PATENT CLAIM ANALYSIS

Application Number: 15744510
Application Type: Utility
Filing Date: 2018-01
Publication Date: 2018-07
Patent Classification: ["514", "222800"]

Abstract:
The invention provides a compound which is a diazine of formula (I) or a tautomer thereof, or a pharmaceutically acceptable salt thereof, for use as an antifungal agent: (I) wherein X, N′, C′, A and E are as defined herein. The invention also provides a compound of Formula (I) as defined herein.

Claim (Index 13):
A compound which is a diazine of formula (I) or a tautomer thereof, or a pharmaceutically acceptable salt thereof wherein the moiety represents -N(D)-C(A)=C(E)- or -N=C(A)-C(R 1 )(E)- as defined in  claim 1 , and wherein X, D, E, R 1 , R 2 , L, T and V are as defined in any one of  claims 2  to  10 , wherein A is -L-T, wherein\n i) L is a linear alkylene or alkenylene moiety comprising from 5 to 12 carbon atoms; wherein L is unsubstituted or is substituted with 1, 2 or 3 groups selected from halogen, C 1 -C 4  alkoxy and \u2014OH; and wherein L may optionally terminate in and/or be interrupted by a heteromoiety selected from \u2014O\u2014, \u2014S\u2014, \u2014C(O)\u2014, \u2014OC(O)\u2014, \u2014C(O)O\u2014, \u2014NR 2 \u2014, \u2014NR 2 C(O)\u2014, and \u2014C(O)NR 2 \u2014; \n and/or \n ii) T is aryl, heteroaryl, cycloalkyl or heterocyclyl; wherein T is unsubstituted or is substituted by 1, 2 or 3 groups V; \n wherein the compound is not: 2-(2-(2-amino-2H-1,3,4-thiadiazin-5-yl)ethyl)isoindoline-1,3-dione; 2-(1-(2-amino-2H-1,3,4-thiadiazin-5-yl)ethyl)isoindoline-1,3-dione; 5-benzyl-6H-1,3,4-thiadiazin-2-amine; 2-amino-5-benzyl-1,3,4-thiadiazine; 5-(3-nitrobenzyl)-6H-1,3,4-thiadiazin-2-amine; 5-(3-methylpentan-3-yl)-6H-1,3,4-thiadiazin-2-amine; or 5-[2-(5-nitro-2-furanyl)ethenyl]-6H-1,3,4-thiadiazin-2-amine.

Metadata:
- Claim Count in Document: 5.0
- Percentile: 86.0
- Lexical Diversity: 1.65
- Patent Class: 514.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['12989410', '14625532', '12601284', '11914516', '12515354']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7176924863382423
- 35 USC 102 Novelty (BERT): 0.5191793146393273
- Combined Prediction Score: 0.6978411691683509
- Mean Citation Score: 288.72395399999994
- Max Citation Score: 300.37643
- Similarity Product: 203.83043630729736

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test