PATENT CLAIM ANALYSIS

Application Number: 15775319
Application Type: Utility
Filing Date: 2018-05
Publication Date: 2019-03
Patent Classification: ["544", "349000"]

Abstract:
There is described herein use of a compound of formula (I) below to make cyclic peptides.

Claim (Index 24):
A compound of formula (III), wherein\n R 1 , R 3 , R 4 , R 5  and R 6  are each independently selected from the group consisting of H; lower alkyl; aryl; heteroaryl; alkenyl; heterocycle; acids of the formula \u2014C(O)OH; esters of the formula \u2014C(O)OR* wherein R* is selected from alkyl and aryl; amides of the formula \u2014C(O)NR**R***, wherein R** and R*** are independently selected from H, alkyl and aryl; \u2014CH 2 C(O)R, wherein R is selected from \u2014OH, lower alkyl, aryl, -loweralkyl-aryl, or \u2014NRaRb, where Ra and Rb are independently selected from H, lower alkyl, aryl or -loweralkyl-aryl; \u2014C(O)Rc, wherein Rc is selected from lower alkyl, aryl or -lower alkyl-aryl; or -lower alkyl-ORd, wherein Rd is a suitable protecting group or OH group; all of which are optionally substituted at one or more substitutable positions with one or more suitable substituents;\n provided that R 3  or R 4  can be covalently linked to R 1  to form a cyclic secondary amine, and/or to R 5  or R 6  to form a ring; R 3  and R 4  may be covalently bound to each other to form a ring; and R 5  and R 6  may be covalently bound to each other to form a ring; \n \n stereocentres 1* and 2* and 3* are independently selected from R and S; and \n Z-L-C\u2550O is an amino acid.

Metadata:
- Claim Count in Document: 1.0
- Percentile: 93.0
- Lexical Diversity: 1.05556
- Patent Class: 544.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['12446343', '13257159', '14962952', '11426287', '12136874']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7919661871376412
- 35 USC 102 Novelty (BERT): 0.5273772969254505
- Combined Prediction Score: 0.7655072981164222
- Mean Citation Score: 315.69614199999995
- Max Citation Score: 351.15
- Similarity Product: 318.58156553506865

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test