PATENT CLAIM ANALYSIS

Application Number: 16106104
Application Type: Utility
Filing Date: 2018-08
Publication Date: 2019-02
Patent Classification: ["514", "301000"]

Abstract:
The present invention is directed to 5-fluoro-C-(aryl or hetercyclyl)-glycoside derivatives, pharmaceutical compositions containing them and their use in the treatment of disorders and conditions modulated by SGLT activity, more particularly dual SGLT1/2 activity.

Claim (Index 12):
A compound as in  claim 4 , selected from the group consisting of\n (2S,3R,4R,5S,6R)-2-(7-((2,3-dihydrobenzo[b][1,4]dioxin-6-yl)methyl)-4-methoxy-2,3-dihydrobenzofuran-5-yl)-5-fluoro-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4-diol; (2S,3R,4R,5S,6R)-2-[5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-methoxy-2,3-dihydrobenzofuran-7-yl]-5-fluoro-6-(hydroxymethyl)tetrahydropyran-3,4-diol; (2S,3R,4R,5S,6R)-2-(7-((2,3-dihydrobenzo[b][1,4]dioxin-6-yl)methyl)-4-hydroxy-2,3-dihydrobenzofuran-5-yl)-5-fluoro-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4-diol; (2S,3R,4R,5S,6R)-5-fluoro-6-(hydroxymethyl)-2-[4-methoxy-7-[(2,2,3,3-tetradeuterio-1,4-benzodioxin-6-yl)methyl]-2,3-dihydrobenzofuran-5-yl]tetrahydropyran-3,4-diol; (2S,3R,4R,5S,6R)-2-[7-[dideuterio(2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-methoxy-2,3-dihydrobenzofuran-5-yl]-5-fluoro-6-(hydroxymethyl)tetrahydropyran-3,4-diol; and isotopologues and pharmaceutically acceptable salts thereof.

Metadata:
- Claim Count in Document: 47.0
- Percentile: 96.0
- Lexical Diversity: 1.08108
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['14593071', '16059072', '16059074', '13634597', '14122836']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8359028762758705
- 35 USC 102 Novelty (BERT): 0.5273771711889197
- Combined Prediction Score: 0.8050503057671754
- Mean Citation Score: 351.143048
- Max Citation Score: 357.37866
- Similarity Product: 295.82409368978983

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 0
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test