PATENT CLAIM ANALYSIS

Application Number: 16091098
Application Type: Utility
Filing Date: 2018-10
Publication Date: 2019-08
Patent Classification: ["514", "340000"]

Abstract:
The present invention provides benzamidazole compounds and methods of using the compounds as galectin-1 inhibitors.

Claim (Index 18):
The compound of  claim 1 , wherein\n R 2a  and R 2b  are each independently selected from the group consisting of \u2014CH 2 CH 2 OH and \u2014CH 2 CH 2 OC(O)CH 3 , or are combined with the nitrogen to which they are attached to form a C 3-8  heterocycloalkyl having from 0 to 2 additional heteroatoms selected from the group consisting of N, O, and S, wherein the heterocycloalkyl is optionally substituted with 1 to 4 R 2c  groups; each R 2c  is independently C 1-6  alkyl; R 3  is selected from the group consisting of hydrogen, C 3-8  cycloalkyl, C 6-12  aryl, and C 5-12  heteroaryl, wherein the aryl and heteroaryl are optionally substituted with 1 to 4 R 3a  groups; each R 3a  is independently selected from the group consisting of halogen, C 1-6  haloalkyl, C 1-6  alkoxy, C 5-12  heteroaryl, and \u2014SO 2 \u2014C 6-12  aryl; X 1  is C 1-6  alkylene; and X 2  is absent or selected from the groups consisting of C 1-6  alkylene, and \u2014C(O)CH(NH 2 )CH 2 \u2014; or pharmaceutically acceptable salts and isomers thereof.

Metadata:
- Claim Count in Document: 24.0
- Percentile: 97.0
- Lexical Diversity: 1.06667
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['12774544', '13048832', '11995928', '14774387', '15634768']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.796952953956514
- 35 USC 102 Novelty (BERT): 0.524702269469786
- Combined Prediction Score: 0.7697278855078412
- Mean Citation Score: 310.190956
- Max Citation Score: 319.20123
- Similarity Product: 232.9642784154689

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test