PATENT CLAIM ANALYSIS

Application Number: 15763248
Application Type: Utility
Filing Date: 2018-03
Publication Date: 2018-09
Patent Classification: ["514", "303000"]

Abstract:
Compounds of formula (I): wherein R 1 , R 2 , R 3 , R 4 , and R 5  are as defined in the description. Medicinal products containing the same which are useful in treating cancer, neurodegenerative disorders and metabolic disorders.

Claim (Index 34):
A compound of formula (I): wherein:\n R 1  represents a cyano group, a halogen atom, or a linear or branched (C 1 -C 6 )alkyl group optionally substituted by from one to three halogen atoms, \n R 2  represents a hydrogen, a linear or branched (C 1 -C 6 )alkyl group, a linear or branched (C 2 -C 6 )alkenyl group, a linear or branched (C 2 -C 6 )alkynyl group, Cy 1 , \u2014(C 1 -C 6 )alkylene-[O] n -Cy 1 , \u2014(C 1 -C 6 )alkenylene-[O]n-Cy 1 , \u2014(C 1 -C 6 )alkylene-NR-Cy 1 , \u2014(C 1 -C 6 )alkylene-S-Cy 1 , \u2014(C 0 -C 6 )alkylene-Cy 2 -Cy 1 , or \u2014Cy 2 -(C 1 -C 6 )alkylene-Cy 1 , wherein the alkyl and alkylene moieties defined hereinbefore may be linear or branched, \n R represents a hydrogen or a linear or branched (C 1 -C 6 )alkyl group, n is 0 or 1, R 3  represents a hydrogen atom, a halogen atom, \u2014NR 6 R 6\u2032 , \u2014NH\u2014(C 0 -C 6 )alkylene-Cy 3 , \u2014NH\u2014CO\u2014(C 0 -C 6 )alkylene-Cy 3 , or \u2014NH\u2014CO\u2014(C 0 -C 6 )alkylene-O-Cy 3 , R 4  and R 5 , each independently represent a hydrogen or a halogen atom, R 6  and R 6 \u2032, each independently represent a hydrogen or a linear or branched (C 1 -C 6 )alkyl group, Cy 1 , Cy 2  and Cy 3 , independently of one another, represent a cycloalkyl group, a heterocycloalkyl group, an aryl or an heteroaryl group, wherein:\n \u201caryl\u201d means a phenyl, naphthyl, biphenyl or indenyl group, \n \u201cheteroaryl\u201d means any mono- or bi-cyclic group composed of from 5 to 10 ring members, having at least one aromatic moiety and containing from 1 to 4 hetero atoms selected from oxygen, sulphur and nitrogen, \n \u201ccycloalkyl\u201d means any mono- or bi-cyclic, non-aromatic, carbocyclic group containing from 3 to 11 ring members, which may include fused, bridged or spiro ring systems, \n \u201cheterocycloalkyl\u201d means any mono- or bi-cyclic, non-aromatic, condensed or spiro group composed of from 3 to 10 ring members and containing from 1 to 3 hetero atoms selected from oxygen, sulphur, SO, SO 2  and nitrogen, which may include fused, bridged or spiro ring systems, \n \u201c\u2014(C 0 -C 6 )alkylene-\u201d refers either to a covalent bond (\u2014C 0 alkylene-) or to an alkylene group containing 1, 2, 3, 4, 5 or 6 carbon atoms, \n wherein the aryl, heteroaryl, cycloalkyl and heterocycloalkyl groups so defined and the alkyl, alkenyl, alkynyl, alkylene, alkenylene may be substituted by from 1 to 4 groups selected from linear or branched (C 1 -C 6 )alkyl, linear or branched (C 2 -C 6 )alkenyl, linear or branched (C 2 -C 6 )alkynyl, linear or branched (C 1 -C 6 )alkoxy, linear or branched (C 1 -C 6 )alkyl-S\u2014, hydroxy, oxo (or N-oxide where appropriate), nitro, cyano, \u2014C(O)\u2014OR\u2032, \u2014C(O)\u2014R\u2032, \u2014O\u2014C(O)\u2014R\u2032, \u2014C(O)\u2014NR\u2032R\u2033, \u2014NR\u2032\u2014C(O)\u2014R\u2033, \u2014NR\u2032R\u2033, linear or branched (C 1 -C 6 )polyhaloalkyl, difluoromethoxy, trifluoromethoxy, or halogen, wherein R\u2032 and R\u2033 independently of one another represent a hydrogen atom or a substituted linear or branched (C 1 -C 6 )alkyl group, its enantiomers and diastereoisomers, and addition salts thereof with a pharmaceutically acceptable acid or base.

Metadata:
- Claim Count in Document: 62.0
- Percentile: 90.0
- Lexical Diversity: 1.41176
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['13266976', '14389336', '10524204', '11939735', '12089050']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7874184434195196
- 35 USC 102 Novelty (BERT): 0.5439518609413049
- Combined Prediction Score: 0.7630717851716982
- Mean Citation Score: 355.59789000000006
- Max Citation Score: 376.5085
- Similarity Product: 316.78277204173804

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test