PATENT CLAIM ANALYSIS

Application Number: 15743079
Application Type: Utility
Filing Date: 2018-01
Publication Date: 2019-03
Patent Classification: ["549", "058000"]

Abstract:
Described herein, inter alia, are compositions and methods for modulating mu opioid receptor activity.

Claim (Index 12):
The compound of  claim 11 , wherein Ring B is R 4 -substituted or unsubstituted (C 3 -C 10 ) cycloalkyl, R 4 -substituted or unsubstituted 5 to 10 membered heterocycloalkyl, R 4 -substituted or unsubstituted (C 6 -C 10 ) aryl, or R 4 -substituted or unsubstituted 5 to 10 membered heteroaryl;\n R 4  is independently oxo, halogen, \u2014CX a 3 , \u2014CN, \u2014SO n1 R 14 , \u2014SO v1 NR 11 R 12 , \u2014NHNR 11 R 12 , \u2014ONR 11 R 12 , \u2014NHC\u2550(O)NHNR 11 R 12 , \u2014NHC\u2550(O)NR 11 R 12 , \u2014N(O) m1 , \u2014NR 11 R 12 , \u2014C(O)R 13 , C(O) \u2014OR 13 , \u2014C(O)NR 11 R 12 , \u2014OR 14 , \u2014NR 11 SO 2 R 14 , \u2014NR 11 C\u2550(O)R 13 , \u2014NR 11 C(O)OR 13 , \u2014NR 11 OR 13 , \u2014CHX 2 , \u2014CH 2 X, \u2014OCX 3 , \u2014OCHX 2 , substituted or unsubstituted alkyl, substituted or unsubstituted heteroalkyl, substituted or unsubstituted cycloalkyl, substituted or unsubstituted heterocycloalkyl, substituted or unsubstituted aryl, or substituted or unsubstituted heteroaryl; two adjacent R 4  substituents may optionally be joined to form a substituted or unsubstituted cycloalkyl, substituted or unsubstituted heterocycloalkyl, substituted or unsubstituted aryl, or substituted or unsubstituted heteroaryl; R 11 , R 12 , R 13 , and R 14  are independently hydrogen, halogen, \u2014CF 3 , \u2014CN, \u2014OH, \u2014NH 2 , \u2014COOH, \u2014CONH 2 , \u2014NO 2 , \u2014SH, \u2014SO 3 H, \u2014SO 4 H, \u2014SO 2 NH 2 , \u2014NHNH 2 , \u2014ONH 2 , \u2014NHC\u2550(O)NHNH 2 , \u2014NHC\u2550(O)NH 2 , \u2014NHSO 2 H, \u2014NHC\u2550(O)H, \u2014NHC(O)OH, \u2014NHOH, \u2014CHF 2 , \u2014CH 2 F, \u2014OCF 3 , \u2014OCHF 2 , substituted or unsubstituted alkyl, substituted or unsubstituted heteroalkyl, substituted or unsubstituted cycloalkyl, substituted or unsubstituted heterocycloalkyl, substituted or unsubstituted aryl, or substituted or unsubstituted heteroaryl; R 11  and R 12  substituents bonded to the same nitrogen atom may optionally be joined to form a substituted or unsubstituted heterocycloalkyl or substituted or unsubstituted heteroaryl;\n m1 and v1 are independently 1 or 2; \n n1 is independently an integer from 0 to 4; and \n X a  is independently \u2014Cl, \u2014Br, \u2014I, or \u2014F.

Metadata:
- Claim Count in Document: 20.0
- Percentile: 86.0
- Lexical Diversity: 1.0625
- Patent Class: 549.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15757238', '15614278', '16301200', '16066285', '14815480']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7704490861503729
- 35 USC 102 Novelty (BERT): 0.566450098859041
- Combined Prediction Score: 0.7500491874212396
- Mean Citation Score: 435.678492
- Max Citation Score: 455.39282
- Similarity Product: 339.51145623341563

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test