PATENT CLAIM ANALYSIS

Application Number: 16104840
Application Type: Utility
Filing Date: 2018-08
Publication Date: 2019-04
Patent Classification: ["544", "105000"]

Abstract:
The present invention relates to compounds including but not limited to of any one of formulas Ia, Ib, IIa, IIb, IIIa, IIIb, and IV to VI, VIIa, VIIb, VIIIa, VIIIb and VIIIc as described herein and their tautomers and/or pharmaceutically acceptable salts, compositions, and methods of uses thereof.

Claim (Index 24):
A compound having a structure of: wherein B 1  is CR 2 ; one of B 2 , B 3 , and B 4  is N, and the remaining are independently CR 2 ; L is selected from the group consisting of a covalent bond, CR 6 2 , C(O)\u2014(CR 6 2 ) m , C(S)\u2014(CR 6 2 ) m , O\u2014(CR 6 2 ) m , S\u2014(CR 6 2 ) m , SO\u2014(CR 6 2 ) m , SO 2 \u2014(CR 6 2 ) m , and NR 6 \u2014(CR 6 2 ) m ; X 1  is O, S, or CH 2 ; the variable p is 0, 1, 2, 3, 4, 5, 6, or 7; the variable k is 1, 2, 3, 4, 5, 6, or 7; R 2  is independently hydrogen, halogen, C 1  to C 6  alkyl, C 1  to C 6  haloalkyl, C 1  to C 6  alkoxy, C 1  to C 6  haloalkoxy, cyano, or nitro; R 3  is independently hydrogen or C 1  to C 6  alkyl; or two R 3  together with the carbon attached thereto form C\u2550O; R 4  is independently C 1  to C 6  alkyl; or two R 4  together with the carbon attached thereto form C\u2550O; R 5  is hydrogen, C 1  to C 6  alkyl, substituted C 1  to C 6  alkyl, cycloalkyl, or acyl; each R 6  independently is selected from the group consisting of hydrogen, halogen, alkyl, substituted alkyl, cycloalkyl, substituted cycloalkyl, alkenyl, substituted alkenyl, alkoxy, substituted alkoxy, alkynyl, substituted alkynyl, amino, substituted amino, aminosulfinyl substituted aminosulfinyl, aminosulfonyl, substituted aminosulfonyl, sulfinyl, sulfonyl, sulfonyloxy, substituted sulfonyloxy, aminosulfonyloxy, aminosulfinyloxy, aminosulfonylamino, acylamino, aminocarbonyloxy, aminocarbonylamino, aminothiocarbonylamino, amidino, substituted amidino, aminocarbonylamino, aminothiocarbonylamino, acyloxy, aryl, substituted aryl, heteroaryl, substituted heteroaryl, cyano, nitro, carboxyl, carboxyl ester, (carboxyl ester)amino, (carboxyl ester)oxy, hydroxyl, acyl, formyl, aminocarbonyl, substituted aminocarbonyl, and substituted aminothiocarbonyl, or two R 6  join together to form a ring selected from the group consisting of C 3 -C 7  cycloalkyl, C 3 -C 7  heterocycloalkyl, and substituted C 3 -C 7  heterocycloalkyl; and R 7  is independently hydrogen or C 1  to C 6  alkyl; or a tautomer, or a pharmaceutically acceptable salt thereof.

Metadata:
- Claim Count in Document: 38.0
- Percentile: 96.0
- Lexical Diversity: 1.4186
- Patent Class: 544.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['15110082', '12669536', '12295967', '12449701', '12449286']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8298474097057469
- 35 USC 102 Novelty (BERT): 0.6274536572055943
- Combined Prediction Score: 0.8096080344557317
- Mean Citation Score: 465.972764
- Max Citation Score: 622.84564
- Similarity Product: 525.5902712475944

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test