PATENT CLAIM ANALYSIS

Application Number: 16063370
Application Type: Utility
Filing Date: 2018-06
Publication Date: 2019-02
Patent Classification: ["514", "339000"]

Abstract:
The present invention covers heteroarylbenzimidazole compounds of general formula (I) in which R 1 , R 2 , R 3 , R 4  and R 5  are as defined herein, methods of preparing said compounds, intermediate compounds useful for preparing said compounds, pharmaceutical compositions and combinations comprising said compounds and the use of said compounds for manufacturing pharmaceutical compositions for the treatment or prophylaxis of diseases, in particular of hyperproliferative and/or inflammatory disorders, as a sole agent or in combination with other active ingredients.

Claim (Index 6):
The compound according to  claim 1 , wherein\n R 1  represents a group selected from in which \u201c*\u201d represents the point of attachment to the rest of the molecule, the ring of said group being, besides R 6 , optionally substituted further one or two times, differently or identically, with a R 7  group; R 2  represents a group in which \u201c*\u201d represents the point of attachment to the rest of the molecule; R 3  represents a hydrogen atom; R 4  represents a hydrogen atom; R 5  represents a hydrogen atom; R 6  represents a group selected from methyl, ethyl, 2,2-difluoroethyl, 2,2,2-trifluoroethyl, (cyclopropyl)-(methyl)-, (2,2-difluorocyclopropyl)-(methyl)-, (2,2-dichlorocyclopropyl)-(methyl)-, (2,2-dimethylcyclopropyl)-(methyl)-, (2-methylcyclopropyl)-(methyl)-, (1-methylcyclopropyl)-(methyl)-, (1-chlorocyclopropyl)-(methyl)-, (cyclobutyl)-(methyl)-, 3,3-difluorocyclobutyl-(methyl)- and (cyclopentyl)-methyl)-; R 7  represents a group selected from methyl, trifluoromethyl, (methoxy)-(methyl)-, ethylamino, isopropylamino, (cyclopropyl)-(methyl)-amino-, cyclopropylamino, cyclobutylamino, dimethylamino, azetidin-1-yl, 3,3-difluoroazetidin-1-yl, 3-trifluoromethylazetidin-1-yl, pyrrolidin-1-yl, piperidin-1-yl, morpholinyl, methoxy, ethoxy, iso-propoxy, 2,2,2-trifluoroethoxy, 2,2-difluoropropoxy and (cyclopropyl)-(methoxy)-; R 9  represents a hydrogen atom or a methyl group; R 10  represents a \u2014C(\u2550O)R 12  group; R 12  represents a group selected from 2,2,2-trifluoroethyl, cyclopropyl, (1-trifluoromethyl)-(cyclopropyl)-, 2,2-difluorocyclopropyl and 2,2-difluoro-1-methylcyclopropyl, or a stereoisomer, a tautomer, an N-oxide, a hydrate, a solvate, or a salt thereof, or a mixture of same.

Metadata:
- Claim Count in Document: 16.0
- Percentile: 94.0
- Lexical Diversity: 1.61404
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15080068', '14772865', '14403151', '13078192', '15083503']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7983009672059921
- 35 USC 102 Novelty (BERT): 0.520748482740537
- Combined Prediction Score: 0.7705457187594467
- Mean Citation Score: 306.67584
- Max Citation Score: 309.4958200000001
- Similarity Product: 217.0263486162437

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test