PATENT CLAIM ANALYSIS

Application Number: 15779435
Application Type: Utility
Filing Date: 2018-05
Publication Date: 2018-09
Patent Classification: ["514", "235800"]

Abstract:
The present invention relates to a novel imidazole compound or a pharmaceutically acceptable salt thereof having a melanocortin receptor agonistic activity, and medical use thereof. The present invention relates to an imidazole compound represented by general formula [I] [wherein: Ring A represents an optionally substituted aryl group or the like; R 1  represents a hydrogen atom, an optionally substituted alkyl group, or the like; R 2  represents a hydrogen atom, a halogen atom, or the like; and R 3  represents an optionally substituted alkyl group] or a pharmaceutically acceptable salt thereof.

Claim (Index 10):
A compound selected from the group consisting of\n 1-(2-{[2-({[(3R,4R)-4-(2,4-difluorophenyl)-3-fluoro-1-(4-methoxy-4-methylpentyl)pyrrolidin-3-yl]carbonyl}amino)-1H-imidazol-1-yl]methyl}-5-methylphenyl)piperidine-4-carboxylic acid; 1-[2-{[2-({[(3R,4R)-4-(2,4-difluorophenyl)-3-fluoro-1-(pentan-3-yl)pyrrolidin-3-yl]carbonyl}amino)-1H-imidazol-1-yl]methyl}-5-(trifluoromethyl)phenyl]piperidine-4-carboxylic acid; 1-[2-{[2-({[(3R,4R)-1-cyclopentyl-4-(2,4-difluorophenyl)-3-fluoropyrrolidin-3-yl]carbonyl}amino)-1H-imidazol-1-yl]methyl}-5-(trifluoromethyl)phenyl]piperidine-4-carboxylic acid; 1-[2-{[2-({[(3R,4R)-4-(2,4-difluorophenyl)-3-fluoro-1-(4-methoxy-4-methylpentyl)pyrrolidin-3-yl]carbonyl}amino)-1H-imidazol-1-yl]methyl}-5-(trifluoromethyl)phenyl]piperidine-4-carboxylic acid; 1-[2-({2-[({(3R,4R)-4-(2,4-difluorophenyl)-3-fluoro-1-[3-(pyrrolidin-1-ylsulfonyl)propyl]pyrrolidin-3-yl}carbonyl)amino]-1H-imidazol-1-yl}methyl)-5-(trifluoromethyl)phenyl]piperidine-4-carboxylic acid; 1-[2-{[2-({[(3R,4R)-1-tert-butyl-4-(2,4-difluorophenyl)-3-fluoropyrrolidin-3-yl]carbonyl}amino)-1H-imidazol-1-yl]methyl}-5-(trifluoromethyl)phenyl]piperidine-4-carboxylic acid; 1-[2-{[2-({[(3R,4R)-1-tert-butyl-3-fluoro-4-(4-fluorophenyl)pyrrolidin-3-yl]carbonyl}amino)-1H-imidazol-1-yl]methyl}-5-(trifluoromethyl)phenyl]piperidine-4-carboxylic acid; 1-[2-{[2-({[(3R,4R)-1-tert-butyl-3-fluoro-4-(4-fluorophenyl)pyrrolidin-3-yl]carbonyl}amino)-1H-imidazol-1-yl]methyl}-5-(propan-2-yl)phenyl]piperidine-4-carboxylic acid; 1-[2-{[2-({[(3R,4R)-1-tert-butyl-3-fluoro-4-(4-methoxyphenyl)pyrrolidin-3-yl]carbonyl}amino)-1H-imidazol-yl]methyl}-5-(trifluoromethyl)phenyl]piperidine-4-carboxylic acid; and 1-[2-{[2-({[(3R,4R)-1-tert-butyl-3-fluoro-4-(4-methoxyphenyl)pyrrolidin-3-yl]carbonyl}amino)-1H-imidazol-1-yl]methyl}-5-(propan-2-yl)phenyl]piperidine-4-carboxylic acid or a pharmaceutically acceptable salt thereof.

Metadata:
- Claim Count in Document: 42.0
- Percentile: 93.0
- Lexical Diversity: 2.03846
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15313407', '15305587', '13154144', '12919973', '14891845']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7692878742346417
- 35 USC 102 Novelty (BERT): 0.5664390922094193
- Combined Prediction Score: 0.7490029960321195
- Mean Citation Score: 313.940092
- Max Citation Score: 427.80472
- Similarity Product: 406.8874881024122

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test