PATENT CLAIM ANALYSIS

Application Number: 15767328
Application Type: Utility
Filing Date: 2018-04
Publication Date: 2018-10
Patent Classification: ["514", "236200"]

Abstract:
The disclosure provides compounds of formula (I) or pharmaceutically acceptable salts thereof: The disclosure also provides processes for their preparation, intermediates used in these processes, pharmaceutical compositions containing them, and their use as modulators of dopamine D 3  receptors, such as treating substance abuse or psychiatric diseases.

Claim (Index 1):
A compound of formula (I) or a pharmaceutically acceptable salt thereof: wherein: G is aryl or a 5-6 membered heteroaromatic group or 8-11 membered heteroaromatic group, which may be benzofused or optionally substituted by 1, 2, 3 or 4 substituents selected from the group consisting of: halogen, cyano, hydroxyl, amino, C 1-4 alkylamino, C 1-4 alkyl, haloC 1-4 alkyl, C 1 -4alkoxy, haloC 1-4 alkoxy, C 1-4 alkanoyl, SF 5 , C(\u2550O)NH 2 , C(\u2550O)OR 4 ; W is S, SO 2 , O, CHR 2 , NR 4 ; n is 0 or 1; m is 1 or 2; p is 0, 1 or 2; q is 0 or 1; z is an integer ranging from 1 to 7; R is independently hydrogen or C 1-4 alkyl; R 1  is hydrogen, C 1-4 alkyl; C 1-4 alkoxy; R 2  is hydrogen, F, C 1-4 alkyl; OH, C 1-4 alkoxy; R 3  is hydrogen, F, C 1-4 alkyl; OH, C 1-4 alkoxy; R 4  is hydrogen, C 1-4 alkyl; G 1  is a phenyl group or a 5-6-membered heteroaromatic group or a 8-11 membered heteroaromatic group, any of which groups may be optionally substituted by 1, 2, 3 or 4 substituents selected from the group consisting of: halogen, cyano, hydroxyl, amino, C 1-4 alkylamino, C 1-4 alkyl, haloC 1-4 alkyl, C 1-4 alkoxy, C 1-4 alkanoyl, SF 5 , C(\u2550O)NH 2 , C(\u2550O)OR 4 ; Y is H or a moiety selected from the group consisting of: 5-6 membered heteroaromatic group, saturated mono 3-7 membered carbocyclic group or 8-11 membered bicyclic carbocyclic group in which one or more atom carbons may be replaced by NR 4 , O, S; any of which groups may be optionally substituted by one or two substituents selected from: halogen, cyano, hydroxyl, amino, C 1-4 alkylamino, C 1-4 alkyl, haloC 1-4 alkyl, C 1-4 alkoxy, haloC 1-4 alkoxy, C 1-4 alkanoyl, SF 5 , C(\u2550O)NH 2 , SO 2 NH 2 , C(\u2550O)O x R 4  wherein x is 0 or 1, or Y\u2032; and Y\u2032 is phenyl, or a 5-6-membered heteroaromatic group optionally substituted by 1 or 2 R 2  groups; with the proviso that n is 0 when q is 0.

Metadata:
- Claim Count in Document: 35.0
- Percentile: 91.0
- Lexical Diversity: 1.25
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15522863', '15750128', '11911035', '11570623', '11569880']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8247422855537362
- 35 USC 102 Novelty (BERT): 0.5447364239719118
- Combined Prediction Score: 0.7967416993955538
- Mean Citation Score: 334.188548
- Max Citation Score: 398.69064
- Similarity Product: 362.2057237146664

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test