PATENT CLAIM ANALYSIS

Application Number: 15775296
Application Type: Utility
Filing Date: 2018-05
Publication Date: 2018-12
Patent Classification: ["514", "300000"]

Abstract:
In crop production in the fields of agriculture, horticulture and the like, the damage caused by insect pests etc. is still immense, and insect pests resistant to existing insecticides have emerged. Under such circumstances, the development of novel agricultural and horticultural insecticides is desired. The present invention provides an agricultural and horticultural insecticide comprising, as an active ingredient, a 3H-pyrrolopyridine compound represented by the general formula (1): (wherein A 1 , A 2 , and A 3  each represent a nitrogen atom or a CH group, R 1  represents an ethyl group, R 2  and R 4  each represent a hydrogen atom, R 3  and R 7  each represent a haloalkyl group, R 5  and R 6  each represent a fluorine atom, and m represents 0 or 2), an N-oxide thereof or a salt thereof; and a method for using the agricultural and horticultural insecticide.

Claim (Index 1):
A 3H-pyrrolopyridine compound represented by the general formula (1): {wherein:\n R 1  represents: \n (a1) a (C 1 -C 6 ) alkyl group; (a2) a (C 3 -C 6 ) cycloalkyl group; (a3) a (C 2 -C 6 ) alkenyl group; or (a4) a (C 2 -C 6 ) alkynyl group,\n R 2  and R 4  may be the same or different and each represent: \n (b1) a hydrogen atom; (b2) a halogen atom; (b3) a hydroxyl group; (b4) a formyl group; (b5) a cyano group; (b6) a (C 1 -C 6 ) alkyl group; (b7) a (C 3 -C 6 ) cycloalkyl group; (b8) a (C 1 -C 6 ) alkoxy group; (b9) a halo (C 1 -C 6 ) alkyl group; (b10) a halo (C 3 -C 6 ) cycloalkyl group; (b11) a halo (C 1 -C 6 ) alkoxy group; (b12) a (C 1 -C 6 ) alkylthio group; (b13) a (C 1 -C 6 ) alkylsulfinyl group; (b14) a (C 1 -C 6 ) alkylsulfonyl group; (b15) a halo (C 1 -C 6 ) alkylthio group; (b16) a halo (C 1 -C 6 ) alkylsulfinyl group; (b17) a halo (C 1 -C 6 ) alkylsulfonyl group; (b18) a (C 3 -C 6 ) cycloalkyl (C 1 -C 6 ) alkoxy group; (b19) a R 9 (R 10 )N group (wherein R 9  and R 10  may be the same or different and each represent a hydrogen atom, a (C 1 -C 6 ) alkyl group, a (C 3 -C 6 ) cycloalkyl (C 1 -C 6 ) alkyl group, a halo (C 1 -C 6 ) alkyl group, a (C 1 -C 6 ) alkylcarbonyl group, a (C 1 -C 6 ) alkoxycarbonyl group or a phenylcarbonyl group); (b20) a mono-(C 1 -C 6 ) alkylaminocarbonyl NH group; (b21) a mono-(C 1 -C 6 ) alkylaminothiocarbonyl NH group; (b22) a C(R 9 )\u2550NOR 10  group (wherein R 9  and R 10  are as defined above); (b23) a carboxyl group; (b24) a (C 1 -C 6 ) alkoxycarbonyl group; (b25) a R 9 (R 10 )N carbonyl group (wherein R 9  and R 10  are as defined above); (b26) an aryl group; (b27) an aryl group having, on the ring, 1 to 5 substituting groups which may be the same or different and are selected from the group consisting of a halogen atom, a (C 1 -C 6 ) alkyl group, a halo (C 1 -C 6 ) alkyl group, a (C 1 -C 6 ) alkoxy group, a halo (C 1 -C 6 ) alkoxy group, a (C 1 -C 6 ) alkylthio group, a halo (C 1 -C 6 ) alkylthio group, a (C 1 -C 6 ) alkylsulfinyl group, a halo (C 1 -C 6 ) alkylsulfinyl group, a (C 1 -C 6 ) alkylsulfonyl group and a halo (C 1 -C 6 ) alkylsulfonyl group; (b28) an aryl (C 1 -C 6 ) alkyl group; (b29) an aryl (C 1 -C 6 ) alkyl group having, on the ring, 1 to 5 substituting groups which may be the same or different and are selected from the group consisting of a halogen atom, a (C 1 -C 6 ) alkyl group, a halo (C 1 -C 6 ) alkyl group, a (C 1 -C 6 ) alkoxy group, a halo (C 1 -C 6 ) alkoxy group, a (C 1 -C 6 ) alkylthio group, a halo (C 1 -C 6 ) alkylthio group, a (C 1 -C 6 ) alkylsulfinyl group, a halo (C 1 -C 6 ) alkylsulfinyl group, a (C 1 -C 6 ) alkylsulfonyl group and a halo (C 1 -C 6 ) alkylsulfonyl group; (b30) an aryl (C 1 -C 6 ) alkyloxy group; (b31) an aryl (C 1 -C 6 ) alkyloxy group having, on the ring, 1 to 5 substituting groups which may be the same or different and are selected from the group consisting of a halogen atom, a (C 1 -C 6 ) alkyl group, a halo (C 1 -C 6 ) alkyl group, a (C 1 -C 6 ) alkoxy group, a halo (C 1 -C 6 ) alkoxy group, a (C 1 -C 6 ) alkylthio group, a halo (C 1 -C 6 ) alkylthio group, a (C 1 -C 6 ) alkylsulfinyl group, a halo (C 1 -C 6 ) alkylsulfinyl group, a (C 1 -C 6 ) alkylsulfonyl group and a halo (C 1 -C 6 ) alkylsulfonyl group; (b32) an aryl (C 1 -C 6 ) alkyl NH group; (b33) an aryl (C 1 -C 6 ) alkyl NH group having, on the ring, 1 to 5 substituting groups which may be the same or different and are selected from the group consisting of a halogen atom, a (C 1 -C 6 ) alkyl group, a halo (C 1 -C 6 ) alkyl group, a (C 1 -C 6 ) alkoxy group, a halo (C 1 -C 6 ) alkoxy group, a (C 1 -C 6 ) alkylthio group, a halo (C 1 -C 6 ) alkylthio group, a (C 1 -C 6 ) alkylsulfinyl group, a halo (C 1 -C 6 ) alkylsulfinyl group, a (C 1 -C 6 ) alkylsulfonyl group and a halo (C 1 -C 6 ) alkylsulfonyl group; (b34) a heterocyclic group; or (b35) a heterocyclic group having, on the ring, 1 to 3 substituting groups which may be the same or different and are selected from the group consisting of a halogen atom, a (C 1 -C 6 ) alkyl group, a halo (C 1 -C 6 ) alkyl group, a (C 1 -C 6 ) alkoxy group, a halo (C 1 -C 6 ) alkoxy group, a (C 1 -C 6 ) alkylthio group, a halo (C 1 -C 6 ) alkylthio group, a (C 1 -C 6 ) alkylsulfinyl group, a halo (C 1 -C 6 ) alkylsulfinyl group, a (C 1 -C 6 ) alkylsulfonyl group and a halo (C 1 -C 6 ) alkylsulfonyl group,\n R 3  and R 7  may be the same or different and each represent: \n (c1) a hydrogen atom; (c2) a halogen atom; (c3) a hydroxyl group; (c4) a formyl group; (c5) a cyano group; (c6) a (C 1 -C 6 ) alkyl group; (c7) a (C 3 -C 6 ) cycloalkyl group; (c8) a (C 1 -C 6 ) alkoxy group; (c9) a halo (C 1 -C 6 ) alkyl group; (c10) a halo (C 3 -C 6 ) cycloalkyl group; (c11) a halo (C 1 -C 6 ) alkoxy group; (c12) a (C 1 -C 6 ) alkylthio group; (c13) a (C 1 -C 6 ) alkylsulfinyl group; (c14) a (C 1 -C 6 ) alkylsulfonyl group; (c15) a halo (C 1 -C 6 ) alkylthio group; (c16) a halo (C 1 -C 6 ) alkylsulfinyl group; (c17) a halo (C 1 -C 6 ) alkylsulfonyl group; (c18) a (C 3 -C 6 ) cycloalkyl (C 1 -C 6 ) alkoxy group; (c19) a R 9 (R 10 )N group (wherein R 9  and R 10  are as defined above); (c20) a mono-(C 1 -C 6 ) alkylaminocarbonyl NH group; (c21) a mono-(C 1 -C 6 ) alkylaminothiocarbonyl NH group; (c22) a C(R 9 )\u2550NOR 10  group (wherein R 9  and R 10  are as defined above); (c23) a carboxyl group; (c24) a (C 1 -C 6 ) alkoxycarbonyl group; (c25) a R 9 (R 10 )N carbonyl group (wherein R 9  and R 10  are as defined above); (c26) an aryl group; (c27) an aryl group having, on the ring, 1 to 5 substituting groups which may be the same or different and are selected from the group consisting of a halogen atom, a cyano group, a (C 1 -C 6 ) alkyl group, a halo (C 1 -C 6 ) alkyl group, a (C 1 -C 6 ) alkoxy group, a halo (C 1 -C 6 ) alkoxy group, a (C 1 -C 6 ) alkylthio group, a halo (C 1 -C 6 ) alkylthio group, a (C 1 -C 6 ) alkylsulfinyl group, a halo (C 1 -C 6 ) alkylsulfinyl group, a (C 1 -C 6 ) alkylsulfonyl group and a halo (C 1 -C 6 ) alkylsulfonyl group; (c28) an aryl (C 1 -C 6 ) alkyl group; (c29) an aryl (C 1 -C 6 ) alkyl group having, on the ring, 1 to 5 substituting groups which may be the same or different and are selected from the group consisting of a halogen atom, a (C 1 -C 6 ) alkyl group, a halo (C 1 -C 6 ) alkyl group, a (C 1 -C 6 ) alkoxy group, a halo (C 1 -C 6 ) alkoxy group, a (C 1 -C 6 ) alkylthio group, a halo (C 1 -C 6 ) alkylthio group, a (C 1 -C 6 ) alkylsulfinyl group, a halo (C 1 -C 6 ) alkylsulfinyl group, a (C 1 -C 6 ) alkylsulfonyl group and a halo (C 1 -C 6 ) alkylsulfonyl group; (c30) an aryl (C 1 -C 6 ) alkyloxy group; (c31) an aryl (C 1 -C 6 ) alkyloxy group having, on the ring, 1 to 5 substituting groups which may be the same or different and are selected from the group consisting of a halogen atom, a (C 1 -C 6 ) alkyl group, a halo (C 1 -C 6 ) alkyl group, a (C 1 -C 6 ) alkoxy group, a halo (C 1 -C 6 ) alkoxy group, a (C 1 -C 6 ) alkylthio group, a halo (C 1 -C 6 ) alkylthio group, a (C 1 -C 6 ) alkylsulfinyl group, a halo (C 1 -C 6 ) alkylsulfinyl group, a (C 1 -C 6 ) alkylsulfonyl group and a halo (C 1 -C 6 ) alkylsulfonyl group; (c32) an aryl (C 1 -C 6 ) alkyl NH group; (c33) an aryl (C 1 -C 6 ) alkyl NH group having, on the ring, 1 to 5 substituting groups which may be the same or different and are selected from the group consisting of a halogen atom, a (C 1 -C 6 ) alkyl group, a halo (C 1 -C 6 ) alkyl group, a (C 1 -C 6 ) alkoxy group, a halo (C 1 -C 6 ) alkoxy group, a (C 1 -C 6 ) alkylthio group, a halo (C 1 -C 6 ) alkylthio group, a (C 1 -C 6 ) alkylsulfinyl group, a halo (C 1 -C 6 ) alkylsulfinyl group, a (C 1 -C 6 ) alkylsulfonyl group and a halo (C 1 -C 6 ) alkylsulfonyl group; (c34) a heterocyclic group; or (c35) a heterocyclic group having, on the ring, 1 to 3 substituting groups which may be the same or different and are selected from the group consisting of a halogen atom, a (C 1 -C 6 ) alkyl group, a halo (C 1 -C 6 ) alkyl group, a (C 1 -C 6 ) alkoxy group, a halo (C 1 -C 6 ) alkoxy group, a (C 1 -C 6 ) alkylthio group, a halo (C 1 -C 6 ) alkylthio group, a (C 1 -C 6 ) alkylsulfinyl group, a halo (C 1 -C 6 ) alkylsulfinyl group, a (C 1 -C 6 ) alkylsulfonyl group and a halo (C 1 -C 6 ) alkylsulfonyl group,\n R 5  and R 6  may be the same or different and each represent: \n (d1) a halogen atom; (d2) a cyano group; (d3) a (C 1 -C 6 ) alkyl group; (d4) a (C 1 -C 6 ) alkylthio group; (d5) a (C 1 -C 6 ) alkylsulfonyl group; or (d6) a (C 1 -C 6 ) alkoxycarbonyl group, or alternatively (d7) R 5  and R 6  are joined together to form a 3- to 6-membered aliphatic ring,\n R 3  and R 4  may be combined to form an aromatic ring, \n A 1 , A 2  and A 3  may be the same or different and each represent a nitrogen atom, N\u2014O or a C\u2014R 8  group (wherein R 8  represents (e1) a hydrogen atom; or (e2) a halogen atom), and \n m represents 0, 1 or 2}, \n an N-oxide thereof or a salt thereof.

Metadata:
- Claim Count in Document: 18.0
- Percentile: 93.0
- Lexical Diversity: 1.94186
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15572107', '14771672', '15545078', '16327236', '14375060']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8118363839996239
- 35 USC 102 Novelty (BERT): 0.5366737033830751
- Combined Prediction Score: 0.784320115937969
- Mean Citation Score: 357.1692720000001
- Max Citation Score: 363.5027
- Similarity Product: 290.0443802687288

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 0
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test