PATENT CLAIM ANALYSIS

Application Number: 16060771
Application Type: Utility
Filing Date: 2018-06
Publication Date: 2018-12
Patent Classification: ["564", "139000"]

Abstract:
Provided is a method of producing an aromatic amide derivative represented by Formula (I), which method includes a process a containing reacting an aniline derivative represented by Formula (II) with a carboxylic acid derivative represented by Formula (III) in the presence of a base to obtain an imide compound represented by Formula (IV) and a process b containing hydrolyzing the imide compound represented by Formula (IV) to obtain the aromatic amide derivative represented by Formula (I): wherein R 1  represents a C 1 -C 4  haloalkyl group, etc.; each of R 2  and R 3  independently represents a hydrogen atom, a halogen atom, etc.; R 4  represents a hydrogen atom, a C 1 -C 4  alkyl group, etc.; each of X 1  and X 2  independently represents a halogen atom, a C 1 -C 4  haloalkyl group, etc.; and Q represents a C 1 -C 4  alkyl group, a phenyl group, a pyridyl group, etc.

Claim (Index 7):
The method of producing an aromatic amide derivative according to  claim 1 , wherein the method further comprises the following process c, process d, and process e, wherein:\n the process c comprises obtaining a carboxylic acid compound represented by the following Formula (V) produced together with the aromatic amide derivative represented by Formula (I) in the process b, and halogenating or esterifying the carboxylic acid compound, to thereby obtain a carboxylic acid derivative reproducing compound represented by the following Formula (IIIa): in Formula (V), R 2  represents a hydrogen atom, a halogen atom, a C 1 -C 4  alkoxy group, a C 1 -C 4  alkylamino group, a di-C 1 -C 4  alkylamino group, a cyano group, or a nitro group;\n R 3  represents a hydrogen atom or a halogen atom; \n R 4  represents a hydrogen atom, a C 1 -C 4  alkyl group, or a C 1 -C 4  haloalkyl group; and \n Q represents: \n a di-C 1 -C 4  alkylaminocarbonyl group; \n a phenyl group; \n a heterocyclic group; \n a phenyl group substituted by 1 to 5 substituents, which may be the same or different, selected from the group consisting of a halogen atom, a cyano group, a nitro group, and a C 1 -C 4  haloalkyl group; or \n a heterocyclic group substituted by 1 to 4 substituents, which may be the same or different, selected from the group consisting of a halogen atom, a cyano group, a nitro group, and a C 1 -C 4  haloalkyl group; \n wherein the heterocyclic group is a pyridyl group, a pyridyl-N-oxide group, a pyrimidyl group, a pyridazyl group, a pyrazyl group, a furyl group, a thienyl group, an oxazolyl group, an isoxazolyl group, an oxadiazolyl group, a thiazolyl group, an isothiazolyl group, an imidazolyl group, a triazolyl group, a pyrrolyl group, a pyrazolyl group, or a tetrazolyl group; \n in Formula (IIIa), R 2 , R 3 , R 4 , X 3  and Q are the same as R 2 , R 3 , R 4 , X 3  and Q in Formula (III);\n the process d comprises allowing the carboxylic acid derivative reproducing compound obtained in the process c and the aniline derivative represented by Formula (II) to react with each other in the presence of a base to obtain the imide compound represented by Formula (IV); and \n the process e comprises hydrolyzing the imide compound represented by Formula (IV) obtained in the process d to obtain the aromatic amide derivative represented by Formula (I).

Metadata:
- Claim Count in Document: 15.0
- Percentile: 94.0
- Lexical Diversity: 2.89231
- Patent Class: 564.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['13016604', '13845664', '14433787', '10587990', '14366715']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.807070997724643
- 35 USC 102 Novelty (BERT): 0.5521912612012366
- Combined Prediction Score: 0.7815830240723024
- Mean Citation Score: 368.154356
- Max Citation Score: 374.60898
- Similarity Product: 276.5478961594605

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test