PATENT CLAIM ANALYSIS

Application Number: 16243301
Application Type: Utility
Filing Date: 2019-01
Publication Date: 2019-05
Patent Classification: ["546", "113000"]

Abstract:
Provided are certain fused tricyclic urea compounds and salts thereof, compositions thereof, and methods of use therefor.

Claim (Index 1):
At least one compound selected from compounds of Formula (I): stereoisomers thereof, and pharmaceutically acceptable salts thereof, wherein:\n Q is selected from C and N; \n R 1 , R 2 , and R 4 , which may be the same or different, are each selected from hydrogen, halogen, alkyl, alkenyl, cycloalkyl, aryl, heterocyclyl, heteroaryl, alkynyl, \u2014CN, \u2014NR 6 R 7 , \u2014OR 55 , COR 6 , \u2014CO 2 R 6 , \u2014CONR 6 R 7 , \u2014C(\u2550NR 6 )NR 7 R 8 , \u2014NR 6 COR 7 , \u2014NR 6 CONR 7 R 8 , \u2014NR 6 CO 2 R 7 , \u2014SO 2 R 6 , \u2014NR 6 SO 2 NR 7 R 8 , \u2014NR 6 SO 2 R 7 , and \u2014NR 6 SO 2 aryl, wherein the alkyl, alkenyl, alkynyl, cycloalkyl, heteroaryl, aryl, and heterocyclyl are independently optionally substituted with at least one substituent R 9 , or (R 1  and R 2 ), and/or (R 3  and R 4 ), together with the ring to which they are attached, form a fused ring selected from heterocyclyl and heteroaryl rings optionally substituted with at least one substituent R 9 , provided that R 1  is absent when Q is N; \n R 5  is each selected from alkyl, cycloalkyl, heterocyclyl, aryl, heteroaryl rings, each of which is optionally substituted with at least one substituent R 9 ; \n R 6 , R 7  and R 8 , which may be the same or different, are each selected from H, alkyl, alkenyl, alkynyl, cycloalkyl, heterocyclyl, aryl, and heteroaryl; or (R 6  and R 7 ), and/or (R 7  and R 8 ) together with the atom(s) to which they are attached, each form a ring selected from heterocyclyl and heteroaryl rings optionally substituted with at least one substituent R 9 ; R 9  is selected from halogen, haloalkyl, alkyl, alkenyl, cycloalkyl, aryl, heteroaryl, heterocyclyl, alkynyl, oxo, -alkyl-NR\u2032R\u2033, \u2014CN, \u2014OR\u2032, \u2014NR\u2032R\u2033, \u2014COR\u2032, \u2014CO 2 R\u2032, \u2014CONR\u2032R\u2033, \u2014C(\u2550NR\u2032)NR\u2033R\u2032\u2033, nitro, \u2014NR\u2032COR\u2033, \u2014NR\u2032CONR\u2032R\u2033, \u2014NR\u2032CO 2 R\u2033, \u2014SO 2 R\u2032, \u2014SO 2 aryl, \u2014NR\u2032SO 2 NR\u2033R\u2032\u2033, NR\u2032SO 2 R\u2033, and \u2014NR\u2032SO 2 aryl, wherein the cycloalkyl, aryl, heteroaryl, or heterocyclyl group are each independently optionally substituented by one, two or three substituents selected from halo, alkyl and haloalkyl, wherein R\u2032, R\u2033, and R\u2032\u2033 are independently selected from H, haloalkyl, alkyl, alkenyl, alkynyl, cycloalkyl, heterocyclyl, aryl, and heteroaryl, or (R\u2032 and R\u2033) and/or (R\u2033 and R\u2032\u2033) together with the atoms to which they are attached, form a ring selected from heterocyclyl optionally substituted by halogen and alkyl, and hetetoaryl rings optionally substituted by halogen and alkyl.

Metadata:
- Claim Count in Document: 80.0
- Percentile: 99.0
- Lexical Diversity: 1.17647
- Patent Class: 546.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15882067', '14901634', '14901556', '14369379', '15882064']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8369842760063847
- 35 USC 102 Novelty (BERT): 0.5990847718696791
- Combined Prediction Score: 0.8131943255927141
- Mean Citation Score: 493.518814
- Max Citation Score: 517.0235
- Similarity Product: 499.521353485167

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test