PATENT CLAIM ANALYSIS

Application Number: 15762878
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2018-09
Patent Classification: ["514", "210180"]

Abstract:
The present invention relates to a compound with formula (I) or a salt and/or a pharmaceutically acceptable solvate thereof, the method for preparing same as well as the uses thereof, in particular the therapeutic use thereof, mainly in the treatment of diseases associated with a hyperactivity of the endocannabinoid system.

Claim (Index 6):
A process for preparing a compound of formula (I) as defined according to  claim 1 , comprising the following steps:\n (i) condensation of 4-methylthiobenzaldehyde with 4-methylthioaniline to obtain the composition of following formula (IV): (ii) Staudinger cycloaddition between the composition of formula (IV) obtained and a ketene of following formula (V): to obtain the composition of following formula (IA): (iii) optionally, deprotection of the phthaloylated amine function of the compound of formula (IA), preferably by action of methylhydrazine to obtain the composition of following formula (IF): then, optionally, coupling of the compound of formula (IF) thus obtained with a compound of formula R 1 \u2014X and/or R 2 \u2014X\u2032, wherein R 1 \u2014X and R 2 \u2014X\u2032 are activated forms, such as acyl chlorides, sulphonyl chlorides and aryl isocyanates, of groups R 1  and R 2  as defined in  claim 1 ; and\n (iv) collection of the compound obtained in step (ii) or in step (iii).

Metadata:
- Claim Count in Document: 41.0
- Percentile: 90.0
- Lexical Diversity: 1.36585
- Patent Class: 514.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['14370951', '14555290', '15771077', '14679846', '15263033']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7271342857095741
- 35 USC 102 Novelty (BERT): 0.5189397279962443
- Combined Prediction Score: 0.7063148299382411
- Mean Citation Score: 269.005014
- Max Citation Score: 274.28796
- Similarity Product: 178.1921970696902

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test