PATENT CLAIM ANALYSIS

Application Number: 16079812
Application Type: Utility
Filing Date: 2018-08
Publication Date: 2019-03
Patent Classification: ["546", "153000"]

Abstract:
The present invention relates to compounds of formula (I) including any stereochemically isomeric form thereof, or pharmaceutically acceptable salts thereof, for the treatment of tuberculosis.

Claim (Index 1):
A compound of formula (I): including any stereochemically isomeric form thereof, wherein: R 1  is -phenyl, optionally mono- or bi-substituted independently with lower alkyl, halogen or alkoxy,\n 5- or 6-membered heteroaryl, optionally mono-, bi- or tri-substituted independently with lower alkyl, halogen, alkoxy, \u2014SCH 3 , \u2014SCH 2 CH 3 , \u2014N(CH 2 CH 3 ) 2  or \u2014N(CH 3 ) 2 , \n benzofuranyl, \n 2,3-dihydrobenzo[b][1,4]dioxin-5-yl, \n 2,3-dihydro-1H-inden-4-yl or \n 5,6,7,8-tetrahydro naphthalene-1-yl; \n R 2  and R 3 , independently of each other, are hydrogen or lower alkyl; R 4  is -phenyl, optionally mono- or bi-substituted independently with halogen or lower alkyl,\n 5- or 6-membered heteroaryl, optionally mono-, bi- or tri-substituted independently with alkoxy, \u2014O-cycloalkyl, \u2014S-loweralkyl, difluoromethoxy or \u2014N(CH 3 ) 2 , \n benzofuranyl, \n benzo[b]thiophenyl or \n 2,3-dihydro-1H-indenyl; and \n R 5  is halogen or cyano, or a pharmaceutically acceptable salt thereof.

Metadata:
- Claim Count in Document: 74.0
- Percentile: 96.0
- Lexical Diversity: 1.11111
- Patent Class: 546.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15325824', '15112294', '11219148', '11015508', '15311817']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7679916220102383
- 35 USC 102 Novelty (BERT): 0.5100674588223985
- Combined Prediction Score: 0.7421992056914544
- Mean Citation Score: 244.50118200000003
- Max Citation Score: 264.78528
- Similarity Product: 188.2167137592316

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test