PATENT CLAIM ANALYSIS

Application Number: 16317341
Application Type: Utility
Filing Date: 2019-01
Publication Date: 2019-06
Patent Classification: ["514", "338000"]

Abstract:
Derivatives of 1,2,4-Triazolo-[3,4-b]-1,3,4-thiadiazoles according to formula (I), as set forth below: processes for production thereof, pharmaceutical compositions containing the same and the use thereof in treatment of cancer.

Claim (Index 1):
A compound of formula (I) or a pharmaceutically acceptable salt thereof: wherein R 1  and R 2  are the same or different and are selected from the group consisting of C 1 -C 5  alkyl, phenyl, methylphenyl, R 3  is selected from the group consisting of CH 2 R 8 , CH 2 CH 2 R 3 , CH\u2550CHR 8 , CH 2 CH 2 CH 2 R 8 , CH 2 CH\u2550CHR 8 , CH\u2550CHCH 2 R 8 , CH\u2550CH\u2014OR 8 , CH 2 \u2014OR 8 , CH 2 CH 2 \u2014OR 8 , CH\u2550CH\u2014NHR 8 , CH 2 \u2014NHRs, CH 2 CH 2 \u2014NHR 8 , CH\u2550CH\u2014SR 8 , CH 2 \u2014SR 8 , CH 2 CH 2 \u2014SR 8 , substituted or unsubstituted phenyl, benzyl, pyridyl, pyrirnidinyl, triazinyi, triazinanyl, oxazinyl, oxazinanyl, cycloexanyl, cycloexenyl, cycloexadienyl, pyranyl, oxathianyl, piperidinyl, cyclopentanyl, cyclopentenyl, cyclopentadienyl, pyrrolidinyl, pyrrolyl, furanyl, oxazolidinyl, pyrazolidinyl, thiophenyl, oxathilnyl, oxathiolyl, oxathiolanyl, wherein the substituent or substituents are selected from the group consisting of rnethyl, F, Cl, Br, I, NO 2 , ON, NH 2 , OCH 2 X, CH 2 X, CX 3 , CH 2 CH 2 X, OH, wherein X is selected from the group consisting of H, F, Cl, Br, I,\n R 4 , R 5 , R 6 , R 7  are the same or different and selected from the group consisting of: \n H, F, Cl, Br, I, NO 2 , ON, NH 2 , OCH 3 , OH, NHCH 2 CH 3 , N(CH 3 ) 2 , \n R 8  is selected from the group consisting of: \n substituted or unsubstituted phenyl, benzyl, pyridyl, pyrimidinyl, triazinyl, triazinanyi, oxazinyl, oxazinanyl, cycloexanyl, cycloexenyl, cycloexadienyl, pyranyl, oxathianyl, piperidinyl, cyclopentanyl, cyclopentenyl, cyclopentadienyl, pyrrolidinyl, pyrrolyl, furanyl, oxazolidinyl, pyrazolidinyl, thiophenyl, oxathiinyl, oxathiolyi, oxathiolanyl, wherein the substituent or substituents are selected from the group consisting of: methyl, F, Cl, Br, I, NO 2 , ON, NH 2 , OCH 2 X, CH 2 X, CX 3 , CH 2 CH 2 X, OH, wherein X is selected from the group consisting of H, F, Cl, Br, I,\n R 9  is selected from the group consisting of: NHR 10 , NR 11 R 12 , \n R 10  is selected from the group consisting of: C 1 -C 5  alkyl, phenyl, \n R 11  and R 12  are the same or different and are C 1 -C 5  alkyl.

Metadata:
- Claim Count in Document: 2.0
- Percentile: 99.0
- Lexical Diversity: 1.11765
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['12187524', '14403014', '13628216', '14927502', '11894900']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7746722254453826
- 35 USC 102 Novelty (BERT): 0.5101525013950791
- Combined Prediction Score: 0.7482202530403523
- Mean Citation Score: 245.702024
- Max Citation Score: 248.3725
- Similarity Product: 166.75574469298124

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test