PATENT CLAIM ANALYSIS

Application Number: 16023232
Application Type: Utility
Filing Date: 2018-06
Publication Date: 2018-10
Patent Classification: ["549", "397000"]

Abstract:
Compounds of Formula (A) are described herein and the uses thereof for the treatment of diseases, conditions and/or disorders mediated by pharmaceutical compositions and the uses thereof as asialoglycoprotein receptor (ASGPR) targeting agents.

Claim (Index 2):
A compound of Formula (A) wherein R 1  is \u2014Z\u2014X\u2014Y, \u2014Z\u2014Y, or \u2014X\u2014Y wherein X is a linker of any of structures L1, L2, L9 or L10 each Q is independently absent or is C(O), C(O)\u2014NR 4 , NR 4 \u2014C(O), O\u2014C(O)\u2014NR 4 , NR 4 \u2014C(O)\u2014O, \u2014CH 2 \u2014, or \u2014O\u2014, wherein at least two carbon atoms separate the \u2014O\u2014 from any other heteroatom group; each T is independently absent or is alkylene, wherein one or more \u2014CH 2 \u2014 groups of the alkylene, may each independently be replaced with a \u2014O\u2014, wherein the \u2014O\u2014 are separated by at least 2 carbon atoms; Y is an amino acid sequence, a nucleic acid sequence, or an oligomer, and Z is absent; each n is independently 0, 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16, 17, 18, 19, 20, 21, 22, 23, 24, 25, 26, 27, 28, 29, 30, 31, 32, 33, 34, 35, 36, 37, 38, 39, or 40, wherein if n is greater than 1, each T and each Q of each (T-Q-T-Q) is independently selected; R 2  is \u2014N(R 3 )\u2014C(O)\u2014R 3  or \u2014N(R 3 )\u2014C(O)\u2014OR 3 ; and each R 3  is independently \u2014H, \u2014(C 1 -C 5 )alkyl, halo-substituted (C 1 -C 5 )alkyl, or (C 3 -C 6 )cycloalkyl; and or a pharmaceutically acceptable salt thereof.

Metadata:
- Claim Count in Document: 13.0
- Percentile: 94.0
- Lexical Diversity: 1.25806
- Patent Class: 549.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15434508', '15093178', '14714484', '14917792', '14779191']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7965372646687389
- 35 USC 102 Novelty (BERT): 0.6117137461678163
- Combined Prediction Score: 0.7780549128186467
- Mean Citation Score: 444.961634
- Max Citation Score: 550.91327
- Similarity Product: 509.4152943313677

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test