PATENT CLAIM ANALYSIS

Application Number: 15866429
Application Type: Utility
Filing Date: 2018-01
Publication Date: 2018-05
Patent Classification: ["544", "234000"]

Abstract:
The invention provides novel compounds having the general formula: wherein R 1  to R 6  are as described herein, compositions including the compounds and methods of using the compounds.

Claim (Index 9):
The compound according to  claim 1 , which compound is selected from the group consisting of:\n 9,10-Dimethoxy-2-oxo-6,7-dihydropyrido[2,1-a]phthalazine-3-carboxylic acid; 9,10-Dimethoxy-6-methyl-2-oxo-7H-pyrido[2,1-a]phthalazine-3-carboxylic acid; 6-Allyl-9,10-dimethoxy-2-oxo-7H-pyrido[2,1-a]phthalazine-3-carboxylic acid; 6-Isopropyl-9,10-dimethoxy-2-oxo-7H-pyrido[2,1-a]phthalazine-3-carboxylic acid; 6-Isobutyl-9,10-dimethoxy-2-oxo-7H-pyrido[2,1-a]phthalazine-3-carboxylic acid; 6-Isobutyl-10-methoxy-9-(3-methoxypropoxy)-2-oxo-7H-pyrido[2,1-a]phthalazine-3-carboxylic acid; 6-Isobutyl-10-methoxy-2-oxo-9-(2,2,2-trifluoroethoxy)-7H-pyrido[2,1-a]phthalazine-3-carboxylic acid; 6-Isobutyl-10-methoxy-2-oxo-9-(tetrahydropyran-4-ylmethoxy)-7H-pyrido[2,1-a]phthalazine-3-carboxylic acid; 6-Isobutyl-10-methoxy-9-(3-methylsulfonylpropoxy)-2-oxo-7H-pyrido[2,1-a]phthalazine-3-carboxylic acid; 6-Isobutyl-10-methoxy-9-(2-morpholinoethoxy)-2-oxo-7H-pyrido[2,1-a]phthalazine-3-carboxylic acid; 9-(3-Hydroxy-2,2-dimethyl-propoxy)-6-isobutyl-10-methoxy-2-oxo-7H-pyrido[2,1-a]phthalazine-3-carboxylic acid; 9-(4-Carboxybutoxy)-6-isobutyl-10-methoxy-2-oxo-7H-pyrido[2,1-a]phthalazine-3-carboxylic acid; 9-(3-Cyanopropoxy)-6-isobutyl-10-methoxy-2-oxo-7H-pyrido[2,1-a]phthalazine-3-carboxylic acid; 9-[5-(Tert-butoxycarbonylamino)pentoxy]-6-isobutyl-10-methoxy-2-oxo-7H-pyrido[2,1-a]phthalazine-3-carboxylic acid; and, 9-(5-Aminopentoxy)-6-isobutyl-10-methoxy-2-oxo-7H-pyrido[2,1-a]phthalazine-3-carboxylic acid hydrochloride; or, a pharmaceutically acceptable salt, or an enantiomers, or a diastereomer thereof.

Metadata:
- Claim Count in Document: 5.0
- Percentile: 86.0
- Lexical Diversity: 1.18519
- Patent Class: 544.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15674810', '14926393', '15144996', '15639966', '14610454']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8152341676862515
- 35 USC 102 Novelty (BERT): 0.552962988316495
- Combined Prediction Score: 0.7890070497492758
- Mean Citation Score: 386.514236
- Max Citation Score: 415.42966
- Similarity Product: 364.57689081934456

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test