PATENT CLAIM ANALYSIS

Application Number: 15763626
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2018-09
Patent Classification: ["514", "210210"]

Abstract:
Compounds of formula (I): wherein R 1 , R 2 , W 3 , W 4 , A 1 , and A 2  are as defined in the description. Medicinal products containing the same which are useful in treating cancer, neurodegenerative disorders and metabolic disorders.

Claim (Index 38):
A compound of formula (I): wherein:\n R 1  and R 2 , each independently of the other, represent a hydrogen atom, a halogen atom, \u2014NR 5 R 5 \u2032 or a linear or branched (C 1 -C 6 )alkyl group, \n W 3  represents a linear or branched (C 1 -C 6 )alkoxy, \u2014O\u2014(C 1 -C 6 )alkylene-Cy 1 , \u2014O\u2014(C 0 -C 6 )-Cy 1 -Cy 2 , \u2014NR a R b , \u2014NR a \u2014(C 0 -C 6 )alkylene-Cy 1 , \u2014NR a -(C 0 -C 6 )alkylene-Cy 1 -Cy 2 , \u2014NR a \u2014(C 0 -C 6 )alkylene-Cy 1 -O\u2014(C 1 -C 6 )alkylene-Cy 2 , -Cy 1 , -Cy 1 -(C 0 -C 6 )alkylene-Cy 2 , -Cy 1 -O\u2014(C 0 -C 6 )alkylene-Cy 2 , \u2014(C 1 -C 6 )alkylene-Cy 1 , \u2014(C 2 -C 6 )alkenylene-Cy 1 , \u2014(C 2 -C 6 )alkynylene-Cy 1 , \u2014(C 1 -C 6 )alkylene-O-Cy 1 , it being understood that the alkylene moieties defined hereinbefore may be linear or branched, \n W 4  represents a cyano group, a cycloalkyl group, a linear or branched (C 1 -C 6 )alkyl group, a linear or branched (C 2 -C 6 )alkenyl group, a linear or branched (C 2 -C 6 )alkynyl group optionally substituted by a cycloalkyl group, \n R 5  and R 5 \u2032 each independently of the others, represent a hydrogen atom or a linear or branched (C 1 -C 6 )alkyl group, \n R a  and R b , each independently of the other, represent a hydrogen atom or a linear or branched (C 1 -C 6 )alkyl group, \n A 1  and A 2 , each independently of the other, represent CH or a nitrogen atom, \n Cy 1 , Cy 2 and Cy 3 , independently of one another, represent a cycloalkyl group, a heterocycloalkyl group, an aryl or an heteroaryl group, \n wherein:\n \u201caryl\u201d means a phenyl, naphthyl, biphenyl or indenyl group, \n \u201cheteroaryl\u201d means any mono- or bi-cyclic group composed of from 5 to 10 ring members, having at least one aromatic moiety and containing from 1 to 4 hetero atoms selected from oxygen, sulphur and nitrogen. \n \u201ccycloalkyl\u201d means any mono- or bi-cyclic, non-aromatic, carbocyclic group containing from 3 to 11 ring members, which may include fused, bridged or spiro ring systems, \n \u201cheterocycloalkyl\u201d means any mono- or bi-cyclic, non-aromatic, condensed or spiro group composed of from 3 to 10 ring members and containing from 1 to 3 hetero atoms or groups selected from oxygen, sulphur, SO, SO 2  and nitrogen, which may include fused, bridged or spiro ring systems, \n \u201c\u2014(C 0 -C 6 )alkylene-\u201d refers either to a covalent bond (\u2014C 0 alkylene-) or to an alkylene group containing 1, 2, 3, 4, 5 or 6 carbon atoms, \n wherein the aryl, heteroaryl, cycloalkyl and heterocycloalkyl groups so defined and the alkyl, alkenyl, alkynyl, alkylene, alkenylene, alkynylene to be substituted by from 1 to 4 groups selected from linear or branched (C 1 -C 6 )alkyl, linear or branched (C 2 -C 6 )alkenyl group, linear or branched (C 2 -C 6 )alkynyl group, linear or branched (C 1 -C 6 )alkoxy optionally substituted by \u2014NR c R d  or by from 1 to 3 halogen atoms, linear or branched (C 1 -C 6 )alkyl-S\u2014, hydroxy, oxo (or N-oxide where appropriate), nitro, cyano, \u2014C(O)\u2014OR c , \u2014C(O)\u2014R c , \u2014O\u2014C(O)\u2014R d , \u2014C(O)\u2014NR c R d , \u2014NR c \u2014C(O)\u2014R d , \u2014NR c R d , linear or branched (C 1 -C 6 )polyhaloalkyl, or halogen, it being understood that R c  and R d  independently of one another represent a hydrogen atom or a linear or branched (C 1 -C 6 )alkyl group, its enantiomers and diastereoisomers, and addition salts thereof with a pharmaceutically acceptable acid or base.

Metadata:
- Claim Count in Document: 20.0
- Percentile: 90.0
- Lexical Diversity: 1.45714
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['16306941', '14435851', '14559294', '15247499', '15738186']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7954365639045538
- 35 USC 102 Novelty (BERT): 0.5201112692018531
- Combined Prediction Score: 0.7679040344342837
- Mean Citation Score: 314.096512
- Max Citation Score: 331.03336
- Similarity Product: 285.316282254796

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 0
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test