PATENT CLAIM ANALYSIS

Application Number: 16394308
Application Type: Utility
Filing Date: 2019-04
Publication Date: 2019-08
Patent Classification: ["514", "253000"]

Abstract:
Compounds of formula (I): wherein R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , R 7 , R 8 , R 14 , W, A and n are as defined in the description. Medicinal products containing the same which are useful in treating conditions requiring a pro-apoptotic agent.

Claim (Index 2):
The method according to  claim 1 , wherein:\n R 1  and R 2  independently of one another represent a halogen atom, a linear or branched (C 1 -C 6 )alkyl group, a hydroxy group, a linear or branched (C 1 -C 6 )alkoxy group, or the substituents of the pair (R 1 , R 2 ), together with the carbon atoms carrying them, form an aromatic ring having from 5 to 7 ring members, which ring may contain from 1 to 3 nitrogen atoms, R 3  represents a hydrogen atom, a halogen atom, a linear or branched (C 1 -C 6 )alkyl group, a hydroxy group, a linear or branched (C 1 -C 6 )alkoxy group, or \u2014O-alkyl(C 1 -C 6 )\u2014NR 11 R 11 \u2032, R 4  and R 5  independently of one another represent a hydrogen atom, a halogen atom, a linear or branched (C 1 -C 6 )alkyl group, a hydroxy group, a linear or branched (C 1 -C 6 )alkoxy group, R 6  and R 7  independently of one another represent a hydrogen atom, a halogen atom, a linear or branched (C 1 -C 6 )alkyl group, a linear or branched (C 1 -C 6 )polyhaloalkyl group, a hydroxy group, a linear or branched (C 1 -C 6 )alkoxy group, a cyano group, a nitro group, -alkyl(C 0 -C 6 )\u2014NR 11 R 11 \u2032, -alkyl(C 0 -C 6 )-Cy 1 , \u2014O-alkyl(C 1 -C 6 )\u2014R 12 , or \u2014C(O)\u2014NR 11 R 11 \u2032, R 8  represents a hydrogen atom, a linear or branched (C 1 -C 8 )alkyl group, or a \u2014CHR a R b  group, R 9  represents a hydrogen atom, a linear or branched (C 1 -C 6 )alkyl group, a linear or branched (C 2 -C 6 )alkenyl group, a linear or branched (C 2 -C 6 )alkynyl group, -Cy 2 , or a halogen atom, R 10  represents a hydrogen atom, a linear or branched (C 1 -C 6 )alkyl group, a linear or branched (C 2 -C 6 )alkenyl group, a linear or branched (C 2 -C 6 )alkynyl group, an arylalkyl(C 1 -C 6 ) group, a cycloalkylalkyl(C 1 -C 6 ) group, a linear or branched (C 1 -C 6 )polyhaloalkyl, or -alkyl(C 1 -C 6 )\u2014O\u2014Cy 4 , or the substituents of the pair (R 9 , R 10 ), when grafted onto two adjacent carbon atoms, together with the carbon atoms carrying them, form a non-aromatic ring having from 5 to 7 ring members, which ring may contain from 1 to 3 heteroatoms selected from oxygen, sulphur and nitrogen, R 11  and R 11 \u2032 independently of one another represent a hydrogen atom, a linear or branched (C 1 -C 6 )alkyl group, or the substituents of the pair (R 11 , R 11 \u2032), together with the nitrogen atom carrying them, form a non-aromatic ring having from 5 to 7 ring members, which ring may contain, in addition to the nitrogen atom, from 1 to 3 heteroatoms selected from oxygen and nitrogen, wherein the nitrogen be substituted by a linear or branched (C 1 -C 6 )alkyl group, R 12  represents -Cy 5  or -Cy 5 -alkyl(C 0 -C 6 )-Cy 6 , W represents a \u2014NH\u2014 group or an oxygen atom, wherein the aryl, heteroaryl, cycloalkyl and heterocycloalkyl groups so defined and the alkyl, alkenyl, alkynyl, alkoxy groups, may be substituted by from 1 to 4 groups selected from optionally substituted linear or branched (C 1 -C 6 )alkyl, optionally substituted linear or branched (C 1 -C 6 )alkoxy, hydroxy, oxo (or N-oxide where appropriate), \u2014C(O)\u2014OR\u2032, \u2014C(O)\u2014NR\u2032R\u2033, \u2014O\u2014C(O)\u2014NR\u2032R\u2033, \u2014NR\u2032R\u2033, \u2014O\u2014P(O)(OR\u2032) 2 , \u2014O\u2014P(O)(O \u2212 M + ) 2 , linear or branched (C 1 -C 6 )polyhaloalkyl, halogen, or an aldohexose of formula: in which each R\u2032 is independent; wherein R\u2032 and R\u2033, independently of one another, represent a hydrogen atom or an optionally substituted linear or branched (C 1 -C 6 )alkyl group and M +  represents a pharmaceutically acceptable monovalent cation.

Metadata:
- Claim Count in Document: 95.0
- Percentile: 100.0
- Lexical Diversity: 1.5
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15738186', '15737479', '15737783', '15738601', '15492306']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8002129151099601
- 35 USC 102 Novelty (BERT): 0.5747077514519726
- Combined Prediction Score: 0.7776623987441613
- Mean Citation Score: 423.82738200000006
- Max Citation Score: 447.99300000000005
- Similarity Product: 411.32288053572177

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test