PATENT CLAIM ANALYSIS

Application Number: 15893804
Application Type: Utility
Filing Date: 2018-02
Publication Date: 2018-06
Patent Classification: ["514", "264110"]

Abstract:
A method for inhibiting androgen activity, including administering an effective amount of a tetrahydropyridopyrimidine compound of formula (I) or a pharmaceutically acceptable salt thereof to a subject in need thereof, and a method for treating tumor, including administering an effective amount of a tetrahydropyridopyrimidine compound of formula (I) or a pharmaceutically acceptable salt thereof to a subject in need thereof

Claim (Index 29):
The method of  claim 23 , wherein, in the formula (I), X is a chlorine atom, a bromine atom, or a trifluoromethyl group, and\n R is selected from the group consisting of: where R 1  is a hydrogen atom, a phenyl group, a hydroxy-C 1-4  alkyl group, a hydroxy-C 3-5  cycloalkyl group, a C 1-4  alkoxy group which is substituted or unsubstituted with Ra, a C 3-5  cycloalkylaminosulfonyl group, a 7-membered monocyclic heterocycloalkylsulfonyl group, a fluoro-C 1-3  alkoxycarbonylamino group, a fluoro-C 1-3  alkylcarbonylamino group, a 6-membered monocyclic heterocycloalkanecarbonyl group substituted with a hydroxy-C 1-4  alkyl group, or \u2014(CH 2 ) n \u2014C(\u2550O)\u2014NHRf, R 2  is a hydrogen atom, a fluorine atom, a chlorine atom, or a trifluoromethyl group; Ra is a C 1-4  alkylpyrazolyl group, a triazolyl group, a tetrazolyl group, or a C 1-4  alkylsulfonylpiperazinyl group, Rf is a fluoro-C 1-3  alkyl group, a hydroxy-C 1-4  alkyl group, a hydroxy-C 3-5  cycloalkyl group, a hydroxy-C 3-5  cycloalkyl-C 1-4  alkyl group, or a C 1-4  alkyl group substituted with Rfa, Rfa is a C 1-4  alkylpyrazolyl group, a fluoro-C 1-3  alkylthiazolyl group, an oxadiazolyl group, or a fluoro-C 1-3  alkyloxadiazolyl group, and n is 0 or 1.

Metadata:
- Claim Count in Document: 2.0
- Percentile: 88.0
- Lexical Diversity: 2.09375
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15203059', '15023894', '15771487', '13391895', '14923525']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8241566106585884
- 35 USC 102 Novelty (BERT): 0.6760085685530902
- Combined Prediction Score: 0.8093418064480385
- Mean Citation Score: 506.41254799999984
- Max Citation Score: 695.1665
- Similarity Product: 646.8169395392836

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test