PATENT CLAIM ANALYSIS

Application Number: 15764283
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2018-09
Patent Classification: ["514", "532000"]

Abstract:
The present invention relates to novel macrocyclic sulfondiimine compounds of general formula (I) as described and defined herein, and methods for their preparation, their use for the treatment and/or prophylaxis of disorders, in particular of hyper-proliferative disorders and/or virally induced infectious diseases and/or of cardiovascular diseases. The invention further relates to intermediate compounds useful in the preparation of said compounds of general formula (I).

Claim (Index 24):
A process for the preparation of a compound of formula (10), in which process a compound of the formula (9), in which R 1 , R 2 , R 3 , R 4  and L are as defined for the compound of formula (I) according to  claim 1 , is oxidised by treatment with an agent selected from iodobenzene diacetate and N-chloro succinimide, followed by the addition of an amine selected from a primary amine of the formula R 5 \u2014NH 2 , in which R 5  is as defined for the compounds of formula (I) according to the invention, and hexamethyldisilazene, to give compounds of the formula (10), and in which process the resulting compound is optionally, if appropriate, converted with the corresponding (i) solvents and/or (ii) bases or acids to the solvates, salts and/or solvates of the salts thereof.

Metadata:
- Claim Count in Document: 20.0
- Percentile: 90.0
- Lexical Diversity: 1.65909
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15303212', '15764289', '14345353', '14443368', '14443180']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8324033441626322
- 35 USC 102 Novelty (BERT): 0.5845887691112588
- Combined Prediction Score: 0.8076218866574948
- Mean Citation Score: 421.604676
- Max Citation Score: 531.68835
- Similarity Product: 403.69587574567794

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test