PATENT CLAIM ANALYSIS

Application Number: 16117107
Application Type: Utility
Filing Date: 2018-08
Publication Date: 2018-12
Patent Classification: ["514", "341000"]

Abstract:
The present invention provides compounds of Formula (I): a stereoisomer, a tautomer, a pharmaceutically acceptable salt, a polymorph, a solvate thereof, wherein all of the variables are as defined herein. These compounds are monoacylglycerol acyltransferase type 2 (MGAT2) inhibitors which may be used as medicaments.

Claim (Index 2):
A compound according to  claim 1 , wherein:\n R 1  is independently selected from: (C 3-6  carbocycle substituted with 0-2 R b  and 0-2 R g ), and (a 5- to 6-membered heteroaryl comprising carbon atoms and 1-4 heteroatoms selected from N, NR e , O and S; wherein said heteroaryl is substituted with 0-1 R b  and 0-2 R g ); R 3  is independently selected from: H, F, C 1-4  alkyl and CN; R 4  is independently selected from: H, F, and C 1-4  alkyl; R b  is, at each occurrence, independently selected from: halogen, C 1-10  alkyl, C 1-10  alkoxy, C 1-10  haloalkyl, C 1-10  haloalkoxy, C 1-10  alkylthio, C 1-10  haloalkylthio, N(C 1-4  alkyl) 2 , \u2014CONH(C 4-20  alkyl), \u2014CONH(C 4-20  haloalkyl), \u2014O(CH 2 ) s O(C 1-6  alkyl), \u2014O(CH 2 ) s O(C 1-6  haloalkyl), R c , and \u2014(CH 2 ) n \u2014(O) t \u2014(CH 2 ) m R c ; and R d  is, at each occurrence, independently selected from: halogen, C 1-4  alkyl, C 1-4  alkoxy, C 1-4  haloalkyl, C 1-4  haloalkoxy, tetrazolyl, OBn and phenyl.

Metadata:
- Claim Count in Document: 56.0
- Percentile: 96.0
- Lexical Diversity: 1.35714
- Patent Class: 514.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['15866871', '15123773', '15602515', '15618182', '15123791']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8155585821022441
- 35 USC 102 Novelty (BERT): 0.5656015266897099
- Combined Prediction Score: 0.7905628765609907
- Mean Citation Score: 398.53599
- Max Citation Score: 441.1919
- Similarity Product: 424.7583247186183

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test