PATENT CLAIM ANALYSIS

Application Number: 16139950
Application Type: Utility
Filing Date: 2018-09
Publication Date: 2019-01
Patent Classification: ["514", "254020"]

Abstract:
A compound, or a pharmaceutically acceptable salt or ester thereof, according to formula I: R 20 -(Z) b -(Y) c —(R 21 ) a —(X) d —R 22 —R 23  wherein R 20  is aryl, substituted aryl, heteroaryl, substituted heteroaryl, cycloalkyl, substituted cycloalkyl, heterocycloalkyl, substituted heterocycloalkyl, alkoxy, aryloxy, a thio-containing group, or a seleno-containing group; Z is alkanediyl, substituted alkanediyl, cycloalkanediyl, or substituted cycloalkanediyl; Y is S, O, S(═O), —S(═O)(═O)—, or NR 10 , wherein R 10  is H or alkyl; R 21  is alkanediyl, substituted alkanediyl, cycloalkanediyl, substituted cycloalkanediyl, alkadienyl, substituted alkadienyl, cycloalkenediyl, substituted cycloalkenediyl, alkatrienyl, substituted alkatrienyl; X is —C(═O)—, —S(═O)(═O)—, or —N(H)C(═O)—; R 22  includes at least one divalent amino radical; R 23  is aryl, substituted aryl, heteroaryl, substituted heteroaryl, cycloalkyl, substituted cycloalkyl, heterocycloalkyl, substituted heterocycloalkyl, alkoxy, aryloxy, a thio-containing group, or a seleno-containing group; a, b, c, and d independently are 0 or 1.

Claim (Index 1):
A compound, or a stereoisomer, pharmaceutically acceptable salt, or ester thereof, selected from:\n (i) a compound according to formula III where the bond represented by \u201c \u201d is a single or double bond,\n R 20  is (a) phenyl substituted with C 2 -C 3  perfluoroalkyl, halo, or pentafluorosulfanyl, (b) thiophenyl substituted with C 1 -C 3  alkyl, or (c) cycloalkyl substituted with C 1 -C 3  perfluoroalkyl, \n R 23  is (a) phenyl mono- or di-substituted with substituents selected from halo, C 1 -C 3  alkyl, C 1 -C 3  perfluoroalkyl, pentafluorosulfanyl, cyano, \u2014C(O)Oalkyl, or \u2014C(O)N(H)alkyl, (b) pyrimidinyl, (c) cycloalkyl, or (d) heterocycloalkyl, \n R 24  and R 25  are absent if the bond represented by \u201c \u201d is a double bond, or R 24  and R 25  independently are hydrogen, deuterium, C 1 -C 3  perhaloalkyl, halo, or cyano, or R 24  and R 25  together form \u2014CH 2 \u2014, and \n R 26  and R 27  independently are hydrogen, deuterium, or halo, \n wherein if R 24 -R 27  are hydrogen, then R 20  is not halogen-substituted phenyl; or\n (ii) a compound in Table A, where each R independently is C 1 -C 3  perfluoroalkyl, halo, pentafluorosulfanyl, \u2014C(O)Oalkyl, or C(O)N(H)alkyl, R 28  is O, N(CH 3 ), or CH 2 , R 29  is N, O, or S, and R 30  is CH or N \n TABLE A

Metadata:
- Claim Count in Document: 40.0
- Percentile: 97.0
- Lexical Diversity: 3.31507
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15961475', '15135334', '15923668', '15222734', '15331777']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7889157273997548
- 35 USC 102 Novelty (BERT): 0.5464470942872098
- Combined Prediction Score: 0.7646688640885003
- Mean Citation Score: 321.965828
- Max Citation Score: 408.1624
- Similarity Product: 287.41756152458186

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test