PATENT CLAIM ANALYSIS

Application Number: 15910307
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2018-07
Patent Classification: ["514", "259300"]

Abstract:
The invention provides novel compounds having the general formula (I) wherein R A , R B , R C , R C1  and W are as defined herein, compositions including the compounds and methods of using the compounds.

Claim (Index 35):
A compound according to  claim 1  and of formula I(b), wherein R A  is selected from the group consisting of\n i) C 1 -C 6 -alkyl, and \n ii) phenyl substituted with R G  and R G1 ; \n R B  is selected from the group consisting of\n i) cyano, and \n ii) halogen; \n R D1  is C 1 -C 6 -alkyl; R G  is selected from the group consisting of\n i) H, \n ii) C 1 -C 6 -alkoxy, \n iii) C 1 -C 6 -alkoxy-C 1 -C 6 -alkylcarbonylamino-C 1 -C 6 -alkyl, \n iv) C 1 -C 6 -alkoxy-C 1 -C 6 -alkylcarbonyl(C 1 -C 6 -alkyl)amino-C 1 -C 6 -alkyl, \n v) C 1 -C 6 -alkoxycarbonyl, \n vi) C 1 -C 6 -alkyl, \n vii) C 1 -C 6 -alkylsulfonyl, \n viii) carboxy, \n ix) cyano, \n x) C 3 -C 8 -cycloalkoxy, \n xi) C 3 -C 8 -cycloalkylcarbonylamino-C 1 -C 6 -alkyl, \n xii) C 3 -C 8 -cycloalkylcarbonyl(C 1 -C 6 -alkyl)amino-C 1 -C 6 -alkyl, \n xiii) halo-C 1 -C 6 -alkyl, \n xiv) halogen, \n xv) aminocarbonyl substituted on the nitrogen atom with R N  and R O , \n xvi) aminocarbonyl-C 1 -C 6 -alkoxy substituted on the nitrogen atom with R N  and R O , \n xvii) heteroaryl substituted with one H, C 1 -C 6 -alkyl, wherein heteroaryl is isoxazolyl, oxazolyl or pyrazolyl, \n xviii) heterocycloalkyl-C 1 -C 6 -alkoxy substituted with one H, C 1 -C 6 -alkyl, wherein heterocycloalkyl-C 1 -C 6 -alkoxy is tetrahydropyranylmethoxy or tetrahydrofuranylmethoxy , and \n xix) heterocycloalkyl-C 1 -C 6 -alkyl substituted with one H, C 1 -C 6 -alkyl, wherein heterocycloalkyl-C 1 -C 6 -alkyl is methyldioxopiperazinylmethyl, oxopyrrolidinylmethyl or oxooxazolidinylmethyl; \n R G2  is H and R G1  is selected from the group consisting of\n i) H, \n ii) halogen, \n iii) C 1 -C 6 -alkyl, and \n iv) halo-C 1 -C 6 -alkoxy; \n R N  is selected from the group consisting of\n i) H, \n ii) C 1 -C 6 -alkoxy, \n iii) C 1 -C 6 -alkoxy-C 1 -C 6 -alkyl, \n iv) C 1 -C 6 -alkoxycarbonyl-C 1 -C 6 -alkyl, \n v) C 1 -C 6 -alkyl, \n vi) carboxy-C 1 -C 6 -alkyl, \n vii) C 3 -C 8 -cycloalkyl, \n viii) C 3 -C 8 -cycloalkyl-C 1 -C 6 -alkyl, \n ix) hydroxy-C 1 -C 6 -alkyl, \n x) phenyl, and \n xi) heteroaryl-C  1 -C 6 -alkyl, wherein heteroaryl-C  1 -C 6 -alkyl is are pyridinylalkyl or thiophenylalkyl; \n R O  is selected from the group consisting of\n i) H, and \n ii) C 1 -C 6 -alkyl; \n or R N  and R O  together with the nitrogen atom to which they are attached form piperidinyl, morpholinyl, pyrrolidinyl or methylpiperazinonyl; or pharmaceutically acceptable salts.

Metadata:
- Claim Count in Document: 1.0
- Percentile: 90.0
- Lexical Diversity: 1.35484
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['12462417', '14844991', '15332398', '12466785', '14376307']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8091614170008097
- 35 USC 102 Novelty (BERT): 0.5385999333933204
- Combined Prediction Score: 0.7821052686400607
- Mean Citation Score: 361.796304
- Max Citation Score: 369.039
- Similarity Product: 275.59526970112324

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test