PATENT CLAIM ANALYSIS

Application Number: 16156447
Application Type: Utility
Filing Date: 2018-10
Publication Date: 2019-08
Patent Classification: ["514", "287000"]

Abstract:
The invention relates to compound of the formula (I′) or a salt thereof, wherein the substituents are as defined in the specification; to its preparation, to its use as medicament and to medicaments comprising it.

Claim (Index 17):
The method of  claim 10 , wherein the compound or a pharmaceutically acceptable salt thereof is selected from:\n 3-cyclobutyl-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 3-cyclobutyl-5-methyl-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 3-isopropyl-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 3-isopropyl-5-methyl-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 8-fluoro-3-isopropyl-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 8-fluoro-3-isopropyl-5-methyl-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 8-chloro-3-isopropyl-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 8-chloro-3-isopropyl-5-methyl-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 3-isopropyl-8-methyl-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 3-isopropyl-5,8-dimethyl-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 9-isopropyl-8-phenyl-1H-indolo[1,7-ab][1,6]naphthyridine-6,7(2H, 8H)-dione; 7-isopropyl-6-phenylthieno[2,3-b][1,6]naphthyridine-4,5(6H,9H)-dione; 7-isopropyl-9-methyl-6-phenylthieno[2,3-b][1,6]naphthyridine-4,5(6H, 9H)-dione; 7-isopropyl-2-methyl-6-phenylthieno[2,3-b][1,6]naphthyridine-4,5(6H,9H)-dione; 7-isopropyl-2,9-dimethyl-6-phenylthieno[2,3-b][1,6]naphthyridine-4,5(6H,9H)-dione; 6-isopropyl-7-phenylthieno[3,2-b][1,6]naphthyridine-8,9(4H,7H)-dione; 6-isopropyl-4-methyl-7-phenylthieno[3,2-b][1,6]naphthyridine-8,9(4H,7H)-dione; 6-isopropyl-2-methyl-7-phenylthieno[3,2-b][1,6]naphthyridine-8,9(4H,7H)-dione; 6-isopropyl-2,4-dimethyl-7-phenylthieno[3,2-b][1,6]naphthyridine-8,9(4H, 7H)-dione; 6-isopropyl-3-methyl-7-phenylthieno[3,2-b][1,6]naphthyridine-8,9(4H,7H)-dione; 6-isopropyl-3,4-dimethyl-7-phenylthieno[3,2-b][1,6]naphthyridine-8,9(4H,7H)-dione; 3-isopropyl-2-phenyl-6,7,8,9-tetrahydrobenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 3-isopropyl-2-phenyl-5,6,7,8-tetrahydro-1H-cyclopenta[b][1,6]naphthyridine-1,9(2H)-dione; 3-cyclobutyl-5-methyl-2-phenyl-5,6,7,8-tetrahydro-1H-cyclopenta[b][1,6]naphthyridine-1,9(2H)-dione; 3-cyclobutyl-2-phenyl-5,6,7,8-tetrahydro-1H-cyclopenta[b][1,6]naphthyridine-1,9(2H)-dione; 3-cyclobutyl-5-methyl-2-phenyl-6,7,8,9-tetrahydrobenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 7-cyclobutyl-9-methyl-6-phenylthieno[2,3-b][1,6]naphthyridine-4,5(6H,9H)-dione; 7-cyclobutyl-2,9-dimethyl-6-phenylthieno[2,3-b][1,6]naphthyridine-4,5(6H,9H)-dione; 7-cyclobutyl-6-phenylthieno[2,3-b][1,6]naphthyridine-4,5(6H, 9H)-dione; 7-cyclobutyl-2-methyl-6-phenylthieno[2,3-b][1,6]naphthyridine-4,5(6H,9H)-dione; 6-cyclobutyl-4-methyl-7-phenylthieno[3,2-b][1,6]naphthyridine-8,9(4H,7H)-dione; 6-cyclobutyl-7-phenylthieno[3,2-b][1,6]naphthyridine-8,9(4H, 7H)-dione; 6-cyclobutyl-2,4-dimethyl-7-phenylthieno[3,2-b][1,6]naphthyridine-8,9(4H,7H)-dione; 6-cyclobutyl-2-methyl-7-phenylthieno[3,2-b][1,6]naphthyridine-8,9(4H,7H)-dione; 3-cyclobutyl-5,8-dimethyl-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 3-cyclobutyl-8-fluoro-5-methyl-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 8-chloro-3-cyclobutyl-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 3-cyclobutyl-8-methyl-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 8-chloro-3-cyclobutyl-5-methyl-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 3-isopropyl-6-methoxy-5-methyl-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 3-cyclobutyl-8-fluoro-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 9-cyclobutyl-8-phenyl-1H-indolo[1,7-ab][1,6]naphthyridine-6,7(2H,8H)-dione; 3-cyclobutyl-6-methoxy-5-methyl-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 3-isopropyl-6-methoxy-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 3-cyclobutyl-6-methoxy-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 3-isopropyl-8-methoxy-5-methyl-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 3-isopropyl-8-methoxy-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 8-hydroxy-3-isopropyl-5-methyl-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 6-hydroxy-3-isopropyl-5-methyl-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 3-cyclobutyl-2-cyclopentylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 3-cyclobutyl-2-cyclopentyl-5-methylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 2-cyclopentyl-3-isopropylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 2-cyclopentyl-3-isopropyl-5-methylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 3-cyclobutyl-2-(pyridin-2-yl)benzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 3-cyclobutyl-5-methyl-2-(pyridin-2-yl)benzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 3-cyclobutyl-2-(pyrrolidin-1-yl)benzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 3-cyclobutyl-5-methyl-2-(pyrrolidin-1-yl)benzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 4-chloro-3-isopropyl-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; 4-chloro-3-isopropyl-5-methyl-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione; and 4-bromo-3-isopropyl-5-methyl-2-phenylbenzo[b][1,6]naphthyridine-1,10(2H,5H)-dione.

Metadata:
- Claim Count in Document: 17.0
- Percentile: 97.0
- Lexical Diversity: 1.24242
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['14728613', '14652102', '15554801', '15315582', '14763468']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7350052989123712
- 35 USC 102 Novelty (BERT): 0.6552720500029056
- Combined Prediction Score: 0.7270319740214246
- Mean Citation Score: 382.642246
- Max Citation Score: 668.1334
- Similarity Product: 572.9820267673731

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test