkenyl, C 2 -C 4 -haloalkenyl, C 2 -C 4 -alkynyl, C 2 -C 4 -haloalkynyl, C 1 -C 4 -alkylcarbonyl, C 1 -C 4 -haloalkylcarbonyl, aminocarbonyl, C 1 -C 4 -alkylaminocarbonyl and di-(C 1 -C 4 -alkyl)aminocarbonyl; or\n two R 16  present on the same carbon atom of a saturated ring may form together \u2550O or \u2550S; and \n \n each R 16  in all other cases is independently selected from the group consisting of halogen, nitro, cyano, \u2014OH, \u2014SH, C 1 -C 6 -alkoxy, C 1 -C 6 -haloalkoxy, C 1 -C 6 -alkylthio, C 1 -C 6 -haloalkylthio, C 1 -C 6 -alkylsulfinyl, C 1 -C 6 -haloalkylsulfinyl, C 1 -C 6 -alkylsulfonyl, C 1 -C 6 -haloalkylsulfonyl, C 1 -C 4 -alkylcarbonyl, C 1 -C 4 -haloalkylcarbonyl, C 1 -C 4 -alkoxycarbonyl, C 1 -C 4 -haloalkoxycarbonyl, aminocarbonyl, C 1 -C 4 -alkylaminocarbonyl, di-(C 1 -C 4 -alkyl)-aminocarbonyl, trimethylsilyl, triethylsilyl, tert-butyldimethylsilyl;\n C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, wherein the three last-mentioned aliphatic radicals may be unsubstituted, partially or fully halogenated and/or may carry 1 or 2 radicals selected from cyano, C 3 -C 4 -cycloalkyl, C 1 -C 4 -alkoxy, C 1 -C 4 -haloalkoxy and oxo; \n C 3 -C 8 -cycloalkyl which may be unsubstituted, partially or fully halogenated and/or may carry 1 or 2 radicals selected from cyano, C 1 -C 4 -alkyl, C 3 -C 4 -cycloalkyl, C 1 -C 4 -alkoxy, C 1 -C 4 -haloalkoxy and oxo; \n phenyl, benzyl, pyridyl and phenoxy, wherein the four last mentioned radicals may be unsubstituted, partially or fully halogenated and/or carry 1, 2 or 3 substituents selected from C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, C 1 -C 6 -alkoxy, C 1 -C 6 -haloalkoxy and (C 1 -C 6 -alkoxy)carbonyl; \n or \n two R 16  present together on the same atom of an unsaturated or partially unsaturated ring may be \u2550O, \u2550S, \u2550N(C 1 -C 6 -alkyl), \u2550NO(C 1 -C 6 -alkyl), \u2550CH(C 1 -C 4 -alkyl) or \u2550C(C 1 -C 4 -alkyl)C 1 -C 4 -alkyl; or \n or two R 16  present on the same S or SO ring member of a heterocyclic ring may together form a group \u2550N(C 1 -C 6 -alkyl), \u2550NO(C 1 -C 6 -alkyl), \u2550NN(H)(C 1 -C 6 -alkyl) or \u2550NN(C 1 -C 6 -alkyl) 2 ; \n or \n two R 16  on two adjacent carbon atoms form together with the carbon atoms they are bonded to a 4-, 5-, 6-, 7- or 8-membered saturated, partially unsaturated or maximally unsaturated ring, wherein the ring may contain 1 or 2 heteroatoms or heteroatom groups selected from N, O, S, NO, SO and SO 2 , as ring members, and wherein the ring optionally carries one or more substituents selected from halogen, C 1 -C 4 -alkyl, C 1 -C 4 -haloalkyl, C 1 -C 4 -alkoxy and C 1 -C 4 -haloalkoxy.

Metadata:
- Claim Count in Document: 62.0
- Percentile: 91.0
- Lexical Diversity: 1.81034
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['15121493', '14757930', '14366161', '14757414', '15539009']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8283296619567898
- 35 USC 102 Novelty (BERT): 0.5649785263342119
- Combined Prediction Score: 0.8019945483945321
- Mean Citation Score: 417.83641
- Max Citation Score: 462.4929
- Similarity Product: 337.3093142307758

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test