PATENT CLAIM ANALYSIS

Application Number: 16106104
Application Type: Utility
Filing Date: 2018-08
Publication Date: 2019-02
Patent Classification: ["514", "301000"]

Abstract:
The present invention is directed to 5-fluoro-C-(aryl or hetercyclyl)-glycoside derivatives, pharmaceutical compositions containing them and their use in the treatment of disorders and conditions modulated by SGLT activity, more particularly dual SGLT1/2 activity.

Claim (Index 7):
A compound as in  claim 4 , wherein\n R 1  is hydroxy-methyl- R 2  is selected from the group consisting of hydrogen, hydroxy, methyl, methoxy, benzyloxy and trideutero-methoxy; R 3  and R 4  are taken together with the carbon atoms to which they are bound to form a ring structure selected from the group consisting of 2,3-dihydro-furanyl, 3-hydroxy-2,2-dimethyl-2,3-dihydro-furanyl, 3-hydroxymethyl-2,3-dihydro-furanyl, 3-hydroxyethyl-2,3-dihydro-furanyl, 3-methyl-3-hydroxymethyl-2,3-dihydro-furanyl and 3-methyl-2,3-dihydro-furanyl; R 5  and R 6  are the same and are selected from the group consisting of hydrogen and deuterium;  is selected from the group consisting of 4-ethyl-phenyl, 4-ethoxy-phenyl, 4-(fluoromethoxy)-phenyl, benzothien-2-yl, chroman-6-yl, 2,3-dihydro-benzo[b][1,4]dioxin-6-yl, 3,4-dihydro-quiunolin-7-yl, 1-methyl-3,4-dihydro-quinolin-7-yl, benzo[b][1,4]oxazin-7-yl-3-one, 2,3-dihydro-benzo[b][1,4]oxathiin-6-yl, 5-(pyrrolidin-1-yl-carbonyl)-6,7-dihydro-thieno[3,2-c]pyridin-2-yl and 2,2,3,3-tetradeutero-2,3-dihydro-benzo[b][1,4]dioxin-6-yl; or a pharmaceutically acceptable salt thereof.

Metadata:
- Claim Count in Document: 47.0
- Percentile: 96.0
- Lexical Diversity: 1.08108
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['14593071', '16059072', '16059074', '13634597', '14122836']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8360977469983987
- 35 USC 102 Novelty (BERT): 0.5280263708642576
- Combined Prediction Score: 0.8052906093849845
- Mean Citation Score: 351.143048
- Max Citation Score: 357.37866
- Similarity Product: 275.2119798228407

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 0
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test