baber/WOPTO huggingface dataset:
Patent CZ-71198-A3 (CZ)
Title: Taxan hydrophobic derivatives supporting hydrolysis
Inventor: MAYHEW ERIC
IPC: C07D305/14
Filed: 1996-09-12
Abstract: Provided herein is a taxane having a hydrocarbon attached at the 2' and/or 7 positions, the hydrocarbon's alpha position being occupied by a "hydrolysis-promoting group" ("HPG"). Substitution of an HPG for the methylene unit ordinarily occupying the alpha position allows for enhanced in vivo hydrolysis of the hydrocarbon-taxane bond, and hence, for enhanced taxane therapeutic activity. Also provided herein are taxane-containing compositions, and methods of administering taxanes to animals, including those afflicted with cancers.
Patent SK-33798-A3 (SK)
Title: Phenylacetic acid derivatives, process for their preparation and their use as pesticides and fungicides
Inventor: MULLER BERND
IPC: C07C251/88
Filed: 1996-09-30
Abstract: The invention concerns phenylacetic acid derivatives of formula (I) in which the substituents and the indices have the following meanings: X denotes NOCH3, CHOCH3 and CHCH3; Y denotes oxygen or NR<a>; R<a> denotes hydrogen or alkyl; R denotes cyano, nitro, trifluoromethyl, halogen, alkyl and alkoxy; m stands for 0, 1 or 2, wherein the rests R can be different if m is 2; R<1> denotes hydrogen or alkyl; R<2> and R<3>, independently of each other, denote hydrogen, cyano, nitro, hydroxy, amino, halogen, optionally substituted alkyl, alkoxy, alkylthio, alkylamino, dialkylamino, alkenyl, alkenyloxy, alkenylthio, alkenylamino, N-alkenyl-N-alkylamino, alkinyl, alkinyloxy, alkinylthio, alkinylamino, N-alkinyl-N-alkylamino, cycloalkyl, cycloalkyloxy, cycloalkylthio, cycloalkylamino, N-cycloalkyl-N-alkylamino, cycloalkenyl, cycloalkenyloxy, cycloalkenylthio, cycloalkenylamino, N-cycloalkenyl-N-alkylamino, heterocyclyl, heterocyclyloxy, heterocyclylthio, heterocyclylamino, N-heterocyclyl-N-alkylamino, aryl, aryloxy, arylthio, arylamino, N-aryl-N-alkylamino, hetaryl, hetaryloxy, hetarylthio, hetarylamino and N-hetaryl-N-alkylamino; R<4> denotes one of the groups mentioned in the case of R<2> or a CR<d>=NOR<e> group; R<d> denotes one of the groups mentioned in the case of R<2>; and R<e> denotes hydrogen, optionally substituted alkyl, cycloalkyl, alkenyl, alkinyl, alkylcarbonyl, alkenylcarbonyl, alkinylcarbonyl, alkylsulphonyl, aryl, arylcarbonyl, arylsulphonyl, hetaryl, hetarylcarbonyl or hetarylsulphonyl. The invention also concerns their salts, a process for the preparation of these substances and their use.
Patent SK-67496-A3 (SK)
Title: Monoclonal anti-idiotypic antibody leading immunity response against receptor of epidermal growth factor, preparation method thereof and pharmaceutical composition containing its
Inventor: CARCELLER ANA
IPC: C07K16/00
Filed: 1996-05-23
Abstract: The present invention relates to anti-idiotypic antibodies which induce an immune response against tumors, bearing as antigen the epidermal growth factor receptor (EGFR). The antibodies of the invention may mimic said antigen. As preferred embodiment the antibodies of the invention derive from mAB 425 (ATCC HB 9629) or a humanized or chimeric derivative thereof.
Patent SK-86997-A3 (SK)
Title: Imides/amides as immunotherapeutic agents, pharmaceutical composition and their use for reducing level of tnf-alpha
Inventor: MULLER GEORGE
IPC: A61K31/4439
Filed: 1995-11-20
Abstract: Novel imide/amide ethers are inhibitors of tumor necrosis factor alpha  and can be used to combat cachexia, endotoxic shock, and retrovirus replication. A typical embodiment is 1-Phthalimido-1-(3',4'-dimethoxyphenyl)propan-1-ol.
Patent SK-94493-A3 (SK)
Inventor: ALBRECHT GERHARD
IPC: C08F20/38
Filed: 1993-09-06
Abstract: Ide o polyméry a vodné polyméme disperzie, ktoré pozostávajú z monomérov zo skupiny nenasýtených karboxylových kyselín, nenasýtených esterov karboxylových kyselín, nenasýtených sulfónových kyselín a nenasýtených N- substituovaných cyklických dikarboxylových kyselín ako aj ich použitie ako prímesí k hydraulickým spojivám.
Patent AT-511026-A3 (AT)
Title: Vorrichtung und verfahren zum wickeln einer faserbahn
Inventor: TIITTA JARI
IPC: B65H19/22
Filed: 2012-01-11
Abstract: Gegenstand der Erfindung ist eine Vorrichtung zum Wickeln einer Faserbahn, insbesondere ein Zwischenwickler für die Faserbahn, wobei der Zwischenwickler einen Abwickler (20), ein Wickelachsenlager (25), eine Ausbreitwalze (21) und einen Aufwickler (3 0) umfasst, und wobei der Aufwickler (30) eine Wickeltrommel (31) zum Bilden eines Wickelwalzenspalts mit einer zu wickelnden Maschinenrolle (15) umfasst. Die Wickeltrommel (31) für den Aufwickler (30) im Zwischenwickler hat mindestens zwei sich im Wesentlichen in vertikaler Richtung befindliche Positionen, von denen die eine eine Wickelposition ist, in der die Wickeltrommel mit der zu bildenden Maschinenrolle (15) einen Wickelwalzenspalt bildet.
Patent CS-187891-A3 (CS)
Title: Pharmaceutical combined preparations containing derivatives of cephalosporin and xanthine and their application
Inventor: KLESEL NORBERT DR
IPC: A61K31/545
Filed: 1991-06-19
Abstract: Pharmaceutical combination products containing at least one cephalosporin derivative and at least one xanthine derivative are suitable for the prophylaxis and treatment of bacterial infectious diseases and for the prophylaxis and treatment of septic shock.
Patent CZ-300492-A3 (CZ)
Title: Process for mixing and applying adhesives and apparatus for making the same
Inventor: VESTERLUND LENNART
IPC: C09J5/00
Filed: 1992-10-01
Abstract: Resin and hardener are supplied via tubes (3,4 respectively) onto the flat, smooth, mixing area (10) of a applicator roll (1). The resin and hardener are mixed in this area by squeezing them repeatedly between the contra-rotating and parallel applicator (1) and dosing rolls (2) whilst causing the mixture to extrude into the threads (11). The adhesive is then spread acoss the threaded area due to the effect of the thread helix and the adhesive is applied from the threads onto the article to be coated. - A partition plate (5) can be used to create a gap (6) that controls the amount of adhesive to be spread. The resin and hardener can be applied in varied relative amounts and will always be mixed in the missing area after being transferred there around the circumference of the rotating applicator roll (1).
Patent CZ-108097-A3 (CZ)
Title: Machine for working sides of building blocks and the like objects
Inventor: DERHAKE THOMAS DR ING
IPC: B24B7/22
Filed: 1995-10-11
Abstract: A machine is disclosed for trimming the sides of building blocks or the like, in particular dried green bricks (Z) or baked bricks (Z) that are centred, vertically clamped and thus conveyed through at least one trimming station with laterally arranged tools. The invention is characterised by a transport device with two endless belts under compression load made of flexible material and designed as conveyor and compression belts (2, 3). The conveyor and compression belts (2, 3) are forcibly guided in the lateral position by at least one groove and spring connection (7a, 8), in particular a keyway and V-rib connection, and run on a rail- or plate-shaped flat support (9) at least in the area of the trimming tools (5).
Patent CZ-131294-A3 (CZ)
Title: Process of environmental friendly stabilization of disposal sites of solid semi-permeable materials containing leacheable heavy metals
Inventor: VOTRUBA JAROSLAV ING CSC
IPC: A62D3/00
Filed: 1994-05-31
Abstract: In this method of ecologically stabilising deposits of solid semi-permeable materials firmly semi-permeable materials are mixed or overlaid by 0.01 to 20 kg/t of the contaminated material of natural or semi-synthetic insoluble humic substances from brown coal.
Patent CZ-154194-A3 (CZ)
Title: Polyvinyl chloride capable of direct working up and process for preparing thereof
Inventor: HARJUHAHTO HANNU
IPC: C08F2/18
Filed: 1992-12-23
Abstract: The invention relates to a homo- or copolymer composition of a vinyl chloride, which is ready for processing and which contains additives necessary from the point of view of the processing, such as stabilizers, lubricants, colourants, reinforcing agents and processing aids, and to a method for its preparation. The polymer has been prepared by adding into the polymerization reactor in the beginning of the polymerization, during it or at the end thereof 0.01-50 weight-% of the amount of vinyl chloride a liquid olefin oligomer and/or ethylene olefin copolymer or olefin terpolymer.
Patent CZ-168697-A3 (CZ)
Title: Liquid-cooled grate element and a grate per se
Inventor: MARTIN JOHANNES JOSEF EDMUND D
IPC: F23H7/04
Filed: 1997-06-02
Abstract: The component has at least one fluid feed channel (13,14) with parallel sections (13) and fluid inlet and outlet. The parallel sections of the channel run crossways to the component longitudinal direction and crossways to the combustible material conveyor direction. The channel sections run in a straight line and have a cross-section determining a compact, dead space-free flow. Two straight-line channel sections are joined by a linkage (14) and thus fluid flows through them in rows. The fluid inflow (15) is provided in the area of the fixture and drive end (5) and the fluid outflow (16) in the head area (7) of the grill component (1,2). All channel sections have a common fluid inlet and a common fluid outlet, with the fluid flowing through in a parallel manner.
Patent CZ-194997-A3 (CZ)
Title: Zinc-sheet roofing
Inventor: RACEK RONALD FRANCIS WALTER
IPC: E04D3/16
Filed: 1995-12-07
Abstract: A galvanised steel or zinc covering essentially comprises an assembly of sheets of said materials, laid over a non-ventilated roof support. The sheet side which faces the support is provided with a resilient, durable, organic coating which is impervious to water vapour and has a thickness of at least 50 microns.
Patent CZ-200443-A3 (CZ)
Title: Heterocyclic compounds and their use as D-Ala-D-Ala ligase inhibitors
Inventor: MOE SCOTT T
IPC: A61K31/525
Filed: 2002-06-28
Abstract: The invention is based on the discovery of a new class of heterocyclic compounds having, for example, antibacterial properties. The D-Ala-D-Ala ligase enzyme is a critical pathway enzyme in the bacterial cell-wall synthesis. The compounds can bind to and inhibit the enzyme D-Ala-D-Ala ligase. The new compounds' activity combined with their ability to cross bacterial cell membranes makes them suitable for use as antibacterial drugs or other antibacterial applications.
Patent CZ-219994-A3 (CZ)
Title: Protective cover of abrasive band grinding machines
Inventor: STRASAK MILAN ING
IPC: B23Q11/08
Filed: 1994-09-09
Abstract: The cover (1) is formed of at least one linear box piece (6) and at least one triangular box piece (7,8). The linear box piece (6) is composed of a flat box equipped with a longitudinal slot (9) on one side, while the triangular box piece (7,8) is composed of a triangular box equipped with a curved slot (16) on one side. All slots (9,16) are arranged at the level of the sanding belt (2).<IMAGE>
Patent CZ-231197-A3 (CZ)
Title: Brain-twister
Inventor: BLAZEK ZDENEK ING
IPC: A63F9/08
Filed: 1997-07-21
Abstract: Brain-twister (1) consists of movable elements which are arranged into the groups (2) of at least four mutually separated and mutually movable flat elements (3, 4) in the scope of 360 DEG , wherein one element of each group (2) creates a central flat element (3) and at least three orbital flat elements (4) are arranged symmetrically around this central flat element (3), wherein at least one of these orbital flat elements (4) is a part of the same number of orbital flat elements (4) of a neighbour group (2) of flat elements (3, 4) again with a central flat element (3), wherein all the groups (2) of flat elements (3, 4) create an infinite and closed chain in all directions and the chains are arranged into a shape of a ball.
Patent CZ-297596-A3 (CZ)
Title: Movable vault as a change-over station
Inventor: PRIMUS ILLO-FRANK DR ING
IPC: E04H5/04
Filed: 1996-10-11
Abstract: The building consists of four wall sections (14,22) combined monolithically with a floor, and a roof in the form of two separately pivotable covers (28,30). One cover is hinged in the vicinity of a gutter carrier (38) and has a skirtlike portion (36) at an angle to the ridge portion. When the building is completed and closed the skirtlike portion constitutes the upper part of one wall. In the depicted double structure the overall length (a1) is more than 4 m, the breadth (e) about 2.3 m and the maximum height (h) 1 m from ground level.
Patent CZ-298398-A3 (CZ)
Title: Pharmaceutical preparation
Inventor: SHANNON HARLAN EDGAR
IPC: A61K31/55
Filed: 1997-03-24
Abstract: The present invention provides a method for treating migraine pain comprising administering an analgesic dosage of olanzapine.
Patent CZ-317996-A3 (CZ)
Title: Binding agent system based on polyurethane for sand mixtures intended for manufacture of casting moulds and cores
Inventor: TORBUS MAREK DR
IPC: C08K5/10
Filed: 1996-10-30
Abstract: The polyurethane-based binder system (I) for foundry mould materials, contains a phenolic resin (A) with free OH groups and a polyisocyanate (B) with monomethyl esters of fatty acid(s) (C) with a chain of 12 or more C atoms as solvent or solvent component for (A) and/or (B). Also claimed are: (i) a process for the production of (I), in which (A) and/or (B) is/are dissolved in (C); and (ii) the production of foundry moulds and cores from a moulding material containing (I) as binder.
Patent CZ-319694-A3 (CZ)
Title: Eatable plastic dispersion containing quickly gelatinizing starch
Inventor: KASICA JAMES
IPC: A23D7/015
Filed: 1993-06-04
Abstract: An edible plastic dispersion not having a continuous fat phase, including at least two condensed phases, at least one of which is continuous, the dispersion comprising a first gel-forming composition and a second gel-forming composition containing 1-8 times the critical concentrations of a gelling starch having a rheological property in an aqueous dispersion characterized by a one-half G'max value at no more than about 7,250 seconds when prepared at a concentration to yield a log G'max value of 5.0 at 15,000 seconds at 11 DEG  C. provided that the aqueous dispersion of the gelling starch is initially prepared at 0 to 40 DEG  C.
Patent CZ-339695-A3 (CZ)
Title: Shifting device built-in forming machine
Inventor: ALLGOWER GERHARD DIPL ING
IPC: B21D43/05
Filed: 1995-05-26
Abstract: The arrangement comprises a cam drive which engages with pushrods to which carriages (2,15) are linked. These carriages run on transfer rails while two carriages at opposite sides are interconnected by a cross traverse (12). The traverse is connected to the carriages via raising and lowering arrangements (1). Each lowering and raising arrangement has its own drive (6) which moves a link block running in a slot, via a torque transmission mechanism in the form of a toothed belt drive or a recirculating ball spindle. <IMAGE>
Patent CZ-9903634-A3 (CZ)
Inventor: FLORIAN MARTIN
IPC: B22C3/00
Filed: 1999-10-13
Abstract: Minerální oleje jsou modifikovány polymery, které tímto
způsobem vytváří systémy Teologických a fýzikálněmechanických
vlastností v důsledku vzájemných interakcí.
Použitými polymery jsou polybutyleny, ethylenové
kopolymery (E/VAC ethylen-vinylacetatu, E/MA ethylenmethylakrylové
kyseliny, E/BA ethylenacetatu) a ataktický
polypropylen, a to v poměru k minerálnímu oleji 1:9 až 3:1
hmotnostně.
Patent CZ-430399-A3 (CZ)
Inventor: BESSODES MICHEL
IPC: C12N15/88
Filed: 1998-06-03
Abstract: Transfekční činidlo obsahující nejménějednu lipofilní oblast
spojenou s kationtovou hydrofilní oblastí, kdy sejmenovaná
kationtová hydrofilní oblast skládá z heterocyklu s 5 nebo 6
atomy, kterýje substituovaný aminoskupinami. Kationtová
*· hydrofilní oblast, kteráje meziproduktempři syntéze činidla
pro přenos nukleové kyseliny má obecný vzorec I, kde yje
celé číslo 0 nebo 1, různé yjsou na sobě nezávislé; Xje atom
kyslíku, atomdusíku, atom síry nebo atomselenu; Zjsou
nezávisle na sobě atom vodíku, skupina OR, kde Rje atom
vodíku, methylová skupina nebo skupina (CH2)n-NR,R2,
kde nje celé číslo i až 6 včetně aRi aR2 jsou nezávisle na
sobě atomvodíku nebo skupina (CH2) q -NH2, kdy se q může
pohybovat mezi 1 až 6 včetně, různá qjsou na sobě nezávislá,
skupma(CH2)m-NRiR2, kdemje celé číslo 1 ažóvčetněa
Ri aR2 jsou definovány výše nebo alternativně Tmůstek"
umožňující vazbu kationtové hydrofilní skupiny k oblasti
lipidu, přičemž nejméně jeden substituent Z nese
aminoskupinu.
Patent CZ-443599-A3 (CZ)
Title: Connecting member for connecting at least two wooden structural elements and connecting board
Inventor: MATTLE PAUL
IPC: F16B25/10
Filed: 1998-06-02
Abstract: The invention relates to a connection between two wooden construction parts (2 and 3). According to the invention, a joint plate (4) is introduced, the base part (5) of said joint plate (4) being connected to the wooden construction part (2) so that it is flush therewith, by means of screws (7). Said joint plate (4) is pushed into a slit (8) in the wooden construction part (3) and the appropriate number of connecting elements (1) are then introduced, passing through the wooden construction part (3) and the joint plate (4). A connecting element of the type used has a boring part (11) at one end and a tool contact part (12) at the other end. The material which is worked off is taken up by a segment with a reduced cross section (14) and corresponding chucking grooves (13). The connecting element can also be secured axially after placement by means of a thread (15) at one end of said connecting element. After placement, the connecting element sits in such a way that it fits perfectly in the self-made bore as a fixing element between the joining plate (4) and the wooden construction part.
Patent SK-101992-A3 (SK)
Title: Method of treatment of worn-out oil and meltable fat contaminated by poly-chlorinated biphenyls
Inventor: CVENGROS JAN
IPC: B01D3/14
Filed: 1992-04-03
Abstract: This patent describes oils and fats able to be melted contaminated with the use of polychlorinated biphenyl (PCB), while they are treated based on the fractional distillation in the wiped film of the short way evaporator so that, the distillation faction is separated, at the temperature of 100 up to 160 Celsius degrees and at the pressure of 1 up 500 Pa, where the above mentioned PCBs are being concentrated. The oil or fat volume, containing toxic PCBs is lowered, when applied this procedure, while this lowering is of a great meaning.
Patent SK-114894-A3 (SK)
Title: Set for treatment of tumors of mammalia
Inventor: BROWN J MARTIN
IPC: A61K33/243
Filed: 1994-09-22
Abstract: Disclosed is a use of a 1,2,4-benzotriazine oxide of general formula (I) or pharmacologically acceptable salts of said compound for the preparation of medicament increasing the cytotoxic effect of chemotherapy agent for the solid tumour, for administering to the mammal from about one half hour to about twenty-four hours after administering the 1,2,4-benzotriazine oxide. The meanings of substituents comprised in general formula (I) are disclosed in patent claims.
Patent SK-122894-A3 (SK)
Title: An absorbent body for an absorbent article
Inventor: GUIDOTTI TED
IPC: A61F13/15
Filed: 1993-04-21
Abstract: An absorbent body intented to form the absorbent element of an absorbent article, such as a diaper, an incontinence guard or a sanitary napkin, includes a first fibre-based absorbent layer (16) which lies proximal to the wearer in use, and a second, fibre-based absorbent layer (17) which is intented to lie distal from the wearer in use, this second layer having a high liquid-dispersing ability. An absorbent body exhibiting particularly good absorption properties has been obtained by including in the first layer (16) a superabsorbent material (18) of high gel-strength and by mixing this superabsorbent essentially uniformly in the fibre material within at least one area of the layer, and by including between the fibre layers (17a, 17b) of the second layer (17) a layer (20) of superabsorbent material.
Patent SK-144794-A3 (SK)
Title: Quaternary nitrogen containing phosphonate compounds for treating abnormal calcium and phosphate metabolism
Inventor: EBETINO FRANK H
IPC: C07F/
Filed: 1993-05-27
Abstract: The present invention relates to a quaternary nitrogen-containing, saturated or unsaturated monocyclic and bicyclic ring containing phosphonate and the pharmaceutically-acceptable salts and esters thereof, having structure (I). The present invention further relates to pharmaceutical compositions containing a safe and effective amount of a compound of the present invention, and pharmaceutically-acceptable excipients. Finally, the present invention relates to methods for treating or preventing pathological conditions characterized by abnormal calcium and phosphate metabolism in humans or other mammals. This method comprises administering to a human or other mammal in need of such treatment of a safe and effective amount of a compound or composition of the present invention.
Patent SK-185399-A3 (SK)
Title: COMPOSITIONS AND METHODS FOR REDUCING RESPIRATORY DEPRESSION ANDì (54) ATTENDANT SIDE EFFECTS OF MU OPIOID COMPOUNDS
Inventor: CHANG KWEN-JEN
IPC: A61K38/08
Filed: 1997-10-01
Abstract: A method of reducing, treating or preventing drug-mediated respiratory depression, muscle rigidity, or nausea/vomiting in an animal, incident to the administration to said animal of a mixed delta/mu opioid agonist or a respiratory depression-mediating drug, comprising administering to the animal receiving said drug an effective amount of a delta receptor agonist compound. The figure shows the effect of the positive isomer of the delta agonist BW373U86 on analgesia and respiratory depression induced by the mu agonist, alfenta. The delta agonist compound may comprise a compound of formula (I), wherein the variables of Ar, G, Z, R<2>, R<3>, R<4>, R<5>, R<6> and R<7> are herein described in the description.
Patent SK-246790-A3 (SK)
Title: The control method of collapse in coal mines
Inventor: SARISSKY DUSAN
IPC: E21C41/18
Filed: 1990-05-21
Abstract: After having worked out the coal seam (2), with the longwall face method, at the end of the mined space (1), 15 up to 35 m long, as a rule, the set of holes is drilled into the overburden (4), along the mined wall (8) and a length of these holes is not less than 15 m and the declination of them related to the normal line is 10 up to 25 degrees in the reverse direction as the sequence of the face wall is. The explosive (7) is placed in the holes (5), with a diameter of 50 up to 70 mm which is blowing up at once.
Patent SK-832015-A3 (SK)
Inventor: ZUZI BOHUSLAV
IPC: E02B3/04
Filed: 2014-04-09
Abstract: Samoplniace protipovodňové vrece pozostáva z dvoch uzavretých komôr (1), ktoré sú medzi sebou prepojené spojovacím mostom (2) v tvare T a ktoré sú vyrobené z polyesterovej tkaniny s vysokou nasiakavosťou vody. Komory (1) sú vyplnené granulovanou alebo gélovou zmesou superabsorbentov (3) vody na báze zosieťovaného polyakrylátu (SAP). Spojovací most (2) obsahuje dve manipulačné kovové oká (4).
Patent WO-0048624-A3 (WO)
Title: Utilisation d'orosomucoide pour la production d'une preparation pharmaceutique
Inventor: AUER WILFRIED
IPC: A61P31/04
Filed: 2000-02-15
Abstract: L'invention concerne l'utilisation d'orosomucoide pour la production d'une préparation pharmaceutique servant au traitement de la pancréatite aiguë.