PATENT CLAIM ANALYSIS

Application Number: 16313360
Application Type: Utility
Filing Date: 2018-12
Publication Date: 2019-06
Patent Classification: ["424", "001110"]

Abstract:
The present invention relates to an aryl ethene derivative, for inhibiting an estrogen-related receptor gamma (ERRγ) activity, a prodrug of same, a solvate of same, a stereoisomer of same or pharmaceutically acceptable salts of same, and a pharmaceutical composition containing same as an active ingredient.

Claim (Index 4):
The pharmaceutical composition of  claim 1 , wherein\n R 1  is (C3-CO 1 )heterocycloalkyl, (C3-C10)heteroaryl, \u2014O\u2014(CH 2 ) m \u2014R 11 , \u2014(CH 2 ) m \u2014R 12 , \u2014NH\u2014(CH 2 ) m \u2014R 13 , \u2014NHCO\u2014(CH 2 ) n \u2014R 14 , or \u2014SiR 16 R 17 \u2014(CH 2 ) m \u2014R 15 ; R 11  to R 15  are independently of one another (C3-C10)heterocycloalkyl; R 16  and R 17  are independently of each other (C1-C10)alkyl; m is an integer of 1 to 3; n is an integer of 0 or 1; Ar is (C6-C12)aryl or (C3-C12)heteroaryl, in which the aryl or heteroaryl of Ar may be further substituted by one or more selected from the group consisting of hydroxy, halogen, (C1-C10)alkyl, halo(C1-C10)alkyl, (C1-C10)alkoxy, nitro, cyano, amino, (C1-C10)alkylsulfonylamino, (C3-C10)cycloalkylsulfonylamino, di((C1-C10)alkylsulfonyl)amino, (C1-C10)alkylcarbonyloxy, (C1-C10)alkylcarbonylamino, guanidino, (C1-C10)alkylsulfonyl, (C1-C10)alkylsulfonyloxy, halo(C1-C10)alkylsulfonyloxy, and (C3-C10)cycloalkylsulfonyloxy; R 2  is hydroxy, fluoro, (C1-C10)alkylcarbonyloxy, or (C1-C10)alkylsulfonyloxy; and the heterocycloalkyl or heteroaryl of R 1  and the heterocycloalkyl of R 11  to R 15  may be further substituted by one or more selected from the group consisting of (C1-C10)alkyl, (C3-C10)cycloalkyl, (C2-C10)alkenyl, amidino, (C1-C10)alkoxycarbonyl, hydroxy(C1-C10)alkyl, and di(C1-C10)alkylamino(C1-C10)alkyl.

Metadata:
- Claim Count in Document: 26.0
- Percentile: 98.0
- Lexical Diversity: 1.43243
- Patent Class: 424.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15102968', '12704343', '11829531', '13098247', '14473147']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.731098864179551
- 35 USC 102 Novelty (BERT): 0.5229539934050796
- Combined Prediction Score: 0.7102843771021038
- Mean Citation Score: 290.742902
- Max Citation Score: 305.64383
- Similarity Product: 209.6487461914396

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 0
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test