PATENT CLAIM ANALYSIS

Application Number: 15899842
Application Type: Utility
Filing Date: 2018-02
Publication Date: 2018-08
Patent Classification: ["544", "331000"]

Abstract:
The present disclosure relates to azetidine compounds. The azetidine compounds are GPR119 modulators and useful for the prevention and/or treatment of diabetes, obesity, dyslipidemia and related disorders. The present disclosure furthermore relates to the use of azetidine compounds as active ingredients in pharmaceuticals, and pharmaceutical compositions comprising them.

Claim (Index 5):
The compound of formula I according to  claim 1 , which is a compound of formula Ia wherein: R4 is (CH 2 ) p ; p is 1 or 2; R5 is CF 3  or cyclopropyl; R7 is OH, COOR13, CONR14R15, S(O) m R16 or COR22; m is 0, 1 or 2; R13 is H or (C 1 -C 2 )-alkyl; R14 and R15 are independently H, (C 3 -C 6 )-cycloalkyl, (C 1 -C 6 )-alkyl or (C 1 -C 6 )-alkyl substituted with 1 to 3 groups selected from the group consisting of CONH 2  and OH; R16 is (C 1 -C 6 )-alkyl; and R22 is azetidinyl, pyrrolidinyl, piperidinyl or piperazinyl;\n wherein the azetidinyl, pyrrolidinyl, piperidinyl or piperazinyl is optionally substituted with 1 to 3 groups selected from the group consisting of OH and COCH 3 , \n in any of its stereoisomeric forms, or a physiologically acceptable salt or solvate of any of the foregoing.

Metadata:
- Claim Count in Document: 128.0
- Percentile: 88.0
- Lexical Diversity: 1.5
- Patent Class: 544.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15284213', '15284334', '14048425', '15301603', '15039607']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7768217187995464
- 35 USC 102 Novelty (BERT): 0.50780499001267
- Combined Prediction Score: 0.7499200459208588
- Mean Citation Score: 240.448416
- Max Citation Score: 281.36795
- Similarity Product: 216.9870893255532

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test