PATENT CLAIM ANALYSIS

Application Number: 15753264
Application Type: Utility
Filing Date: 2018-02
Publication Date: 2018-08
Patent Classification: ["514", "080000"]

Abstract:
Various embodiments relate to a compound of the formula (I): wherein X, X 1 , R 1 -R 4  and R 7  are defined herein, as well as pharmaceutical compositions comprising compounds of the formula (I) and methods of treating an HIV infection comprising administering a therapeutically effective amount of one or more compounds of formula (I), or a pharmaceutical compositions comprising compounds of the formula (I), to a patient in need thereof.

Claim (Index 1):
A compound of the formula (I): or a pharmaceutically acceptable salt, polymorph, prodrug, solvate or clathrate thereof, wherein: n is an integer from 0 to 3; X and X 1  are each, independently, (\u2014CH 2 \u2014) m , wherein m is 1 or 2; R 1  is \u2014N 3  or \u2014NR 5 2 , wherein each R 5  is, independently, H, unsubstituted or substituted alkyl, unsubstituted or substituted alkenyl or a nitrogen protecting group, such as an alkyloxycarbonyl group, including a t-butyl oxycarbonyl group; R 7  is H or unsubstituted or substituted alkyl or R 1  and R 7 , together with the carbon atom to which they are attached, form a heterocycle; R 2  is unsubstituted or substituted alkyl, unsubstituted or substituted alkenyl, unsubstituted or substituted alkoxy, unsubstituted or substituted hydroxyalkyl, halo, unsubstituted or substituted heterocyclylalkyloxy, \u2014O\u2014(CH 2 ) 0-2 P(O)(OR 6 ) 2 , wherein each R 6  is independently H or unsubstituted or substituted alkyl or substituted or unsubstituted aryl or R 1  is \u2014NR 5 2 , wherein one R 5  and one R 2  are joined to represent the group \u2014(CH 2 ) p (CHCH) d (CH 2 ) q O\u2014 wherein p is an integer from 0 to 5, d is 0 or 1, and q is an integer from 0 to 5; R 3  is substituted or unsubstituted alkyl; and R 4  is unsubstituted or substituted aryl, unsubstituted or substituted benzthiazole, unsubstituted or substituted benzoxazole, unsubstituted or substituted benzofuranyl or unsubstituted or substituted indolyl.

Metadata:
- Claim Count in Document: 50.0
- Percentile: 88.0
- Lexical Diversity: 1.8125
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15311806', '15400766', '10166979', '14820488', '14238374']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7433195691193882
- 35 USC 102 Novelty (BERT): 0.5247067730448167
- Combined Prediction Score: 0.721458289511931
- Mean Citation Score: 246.022912
- Max Citation Score: 313.0263
- Similarity Product: 243.7591566477477

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test