PATENT CLAIM ANALYSIS

Application Number: 15767945
Application Type: Utility
Filing Date: 2018-04
Publication Date: 2018-10
Patent Classification: ["514", "064000"]

Abstract:
The present invention provides a urea peptidomimetic boronic compound and pharmaceutical compositions thereof, their preparative methods and uses. The compounds are represented by the following formula (1).

Claim (Index 14):
A method for preparation of the compound according to  claim 1 , wherein: the compound is prepared according to process (B);\n the process (B) comprising:\n (B1) formation of carbamido group by coupling; \n (B2) hydrolysis of methyl ester group; (B3) formation of amido group; (B4) optionally forming boronic acid compounds or diol ester compounds; optionally hydrolyzing the pinacol ester obtained by step (B3) to obtain the corresponding boronic acid compound; optionally, further esterifying the boronic acid compound with a diol, to obtain the corresponding diol ester compounds.

Metadata:
- Claim Count in Document: 13.0
- Percentile: 91.0
- Lexical Diversity: 1.10345
- Patent Class: 514.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['13379142', '16300162', '14567480', '14734233', '13582678']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7117379932406227
- 35 USC 102 Novelty (BERT): 0.505566930449029
- Combined Prediction Score: 0.6911208869614633
- Mean Citation Score: 214.68997
- Max Citation Score: 237.31741
- Similarity Product: 167.18043050898555

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test