PATENT CLAIM ANALYSIS

Application Number: 16110698
Application Type: Utility
Filing Date: 2018-08
Publication Date: 2018-12
Patent Classification: ["546", "314000"]

Abstract:
The present invention features compounds having soluble epoxide hydrolase inhibitory activity. The compounds of the invention, alone or in combination with other pharmaceutically active agents, can be used for treating or preventing various medical conditions, such as cardiovascular diseases, respiratory diseases, inflammation, and diabetes.

Claim (Index 1):
A compound having the structure: wherein one of X 1  or X 2  is N and the other is CH; R 1  is hydrogen, C 1 -C 6  acyl, C 1 -C 6  alkyl, C 2 -C 6  alkenyl, C 2 -C 6  alkynyl, C 1 -C 6  heteroalkyl, C 2 -C 6  heteroalkenyl, C 2 -C 6  heteroalkynyl, C 3 -C 10  carbocyclyl, C 6 -C 10  aryl, C 6 -C 10  aryl C 1 -C 6  alkyl, C 2 -C 9  heterocyclyl, C 2 -C 9  heterocyclyl C 1 -C 6  alkyl; R 2  is hydrogen or C 1 -C 6  alkyl; R 3  is hydrogen, hydroxyl, halogen, thiol, C 1 -C 6  acyl, C 1 -C 6  alkyl, C 2 -C 6  alkenyl, C 2 -C 6  alkynyl, C 1 -C 6  heteroalkyl, C 2 -C 6  heteroalkenyl, C 2 -C 6  heteroalkynyl, C 3 -C 10  carbocyclyl, C 6 -C 10  aryl, C 6 -C 10  aryl C 1 -C 6  alkyl, C 2 -C 9  heterocyclyl, C 2 -C 9  heterocyclyl C 1 -C 6  alkyl, \u2014C(O)NHR 4 ; and R 4  is hydrogen, C 1 -C 6  acyl, C 1 -C 6  alkyl, C 2 -C 6  alkenyl, C 2 -C 6  alkynyl, C 1 -C 6  heteroalkyl, C 2 -C 6  heteroalkenyl, C 2 -C 6  heteroalkynyl, C 3 -C 10  carbocyclyl, C 6 -C 10  aryl, C 6 -C 10  aryl C 1 -C 6  alkyl, C 2 -C 9  heterocyclyl, C 2 -C 9  heterocyclyl C 1 -C 6  alkyl; or a pharmaceutically acceptable salt thereof.

Metadata:
- Claim Count in Document: 47.0
- Percentile: 96.0
- Lexical Diversity: 1.26829
- Patent Class: 546.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15504223', '15660114', '15737683', '15114895', '14776184']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7919545276222443
- 35 USC 102 Novelty (BERT): 0.499851009638273
- Combined Prediction Score: 0.7627441758238471
- Mean Citation Score: 263.28891000000004
- Max Citation Score: 303.49783
- Similarity Product: 297.3643475289822

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test