PATENT CLAIM ANALYSIS

Application Number: 16438135
Application Type: Utility
Filing Date: 2019-06
Publication Date: 2019-10
Patent Classification: ["544", "281000"]

Abstract:
Compounds of Formula (00A) and methods of use as Janus kinase inhibitors are described herein.

Claim (Index 3):
The compound of  claim 1 , further defined as a compound of Formula (Ia) or Formula (Ib): wherein:\n R a  is H or NH 2 ; \n R 1a  is bound to a nitrogen atom of Ring A in (Ia) or is bound to a carbon atom of Ring B in (Ib), and is selected from the group consisting of:\n a. H, \n b. C 1 -C 6  alkyl optionally substituted by OH, halo, \u2014O\u2014(C 1 -C 6  alkyl), \u2014SO 2 \u2014(C 1 -C 6  alkyl), -(2-oxoindolin-1-yl), \u2014OC(O)-3-6 membered cycloalkyl, \u2014OC(O)-4-6 membered heterocycloalkyl, or phenyl; \n c. \u2014(C 1 -C 6  alkylene)-O\u2014(C 1 -C 6  alkylene)-phenyl wherein the phenyl is optionally substituted by halo; \n d. \u2014(C 1 -C 6  alkylene)-3-6 membered cycloalkyl wherein the cycloalkyl is optionally substituted by halo, OH, or CN; \n e. \u2014(C 1 -C 6  alkylene)-4-6 membered heterocycloalkyl, wherein the heterocycloalkyl is optionally substituted by oxo, C 1 -C 6  alkyl, \u2014C(O)\u2014(C 1 -C 6  alkyl), \u2014C(O)O\u2014(C 1 -C 6  alkyl), \u2014SO 2 \u2014(C 1 -C 6  alkyl), \u2014C(O)-4-6 membered heterocycloalkyl, or \u2014C(O)N(C 1 -C 6  alkyl)(C 1 -C 6  alkyl); \n f. \u2014C(O)O\u2014(C 1 -C 6  alkylene)-OH; and \n g. \u2014C(O)O\u2014(C 1 -C 6  alkylene)-phenyl; \n h. \u2014NR a R b , wherein R a  and R b  are independently selected from the group consisting of H and C 1 -C 6  alkyl optionally substituted by OH, halo, CN, phenyl, and 3-7 membered heterocycloalkyl; \n \n R 2a  is selected from the group consisting of H, C 1 -C 6  alkyl optionally substituted by OH, and phenyl; \n R 3a  is selected from the group consisting of H, C 1 -C 6  alkyl optionally substituted by OH, and phenyl; \n Ring A is a 3-7 membered heterocycloalkyl; and \n Ring B is a 3-7 membered heterocycloalkyl or a 3-7 membered heterocyclyalkenyl, wherein p 1a  is 0, 1 or 2 and p 2a  is 0, 1 or 2, \n provided that Ring A and Ring B together form a 6-11 membered bicyclic heterocycloalkyl.

Metadata:
- Claim Count in Document: 50.0
- Percentile: 100.0
- Lexical Diversity: 1.05882
- Patent Class: 544.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15139164', '15543826', '14904801', '14451600', '15257926']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8095525706175551
- 35 USC 102 Novelty (BERT): 0.584021293230305
- Combined Prediction Score: 0.7869994428788301
- Mean Citation Score: 405.063252
- Max Citation Score: 495.0762
- Similarity Product: 429.7903089289426

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 0
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test