PATENT CLAIM ANALYSIS

Application Number: 16180612
Application Type: Utility
Filing Date: 2018-11
Publication Date: 2019-03
Patent Classification: ["549", "029000"]

Abstract:
Disclosed are compounds, compositions and methods for treating of disorders that are affected by the modulation of the GPR120 receptor. Such compounds are represented by Formula (I) and Formula (II) as follows: wherein Y, R 1 , G, and Q are defined herein;and  wherein R 11 , R 21 , R 41 , R B1  and G 1 , are defined herein.

Claim (Index 31):
A compound of Formula (II) selected from the group consisting of Cpd 1, 3-(4-{[3-(4-Ethylphenyl)-5-fluorothiophen-2-yl]methoxy}-2,3-dimethylphenyl)propanoic acid; Cpd 2, 3-(4-{[5-Chloro-3-(4-chlorophenyl)thiophen-2-yl]methoxy}-3,5-difluorophenyl)propanoic acid; Cpd 3, 3-(4-{[3-(4-Chlorophenyl)-5-fluorothiophen-2-yl]methoxy}-2,3-dimethylphenyl)propanoic acid; Cpd 4, 3-(4-{[3-(4-Ethylphenyl)thiophen-2-yl]methoxy}-2,3-difluorophenyl)propan-1-ol; Cpd 5, 3-(4-{[5-Chloro-3-(4-ethylphenyl)thiophen-2-yl]methoxy}-2,3-dimethylphenyl)propanoic acid; Cpd 6, 3-(4-{[5-Chloro-3-(4-chlorophenyl)thiophen-2-yl]methoxy}-2,3-dimethylphenyl)propanoic acid; Cpd 7, 3-(4-{[3-(4-Ethylphenyl)-5-fluorothiophen-2-yl]methoxy}-3,5-difluorophenyl)propanoic acid; Cpd 8, 3-(4-{[5-Chloro-3-(4-ethylphenyl)thiophen-2-yl]methoxy}-3,5-difluorophenyl)propanoic acid; Cpd 9, 3-(4-{[5-Chloro-3-(4-ethylphenyl)thiophen-2-yl]methoxy}-3,5-difluorophenyl)propan-1-ol; Cpd 10, 3-(4-{[3-(4-Chlorophenyl)-5-fluorothiophen-2-yl]methoxy}-3,5-difluorophenyl)propanoic acid; Cpd 11, 3-(4-{[5-Chloro-3-(4-ethylphenyl)thiophen-2-yl]methoxy}-2,3-difluorophenyl)propanoic acid; Cpd 12, 3-(4-{[3-(4-Ethylphenyl)-5-fluorothiophen-2-yl]methoxy}-2,3-difluorophenyl)propanoic acid; Cpd 13, 3-(4-{[3-(4-Ethylphenyl)-5-methylthiophen-2-yl]methoxy}-2,3-dimethylphenyl)propanoic acid; Cpd 14, 3-(4-{[5-Chloro-3-(4-ethylphenyl)thiophen-2-yl]methoxy}-2,3-difluorophenyl)propan-1-ol; Cpd 15, 3-(4-{[5-Chloro-3-(4-chlorophenyl)thiophen-2-yl]methoxy}-2,3-dimethylphenyl)propan-1-ol; Cpd 16, 3-(3,5-Difluoro-4-{[3-(1-methylethoxy)-5-(trifluoromethyl)thiophen-2-yl]methoxy}phenyl)propanoic acid; Cpd 17, 3-(4-{[3-(4-Ethylphenyl)-5-fluorothiophen-2-yl]methoxy}-2,3-difluorophenyl)propan-1-ol; Cpd 18, 3-(4-{[3-(4-Chlorophenyl)-5-fluorothiophen-2-yl]methoxy}-3,5-difluorophenyl)propan-1-ol; Cpd 19, 3-(4-{[5-Chloro-3-(4-chlorophenyl)thiophen-2-yl]methoxy}-3,5-difluorophenyl)propan-1-ol; Cpd 20, 3-(4-{[3-(4-Ethylphenyl)thiophen-2-yl]methoxy}-3,5-difluorophenyl)propan-1-ol; Cpd 21, 3-(4-{[3-(4-Ethylphenyl)-5-(trifluoromethyl)thiophen-2-yl]methoxy}-2,3-difluorophenyl)propanoic acid; Cpd 22, 3-(4-{[3-(4-Ethylphenyl)-5-(trifluoromethyl)thiophen-2-yl]methoxy}-3,5-difluorophenyl)propanoic acid; Cpd 23, 3-(4-{[3-(4-Ethylphenyl)-5-methylthiophen-2-yl]methoxy}-2,3-difluorophenyl)propan-1-ol; Cpd 24, 3-(4-{[3-(4-Ethylphenyl)-5-methylthiophen-2-yl]methoxy}-3,5-difluorophenyl)propan-1-ol; Cpd 25, 3-(4-{[3-(4-Ethylphenyl)-5-methylthiophen-2-yl]methoxy}-3,5-difluorophenyl)propanoic acid; Cpd 26, 3-(4-{[3-(4-Ethylphenyl)-5-methylthiophen-2-yl]methoxy}-2,3-difluorophenyl)propanoic acid; Cpd 27, 3-(4-{[3-(4-Ethylphenyl)-5-fluorothiophen-2-yl]methoxy}-3,5-difluorophenyl)propan-1-ol; Cpd 28, 3-(4-{[5-Chloro-3-(4-chlorophenyl)thiophen-2-yl]methoxy}-2,3-difluorophenyl)propanoic acid; Cpd 29, 3-(4-{[5-Chloro-3-(4-chlorophenyl)thiophen-2-yl]methoxy}-2,3-difluorophenyl)propan-1-ol; Cpd 30, 3-(4-{[3-(4-Chlorophenyl)-5-fluorothiophen-2-yl]methoxy}-2,3-dimethylphenyl)propan-1-ol;\n or a pharmaceutically acceptable salt form thereof.

Metadata:
- Claim Count in Document: 68.0
- Percentile: 98.0
- Lexical Diversity: 1.7619
- Patent Class: 549.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['14200108', '14200127', '14200097', '14200114', '15228042']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8457796132920781
- 35 USC 102 Novelty (BERT): 0.6673735628165711
- Combined Prediction Score: 0.8279390082445274
- Mean Citation Score: 547.1481980000002
- Max Citation Score: 687.37866
- Similarity Product: 645.795306192609

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test