PATENT CLAIM ANALYSIS

Application Number: 16125401
Application Type: Utility
Filing Date: 2018-09
Publication Date: 2019-01
Patent Classification: ["546", "153000"]

Abstract:
The present invention relates a new process to synthesize 1-((4-(4-Fluoro-2-methyl-1H-indol-5-yloxy)-6-methoxyquinolin-7-yloxy)methyl)cyclopropanamine (AL3818). A stable crystalline form of Al3818 has been prepared. Salts and their crystalline forms of AL3818 have been also prepared. Anti-cancer and optometric activities of AL3818 and its salts have been further tested. New process has been outlined in Scheme I.

Claim (Index 3):
The compound of  claim 1 , wherein the peaks have d values of: NO. d value 1 11.56173 2 10.22328 3 9.43969 4 8.75881 5 6.43957 6 6.11252 7 5.82962 8 5.61643 9 5.14957 10 4.77448 11 4.60215 12 4.42696 13 3.99909 14 3.89483 15 3.79886 16 3.63702 17 3.48708 18 3.33576 19 3.25978 20 3.17732 21 3.09732 22 2.99133 23 2.85271 24 2.82721 25 2.72504 26 2.65632 27 2.34534

Metadata:
- Claim Count in Document: 50.0
- Percentile: 97.0
- Lexical Diversity: 1.52174
- Patent Class: 546.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15659510', '15143630', '14760549', '12036244', '15460633']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.785671466693245
- 35 USC 102 Novelty (BERT): 0.5848788493840859
- Combined Prediction Score: 0.765592204962329
- Mean Citation Score: 366.803362
- Max Citation Score: 538.4721
- Similarity Product: 381.8533581847786

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test