PATENT CLAIM ANALYSIS

Application Number: 16007417
Application Type: Utility
Filing Date: 2018-06
Publication Date: 2018-12
Patent Classification: ["514", "235800"]

Abstract:
Aminothiazole compounds of Formula (I) shown below and pharmaceutical compositions containing one of such compounds: Also disclosed are methods of inhibiting a tyrosine kinase and treating cancer associated with a tyrosine kinase with one of the aminothiazole compounds.

Claim (Index 1):
A compound of formula (I) below or a pharmaceutically acceptable salt thereof: wherein\n R 1  is C 1-6  alkyl or C 1-6  thioalkyl; \n X is O or NR a , in which R a  is H or C 1-6  alkyl; \n Y is CR b R c  or NR d , in which each of R b  and R c , independently, is H, halo, C 1-6  alkyl, C 1-6  alkoxyl, or amino, or R b , together with R a , the carbon atom bonded to R b , and the nitrogen atom bonded to R a , is C 3-10  heterocycloalkyl; and R d  is H or C 1-6  alkyl, or R d , together with R a  and the nitrogen atoms bonded to R d  and R a , is C 3-10  heterocycloalkyl; \n R 2  is \u2014CH 2 CH 2 R e  or NR f R g , in which R e  is H, halo, C 1-6  alkyl, or OR b  and each of R f  and R g , independently, is C 1-6  alkyl or C 3-8  cycloalkyl, R h  being H or C 1-6  alkyl, or R h , together with R d , the oxygen atom bonded to R h , and the nitrogen atom bonded to R d , being C 3-10  heterocycloalkyl; and \n R 3  is heteroaryl.

Metadata:
- Claim Count in Document: 39.0
- Percentile: 94.0
- Lexical Diversity: 1.35484
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15419183', '15257926', '15861688', '14670421', '14670425']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.774959781604317
- 35 USC 102 Novelty (BERT): 0.5410036364338358
- Combined Prediction Score: 0.7515641670872689
- Mean Citation Score: 323.369304
- Max Citation Score: 366.57004
- Similarity Product: 307.19124306156874

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test