PATENT CLAIM ANALYSIS

Application Number: 15759119
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2018-10
Patent Classification: ["564", "057000"]

Abstract:
Provided are a cyclohexane derivative as shown by formula IB or a stereoisomer or a salt thereof, and the preparation and use thereof. The cyclohexane derivative has a high affinity for D 3  receptors and 5-hydroxytryptamine, has a lower affinity for D 2  receptors, shows a high selectivity for D 3 /D 2  receptors, and can be used as a therapeutic drug against neuropsychiatric diseases; and the preparation method thereof is simple and easy.

Claim (Index 11):
The method according to  claim 10 , wherein the pharmaceutical composition is a solid tablet consisting of N\u2032-[trans-4-[2-[4-(benzo[b]thiophene)-7-piperazinyl]ethyl]cyclohexyl]-N,N-dimethylurea as an active ingredient and pharmaceutical excipients; and the solid tablet consists of the following components based on weight:\n active ingredient: 1-40 mg; diluent: 10-200 mg; adhesive: 5-25 mg; disintegrant: 5-50 mg; and lubricant: 1-5 mg; wherein the diluent is selected from starch, lactose or microcrystalline cellulose; the adhesive is selected from hydroxybenzyl cellulose, hydroxypropylmethyl cellulose or polyvinylpyrrolidone; the disintegrant is selected from sodium hydroxyethyl starch or crospovidone; and the lubricant is magnesium stearate.

Metadata:
- Claim Count in Document: 39.0
- Percentile: 90.0
- Lexical Diversity: 1.7234
- Patent Class: 564.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['14889831', '15124264', '15029218', '13123368', '13056365']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7264579889342867
- 35 USC 102 Novelty (BERT): 0.5390437161731316
- Combined Prediction Score: 0.7077165616581712
- Mean Citation Score: 248.190766
- Max Citation Score: 269.30753
- Similarity Product: 167.26111440414428

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test