PATENT CLAIM ANALYSIS

Application Number: 15953494
Application Type: Utility
Filing Date: 2018-04
Publication Date: 2018-08
Patent Classification: ["514", "235800"]

Abstract:
Disclosed are novel compounds of Formula I that are cGAS antagonists, methods of preparation of the compounds, pharmaceutical compositions comprising the compounds, and their use in medical therapy.

Claim (Index 4):
The compound of  claim 1 , or a pharmaceutically acceptable salt thereof, wherein X is S, Y is O or S, and R 2a  is pyridyl group with 0-3 substituents independently selected from the group consisting of halogen, \u2014SR 3a , \u2014S(O)R 3a , \u2014OR 3a , \u2014OCH 2 R 3b , \u2014OCH(CH 3 )R 3b , \u2014OC(O)NHR 3a , \u2014NR 3a R 4a , \u2014NHSO 2 R 3a , azido, \u2014CHO, CO 2 R 3a , cyano, C 1-6 alkyl or \u2014CR 5a R 6a R 7a , C 2-6 alkeny, \u2014C(R 5a )\u2550C(R 8a )(R 9a ), C 2-6 alkynyl, and \u2014C\u2261CR 8a .

Metadata:
- Claim Count in Document: 14.0
- Percentile: 91.0
- Lexical Diversity: 1.33333
- Patent Class: 514.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: False
- Related Applications: ['15953492', '12096432', '14343410', '12312749', '15522969']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7890929418775027
- 35 USC 102 Novelty (BERT): 0.5617204382280061
- Combined Prediction Score: 0.766355691512553
- Mean Citation Score: 329.689702
- Max Citation Score: 430.0401
- Similarity Product: 356.34170595413445

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test