PATENT CLAIM ANALYSIS

Application Number: 15896851
Application Type: Utility
Filing Date: 2018-02
Publication Date: 2018-06
Patent Classification: ["514", "428000"]

Abstract:
Novel amisulpride derivatives and pharmaceutical compositions thereof are disclosed. The amisulpride derivative disclosed herein or a pharmaceutical composition thereof may have better membrane permeability compared to amisulpride. The amisulpride derivative disclosed herein or a pharmaceutical composition thereof may be used for antagonizing dopamine and/or serotonin (e.g., 5-HT2a) and/or α2 receptor in a subject, either individually or in combination with other CNS active agents. The amisulpride derivative disclosed herein or a pharmaceutical composition thereof may be used for treating one or more conditions responsive to modulation of dopamine and/or serotonin (e.g., 5-HT2a) and/or α2 receptor in a subject, either individually or in combination with other CNS active agents. The amisulpride derivative disclosed herein or a pharmaceutical composition thereof may be used for treating one or more disorders associated with an abnormality in levels of dopamine and/or serotonin in the brain, either individually or in combination with other CNS active agents.

Claim (Index 27):
The method of  claim 10 , wherein the serotonin receptor is 5-HT 2a  receptor.

Metadata:
- Claim Count in Document: 162.0
- Percentile: 88.0
- Lexical Diversity: 2.67213
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15824966', '15416964', '15836261', '15593654', '11643190']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7658343570117302
- 35 USC 102 Novelty (BERT): 0.5611840252058675
- Combined Prediction Score: 0.745369323831144
- Mean Citation Score: 292.8562740000001
- Max Citation Score: 456.31693
- Similarity Product: 334.54723654441835

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test