PATENT CLAIM ANALYSIS

Application Number: 16129867
Application Type: Utility
Filing Date: 2018-09
Publication Date: 2019-01
Patent Classification: ["514", "471000"]

Abstract:
The invention relates to 1-(3-sulfonylphenyl)-3-(cyclopent-2-en-1-yl)urea derivatives, and their use in treating or preventing diseases and conditions mediated by the CXCR2 receptor. In addition, the invention relates to compositions containing the derivatives and processes for their preparation.

Claim (Index 6):
The method according to  claim 1 , wherein R 4  is selected from the group consisting of:\n a) C 1-4 alkyl optionally substituted by one, two or three substituents independently selected from the group consisting of: fluoro, C 1-3 alkoxy and C 1-3 fluoroalkyl; d) a 5 or 6-membered, saturated heterocyclyl group directly attached to the sulfone via a ring carbon atom, which heterocyclyl group is optionally substituted by one, two or three substituents independently selected from the group consisting of C 1-3 alkyl optionally substituted by one or more deuterium, fluoro, C 1-3 fluoroalkyl, hydroxy, C 1-3 alkoxy and \u2014NR 4c R 4d , wherein R 4c  and R 4d  are independently C 1-3 alkyl; and which heterocyclyl group contains one or two ring-heteroatoms independently selected from nitrogen and oxygen; and e) a C 4-6 cycloalkyl group directly attached to the sulfone; which cycloalkyl group is optionally substituted by one or two substituents independently selected from the group consisting of fluoro, C 1-3 fluoroalkyl, hydroxy, C 1-3 alkoxy and \u2014(CH 2 ) t NR 4e R 4f ; wherein t is 0 or 1, and wherein R 4e  and R 4f  are independently C 1-3 alkyl, or R 4e  and R 4f , together with the nitrogen to which they are attached, form a 4, 5 or 6-membered saturated ring which ring is optionally substituted by one or more fluoro substituent.

Metadata:
- Claim Count in Document: 3.0
- Percentile: 97.0
- Lexical Diversity: 1.37143
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15314124', '15175363', '15502356', '15799771', '14354500']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.792836414504341
- 35 USC 102 Novelty (BERT): 0.6242476989415601
- Combined Prediction Score: 0.7759775429480629
- Mean Citation Score: 405.007728
- Max Citation Score: 570.4564
- Similarity Product: 522.4368097837448

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test