PATENT CLAIM ANALYSIS

Application Number: 16155846
Application Type: Utility
Filing Date: 2018-10
Publication Date: 2019-02
Patent Classification: ["544", "281000"]

Abstract:
The present teachings provide a compound represented by structural formula (I-0), or a pharmaceutically acceptable salt thereof. Also described are pharmaceutical compositions and methods of use thereof.

Claim (Index 29):
The compound of any one of  claims 1 - 7  and  20 - 25 , wherein R 2  is\n 4-10 membered heterocycloalkyl containing one ring heteroatom which is nitrogen optionally substituted with hydroxy, hydroxy(C 1 -C 3 )alkyl, \u2014C(\u2550O)(C 1 -C 3 )alkyl, or (C 3 -C 7 )cycloalkyl; \n 5-10 membered nitrogen-containing heteroaryl; \n OR c2 , wherein R c2  is phenyl optionally substituted with halogen, (C 1 -C 3 )alkyl, \u2014N(R a1 ) 2  or 4-6 membered heterocycloalkyl containing one ring heteroatom which is nitrogen; pyridinyl optionally substituted with halogen or (C 1 -C 3 )alkyl; piperidinyl optionally substituted with 4-6 membered heterocycloalkyl containing one ring heteroatom which is oxygen, or (C 1 -C 3 )alkoxy; pyrrolidinyl optionally substituted with 4-6 membered heterocycloalkyl containing one ring heteroatom which is oxygen or (C 1 -C 3 )alkoxy; or azetidinyl optionally substituted with 4-6 membered heterocycloalkyl containing one ring heteroatom which is oxygen or (C 1 -C 3 )alkoxy; wherein R a1  is H or (C 1 -C 3 )alkyl, or \n NHR b2  or N((C 1 -C 3 )alkyl)R b2  wherein R b2  is (C 1 -C 4 )alkyl, (C 3 -C 7 )cycloalkyl, 3-7 membered heterocycloalkyl containing one ring heteroatom which is oxygen, phenyl, or 5-6 membered nitrogen-containing heteroaryl;\n wherein the (C 1 -C 4 )alkyl represented by R b2  is optionally substituted with one or more groups selected from hydroxy, \u2014C(\u2550O)NH 2 , (C 1 -C 4 )alkyl, hydroxy(C 1 -C 3 )alkyl, (C 3 -C 7 )cycloalkyl, 3-7 membered heterocycloalkyl containing one ring heteroatom which is oxygen, and wherein the (C 3 -C 7 )cycloalkyl, 3-7 membered heterocycloalkyl, phenyl, and 5-6 membered nitrogen-containing heteroaryl substituents in the group represented by R b2  are optionally substituted with hydroxy, halogen, (C 1 -C 3 )alkyl, (C 1 -C 3 )alkoxy, hydroxy(C 1 -C 3 )alkyl.

Metadata:
- Claim Count in Document: 113.0
- Percentile: 97.0
- Lexical Diversity: 1.10345
- Patent Class: 544.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['14443072', '15434275', '14351381', '15543826', '14382123']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7949389914218765
- 35 USC 102 Novelty (BERT): 0.590865894231983
- Combined Prediction Score: 0.7745316817028872
- Mean Citation Score: 421.832804
- Max Citation Score: 504.46133
- Similarity Product: 441.4197201892936

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test