baber/WOPTO huggingface dataset:
Patent AU-608821-B2 (AU)
Title: Methods of treating gout with chalcone derivatives
Inventor: EDWARDS MICHAEL L
IPC: A61K31/165
Filed: 1988-04-05
Granted: 1991-04-18
Abstract: Certain chalcone derivatives are reported to inhibit the polymerization of tubulin to form microtubules and are therefore antimitotic agents which can be used to control the growth of tumor tissue and can be used as antigout agents. The chalcone derivatives are also reported to inhibit the destruction of the myelin sheath in the central nervous system of multiple schlerosis patients and are thus useful in controlling the progressive nature of the disease.
Patent AU-695931-B2 (AU)
Title: PNA synthesis using an amino protective group which is labile to weak acids
Inventor: BREIPOHL GERHARD
IPC: C07D473/18
Filed: 1995-03-10
Granted: 1998-08-27
Abstract: A process is claimed for preparing peptide nucleic acid (PNA) oligomers of formula (I) B-X = a gp. of formula (i)-(viii): f = 1-4; g = 0-3; Ro = H, 1-18C alkanoyl, 2-19C alkoxycarbonyl, 3-8C cycloalkanoyl (sic), 7-15C aroyl, 3-13C heteroaroyl or a gp. which enhances intracellular uptake of the oligomer or interacts with a target nucleic acid during hybridisation; A and Q = amino acid residues; k and m = 0-10; B = a natural or non-natural nucleotide base, opt. in prodrug form, or a base substitute; Qo = OH, NH2 or NHR"; R" = 1-18C alkyl, 2-18C aminoalkyl or 2-18C hydroxyalkyl; n = 1-50. The process comprises: (a) opt. coupling amino acids (Q<1>) to a support of formula L-(Polymer) by solid-phase synthesis, where L = a linking gp. contg. Qo in latent form and Q<1> = Q with optional side-chain protecting; (b) opt. removing the protecting gp. PG (sic) with a suitable reagent; (c) repeating steps (a) and (b) m-1 times to give (Q<1>)m-L-(Polymer); (d) coupling a cpd. of formula (II) to L-(Polymer) or (Q<1>)m-L-(Polymer): PG-X(B<1>)-OH (II) where PG is a weak-acid-labile protecting gp. and B<1> is B with opt. protected exocyclic amino or OH gps.; (e) removing PG; (f) repeating steps (d) and (e) n-1 times; (g) opt. coupling amino acids (A<1>) to the prod. by solid-phase synthesis, where A<1>=A with optional side-chain protection; (h) removing the protecting gp. PG (sic) with a suitable reagent; (i) repeating steps (g) and (h) k-1 times; (j) introducing Ro if Ro is other than H; and (k) cleaving the PNA oligomer from the prod. of formula (III) and simultaneously or subsequently deprotecting B<1>, A<1> and Q<1>: Ro-(A<1>)k-(X(B<1>))n-(Q<1>)m-L-(Polymer) (III).
Patent AU-609120-B2 (AU)
Title: Use of ODC inhibitors, dacarbazine, and interferon in the treatment of malignant melanoma
Inventor: SUNKARA SAI P
IPC: A61K31/195
Filed: 1988-04-21
Granted: 1991-04-26
Abstract: This invention relates to the improvement of the polyamine depletion effects of ornithine decarboxylase inhibitors, the improvement being effected by the use of Interferon and Dacarbazine in conjunctive therapy with said inhibitors.
Patent AU-766991-B2 (AU)
Title: Method and rock drilling apparatus for controlling rock drilling
Inventor: AHTOLA UNTO
IPC: E21B47/022
Filed: 1999-12-08
Granted: 2003-10-30
Abstract: A method and a rock drilling apparatus for drilling holes in rock according to a predetermined drilling plan. The method comprises measuring the location of each hole in the rock by inserting a measuring device into the hole, and calculating the deviation of the end of the measured hole from the location determined in the drilling plan. The rock drilling apparatus comprises a measuring device that can be inserted into a drill hole, and means for transferring the measurement values measured by the measuring device to control means of the rock drilling apparatus.
Patent AU-772001-B2 (AU)
Title: A self-expanding stent-graft
Inventor: DAVILA LUIS A
IPC: A61F2/06
Filed: 2001-01-29
Granted: 2004-04-08
Abstract: In accordance with the present invention, there is provided a stent-graft for insertion into target site within a vessel of a patient. The graft has a crimped state for delivery to the target site, and an expanded state for implantation therein. The graft has a self-expanding outer stent, which is a tubular member made from an elastic material. The graft further includes a tubular flexible porous graft member extending along the interior of the outer stent. The graft member has front and back ends which are folded over and bonded to the front and back ends of the outer stent to form cuffs. In addition, the stent-graft has a self-expanding inner stent which also is a tubular member made from an elastic material. The inner stent is disposed within the interior of the graft member such that the inner stent, the graft member and the outer stent are all abutting. <IMAGE>
Patent AU-662742-B2 (AU)
Title: Circular saw blade straightening machine
Inventor: OPPLIGER WALTER
IPC: B23D63/18
Filed: 1992-06-30
Granted: 1995-09-14
Abstract: This invention relates to a saw blade straightening machine for removing unevenness in circular saw blades with straightening rollers or drums arranged on both sides of the saw blade for correcting uneven regions of the saw blade, in that straightening rollers or drums (14, 14', 17, 17') for smoothing unevenness in the different directions of the saw blade (1) are arranged opposite one another on a straight line leading through the middle of the saw blade, at equal distances from the centre, and a dial gauge (26) for scanning one surface of the saw blade and for generating a signal if unevenness is detected is arranged offset by a specific angle in relation to the straightening rollers and at the same distance from the centre of the saw blade. <IMAGE>
Patent AU-578232-B2 (AU)
Title: Composite apparatus for generation of electrical energy from solar energy
Inventor: NAGAI TOKI
IPC: H01L31/052
Filed: 1983-10-26
Granted: 1988-10-20
Abstract: PCT No. PCT/JP83/00379 Sec. 371 Date May 9, 1985 Sec. 102(e) Date May 9, 1985 PCT Filed Oct. 26, 1983 PCT Pub. No. WO84/02584 PCT Pub. Date Jul. 5, 1984.This invention deals with a composite electromotive apparatus utilizing solar energy and the like, comprising composite electromotive elements such as a thermoelectromotive unit, a photovoltaic unit, a magnetic electromotive unit utilizing convection, radiation, and/or other phenomena and so forth, to aim to gain electromotive even if momentarily small but as often as possible, with less limits in spite of any conditions, environment, etc., but without taking huge spaces and the like.
Patent AU-655838-B2 (AU)
Title: Process for the preparation of a cephalosporin antibiotic
Inventor: LIM GARY M F
IPC: C07D501/56
Filed: 1992-09-09
Granted: 1995-01-12
Abstract: The present invention provides an anhydrous acylation process for the preparation of antibiotic, cefepime dihydrochloride hydrate which is substantially free of the anti-isomer and the  DELTA <2> isomer comprising the N-acylation of a silylated derivative of 7-amino-3-[(1-methyl-1-pyrrolidinio)-methyl]ceph-3-em-4-carboxylate with the syn-isomer of 2-(2-aminothiazol-4-yl)-2-methoxyimino acetyl chloride hydrochloride.
Patent AU-670734-B2 (AU)
Title: Process and device for the separation of substances by crystallization of molten material
Inventor: KONIG AXEL
IPC: B01D9/00
Filed: 1995-04-28
Granted: 1996-07-25
Abstract: PCT No. PCT/EP95/01617 Sec. 371 Date Mar. 29, 1996 Sec. 102(e) Date Mar. 29, 1996 PCT Filed Apr. 28, 1995 PCT Pub. No. WO95/30466 PCT Pub. Date Nov. 16, 1995Crystallization of a melt is induced by causing the melt to flow downwardly in a gap which is defined by upwardly moving cooled walls so that crystallate adheres to the walls and is carried upwardly for recovery. The walls are formed by endless belts which are cooled by fluid sprayed from nozzles. The walls are adjustable so as to be parallel or upwardly divergent.
Patent AU-726914-B2 (AU)
Title: Bioactivated diagnostic imaging contrast agents
Inventor: LAUFFER RANDALL B
IPC: A61K49/14
Filed: 1997-03-25
Granted: 2000-11-23
Abstract: The present invention relates to improved diagnostic agents for Magnetic Resonance Imaging and optical imaging. In particular, this invention relates to MRI and optical imaging agents that allow for the sensitive detection of a specific bioactivity within a tissue. These agents are prodrug contrast agents which are bioactivated in vivo in the presence of the specific bioactivity. This invention also relates to pharmaceutical compositions comprising these agents and to methods of using the agents and compositions comprising the agents.
Patent AU-658007-B2 (AU)
Title: Synergistic combinations of 2-(thiocyanomethylthio)benzothiazole with a mixture of 4,4-dimethyloxazolidine and 3,4,4-trimethyloxazolidine in controlling fungal and bacterial growth in aqueous fluids
Inventor: OPPONG DAVID
IPC: C10M173/02
Filed: 1992-09-24
Granted: 1995-03-30
Abstract: Synergistic combinations of 2-(Thiocyanomethylthio)-benzothiazole and a mixture of 4,4-dimethyloxazolidine and 3,4,4-trimethyloxazolidine for use in controlling the growth of at least one microorganism, such as fungi and bacteria, in aqueous fluids, such as metalworking fluids.
Patent AU-752849-B2 (AU)
Title: Self-heating or self-cooling containers
Inventor: SEARLE MATTHEW JOHN
IPC: A47J36/28
Filed: 2000-02-28
Granted: 2002-10-03
Abstract: A self-heating container (10) has an internal cavity (22) for its contents and an external cavity (20) for a heating mechanism, for example, comprised of first and second chemically reactive materials which are arranged to be mixed when heating is required. A closure (30) closes the external cavity (20). When the heating mechanism is operated to mix the chemicals and cause an exothermic reaction, vapor, such as steam and hot air, is produced. The vapor is constrained to flow to the exterior of the closure (30) through grooves (62) therein. A sleeve (60) is arranged around the container (10) contiguous to the closure (30) such that the exiting vapor is constrained to flow between the sleeve (30) and the can (10). By this means, a user of the can is protected from coming into contact with the hot steam and air and the heat in the vapor generated can enhance the heating process. Preferably, the sleeve (60) is constructed of an absorbent material, such as a cardboard, to absorb any condensates and this absorbent material is surrounded by an impermeable plastics material to insulate the user from the heat of the reaction.
Patent AU-685971-B2 (AU)
Title: Process for the preparation of the (-)-N-methyl-N-{4-(4- phenyl-4-acetylaminopiperidin-1-yl)-2-(3,4-dichlorophenyl) butyl}benzamide and its pharmaceutically acceptable salts
Inventor: DESCAMPS MARCEL
IPC: A61K31/445
Filed: 1995-08-23
Granted: 1998-01-29
Abstract: A process is described for the preparation of (+)-2-(3,4-dichlorophenyl)-4-hydroxybutylamine of formula (I) and for the preparation of the (-)-N-methyl-N-Ä4-(4-phenyl-4-acetylamino-piperidin-1-yl)-2-(3,4-dichl orophenyl)butylÜ benzamide and of its pharmaceutically acceptable salts using the compound of formula (I) as synthesis intermediate.
Patent AU-718770-B2 (AU)
Title: Beat onset detector
Inventor: POLIAC MARIUS O
IPC: A61B5/0245
Filed: 1997-05-28
Granted: 2000-04-20
Abstract: A method for identifying an onset of a first heart beat includes sensing blood pressure over time to produce a plurality of blood pressure samples, each sample having a corresponding blood pressure amplitude in time, identifying a post onset point in time following an onset of the first heart beat and preceding an onset of a second heart beat, and identifying an onset of the heart beat based upon the blood pressure samples and the post onset point.
Patent AU-664592-B2 (AU)
Title: Transparent file mark
Inventor: GARCIA JOSE A
IPC: G11B27/32
Filed: 1993-02-24
Granted: 1995-11-23
Abstract: Separations between the end of one data file (150) and the beginning of the next data file (151) are recognized, without utilizing an entire data storage block by means of a controlling program for a peripheral recording device monitoring the control information headers (156) of helically stored data on a magnetic tape. When files are stored on the magnetic tape, the controlling program increments an increase of a file section number (152) by one and increments to zero a data block number (154) at the beginning of a new data file. When the recording device is reading the magnetic tape and there is detected an incrementation of the file section number (152) and a zero value for a data block number (154), a recognition is made that this data indicates the end of one data file and the beginning of another data file. <IMAGE>
Patent AU-750613-B2 (AU)
Title: Synchronisation and/or data exchange method for secure, fault-tolerant computers and corresponding device
Inventor: SCHMERBECK FRIEDRICH
IPC: G06F11/16
Filed: 1999-02-17
Granted: 2002-07-25
Abstract: The invention relates to a synchronisation and/or data exchange method for secure, fault-tolerant computers. The method enables the synchronisation of or the exchange of data between several individual computers working in parallel. The synchronisation or exchange of data is carried out with interrupt signals and using standard components. The invention also relates to a device for carrying out the inventive method.
Patent AU-693939-B2 (AU)
Title: Novel crystal forms of 1-(5-methanesulfonamidoindolyl-2- carbonyl)-4-(3-(1-methylethylamino)-2-pyridinyl) piperazine
Inventor: HAVENS JEFFREY L
IPC: A61K31/496
Filed: 1995-03-01
Granted: 1998-07-09
Abstract: The present invention relates to two novel crystal forms of a known compound, 1-[5-Methanesulfonamidoindolyl-2-carbonyl]-4-[3-(1-methylethylamino)-2-pyridinyl] piperazine monomethanesulfonate salt, which are useful for treating humans who are HIV positive, which are identified by a powder X-ray diffraction spectrum known commonly as the "S" and "T" forms.
Patent AU-671436-B2 (AU)
Title: Elevated temperature dimensionally stable polyester with low gas permeability
Inventor: DALGEWICZ EDWARD J III
IPC: B29C49/00
Filed: 1993-02-03
Granted: 1996-08-29
Abstract: Polyester composition with improved impact properties, improved oxygen permeability and improved dimensional skrinkage during heating. Impact modifiers are dissolved into a molten polyester to form a eutectic alloy. On slow cooling, the eutectic alloy of the invention freezes to form a mixture of particles of the impact modifier embedded in a matrix of the polyester. By controlling the solidification of the melt, the size and distribution of the precipitates from the melt can be controlled, which allows control of the mechanical properties. The precipitation can also be controlled either by homogenous nucleation or by heterogeneous nucleation through the addition of a nucleating agent or the introduction of a suitable surface for nucleation. The invention also provides a process of manufacturing the above polyester, an article comprising this polyester and a process for making this article. The crystalline polyester article is useful as a container for microwavable, ovenable and/or frozen foods, and has improved gas barrier properties, impact strength, and post-mold dimensional stability between -60  DEG C and 200  DEG C.
Patent AU-573664-B2 (AU)
Title: Wireline jar
Inventor: ZWART KLAAS
IPC: E21B31/107
Filed: 1984-12-18
Granted: 1988-06-16
Abstract: An upstroke wireline jar having a hammer 12 at the bottom end of an operating rod 3 which is axially slidable in a casing 2 having an anvil 13 at its upper end. This casing also includes a releasable coupling means which is biased downwards by a spring 5 to a rest position, said coupling means comprising a sleeve 4 which receives the rod 3 into its upper end and a plurality of arcuate segments 9 which are contained in apertures in the sleeve and engage in a circumferential groove 10 in the rod. Circumferential recesses 11 and 17 in the interior wall of the casing 2 are adapted to partially receive the segments when the sleeve is in appropriate registration therewith thereby facilitating disconnection and subsequent re-engagement of the operating rod with the sleeve. The spring 5 is mounted below the hammer so as to allow free travel of the latter along a substantial portion of the casing. The spring is provided with an upper abutment 6 mounted on a rod 7 the axial position of which is adjustable from outside the jar. At its bottom end the spring 5 abuts a flanged bush 15 which depends from the sleeve 4. A second spring 6 assists in biasing the sleeve to its rest position.
Patent AU-762973-B2 (AU)
Title: Methods and compositions for producing viral particles
Inventor: TORRENT CHRISTOPHE
IPC: C12N7/00
Filed: 1999-05-18
Granted: 2003-07-10
Abstract: The invention concerns methods and constructs for producing retroviral particles, in vitro, ex vivo or in vivo. It also concerns the use of said methods and constructs for transferring nucleic acids into cells. More particularly, the invention concerns a composition comprising the whole set of genetic elements required for constituting a retroviral particle, incorporated in one or several recombinant adenoviruses defective for all or part of the regions E1 and E4 at least (adenoviral/retroviral chimeric vectors).
Patent AU-667715-B2 (AU)
Title: Carrier system against GnRH
Inventor: ZEE ANNA VAN DER
IPC: A61K47/48
Filed: 1993-06-18
Granted: 1996-04-04
Abstract: The present invention is concerned with vaccination of mammals against GnRH. The vaccine comprises a GnRH peptide conjugate to E. coli fimbrial-filaments and elicits an immune response against GnRH.
Patent AU-764108-B2 (AU)
Title: A novel VLA-4 inhibitor: oMePUPA-V
Inventor: LEE WEN-CHERNG
IPC: A61K31/40
Filed: 1999-05-28
Granted: 2003-08-07
Abstract: OMePUPA-V, (R)-N-[[4-[[(2-methylphenylamino)carbonyl]amino]phenyl]acetyl]-L-prolyl-3-methyl)-beta-Alanine, a cell adhesion inhibitor, pharmaceutical compositions, and methods of treatment of cell-adhesion mediated pathologies.
Patent AU-668737-B2 (AU)
Title: Contact lenses comprising lipophilised cyclodextrins
Inventor: HERBRECHTSMEIER PETER
IPC: C08G77/42
Filed: 1993-07-30
Granted: 1996-05-16
Abstract: The present invention relates to a contact lens which contains a crosslinked cyclodextrin derivative which has been rendered lipophilic and which is characterised by repeating units of the formula V <IMAGE> in which n is a number from 6 to 15, each of the R<1> radicals is, independently of the others, R<2> or R<7>, where at least one R<1> radical of the (3 times n) R<1> radicals has the meaning of R<7> and the remaining R<1> radicals are hydrogen or have the meaning of R<2>, in which R<2> is unsubstituted or halogen-substituted alkyl or alkyl-substituted aryl, and in which R<7> is a divalent or polyvalent radical of the formula VI <IMAGE> in which x is a number from 1 to 10,000, R<4>, R<5> and R<8> are, independently of one another, hydrogen, alkyl, unsubstituted or halogen-substituted alkylene or alkenylene, phenyl or hydroxyl, with the proviso that in one radical of the formula VI at least two of the radicals R<4>, R<5> and R<8> are unsubstituted or halogen-substituted alkylene or alkenylene. The invention likewise relates to the use of such crosslinked lipophilic cyclodextrin derivatives for producing contact lenses.
Patent AU-575964-B2 (AU)
Title: Pineapple ketone carbonate derivatives
Inventor: BYRNE BRIAN
IPC: C07D307/58
Filed: 1985-07-01
Granted: 1988-08-11
Abstract: A compound of the general formula, <CHEM> wherein R1 and R2 independently are -H, -CH3, or -CH2CH3; and R3 is alkyl of from 1 to 10 carbons or aryl of from 6 to 10 carbons.
Patent AU-751489-B2 (AU)
Title: Method of preparing dry animal feed
Inventor: MOLOGNI BATTISTA
IPC: A23K1/00
Filed: 1999-05-05
Granted: 2002-08-15
Abstract: The present invention relates to a method of preparing a ground dry animal feed with a predetermined water content. According to the method, there is added to a dry animal feed mixture an emulsion of water emulsified in a hydrophobic component having a melting point of at least 15° C., suitably at least 20° C., in such an amount that the animal feed obtains the predetermined water content.
Patent AU-762174-B2 (AU)
Title: Fishing reel
Inventor: WHITTLE-HERBERT GILES
IPC: A01K89/016
Filed: 1999-07-28
Granted: 2003-06-19
Abstract: This invention relates to a fishing reel (10) which comprises a reel body (12), a spool (14) rotatable relative to the reel body, a handle (16) for rotating the spool, and a drive bearing (32) connecting the handle to the spool. The drive bearing (32) is in the form of a ball-bearing including a plurality of balls (34) which are mounted to the handle (16) and which are arranged to rotate so that rotation of the handle (16) at a first velocity is transferred to the spool (14) at a second velocity greater than the first velocity.
Patent AU-745191-B2 (AU)
Title: A diffuser for aerating a fluid
Inventor: LAWSON THOMAS URIE
IPC: F16K24/06
Filed: 1997-11-12
Granted: 2002-03-14
Abstract: A diffuser for aerating a fluid, and particularly for aeration in waste water treatment tanks, is formed in an elongate configuration by manufacturing a base plate from an extrusion cut to the desired length. A perforated elastomeric membrane is secured to the base plate by pressing sealing strips along the elongate edges of the membrane into corresponding grooves formed in the base plate extrusion. The ends of the membrane are sealed to the base plate by end strips or clamps. Air is introduced through apertures in the base plate causing the membrane to inflate away from the base plate forming an interior compartment for the passage of air along the diffuser. Apparatus for securing the diffuser to a horizontal header pipe is also described.
Patent AU-581944-B2 (AU)
Title: Apparatus for the rapid determination of the moisture content of a material
Inventor: PHILIPPE JEAN
IPC: G01N5/04
Filed: 1985-11-18
Granted: 1989-03-09
Abstract: A device for determining the moisture content of a material which includes a micro wave heating unit (1) for heating a sample of the material which is under investigation and a weighing device (3) for weighing the sample during heating and providing signals representing a series of measurements of the weight of the sample at specific times. The weighing device is connected to a processing unit (4) which is a microprocessor and which includes a computer (9) which produces signals representing the loss of weight of the sample in the course of heating and which computes the parameters of a asymptotic function and which represents the loss of weight of the sample in the course of time. There is also a calculator (11) for determining the differences between two asymptotic values, and a comparator (12) for comparing the differences with a reference value representing the acceptable uncertainty in regard to the moisture content of the material. There is also a restoring device for restoring the asymptotic values when the differences reach values which are equal to or less than the reference value.
Patent AU-631190-B2 (AU)
Title: Ultraviolet absorbing lenses and methods of making the same
IPC: G02B1/04
Filed: 1990-03-06
Granted: 1992-11-19
Abstract: An ultraviolet radiation absorbing contact or intraocular lens and method of making the same, comprising a polymeric lens material to which is covalently bonded at least one halotriazine reactive ultraviolet radiation absorbing agent of the formula <CHEM> wherein A and E2 are ultraviolet radiation absorbing groups which are either identical to or dissimilar to each other, or of the formula IB   <CHEM> wherein X is Cl or F; A is an ultraviolet radiation absorbing group; and E1 is an aqueous soluble group.