PATENT CLAIM ANALYSIS

Application Number: 15748514
Application Type: Utility
Filing Date: 2018-01
Publication Date: 2018-08
Patent Classification: ["514", "506000"]

Abstract:
A method for the synthesis of a aryl compound of Formula (1). Formula (1) UT-W—R 1 ) n    (1)

Claim (Index 1):
A method for the synthesis of a compound of Formula (1);\n U\ue8a0T-W\u2014R 1 ) n \u2003\u2003 Formula (1) \n the method comprising the step of: reacting a compound of Formula (2);\n U\ue8a0X) n \u2003\u2003 Formula (2) \n \n with a compound of Formula (3);\n V\u2014Y\u2003\u2003 Formula (3) \n \n under a first set of reaction conditions, to produce a compound of Formula (4):\n U\ue8a0V) n \u2003\u2003 Formula (4) \n \n then reacting the compound of Formula (4) with one or more reagents under a second set of reaction conditions to produce the compound of Formula (1); where; n is 1-6; U is a benzene or pyridine; T is -, = or \u2261; V is = or \u2261; W is a benzene or pyridine; Y is \u2014B K- G I M J+ ; G is a halogen; M is any Group (I) or Group (II) metal; K is 1 or 2; I is 3 or 4; J is 1 or 2; X is a halogen; each R 1  may be independently selected from any one or more of i-xxxiii: i. H; ii. C 1-8  alkyl; iii. C 1-8  heteroalkyl; iv. carboxylic acids and related derivatives independently selected from: a) carboxylic acid, b) alkyl carboxylic acid, \u2003where n=1-8; c) thiocarboxylic acid, d) alkyl thiocarboxylic acid, \u2003where n=1-8; e) esters, f) alkyl esters, \u2003where n=1-8; g) thioesters, h) alkyl thioesters, \u2003where n=1-8 i) dithioesters, j) alkyl dithioesters, \u2003where n=1-8 v. amide derivatives of carboxylic acids independently selected from: k) amides, l) thioamides, vi. aldehydes, ketones and their derivatives independently selected from: m) aldehyde, n) thial, o) ketones, p) thioketones, q) acetals, \u2003where n=1-3 r) dithioacetals, \u2003where n=1-3 vii. amines, alkyl amines and their derivatives independently selected from: s) amines, t) amides, u) thioamides, v) ammonium salts, w) alkyl amines, \u2003where n=1-8 x) alkyl amides, \u2003where n=1-8 y) alkyl thioamides, \u2003where n=1-8 z) alkyl ammonium salts, \u2003where n=1-8, aa) imines, bb) guanidines, cc) amidines, viii. nitrile (cyano), \u2014C\u2261N, ix. isonitrile, \u2014N + \u2261C \u2212 , X. cyanate, \u2014O\u2014C\u2261N, xi. isocyanate, \u2014N\u2550C\u2550O, xii. thiocyanate, \u2014S\u2014C\u2261N, xiii. isothiocyanate, \u2014N\u2550C\u2550S, xiv. azo, \u2014N\u2550NH, xv. nitro, xvi. nitrite, \u2014O\u2014N\u2550O, xvii. nitriso, \u2014N\u2550O, xviii. N-terminal peptide sequences, \u2003where q=1-3 and R pep  is any group resulting in the formation of an amino acid, xix. C-terminal peptide sequences, \u2003where q=1-3 and R pep  is any group resulting in the formation of an amino acid, xx. phosphorus based substituents, where the phosphorus atom is in either the 3 +  or 5 +  oxidation state, independently selected from: dd) alkyl phosphines, \u2003where n=1-8 ee) alkyl phosphonium salts, \u2003where n=0-8 ff) phosphines, gg) phosphine oxides, hh) phosphites, ii) phosphates, jj) phosphinites, kk) phosphinates, ll) phosphinites, mm) phosphonates, xxi. sulfur based substituents, nn) sulfate, oo) sulfone, pp) sulfoxide, qq) sulfinic acids, rr) sulfimines, ss) sulfon amides, tt) triflates, xxii. boron based substituents, uu) boronic acid, vv) boronic esters, xxiii. semicarbazones, xxiv. thiosemicarbazones, xxv. cyanimide, xxvi. hydrazone, xxvii. oxime, xxviii. nitroamine, xxix. nitronate, xxx. nitrone, xxxi. carbonates, xxxii. carbamates, xxxiii. dithiocarbamates, where R a , R b , R c  and R d  in i-xxxiii are independently selected from hydrogen or alkyl (C 1-4 ).

Metadata:
- Claim Count in Document: 47.0
- Percentile: 86.0
- Lexical Diversity: 1.625
- Patent Class: 514.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['12446343', '12407857', '14518480', '14609612', '10623196']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7025547790595608
- 35 USC 102 Novelty (BERT): 0.5016774886396692
- Combined Prediction Score: 0.6824670500175716
- Mean Citation Score: 196.937276
- Max Citation Score: 201.06427
- Similarity Product: 132.44260245313706

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test