PATENT CLAIM ANALYSIS

Application Number: 15864750
Application Type: Utility
Filing Date: 2018-01
Publication Date: 2018-07
Patent Classification: ["514", "253100"]

Abstract:
The invention relates to compounds of formula IA and pharmaceutically acceptable derivatives thereof, compositions comprising an effective amount of a compound of formula IA or a pharmaceutically acceptable derivative thereof, and methods for treating or preventing a condition such as pain, UI, an ulcer, IBD and IBS, comprising administering to an animal in need thereof an effective amount of a compound of formula IA or a pharmaceutically acceptable derivative thereof.

Claim (Index 5):
A compound of formula III: or a pharmaceutically acceptable salt thereof, wherein\n X is O, S, N\u2014CN, N\u2014OH, or N\u2014OR 10 ; \n W is N or C; \n the dashed line denotes the presence or absence of a bond, and when the dashed line denotes the presence of a bond or W is N then R 4  is absent, otherwise R 4  is \u2014H, \u2014OH, \u2014OCF 3 , -halo, \u2014(C 1 -C 6 )alkyl, \u2014CH 2 OH, \u2014CH 2 Cl, \u2014CH 2 Br, \u2014CH 2 I, \u2014CH 2 F, \u2014CH(halo) 2 , \u2014CF 3 , \u2014OR 10 , \u2014SR 10 , \u2014COOH, \u2014COOR 10 , \u2014C(O)R 10 , \u2014C(O)H, \u2014OC(O)R 10 , \u2014OC(O)NHR 10 , \u2014NHC(O)R 13 , \u2014CON(R 13 ) 2 , \u2014S(O) 2 R 10 , or \u2014NO 2 ; \n each R 3  is independently: \n (a) \u2014H or \u2014(C 1 -C 6 )alkyl; or \n (b) two R 3  groups together form a (C 2 -C 6 )bridge, which is unsubstituted or substituted with 1, 2 or 3 independently selected R 8  groups, and which bridge optionally contains \u2014HC\u2550CH\u2014 within the (C 2 -C 6 )bridge; or \n (c) two R 3  groups together form a \u2014CH 2 \u2014N(R a )\u2014CH 2 \u2014 bridge, a \n bridge, or a bridge;\n R a  is \u2014H, \u2014(C 1 -C 6 )alkyl, \u2014(C 3 -C 8 )cycloalkyl, \u2014CH 2 \u2014C(O)\u2014R c , \u2014(CH 2 )\u2014C(O)\u2014OR c , \u2014(CH 2 )\u2014C(O)\u2014N(R c ) 2 , \u2014(CH 2 ) 2 \u2014O\u2014R c , \u2014(CH 2 ) 2 \u2014S(O) 2 \u2014N(R c ) 2 , or \u2014(CH 2 ) 2 \u2014N(R c )S(O) 2 \u2014R c ; \n R b  is: \n (a) \u2014H, \u2014(C 1 -C 6 )alkyl, \u2014(C 3 -C 8 )cycloalkyl, -(3- to 7-membered)heterocycle, \u2014N(R c ) 2 , \u2014N(R c )\u2014(C 3 -C 8 )cycloalkyl, or \u2014N(R c )-(3- to 7-membered)heterocycle; or \n (b) -phenyl, -(5- or 6-membered)heteroaryl, \u2014N(R c )-phenyl, or \u2014N(R c )-(5- to 10-membered)heteroaryl, each of which is unsubstituted or substituted with 1, 2 or 3 independently selected R 7  groups; \n each R c  is independently \u2014H or \u2014(C 1 -C 4 )alkyl; \n m is the integer 0, 1, or 2; \n wherein Ar 1  is: \n R 1  is \u2014Cl, \u2014F, \u2014CF 3 , or \u2014CH 3 ; wherein Ar 2  is: R 14  is \u2014H, \u2014Cl, \u2014F, \u2014Br, \u2014CF 3 , \u2014OCF 3 , \u2014(C 1 -C 6 )alkyl, \u2014SO 2 CF 3 , \u2014SO 2 (C 1 -C 6 )alkyl, \u2014OCH 3 , \u2014OCH 2 CH 3 , or \u2014OCH(CH 3 ) 2 ; R 14\u2032  is \u2014H, \u2014Cl, \u2014F, \u2014Br, \u2014CF 3 , \u2014OCF 3 , \u2014(C 1 -C 6 )alkyl, \u2014SO 2 CF 3 , \u2014SO 2 (C 1 -C 6 )alkyl, \u2014OCH 3 , \u2014OCH 2 CH 3 , or \u2014OCH(CH 3 ) 2 ; and R 8  and R 9  are independently \u2014H, \u2014Cl, \u2014Br, \u2014F, \u2014CH 3 , \u2014OCH 3 , \u2014OCH 2 CH 3 , \u2014CF 3 , \u2014OCF 3 , iso-propyl, or tert-butyl.

Metadata:
- Claim Count in Document: 32.0
- Percentile: 86.0
- Lexical Diversity: 1.925
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['14498724', '13396450', '12110155', '15179612', '14237848']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8827271273613775
- 35 USC 102 Novelty (BERT): 0.7504262914312695
- Combined Prediction Score: 0.8694970437683668
- Mean Citation Score: 842.7405679999997
- Max Citation Score: 945.5279
- Similarity Product: 840.0100469071091

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test