PATENT CLAIM ANALYSIS

Application Number: 16003600
Application Type: Utility
Filing Date: 2018-06
Publication Date: 2019-02
Patent Classification: ["514", "220000"]

Abstract:
The present invention relates to tricyclic quinoline and quinoxaline derivatives, to a pharmaceutical composition containing such compounds, to their use as modulators, especially agonists or partial agonists, of the 5-HT 2C  receptor, their use for preparing a medicament for the prevention or treatment of conditions and disorders which respond to the modulation of 5-HT 2C  receptor, and to a method for preventing or treating conditions and disorders which respond to the modulation of 5-HT 2C  receptor.

Claim (Index 51):
A compound selected from the group consisting of\n trans-12a-methyl-4,5,6,7,10,11,12,12a-octahydrocyclopenta[c][1,4]diazepino[6,7,1-ij]quinolin-9(9aH)-one; cis-12a-methyl-4,5,6,7,10,11,12,12a-octahydrocyclopenta[c][1,4]diazepino[6,7,1-ij]quinolin-9(9aH)-one; cis-12a-methyl-4,5,6,7,9,9a,10,11,12,12a-decahydrocyclopenta[c][1,4]diazepino[6,7,1-ij]quinoline; trans-12a-methyl-4,5,6,7,9,9a,10,11,12,12a-decahydrocyclopenta[c][1,4]diazepino[6,7,1-ij]quinoline; (R)-5,6,7,9,9a,10,11,12-octahydro-4H-[1,4]diazepino[1,7,6-de]pyrrolo[1,2-a]quinoxaline; (S)-5,6,7,9,9a,10,11,12-octahydro-4H-[1,4]diazepino[1,7,6-de]pyrrolo[1,2-a]quinoxaline; and 3-benzyl-2\u2032,3\u2032,7\u2032,8\u2032,9\u2032,10\u2032-hexahydro-1H-3\u2032,8\u2032,10a\u2032-triaza-cyclohepta[de]naphthalene; or a pharmaceutically acceptable salt thereof.

Metadata:
- Claim Count in Document: 140.0
- Percentile: 94.0
- Lexical Diversity: 1.88636
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['14026354', '13838788', '14868835', '14657916', '14657840']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7758532183576378
- 35 USC 102 Novelty (BERT): 0.5273087749599029
- Combined Prediction Score: 0.7509987740178643
- Mean Citation Score: 284.69573
- Max Citation Score: 312.41757
- Similarity Product: 203.0603518576456

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test