PATENT CLAIM ANALYSIS

Application Number: 16055362
Application Type: Utility
Filing Date: 2018-08
Publication Date: 2019-01
Patent Classification: ["514", "259300"]

Abstract:
This invention relates to compounds of the general formula: in which the variable groups are as defined herein, and to their preparation and use.

Claim (Index 23):
A compound of the formula: wherein:\n Ring A is a 5- or 6-membered aryl or heteroaryl ring; \n Ring B is a 5- or 6-membered aryl or heteroaryl ring; \n L 1  is chosen from NR 1 C(O), C(O)NR 1 , NR 1 C(O)O, NR 1 C(O)NR 1 , and OC(O)NR 1 ; \n each occurrence of R a  and R b  is independently halo, \u2014CN, \u2014NO 2 , \u2014R 4 , \u2014OR 2 , \u2014NR 2 R 3 , \u2014C(O)YR 2 , \u2014OC(O)YR 2 , \u2014NR 2 C(O)YR 2 , \u2014SC(O)YR 2 , \u2014NR 2 C(\u2550S)YR 2 , \u2014OC(\u2550S)YR 2 , \u2014C(\u2550S)YR 2 , \u2014YC(\u2550NR 3 )YR 2 , \u2014YP(\u2550O)(YR 4 )(YR 4 ), \u2014Si(R 2 ) 3 , \u2014NR 2 SO 2 R 2 , \u2014S(O) r R 2 , \u2014SO 2 NR 2 R 3  or \u2014NR 2 SO 2 NR 2 R 3 , wherein each Y is independently a bond, \u2014O\u2014, \u2014S\u2014 or \u2014NR 3 \u2014; \n R e , at each occurrence, is independently halo, \u2014CN, \u2014NO 2 , \u2014R 4 , \u2014OR 2 , \u2014NR 2 R 3 , \u2014C(O)YR 2 , \u2014OC(O)YR 2 , \u2014NR 2 C(O)YR 2 , \u2014SC(O)YR 2 , \u2014NR 2 C(\u2550S)YR 2 , \u2014OC(\u2550S)YR 2 , \u2014C(\u2550S)YR 2 , \u2014YC(\u2550NR 3 )YR 2 , \u2014YP(\u2550O)(YR 4 )(YR 4 ), \u2014Si(R 2 ) 3 , \u2014NR 2 SO 2 R 2 , \u2014S(O) r R 2 , \u2014SO 2 NR 2 R 3  or \u2014NR 2 SO 2 NR 2 R 3 , wherein each Y is independently a bond, \u2014O\u2014, \u2014S\u2014 or \u2014NR 3 \u2014; \n R 1 , R 2  and R 3  are each independently H, alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, heterocyclyl, or heteroaryl; \n or R 2  and R 3 , taken together with the atom to which they are attached, form a 5- or 6-membered saturated, partially saturated or unsaturated ring, which contains 0-2 heteroatoms selected from N, O and S(O) r ; \n each occurrence of R 4  is independently alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, heterocyclyl, or heteroaryl; \n each of the alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl and heterocyclyl moieties is optionally substituted with one or more groups chosen from halo, \u2014CN, \u2014R 4 , \u2014OR 2 , \u2014S(O) r R 2 , \u2014SO 2 NR 2 R 3 , \u2014NR 2 R 3 , \u2014(CO)YR 2 , \u2014O(CO)YR 2 , \u2014NR 2 (CO)YR 2 , \u2014S(CO)YR 2 , \u2014NR 2 C(\u2550S)YR 2 , \u2014OC(\u2550S)YR 2 , \u2014C(\u2550S)YR 2 , \u2014YC(\u2550NR 3 )Y\u2032R 2 , \u2014COCOR 2 , \u2014COMCOR 2 , \u2014YP(\u2550O)(YR 4 )(YR 4 ), \u2014Si(R 2 ) 3 , \u2014NO 2 , \u2014NR 2 SO 2 R 2 , \u2014NR 2 SO 2 NR 2 R 3 , \u2550O, \u2550S, \u2550NH, \u2550NNR 2 R 3 , \u2550NNHC(O)R 2 , \u2550NNHCO 2 R 2 , and \u2550NNHSO 2 R 2 , wherein M is a 1-6 carbon alkyl group; \n each of the aryl and heteroaryl moieties is optionally substituted on an unsaturated carbon atom with one or more groups chosen from halo, \u2014CN, \u2014R 4 , \u2014OR 2 , \u2014S(O) r R 2 , \u2014SO 2 NR 2 R 3 , \u2014NR 2 R 3 , \u2014(CO)YR 2 , \u2014O(CO)YR 2 , \u2014NR 2 (CO)YR 2 , \u2014S(CO)YR 2 , \u2014NR 2 C(\u2550S)YR 2 , \u2014OC(\u2550S)YR 2 , \u2014C(\u2550S)YR 2 , \u2014YC(\u2550NR 3 )Y\u2032R 2 , \u2014COCOR 2 , \u2014COMCOR 2 , \u2014YP(\u2550O)(YR 4 )(YR 4 ), \u2014Si(R 2 ) 3 , \u2014NO 2 , \u2014NR 2 SO 2 R 2 , and \u2014NR 2 SO 2 NR 2 R 3 ; \n m is 0, 1, 2, 3 or 4; \n p is 0, 1, 2, 3, 4 or 5; \n r is 0, 1 or 2; and \n s is 0, 1, 2, 3 or 4, \n or a pharmaceutically acceptable salt thereof.

Metadata:
- Claim Count in Document: 56.0
- Percentile: 96.0
- Lexical Diversity: 1.125
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['14296016', '13801619', '13614838', '12227002', '13801116']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7747536576848669
- 35 USC 102 Novelty (BERT): 0.5370379171237779
- Combined Prediction Score: 0.7509820836287581
- Mean Citation Score: 333.1144020000001
- Max Citation Score: 358.56778
- Similarity Product: 330.9204378179192

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test