baber/WOPTO huggingface dataset:
Patent IL-135108-A (IL)
Title: Homopiperazine derivatives, pharmaceutical compositions comprising them and their use in the preparation of medicaments for treating diseases in the central or peripheral nervous system
IPC: C07D417/04
Filed: 2000-03-16
Abstract: Heteroaryl diazacycloalkane derivatives (I) are new. Heteroaryl diazacycloalkane derivatives of formula (I) and their enantiomers or mixtures, isotopes and salts are new. [Image] n : 1-3 m : 0-2; R : H, alkyl, cycloalkyl, cycloalkylalkyl or aralkyl; R 1>aminophenyl; nitrophenyl; hydroxyphenyl; alkoxyphenyl; monocyclic 5-6 membered heterocyclyl (optionally substituted by alkyl, cycloalkyl, cycloalkylalkyl, alkenyl, alkynyl, alkoxy, cycloalkoxy, alkenoxy, alkynoxy, methylenedioxy, halo, CF 3, OCF 3, CN, amino, NO 2, COOR 3, CONR 2R 3, NHCO 2R 2and/or OCONR 2R 3); aryl (optionally substituted by alkyl, cycloalkyl, cycloalkylalkyl, alkenyl, alkynyl, alkoxy, cycloalkoxy, alkenoxy, alkynoxy, methylenedioxy, halo, CF 3, OCF 3, CN, amino and/or NO 2); X-alkyl-Y-alkyl (optionally alkyl substituted by alkoxy or thioalkoxy); X-(alkyl) o-aryl (optionally substituted by alkyl, cycloalkyl, cycloalkylalkyl, alkenyl, alkynyl, alkoxy, cycloalkoxy, alkenoxy, alkynoxy, methylene-dioxy, halo, CF 3, OCF 3, CN, amino and/or NO 2); X-(alkyl) o-Z (optionally substituted by alkyl, cycloalkyl, cycloalkylalkyl, alkenyl, alkynyl, alkoxy, cycloalkoxy, alkenoxy, alkynoxy, methylenedioxy, halo, CF 3, OCF 3, CN, amino and/or NO 2), monocyclic 5-6 membered heterocyclyl (optionally substituted by alkyl, cycloalkyl, cycloalkylalkyl, alkenyl, alkynyl, alkoxy, cycloalkoxy, alkenoxy, alkynoxy, methylenedioxy, halo, CF 3, OCF 3, CN, amino and/or NO 2) (sic), bicyclic heterocyclyl comprising a 5-6 membered monocyclic heterocyclyl fused to a benzene ring (optionally substituted by alkyl, cycloalkyl, cycloalkylalkyl, alkenyl, alkynyl, alkoxy, alkoxy-alkoxy, cycloalkoxy, alkenoxy, alkynoxy, methylenedioxy, halo, CF 3, OCF 3, CN, amino, NO 2, aryl optionally substituted by alkyl, cycloalkyl, cycloalkylalkyl, alkenyl, alkynyl, alkoxy, cycloalkoxy, alkenoxy, alkynoxy, methylenedioxy, halo, CF 3, OCF 3, CN, amine and/or NO 2) or monocyclic 5-6 membered heterocyclyl (optionally substituted by alkyl, cycloalkyl, cycloalkylalkyl, alkenyl, alkynyl, alkoxy, cycloalkoxy, alkenoxy, alkynoxy, methylenedioxy, halo, CF 3, OCF 3, CN, amino and/or NO 2); X, Y : O, S or NH, N-alkyl or Se; o : 0 or 1 and Z : 5-6 membered monocyclic heterocyclyl. ACTIVITY : Analgesic; Neuroprotective; Nootropic; Tranquilizer; Antiinflammatory; Antiaddictive; Antismoking; Anticonvulsant; Neuroleptic; Antidepressant; Antiasthmatic; Antianginal; Antimigraine. The affinity of 1-(6-chloro-5-methoxy-3-pyridyl)-homopiperazine fumaric acid salt for nicotinic Ach receptors was investigated in a test for in vitroinhibition of 3H-cytisine binding. The compound exhibited and IC 50value of 0.0007 mu M. MECHANISM OF ACTION : Nicotinic acetyl choline receptor ligand.
Patent IL-141828-A (IL)
Title: Multi-purpose end-mill
IPC: B23C5/10
Filed: 2001-03-05
Abstract: A multi-purpose end-mill to be used for different machining purposes, in particularly useful for closed or open contours machining. The end-mill comprises a cylindrical shank portion connected to a first cutting portion provided with a plurality of spaced-apart cutting teeth and a second portion provided with a plurality of different spaced-apart cutting teeth.
Patent IL-160358-A (IL)
Title: Isolated human monoclonal antibodies specific for interleukin 15 (il-15)
IPC: C07K16/24
Filed: 2004-02-12
Abstract: Isolated human monoclonal antibodies which specifically bind to IL-15 (e.g., human IL-15), and related antibody-based compositions and molecules, are disclosed. The human antibodies can be produced in a transfectoma or in a non-human transgenic animal, e.g., a transgenic mouse, capable of producing multiple isotypes of human monoclonal antibodies by undergoing V-D-J recombination and isotype switching. Also disclosed are pharmaceutical compositions comprising the human antibodies, non-human transgenic animals, and hybridomas which produce the human antibodies, and therapeutic and diagnostic methods for using the human antibodies.
Patent IL-160983-A (IL)
Title: Use of pyy for preparation of a medicament for modification of feeding behavior
IPC: A61P3/04
Filed: 2004-03-21
Abstract: Methods are disclosed for decreasing calorie intake, food intake, and appetite in a subject. The methods include peripherally administering a therapeutically effective amount of PYY or an agonist thereof to the subject, thereby decreasing the calorie intake of the subject.
Patent IL-200056-A (IL)
Title: Composition comprising an isolated agonistic antibody which specifically cross reacts with different apo - 2l receptors for use in inducing apoptosis in mammalian cancer cells
IPC: C12N5/10
Filed: 2009-07-23
Abstract: A method of making monoclonal antibodies according to a mixed antigen immunization protocol is described. In addition, antibodies obtainable by the method are disclosed which specifically cross-react with two or more different receptors to which Apo-2 ligand (Apo-2L) can bind.
Patent IN-2015DE00012-A (IN)
Inventor: NOBUYUKI SHIMOMURA
IPC: F02B1/00
Filed: 2015-01-02
Abstract: A carburetor air vent tube piping structure for a I saddle ,riding type vehicle, the saddle riding type vehicle 1 having an internal combustion engine 3 and an air cleaner case 7 arranged longitudinally be1ow.a fuel tank 16, and having an intake air passage formed by an upstream side intake pipe 62 and a downstream side intake pipe 61 with a carburetor 5 interposed between the upstream side intake pipe 62and the downstream side .intake pipe 61, wherein a detouring portion top portion 80 of an air vent tube 8 connected to a side portion of one of a left and a right of the carburetor 5, the air vent tube 8 detouring above,the upstream side intake pipe. 62 and extending to a side of the other of the left and the right of the carburetor 5, is supported at a higher 42 position than an upper portion of the upstream side intake pipe 62 by a supporting rib 71 provided to the air cleaner case' 7,upstream of the carburetor 5.
Patent JP-S62256679-A (JP)
Title: Printer
Inventor: WATARAI SHINICHI
IPC: B41J21/00
Filed: 1986-04-30
Abstract: PURPOSE:To ensure that a printing head is constantly positioned within the width of a printing medium, by outputting a moving quantity for moving the printing head in a spacing direction according to the with of the printing medium fed to a printing part, to a spacing driving part. CONSTITUTION:When a printing medium 4 is set to a tractor 12 and a paper- supplying command T is given to a controlling part 10, the tractor 12 is driven, and a leading end part of the medium 4 is moved as indicated by an arrow D, on which the width of the medium 4 is detected through an output signal from a detector 7, a moving quantity L is outputted from a calculating part 8 to a spacing driving part 5, and a printing head 1 is moved in a spacing direction by the moving quantity L by the part 5. Next, a platen 2 is driven to feed the medium 4. Accordingly, the head 1 is constantly positioned at a predetermined position according to the width of the printing medium 4 by moving the head 1 in the spacing direction.
Patent JP-S63268516-A (JP)
Title: Tension reel
Inventor: OGAWA TAKAO
IPC: B21C47/28
Filed: 1987-04-24
Abstract: PURPOSE:To improve the yield of a product strip by providing a crown on a take-up shaft of a metal strip. CONSTITUTION:A proper amount of crown is provided in advance on the take-up shaft 2 of a tension reel 1. When the strip is taken up by the take-up shaft 2 fitted with the crown, stress is prevented from concentrating at the lug parts of the metal strip and the amount of deflection generated in the take-up shaft 2 of its own is reduced. Accordingly, the optimum range of tension in taking up the strip can be prevented from decreasing even after a long period of use of the take-up shaft 2. Thereby, the lug is prevented from extending in the metal strip after it has been taken up and that strip is improved in yield.
Patent JP-H06289328-A (JP)
Title: Method for processing lens, manufacture of lens, and lens
Inventor: HAGA SHUNPU
IPC: G02B3/00
Filed: 1993-04-01
Abstract: PURPOSE:To easily obtain the lens which have both its surfaces processed differently. CONSTITUTION:The plane or concave surface side of the lens is shielded by a shield member which can contact the peripheral edge part of the lens, the part contacting the lens is sealed with a removable sealing means, and the lens is coated with a hard coat, etc. The shield member which contact with the peripheral edge part of the lens and has the surface, facing the lens, formed into a plane or concave surface is usable as the shield member. After the coating process, the seal part is removed to obtain the lens which has both its surfaces processed differently. After the seal part is removed, at least the internal surface can be coated differently from the external surface. The lens which has its external surface coated with the hard coat and its internal surface coated for fog protection is suitably used for a spectacle lens with high practicality.
Patent JP-H02279133-A (JP)
Title: Small-sized cardiogram analyzing apparatus
Inventor: HOSOYA MANABU
IPC: A61B5/332
Filed: 1989-04-21
Abstract: PURPOSE:To reduce the size of a measurement-analyzing apparatus which digitizes cardiogram information and stores the same in a memory and to reduce the patient's burden during the measurement by providing the abovementioned measurement analyzing apparatus and a monitor device which reads out and displays the cardiogram information in the memory. CONSTITUTION:The cardiac electromotive forces appearing on the surface of a human body are introduced from the plural electrodes through an electrode cable 116 which is mounted to a patient 15 and has plural electrodes to a cardiogram inputting section 3 and the signals outputted by each of the inductions corresponding to the respective electrodes from the cardiogram inputting section 3 are amplified in a main amplifier section 4 and are digitized in an A/D converting section 5. The digital signals are supplied to a digital signal processing section 6 from which the signals are passed through digital filters and are subjected to the analyzation processing of the cardiogram. The signals are then stored in the memory 7. The memory information stored in the memory 7 is read out by an operating section 12 and is displayed on a display section 10. The sending of the memory information stored in the memory 7 to a remote place by providing a modem or the like to the monitor device 2 is possible as well. The patient 15 is merely required to carry the measuring analysis apparatus 1 alone. The size and weight are reduced by as mush as the size and weight of the monitor device 2 and the patient's burden 15 can be reduced.
Patent JP-H06289951-A (JP)
Title: Picture reproduction system
Inventor: FUKAYA MASAHARU
IPC: G06T1/00
Filed: 1993-04-02
Abstract: PURPOSE:To reduce a time long occurring between a continuous reproduction processing and a reproduction processing which is processed in parallel with the continuous reproduction processing. CONSTITUTION:First and second processors 26 and 54 executing the continuous reproduction processing and the parallel processing by a command from a host computer 10a, a clock signal generation circuit 56 supplying a clock signal to the first and second processors 26 and 54, a second clock 58 outputting a time by the clock signal of the clock signal generation circuit 56, a reset means resetting the first and second clocks 22 and 58 at the time of issuing a continuous reproduction command and a comparison control means comparing the times of the first and second clocks 22 and 58 whenever a prescribed time T elapses from a time when issuing a continuous reproduction command and setting the time of the first clock 22 equal to the time of the second clock 58 when they are unequal are provided. The processing timing of the first processor 26 and that of the second processor 54 are synchronized and the time of the first clock 22 is set equal to the time of the second clock 58 at prescribed time intervals T.
Patent JP-H02280859-A (JP)
Title: Thermal spraying repairing apparatus of coke oven
Inventor: NISHINO NO
IPC: C10B29/06
Filed: 1989-04-21
Abstract: PURPOSE:To achieve the supply of air in a same way as a stationary case even during the rotation of a pipe by providing an outer cylindrical pipe to a main pipe on the outside through a bush and an air seal packing and supplying air into the main pipe from the outside through the introducing hole opened to said pipe. CONSTITUTION:The base part of a main pipe 4 having thermal spraying equipment fixed to the leading end thereof and receiving various pipings is sealed in an airtight manner and a sprocket wheel 5 is mounted thereto on the outside and an outer cylindrical pipe 8 is provided to the main pipe 4 on the outside through bushes 6 and air seal packings 7. Cooling air is supplied into the pipe 4 from the air introducing pipe 9 of the outer cylindrical pipe 8 through the air introducing hole 10 opened to the pipe 4 and the sprocket wheel 5 is rotated by a drive device. As a result, especially, in a case having no allowance of pipings in connection with a space, cooling air can be directly introduced into a rotary body without using a pipe.
Patent JP-S582261-A (JP)
Inventor: MITSUOKA YOSHIAKI
IPC: C04B28/08
Filed: 1981-06-26
Abstract: (57)【要約】本公報は電子出願前の出願データであるた め要約のデータは記録されません。
Patent JP-H05270694-A (JP)
Title: Sheet conveying device
IPC: G03G15/00
Filed: 1992-03-26
Abstract: PURPOSE:To simplify a jam treatment with a single operation knob even in the case where respective conveying rollers are rotation-driven by two driving motors, for example, in a large-size machine. CONSTITUTION:A first rotation transmission system 19 is provided for transmitting rotation of a first driving motor 16 to a conveying roller 10 upstream in the sheet conveying direction. A second rotation transmission system 29 is provided for transmitting rotation of a second driving motor 26 to a conveying roller 20 downstream of the conveying roller 10. A third rotation transmission system 30 to be freely rotation-driven by means of an operation knob 40 is provided between the first and the second transmission systems 19, 29 for joining both. A one way clutch mechanism is provided for preventing rotation transmission from the first and the second rotation transmission systems 19, 29 to the third rotation transmission system 30.
Patent JP-H0771488-A (JP)
Title: Free wheel related to direction of rotation
Inventor: FURANTSU GURATSUTSUERU
IPC: F16D41/10
Filed: 1994-04-05
Abstract: PURPOSE: To operate a free wheel only during forward run by allowing a pawl provided between a ring as a driving portion and a cage to be oscillated around an axis and to be disengageable from a recess in the cage forming a pawl stopper. CONSTITUTION: During forward run in towing operation, a ring 2 drives a ring 4 via a transmission roller 7. A pawl 12 is associated therewith via a shaft 11 provided on the ring 2, and its lock 14 is pushed into a recess 15 in a cage 5 by a holding spring 21. An arm 17 of the pawl 12 is hauls off an arm 20 of a dragging spring 18 to cause a loop 19 to rotate on a fixed ring 10. A spring arm 20 gives slight force for assisting the holding spring 21 to the pawl 12. At a high speed of rotating, the loop 19 is spread through the action of centrifugal force, resulting in the free wheel to be operated without friction. At this time, when a drive shaft 1 is braked, the ring 4 runs over the ring 2 to become a drive portion.  The ring 4 is associated with a cage 5 via a friction member 8, and the stopper 16 hits the key 14 to hold the cage 5 at a neutral position, so that the transmission roller 7 will not transmit torque.
Patent JP-S61260770-A (JP)
Title: Synchronous control circuit
Inventor: GOTO YOSHIYUKI
IPC: G11C11/401
Filed: 1985-05-14
Abstract: PURPOSE:To apply synchronous control while keeping the periodicity of a timing circuit by providing a prescribed width to an output condition of a counter circuit controlling an initial value setting signal. CONSTITUTION:A counter circuit 102 has initial value input terminals (A-C) 103-105, output terminals (QA-QC) 106-108, a clock input 109, and an initial value setting terminal (load signal input terminal) 110, the initial value is selected as (A, B, C)=(1,1,1) and the condition that the synchronizing signal passes through a gate circuit 111 and is given as a load signal is selected as (QA, QB)=(1.1). When the 1st clock-8th clock are in the relation of (QA, QB, QC)=(1.1,0) in normal one period, if no load signal is recognized in the 16th clock, when the succeeding relation of (QA, QB, QC)=(1,1,1) exists, it is recognized by the 17th clock, the initializing is obtained and the period processing is attained as if the 16th clock were transferred to the initializing operation.
Patent JP-H06295680-A (JP)
Title: Gas discharge display panel and manufacture thereof
Inventor: NAKAJIMA FUMIO
IPC: H01J17/49
Filed: 1993-04-02
Abstract: PURPOSE:To increase light emission efficiency in a discharge cell, and provide display of an extremely high brightness by forming a columnar cathode which is embedded in a cathode holding layer on one end side, and protruded out of the cathode holding layer on the other end side. CONSTITUTION:A columnar cathode 20 which is embedded in a cathode holding layer 22 on one end side, and protruded out of the layer 22 on the other end side is formed to stand in a surface of a cathode pulling pattern 18. A DC voltage is applied between a transparent electrode 24 and the cathode 20 to generate discharge inside a discharge cell 30, and UV-ray is generated. This UV-ray excites phosphor 32 in the cell 30, and light having a specified emission color is radiated through the anode 24 and a front surface substrate 14 to the external. This voltage application is executed selectively through a control and drive circuit to generate discharge light emission in the desired cell 30, and a desired character or figure can be displayed on the substrate 14. At this time, not only an upper end part of the cathode 20 but also a side circumferential surface of it contribute to discharge, and it is radiated sufficiently to the phosphor 32 as well, thereby extremely high brightness display can be provided.
Patent JP-H05274388-A (JP)
Title: Input pattern generation method for logic circuit simulation
IPC: G06F11/25
Filed: 1992-03-25
Abstract: PURPOSE:To generate an input pattern without erroneous input in a short time. CONSTITUTION:The input pattern generation method for logic circuit simulation generates or edits an input pattern to be inputted to the logic circuit simulator to be used for the inspection whether or not the designed logic circuit exhibits the required performance. A given input pattern is selected (S1 and S2) based on the stored input pattern, performing edition for the input pattern (S3 and S4). The edited input pattern is collated with the definition rule stored in advance, checking whether or not it is legal.
Patent JP-H05269976-A (JP)
Title: Method for detecting register mark on transparent web
IPC: B41F33/14
Filed: 1992-03-26
Abstract: PURPOSE:To make both of a register mark by visible ink and a register mark by transparent ink detectable in the case where a web is of a transparent one. CONSTITUTION:Shedding is made by light from a light source covering a range from ultraviolet light to visible light over a transparent web 3 that is conveyed, and watching is made by a sensor 2 on receiving of the light transmitted through the transparent web 3. Then, both of a register mark 4 printed with transparent ink and a register mark 4 printed with visible ink are detected through damping of light-receiving intensity in each of wavelength areas in distribution of the wavelength of the received light.
Patent JP-S60246229-A (JP)
Inventor: PIITAA BIRUKU
IPC: B26D1/08
Filed: 1985-05-14
Abstract: (57)【要約】本公報は電子出願前の出願データであるた め要約のデータは記録されません。
Patent JP-S5528023-A (JP)
Title: Production of covered lens
Inventor: MAEDA YUUJI
IPC: G02B1/10
Filed: 1978-08-18
Abstract: PURPOSE: To produce the covered lens surely with a simple constitution by forming undulations on the surface of the lens body and applying films.  
     CONSTITUTION: Raw liquid 2 is injected into molds 1 and is set after heating to mold a lens body 3. The burrs 4 of the circumferential edge portions thereof are ground away and the surfaces of the resultant lens body 5 are suitably polished, whereby flaws of 2 to 5 microns are formed on said surfaces, whereby the surfaces are roughened. Next, the lens body 5 is dipped in the solution of desired film forming material, after which it is dried, whereby films 6 are formed on the surfaces of the body 5. Hence, the films 6 are deposited by having undulations and will not peel from the body 5. 
     COPYRIGHT: (C)1980,JPO&Japio
Patent JP-S59227690-A (JP)
Inventor: ISHII SUEJI
IPC: B66C23/88
Filed: 1983-06-08
Abstract: (57)【要約】本公報は電子出願前の出願データであるた め要約のデータは記録されません。
Patent JP-S61258376-A (JP)
Title: Polishing device for magnetic head
Inventor: KITSUNAI TSUNEYUKI
IPC: G11B21/21
Filed: 1985-05-13
Abstract: PURPOSE:To attain a polishing process with high efficiency in a constant radius state of high accuracy by giving the radius polishing to the corner of contact face of a magnetic head against a magnetic recording medium with a contact secured to a lapping tape so that the coincidence is obtained between the direc tion of the head and the driving direction of the recording medium. CONSTITUTION:A lapping tape 3 is set between guide rolls 1 and 2 engaged with each other through their recess and projection parts. Thus the tape 3 is deformed into the shapes of both rolls 1 and 2. The recess/projection forms of rolls 1 and 2 is approximate or equal to the radius shape of the contact face of a magnetic head against a recording medium which requires the processing. Thus the apexes of the recess/projection parts of the polishing sur face of the deformed tape 3 have no contact with the part of the head requiring no processing. Then the magnetic head is fixed to a tool 5 and has a slight touch to the tape 3 so that the coincidence is secured between the head direction and the driving direction of the recording medium. Thus the head is polished in an radius shape. In this case, the polishing time is set by a timer. Then the tape 3 is moved up after polishing to secure a fixed radius state.
Patent JP-H06304296-A (JP)
Title: Slot machine
Inventor: NAKAZAWA HIROTO
IPC: A63F11/00
Filed: 1993-04-27
Abstract: PURPOSE:To obtain a slot machine which permits the easy handling such as in transport and storage, suppresses the generation of the rust which deteriorates the quality of products, and is protected from the influence of the static electric ity as the cause of the faulty operation, and can contribute to the protection of environment. CONSTITUTION:A case body for accommodating a mechanism part is made of plastics having electric conductivity, and is constituted of side plates 90, a top plate 100, a bottom plate 110, a back plate 120, and a front door 130.
Patent JP-S58216533-A (JP)
Inventor: FUJISAWA SHIYOUTAROU
IPC: B08B9/34
Filed: 1982-06-11
Abstract: (57)【要約】本公報は電子出願前の出願データであるた め要約のデータは記録されません。