PATENT CLAIM ANALYSIS

Application Number: 15759084
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2019-02
Patent Classification: ["514", "210000"]

Abstract:
The present application relates to novel azetidinimine of formula (I). Wherein R 1 -R 6  are as defined in claim  1 . The azetidinimine of the invention are useful as antibiotics and as inhibitors of a carbapenemases. The present invention thus further relates to their use in antibiotic therapies and their methods of synthesis.

Claim (Index 3):
Compound according to  claim 1  or  2 , characterized in that R 1  represents a monocyclic aryl fragment optionally substituted by\n one or several (notably 1 to 3) OH, C 1 -C 6  alkyl, C 1 -C 6  thioalkyl, halogen, amino-(C 1 -C 10  alkoxy), (carboxylic acid)-(C 1 -C 10  alkoxy), (carboxylic (C 1 -C 6 )alkyl ester)-C 1 -C 10  alkoxy, (1,2 diol)-C 2 -C 10  alkoxy, \u2014O\u2014(C 1 -C 6 )alkyl-O\u2014(C 1 -C 6 )alkyl-OH, (C 5 -C 12 )-aryl-(C 1 -C 6 )-alkyl ester, nitro and/or a C 1 -C 6  alkoxy group optionally substituted by a mono or polycyclic C 5 -C 12  aryl group, and/or \n a bridging group of formula \u2014O\u2014CH 2 \u2014O\u2014 or \u2014O\u2014CH 2 CH 2 \u2014O\u2014, \n preferably R 1  represents a monocyclic aryl fragment optionally substituted by one or several C 1 -C 6  alkoxy, C 1 -C 6  thioalkyl, halogen, amino-(C 1 -C 10  alkoxy), (carboxylic acid)-(C 1 -C 10  alkoxy), (1,2 diol)-(C 2 -C 10  alkoxy), (C 5 -C 12 )-aryl-(C 1 -C 6 )-alkyl ester and/or nitro fragments.

Metadata:
- Claim Count in Document: 28.0
- Percentile: 90.0
- Lexical Diversity: 1.51282
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15029377', '14785034', '14382232', '13356729', '13538399']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8193369020423895
- 35 USC 102 Novelty (BERT): 0.5341240144604641
- Combined Prediction Score: 0.790815613284197
- Mean Citation Score: 357.41369799999984
- Max Citation Score: 368.19736
- Similarity Product: 285.3378242394972

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test