PATENT CLAIM ANALYSIS

Application Number: 15874500
Application Type: Utility
Filing Date: 2018-01
Publication Date: 2018-08
Patent Classification: ["514", "236500"]

Abstract:
Disclosed are compounds, such as pyridazinones, that can be, inter alia, used for treating cancer.

Claim (Index 32):
A compound of Formula I or a pharmaceutically acceptable salt, ester or prodrug thereof: wherein: X 1  is -A 1 -A 2 -A 3 -A 4 - X 2  is C or N, X 3  is C or N R 1  is H, halo, optionally substituted alkyl, optionally substituted alkenyl, alkynyl, haloalkyl, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted carbocycle, optionally substituted heterocycle, optionally substituted alkoxy, optionally substituted amine, cyano, or optionally substituted arylalkyl, R 2  is optionally substituted C 1 -C 8  alkyl, haloalkyl, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted carbocycle, optionally substituted heterocycle, halo, H, \u2014OH, optionally substituted alkoxy, optionally substituted amine, cyano, or optionally substituted arylalkyl, R 3  is an optionally substituted, saturated or unsaturated alkyl, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted carbocycle, or optionally substituted heterocycle, H, halo, alkoxy, haloalkyl, optionally substituted alkoxy, cyano, optionally substituted arylalkyl, R 4  is C 1 -C 6  alkyl, C 1 -C 6 , alkenyl, cycloalkyl, cycloalkenyl, heteroaryl, OR 5 , NR 5 R 6 , NR 5 C(\u2550O)R 6 , or or R 4  and R 1  together with the atoms to which they are connected form an aryl, heteroaryl, heterocycle or carbocycle ring of 5-8 atoms, wherein A 1 , A 2 , A 3 , and A 4  are independently carbon or null, wherein when two or more of A 1 , A 2 , A 3 , and A 4  are carbons, the bonds between the carbons are optionally double bonds, wherein each R 2  connected to each of A 1 , A 2 , A 3 , and A 4  is independent of one another, wherein R 5  and R 6  are independently null, H, \u2014OH, \u2550O, halo, haloalkyl, alkyl, alkynyl, alkenyl, aryl, arylalkyl, heteroaryl, carbocycle, heterocycle, cyano, alkoxy, amine, wherein R 5  and R 6  can be further substituted, wherein R 10  is C, N, O, or S.

Metadata:
- Claim Count in Document: 2.0
- Percentile: 86.0
- Lexical Diversity: 1.17647
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['10325087', '12588882', '12588883', '14775354', '13646143']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8319219812013711
- 35 USC 102 Novelty (BERT): 0.5405266334130229
- Combined Prediction Score: 0.8027824464225363
- Mean Citation Score: 365.953898
- Max Citation Score: 385.04922
- Similarity Product: 281.3766317888188

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test