PATENT CLAIM ANALYSIS

Application Number: 15753157
Application Type: Utility
Filing Date: 2018-02
Publication Date: 2018-08
Patent Classification: ["514", "210170"]

Abstract:
Disclosed are functionalized aminobenzoboroxoles compounds, method for preparing these compounds, and methods for treating cancers.

Claim (Index 1):
A compound having the structure of formula (I): or a pharmaceutically acceptable salt thereof, wherein R 1  is selected from hydrogen, C 1-6  alkyl, C 2-6  alkenyl, C 2-6  alkynyl, optionally substituted C 6-10  aryl, optionally substituted 5-10 membered heteroaryl, optionally substituted C 3-10  carbocyclyl, or optionally substituted 3-10 membered heterocyclyl; each of R 2 , R 3 , R 4  and R 5  is independently selected from hydrogen, halogen, hydroxy, optionally substituted C 1-6  alkyl, optionally substituted C 2-6  alkenyl, optionally substituted C 2-6  alkynyl, optionally substituted C 1-6  alkoxy, optionally substituted C 1-6  alkylthio, optionally substituted C 2-8  alkoxyalkyl, C 1-6  haloalkyl, C 1-6  hydroxyalkyl, \u2014CN, \u2014NO 2 , O-carboxy, C-carboxy, O-amido, C-amido, sulfinyl, sulfonyl, S-sulfonamido, N-sulfonamido, amino, optionally substituted aminoalkyl, optionally substituted C 6-10  aryl, optionally substituted C 7-14  aralkyl, optionally substituted 5-10 membered heteroaryl, optionally substituted C 3-10  carbocyclyl, or optionally substituted 3-10 membered heterocyclyl; R 6  is selected from hydrogen, optionally substituted C 1-6  alkyl, \u2014N(\u2550O), or \u2014C(\u2550O)NR 8 R 9 ; R 7  is selected from C 1-6  alkyl, \u2014(CH 2 ) m \u2014(C 6-10  aryl), \u2014(CH 2 ) m -(5-10 membered heteroaryl), \u2014(CH 2 ) m \u2014(C 3-10  carbocyclyl), and \u2014(CH 2 ) m -(3-10 membered heterocyclyl), each optionally substituted with one or more R 10 ; each R 8  and R 9  is independently selected from hydrogen, optionally substituted C 1-6  alkyl, C 1-6  haloalkyl, optionally substituted C 2-6  alkenyl, optionally substituted C 2-6  alkynyl, optionally substituted C 2-8  alkoxyalkyl, optionally substituted C 3-10  carbocyclyl, optionally substituted C 6-10  aryl, optionally substituted C 7-14  aralkyl, optionally substituted 5-10 membered heteroaryl, or optionally substituted 3-10 membered heterocyclyl; R 10  is selected from hydroxy, halogen, optionally substituted C 1-6  alkyl, optionally substituted C 2-6  alkenyl, optionally substituted C 2-6  alkynyl, optionally substituted C 1-6  alkoxy optionally substituted C 1-6  alkylthio, optionally substituted C 2-8  alkoxyalkyl, C 1-6  haloalkyl, C 1-6  hydroxyalkyl, optionally substituted C 3-10  carbocyclyl, optionally substituted C 6-10  aryl, optionally substituted C 7-14  aralkyl, optionally substituted 5-10 membered heteroaryl, or optionally substituted 3-10 membered heterocyclyl, \u2014CN, \u2014NO 2 , O-carboxy, C-carboxy, O-amido, C-amido, sulfinyl, sulfonyl, S-sulfonamido, N-sulfonamido, amino, or optionally substituted aminoalkyl; m is an integer selected from 1 to 6; and n is 0 or 1.

Metadata:
- Claim Count in Document: 47.0
- Percentile: 88.0
- Lexical Diversity: 1.2
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15636424', '15024504', '15518541', '15435003', '14358606']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7850694913011292
- 35 USC 102 Novelty (BERT): 0.5306384139176803
- Combined Prediction Score: 0.7596263835627843
- Mean Citation Score: 344.75435000000016
- Max Citation Score: 356.21725
- Similarity Product: 289.795871022284

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test