PATENT CLAIM ANALYSIS

Application Number: 16055362
Application Type: Utility
Filing Date: 2018-08
Publication Date: 2019-01
Patent Classification: ["514", "259300"]

Abstract:
This invention relates to compounds of the general formula: in which the variable groups are as defined herein, and to their preparation and use.

Claim (Index 27):
The compound of  claim 23 , having the formula: wherein:\n Ring D represents a 5- or 6-membered heterocyclyl or heteroaryl ring comprising carbon atoms and 1-3 heteroatoms independently chosen from O, N and S(O) r ; \n L 2  is chosen from (CH 2 ) z , O(CH 2 ) x , NR 3 (CH 2 ) x , S(CH 2 ) x  and (CH 2 ) x NR 3 C(O)(CH 2 ) x  in either direction; \n R d , at each occurrence, is H, halo, \u2550O, \u2014CN, \u2014NO 2 , \u2014R 4 , \u2014OR 2 , \u2014NR 2 R 3 , \u2014C(O)YR 2 , \u2014OC(O)YR 2 , \u2014NR 2 C(O)YR 2 , \u2014SC(O)YR 2 , \u2014NR 2 C(\u2550S)YR 2 , \u2014OC(\u2550S)YR 2 , \u2014C(\u2550S)YR 2 , \u2014YC(\u2550NR 3 )YR 2 , \u2014YP(\u2550O)(YR 4 )(YR 4 ), \u2014Si(R 2 ) 3 , \u2014NR 2 SO 2 R 2 , \u2014S(O) r R 2 , \u2014SO 2 NR 2 R 3  or \u2014NR 2 SO 2 NR 2 R 3 , wherein each Y is independently a bond, \u2014O\u2014, \u2014S\u2014 or \u2014NR 3 \u2014; \n R 2  and R 3  are independently H, alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, heterocyclyl, or heteroaryl; \n or R 2  and R 3 , taken together with the atom to which they are attached, form a 5- or 6-membered saturated, partially saturated or unsaturated ring, which contains 0-2 heteroatoms selected from N, O and S(O) r ; \n each occurrence of R 4  is independently alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, heterocyclyl, or heteroaryl; \n each of the alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl and heterocyclyl moieties is optionally substituted with one or more groups selected from halo, \u2014CN, \u2014R 4 , \u2014OR 2 , \u2014S(O) r R 2 , \u2014SO 2 NR 2 R 3 , \u2014NR 2 R 3 , \u2014(CO)YR 2 , \u2014O(CO)YR 2 , \u2014NR 2 (CO)YR 2 , \u2014S(CO)YR 2 , \u2014NR 2 C(\u2550S)YR 2 , \u2014OC(\u2550S)YR 2 , \u2014C(\u2550S)YR 2 , \u2014YC(\u2550NR 3 )Y\u2032R 2 , \u2014COCOR 2 , \u2014COMCOR 2 , \u2014YP(\u2550O)(YR 4 )(YR 4 ), \u2014Si(R 2 ) 3 , \u2014NO 2 , \u2014NR 2 SO 2 R 2 , \u2014NR 2 SO 2 NR 2 R 3 , \u2550O, \u2550S, \u2550NH, \u2550NNR 2 R 3 , \u2550NNHC(O)R 2 , \u2550NNHCO 2 R 2 , and \u2550NNHSO 2 R 2 , wherein M is a 1-6 carbon alkyl group; \n each of the aryl and heteroaryl moieties is optionally substituted on an unsaturated carbon atom with one or more groups selected from halo, \u2014CN, \u2014R 4 , \u2014OR 2 , \u2014S(O) r R 2 , \u2014SO 2 NR 2 R 3 , \u2014NR 2 R 3 , \u2014(CO)YR 2 , \u2014O(CO)YR 2 , \u2014NR 2 (CO)YR 2 , \u2014S(CO)YR 2 , \u2014NR 2 C(\u2550S)YR 2 , \u2014OC(\u2550S)YR 2 , \u2014C(\u2550S)YR 2 , \u2014YC(\u2550NR 3 )Y\u2032R 2 , \u2014COCOR 2 , \u2014COMCOR 2 , \u2014YP(\u2550O)(YR 4 )(YR 4 ), \u2014Si(R 2 ) 3 , \u2014NO 2 , \u2014NR 2 SO 2 R 2 , and \u2014NR 2 SO 2 NR 2 R 3 ; \n w is 0, 1, 2, 3, 4 or 5; \n x is 0, 1, 2 or 3; and \n z is 1, 2, 3 or 4.

Metadata:
- Claim Count in Document: 56.0
- Percentile: 96.0
- Lexical Diversity: 1.125
- Patent Class: 514.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['14296016', '13801619', '13614838', '12227002', '13801116']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7531228872425877
- 35 USC 102 Novelty (BERT): 0.5343007031525567
- Combined Prediction Score: 0.7312406688335846
- Mean Citation Score: 333.1144020000001
- Max Citation Score: 358.56778
- Similarity Product: 346.59969518710966

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test