PATENT CLAIM ANALYSIS

Application Number: 15751007
Application Type: Utility
Filing Date: 2018-02
Publication Date: 2018-08
Patent Classification: ["549", "213000"]

Abstract:
Disclosed are a range of protected organoboronic acid reagents useful in the modular assembly of complex organic compounds. The reactivities of the protected organoboronic acid reagents may be varied predictably by changes to the number and identities of their substituents. Also disclosed are methods of using the protected organoboronic acid reagents in the synthesis of organic compounds.

Claim (Index 1):
A compound represented by formula I wherein independently for each occurrence\n R 10  is an organic group; \n B is a boron having sp 3  hybridization; \n R 20  is an organic group; \n each of R 21  and R 24  is selected from the group consisting of H, alkyl, alkenyl, alkynyl, aryl, heteroaryl, aralkyl, and heteroaralkyl; or R 21  and R 24  taken together form a substituted or unsubstituted C 1 -C 5  alkylene or C 2 -C 5  alkenylene bridge between the carbon atoms to which they are attached, wherein any substituent on the C 1 -C 5  alkylene or C 2 -C 5  alkenylene bridge is alkyl or halogen, or a 3- to 6-membered spirocyclic carbocyclic or heterocyclic ring attached to one bridging carbon atom, or a 3- to 6-membered carbocyclic or heterocyclic ring fused to two adjacent bridging carbon atoms; \n each of R 22  and R 23  is selected from the group consisting of H, alkyl, alkenyl, alkynyl, aryl, heteroaryl, aralkyl, and heteroaralkyl; \n R 21  and R 22 , together with the carbon atom to which they are attached, may form a substituted or unsubstituted cycloalkyl, heterocycloalkyl, cycloalkenyl, or heterocycloalkenyl group; or R 21  and R 22 , together with the carbon to which they are attached, may form a substituted or unsubstituted 3- to 6-membered carbocyclic or heterocyclic ring; and \n R 23  and R 24 , together with the carbon atom to which they are attached, may form a substituted or unsubstituted cycloalkyl, heterocycloalkyl, cycloalkenyl, or heterocycloalkenyl group; or R 23  and R 24 , together with the carbon to which they are attached, may form a substituted or unsubstituted 3- to 6-membered carbocyclic or heterocyclic ring; \n provided that if (i) R 21  and R 24  taken together do not form a substituted or unsubstituted C 1 -C 5  alkylene or C 2 -C 5  alkenylene bridge; and (ii) R 21  and R 22 , together with the carbon to which they are attached, do not form a substituted or unsubstituted 3- to 6-membered carbocyclic or heterocyclic ring; and (iii) R 23  and R 24 , together with the carbon to which they are attached, do not form a substituted or unsubstituted 3- to 6-membered carbocyclic or heterocyclic ring, then: \n (a) if R 20  is selected from the group consisting of methyl, isopropyl, 1-phenylethyl, 6,6-dimethylbicyclo[3.1.1]heptan-3-yl, 1-cyclohexylethyl, 2,6,6-trimethylbicyclo[3.1.1]heptan-3-yl, 1-benzyloxy-5-cyclopentyl, 2-(benzyloxy)cyclopentyl, 1,2,3,4-tetrahydronaphthalen-1-yl, 1-(4-methoxyphenyl)ethyl, 3,3-dimethylbutan-2-yl, 1-(naphthalen-1-yl)ethyl, and 1-phenylbutan-2-yl, then at least one of R 21 , R 22 , R 23 , and R 24  is not H; \n (b) if R 10  is phenyl and R 20  is methyl and R 21  is o-, m-, or p-CH 3 C 6 H 4 CH 2 \u2014, then at least one of R 22 , R 23 , and R 24  is not H; \n (c) if R 10  is phenyl and R 20  is methyl and R 22  is o-, m-, or p-CH 3 C 6 H 4 CH 2 \u2014, then at least one of R 21 , R 23 , and R 24  is not H; \n (d) if R 10  is phenyl and R 20  is benzyl and R 21  is a radical selected from the group consisting of methyl, ethyl, n-propyl, and n-butyl, then at least one of R 22 , R 23 , and R 24  is not H; and \n (e) if R 10  is phenyl and R 20  is benzyl and R 22  is a radical selected from the group consisting of methyl, ethyl, n-propyl, and n-butyl, then at least one of R 21 , R 23 , and R 24  is not H.

Metadata:
- Claim Count in Document: 65.0
- Percentile: 88.0
- Lexical Diversity: 1.62162
- Patent Class: 549.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['14035408', '15142418', '13030833', '12567443', '13669906']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8021682653496336
- 35 USC 102 Novelty (BERT): 0.520090064917649
- Combined Prediction Score: 0.7739604453064352
- Mean Citation Score: 318.94072199999994
- Max Citation Score: 330.1366
- Similarity Product: 244.859421492362

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 0
- Claim Label 112: 0
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test