PATENT CLAIM ANALYSIS

Application Number: 15751515
Application Type: Utility
Filing Date: 2018-02
Publication Date: 2018-10
Patent Classification: ["504", "100000"]

Abstract:
The invention relates inter alia to compounds of the general formula (I). Also described are methods for preparing the compounds of the formula (I). The compounds according to the invention are especially suitable for controlling insects, arachnids and nematodes in agriculture, and ectoparasites in veterinary medicine and also as herbicides.

Claim (Index 1):
Compound of formula (I\u2032) in which U is \u2014C(\u2550W)-Q or \u2014S(O) 2 -Q, R 1  is H, in each case optionally substituted C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 7 -cycloalkyl, C 1 -C 6 -alkylcarbonyl, C 1 -C 6 -alkoxycarbonyl, aryl(C 1 -C 3 )-alkyl, heteroaryl(C 1 -C 3 )-alkyl, or R 1  is H in each case optionally substituted C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 7 -cycloalkyl, C 1 -C 6 -alkylcarbonyl, C 1 -C 6 -alkoxycarbonyl, C 3 -C 7 -cycloalkyl(C 1 -C 3 )-alkyl, aryl(C 1 -C 3 )-alkyl, heteroaryl(C 1 -C 3 )-alkyl, the moieties are as follows: A 1  is CR 2  or N, A 2  is CR 3  or N, A 3  is CR 4  or N, A 4  is CR 5  or N, A 5  is C, B 1  is CR 6  or N, B 2  is CR 7  or N, B 3  is CR 8  or N, B 4  is CR 9  or N, and B 5  is CR 10  or N, but not more than three of the A 1  to A 4  moieties are N and not more than three of the B 1  to B 5  moieties are simultaneously N; M 1 , M 2  are each independently H, in each case optionally substituted C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 7 -cycloalkyl, C 1 -C 6 -alkylcarbonyl, C 1 -C 6 -alkoxycarbonyl, aryl(C 1 -C 3 )-alkyl, heteroaryl(C 1 -C 3 )-alkyl, or M 1  and M 2  with the carbon atom to which they are attached form an optionally substituted 3-, 4-, 5- or 6-membered ring which optionally contains 0, 1 or 2 nitrogen atoms and/or 0, 1 or 2 oxygen atoms and/or 0, 1 or 2 sulfur atoms, or M 1  or M 2  with R 4  from A 3 , the carbon atom of A 3 , A 5  and D form a 5- or 6-membered ring optionally substituted by F, Cl, Br, I, C 1 -C 3 -alkyl, which may contain 0, 1 or 2 nitrogen atoms and/or 0, 1 or 2 oxygen atoms and/or 0, 1 or 2 sulfur atoms, R 2 , R 3 , R 4 , R 5 , R 6 , R 7 , R 9  and R 10  are each independently H, halogen, cyano, nitro, in each case optionally substituted C 1 -C 6 -alkyl, C 3 -C 6 -cycloalkyl, C 1 -C 6 -alkoxy, N\u2014C 1 -C 6 -alkoxyimino-C 1 -C 3 -alkyl, C 1 -C 6 -alkylsulfanyl, C 1 -C 6 -alkylsulfinyl, C 1 -C 6 -alkylsulfonyl, N\u2014C 1 -C 6 -alkylamino or N,N-di-C 1 -C 6 -alkylamino,\n if neither of the A 2  and A 3  moieties is N, R 3  and R 4  together with the carbon atom to which they are attached may form a 5- or 6-membered ring containing 0, 1 or 2 nitrogen atoms and/or 0 or 1 oxygen atom and/or 0 or 1 sulfur atom, or \n if neither of the A 1  and A 2  moieties is N, R 2  and R 3  together with the carbon atom to which they are attached may form a 6-membered ring containing 0, 1 or 2 nitrogen atoms; \n R 8  is halogen, cyano, nitro, in each case optionally substituted C 1 -C 6 -alkyl, C 3 -C 6 -cycloalkyl, C 1 -C 6 -alkoxy, N\u2014C 1 -C 6 -alkoxyimino-C 1 -C 3 -alkyl, C 1 -C 6 -alkylsulfanyl, C 1 -C 6 -alkylsulfinyl, C 1 -C 6 -alkylsulfonyl, N\u2014C 1 -C 6 -alkylamino or N,N-di-C 1 -C 6 -alkylamino; W is O or S, Q is H, formyl, hydroxyl, amino or in each case optionally substituted C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 6 -cycloalkyl, C 1 -C 5 -heterocycloalkyl, C 1 -C 4 -alkoxy, C 1 -C 6 -alkyl-C 3 -C 6 -cycloalkyl, C 3 -C 6 -cycloalkyl-C 1 -C 6 -alkyl, C 6 -,C 10 -C 14 -aryl, C 1 -C 5 -heteroaryl, C 6 -,C 10 -,C 14 -aryl-(C 1 -C 3 )-alkyl, C 1 -C 5 -heteroaryl-(C 1 -C 3 )-alkyl, N\u2014C 1 -C 4 -alkylamino, N\u2014C 1 -C 4 -alkylcarbonylamino, or N,N-di-C 1 -C 4 -alkylamino; or\n is an optionally poly-V-substituted unsaturated 6-membered carbocycle; or \n is an optionally poly-V-substituted unsaturated 4-, 5- or 6-membered heterocyclic ring, where \n V is independently halogen, cyano, nitro, in each case optionally substituted C 1 -C 6 -alkyl, C 1 -C 4 -alkenyl, C 1 -C 4 -alkynyl, C 3 -C 6 -cycloalkyl, C 1 -C 6 -alkoxy, N\u2014C 1 -C 6 -alkoxyimino-C 1 -C 3 -alkyl, C 1 -C 6 -alkylsulfanyl, C 1 -C 6 -alkylsulfinyl, C 1 -C 6 -alkylsulfonyl, or N,N-di-(C 1 -C 6 -alkyl)amino; T is one of the 5-membered heteroaromatic systems T1-T8 shown below, where the bond to the ring (C-B1-B2-B3-B4-B5) is indicated by an asterisk, where R 11  is independently H, optionally halogenated C 1 -C 6 -alkyl or halogen, and/or a salt, N-oxide and/or tautomeric form of a compound of the formula (Ia\u2032).

Metadata:
- Claim Count in Document: 16.0
- Percentile: 88.0
- Lexical Diversity: 1.55263
- Patent Class: 504.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15033415', '15033464', '15554501', '15533565', '14906797']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7716801675311792
- 35 USC 102 Novelty (BERT): 0.5469997741033558
- Combined Prediction Score: 0.7492121281883969
- Mean Citation Score: 327.66451
- Max Citation Score: 347.75168
- Similarity Product: 305.5519133435059

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test