PATENT CLAIM ANALYSIS

Application Number: 15780419
Application Type: Utility
Filing Date: 2018-05
Publication Date: 2018-12
Patent Classification: ["549", "292000"]

Abstract:
The invention relates to compounds of Formula (I), wherein the variables are as defined in the claims, which are useful in the treatment and/or prevention of bacterial infections in a subject. The invention further relates to the use of a compound of Formula (I) in the manufacture of a medicament, and medical devices when used in a method of treating or preventing a bacterial infection in a subject, and related aspects.

Claim (Index 1):
A compound of Formula I: wherein R 1  is substituted or unsubstituted C 1 -C 20 alkyl, C 2 -C 20 alkenyl, C 2 -C 20 alkynyl, C 1 -C 6 alkoxyC 1 -C 3 alkyl or C 3-6  cycloalkylC 1 -C 3 alkyl; R 2  is substituted or unsubstituted C 1 -C 20 alkyl, C 2 -C 20 alkenyl, C 2 -C 20 alkynyl, C 1 -C 6 alkoxyC 1 -C 3 alkyl, C 1 -C 6  cycloalkylC 1 -C 3 alkyl or C 1 -C 6 cycloalkenylC 1 -C 3 alkyl; R 3  is H or a bond along with the adjacent carbon defining a keto group, R 5 , C(O)R 5 , CR a R b OR 5 , CR a R b OC(O)R 5 , CR a R b OC(O)OR 5  or C(O)CHR 7 NH 2 ; R 4  is R 5 , C(O)R 5 , CR a R b OR 5 , CR a R b OC(O)R 5 , CR a R b OC(O)OR 5  or C(O)CHR 7 NH 2 ; R 5  and R 6  are independently H, or selected from the group consisting of substituted or unsubstituted C 1 -C 6 alkyl, C 3 -C 6 cycloalkyl and C 3 -C 6 cycloalkylC 1 -C 3 alkyl; R 7  is H, C 1 -C 6 alkyl, C 3 -C 6 cycloalkyl and C 3 -C 6 cycloalkylC 1 -C 3 alkyl; wherein R a  and R b  are independently selected from H and methyl; or a pharmaceutically acceptable salt, stereoisomer, N-oxide or hydrate thereof; with the provisos that\n when R 3  is a bond, R 4  is H, and R 1  and R 2  are both unsubstituted alkyl, then if R 1  is C 6 -alkyl, R 2  has at least two carbon atoms, and \n when R 3  is a bond, R 4  is H, and R 1  and R 2  are both unsubstituted C 1 -C 20  alkyl, then R 1  has at least 2 more carbon atoms than R 2 .

Metadata:
- Claim Count in Document: 14.0
- Percentile: 93.0
- Lexical Diversity: 1.76087
- Patent Class: 549.0
- Transitional Phrase Type: closed
- Component Type: 1
- Foreign Priority: True
- Related Applications: ['11204269', '12503286', '10718337', '10777455', '14880834']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.734408786866811
- 35 USC 102 Novelty (BERT): 0.5028610104501302
- Combined Prediction Score: 0.7112540092251429
- Mean Citation Score: 235.214476
- Max Citation Score: 249.48485
- Similarity Product: 187.43680224677323

Labels:
- Claim Label 101: 1
- Claim Label 102: 0
- Claim Label 103: 1
- Claim Label 112: 1
- Combined Label: 0
- Label 101 Adjusted: 1

Dataset: test