PATENT CLAIM ANALYSIS

Application Number: 15987458
Application Type: Utility
Filing Date: 2018-05
Publication Date: 2018-09
Patent Classification: ["544", "237000"]

Abstract:
The present invention relates to a class of substituted triazolopiperazine compounds, tautomers, enantiomers, diastereomers, racemates, metabolites, metabolic precursors, and pharmaceutically acceptable salts, esters, prodrugs or hydrate thereof, a preparation methods therefor, intermediates and a use thereof in the preparation of drugs for prevention and treatment of diseases associated with PARP including various ischemic diseases, neurodegenerative diseases and cancers.

Claim (Index 3):
The substituted triazolopiperazine compound represented by formula (I) according to  claim 1 , tautomers, enantiomers, diastereomers, racemates, metabolites, metabolic precursors, pharmaceutically acceptable salts, esters, prodrugs or hydrates thereof,\n wherein, Y is A and B are each independently hydrogen or methyl; alternatively, A and B together with the carbon atoms to which they are attached form a benzene ring; X is hydrogen or halogen; R is halogen, COOR 1 , substituted or unsubstituted phenyl, substituted or unsubstituted 5- and 6-membered heterocyclic ring, substituted or unsubstituted 5- and 6-membered heteroaromatic ring, wherein the substituent in the substituted phenyl, heterocyclic ring, or heteroaromatic ring is selected from one or more of the group consisting of methyl, halogen, trifluoromethyl, methoxy, hydroxymethyl; R 1  is selected from hydrogen, methyl and ethyl.

Metadata:
- Claim Count in Document: 9.0
- Percentile: 93.0
- Lexical Diversity: 1.44898
- Patent Class: 544.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['14418705', '15708917', '13035640', '16060701', '11849230']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8300685500688227
- 35 USC 102 Novelty (BERT): 0.5514197894449151
- Combined Prediction Score: 0.802203674006432
- Mean Citation Score: 337.94636
- Max Citation Score: 431.5869
- Similarity Product: 361.21740373778334

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test