PATENT CLAIM ANALYSIS

Application Number: 15750103
Application Type: Utility
Filing Date: 2018-02
Publication Date: 2018-08
Patent Classification: ["514", "338000"]

Abstract:
Compounds of formula (I) as described herein, processes for their production and their use as pharmaceuticals.

Claim (Index 2):
The compound of formula (I) according to  claim 1 , wherein:\n G represents a group selected from: wherein * indicates the points of attachment of said group with the rest of the molecule; X represents CH 2 , or C\u2550O; R 1  represents hydrogen or C 1 -C 4 -alkyl; R 2  represents hydrogen, C 1 -C 4 -alkyl, R 10 \u2014O\u2014C(O)\u2014 or R 7 R 8 N\u2014C(O)\u2014; R 3  represents hydrogen or C 1 -C 4 -alkyl; A represents a group selected from: wherein * indicates the point of attachment of said group with the rest of the molecule and said group is optionally substituted, one or more times, independently from each other, with R 4 ; R 4  represents halogen, hydroxy, nitro, cyano, C 1 -C 4 -alkyl, C 1 -C 4 -alkoxy, C 1 -C 4 -haloalkyl, C 1 -C 4 -haloalkoxy, C 1 -C 4 -hydroxyalkyl, C 1 -C 4 -alkyl-C(O)\u2014, or R 10 \u2014O\u2014C(O)\u2014; E represents a group wherein * indicates the point of attachment of said group with the rest of the molecule; R 5  represents, independently from each other, halogen, hydroxy, nitro, cyano, R 9 R 10 N\u2014, (R 13 \u2014C(O)\u2014)(R 14 \u2014C(O)\u2014)N\u2014, C 1 -C 3 -alkyl, C 3 -C 4 -cycloalkyl, C 1 -C 3 -alkoxy, C 1 -C 3 -haloalkyl, C 1 -C 3 -haloalkoxy, R 6 \u2014C(O)\u2014NR 9 \u2014, R 6 \u2014O\u2014C(O)\u2014NR 9 \u2014, R 6 \u2014SO 2 \u2014NR 9 \u2014 or R 7 R 8 N\u2014C(O)\u2014NR 9 \u2014, Q represents O; R 6  represents, independently from each other, C 1 -C 6 -alkyl, C 3 -C 6 -cycloalkyl, 4- to 6-membered heterocycloalkyl, phenyl or heteroaryl,\n wherein said C 1 -C 6 -alkyl is optionally substituted, one or more times, independently from each other, with halogen, hydroxy, nitro, cyano, C 1 -C 4 -alkoxy, C 1 -C 4 -haloalkoxy, C 3 -C 6 -cycloalkyl, R 7 R 8 N\u2014 or phenyl optionally substituted, one or more times, independently from each other, with R 4 , \n wherein said C 3 -C 6 -cycloalkyl, 4- to 6-membered heterocycloalkyl, phenyl or heteroaryl groups are optionally substituted, one or more times, independently from each other, with halogen, hydroxy, nitro, cyano, C 1 -C 6 -alkyl, C 1 -C 4 -alkoxy, C 1 -C 4 -haloalkyl, R 10 \u2014O\u2014C(O)\u2014 or C 1 -C 4 -haloalkoxy; \n R 7 , R 8  represent, independently from each other, hydrogen, C 1 -C 6 -alkyl, C 3 -C 6 -cycloalkyl, R 10 \u2014O\u2014C(O)\u2014 or phenyl,\n wherein said C 1 -C 6 -alkyl is optionally substituted, one or more times, independently from each other, with halogen, hydroxy, C 1 -C 4 -alkoxy, C 1 -C 4 -haloalkoxy, C 3 -C 6 -cycloalkyl optionally substituted one time with hydroxy, 4- to 6-membered heterocycloalkyl, heteroaryl, or R 9 R 10 N\u2014, \n wherein said phenyl group is optionally substituted, one or more times, independently from each other, with R 4 ; \n or, \n R 7  and R 8  together with the nitrogen atom to which they are attached form a 5- to 6-membered nitrogen containing heterocyclic ring, optionally containing one additional heteroatom selected from O, and NR 9 ; R 9  represents hydrogen, or C 1 -C 4 -alkyl; R 10  represents hydrogen, C 1 -C 4 -alkyl or C 3 -C 4 -cycloalkyl; R 13 , R 14  represent, independently from each other, C 1 -C 3 -alkyl, or C 3 -C 4 -cycloalkyl,\n wherein said C 3 -C 4 -cycloalkyl is optionally substituted, one or more times, independently from each other, with halogen; \n m represents 0, 1 or 2; or an N-oxide, a salt, a tautomer or a stereoisomer of said compound, or a salt of said N-oxide, tautomer or stereoisomer.

Metadata:
- Claim Count in Document: 8.0
- Percentile: 88.0
- Lexical Diversity: 1.11111
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15317924', '15737182', '14004515', '14350160', '14900599']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.761821441772058
- 35 USC 102 Novelty (BERT): 0.5438808936873665
- Combined Prediction Score: 0.7400273869635888
- Mean Citation Score: 301.259288
- Max Citation Score: 372.99286
- Similarity Product: 281.44464528805497

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test