PATENT CLAIM ANALYSIS

Application Number: 15889578
Application Type: Utility
Filing Date: 2018-02
Publication Date: 2018-08
Patent Classification: ["546", "112000"]

Abstract:
The present invention provides compounds of formula I: or a pharmaceutically acceptable salt, tautomer, or stereoisomer, thereof, wherein the variables are as defined herein. The present invention further provides pharmaceutical compositions comprising such compounds and methods of using such compounds for treating, preventing, inhibiting, ameliorating, or eradicating the pathology and/or symptomology of a disease caused by a  Plasmodium  parasite, such as malaria.

Claim (Index 9):
The compound of  claim 1 , wherein the compound is of Formula Ia: or a pharmaceutical acceptable salt, tautomer or stereoisomer thereof,\n wherein\n n is 1 or 2; \n n is 1 or 2; \n Ring A is phenyl, pyridinyl, or pyrimidinyl; \n Ring C is phenyl or pyridinyl; \n L is *\u2014C(O)NR 2 \u2014 or *\u2014NR 2 C(O)\u2014, wherein R 2  is selected from hydrogen, C 1-4 alkyl, C 1-4 alkylamino-(C 0-4 )alkylene, C 3-6 cycloalkyl-(C 0-4 )alkylene, C 4-6 heterocycloalkyl-(C 0-4 )alkylene, wherein the C 4-6 heterocycloalkyl is selected from the group consisting of piperazinyl, morpholinyl, thiomorpholinyl, tetrahydropyranyl, and oxetanyl, and wherein the C 3-6 cycloalkyl is selected from cyclopropyl, cyclobutyl, cyclopentyl and cyclohexyl; \n each R 1  is independently *\u2014C(O)NR 7 R 8  or \u2014NH 2 \u2014, wherein R 7  and R 8  are each independently hydrogen or C 1-4 alkyl; and \n R 17  is selected from the group consisting of cyano, halo, \u2014NH 2 \u2014, \u2014C(O)NH 2 , \u2014C(O)NH(CH 3 ), and \u2014C(O)N(CH 3 ) 2 .

Metadata:
- Claim Count in Document: 32.0
- Percentile: 88.0
- Lexical Diversity: 1.5102
- Patent Class: 546.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['14443609', '14083203', '15220149', '15150038', '14382210']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8157414653329222
- 35 USC 102 Novelty (BERT): 0.6521689981922579
- Combined Prediction Score: 0.7993842186188558
- Mean Citation Score: 451.795378
- Max Citation Score: 627.8209
- Similarity Product: 604.8105143368184

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test