PATENT CLAIM ANALYSIS

Application Number: 16097440
Application Type: Utility
Filing Date: 2018-10
Publication Date: 2019-05
Patent Classification: ["514", "340000"]

Abstract:
Compounds of the formula I in which X, Y, R 1  and R 2  have the meanings indicated in claim  1 , are inhibitors of pyruvate dehydrogenase kinase (PDHK), and can be employed, inter alia, for the treatment of diseases such as cancer.

Claim (Index 1):
Compounds of the formula I in which\n X\u2014Y denotes CO\u2014NA\u2033 or NA\u2033-CO, \n R 1  denotes Ar or Het, \n R 2  denotes H or CH 3 , \n R 3  denotes H or A\u2032, \n Ar denotes phenyl, which is unsubstituted or mono-, di- or trisubstituted by Hal, NO 2 , CN, A, OR 3 , S(O) m R 3 , N(R 3 ) 2 , COA, COOR 3 , CON(R 3 ) 2 , SO 2 N(R 3 ) 2 , NR 3 COR 3 , NR 3 SO 2 A and/or NR 3 CON(R 3 ) 2 , \n Het denotes a mono- or bicyclic saturated, unsaturated or aromatic heterocycle having 1 to 4 N, O and/or S atoms, which is unsubstituted or mono- or disubstituted by Hal, NO 2 , CN, A, OR 3  S(O) m R 3 , N(R 3 ) 2 , COA, COOR 3 , CON(R 3 ) 2 , SO 2 N(R 3 ) 2 , NR 3 COR 3 , NR 3 SO 2 A and/or NR 3 CON(R 3 ) 2 , \n A denotes unbranched or branched alkyl with 1-10 C-atoms, wherein one or two non-adjacent CH- and/or CH 2 -groups may be replaced by N-, O- and/or S-atoms and/or wherein 1-7H-atoms may be replaced by R 4 , \n R 4  denotes F, Cl or OH, \n A\u2032 denotes unbranched or branched alkyl with 1-6 C-atoms, wherein 1-5H-atoms may be replaced by F, \n A\u2033 denotes unbranched or branched alkyl with 1-4 C-atoms, \n Hal denotes F, Cl, Br or I, \n m denotes 0, 1 or 2,\n and pharmaceutically acceptable salts, tautomers and stereoisomers thereof, including mixtures thereof in all ratios.

Metadata:
- Claim Count in Document: 32.0
- Percentile: 97.0
- Lexical Diversity: 1.34211
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15105154', '15748786', '14420003', '16069326', '15039226']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7811899948270586
- 35 USC 102 Novelty (BERT): 0.5639952883093821
- Combined Prediction Score: 0.759470524175291
- Mean Citation Score: 359.29564
- Max Citation Score: 434.02216
- Similarity Product: 346.3780791308022

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test