baber/WOPTO huggingface dataset:
Patent HU-T43063-A (HU)
Title: Process for preparing imidazo/1,2-a/quinoline derivatives and pharmaceutical compositions containing such compounds
Inventor: GEORGE PASCAL
IPC: C07D471/04
Filed: 1987-01-21
Abstract: 1. Claims for the Contracting States : BE, CH, DE, FR, GB, IT, LI, LU, NL, SE Imidazo[1,2-_a]quinoline derivatives corresponding to the formula (I)  see diagramm : EP0233800,P14,F1  in which X denotes hydrogen, a halogen or a (C1-4 )alkyl, (C1-4 )-alkoxy, (C1-4 )alkylthio, methylsulphonyl, amino, (C1-4 )-alkylamino, di(C1-4 )alkylamino, nitro or trifluoroalkyl group, Y denotes hydrogen, a halogen or a methyl group at position 6, 7 or 8, and R1 and R2, taken separately, each denote hydrogen or a (C1-6 )alkyl group, or alternatively R1 and R2 together form a tetramethylene, pentamethylene, 3-methyl-3-azapentamethylene or 3-oxapentamethylene chain, as well as their addition salts which are acceptable in pharmacology. 1. Claims for the Contracting States : AT, ES, GR Process for the preparation of imidazo[1,2-_a]quinoline derivatives corresponding to the formula (I)  see diagramm : EP0233800,P16,F1  in which X denotes hydrogen, a halogen or a (C1-4 )alkyl, (C1-4 )-alkoxy, (C1-4 )alkylthio, methylsulphonyl, amino, (C1-4 )-alkylamino, di(C1-4 )alkylamino, nitro or trifluoroalkyl group, Y denotes hydrogen, a halogen or a methyl group at position 6, 7 or 8, and R1 and R2, taken separately, each denote hydrogen or a (C1-6 )alkyl group, or alternatively R1 and R2 together form a tetramethylene, pentamethylene, 3-methyl-3-azapentamethylene or 3-oxapentamethylene chain, which process is characterized in that the quinoline of formula (II)  see diagramm : EP0233800,P16,F2  is first subjected to the action of an alpha-bromoacetophenone bearing the substituent X defined above, in the heated state in a solvent such as methylene chloride or 1,2-dichloroethane ; an ionic compound of formula (III)  see diagramm : EP0233800,P16,F3  is obtained, which is cyclized in the presence of ammonium acetate, in an acidic organic solvent such as acetic or propionic acid, at a temperature of 90 degrees C, to obtain the compound of formula (IV)  see diagramm : EP0233800,P16,F4  the compound obtained (IV) is reacted with glyoxylic acid in a solvent such as acetic acid at 80 degrees C ; the alpha-hydroxy acid obtained (V)  see diagramm : EP0233800,P17,F1  is acetylated using acetic anhydride in the presence of pyridine, and then converted to the alpha-acetoxyacetamide  see diagramm : EP0233800,P17,F2  via the imidazolide, which is prepared in situ ; the compound (VI) is deacetylated to the alpha-hydroxyacetamide (VII) see diagramm : EP0233800,P17,F3  by treatment with potassium carbonate in ethanol ; the compound (VII) is reacted with sulphonyl chloride SOCl2 in a chlorinated solvent such as dichloromethane, to obtain the chlorinated compound (VIII)  see diagramm : EP0233800,P17,F4  which is reduced using Rongalite**(r) in methylene chloride to the compound (I).
Patent HU-T34452-A (HU)
Title: Process for producing piperonyl-butoxide
Inventor: REEPAASY OTTO
IPC: C07D317/54
Filed: 1983-02-04
Abstract: Piperonyl-butoxide is prepd. by first hydrogenating and chloromethylating safrol contg. etheric oils to obtain chloromethyl-dihydro-safrol. This is further reacted with diethylene-glycol-monobutyl-ether at 100-120 deg.C in the presence of alkali and/or alkaline earth metal hydroxides and/or oxides in an inert solvent forming an azeotrope with water, pref. benzene and/or toluene and/or xylene in water free or aq. soln., or directly without solvents in water free conditions in the presence of alkali or alkaline earth metal carbonates, observing a mole ratio chloromethyl-dihydro-safrol: diethylene-glycol-monobutyl-ether: alkali of 1: (1.5-2.1): (1.3-2.0). - The raw prod. is freed from salts by filtration and/or washinq, the solvent is taken off by distn. at atmos. pressure or in a slight vacuum, and part of the diethylene-glycol-monobutyl-ether is eliminated.
Patent HU-T39408-A (HU)
Title: Method for processing blast furnace and converter slags into phosphorous fertilizer
Inventor: PENTEK ISTVAN
IPC: C05B13/00
Filed: 1985-02-15
Abstract: The latent heat of the molten slag and phosphorus mineral from the convertor are utilised in production of an alkaline fertiliser comprising also Zn, Cu, Co, Fe and Mn. The solubility of citrates in 20 wt. % P2O5 fertiliser is above 90% w/w and in a 36-40 wt. % CaO+MgO it is 60-70 wt. %.
Patent JP-S5283931-A (JP)
Title: Antigen of catechol amine derivatives
Inventor: YOSHIOKA MASANORI
IPC: G01N33/53
Filed: 1976-01-01
Abstract: PURPOSE: An antigen containing catechol amine as hapten which can produce antibody having high specificity, by reacting the benzene ring the catechol amine protein carrier by Mannig reaction. 
     COPYRIGHT: (C)1977,JPO&Japio
Patent JP-H06247351-A (JP)
Title: Truck bushing
Inventor: KENISU AARU WATSUTSU
IPC: F16C11/02
Filed: 1994-01-06
Abstract: PURPOSE: To raise strength and elongate life of a track bush by forming an outer peripheral surface and an inner central portion of the track bush so that Rockwell hardness thereof, respectively, shows a specific value. CONSTITUTION: A track bush 10 which is used for the endless track of a work vehicle, such as an endless track tractor or the like, has a cylindrical form in its entirety and comprises an outer peripheral surface 12 extending substantially the entire length, a pair of radial end surfaces 14, 16 and a longitudinal bore 18. As far as first and second end portions 24, 26 having comparatively small radiuses and the central portion 28 of the bush 10 are concerned, Rockwell hardness C of the outer peripheral surface of the bush 10 is set to about 57-62, and the Rockwell hardness C of the inner peripheral surfaces of the first and the second end portions 24, 26 is set to about 57-62, and the Rockwell hardness C of the inner central portion 28 is set to about 15-50. The central portion 28 is formed so as to occupy approximately 50% of an entire length L of the bush 10.
Patent JP-H07197699-A (JP)
Title: Fence
Inventor: KIMURA TETSUYA
IPC: E04H17/16
Filed: 1994-01-07
Abstract: PURPOSE:To improve the appearance of a fence by burying buried nuts to both side end faces of a concrete board disposed between a pair of struts, screwing adjusting nuts and the buried nuts to bolts penetrated to the struts and covering the struts with covers. CONSTITUTION:A concrete board 2 is arranged between a pair of oppositely faced struts 1, 1, and adjusting nuts 5 are screwed to bolts 6 passed into bolt inserting holes and penetrated to the struts 1 while the front end sections of the bolts 6 are screwed to buried nuts 4 buried to the concrete board 2. The operation is conducted similarly at both side edge sections of the concrete board 2, and the bolts 6 and the adjusting nuts 5 are operated and adjusted so that clearances D among the concrete board 2 and the struts 1 are equalized at both sides. The operation is performed repeatedly, and the concrete boards 2 are stacked successively from lower stages. Lastly, covers 11 with tongue pieces 12 inserted to sections, from which the bolts 6 and the adjusting nuts 5 are removed, in the clearances D are inserted from the upper ends of the struts 1, thus completing a fence.
Patent JP-S63170070-A (JP)
Title: Recorder
Inventor: ASANO SHINYA
IPC: B41J29/36
Filed: 1987-01-07
Abstract: PURPOSE:To save consumption of ink ribbon, when making a correcting operation with a correction ribbon being placed between a recording medium and the ink ribbon, by controlling the feeding quantity of ink ribbon variably based on specific conditions. CONSTITUTION:Upon provision of a correction command, CPU16 reads out a feeding quantity data N corresponding to the width of type of a character to be corrected from a correcting time ink ribbon feeding quantity data memory 18 in ROM17, and sotres said data N in a correcting time ink ribbon feed counter 20. Upon finish of correction of character, a step motor 24 for feeding an ink ribbon is rotated. The ink ribbon feeding quantity data N stored in said counter 20 is employed for said rotation control, and the content of counter is subtracted one by one every time when the step motor rotates by single step, and the rotation is stopped when the content goes to 0, thus finishing correction. When correction is made, the ink ribbon is fed by a predetermined width corresponding to the width of type, thereby it can be utilized effectively within minimum feeding quantity range without causing breaking nor cutting.
Patent JP-H04242740-A (JP)
Title: Powder coating device
Inventor: HONMA YOSHIYASU
IPC: G03D13/00
Filed: 1991-01-08
Abstract: PURPOSE:To uniformly apply a developer to a support body by driving a carrier and a feeding body after applying an electric field at the time of applying a powder onto the support body, stopping the carrier and feeding body at the time of finishing the application, and then stopping the electric field. CONSTITUTION:The moment when a general paper P comes in a transfer area 27 is judged by a sensor, a developer carrying roller 22 and a feed roller 21 are driven, and a developer S is stirred, adhered onto the developer carrying roller 22 and transferred to the transfer area 27. An electric field suitable to the polarity of the electrified developer S is preliminarily added to an electrode roller 23 by a power source 26, whereby the developer S electrified by the electrostatic power is flown from the developer carrying roller 22 to the general paper P. The moment when the general paper P gets out of the transfer area 27 is judged by the sensor, and the developer carrying roller 22 and the feed roller 21 are turned off. Thereafter, the power source 26 is turned off, and the electrode roller 23 is turned off after the general paper P gets out of an output port 28.
Patent JP-S63171658-A (JP)
Title: Rotary atomizing head for electrostatic painting
Inventor: HAYASHI NOBUYUKI
IPC: B05B5/04
Filed: 1987-01-06
Abstract: PURPOSE:To atomize a paint for electrostatic painting in the form of fine particles having uniform sizes, by inclining the side walls on the rear side of guide grooves in the rotating direction thereof more steeply than the inclination of the side walls on the front side of the rotating direction. CONSTITUTION:A rotary atomizing head 7 is connected to a high-voltage generator to form an electrostatic field between side head and a material to be coated. The rotary atomizing head 7 is rotated at a high speed. The liquid paint dropped from a paint supplying pipe 14 into an inside chamber 4 is supplied from a supply port 5 by centrifugal force to the inside peripheral face of the rotary atomizing head 7 from which the paint spreads in the form of a thin film and arrives at a steeply inclined part 10. The centrifugal force in said part is increased and accelerated by which the paint is finely divided in flow along the many guide grooves 12 and is released as fine liquid yarn from the apertures of the respective guide grooves 12. The released liquid is pulverized by the centrifugal force and electrostatic effect and is deposited on the material to be coated. The side walls 12a of the rear side of the respective guide grooves 12 in the rotating direction thereof are more steeply inclined than the inclination of the side walls 12b on the rear side of the rotating direction in this constitution. The flow of the paint over the side walls 12a is prevented when the paint divided in flow in the respective guide grooves 12 is pressed to the side walls by the centrifugal force. The release of the paint from a front end edge 11 in the state of the thin film is thus averted.
Patent JP-H09190798-A (JP)
Title: Charged particle measuring method
Inventor: MAEDA FUMIHIKO
IPC: H01J49/44
Filed: 1996-01-08
Abstract: PROBLEM TO BE SOLVED: To shorten the measurement time and make high speed measurement possible by taking in charged particles in the specified energy range at a time without scanning the blocking potential of an analyzer when the charged particle is detected by the separation of energy. SOLUTION: Photo-electron spectrum measurement is performed by using a photo-electron analyzer having a hemispherical electron energy analyzers 4, 5, an electric field correction electrode 1 arranged on the output side of the analyzers 4, 5, and a detecting part comprising an MCP(multi-channel plate) of 128 channels, and a position sensitive detector 3. The blocking potential of an electrostatic lens 6 is set, then the potential is applied to the analyzers 4, 5, and the energy of an electron passing through the analyzers 4, 5 is set. The electrons passed through the analyzers 4, 5 by the set gate time of the detector 3 are measured. The kinetic energy of the photo-electrons is calculated, and data obtained is converted into energy.
Patent JP-H11264093-A (JP)
Title: Production of zinc oxide film, production of photovoltaic element and production of semiconductor device substrate
Inventor: NISHIO YUTAKA
IPC: C25D9/04
Filed: 1999-01-06
Abstract: PROBLEM TO BE SOLVED: To produce at low cost a solar cell high in efficiency by forming in a short time and stably a zinc oxide film having an excellent optical confinement effect and using the film as the photovoltaic element. SOLUTION: In the production method of the zinc oxide film forming the zinc oxide film on the conductive substrate 103 by energizing between a conductive substrate 103 immersed in an electrodeposition bath 104 and a counter electrode 105 immersed in the electrodeposition bath 104, the temp. of the electrodeposition bath is kept at >=50 deg.C, and a temp. profile in which the temp. of the electrodeposition bath at a final stage of the electrodeposition is lower than that at an initial stage is given.
Patent JP-S62158935-A (JP)
Title: Operation frequency control device for air-conditioning machine
Inventor: NISHIHARA YOSHIKAZU
IPC: F24F11/02
Filed: 1986-01-07
Abstract: PURPOSE:To reduce the change of indoor temperature as well as vibration and noise due to the fluctuation of operation frequency by a method wherein the maximum operation frequency of a compressor is reduced stepwisely in accordance with the rise of an atmospheric temperature when the amount of indoor airflow is changed. CONSTITUTION:The operation frequency control device of a compressor for an air-conditioning machine is provided with an indoor airflow amount setting means A, changing the amount of indoor airflow, and a means B for detecting an atmospheric temperature. After starting the operation of the compressor, a set temperature 1 or another set temperature 2 is selected and the set temperature is compared with a signal from the atmospheric temperature detecting means A by a comparing means C. The output signal from the comparing means C is outputted at every predetermined times to change the maximum frequency (f1)-(f3) of the compressor stepwisely so that the compared temperature T is within a predetermined set temperature range T1'-T3. According to this method,the fluctuation of the operation frequency may be reduced and vibration or noise may be restrained.
Patent JP-S57113453-A (JP)
Title: Cassette holding mechanism of cassette deck
Inventor: TAKEMASA KAORU
IPC: G11B15/675
Filed: 1981-01-07
Abstract: PURPOSE:To reduce size and thickness by providing an auxiliary member which touches the main surface of a cassette half at one point in addition to a couple of members which sandwich the cassette half, and by positioning the cassette half in parallel to reel shafts while sandwiching the cassette half by those interlocking members. CONSTITUTION:A cassette half 15, when inserted, is supported by a cassette supporting plate 19 and an auxiliary arm 20 and also held by a cassette holder 16 from above. The cassette supporting plate 19 is rotatably freely around a fulcrum 19c to and from an underframe, and engages with the read end of a rotary arm 11 through a life-up arm 21, fitted rotatably to a back frame, to be held at a position shown in a figure. When the cassette frame 15 is lowered, the cassette holder 16 and cassette supporting plate 19 couple with the rotary arm 11 to turn while sandwiching the cassette half 15, and thus lowers the cassette half 15 to equip it to reel units 18a and 18b. Further, the auxiliary arm 20 secures the supporting the cassette half 15 more.
Patent JP-2000200895-A (JP)
Title: Method for designing light shielding layer pattern in photosemiconductor integrated circuit
Inventor: MICHINAKA SEIJI
IPC: H01L27/14
Filed: 1999-01-06
Abstract: PROBLEM TO BE SOLVED: To obtain a light shielding layer pattern having an appropriate opening space in a short time by converting a pattern data of light shielding layer determined through geometrical operation into an arbitrary layer and verifying it while superposing on a preset layout of a photosemiconductor integrated circuit. SOLUTION: A light shielding layer 14 is formed using a CAD system by forming the layout data of a photosemiconductor integrated circuit. 10 provided with no light shielding layer 14 and then processing the layout data geometrically using a CAD tool for verifying the layout. A verification is made whether there is no special problem as a photosemiconductor integrated circuit. 10 and in the fabrication process or not and if there is no problem, that layout data is outputted as a design layout data to a file. Pattern of the light shielding layer 14 is then designed to expose the parts of the photosemiconductor integrated circuit. 10 other than the photodiode part 15 and the capacitor part 11 are exposed from an opening space.
Patent JP-S55106601-A (JP)
Title: Manufacture of slab for thick steel plate by continuous casting
Inventor: OKADO TSUYOSHI
IPC: B21B1/46
Filed: 1979-01-11
Abstract: PURPOSE:To increase the rolling pressure for the middle part of the material, and to improve the effect of pressure welding for the porosity, by giving material the strong reduction with the stepped rolls and flat rolls, while the bloomed slab still keeping a temperature difference between its surface and central zone. CONSTITUTION:While the continuously cast and bloomed slab still keeps a temperature difference between its surface and central zone, a strong reduction is given by the stepped rolls 1 to the middle part A of the material 2. Hereby, the compression stress acting in the longitudinal direction of the sheet generates at the part A, and the tensile stress generates at the part B being left free from above reduction, and the compression stress of the part A increases. Next, the material 2 is rolled by the flat rolls 3, and the part B receives reduction under the compression stress acting in the longitudinal direction of the sheet, and a high rolling force can be obtained. According to this method, the porosity at the central zone of the slab is effectively pressure welded, and the cast structure is efficiently forged; as a result, the manufacturing limit for the sound, high equality thick steel plate is widened.
Patent MA-43354-A (MA)
Title: Conjugués médicamenteux à pont disulfure encombré
Inventor: CHEN JINHUA
IPC: A61P35/00
Abstract: L'invention concerne généralement des conjugués de médicament disulfure dans lesquels un lieur comprenant un atome de carbone soufré substitué par au moins un hydrocarbyle ou hydrocarbyle substitué est conjugué par une liaison disulfure à un atome de soufre de cystéine d'un support de ciblage et dans lequel le lieur est en outre conjugué à un fragment de médicament. L 'invention concerne en outre des conjugués activés de médicament lieur pouvant être conjugués à un porteur de ciblage par une liaison disulfure. L'invention concerne en outre des procédés de préparation de conjugués de médicament à base de disulfure encombré.
Patent ME-00591-A (ME)
Inventor: WIEGAND STANLEY J
IPC: A61K39/39
Filed: 2007-08-07
Abstract: Terapijski postupak za liječenje ishemijskih ili vaskularnih poremećaja primjenjivanjem sredstva koje može inhibisati akti vnost humanog delta-sličnog liganda 4 (DII4) subjektu kome je to neophodno. Poželjno, sredstvo je anti - DII4 anti ti jelo ili fragment anti ti jela koji mogu inhibisati vezivanje DII4 za Notch receptor. U jednom ostvarenju, ishemijski ili vaskularni poremećaj je: ishemijska povreda, cerebralna ishemija, srčana ishemija, ishemijska stanja koja se javljaju u udovima i drugim organima ili tkivima, arteriovenska malformacije, zarastanje rana, transplatacija organa ili tkiva, insufi cijencija placente, arterijalno sužavanje i okluzija, arteroskleroze i sistematska ili plućna hipertenzija. U drugom ostvarenju, liječena bolest je bolest oka ili stanje kao što je: reti nopati ja kod preranog rođenja, ishemijska reti nopati ja, okluzija vene ili arterije mrežnjače, reti nopati ja posledica dijabeta, horoidna neovaskularizacija, makularna degeneracija povezana sa starenjem, neovaskularizacija rožnjače, neovaskularni glaukom i transplatacija rožnjače.
Patent ME-P7609-A (ME)
Inventor: TAKEUCHI KOJI
IPC: A61K31/4439
Filed: 2006-12-27
Abstract: Ovaj pronalazak se odnosi na agnes za zašti tu pankreasa koji sadrži kombinaciju lijeka koji snižava glukoyu krvi, a ne sti muliše izlučivanje insulina, i jedinjenja predstavljenog formulom (II), gdje je svaki simbol defi nisan u opisu, ili njegove soli, u jedinjenja predstavljenog formulom (II), gdje je svaki sinbol defi nisan u opisu, ili njegove soli.
Patent OA-07257-A (OA)
Inventor: BRIET PHILIPPE
IPC: A61K31/38
Filed: 1982-11-25
Abstract: The invention concerns [oxo-4-4H-[1]-benzopyran-8-yl]-alcanoic acids and their derivatives, their manufacture, represented by the formula. <IMAGE>   where AR is hydrogen, a phenyl radical which may or may not be substituted thenyl, furyl, naphthyl, a lower alkyl, cycloalkyl, aralkyl radical; B is a linear or branched lower alkyl radical, either saturated or ethylinically unsaturated; R1 is hydrogen or a phenyl radical; X is hydrogen or a lower alkyl or alkoxy radical and n=1, as well as salts, esters, aminoesters and amides. Compounds and their derivatives may be used as medicines, in particular in the control of tumors.
Patent PH-30442-A (PH)
Title: Process for the enzymatic preparation ofgrf (1-44)nh2
Inventor: FELIX ARTHUR MARTIN
IPC: C07K14/00
Filed: 1991-12-09
Abstract: GRF(1-44)-NH2 is prepared by the trypsin catalyzed enzymatic coupling of Leu-NH2 to GRF(1-43)-OH. The latter compound may be obtained by recombinant DNA synthesis. Thus the present method provides an economical way to obtain the clinically important GRF(1-44)-NH2.
Patent PH-29957-A (PH)
Title: Use of tyloxapol as a nano-particle stabilizer and dispersant
Inventor: JUNE SIEGFRIED K
IPC: A61K47/00
Filed: 1993-09-24
Abstract: A composition comprising nanoparticles having tyloxapol adsorbed on the surface thereof, preferably containing a diagnostic or therapeutic agent, and most preferably including a further surface modifier associated therewith is described. A method of making such nanoparticles and a method of diagnosis comprising administering to a mammal of a contrast effective amount of particles of nanoparticles having tyloxapol adsorbed on the surface thereof is also described.
Patent PH-31459-A (PH)
Title: Absorbent article having elasticized side flaps and wings.
Inventor: YASUKO MORITA
IPC: A61F13/514
Filed: 1993-11-26
Abstract: An absorbent article having a liquid permeable topsheet, a liquid impermeable backsheet and a liquid absorbent pad for absorbing a liquid exuded from the human body positioned there between, and having an elasticized side flap and an extended wing along each side edge of the absorbent article. The side flap has a loop member formed from either the topsheet or the backsheet, or an optional secondary non-woven sheet, which extends from and loops back toward said side edge of said absorbent pad, and an inserted member formed from a layer which extends from said side edge of said absorbent pad. An elastic material is affixed along a portion of the length of the inserted member, and a seal affixes the inserted member inside the loop member at its base end. The wing can be a separate material or can be formed from one of the layer materials used to form the elasticized flap. The absorbent sanitary article provides improved fit and leakage protection with better comfort.