PATENT CLAIM ANALYSIS

Application Number: 16331920
Application Type: Utility
Filing Date: 2019-03
Publication Date: 2019-06
Patent Classification: ["514", "261100"]

Abstract:
Triazolo(4,5-d)pyrimidine derivatives for use in treatment or prevention of bacterial infection in a host mammal in need of such treatment or use as inhibitor of biofilm formation on a surface of biomaterial or medical device, particularly of cardiovascular device such as prosthetic heart valve or pacemakers.

Claim (Index 5):
The triazolo(4,5-d) pyrimidine derivative according to  claim 1  selected from the group consisting of:\n (1R-(1a, 2a, 3\u03b2(1R*, 2*),5\u03b2))-3-(7-((2-(3,4-difluorophenyl)cyclopropyl)amino)-5-((3,3,3-trifluoropropyl)thio)3H-1,2,3-triazolo(4,5d)pyrimidin-3-yl)5(hydroxy)cyclopentane-1,2-diol; \n (1S-(1a, 2a, 3\u03b2(1R*, 2*),5\u03b2))-3-(7-((2-(3,4-difluorophenyl)cyclopropyl)amino)-5-(propylthio)(3H-1,2,3-triazolo(4,5d)pyrimidin-3-yl)5 (2-hydroxyethoxy)cyclopentane-1,2-diol; \n (1S,2S,3R,5S)-3-[7-[(1R,2S)-2-(3,4-difluorophenyl)cyclopropylamino]-5-(propylthio)-3H-[1,2,3]-triazolo[4,5-d]pyrimidin-3-yl]-5-(2-hydroxyethoxy)-1,2-cyclopentanediol); \n (1S,2S,3R,5S)-3-[7-[(1R,2S)-2-(4-fluorophenyl)cyclopropylamino]-5-(propylthio)-3H-[1,2,3]-triazolo[4,5-d]pyrimidin-3-yl]-5-(2-hydroxyethoxy)-1,2-cyclopentanediol); \n (1S,2R,3S,4R)-4-[7-[[(1R,2S)-2-(3,4-Difluorophenyl)cyclopropyl]amino]-5-(propylthio)-3H-1,2,3-triazolo[4,5-d] pyrimidin-3-y]-1,2-3 cyclopentanetriol; and \n a pharmaceutical acceptable salt or solvate thereof, or a solvate thereof or a solvate of such a salt.

Metadata:
- Claim Count in Document: 13.0
- Percentile: 99.0
- Lexical Diversity: 1.40541
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['11841030', '11980907', '11981071', '14958619', '16025170']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.781916766706436
- 35 USC 102 Novelty (BERT): 0.5181789143188974
- Combined Prediction Score: 0.7555429814676822
- Mean Citation Score: 263.689836
- Max Citation Score: 313.5044
- Similarity Product: 268.3218911759853

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 0
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test