PATENT CLAIM ANALYSIS

Application Number: 16264097
Application Type: Utility
Filing Date: 2019-01
Publication Date: 2019-05
Patent Classification: ["548", "469000"]

Abstract:
The present invention relates to indole compounds, and pharmaceutically acceptable compositions thereof, useful as antagonists of P2X7, and for the treatment of P2X7-related disorders.

Claim (Index 30):
A process for manufacturing a compound of  claim 19 , comprising the steps of:\n reacting a compound of formula A: wherein X is CH and Y is Cl; and wherein LG is group that is able to be displaced; with a compound of formula LG-R 1 ; wherein R 1  is as defined in  claim 19 ; to yield a compound of formula B: and reacting a compound of formula B with a compound of formula NH 2 \u2014R 2 ; wherein R 2  is as defined in  claim 19  to provide the compound.

Metadata:
- Claim Count in Document: 8.0
- Percentile: 99.0
- Lexical Diversity: 1.16667
- Patent Class: 548.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['15370645', '14969328', '14814659', '14730351', '15626138']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.738564558110403
- 35 USC 102 Novelty (BERT): 0.498567490468723
- Combined Prediction Score: 0.714564851346235
- Mean Citation Score: 266.416144
- Max Citation Score: 289.2787
- Similarity Product: 254.45142059848308

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test