PATENT CLAIM ANALYSIS

Application Number: 15906268
Application Type: Utility
Filing Date: 2018-02
Publication Date: 2018-07
Patent Classification: ["514", "233200"]

Abstract:
The present invention is directed to novel compounds of formula I and their use as therapeutic compounds.

Claim (Index 21):
The pharmaceutical composition according to  claim 20  comprising a compound selected from formulae Ie-1, Ie-2 and Ie-3 or a pharmaceutically acceptable salt or solvate thereof and at least one pharmaceutically acceptable carrier, diluent, excipient and/or adjuvant, wherein a depicts the bond linking R 1  to the piperazine moiety; and Ar 2 , R 1 , X 1  and X 2  are as defined in claim  2 ; and R 5  and R 6  are independently selected from H, halo, cyano, alkyl, cyclopropyl, aryl, heteroaryl, each of said aryl and heteroaryl groups being optionally substituted by one or more group(s) selected from halo, alkyl, cyclopropyl, or R 5  and R 6  together form a phenyl moiety fused to the phenyl ring they are attached to; and R 8 , R 8\u2032 , R 9 , R 9\u2032  and R 10  are independently selected from H, halo, haloalkyl, cyclopropyl or haloalkoxy, or R 8 , R 8\u2032 , R 9 , R 9\u2032  are H and R 10  is phenoxy; M 1  and M 2  are as defined in claim  4 ; and wherein, in formula Ie-1 when: R 1  is H, and R 5  and R 6  are independently selected from H, halo, cyano, C1-C3 alkyl, and Ar 2  is a 5- to 6-membered aryl or heteroaryl group optionally substituted by one or more group(s) selected from halo, C1-C3alkyl, hydroxyl, alkoxy, or fused to an aryl group optionally substituted by one or more further halo, C1-C3 alkyl, hydroxyl, methoxy then, R 6  is H and R 5  is H, halo, or R 5  is H and R 6  is halo, cyano, C1-C3 alkyl, C1 haloalkyl, or R 5  and R 6  are independently halo, and Ar 2  is, quinolin-2-yl, isoquinolin-3-yl, 8-haloquinolin-2-yl, benzothiazol-2-yl, 4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl.

Metadata:
- Claim Count in Document: 32.0
- Percentile: 88.0
- Lexical Diversity: 1.05882
- Patent Class: 514.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['14349595', '14799208', '13627091', '15259922', '15205304']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8138521764291394
- 35 USC 102 Novelty (BERT): 0.6253844343535592
- Combined Prediction Score: 0.7950054022215813
- Mean Citation Score: 548.391766
- Max Citation Score: 607.86743
- Similarity Product: 513.2024180211723

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test