PATENT CLAIM ANALYSIS

Application Number: 15773975
Application Type: Utility
Filing Date: 2018-05
Publication Date: 2018-11
Patent Classification: ["514", "269000"]

Abstract:
The present teachings relate to hydroxypyridinone and hydroxypyrimidinone derivatives, pharmaceutical compositions thereof, and methods of using such compounds to treat bacterial infections.

Claim (Index 15):
The compound of  claim 14 , wherein\n L 2  is a bivalent radical selected from \u2014(C(R 4 )(R 5 )) n \u2014(C 0-3  alkylene)-, \u2014(C(R 4 )(R 5 )) n \u2014C 0-3  alkylene)\u2014(C\u2014OR c )\u2014, \u2014(C(R 4 )(R 5 )) n \u2014(C 0-3  alkylene)-C(\u2550O)\u2014, \u2014(C(R 4 )(R 5 )) n \u2014(C 0-3  alkylene)-O\u2014, \u2014(C(R 4 )(R 5 )) n \u2014(C 0-3  alkylene)-N(R 5 )\u2014, \u2014(C(R 4 )(R 5 )) n \u2014(C 0-3  alkylene)-S(\u2550O) 2 \u2014; wherein each R 4  is H or optionally substituted C 1-6  alkyl; and each R 5  is independently H, an optionally substituted C 1-6  alkyl, an optionally substituted C 1-6  heteroalkyl, an optionally substituted C 1-6  alkenyl, an optionally substituted C 1-6  alkynyl, an optionally substituted C 6-14  aryl, an optionally substituted 5- to 14-membered heteroaryl, an optionally substituted C 3 -C 8  cycloalkyl, on optionally substituted \u2014(C 0-4  alkylene)-OR f , \u2014(C 0-4  alkylene)-(C 1-4  alkene), \u2014(C 0-4  alkylene)-(C 1-4  alkyne), C 2 -C 7  heterocycle, \u2014(C 0-4  alkylene)-C(\u2550O)\u2014(C 1 -C 6  alkyl), \u2014(C 0-4  alkylene)-C(\u2550O)H, alkylene)-C(\u2550O)OR f , alkylene)-CN, \u2014(C 0-4  alkylene)-halo, \u2014(C 0-4  alkylene)-NO 2 , alkylene)-N(R f ) 2 , \u2014(C 0-4  alkylene)-S(\u2550O) 2 -(R f ), \u2014(C 0-4  alkylene)-(C 6-14  aryl), \u2014(C 1-4  alkylene)-(5- to 14-membered heteroaryl), \u2014(C 0-4  alkylene)- C(\u2550O)NR b R f  or \u2014(C 0-4  alkylene)-NR b C(\u2550O)R f ; wherein each R f  is independently H, an optionally substituted alkyl, an optionally substituted cycloalkyl, an optionally substituted heterocyclyl, or an optionally substituted alkoxy; L 3  is \u2014(C 2-6  alkynylene)-; L 4  is a bivalent radical selected from \u2014C(\u2550O)\u2014, \u2014(C(\u2550O)O)\u2014, \u2014(C(\u2550O)NR e )\u2014, \u2014N(R e )C(\u2550O)\u2014, or \u2014(C 1-4  alkylene)-; G 3  is H, C 3-7  cycloalkyl, C 3-10  heterocycloalkyl, C 6-14  aryl, 5- to 14-membered heteroarylene, (C 1-4  alkylene)-(C 1-4  heteroalkyl), (C 3-10  heterocycloalkylene)-(C 1-4  alkyl), (C 3-10  heterocycloalkylene)-(C 1-4  heteroalkyl), an optionally substituted alkyl, an optionally substituted heteroalkyl, an optionally substituted alkenyl, an optionally substituted alkynyl, an optionally substituted cycloalkyl, an optionally substituted heterocyclyl, or an optionally substituted alkoxy; and R a , R b , R c , R d , and R e  are each independently, at each occurrence, H or C 1-6  alkyl; and n is 1 or 2.

Metadata:
- Claim Count in Document: 1.0
- Percentile: 93.0
- Lexical Diversity: 1.13636
- Patent Class: 514.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: False
- Related Applications: ['15773976', '15123232', '13460524', '14222500', '13121157']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7865593199548948
- 35 USC 102 Novelty (BERT): 0.5822766320661309
- Combined Prediction Score: 0.7661310511660184
- Mean Citation Score: 375.364822
- Max Citation Score: 519.7719999999998
- Similarity Product: 396.87992605829226

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 1
- Claim Label 112: 0
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test