baber/WOPTO huggingface dataset:
Patent HU-T62573-A (HU)
Title: Process for producing piperidine derivatives and pharmaceutical compositions comprising such compounds
Inventor: JEGHAM SAMIR
IPC: A61K31/445
Filed: 1992-04-02
Abstract: Compounds corresponding to the general formula (I) 
<IMAGE>
 in which 
 
  R<1> represents either a hydrogen atom, or a linear or branched (C1-6)alkyl group or a cyclo(C3-8)alkyl group, 
  X represents either an oxygen atom or a sulphur atom or a group of general formula N-R3 in which R3 is a hydrogen atom, a linear or branched (C1-8)alkyl group, a cyclo(C3-6)alkyl group, a cyclo(C3-6)alkylmethyl group, a (C1-4)alkoxy(C1-4)alkyl group, a phenyl group, a 4-pyridyl group or a 3-pyridyl group, 
  Z represents a hydrogen or fluorine atom as well as their addition salts with pharmaceutically acceptable acids. 
 
<??>Application in therapy.
Patent HU-T63055-A (HU)
Title: Process for producing pharmaceutical compositions for relieving diuria
Inventor: MORIOKA YUKO
IPC: C07D473/06
Filed: 1992-12-10
Abstract: Pharmaceutical compositions for the improvement of dysuria comprising a pharmaceutical carrier and a therapeutically effective amount of a xanthine derivative represented by the general formula I <CHEM> wherein R1 denotes a group of the formula R4-CO- or R5R6(OH)C-or a carboxyl group, wherein R4 and R5 independently denote an alkyl group having 1-3 carbon atoms, and R6 denotes a hydrogen atom or an alkyl group having 1-3 carbon atoms, R2 denotes a hydrogen atom, an alkyl group having 1-5 carbon atoms or an alkyloxy group having 1-5 carbon atoms, R3 denotes an alkyl group having 1-3 carbon atoms and n denotes 1-6 or a pharmaceutically acceptable acid addition salt thereof. They are active in prolonging urination intervals and increasing urination threshold pressure with almost no influence upon constrictive force of the bladder. Thus, they are effective in treatment and prevention of dysuria such as pollakiuria and incontinence of urine.
Patent HU-T71397-A (HU)
Title: Process for producing peptide derivates
Inventor: MATSUO MASAAKI
IPC: A61K38/06
Filed: 1993-04-09
Abstract: Disclosed herein are compounds of the following formula:   <IMAGE>   wherein R1 is a group of the formula   <IMAGE>   "X" is CH2 or N, "Z" is O, S, or N-R6, "A" is an amino acid residue, and Y, R2, R3, R4, R5, R6, and R7 are substituent variables as defined herein. The compounds are antagonists of tachykinin, and as such are useful for alleviation of pain and for treatment of disorders including asthma, bronchitis, rhinitis, conjunctivitis, dermatitis, arthritis, and urticaria.
Patent HU-T72086-A (HU)
Title: Dioxcyclobutene derivatives, pharmaceutical compositions containing them and process for their production
Inventor: BIRCH ALAN MARTIN
IPC: C11D7/26
Filed: 1993-07-03
Abstract: The invention provides compounds of formula (I), and pharmaceutically acceptable salts thereof; wherein R50 is hydrogen or C1-4 alkyl, A51 is oxygen, sulphur or a group of the formula -NR52- wherein R52 is hydrogen or C1-4 alkyl; A50 comprises (i) a mono or bicyclic aromatic ring optionally containing one or more nitrogen, oxygen or sulphur atoms, (ii) a cycloalkendiyl group, or (iii) an acyclic bridging group having a chain of one, two or three atoms between the cyclobutenedione group and X50, said chain being a chain of one or two carbon atoms or a chain of one carbon atom and one or more nitrogen, oxygen or sulphur atoms or (iv) a bond; X50 is either a bond or a spacer group providing a chain between A50 and B50 of one or two atoms length; B50 is a mono or bicyclic aromatic ring optionally containing one or more nitrogen, oxygen or sulphur atoms; r is an integer from 1 to 6; and Het is a ring system optionally containing one or more nitrogen, oxygen or sulphur atoms or is a phosphonate, phosphinate or amine derivate (wherein each of A50, X50, B50 and Het are optionally substituted). The compounds have angiotensin II antagonist activity and are useful in the treatment of cardiovascular disorders such as hypertension.
Patent HU-T70682-A (HU)
Title: Roof structure, cask-making machine for that roof structure and method for production of that cask-making machine
Inventor: JACOBSEN PER
IPC: E04D13/147
Filed: 1993-09-09
Abstract: PCT No. PCT/DK93/00289 Sec. 371 Date Feb. 10, 1995 Sec. 102(e) Date Feb. 10, 1995 PCT Filed Sep. 9, 1993 PCT Pub. No. WO94/08108 PCT Pub. Date Apr. 14, 1994For sealingly joining an underroof to a skylight or another roof installation a fitting collar is provided comprising a film element (7, 8) with a substantially U-shaped plane configuration with a cutout, at the sides of which there are flange parts (9, 10) for attachment of the fitting collar to mutually adjoined exterior sides (1-4) of the main frame structure of the window or the roof installation, in such manner that the film element is brought to extend substantially in parallel with the roof surface, in order to connect with adjacent parts (5, 6) of the underroof. The fitting collar can be manufactured in a simple manner, in that there in two overlapping lengths of film is produced transversal welds, at distances corresponding to a prescribed main frame width, whereby an obliquely extending part of each weld is formed with two parallel welded seams, while there in the edge zones at the opposite side edges of the lengths of film in extension of one and the other, respectively, of the two parallel welded seams are produced welded seams, which are perpendicular to the side edges. The collar elements are then separated by cutting along the cutting lines (22) between the parallel welded seams and parallel to the welded seams perpendicular to the side edges, and the collar is completed by cutting one length of film along the mid line between the welded seams with a subsequent bending upwards of the attachment flange parts.
Patent IL-43544-A (IL)
Title: 10(3-(4-(2-hydroxyethoxy)-4-alkyl)piperidino)-propyl-2-trifluoromethyl-phenothiazine derivatives,process for preparing them and pharmaceutical compositions containing them
IPC: C07D417/06
Filed: 1973-11-01
Abstract: 1393490 Phenothiazine derivatives ROUSSEL UCLAF 9 Nov 1973 [9Nov 1972] 52171/73 Addition to 1383773 Heading C2C Novel compounds of Formula I (in which R 1 = Me or Et and R 2 = decanoyloxy or, when R 1 = Me, 2-methylheptanoyloxy or hexadecanoyloxy) and physiologically acceptable acid addition salts thereof, and the novel maleic acid addition salt of the compound of Formula I wherein R 1 = Et and R 2 = OH, are prepared by reacting 10-(3-chloropropyl)-2- trifluoromethyl-phenothiazine with a piperidine derivative of Formula II to produce a compound of Formula III which is reacted, when R 3 = C 2 H 5 with decanoic acid chloride or maleic acid, or, when R 3 = CH 3 with decanoyl, 2-methylheptanoyl or hexadecanoyl chloride. The physiologically acceptable acid addition salts of compounds I are prepared by reacting the parent compound with an appropriate acid. Pharmaceutical compositions having neuroleptic activity, for oral or parenteral administration comprise one of the above novel compounds together with a pharmaceutical carrier.
[GB1393490A]
Patent IL-46802-A (IL)
Title: Method for preparing stable betalactam-type-antibiotic susceptibility test discs
IPC: C07G11/00
Filed: 1975-03-12
Abstract: Stable antibiotic susceptibility test discs are prepared by depositing crystals of a .beta.-lactam-type-antibiotic on said discs, said crystals being dispersed in a volatile unreactive non-solvent vehicle, such dispersion being contacted with such discs and the vehicle evaporated therefrom.[US3937655A]
Patent IL-61917-A (IL)
Title: Counterflow heat exchanger construction
IPC: F28D9/00
Filed: 1981-01-16
Abstract: In a counterflow heat exchanger a manifold is attached at two points to the ram and bleed closure bars. The bleed closure bar defines a bleed inlet from the manifold and is constructed to reduce the mechanical stresses in the ram closure bar between those attachment points.
Patent IL-82943-A (IL)
Title: Total esters of alginic acid with alcohols, their preparation and pharmaceutical and cosmetic compositions containing them
IPC: A23L29/00
Filed: 1987-06-22
Abstract: The present invention relates to total and partial esters of alginic acid with alcohols of the aliphatic, araliphatic, cycloaliphatic, aliphatic-cycloaliphatic and heterocyclic radicals, and salts of said partial esters with inorganic and organic bases. The said partial ester are not a partial ester of bivalent aliphatic alcohols. These compounds are intended to be used in pharmaceutical. applications.
[EP0251905A2]
Patent IL-87884-A (IL)
Title: Catalyst and process for olefin polymerization
IPC: C08F4/64
Filed: 1988-09-29
Abstract: A catalyst for olefin polymerization which comprises:   (A) a catalyst component obtained by reacting (a) pentadiene or a derivative thereof with (b) an alkali metal and subsequently reacting the reaction product with (c) a titanium compound or zirconium compound, and   (B) aluminoxane. t
Patent IL-88208-A (IL)
Title: Pharmaceutical compositions containing acyl-substituted uridines and cytidines and some novel compounds of this type
IPC: A61P9/10
Filed: 1988-10-28
Abstract: General methods for delivering exogenous cytidine or uridine to the tissue of an animal comprising the administration of acylated cytidine or acylated uridine, respectively, are disclosed. Methods of treating myocardial infarction and cardiac insufficiency comprising the administration of acylated cytidine or acylated uridine, are also disclosed.
Patent IL-89124-A (IL)
Title: Composition for reducing immunoglobulin e response comprising an antagonist to human interleukin - 4
IPC: C12P21/00
Filed: 1989-01-31
Abstract: A method of reducing immunoglobulin E responses associated with certain immune disorders is provided. The method comprises administering an effective amount of an antagonist to human interleukin-4. Preferably the antagonist is a blocking monoclonal antibody specific for human interleukin-4, or a fragment or binding composition derived therefrom.
Patent IL-95507-A (IL)
Title: Fluid dispensing devices
IPC: B65D81/32
Filed: 1990-08-28
Abstract: A method is described for producing a dispenser including a plastic body which defines two vertically spaced compartments (2, 3) connected by an orifice closable by a plug valve (6) which co-operates with a seating (5) set in the internal periphery of the orifice to provide a seal between the two compartments (2, 3). The body section (2) which defines the upper of the two compartments is of tubular construction and the body section (3) which defines the lower of the two compartments is capable of flexing movement towards and away from the mid section of the body in which the orifice between the two compartments (2, 3) is defined. The method includes the steps of producing by an injection moulding technique a semi-finished product comprising the upper and mid body sections and a parison dependent from the mid body section, and subsequently blow moulding the parison to produce the lower compartment of the dispenser.
Patent JP-H01308517-A (JP)
Title: Cable take-up device for dust suction machine
Inventor: RORUFUUYURUGEN KUREEMERU
IPC: A47L9/26
Filed: 1989-01-20
Abstract: PURPOSE: To pull a cable without applying and removing a load to a braking device by separating a sidewall of a cable winding frame from the remainder of the frame and connecting the frame to an attachable winding frame via a one-directional clutch. CONSTITUTION: A sidewall 3 is supported by a braking machine 20 and moves to A direction together with a winding frame bottom 2 in the case of taking out a cable 22. An axis 5 rotates similarly to the direction and a part 7 of the one-directional clutch rotates freely. In the case of taking out the cable, however, a recovery spring 21 on a sidewall 4 is simultaneously pulled and rotates the cable oppositely in E direction if tensile strength on the cable 22 is decreased. Thereby, the axis 5 also rotates oppositely but prevented from doing so by means of the part 7 of the one-directional clutch together with the sidewall 4 and the winding frame bottom 2. Once the braking machine 20 being relaxed, both sidewalls of the cable winding frame 1 can be returned to E direction and thus centrifugal braking weights 11 and 12 can be in operation.
Patent JP-S55102935-A (JP)
Title: System and device for amplitude equalization
Inventor: NAMIKI JIYUNJI
IPC: H04B3/14
Filed: 1979-01-31
Abstract: PURPOSE:To equalize the amplitude of an amplitude-distorted input signal accurately and rapidly by exercising control over an increase and decrease in center frequency according to a difference in level value between a 2nd-level interpolation, interpolated from a gradient obtained from a 1st level and 3rd level, and actual value. CONSTITUTION:Signal detector 1090 detects levels P1, P2 and P3 of outputs of band-pass filters provided at three points in a transmission band after the output of a variable resonance circuit whose center frequency omega0 and frequency selectivity Q0 are variable. Then, control (1097) over an increase and decrease in frequency omega0 is exercised according to a difference between actual level P2 and the interpolation value of level P2 interpolated from a gradient found from levels P1 and P3, so that the amplitude of an input signal influenced by amplitude distortion close to reverse characteristics of circuit 1090 can be equalized by variable resonance circuit 1090.
Patent JP-S55102960-A (JP)
Title: Signal transmission system
Inventor: SANAGI MUTSUTAKE
IPC: H04L27/26
Filed: 1979-01-31
Abstract: PURPOSE: To exercise a supervision over a transmission line by the output of the detection of a specific signal, obtained by combining several frequencies, by a reception office when no information input arrives at the terminal of a transmission office.  
     CONSTITUTION: Corresponding to information inputs 2∼2''' from transmission office 1, a signal obtained by combining specific frequencies among several frequencies is transmitted to reception office 7 via transmission line 6, and reception office 7 extracts information outputs corresponding to information inputs. Between information inputs 2∼2''' of transmission office 1, and coding part 3, AND circuit 15 is connected and when none of information inputs 2∼2''' arrives, an output is generated by circuit 15 and coded by coding part 3, and frequencies of oscillation parts 4∼4''' are combined and sent to reception office 7. Those combined frequencies are applied to detection circuits 9∼9''' via band-pass filters 8∼8''' of  reception office 7 and when a specific frequency is detected, decoding part 10 outputs information outputs 11∼11''' and transmission-line supervisory output 18 is  sent out from OR circuit 17. 
     COPYRIGHT: (C)1980,JPO&Japio
Patent JP-S62168677-A (JP)
Title: Welding start point detecting device in weld line copying device
Inventor: KUGA MINORU
IPC: B23K9/12
Filed: 1986-01-22
Abstract: PURPOSE:To improve the detection accuracy by fixing a slit light source and an observation use optical system together with a welding torch, and also, making a point where each center axis of the slit light source and the observation use optical system crosses coincide, etc. with a welding target point of the welding torch. CONSTITUTION:A slit light source 6 and an observation use optical system 10 of a semiconductor laser, etc. are fixed together with a welding torch 2, to fixing jig 4 which has been provided on a wrist 3 of a robot. In this case, a point where the center axis of the light source 6 and the center axis of the optical axis cross is made to coincide with a welding target point of the welding torch 2. Also, a plane which is formed by a slit light beam 5 and each center axis of the optical system 10 is constituted so as to make a prescribed angle against the center axis of the torch 2. According to this method, since a detecting optical system 1 is fixed together with the torch 2, even in case an object to be measured 11 and the torch 2 approach each other, the detection can be executed, and the accuracy for detecting a welding start point is improved.
Patent JP-S63180414-A (JP)
Title: Electric discharge machining source device
Inventor: FUTAMURA SHOJI
IPC: B23H1/02
Filed: 1987-01-20
Abstract: PURPOSE:To prevent the occurrence of unevenness in a machined surface and consumption of an electrode during machine on an electrode consumption condition, by a method wherein a current control means is situated, a current peak value during restarting of electric discharge after elapse of a stop period of electric discharge machining is decreased over a normal value, and the current peak value is gradually restored to the normal value. CONSTITUTION:The phase of a control rectifying circuit 9, being a current control means, is controlled by means of a signal from a phase control circuit 10. Namely, a signal for rising and lowering of an electrode is provided from a terminal 12. When an electrode is raised, phase control is effected so that the output voltage of the control circuit 9 is slightly decreased, and the output voltage is so decreased that a current peak value prevailing when discharge is restarted at a decreased voltage is decreased over a set normal value. Thereafter, when, through monitoring of a voltage applied between an electrode 6 and a workpiece 7, it is detected by a machining starting detecting circuit 11 for detecting the starting of electric discharge machining that electric discharge machining is restarted, the phase of the control circuit 9 is controlled by a phase control circuit 10 so that a peak value is gradually restored to a normal value according to a given function.
Patent JP-S56107692-A (JP)
Title: Monitoring control unit
Inventor: YAMADA SHINKICHI
IPC: H04Q9/00
Filed: 1980-01-31
Abstract: PURPOSE:To simplify an interface by executing remote monitorial control of straight forward system of an currnt reverse system, and shunning an erroneous signal of the control output from a controlling computer by means of software. CONSTITUTION:By the output point selective program 1-2 of an apparatus to be contolled, the output point of this apparatus is encoded, and it is output to the selective matrix 2. A control output command of on or off is output to the control master output program 1-2 by the control program 1-1, and the control master output program 1-2 outputs a common command of on or off as a pulse output to the master station 3-1. And, a state or a fault of apparatus to be controlled, which has been detected is changed to a group by the address circuit 6, and it is input to the controlling computer 1. On the other hand, the fault or state input is loaded in advance by the state input processing program 1-4, and the state input table of the point where the fault has occurred is turned off unconditionally.
Patent JP-H06218383-A (JP)
Title: Ozone injection method
Inventor: ISHIDA KOJI
IPC: C02F1/78
Filed: 1993-01-26
Abstract: PURPOSE:To limit the consumption of ozone as a whole and efficiently decompose organic matters by setting injection rates of ozone corresponding to the properties of water to be treated in a reaction region and injecting ozone gas in a multistage manner so that the total amount of absorbed ozone exceeds the total amount of consumed ozone. CONSTITUTION:By actuating a flow control valve 5, the injection rate of ozone in each reaction region 1b is controlled so as to maintain a specific ozone absorption efficiencies of suitable value corresponding to the property of water to be treated in respective reaction region, whereby a best ozone injection method is achieved when an attempt is made to decrease the initial concentration of organic matter in water to be treated to a specified value. And ozone injection rates are not increased by one-stage process but by a method wherein ozone is divided and injected in a multistage manner to increase the ozone injection rates as a whole. That is, since three-stage treatment is better than one-stage treatment and six-stage is better than three-stage, ozone is injected in such a manner that ozone injection rate per one tank satisfies conditions of ozone absorption efficiency, thereby efficiently effecting removal of organic matters.
Patent JP-S60153883-A (JP)
Inventor: TSUCHIKURA MITSURU
IPC: A63B43/00
Filed: 1984-01-23
Abstract: (57)【要約】本公報は電子出願前の出願データであるた め要約のデータは記録されません。
Patent JP-S56107507-A (JP)
Title: Transformer
Inventor: SATOU TATSUO
IPC: H01F27/33
Filed: 1980-01-29
Abstract: PURPOSE:To make incombustible, miniaturize and lighten a transformer by a method wherein an insulating gas is enclosed into a tank and a cooler, and the insulating gas is circulated by means of a blower. CONSTITUTION:A tank 8 and a cooler 9 are communicated by means of pipings 10a, 10b, and an insulating gas is enclosed into the tank 8 and the cooler 9. Heat generated in the tank 1 is transmitted to the insulating gas, forwarded to the cooler 9 by means of a blower 11 and thermally radiated into air.
Patent JP-S61170621-A (JP)
Title: Method for measuring coefficient of cubical expansion of hydrogen occluding alloy
Inventor: NASAKO KENJI
IPC: G01N7/00
Filed: 1985-01-25
Abstract: PURPOSE:To make easily and economically the measurement to determine the coefft. of cubical expansion of a hydrogen occluding alloy in the stage of releasing hydrogen and in the stage of occluding hydrogen by incorporating an inert gas into a system including hydrogen and the hydrogen occluding alloy and measuring the fluctuation of the internal pressure of the inert gas. CONSTITUTION:The volume of respective piping parts A-C is first measured while the hydrogen occluding alloy 2 is not packed into a thermostatic chamber 1. The alloy 2 is then packed into a container 3 and the inert gas is introduced into the piping parts A, C from an inert gas cylinder 12 and the pressure change of the parts A, C is measured, by which the volume of the part A is determined. The gas in the system is then discharged by a vacuum pump 7 and thereafter the hydrogen is introduced into the parts A, B from a gaseous hydrogen cylinder 11 so that the hydrogen is occluded into the alloy 2. The inert gas is thereafter discharged from the part C to the part A and the pressures in the parts A, C are measured. The volume of the part A in the stage of occluding the hydrogen is measured. The coefft. of cubical expansion of the alloy is calculated from the results of the above-mentioned measurement.
Patent JP-S55104402-A (JP)
Title: Sliding material
Inventor: FUTAMURA KENICHIROU
IPC: C22C38/00
Filed: 1979-01-31
Abstract: PURPOSE: To improve the hardness, wear resistance and impact resistance of the sliding material obtained, by spreading powder mixture of Mo, B and Fe metal for the rest at specified ratio thinly on the backing metal of Fe base alloy, and baking.  
     CONSTITUTION: Powder mixture is prepared in paste form by containing, by wt%, Mo; 30W10%, B; 8W30%, and, if necessary, Pb; ≤10%, and one or both of P; ≤10% and P; 8%, and Fe metal group for the rest. For example, by using mixture solution of starch glue carbonized by baking or resin base adhesive, and water or alcohol, a paste form is obtained, which is spread on the backing metal consisting of Fe base alloy to a thickness of less than 0.3mm to form a sliding adhesive layer. By baking this layer, the sliding adhesive layer and backing metal is formed into an integral body. By adding Pb and P, the surface performance such as sliding property and false adhesion resistance may be improved. 
     COPYRIGHT: (C)1980,JPO&Japio