PATENT CLAIM ANALYSIS

Application Number: 15781848
Application Type: Utility
Filing Date: 2018-06
Publication Date: 2018-12
Patent Classification: ["514", "300000"]

Abstract:
The present application relates to novel (2-phenylimidazo[1,2-a]pyridin-3-yl)methyl-substituted perhydropyrrolo[3,4-c]pyrrole derivatives, to methods for the preparation thereof, to the use thereof alone or in combinations for treatment and/or prevention of diseases, and to the use thereof for production of medicaments for treatment and/or prevention of diseases, especially for treatment and/or prevention of respiratory disorders including sleep-related respiratory disorders such as obstructive sleep apneas and central sleep apneas and snoring.

Claim (Index 3):
The compound of  claim 1 , in which\n R 1  represents chlorine, bromine or isopropyl, and R 2  represents cyclobutyl or cyclopentyl, or R 2  represents a phenyl group of the formula (a) or a pyridyl group of the formula (b) in which * marks the bond to the adjacent carbonyl group and R 3  represents fluorine, chlorine, methyl, trifluoromethyl or methoxy,\n R 4  represents hydrogen or fluorine, \n R 5  represents hydrogen, fluorine or methyl \n and \n R 6  represents methoxy, \n or R 2  represents an \u2014OR 7  or \u2014NR 8 R 9  group in which R 7  represents isopropyl, cyclopentyl, phenyl or benzyl,\n where phenyl and the phenyl group in benzyl may be up to disubstituted by identical or different radicals selected from the group consisting of fluorine, chlorine, methyl, trifluoromethyl, methoxy and ethoxy, \n R 8  represents phenyl or 1-phenylethyl,\n where phenyl and the phenyl group in 1-phenylethyl may be up to disubstituted by identical or different radicals selected from the group consisting of fluorine, chlorine, methyl, trifluoromethyl, methoxy and ethoxy, \n and \n R 9  is hydrogen, \n or \n R 8  and R 9  are attached to one another and, together with the nitrogen atom to which they are bonded, form a tetrahydroquinoline ring of the formula (c), in which ** marks the bond to the carbonyl group, and the salts, solvates and solvates of the salts thereof.

Metadata:
- Claim Count in Document: 4.0
- Percentile: 94.0
- Lexical Diversity: 1.66
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15027519', '15735138', '14895793', '13819337', '13945675']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7972919891451068
- 35 USC 102 Novelty (BERT): 0.5251638679294768
- Combined Prediction Score: 0.7700791770235438
- Mean Citation Score: 325.011188
- Max Citation Score: 333.57864
- Similarity Product: 286.4509097383118

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test