PATENT CLAIM ANALYSIS

Application Number: 16041836
Application Type: Utility
Filing Date: 2018-07
Publication Date: 2019-01
Patent Classification: ["514", "424000"]

Abstract:
Provided herein are compounds, derivatives thereof, composition comprising one or more of said compounds and derivatives, and methods for prevention and/or treatment of microbial infections and/or related diseases or conditions. The present compounds and/or derivatives thereof can be represented by Formula (I): The present methods include administering to a subject an effective amount of one or more compounds of Formula (I). In one embodiment, said microbial infections are bacterial infections. More specifically, said bacterial infections are staphylococcal infections.

Claim (Index 8):
A method of treating and/or preventing microbial infections and/or related diseases or conditions in a subject comprising:\n administering to said subject an effective amount of one or more compounds of formula (I), wherein R 1 , R 2 , and R 3  are independently or jointly selected from the group consisting of: H; F; Cl; Br; I; OH; CN; (C 1-4 )alkyl comprising methyl, ethyl, n-propyl, isopropyl, n-butyl, sec-butyl, isobutyl, and tert-butyl; (C 2-4 )alkenyl comprising ethenyl, propenyl, butenyl, wherein a double bond is optionally located at any position in the alkenyl carbon chain, and any alkenyl conformational isomers thereof; alkynyl; aralkyl; alkaryl; halogenated alkyl; heteroalkyl; aryl; heterocyclyl; cycloalkyl; cycloalkenyl; cycloalkynyl; hydroxyalkyl; aminoalkyl; amino; alkylamino; arylamino; dialkylamino; alkylarylamino; diarylamino; acylamino; hydroxyl; thiol; thioalkyl; alkoxy; alkylthio; alkoxyalkyl; aryloxy; arylalkoxy; acyloxy; nitro; carbamoyl; trifluoromethyl; phenoxy; benzyloxy; phosphonic acid; phosphate ester; sulfonic acid (\u2014SO 3 H); sulfonate ester; sulfonamide; alkaryl; arylalkyl; carbamate; amino; alkylamino; arylamino; dialkylamino; alkylarylamino; diarylamino; alkylthio; hetero alkyl; alkyltriphenylphosphonium; heterocyclyl; ketone (\u2550O); ether (\u2014OR 4 ); and ester (\u2014COOR 5  and \u2014OC(\u2550O)R 5 ), wherein R 1  and R 2  are optionally bonded together to form a four-, five-, or six-membered heterocyclyl, cycloalkenyl, or cycloalkyl; and wherein R 4  and R 5  are independently or jointly selected from the group consisting of: a (C 1-4 )alkyl comprising methyl, ethyl, n-propyl, isopropyl, n-butyl, sec-butyl, isobutyl, and tert-butyl; (C 2-4 )alkenyl comprising ethenyl, propenyl, butenyl, wherein a double bond is optionally located at any position in the alkenyl carbon chain, and any alkenyl conformational isomers thereof; and alkynyl.

Metadata:
- Claim Count in Document: 11.0
- Percentile: 95.0
- Lexical Diversity: 1.80392
- Patent Class: 514.0
- Transitional Phrase Type: open
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['12299934', '13364082', '15973569', '12764503', '15107531']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7556739434913394
- 35 USC 102 Novelty (BERT): 0.4994336884432622
- Combined Prediction Score: 0.7300499179865317
- Mean Citation Score: 241.809452
- Max Citation Score: 255.79655
- Similarity Product: 190.5947619558662

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test