PATENT CLAIM ANALYSIS

Application Number: 16060714
Application Type: Utility
Filing Date: 2018-06
Publication Date: 2019-01
Patent Classification: ["514", "274000"]

Abstract:
The present invention provides a modulator of Kv3.1 and/or Kv3.2 and/or Kv3.3 channels for use in the prophylaxis or treatment of pain. Modulators for use in the prophylaxis or treatment of pain include compounds of formula (I) or a pharmaceutically acceptable salt and/or solvate thereof and/or derivative thereof: (I).

Claim (Index 27):
The method according to  claim 26 , wherein the modulator of Kv3.1 and/or Kv3.2 and/or Kv3.3 is selected from a compound of formulae (IA), (IB), (IC), (ID), (IE) and (IF): wherein:\n R 1  is H, C 1-4  alkyl, halo, haloC 1-4  alkyl; \n R 2  is H, C 1-4  alkyl, C 3-5  spiro carbocyclyl, or haloC 1-4  alkyl; \n R 3  is H, C 1-4  alkyl, haloC 1-4  alkyl or halo; or R 3  is absent \n R 13  is H or is absent; \n R 14  is H or is absent; \n A is a 5 or 6 membered saturated or unsaturated heterocycle, with at least one O atom; \n R 4  is C 1-4  alkyl; \n R 5  is H or C 1-4  alkyl;\n wherein when R 5  is present, R 4  and R 5  have the stereochemical arrangement: \n \n R 16  is C 1-4  alkyl, C 1-4  alkoxy, halo-C 1-4  alkyl, halo-C 1-4  alkoxy; R 17  is H, cyano or C 1-4  alkyl; with the proviso that when R 17  is H, R 16  is not in the para position; R 23  is C 1-4  alkyl, Cl, CF 3 , O\u2014C 1-4  alkyl, OCF 3  or N(CH 3 ) 2 ; R 24  is H, Cl, F, C 1-4  alkyl, O\u2014C 1-4  alkyl, CN, OCF 3 ; R 22 , R 25  and R 26  are H; X is CH or N and Y is CH or N.

Metadata:
- Claim Count in Document: 54.0
- Percentile: 94.0
- Lexical Diversity: 1.6
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['14403011', '15730559', '14361510', '15208329', '14403048']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8172663369831011
- 35 USC 102 Novelty (BERT): 0.6224721300121058
- Combined Prediction Score: 0.7977869162860016
- Mean Citation Score: 527.578932
- Max Citation Score: 633.7182
- Similarity Product: 485.2358617053866

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test