PATENT CLAIM ANALYSIS

Application Number: 16270965
Application Type: Utility
Filing Date: 2019-02
Publication Date: 2019-08
Patent Classification: ["514", "510000"]

Abstract:
The present disclosure provides treprostinil derivatives that can act as prodrugs of treprostinil. The treprostinil derivatives can be used to treat any conditions responsive to treatment with treprostinil, including pulmonary hypertension, such as pulmonary arterial hypertension.

Claim (Index 25):
A compound of Formula (I): wherein:\n R 1  and R 2  independently are hydrogen, \n wherein:\n R 6  in each occurrence independently is hydrogen, R 3 , \u2014C(\u2550O)R 3 , \u2014C(\u2550O)OR 3  or \u2014C(\u2550O)NR 9 R 10 ; \n R 3  in each occurrence independently is alkyl, haloalkyl, -alkylaryl, cycloalkyl, heterocyclyl, aryl or heteroaryl, each of which may optionally be substituted; \n R 9  and R 10  in each occurrence independently are hydrogen, alkyl, -alkylaryl, cycloalkyl, heterocyclyl, aryl or heteroaryl; or\n R 9  and R 10  and the nitrogen atom to which they are connected form a heterocyclic or heteroaryl ring; \n \n j in each occurrence independently is an integer from 0 to 4; and \n t in each occurrence independently is an integer from 1 to 9; \n with the proviso that both R 1  and R 2  are not hydrogen; \n or a pharmaceutically acceptable salt, solvate, hydrate, clathrate, polymorph or stereoisomer thereof.

Metadata:
- Claim Count in Document: 122.0
- Percentile: 99.0
- Lexical Diversity: 1.42857
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['14742544', '15617243', '15927636', '15473434', '15178637']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8061029568928312
- 35 USC 102 Novelty (BERT): 0.5633409821538793
- Combined Prediction Score: 0.781826759418936
- Mean Citation Score: 245.799044
- Max Citation Score: 255.80673
- Similarity Product: 194.9080692155707

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test