PATENT CLAIM ANALYSIS

Application Number: 16109456
Application Type: Utility
Filing Date: 2018-08
Publication Date: 2018-12
Patent Classification: ["546", "074000"]

Abstract:
Provided are compounds, including those of Formula I; and pharmaceutically acceptable salts and solvates thereof. The compounds described herein relate to and/or have application(s) in (among others) the fields of drug discovery, pharmacotherapy, physiology, organic chemistry and polymer chemistry.

Claim (Index 1):
A compound selected from the formula: wherein:\n R 1  is selected from hydrogen, optionally substituted alkyl, optionally substituted aryl, and X-POLY; \n R 2  is selected from optionally substituted alkyl and \u2014X-POLY; \n R 3  is selected from hydroxyl, optionally substituted alkyl, optionally substituted amino, optionally substituted heterocyclyl, and \u2014X-POLY; or \n R 1  and R 3  are taken together with their intervening atoms to form a fused, optionally substituted heteroaryl or optionally substituted heterocyclyl; or \n R 3  and R 5  are taken together with their intervening atoms to form a fused, optionally substituted heteroaryl; \n  is optionally a single bond or a double bond; \n G is \u2014O\u2014R 4  or NH\u2014R 4  when   represents a single bond or G is \u2550O or \u2550N\u2014R 4  when   represents a double bond; \n X is a spacer moiety (e.g. a covalent bond, \u2014C(O)\u2014, \u2014NHC(O)\u2014, \u2014NH\u2014, \u2014CH 2 CHOHCH 2 NH\u2014, and \u2014O\u2014); \n POLY is a water soluble, non-peptidic oligomer; \n R 4  is -L-POLY or \u2014X-POLY, wherein L is an optional amino acid residue; \n R 5  is selected from hydrogen and X-POLY; and \n provided one of R 1 , R 2 , R 3 , R 4 , and R 5  comprises a POLY group; \n and pharmaceutically acceptable salts and solvates thereof.

Metadata:
- Claim Count in Document: 2.0
- Percentile: 96.0
- Lexical Diversity: 1.275
- Patent Class: 546.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15603942', '15511360', '15039686', '14075176', '15308987']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.839245512177407
- 35 USC 102 Novelty (BERT): 0.6264234466480851
- Combined Prediction Score: 0.8179633056244748
- Mean Citation Score: 476.83773600000006
- Max Citation Score: 680.4591
- Similarity Product: 518.354106019789

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test