PATENT CLAIM ANALYSIS

Application Number: 15935120
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2019-09
Patent Classification: ["514", "211120"]

Abstract:
Novel heterocyclic fused systems are disclosed herein which possess numerous biological activities, including but not limited to antibacterial activity, and usefulness to the treatment of many disease states, such as pathogenic infections. In particular, new imidazoles are disclosed along with related processes of preparation and methods of use as antibacterial agents. The disclosed compounds were found to be active against several Gram-positive bacteria, including  Enterococcus faecalis  and  Bacillus subtilis , and were also found to be active against several species of multi-drug resistant  Staphylococcus , such as  S. aureus, S. saprophyticus, S. haemolyticus , and  S. epidermidis.

Claim (Index 14):
A compound having the following general formula: wherein: is a 5, 6, or 7 membered heteroaryl or heteroalicyclic ring that is either unsubstituted or substituted with 1, 2, 3, or 4 substituents independently selected from the group consisting of: a halogen atom, CN, R 3 , OR 3 , SR 3 , N(R 3 ) 2 , C(O)R 3 , C(O)OR 3 , NR 3 C(O)R 3 , C(O)NR 3 , SO 2 R 3 , NR 3 SO 2 R 3 , and SO 2 N(R 3 ) 2 ; n=1, 2, 3 and ring B has 6, 7, or 8 members; R 1  is hydrogen or an unsubstituted or substituted alkyl, aryl, or heteroaryl group; R 2  is selected from the group consisting of: C(O)OR 3 , CN, N(R 3 ) 2 , C(O)R 3 , C(O)NR 3 , SO 2 R 3 , SO 2 N(R 3 ) 2 , and PO 2 R 3 ; and is a 5, 6, or 7 membered aryl or heteroaryl ring that is either unsubstituted or substituted with 1, 2, 3, or 4 substituents independently selected from the group consisting of: a halogen atom, CN, \u2014R 3 , OR 3 , SR 3 , N(R 3 ) 2 , C(O)R 3 , C(O)OR 3 , NR 3 C(O)R 3 , C(O)NR 3 , SO 2 R 3 , NR 3 SO 2 R 3 , and SO 2 N(R 3 ) 2 , or a pharmaceutically acceptable salt, pro-drug, or derivative thereof.

Metadata:
- Claim Count in Document: 20.0
- Percentile: 90.0
- Lexical Diversity: 1.55072
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['14902004', '15107531', '15897571', '15023413', '15301270']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7970616105359783
- 35 USC 102 Novelty (BERT): 0.5260473637658817
- Combined Prediction Score: 0.7699601858589686
- Mean Citation Score: 321.87749599999995
- Max Citation Score: 331.52615
- Similarity Product: 267.5191687190353

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test