PATENT CLAIM ANALYSIS

Application Number: 15899844
Application Type: Utility
Filing Date: 2018-02
Publication Date: 2019-01
Patent Classification: ["536", "007100"]

Abstract:
The invention described herein relates to processes for preparing ketolide antibacterial agents. In particular, the invention relates to intermediates and processes for preparing ketolides that include a 1,2,3-triazole substituted side chain.

Claim (Index 34):
An intermediate of the formulae wherein:\n A is CH 2 , C(O), C(O)O, C(O)NH, S(O) 2 , S(O) 2 NH, or C(O)NHS(O) 2 ; \n B is saturated C 0 C 10 ; or B is unsaturated C 2 C 10 ; or \n AB taken together is alkylene, alkenylene, cycloalkylene, or arylene; \n C is hydrogen, halogen, hydroxy, acyl, acyloxy, sulfonyl, ureyl, and carbamoyl, and alkyl, alkoxy, heteroalkyl, aryl, heteroaryl, arylalkyl, and heteroarylalkyl, each of which is optionally substituted; or C is C P , where C P  is a protected form of C; \n R 100  is hydrogen or a hydroxyl protecting group; and \n N P  is NH 2  or protected amino.

Metadata:
- Claim Count in Document: 14.0
- Percentile: 88.0
- Lexical Diversity: 1.25926
- Patent Class: 536.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['14774843', '12739652', '15262277', '13821314', '14387643']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.633684761816705
- 35 USC 102 Novelty (BERT): 0.5097971316282132
- Combined Prediction Score: 0.6212959987978558
- Mean Citation Score: 242.742502
- Max Citation Score: 301.2052
- Similarity Product: 226.91789837112427

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test