PATENT CLAIM ANALYSIS

Application Number: 16327854
Application Type: Utility
Filing Date: 2019-02
Publication Date: 2019-06
Patent Classification: ["546", "269700"]

Abstract:
The present invention relates to novel substituted phenoxy- and benzyloxy-piperidine compounds of formula (I) having P2X7 receptor (P2X7) antagonistic properties, pharmaceutical compositions comprising these compounds, chemical processes for preparing these compounds and their use in the treatment or prophylaxis of diseases associated with P2X7 receptor activity in animals, in particular humans.

Claim (Index 2):
The compound of Formula (I) according to  claim 1  or a pharmaceutically acceptable salt thereof including any stereochemically isomeric form thereof, wherein:\n n is 0 or 1; \n R 1  is methyl, or difluoromethyl; \n each of R 2 , R 3 , and R 4  independently is hydrogen, fluorine, chlorine or the R 2  and R 4  groups, taken together, form a six membered heterocyclic ring containing a nitrogen atom provided that at least one of R 2 , R 3 , and R 4  is not hydrogen; \n each of R 5  and R 6  is hydrogen, fluorine or chlorine provided that at least one of R 5  and R 6  is halogen.

Metadata:
- Claim Count in Document: 4.0
- Percentile: 99.0
- Lexical Diversity: 1.31111
- Patent Class: 546.0
- Transitional Phrase Type: none
- Component Type: 0
- Foreign Priority: True
- Related Applications: ['15115963', '14747485', '15763281', '15176597', '13057510']

Analysis Scores:
- 35 USC 101 Eligibility (BERT): 0.7967642385937952
- 35 USC 102 Novelty (BERT): 0.523182398257337
- Combined Prediction Score: 0.7694060545601494
- Mean Citation Score: 282.820674
- Max Citation Score: 340.03296
- Similarity Product: 256.74981225746154

Labels:
- Claim Label 101: 1
- Claim Label 102: 1
- Claim Label 103: 0
- Claim Label 112: 1
- Combined Label: 1
- Label 101 Adjusted: 1

Dataset: test