PATENT CLAIM ANALYSIS

Application Number: 15757816
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2018-12
Patent Classification: ["514", "302000"]

Abstract:
The present invention relates to compounds of general formula I wherein the groups R, R 1 , R 2 , m and n are defined as in claim  1 , which have valuable pharmacological properties, in particular bind to the GPR40 receptor and modulate its activity. The compounds are suitable for treatment and prevention of diseases which can be influenced by this receptor, such as metabolic diseases, in particular diabetes type 2. Furthermore, the invention relates to novel intermediates, useful for the synthesis of compounds of formula I.

Claim (Index 3):
The compound according to  claim 1 , wherein\n R is selected from the group consisting of F, Cl, NC\u2014, H 2 NC(\u2550O)\u2014, H 3 CHN\u2014C(\u2550O)\u2014, (H 3 C) 2 N\u2014C(\u2550O)\u2014, HOOC\u2014, H 2 N\u2014, HO\u2014;\n C 1-3 -alkyl optionally substituted with 1 or more F or optionally monosubstituted with HO\u2014; \n cyclopropyl optionally monosubstituted with NC\u2014; \n H 3 C\u2014O\u2014 optionally monosubstituted with C 1-4 -alkyl, HOOC\u2014, oxetanyl, tetrahydrofuranyl, tetrahydropyranyl, 1,1-dioxotetrahydrothiopyranyl, or phenyl, wherein said C 1-4 -alkyl group is optionally monosubstituted with NC\u2014, HO\u2014 or H 3 C\u2014S(\u2550O) 2 \u2014, and wherein each of said oxetanyl, tetrahydrofuranyl, tetrahydropyranyl, 1,1-dioxotetrahydrothiopyranyl groups is optionally monosubstituted with H 3 C\u2014 or HO\u2014; \n cyclopropyl-O\u2014, tetrahydrofuranyl-O\u2014 and tetrahydropyranyl-O\u2014; and \n a heteroaryl group selected from the group consisting of pyrazolyl, [1,2,4]oxadiazolyl, tetrazolyl, pyridyl, pyridin-2-onyl, pyrazinyl, pyrimidinyl, and pyrimidin-4-onyl, wherein each of said heteroaryl groups is optionally monosubstituted with H 3 C\u2014 and wherein each H\u2014N group in said heteroaryl groups is optionally replaced with H 3 C\u2014N or (H 3 C) 2 C(OH)\u2014H 2 C\u2014N; \n or a salt thereof.

Metadata:
- Claim Count in Document: 26.0
- Percentile: 90.0
- Lexical Diversity: 1.70175
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['15225038', '16484124', '15818790', '13803237', '15876237']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8179017387885867
- 35 USC 102 Novelty (BERT): 0.5503863959339618
- Combined Prediction Score: 0.7911502045031242
- Mean Citation Score: 390.195968
- Max Citation Score: 394.82303
- Similarity Product: 390.8766625949556

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test