PATENT CLAIM ANALYSIS

Application Number: 15773975
Application Type: Utility
Filing Date: 2018-05
Publication Date: 2018-11
Patent Classification: ["514", "269000"]

Abstract:
The present teachings relate to hydroxypyridinone and hydroxypyrimidinone derivatives, pharmaceutical compositions thereof, and methods of using such compounds to treat bacterial infections.

Claim (Index 7):
The compound of  claim 6 , wherein:\n R 1  is H or C 1-6  alkyl; R 2  is H or C 1-6  alkyl; L 1  is a bivalent radical selected from a bond, \u2014(C(\u2550O)O)\u2014, \u2014(C(\u2550O)NR b )\u2014, \u2014N(R b )C(\u2550O)\u2014, a bond, \u2014(C 1-4  alkylene)-O\u2014, \u2014(C 1-4  alkylene)-N(R b )\u2014, or \u2014(C 1-4  alkylene)-S(\u2550O) 2 \u2014; L 2  is a bivalent radical is selected from \u2014(C(R 4 )(R 5 )),\u2014(C 0-3  alkylene), or \u2014(C(R 4 )(R 5 )) n \u2014(C  0-3  alkylene)-N(R 5 )\u2014; wherein each R 4  is H or an optionally substituted C 1-6  alkyl; and each R 5  is H or C 1-6  alkyl, \u2014C(\u2550O)NR b R f  or \u2014(C 1-4  alkylene)-NR b C(\u2550O)R f ; wherein R f  is H, an optionally substituted C 1-6  alkyl, an optionally substituted C 1-6  heteroalkyl, an optionally substituted C 1-6  alkenyl, an optionally substituted C 1-6  alkynyl, an optionally substituted C 6-14  aryl, an optionally substituted 5- to 14-membered heteroaryl, an optionally substituted C 3 -C 8  cycloalkyl; L 4  is a bivalent radical selected from \u2014C(\u2550O)\u2014, \u2014(C(\u2550O)O)\u2014, \u2014(C(\u2550O)NR e )\u2014, \u2014N(R e )C(\u2550O)\u2014, or \u2014(C 1-4  alkylene)-; G 1  and G 2  are each independently, at each occurrence, a bivalent radical selected from \u2014(C 6-14  arylene)- or -(5- to 14-membered heteroarylene)-;\n G 3  is H, C 3-7  cycloalkyl, C 3-10  heterocycloalkyl, C 6-14  aryl, 5- to 14-membered heteroarylene, (C 1-4  alkylene)-(C 1-4  heteroalkyl), (C 3-10  heterocycloalkylene)-(C 1-4  alkyl), (C 3-10  heterocycloalkylene)-(C 1-4  heteroalkyl), an optionally substituted alkyl, an optionally substituted heteroalkyl, an optionally substituted alkenyl, an optionally substituted alkynyl, an optionally substituted cycloalkyl, an optionally substituted heterocyclyl, or an optionally substituted alkoxy; and \n R b  and R e  are each independently, at each occurrence, H or C 1-6  alkyl; and \n n is 1 or 2.

Metadata:
- Claim Count in Document: 1.0
- Percentile: 93.0
- Lexical Diversity: 1.13636
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15773976', '15123232', '13460524', '14222500', '13121157']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7884960878649003
- 35 USC 102 Novelty (BERT): 0.575395802914027
- Combined Prediction Score: 0.767186059369813
- Mean Citation Score: 375.364822
- Max Citation Score: 519.7719999999998
- Similarity Product: 364.9514281651972

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test