PATENT CLAIM ANALYSIS

Application Number: 16119445
Application Type: Utility
Filing Date: 2018-08
Publication Date: 2018-12
Patent Classification: ["546", "300000"]

Abstract:
The present invention relates to a compound of formula (I), or a tautomer and/or a pharmaceutically acceptable salt thereof, wherein R 1  is alkyl, Cl, F or Br, R 2  is H or F; R 3  is selected from H and alkyl; R 4  is selected from H and C(O)R 6 ; R 5  is H or R 4  and R 5  are linked to form a heterocyclic group which is optionally substituted with one or more R 10  groups R 6  is selected from R 7 , OR 7  and NR 8 R 6 ; R 7 R 8  and R 9  are each independently selected from alkyl, cycloalkyl, aralkyl, cycloalkenyl, heterocycyl and aryl, each of which is optionally substituted with one or more R 10  groups; each R 10  is independently selected from halogen. OH, CN NO 2 , COO-alkyl, aralkyl, SO 2 -alkyl, SO 2 -aryl, COOH, CO-alkyl, CO-aryl, NH 2 , NH-alkyl, N(alkyl) 2 , CF 3 , alkyl and alkoxy, X and Z are each independently CR 11  and Y is selected from CR 11  and N and R 11  is H or F; for use in treating a disorder associated with protein misfolding stress and in particular associated with accumulation of misfolded proteins.

Claim (Index 9):
The method according to  claim 1  wherein R 4  and R 5  are linked to form a heterocyclic group which is optionally substituted with one or more R 10  groups.

Metadata:
- Claim Count in Document: 1.0
- Percentile: 96.0
- Lexical Diversity: 2.44
- Patent Class: 546.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15467613', '14760350', '15316797', '15749485', '13806602']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8234644802800667
- 35 USC 102 Novelty (BERT): 0.6358739389012
- Combined Prediction Score: 0.8047054261421801
- Mean Citation Score: 434.217756
- Max Citation Score: 622.9989
- Similarity Product: 563.4504855900942

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test