PATENT CLAIM ANALYSIS

Application Number: 16060142
Application Type: Utility
Filing Date: 2018-06
Publication Date: 2018-09
Patent Classification: ["546", "082000"]

Abstract:
The present invention relates to a process for phospholipidation of imidazoquinolines and oxoadenines. More particularly, the present invention relates to a high-yielding and scalable procedure for the phospholipidation of imidazoquinolines and oxoadenines which obviates the need to isolate unstable phosphoramidite intermediates. This process may be used for the phospholipidation of toll-like receptor 7 (TLR7)-active and toll-like receptor (TLR8)-active imidazoquinolines and oxoadenines.

Claim (Index 17):
The process of  claim 15  wherein imidazolium triflate is added with the compound of formula (VII) to the same reaction mixture produced by the reaction of compound of formula (V) with the compound of formula (III).

Metadata:
- Claim Count in Document: 29.0
- Percentile: 94.0
- Lexical Diversity: 1.775
- Patent Class: 546.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15781905', '14008805', '12578020', '13389307', '15126245']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7766058880128307
- 35 USC 102 Novelty (BERT): 0.520689232606413
- Combined Prediction Score: 0.751014222472189
- Mean Citation Score: 259.280824
- Max Citation Score: 305.36798
- Similarity Product: 184.97728015704988

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test