PATENT CLAIM ANALYSIS

Application Number: 16142907
Application Type: Utility
Filing Date: 2018-09
Publication Date: 2019-03
Patent Classification: ["514", "442000"]

Abstract:
The present invention relates to 1-[1-(benzoyl )-pyrrolidine-2-carbonyl]-pyrrolidine-2-carbonitrile derivatives having pharmacological activity formula (I) to processes of preparation of such compounds, to pharmaceutical compositions comprising them, and to their use in therapy and/or prophylaxis of a cognitive disorder.

Claim (Index 14):
A method for the treatment or prophylaxis of a cognitive disorder in a patient, comprising administering to the patient in need of such treatment or prophylaxis a therapeutic amount of a compound of formula (I): wherein R 1 , R 2 , R 3  and R 4  are independently selected from the group consisting of C 1-4  alkoxy, C 1-4  alkylcarbonyloxy, benzyloxy, phenylcarbonyloxy, naphthylcarbonyloxy, quinolinylcarbonyloxy, isoquinolinylcarbonyloxy, trifluoromethyl, halogen and hydrogen; R 5  is selected from the group consisting of halogen, nitrile, C 1-4  alkoxy, C 1-4  alkylthio, C 1-4  alkyl, phenyl, phenoxy, phenylthio and trifluoromethyl; R 6  is selected from the group consisting of hydrogen, fluor and methyl; or a pharmaceutically acceptable salt, isomer, prodrug or solvate thereof.

Metadata:
- Claim Count in Document: 56.0
- Percentile: 97.0
- Lexical Diversity: 1.225
- Patent Class: 514.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['14436715', '15776296', '12468632', '15738900', '10481543']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7189114258174081
- 35 USC 102 Novelty (BERT): 0.597643253505252
- Combined Prediction Score: 0.7067846085861925
- Mean Citation Score: 310.28643
- Max Citation Score: 611.5246
- Similarity Product: 400.8545907906652

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test