PATENT CLAIM ANALYSIS

Application Number: 16067619
Application Type: Utility
Filing Date: 2018-07
Publication Date: 2019-01
Patent Classification: ["514", "345000"]

Abstract:
The present invention provides compounds of Formula (I): or stereoisomers, tautomers, or pharmaceutically-acceptable salts thereof wherein all the variables are as defined herein. These compounds are selective ROCK inhibitors. This invention also relates to pharmaceutical compositions comprising these compounds and methods of treating cardiovascular, smooth muscle, oncologic, neuropathologic, autoimmune, fibrotic, and/or inflammatory disorders using the same.

Claim (Index 13):
The compound of  claim 12  or a stereoisomer, an enantiomer, a diastereoisomer, a tautomer, a pharmaceutically-acceptable salt thereof, wherein:\n R 5  is selected from H, C 1-4  alkyl substituted with 1-4 R 7 , \n alternatively, R 5  and R 5  are taken together with the nitrogen atom to which they are attached to form a heterocycle selected from R 7 , at each occurrence, is independently selected from H, halogen, C 1-4  alkyl, C 1-4  alkoxy, CN, OH, CF 3 , \u2014NR 8 R 8 , SO 2 C 1-4 alkyl, \u2014(CH 2 ) n -carbocycle, and \u2014(CH 2 ) n -heterocycle, wherein said alkyl, alkoxyl, carbocycle, and heterocycle are substituted with 0-4 R 9 . R 8 , at each occurrence, is independently selected from H and C 1-4  alkyl; and R 9 , at each occurrence, is independently selected from halogen, OH, NO 2 , CHF 2 , CF 3 , C 1-4  alkyl, C 1-4  alkoxy, CH 2 OH, CO 2 H, CO 2 (C 1-4  alkyl), CONH 2 , \u2014NH 2 , and a 4- to 10-membered heterocycle.

Metadata:
- Claim Count in Document: 1.0
- Percentile: 95.0
- Lexical Diversity: 1.2963
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['14797414', '14759495', '15890436', '14157564', '14900238']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8304860959355421
- 35 USC 102 Novelty (BERT): 0.6172393116608765
- Combined Prediction Score: 0.8091614175080756
- Mean Citation Score: 524.2081519999998
- Max Citation Score: 581.0306400000002
- Similarity Product: 487.83192088665976

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test