PATENT CLAIM ANALYSIS

Application Number: 15893341
Application Type: Utility
Filing Date: 2018-02
Publication Date: 2018-11
Patent Classification: ["546", "193000"]

Abstract:
Compounds of formula I that modulate or inhibit the enzymatic activity of indoleamine 2,3-dioxygenase, pharmaceutical compositions including such compounds and methods of treating diseases, conditions or disorders utilizing such compounds and compositions.

Claim (Index 1):
A compound of formula I wherein:\n X is N or CR; \n Y is N or CR; \n Y 1  is N or C; \n R is H, halogen, optionally substituted C1-C3 alkyl or optionally substituted C1-C3 alkoxy; \n X 1  is selected from CH 2 , O, S or NR 1 , where R 1  is H or C1-C3 alkyl; \n n is selected from 1, 2 or 3; \n R 2  and R 3  independently is H or C1-C2-alkyl or together with the carbon to which they are attached to form is C3-C4 cycloalkyl; \n R 4  is \u2014CONHR 5 , \u2014CSNHR 5 , C(\u2550NH)NHR 5 , \u2014SO 2 R 6 , \u2014COR 6 , optionally substituted C1-C6 alkyl, optionally substituted C3-C8 heteroaryl, optionally substituted C3-C8 alkylheteroaryl, optionally substituted C3-C8 alkoxylheteroaryl, optionally substituted C3-C8 heterocycle, optionally substituted C3-C8 alkylheterocycle or optionally substituted C3-C8 alkoxyheterocycle; \n R 5  is optionally substituted C1-C6 alkyl, optionally substituted C2-C6 alkenyl, optionally substituted C2-C6 alkynyl, optionally substituted C3-C7 cycloalkyl, or optionally substituted C4-C7 cycloalkenyl; optionally substituted aryl, optionally substituted C7-C10 alkylaryl, optionally substituted C7-C10 alkoxyaryl, optionally substituted C3-C10 heteroaryl, optionally substituted C3-10-alkyl heteroaryl or C3-C8 heterocycle; and \n R 6  is CF 3 , optionally substituted C1-C5 alkyl, optionally substituted aryl, optionally substituted C7-C10 alkylaryl, optionally substituted C7-C10 alkoxyaryl, optionally substituted C3-C10 heteroaryl, optionally substituted C3-10-alkyl heteroaryl or C3-C8 heterocycle.

Metadata:
- Claim Count in Document: 28.0
- Percentile: 88.0
- Lexical Diversity: 1.2963
- Patent Class: 546.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['13780510', '11641284', '15613361', '14795466', '15698788']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7360763502220216
- 35 USC 102 Novelty (BERT): 0.49983909240359
- Combined Prediction Score: 0.7124526244401784
- Mean Citation Score: 242.17147600000004
- Max Citation Score: 245.82295
- Similarity Product: 188.6435272993237

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test