PATENT CLAIM ANALYSIS

Application Number: 15938409
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2018-08
Patent Classification: ["546", "014000"]

Abstract:
A compound having the general structure shown in Formula I: or pharmaceutically acceptable salts and/or solvates thereof are useful in treating diseases or conditions mediated by NK 1  receptors, for example various physiological disorders, symptoms or diseases, including emesis, depression, anxiety and cough.

Claim (Index 2):
The method of  claim 1 , wherein the physiological disorder, symptom or disease is depression, anxiety, a bladder disorder or a genitourinary disorder and the compound is selected from the group consisting of a compound having the Formula IB wherein R 1  and R 2  are selected from the group consisting of: Compound R 1 R 2 \u20021 \u2014CN   \u20022 \u2014CN   \u20023   \u20024   \u20025 \u2014CH 2 CN   \u20026 \u2014CH 3   \u20027 \u2014CN   \u20028 \u2014C(O)\u2014O\u2014CH 3   \u20029 \u2014CN   10 \u2014C(O)\u2014NH 2   11 \u2014CH 2 C(OH)(CH 3 ) 2   12 \u2014CH 2 OH   13 \u2014CH 2 OCH 3   14 \u2014CH 2 OCH 3   15 \u2014CH 2 \u2014NH\u2014S(O 2 )\u2014CH 3   16 CH 2 C(O)\u2014NH(CH 2 CH 3 )   17 CH 2 \u2014C(O)O\u2014CH 2 CH 3   18 \u2014C(\u2550N\u2014OH)\u2014CH 2 CH 3   19 \u2014C(O)\u2014CH 2 CH 3   20 \u2014CH 2 OCH 3   21 \u2014C(O)\u2014NH(CH 3 )   22 C(O)\u2014NH(CH 3 )   23 \u2014CH 2 OH   24 \u2014CH 2 CH 2 OH   25 \u2014CH 2 CH 2 CH 3   26 \u2014CH 2 OCH 3   27 \u2014CH 2 OCH 3   28 H   29 \u2014CH 2 C(O)\u2014NH 2   30 \u2014CH 2 \u2014C(O)\u2014CH 3   31 \u2014CH 2 \u2014C(O)O\u2014CH 3   32 \u2014CN   33 \u2014CN   34 \u2014CN   35 \u2014CN   36 NH\u2014S(O 2 )\u2014CH 3 \u2014CN 37 \u2014CN \u2014NH\u2014S(O 2 )\u2014CH 3   38 \u2014CH 2 CN   39 \u2014CN \u2014NH 2 40 \u2014NH 2 \u2014CN 41 NH\u2014C(O)\u2014NH 2 \u2014CN   42 \u2014CN   43 H   44 H   45 H   46 H   47 H   48 H   49 H   50 H   51 \u2014C(O)\u2014NH 2   52 \u2014C(\u2550N\u2014OCH 3 )\u2014CH 3   53 \u2014C(O)\u2014CH 3   54 \u2014C(\u2550N\u2014OH)\u2014CH 3   55 \u2014C(O)OCH 3   56 \u2014CH 2 Cl   57 \u2014CH 3   58 C(\u2550N\u2014OCH 3 )\u2014CH 2 CH 3   59 \u2014NHC(O)CH 3   60 H   61 H

Metadata:
- Claim Count in Document: 11.0
- Percentile: 90.0
- Lexical Diversity: 1.19048
- Patent Class: 546.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['13245403', '12750420', '11432133', '11653558', '10741056']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8500145246812101
- 35 USC 102 Novelty (BERT): 0.5255089002285234
- Combined Prediction Score: 0.8175639622359414
- Mean Citation Score: 343.390956
- Max Citation Score: 362.47183
- Similarity Product: 261.24008988165923

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 0
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test