PATENT CLAIM ANALYSIS

Application Number: 15751316
Application Type: Utility
Filing Date: 2018-02
Publication Date: 2018-08
Patent Classification: ["564", "134000"]

Abstract:
The present invention relates to processes, process steps and intermediates useful in the asymmetric bisamidation of malonic ester derivatives wherein the new processes, process steps and intermediates are, for example, useful in the preparation of asymmetric malonic acid bisanilides such as cabozantinib.

Claim (Index 7):
The process of  claim 1 , wherein converting the M a  salt of formula (II) and/or of formula (II\u2032) to the compound of formula (IV) according to (ii) comprises\n (ii.a.1) converting the M a  salt of formula (II) to a compound of formula (III) \u2003or the M a  salt of formula (II\u2032) to a compound of formula \u2003or the mixture of the M a  salt of formula (II) and the M a  salt of formula (II\u2032) to a mixture of the compounds of formula (III) and formula (III\u2032).

Metadata:
- Claim Count in Document: 11.0
- Percentile: 88.0
- Lexical Diversity: 1.46875
- Patent Class: 564.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['14494631', '10994983', '12067612', '15750339', '15453953']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7343556688266604
- 35 USC 102 Novelty (BERT): 0.5157964362984706
- Combined Prediction Score: 0.7124997455738413
- Mean Citation Score: 227.855124
- Max Citation Score: 238.50386
- Similarity Product: 177.58114558093789

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 0
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test