PATENT CLAIM ANALYSIS

Application Number: 16228284
Application Type: Utility
Filing Date: 2018-12
Publication Date: 2019-04
Patent Classification: ["544", "376000"]

Abstract:
The present invention provides a heterocyclic compound represented by the general formula (1): The compound of the present invention has a wide treatment spectrum for mental disorders including central nervous system disorders, no side effects and high safety.

Claim (Index 16):
A process for producing a heterocyclic compound represented by the formula (1): [wherein ring Q represented by represents (wherein represents \u2014NH\u2014CH 2 \u2014, \u2014N\u2014CH\u2014, \u2014CH 2 \u2014NH\u2014 or \u2014CH\u2014N\u2014; and\n the carbon-carbon bond\n \n \n between the 3-position and 4-position of the heterocyclic skeleton containing Z and Y represents a single bond or a double bond);\n the ring Q may have at least one substituent selected from the group consisting of a lower alkyl group, a lower alkenyl group, a lower alkynyl group, a hydroxy group, a lower alkoxy group, a halogenated lower alkyl group, an aryl group, an aryl lower alkyl group, an aryl lower alkoxy group, an arylcarbonyl group, a lower alkenyloxy group, a lower alkanoyl group, a lower alkanoyloxy group, a cycloalkyl group, a cycloalkyl lower alkyl group, a halogen atom, a carbamoyl group which may have a lower alkyl group, a carboxy group, a lower alkoxycarbonyl group, an amino group which may have a lower alkanoyl group, a nitro group, a hydroxy lower alkyl group, an amino lower alkyl group which may have a lower alkyl group, a thienyl group, a saturated 3- to 8-membered heteromonocyclic group containing 1 to 2 nitrogen atoms-substituted lower alkyl group and an oxo group; \n R 2  represents a hydrogen atom or a lower alkyl group; and \n A represents \u2014O-A 1 - (wherein A 1  represents an alkylene group which may be substituted with a hydroxy group (wherein the alkylene group may contain one oxygen atom) or a lower alkenylene group) or a lower alkylene group; \n provided that when A represents a lower alkylene group, the ring Q represents a bicyclic group selected from the group consisting of: \n (wherein the carbon-carbon bond\n \n represents a single bond or a double bond)] or a salt thereof,\n characterized by comprising a reaction of a compound represented by the formula: \n (wherein the ring Q and A are the same as defined above, and X 1  represents a halogen atom or a group which causes a substitution reaction the same as in a halogen atom) or a salt thereof with a compound represented by the formula: (wherein R 2  is the same as defined above) or a salt thereof.

Metadata:
- Claim Count in Document: 2.0
- Percentile: 98.0
- Lexical Diversity: 1.19444
- Patent Class: 544.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15697196', '12970690', '14089504', '11659005', '14928972']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8245064692192714
- 35 USC 102 Novelty (BERT): 0.6261314961829282
- Combined Prediction Score: 0.804668971915637
- Mean Citation Score: 556.557896
- Max Citation Score: 585.1553299999998
- Similarity Product: 567.1532024146973

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 0

Dataset: test