PATENT CLAIM ANALYSIS

Application Number: 16155846
Application Type: Utility
Filing Date: 2018-10
Publication Date: 2019-02
Patent Classification: ["544", "281000"]

Abstract:
The present teachings provide a compound represented by structural formula (I-0), or a pharmaceutically acceptable salt thereof. Also described are pharmaceutical compositions and methods of use thereof.

Claim (Index 3):
A compound represented by the following structural formula: or a pharmaceutically acceptable salt thereof, wherein:\n R is phenyl or monocyclic 5-6 membered heteroaryl, both of which are substituted with \u2014C(\u2550O)NR d R e , \u2014NHC(\u2550O)R 5 , \u2014C(\u2550S)NR d R e , or \u2014NHC(\u2550S)R 5  and optionally substituted with one or more groups selected from halogen, hydroxy, (C 1 -C 3 )alkyl, (C 1 -C 3 )haloalkyl, (C 1- C 3 )alkoxy, and (C 1 -C 3 )haloalkoxy; \n R 1  is \u2014NR a1 R b1 , \u2014OR c1 , \u2014SR c1 , \u2014SOR c1 , or \u2014SO 2 R c1 ; \n R 2  is \u2014NR a2 R b2 , \u2014OR c2 , \u2014SR c2 , optionally substituted phenyl or optionally substituted 5-6 membered monocyclic heteroaryl; \n R 5  is optionally substituted (C 1 -C 3 )alkyl, optionally substituted (C 3 -C 7 )cycloalkyl, optionally substituted 3-7 membered monocyclic heterocycloalkyl, optionally substituted phenyl, or optionally substituted 5-6 membered monocyclic heteroaryl; \n R a1  and R b1  are each independently selected from \u2014H, optionally substituted (C 1 -C 6 )alkyl, optionally substituted (C 3 -C 7 )cycloalkyl, optionally substituted 3-7 membered monocyclic heterocycloalkyl, optionally substituted phenyl, and optionally substituted 5-6 membered monocyclic heteroaryl; \n R a2  and R b2  are each independently selected from \u2014H, optionally substituted (C 1 -C 6 )alkyl, optionally substituted (C 3 -C 7 )cycloalkyl, optionally substituted 3-7 membered monocyclic heterocycloalkyl, optionally substituted phenyl, and optionally substituted 5-6 membered monocyclic heteroaryl; or \n R a2  and R b2 , together with the nitrogen to which they are attached, form an optionally substituted 3-7 membered ring; \n R c1  is optionally substituted (C 1 -C 6 )alkyl, optionally substituted (C 3 -C 7 ) cycloalkyl, optionally substituted 3-7 membered monocyclic heterocycloalkyl, optionally substituted phenyl, or optionally substituted 5-6 membered monocyclic heteroaryl; \n R c2  is optionally substituted (C 1 -C 6 )alkyl, optionally substituted (C 3 -C 7 )cycloalkyl, optionally substituted 3-7 membered monocyclic heterocycloalkyl, optionally substituted phenyl, or optionally substituted 5-6 membered monocyclic heteroaryl; and \n R d  and R e  are each independently selected from \u2014H, optionally substituted (C 1 -C 7 )alkyl, optionally substituted (C 3 -C 7 )cycloalkyl, optionally substituted 3-7 membered monocyclic heterocycloalkyl, optionally substituted phenyl, and optionally substituted 5-6 membered monocyclic heteroaryl; or \n R d  and R e , together with the nitrogen to which they are attached, form an optionally substituted 3-7 membered ring.

Metadata:
- Claim Count in Document: 113.0
- Percentile: 97.0
- Lexical Diversity: 1.10345
- Patent Class: 544.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['14443072', '15434275', '14351381', '15543826', '14382123']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7916642280023092
- 35 USC 102 Novelty (BERT): 0.6023103076160806
- Combined Prediction Score: 0.7727288359636864
- Mean Citation Score: 421.832804
- Max Citation Score: 504.46133
- Similarity Product: 499.6592519216717

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test