PATENT CLAIM ANALYSIS

Application Number: 15945429
Application Type: Utility
Filing Date: 2018-04
Publication Date: 2018-08
Patent Classification: ["514", "210180"]

Abstract:
The invention relates to a compound of formula (I) wherein R 1  and R 2  are defined as in the description and in the claims. The compound of formula (I) can be used as a medicament.

Claim (Index 23):
The compound according to  claim 1  which compound is selected from the group consisting of:\n (S)\u2014N-(3-(3-chloro-4-(trifluoromethoxy)phenyl)-1-(1-cyanocyclopropylamino)-1-oxopropan-2-yl)-2-(4-fluorophenyl)-2H-1,2,3-triazole-4-carboxamide; \n (S)\u2014N-(3-(3-chloro-4-(trifluoromethoxy)phenyl)-1-(1-cyanocyclopropylamino)-1-oxopropan-2-yl)-3-phenylisoxazole-5-carboxamide; \n (S)\u2014N-(3-(3-chloro-4-(trifluoromethoxy)phenyl)-1-(1-cyanocyclopropylamino)-1-oxopropan-2-yl)-2-phenyl-2H-1,2,3-triazole-4-carboxamide; \n 2-(4-chlorophenyl)-N-[(2S)-3-[3-chloro-4-(trifluoromethoxy)phenyl]-1-[(1-cyanocyclopropyl)amino]-1-oxopropan-2-yl]triazole-4-carboxamide; \n N-[(2S)-3-[3-chloro-4-(trifluoromethoxy)phenyl]-1-[(1-cyanocyclopropyl)amino]-1-oxopropan-2-yl]-2-pyridin-3-yltriazole-4-carboxamide; \n N-[(2S)-1-[(1-cyanocyclopropyl)amino]-3-(3,4-dichlorophenyl)-1-oxopropan-2-yl]-2-(4-fluorophenyl)triazole-4-carboxamide; \n N-[(2S)-3-[3-chloro-4-(trifluoromethoxy)phenyl]-1-[(1-cyanocyclopropyl)amino]-1-oxopropan-2-yl]-2-(6-fluoropyridin-3-yl)triazole-4-carboxamide; \n N-[(2S)-3-[3-chloro-4-(trifluoromethoxy)phenyl]-1-[(1-cyanocyclopropyl)amino]-1-oxopropan-2-yl]-2-propan-2-yltriazole-4-carboxamide; \n N-[(2S)-3-[3-chloro-4-(trifluoromethoxy)phenyl]-1-[(1-cyanocyclopropyl)amino]-1-oxopropan-2-yl]-2-methyltriazole-4-carboxamide; \n N-[(2S)-3-[3-chloro-4-(2-methoxyethoxy)phenyl]-1-[(1-cyanocyclopropyl)amino]-1-oxopropan-2-yl]-2-(4-fluorophenyl)triazole-4-carboxamide; and \n 2-tert-butyl-N-[(2S)-3-[3-chloro-4-(trifluoromethoxy)phenyl]-1-[(1-cyanocyclopropyl)amino]-1-oxopropan-2-yl]triazole-4-carboxamide; or, a pharmaceutically acceptable salt thereof.

Metadata:
- Claim Count in Document: 14.0
- Percentile: 91.0
- Lexical Diversity: 1.5
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['12761427', '15567668', '13148296', '15320155', '13049941']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8120994462123268
- 35 USC 102 Novelty (BERT): 0.5133365705686301
- Combined Prediction Score: 0.7822231586479571
- Mean Citation Score: 279.468204
- Max Citation Score: 312.96332
- Similarity Product: 250.9480590826464

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test