PATENT CLAIM ANALYSIS

Application Number: 15911546
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2019-02
Patent Classification: ["544", "329000"]

Abstract:
The present invention provides compounds and compositions thereof which are useful as inhibitors of Bruton's tyrosine kinase and which exhibit desirable characteristics for the same.

Claim (Index 28):
A pharmaceutical composition comprising a compound of Formula I, or pharmaceutically acceptable salt thereof; and one or more pharmaceutically acceptable excipients;\n wherein the compound is of Formula I: wherein:\n each R 1  is independently hydrogen, an optionally substituted C 1-6  aliphatic group, an optionally substituted 3-7 membered monocyclic heterocyclic group, or an optionally substituted heterocyclylalkyl group having 3-7 carbon atoms and 1-3 heteroatoms independently selected from nitrogen, oxygen, or sulfur;\n or two R 1  groups are taken together with their intervening atoms to form an optionally substituted 3-7 membered saturated or partially unsaturated monocyclic heterocyclic ring having 1-2 heteroatoms independently selected from nitrogen, oxygen, or sulfur; \n \n wherein optionally substituted groups may be substituted with halogen, \u2014NO 2 , \u2014CN, \u2014OR, \u2014SR, \u2014N(R) 2 , \u2014C(O)R, \u2014CO 2 R, \u2014N(R)C(O)OR, \u2014C(O)N(R) 2 , \u2014OC(O)R, \u2014N(R)C(O)R, \u2014S(O)R, \u2014S(O) 2 R, or \u2014S(O) 2 N(R) 2 ; \n each R is independently hydrogen or C 1-6  aliphatic;\n or two R groups attached to the same nitrogen are taken together with their intervening atoms to form an optionally substituted 3-7 membered saturated or partially unsaturated monocyclic heterocyclic ring having 1-2 heteroatoms, in which any second heteroatom is independently selected from nitrogen, oxygen, or sulfur; \n \n Ring A is \n R 2  is \u2014Cl or \u2014F; and R 3  is \u2014CF 3 , \u2014OCF 3 , or \u2014F.

Metadata:
- Claim Count in Document: 54.0
- Percentile: 90.0
- Lexical Diversity: 1.08
- Patent Class: 544.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['14406315', '14316710', '15698171', '13393192', '15006061']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7548293438949453
- 35 USC 102 Novelty (BERT): 0.5393932057033957
- Combined Prediction Score: 0.7332857300757903
- Mean Citation Score: 346.835098
- Max Citation Score: 378.47186
- Similarity Product: 355.32056268331775

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 0

Dataset: test