PATENT CLAIM ANALYSIS

Application Number: 15946601
Application Type: Utility
Filing Date: 2018-04
Publication Date: 2018-08
Patent Classification: ["548", "240000"]

Abstract:
Disclosed is a method for preparing a compound of Formula 1 wherein Q and Z are as defined in the disclosure comprising distilling water from a mixture comprising a compound of Formula 2, a compound of Formula 3, a base comprising at least one compound selected from the group consisting of alkaline earth metal hydroxides of Formula 4 wherein M is Ca, Sr or Ba, alkali metal carbonates of Formula 4a wherein M 1  is Li, Na or K, 1,5-diazabicyclo[4.3.0]non-5-ene and 1,8-diazabicyclo[5.4.0]undec-7-ene, and an aprotic solvent capable of forming a low-boiling azeotrope with water. Also disclosed is a method for preparing a compound of Formula 2 comprising (1) forming a reaction mixture comprising a Grignard reagent derived from contacting a compound of Formula 5 wherein X is Cl, Br or I with magnesium metal or an alkylmagnesium halide in the presence of an ethereal solvent, and then (2) contacting the reaction mixture with a compound of Formula 6 wherein Y is OR 11  or NR 12 R 13 , and R 11 , R 12  and R 13  are as defined in the disclosure. Further disclosed is a method for preparing a compound of Formula 7 wherein Q and Z are as defined in the disclosure, using a compound of Formula 1 characterized by preparing the compound of Formula 1 by the method disclosed above or using a compound of Formula 1 prepared by the method disclosed above.

Claim (Index 13):
The method of  claim 12  wherein Z is R 2a  is F, Cl, Br, C 1 -C 2  fluoroalkyl or C 1 -C 2  fluoroalkoxy; R 2b  is H, F, Cl or Br; and R 2c  is H, F, Cl, Br or CF 3 .

Metadata:
- Claim Count in Document: 21.0
- Percentile: 91.0
- Lexical Diversity: 2.5534
- Patent Class: 548.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['12933493', '15159322', '14683423', '12679382', '13544113']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8729053319932301
- 35 USC 102 Novelty (BERT): 0.559707417412993
- Combined Prediction Score: 0.8415855405352064
- Mean Citation Score: 422.608154
- Max Citation Score: 456.38446
- Similarity Product: 353.83053125520706

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test