baber/WOPTO huggingface dataset:
Patent AR-013079-A1 (AR)
Title: Derivados sustituidos de tetrahidrofurano-3-onas, de tetrahidropirano-3- onas y tetrahidrotiofen-3-onas, un procedimiento para su preparacion unacomposicion farmaceutica de un medicamento util como inhibidores de proteasas e intermediarios
IPC: C07D409/12
Filed: 1998-05-04
Abstract: Derivados sustituidos de tetrahidrofurano-3-onas, de tetrahidropirano-3- onas y tetrahidrotiofen-3-onas, caracterizados porque comprenden un compuestosegun la formula (I) en la que: R1 es R, RC(O), RC(S), RSO2, ROC(O), RRNC(O), o ROC(O)NRCH(R6)C(O); R2 es H, alquilo C1-6, alquenilo C2-6,Ar-alquilo C0-6, o Het-alquilo C0-6; R3 es H, alquilo C1-6, alquenilo C2-6, alquinilo C2-6, cicloalquil C3-6-alquilo C0-6, Ar-alquilo C0-6, o Het-alquiloC0-6; R4 es H, alquilo C1-6, alquenilo C2-6, Ar-alquilo C0-C6, o Het-alquilo C0-6; R5, en cada caso, es independientemente H, alquilo C1-6, alquenilo C2-6,Ar-alquilo C0-6, o Het-alquilo C0-6; R6 es H, alquilo C1-6, alquenilo C2-6, cicloalquil C3-6-alquilo C0-6, Ar-alquilo C0-6, o Het-alquilo C0-6; Res H,alquilo C1-6, alquenilo C2-6, Ar-alquilo C0-6, o Het-alquilo C0-6; R es alquilo C1-6, Ar-alquilo C0-6, Het-alquilo C0-6, Ar-alquenilo C2-6, oHet-alquenilo C2-6, o Het-alquenilo C2-6; X es O o S; y n es 1, 2 o 3; o una de sus sales faramcéuticamente aceptables, que son inhibidores de cisteínaproteasas, particularmente catepsina K, y son utiles en el tratamietno de enfermedades uno de cuyos factores es la inhibicion de pérdida osea,procedimiento para su preparacion, una composicion farmacéutica que los comprende, el uso de los mismos para la fabricacion de un medicamento eintermediarios.
Patent AR-013535-A1 (AR)
Title: Un conjugado polimerico de 20-0-[glicil-aminoacil-glicil] camptotecina, un procedimiento para producir dicho conjugado polimerico, un derivado de 20-0-acilamino-glicil-camptotecina, un derivado de 20-0-[metacriloil-glicil- (aminoacil)-glicil] camptotecina, procedimientos para producir dichos derivad
IPC: A61K47/48
Filed: 1998-09-30
Abstract: Un conjugado polimérico de 20-0-[glicil-aminoacil-glicil]camptotecina compuesto de: (i) entre un 85 y un 97% mol de unidades de N-(2-hidroxipropil)metacriloilamida representadas por la formula (3); (ii) entre un 3 y un 15% mol de unidadesd e 20-0-(N-metacriloil-glicil-aminoacil-glicil)-camptotecinarepresentadas por la formula (4), en la que n oscila entre 2 y 8, -[o-CPT] representa el residuo de una camptotecina de la formula (2), que se encuentraunida a la posicion C-20 y enla q ue, cada una entre R1, R2, R3, R4 y R5 que pueden ser iguales o diferentes, es: hidrogeno, alquilo C1-12 lineal oramificado, nitro, amino, (CH2)aNR6R7, donde a oscila entre 0 y 4 y R6 y R7 son hidrogeno o una entre R6 y R7 es hidrogeno y laotra e ntre R6 y R7 es alquiloC1-6, o NR6R7 representa un anillo de piperazino o N-alquil-piperazino opcionalmente sustituido con alquilo C1-6 lineal o ramificado o un anillode piperidino, (CH2)aNHCOR8 donde a es tal como se definiera antesy R8 es alquilo C1-8 lineal o ramificado o un grupo NR6R7 tal como se expresara antes,hidroxi o O-CO-R8, donde R8 es tal como se definiera antes o representa un anillo 1-piperidino o 1,4-bipiperidino, o R2 y R3 tomadas en formaconjunta,representa n el residuo de O-(CH2)b-O, en el que b es 1 o 2; o R4 y R5 representan el residuo de (CH2)m, en el que m oscila entre 2 y 4, o el residuoCH2-O-CH2 o CH2NHCH2; y (iii) entre un 0 y un 12% mol de unidades de N-metacriloil-glicina o N-(2-hidroxi-propil)metacriloil-glicinamida representadaspor la formula (5), en la que [Z] representa un grupo hidroxi o un residuo de la formula -NH-CH2-CH(OH)-CH3. Este conjugado polimérico posee una actividadantitumoralmejorada y una toxicidad reducida con respecto al fármaco libre. Un procedimiento para producir a este conjugado polimérico, un derivado de
Patent AR-015998-A1 (AR)
Title: PROCESO PARA PRODUCIR MATERIAL BIOLoGICO SECO, TOTALMENTE AMORFO Y ESTABILIZADO.
IPC: A61K9/16
Filed: 1998-10-30
Abstract: Proceso para la produccion de productos amorfos secos que, además de material biologicamente activo, en particular material terapéuticamente activo,contienen mezclas de substancias para la estabilizacion, que una solucion o suspension de material biologico y una mezcla de substancias que consiste en:(a) un carbohidrato y al menos un zwitterion con un radical polar o apolar o derivados del mismo, y/o (b) al menos dos zwitteriones con radicales polareso apolares o derivados de los mismos, y/o (c)al menos un zwitterion con un radical polar o apolar o una pluralidad de zwitteriones con radicales polares oapolares o derivados de los mismos; se produce y se seca mediante secado por conveccion con ajuste del contenido en humedad a < 70% en la faseestacionaria, y una temperatura de entrada de flujo de aire de 50 - 300*C. Se refiere asimismo a los productos amorfos microcopicamente homogéneos que sonobtenidos mediante este proceso, que están en forma de polvo y que presentan una forma geométirca uniforme, en particular esférica. También se refiereadicionalmente al uso de mezclas de substancias para la estabilizacion de material biologicamente activo, en particular proteínas mediante secado porpulverizacion.
Patent AR-014632-A1 (AR)
Title: Un radio receptor para recibir una senal de television digital selaccionada
IPC: H04L27/06
Filed: 1999-02-23
Abstract: Un receptor de television digital (DTV) de QAM/VSB del tipo de conversion multiple que utiliza los mismos circuitos hasta un penultimo amplificador defrecuencia intermedia para recibir senales de DTV, ya sea que éstas utilicen modulacion de QAMo VSB. El conversor utilizado para generar senales defrecuencia intermedia final cuando se recibe la modulaci[on de QAM y el conversor utilizado para generar las senalescuando se recibe la modulacion de VSB se tienen respectivos mezcladores yresp ectivos osciladoreslocales con control automático de frecuencia y fase separados. El uso de estos conversores separados evite el bloque de la modalidad de recepcion de VSB que,de lo contrario, se puede producir durante la recepcion de senalesde DT V con modulacion de VSB.
Patent AR-014985-A1 (AR)
Title: Vaina protectora
IPC: D04C1/02
Filed: 1999-04-15
Abstract: Una vaina protectora que comprende una pared tubular la cual a su vez comprende una pluralidad de vainas similares de material flexible que estánformadas de manera de conforma una tela. Dicha pared también comprende por lo menos un hilo adicional que compren un nucleo sustancialmente inextensiblesobre el cual está formada una capa de material amortiguador. El material amortiguador forma proyecciones amortiguadoras sobre por lo menos una de lassuperficies externa e interna de la pared.
Patent AR-020752-A1 (AR)
Title: Procedimiento para controlar una distribucion sobre una superficie o en el espacio.
IPC: G06T7/41
Filed: 1999-10-08
Abstract: Procedimiento para el control de la distribucion de estructuras sobre una superficie o de partículas en el espacio donde, por ejemplo con técnicas de video, se genera una imagen optica bidimensional de la distribucion, se la descompone en elementos de imagen determinando la luminosidad media de cada elemento deimagen y se calculan las diferencias entre los valores de luminosidad de elementos de imagen vecinos a lo largo de filas de elementos de imagenpreseleccionadas. Estos valores de diferencias se almacenan sobre un portador de datos y/o se emiten de manera tal que se mantenga una correlacion entre losvalores de diferencia con la ubicacion de los elementos de imagen sobre la imagen. De esta forma se puede determinar en cuales lugares apareceninhomogeneidades en la distribucion de estructuras sobre una superficie o de partículas en el espacio. Por ejemplo, el procedimiento puede aplicarse en laevaluacion de la homogeneidad de superficies, en la deteccion de efectos de superficie y para el control del ángulo de apertura y de la homogeneidad de unchorro de rociado.
Patent WO-2007147193-A1 (WO)
Inventor: ZEILLINGER ROLAND
IPC: F02K1/72
Filed: 2007-06-22
Abstract: Die Erfindung betrifft Führungs träger (6, 7) für die Verkleidung (1) von Strahltriebwerken für Flugzeuge, umfassend einen durch ein Hohlprofil 14, 15 mit im Wesentlichen geschlossenem Querschnitt gebildeten Grundkörper (8, 9) mit zumindest einer Gleiteinrichtung (10, 11) zur verschieblichen Lagerung einer Schubumkehreinrichtung (2), mit einer Anbindung für eine innere Triebwerksverkleidung (5), und mit Beschlägen (12, 13) zur lösbaren und schwenkbaren Befestigung an einer Tragkonstruktion zu Verbindung mit einem anderen Führungs träger (7). Zur Schaffung eines derartigen Führungs trägers (6, 7), welcher besonders niedriges Gewicht aufweist und dennoch ausreichend steif ist, ist das Hohlprofil (14, 15) aus kohlenstoff faserverstärktem Kunststoffmaterial nach der Harz Infusions-Methode hergestellt ist. Zur Anbindung an die innere Triebwerksverkleidung (5) befinden sich zwei Flansche (18, 19) am Hohlprofil (14, 15) des Grundkörpers (8, 9) des Führungs trägers (6, 7).
Patent WO-2013090951-A1 (WO)
Title: Châssis de tiroir à double paroi, comportant une paroi intérieure et une paroi extérieure
Inventor: FEUERSTEIN MARKUS
IPC: A47B88/00
Filed: 2012-11-02
Abstract: L'invention concerne un châssis de tiroir à double paroi (1), comportant une paroi intérieure (2) et une paroi extérieure (3) qui peuvent être reliées l'une à l'autre, de préférence par collage. La paroi intérieure (2) possède une partie de liaison de paroi intérieure (2a) et la paroi extérieure (3) possède une partie de liaison de paroi extérieure (3a). Dans la position de montage, la partie de liaison de paroi intérieure (2a) et la partie de liaison de paroi extérieure (3a) sont disposées à l'intérieur du châssis de tiroir à double paroi (1) et peuvent être reliées l'une à l'autre pour raccorder la paroi intérieure (2) à la paroi extérieure (3). Grâce à un dispositif de retenue mécanique (4) pouvant être relié à la partie de liaison de paroi intérieure (2a) et à la partie de liaison de paroi extérieure (3a), la paroi intérieure (2) peut être immobilisée de manière stable par rapport à la paroi extérieure (3).
Patent WO-2014078880-A1 (WO)
Title: Vorrichtung zum bohren von ankerlöchern im untertagebau
Inventor: LEOPOLD HORST
IPC: E21B7/02
Filed: 2012-11-21
Abstract: Es wird eine Vorrichtung zum Bohren von Ankerlöchern im Untertagebau mit einem Gestell (1) beschrieben, das parallele Verschiebeführungen (2) einerseits für einen an der zu bohrenden Fläche (9) abstützbaren Schlitten (3) und anderseits für eine Bohreinrichtung (4) bildet, deren Vorschubantrieb (10) am Schlitten (3) abgestützt ist. Um die Bohrlochtiefe genau bestimmen zu können, wird eine magnetostriktive Messeinrichtung mit entlang der Verschiebeführungen (2) verlaufenden, an eine Auswerteschaltung angeschlossenen Messfühlern (17) und mit dem Schlitten (3) und der Bohreinrichtung (4) zugehörigen, mit dem jeweiligen Messfühler (17) zusammenwirkenden magnetischen Lagegebern (18) vorgeschlagen.
Patent AU-2002225953-A1 (AU)
Title: Injection high frequency noise into pulse excitation for low bit rate celp
Inventor: GAO YANG
IPC: G10L19/12
Filed: 2001-12-10
Abstract: This method for speech coding comprises generating (602) an excitation signal by use of at least one pulse codebook (202, 204) applied to a speech signal (s(n)); and providing a high frequency enhancement (610) of the excitation signal based on one or more criteria. In the method the one or more criteria includes an energy content of the speech signal.
Patent AU-2002352569-A1 (AU)
Title: Nonwoven separator for electrochemical cell
Inventor: AUDEBERT JEAN-FRANCOIS
IPC: H01M50/429
Filed: 2002-11-08
Abstract: A low volume nonwoven separator and an electrochemical cell employing the separator are provided. The cell includes a positive electrode and a negative electrode. The nonwoven separator is disposed between the positive electrode and negative electrode. The nonwoven separator comprises, prior to insertion in the cell, a non-compressed single layer dry thickness in the range of 0.04 to 0.09 mm, and an average pore size of no greater than 14 mum. The cell further includes an electrolyte in contact with the separator and the positive and negative electrodes.
Patent AU-2002360133-A1 (AU)
Title: Motor fan system which is intended, in particular, for a motor vehicle heating and/or air-conditioning system
Inventor: GATINOIS JEAN
IPC: B60H1/00
Filed: 2002-10-18
Abstract: The invention relates to a speed control unit for the motor of a motor fan system comprising a printed circuit board (40). Electronic components (50), which are disposed on said board, are interconnected by means of electric strips (50) and thermally coupled to a radiator (60). Said one-piece radiator (60) extends along the entire lower surface of the board (40) and comprises first contact areas (61, 62), which are directly thermally coupled to several electronic components (51, 52), and second contact areas (63) which are thermally coupled to equipotential areas located on the lower surface of the printed circuit board (40).
Patent AU-2003213738-A1 (AU)
Title: Heavy hydrocarbon recovery from pressure swing adsorption unit tail gas
Inventor: DOLAN WILLIAM B
IPC: C07C7/12
Filed: 2003-03-07
Abstract: A pressure swing adsorption process for the separation of impurities such as nitrogen and carbon dioxide and recovery of hydrocarbons from a natural gas stream utilizes two separate adsorption systems, the first containing an adsorbent selective for nitrogen, carbon dioxide or both and the second containing a hydrocarbon-selective adsorbent. In the process, the natural gas stream is passed through a first adsorbent to form a product stream enriched with methane and to adsorb nitrogen and/or carbon dioxide and which further co-adsorbs at least a portion of the hydrocarbons contained in the feed stream. The hydrocarbons are recovered by passing a low pressure waste stream from the first pressure swing adsorption stage which contains co-adsorbed nitrogen and/or carbon dioxide and hydrocarbons and directing the waste stream to the second pressure swing adsorption stage to adsorb the hydrocarbons and produce a product stream enriched in nitrogen and/or carbon dioxide. The hydrocarbons are recovered from the hydrocarbon-selective adsorbent by an intermediate pressure methane-containing stream from the first pressure swing adsorption stage which purges the adsorbent in the second stage and forms a combined stream comprising methane and C3+ hydrocarbons. The C3+ hydrocarbons can be separated from the methane such as by compression with flash separation or refrigeration.
Patent AU-2003218945-A1 (AU)
Title: Method for the continuous production of biomethanol diesel
Inventor: ADLER BERNHARD
IPC: C11B3/00
Filed: 2003-03-06
Abstract: In the production of biomethanol diesel from rapeseed oil in relatively small amounts by catalytic ester exchange in a microreactor cascade, the freshly expressed oil is washed twice with methanol, before actual ester exchange in the cascade, so that acid numbers at most 0.1 are attained.
Patent AU-2003227771-A1 (AU)
Title: Vacuum pump for bottles
Inventor: BONICH MARTA BRUCART
IPC: B65B31/04
Filed: 2003-05-20
Abstract: The invention relates to a vacuum pump for bottles, which is particularly suitable for wine bottles which have been opened but not completely consumed. The inventive pump consists of a support (1) which can be connected to the neck (4) of the bottle and which comprises an inner constriction (2) that rests on the mouth (3) of said bottle. The aforementioned constriction forms the support and the head (7) of a stopper (8) which penetrates the mouth (4) of the bottle and which is solidly fixed thereto. Moreover, the invention also comprises a cover (19) which can be moved axially in relation to the support (1) and which forms a variable-volume chamber (22) along with said support and the head (7) of the stopper. According to the invention, a unidirectional valve (11-14-16) is formed in the stopper (8) and a second unidirectional valve (20-21) is formed between the support (1) and the cover (19) such that, when the chamber (22) increases, air is drawn from inside the bottle and, when the chamber decreases, said air is released to the exterior. <IMAGE>
Patent AU-2003240977-A1 (AU)
Title: Abrasive product, method of making and using the same, and apparatus for making the same
Inventor: CHESLEY JASON A
IPC: B24D3/28
Filed: 2003-06-02
Abstract: The invention provides a method and apparatus for making an abrasive product comprising providing a substantially horizontally deployed flexible backing having a first surface bearing an at least partially cured primer coating and an opposite second surface; providing a dry flowable particle mixture comprising abrasive particles and particulate curable binder material; depositing a plurality of temporary shaped structures comprised of said particle mixture on the at least partially cured primer coating of the first surface of the backing; softening said particulate curable binder material to provide adhesion between adjacent abrasive particles; and curing the softened particulate curable binder material to convert said temporary shaped structures into permanent shaped structures and cure the at least partially cured primer coating on the first surface of the backing. The invention also provides an abrasive product made by the method.
Patent AU-2003250927-A1 (AU)
Title: A continuous metal strip casting plant
Inventor: KAPAJ NUREDIN
IPC: B22D11/06
Filed: 2003-07-09
Abstract: A continuous metal strip casting plant on which is mounted, at the casting location, a mobile ingot mould comprising two cylindrical metallic casting rolls in addition to other components, amongst which there are a tundish and/or under tundish and/or an unloader and/or lateral plates, respective preheating stations located in positions separated from the position of casting, and rotating arms located on a turret itself also placed on the casting plane to transfer the components from the casting line to their preheating stations.
Patent AU-2003254493-A1 (AU)
Title: Plant watering system
Inventor: GRAHAM GRAHAM
IPC: A01G31/00
Filed: 2003-07-24
Abstract: The invention relates to a plant watering system and in particular a system which allows the long-term watering of plants without the need for an open reservoir. The invention uses a water insoluble polymer contained within a porous bag or enclosure ( 1 ) to hold water in a reservoir type manner, which can then be provided to the plant ( 7 ) as required.
Patent AU-2003267283-A1 (AU)
Title: Methods for measuring rates of reserve cholesterol transport in vivo, as an index of anti-atherogenesis
Inventor: HELLERSTEIN MARC K
IPC: G01N33/15
Filed: 2003-09-15
Abstract: The present invention relates to biochemical methods for determining reverse cholesterol transport. Specifically, the rates of the two arms of reverse cholesterol transport (HDL or first arm and post-HDL or second arm) are obtained by measuring the flow of unlabeled cholesterol from tissues into plasma HDL and from plasma HDL to bile acids.
Patent AU-2003289691-A1 (AU)
Title: Vehicle cab
Inventor: FORSMAN LARS
IPC: B62D25/04
Filed: 2003-12-10
Abstract: A vehicle cab having a frame construction comprising a pair of front supporting A-pillars, a pair of rear supporting B- or C-pillars, at least one front transverse beam, which mutually connects said front supporting A-pillars, and a rear transverse beam, which mutually connects said rear supporting B or C-pillars, and a pair of roof bars, which are supported by and connect said front supporting A-pillars to said rear supporting B or C-pillars.
Patent AU-2003294453-A1 (AU)
Title: Polyhydropolyborates as polymerization catalysts
Inventor: LEMMON JOHN PATRICK
IPC: C08G64/30
Filed: 2003-11-21
Abstract: The present invention relates to a synthetic method comprising contacting at least one diaryl carbonate with one or more dihydroxy aromatic compounds in the presence of a transesterification catalyst under melt polymerization conditions to afford a product polycarbonate. The transesterifcation catalysts used according to the method of the present invention are polyhydropolyborates in combination with tetraalkylammonium or tetraalkylphosphonium compounds which serve as co-catalysts. The transesterification catalysts employed according to the method of the present invention provide polycarbonates having reduced levels of Fries rearrangement product relative to conventionally employed catalysts such as sodium hydroxide in combination with tetramethylammonium hydroxide co-catalyst.
Patent AU-2003303714-A1 (AU)
Title: Improved linkers for radiopharmaceutical compounds
Inventor: HAEN CHRISTOPH DE
IPC: A61K38/095
Filed: 2003-12-24
Abstract: A new and improved method for extending the half life of pharmaceutical compounds for use in diagnostic imaging or therapy uses a novel linker to attach a diagnostic or therapeutic moiety to a targeting peptide or another diagnostic or therapeutic moiety. The resulting compound may have the general formula M-N—O—P-Q, wherein M is the diagnostic or therapeutic moiety, N—O—P is the linker of the present invention, and Q is the targeting peptide. In another embodiment the compounds may have the formula M-N—O—P-M, wherein M is independently a diagnostic or therapeutic moiety and N—O—P is the linker of the invention. Methods for imaging or treating a patient using the compounds of the invention are also provided. Methods and kits for preparing a diagnostic imaging agent from the compound are further provided. Methods for radiotherapy of a patient using the compounds are further provided, as are methods for preparing a radiotherapeutic agent from the compounds.
Patent WO-2004092079-A1 (WO)
Title: Appareil et procede de traitement de dechets
Inventor: AMES ROY VICTOR
IPC: C02F1/44
Filed: 2004-04-16
Abstract: L'invention concerne un système de traitement de déchets, qui convient pour un usage domestique et peut produire de l'eau de recyclage appropriée pour le ménage. Le système comprend un bioréacteur (30) et une chambre de décomposition (16). Le bioréacteur (30) est conçu pour digérer des matières-déchets liquides à l'aide de bactéries, et peut être mis en oeuvre dans des conditions anaérobies, anoxiques et/ou aérobies. La chambre de décomposition (16) décompose les déchets sensiblement solides générés dans le bioréacteur. Le bioréacteur et la chambre de décomposition communiquent librement, si bien que les déchets sensiblement solides générés dans le bioréacteur peuvent être transférés vers la chambre de décomposition pour un traitement ultérieur. Les matières solides résultantes peuvent facultativement être acheminées vers une cellule de végétation (24), et le liquide (34) sortant du bioréacteur peut facultativement être transféré vers une unité de traitement à membrane (40) et une unité de désinfection (50).
Patent WO-2005019080-A1 (WO)
Inventor: PYE WARRICK KEITH
IPC: B32B37/20
Filed: 2004-08-25
Abstract: L'invention concerne un applicateur de bande (51) permettant d'appliquer une bande sur un substrat, l'applicateur de bande comprenant une paire de rouleaux pinceurs, lesdits rouleaux pinceurs comprenant un rouleau de bande (55) et un rouleau de substrat (56), l'applicateur de bande comprenant également un rouleau de tension (57) disposé en face du rouleau de substrat (56) afin de tendre le substrat préalablement à l'alimentation entre les rouleaux pinceurs, un mécanisme d'alimentation de bande et un mécanisme d'entraînement pour faire tourner les rouleaux pinceurs.
Patent AU-2004213716-A1 (AU)
Title: Signal amplification method for detecting mutant gene
Inventor: FUJIKAWA TOSHIHIKO
IPC: C12Q1/68
Filed: 2004-02-20
Abstract: There is provided a signal amplification method for detecting a mutated gene, which can increase the detection sensitivity of mutated genes on a DNA chip according to the PALSAR method, can establish efficient signal amplification and can establish simple detection by contriving design of oligonucleotide probes for use in the PALSAR method. The signal amplification method comprises a ligation reaction with a DNA ligase and a self-assembly reaction which forms a double-stranded self-assembly substance having a regular higher-order structure of oligonucleotides, wherein the detection sensitivity of the mutated gene on a DNA chip is improved. <IMAGE>