PATENT CLAIM ANALYSIS

Application Number: 16081904
Application Type: Utility
Filing Date: 2018-09
Publication Date: 2019-06
Patent Classification: ["514", "064000"]

Abstract:
Compounds, pharmaceutical formulations, and methods of treating bacterial infections are disclosed.

Claim (Index 1):
A compound, or a salt or a hydrate or a solvate thereof, having a structure which is: wherein W is H or a bond to X; X is wherein\n R a  and R b  are each independently selected from the group consisting of R 15 , \u2014OR 15 , \u2014NR 15 R 16 , \u2014SR 15 , \u2014S(O)R 15 , \u2014S(O) 2 R 15 , \u2014S(O) 2 NR 15 R 16 , \u2014C(O)R 15 , \u2014C(O)OR 15 , and \u2014C(O)NR 15 R 16  \n wherein R 15  and R 16  are each independently selected from the group consisting of H, halogen, cyano, nitro, \u2014OR 17 , \u2014NR 17 R 18 , substituted or unsubstituted alkyl, substituted or unsubstituted heteroalkyl, substituted or unsubstituted cycloalkyl, substituted or unsubstituted heterocycloalkyl, substituted or unsubstituted aryl, and substituted or unsubstituted heteroaryl\n wherein R 17  and R 18  are each independently selected from the group consisting of H, substituted or unsubstituted alkyl, substituted or unsubstituted heteroalkyl, substituted or unsubstituted cycloalkyl, substituted or unsubstituted heterocycloalkyl, substituted or unsubstituted aryl, and substituted or unsubstituted heteroaryl \n \n \n and wherein R 15  and R 16 , and/or R 17  and R 18 , along with the nitrogen to which they are connected, are optionally joined to form a substituted or unsubstituted 4- to 8-membered ring \n with the proviso that R a  and R b  are not both H; \n or X is wherein\n R c  is \u2014OR 15 , \u2014NR 15 R 16 , \u2014SR 15 , \u2014S(O)R 15 , \u2014S(O) 2 R 15 , \u2014S(O) 2 NR 15 R 16 , \u2014C(O)R 15 , \u2014C(O)OR 15 , and \u2014C(O)NR 15 R 16  \n wherein R 15  and R 16  are each independently selected from the group consisting of H, halogen, cyano, nitro, substituted or unsubstituted alkyl, substituted or unsubstituted heteroalkyl, substituted or unsubstituted cycloalkyl, substituted or unsubstituted heterocycloalkyl, substituted or unsubstituted aryl, and substituted or unsubstituted heteroaryl \n and wherein R 15  and R 16 , along with the nitrogen to which they are connected, are optionally joined to form a substituted or unsubstituted 4- to 8-membered ring \n \n or X is H wherein\n R d  and R e  are each independently selected from the group consisting of H, halogen, cyano, nitro, substituted or unsubstituted alkyl, substituted or unsubstituted heteroalkyl, substituted or unsubstituted cycloalkyl, substituted or unsubstituted heterocycloalkyl, substituted or unsubstituted aryl, and substituted or unsubstituted heteroaryl, \u2014OR 15 , \u2014NR 15 R 16 , \u2014SR 15 , \u2014S(O)R 15 , \u2014S(O) 2 R 15 , \u2014S(O) 2 NR 15 R 16 , \u2014C(O)R 15 , \u2014C(O)OR 15 , and \u2014C(O)NR 15 R 16  \n wherein R 15  and R 16  are each independently selected from the group consisting of H, halogen, cyano, nitro, substituted or unsubstituted alkyl, substituted or unsubstituted heteroalkyl, substituted or unsubstituted cycloalkyl, substituted or unsubstituted heterocycloalkyl, substituted or unsubstituted aryl, and substituted or unsubstituted heteroaryl \n and wherein R d  and R e , along with the atom to which they are connected, are optionally joined to form a substituted or unsubstituted 3- to 8-membered ring \n and wherein R 15  and R 16 , along with the nitrogen to which they are connected, are optionally joined to form a substituted or unsubstituted 4- to 8-membered ring \n with the proviso that R d  and R e  are not both H \n \n wherein X optionally comprises an attachment point to W; Y is selected from the group consisting of a bond, \u2014O\u2014, \u2014S\u2014, \u2014NH\u2014, substituted or unsubstituted alkylene, and substituted or unsubstituted heteroalkylene; and Z is a substituted or unsubstituted heterocyclic ring or ring system containing at least one endocyclic boron.

Metadata:
- Claim Count in Document: 5.0
- Percentile: 97.0
- Lexical Diversity: 1.07692
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['16081902', '15718422', '15986747', '13606949', '14688581']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7241256913077775
- 35 USC 102 Novelty (BERT): 0.546364110228837
- Combined Prediction Score: 0.7063495331998835
- Mean Citation Score: 255.67250400000003
- Max Citation Score: 390.4352
- Similarity Product: 243.38705353469848

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test