PATENT CLAIM ANALYSIS

Application Number: 16077561
Application Type: Utility
Filing Date: 2018-08
Publication Date: 2019-01
Patent Classification: ["548", "374100"]

Abstract:
The present invention concerns a process for the manufacture of carboxamides, in particular agrochemical or pharmaceutically active ingredients, from pyrazole ketone compounds.

Claim (Index 1):
A process for the manufacture of carboxamides, the process comprising the step of reacting a pyrazole compound of the formula (I) with a compound of the formula (II) NR 3 H(A*)Q to obtain a compound of the formula (III) wherein R 1  is selected from the group consisting of H, R\u2032, X\u2032, CN, COOR\u2032, OR\u2032, SR\u2032 and C(O)NR\u2032 2 , wherein R\u2032 is selected independently from the group consisting of hydrogen, CN, C 1 -C 12 -alkyl, C 1 -C 12 -alkyl, C 2 -C 6  alkenyl, aryl, cycloalkyl, aralkyl and heteroaryl, each of which is optionally substituted, and X\u2032 is selected from the group consisting of F, Cl, Br and I;\n wherein R 2  is selected from the group consisting of optionally substituted C 1 -C 12 -alkyl, C 2 -C 6  alkenyl, cycloalkyl, aryl, heteroaryl, and aralkyl; wherein R 3  is selected from the group consisting of H, optionally substituted C 1 -C 12 -alkyl, C 2 -C 6  alkenyl [[or]] and C 3 -C 8 -cycloalkyl group; \n wherein R 4  is selected from the group consisting of H, X\u2032, COOR\u2032, OR\u2032, SR\u2032, and C(O)NR\u2032 2 , wherein R\u2032 and X\u2032 are as defined above; \n wherein R 5  is selected from the group consisting of C 1 -C 12 -alkyl, C 2 -C 6  alkenyl, cycloalkyl, aryl, heteroaryl, and aralkyl, each of which is optionally substituted; \n wherein A* is absent or an optionally substituted C 1 -C 4 -alkylene group; \n wherein Q is an optionally substituted aryl or heteroaryl group.

Metadata:
- Claim Count in Document: 12.0
- Percentile: 96.0
- Lexical Diversity: 1.04167
- Patent Class: 548.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15199528', '11033079', '12087185', '11830733', '13881366']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.6920662763717613
- 35 USC 102 Novelty (BERT): 0.4984428732067328
- Combined Prediction Score: 0.6727039360552585
- Mean Citation Score: 222.989906
- Max Citation Score: 224.82187
- Similarity Product: 159.81532319750306

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test