PATENT CLAIM ANALYSIS

Application Number: 15917866
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2018-09
Patent Classification: ["514", "210170"]

Abstract:
The present invention provides a genus of polycyclic amines that are useful as opioid receptor modulators. The compounds of the invention are useful in both therapeutic and diagnostic methods, including for treating pain, neurological disorders, cardiac disorders, bowel disorders, drug and alcohol addiction, drug overdose, urinary disorders, respiratory disorders, sexual dysfunction, psoriasis, graft rejection or cancer.

Claim (Index 1):
A compound having a structure according to Formula I: wherein: A is substituted or unsubstituted: alkyl, heteroalkyl, cycloalkyl, heterocycloalkyl, aryl, heteroaryl, and arylalkyl; Y is substituted or unsubstituted: alkyl, heteroalkyl, cycloalkyl, and heterocycloalkyl; Q is substituted or unsubstituted: aryl, heteroaryl, and null; W is substituted or unsubstituted, saturated or unsaturated: (i) 4- to 8-membered heterocyclic rings including an N-substituent; or (ii) 4- to 10-membered bicyclic or heterobicyclic rings, wherein at least one or the rings includes an N-substituent; G is substituted or unsubstituted alkyl or an N atom; Z includes substituted or unsubstituted aryl, substituted or unsubstituted heteroaryl, and null; If Z is null then T is null, but if Z is not null, T is selected from: (i) the moieties H, OH, NH 2 , NO 2 , \u2014SO 2 NH 2 , halogen, and (ii) substituted or unsubstituted: alkyl, heteroalkyl, cycloalkyl, heterocycloalkyl, aryl, and heteroaryl; n is an integer from 1-4 when G is alkyl and is 1 when G is an N atom; R 1  and R 3  are members independently selected from H and substituted or unsubstituted: alkyl, heteroalkyl, 3- to 7-membered cycloalkyl, 3- to 7-membered heterocycloalkyl, aryl, and heteroaryl; m is an integer from 0-8 and can be same or different for each of R 2 , R 4 , R 5  and R 6 , and wherein R 2 , R 4 , R 5  and R 6  are each independently selected from H and substituted or unsubstituted: alkyl, heteroalkyl, 3- to 7-membered cycloalkyl, 3- to 7-membered heterocycloalkyl, and where m is greater than 1 for any of R 2 , R 4 , R 5  and R 6 , each member in said multi-member R 2 , R 4 , R 5  and R 6  chain can be the same or different; and further provided that the total number of R 2 , R 4 , R 5  and R 6  for which m is greater than 0 is always less than or equal to the number of W ring positions available for covalent bonding; and R 1  and R 3 , or R 1  or R 3  and Z, or R 2  and A, or R 2  and Y together with groups to which they may be joined, optionally form a substituted or unsubstituted 3- to 7-membered ring.

Metadata:
- Claim Count in Document: 5.0
- Percentile: 90.0
- Lexical Diversity: 1.46809
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['11464057', '11105938', '12312749', '12814964', '11643190']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7990597918102462
- 35 USC 102 Novelty (BERT): 0.5266156325317674
- Combined Prediction Score: 0.7718153758823983
- Mean Citation Score: 336.9528200000001
- Max Citation Score: 345.2538
- Similarity Product: 259.38649686870576

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test