PATENT CLAIM ANALYSIS

Application Number: 15748027
Application Type: Utility
Filing Date: 2018-01
Publication Date: 2018-08
Patent Classification: ["548", "307400"]

Abstract:
The present invention relates to a method for preparing substituted 3-(2-anilino-1-cyclohexyl-1H-benzimidazol-5-yl)propanoic acid derivatives of the general formula (I) in which R 1  represents a hydrogen atom or R 1  represents a group selected from the series of C 1 -C 3 -alkyl-, C 1 -C 3 -alkoxy-, C 1 -C 3 -haloalkyl- and C 1 -C 3 -haloalkoxy-, R 2  represents a hydrogen atom or a C 1 -C 3 -alkyl group, R 3  represents a hydrogen atom or a C 1 -C 3 -alkyl group, R 4  represents a cyclohexyl group, which is optionally singly or multiply substituted by a C 1 -C 3 -alkyl group, and R 5  represents a hydrogen atom or a C 1 -C 6 -alkyl group; and also intermediates which may be used to prepare substituted 3-(2-anilino-1-cyclohexyl-1H-benzimidazol-5-yl)propanoic acid derivatives. The present invention also relates to a crystalline form of 3-(2-{[4-(trifluoromethoxy)phenyl]amino}-1-[(1R,5R)-3,3,5-trimethylcyclohexyl]-1H-benzimidazol-5-yl)propanoic acid, pharmaceutical compositions comprising this crystalline form, and also the use of this crystalline form for preparing a medicament for the treatment of a disease.

Claim (Index 2):
The method according to  claim 1 , wherein R 2  is a hydrogen atom, R 3  is a hydrogen atom and R 1  represents a group selected from the group consisting of C 1 -C 3 -alkyl-, C 1 -C 3 -alkoxy-, C 1 -C 3 -haloalkyl- and C 1 -C 3 -haloalkoxy-.

Metadata:
- Claim Count in Document: 11.0
- Percentile: 86.0
- Lexical Diversity: 2.52941
- Patent Class: 548.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15744641', '15118154', '15748014', '15118157', '15742363']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8071318771261228
- 35 USC 102 Novelty (BERT): 0.60693685543131
- Combined Prediction Score: 0.7871123749566415
- Mean Citation Score: 468.837484
- Max Citation Score: 542.7752
- Similarity Product: 486.8758004559517

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test