PATENT CLAIM ANALYSIS

Application Number: 16313956
Application Type: Utility
Filing Date: 2018-12
Publication Date: 2019-05
Patent Classification: ["546", "197000"]

Abstract:
Compounds of formula I, wherein R a  and R b  are as defined in the claims, exhibit alpha2C antagonistic activity and are thus useful as alpha2C antagonists.

Claim (Index 6):
The compound according to  claim 1 , wherein R a  and R b  form, together with the nitrogen atom to which they are attached any one of the following groups wherein; group (4), (5), (6), or (7) is optionally further substituted with R 3 , R 4 , and/or R 5 ; Z is N or O; R 1  is oxo; R 2  is oxo; R 3  is (C 1 -C 6 )alkyl, (R 6 ) 2 N\u2014(C 1 -C 6 )alkyl, (R 6 ) 2 N\u2014(C\u2550O)\u2014(C 1 -C 6 )alkyl, cyclo(C 3 -C 6 )alkyl, cyclo(C 3 -C 6 )alkyl(C 1 -C 6 )alkyl, phenyl, phenyl(C 1 -C 6 )alkyl, heterocyclyl, or heterocyclyl(C 1 -C 6 )alkyl, wherein said phenyl, cyclo(C 3 -C 6 )alkyl, or heterocyclyl is optionally substituted with 1 or 2 substituent(s) each independently being halogen or (C 1 -C 6 )alkyl-(C\u2550O); R 4  is oxo or (C 1 -C 6 )alkyl; R 5  is (C 1 -C 6 )alkyl; R 6  is (C 1 -C 6 )alkyl; or two of R 3 , R 4  and R 5 , both attached to the same carbon ring atom form, together with the carbon ring atom to which they are attached, a 3 membered unsubstituted carbocyclic ring; and the atom marked with * is bonded to the parent molecular moiety.

Metadata:
- Claim Count in Document: 14.0
- Percentile: 98.0
- Lexical Diversity: 1.25
- Patent Class: 546.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['12668918', '14192131', '13917745', '14747485', '14725683']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.8079665030749448
- 35 USC 102 Novelty (BERT): 0.529305273191619
- Combined Prediction Score: 0.7801003800866122
- Mean Citation Score: 313.98425400000013
- Max Citation Score: 358.68304
- Similarity Product: 241.90774031981468

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test