PATENT CLAIM ANALYSIS

Application Number: 15766222
Application Type: Utility
Filing Date: 2018-04
Publication Date: 2018-10
Patent Classification: ["514", "277000"]

Abstract:
The present invention relates to compounds of formula (I) and salts thereof, pharmaceutical compositions containing such compounds and to their use in therapy.

Claim (Index 27):
A compound of Formula (I) or a pharmaceutically acceptable salt thereof: wherein\n R 1  is C 1-3 alkyl or cyclopropyl; \n R2 is \u2014CH 3 , C 2-6 alkyl, \u2014C 2-6 alkylOR 5 , \u2014C 2-6 alkylNR 5 R 6 , \u2014(CH 2 ) m SO 2 C 1-3 alkyl, \u2014(CH 2 ) m C(O)NR 5 R 6 , \u2014(CH 2 ) m CN, \u2014(CH 2 ) m CO 2 R 5 , \u2014(CH 2 ) m NHCO 2 C(CH 3 ) 3 , or \u2014(CH 2 ) n C 5-6 heteroaryl, \n wherein said C 2-6 alkyl is optionally substituted by one, two, three, four, or five times by fluoro; or said C 5-6 heteroaryl is optionally substituted by one or two substituents independently selected from halo, C 1-4 alkyl, C 3-4 cycloalkyl, and \u2014OR 5 ; \n R 3  is phenyl, C 5-6 heteroaryl, C 9-11 heteroaryl, or \u2014(CH 2 ) q -phenyl, \n wherein said phenyl is optionally substituted one, two, or three times by R 9 , said C 5-6 heteroaryl is optionally substituted by C 1-3 alkyl, C 3-4 cycloalkyl, C 1-3 alkoxy, or halo; or said C 9-11 heteroaryl is optionally substituted one, two, or three times independently selected from \u2014C 1-3 alkylR 10 , \u2014OCH 3 , \u2014OCHF 2 , \u2014OCF 3 , \u2014OC 2-3 alkylR 10 , halo, oxo, and \u2014CN; \n R 4  is \u2014H, C 1-4 alkyl, cyclopropyl, \u2014CH 2 OR 11 , or \u2014CH 2 CH 2 OR 11 ; \n R 5  and R 6  are each independently selected from \u2014H, C 1-3 alkyl, and C 2-4 alkylOC 0-3 alkyl; \n each R 9  is independently selected from \u2014NR 12 R 13 , fluoro, \u2014CN, \u2014CH 2 CN, \u2014CO 2 R 11 , \u2014C(O)C 1-3 alkyl, \u2014OH, \u2014OCHF 2 , \u2014OCF 3 , \u2014O\u2014C 2-6 alkylR 10 , \u2014OCH 3 , \u2014OCH 2 CH 2 NR 12 R 13 , \u2014C 1-6 alkylR 10 , \u2014OC 4-7 heterocyclyl, \u2014OCH 2 C 4-7 heterocyclyl, \u2014CH 2 C 4-7 heterocyclyl, \u2014CH 2 CH 2 C 4-7 heterocyclyl, \u2014NHC(O)R 11 , \u2014SO 2 R 11 , and \u2014SOR 11 ; \n R 10  is \u2014H, \u2014OR 11 , or \u2014NR 12 R 13 ; \n R 11  is \u2014H or C 1-3 alkyl; \n R 12  and R 13  are each independently selected from \u2014H and C 1-3 alkyl; or R 12  and R 13  may join together with nitrogen to which they are attached to form a C 4-7 heterocyclyl optionally containing a further heteroatom selected from nitrogen, oxygen, and sulphur and optionally substituted by one or two substituents independently selected from C 1-3 alkyl, \u2014OH, and fluoro; \n m is selected from 0, 1, 2, 3, and 4; \n n is selected from 2, 3, and 4; and \n q is selected from 1 and 2.

Metadata:
- Claim Count in Document: 2.0
- Percentile: 91.0
- Lexical Diversity: 1.125
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15762229', '15757199', '16091577', '14190477', '14977508']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7642629887063928
- 35 USC 102 Novelty (BERT): 0.5923800012591791
- Combined Prediction Score: 0.7470746899616715
- Mean Citation Score: 410.926672
- Max Citation Score: 523.60333
- Similarity Product: 409.2312592926574

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test