baber/WOPTO huggingface dataset:
Patent JP-H08510620-A (JP)
Title: 線形電力増幅器における振幅トレーニング方法
IPC: H03G3/20
Filed: 1995-03-02
Abstract: (57)【要約】
帰還回路の入力トレーニング信号を適応変化することにより電力増幅器の振幅トレーニングを行う方法を提供する。
Patent JP-2000502395-A (JP)
Title: ポリアミドまたはポリエステル組成物
IPC: C08K5/54
Filed: 1996-12-20
Abstract: (57)【要約】
本発明は、ポリエステルおよびポリアミド組成物用の難燃剤に関し、さらに詳細には、（１）約３０〜約７０重量％のポリエステルまたは合成脂肪族ポリアミドまたはそれらの混合物と；（２）約１５〜約４０重量％のガラスまたは無機補強剤と；（３）（ａ）約２０〜約３０重量％のメラミンホスフェートおよび約１０重量％以下のチャー化触媒、（ｂ）約１５〜約３０重量％のメラミンホスフェート、約１０重量％以下のチャー化触媒および約１０重量％以下のチャー形成体、（ｃ）約５〜約４５重量％のメラミンピロホスフェート、（ｄ  約１５〜約３０重量％のメラミンピロホスフェートおよび約１０重量％以下のチャー化触媒、（ｅ）約１５〜約３０重量％のメラミンピロホスフェート、約１０重量％以下のチャー化触媒および約１０重量％以下のチャー形成体、もしくは（ｆ）約２０〜約３０重量％のメラミンピロホスフェート、および約１０重量％以下のメラミンシアヌレート、メラミンまたはホウ酸亜鉛の少なくとも１種からなる群から選ばれる難燃剤と［但し、全ての重量％は（１）＋（２）＋（３）のみの合計重量に対するものである］、を含有する組成物に関する。
Patent JP-H08509640-A (JP)
Title: 便座カバー
IPC: A47K13/16
Filed: 1994-04-28
Abstract: (57)【要約】
便座の形状に順応する洗い流し可能な便座カバー（２０）。便座の形状に順応することによって、便座カバーは、使用者が据え付けた後、適所にとどまる。便座カバー（２０）は又、汗を逃がし、使用時に便座カバーが使用者にくっついて適所から移動するのを防止する。
Patent JP-H11500025-A (JP)
Title: 血圧を算出する方法および装置
IPC: A61B5/0245
Filed: 1995-12-01
Abstract: (57)【要約】
本発明は、パルスを有する動脈の血圧を計測する方法および装置(20)である。この方法は、変動圧力を動脈に付与することを含む。圧力波形(450)を感知して圧力波形データを生成する。波形パラメータ(510、530)は、感知した圧力波形データから求める。そして、求められたパラメータを用いて血圧を決定する。
Patent JP-2001505982-A (JP)
IPC: F16D55/00
Filed: 1997-12-08
Abstract: A disc brake comprises an operating mechanism operable to move friction material pads into contact with a disc. The operating mechanism comprises a support body located on one side of the disc, a cylinder defined by the support body, and a piston in the cylinder. The operating mechanism also comprises a guidance member for the pads. The guidance member projects from the support body past the disc and supports an abutment on which one of said pads is mounted. The guidance member is mounted on the support body by means of a plurality of bolts which extend through bores in the guidance member to said abutment. The bolts take the load during application of the brake.
Patent JP-2002512596-A (JP)
Title: 新規なカルボキシ置換された環状カルボキサミド誘導体
IPC: A61K31/495
Filed: 1997-11-21
Abstract: (57)【要約】
本発明は、式(１)
 を有する新規なカルボキシ置換された環状カルボキサミド誘導体およびその立体異性体および医薬的に許容し得る塩およびタキキニン受容体アンタゴニストとしてのこれらの化合物の使用に関するものである。このようなアンタゴニストは、喘息、咳および気管支炎を包含する明細書において説明されたタキキニン−仲介疾患および状態の治療に有用である。
Patent JP-H10500056-A (JP)
IPC: B08B15/00
Filed: 1995-04-27
Abstract: PCT No. PCT/SE95/00463 Sec. 371 Date Oct. 24, 1996 Sec. 102(e) Date Oct. 24, 1996 PCT Filed Apr. 27, 1995 PCT Pub. No. WO95/29771 PCT Pub. Date Nov. 9, 1995An electric current carrying device at an exhausting device for use in exhausting or sucking-out unhealthy gases, preferably exhausts from vehicles. At least one electric current carrying line (24 and/or 25), extending along a guide rail (4), is included in or forms part of a sealing strip (14 and/or 15).
Patent JP-2001511717-A (JP)
Title: 紫外線に対する露光による架橋結合／高密度化を使用して多層光材料を製造する方法と当該方法で製造された光材料
IPC: B32B37/00
Filed: 1998-02-06
Abstract: (57)【要約】
本発明は、各層が少なくとも１つの金属酸化物又は半金属酸化物を含み、堆積された層が紫外線に対する露光によって高密度化架橋結合される、無機ポリマー材料から成る少なくとも２つの層を基板上に堆積することによって、光学材料を製造する方法に関する。本発明はまた、本方法を用いて製造される光学材料にも関する。前記の方法を用いて製造される光学材料は、反射防止材及び反射材などの特に複数層の材料である。
Patent JP-2001513787-A (JP)
Title: アルキル−（１−アルコキシエチル）ホスフィン酸の製造方法
IPC: C07F9/30
Filed: 1998-02-20
Abstract: (57)【要約】
アルキルジクロロホスフィンをアセトアルデヒドジアルキルアセタールと反応させ、次いで反応混合物を水と反応させることにより、アルキル−（１−アルコキシエチル）ホスフィン酸を製造する。この方法は高収率を与え、簡単に実施できる。
Patent JP-H11510458-A (JP)
Title: ベルトテンショナ用点火装置駆動手段
IPC: F42B3/04
Filed: 1997-05-30
Abstract: (57)【要約】
本発明はベルトテンショナ用点火装置駆動手段に関し、前記装置はハウジング内に構成された作動室（２４）、および前記ハウジング内で移動可能でかつ推進装薬（４６）が作動室（２４）内で作動せしめられるとき上昇するガス圧によって加圧されるピストンを有する。別々にまたは同時に点火可能で、かつハウジングの別々のうけ入れ室（３２，３４）に配置された少なくとも二つの推進装薬（３６，３８）が、複数段で駆動エネルギを供給するため設けられている。二つのうけ入れ室（３２，３４）および作動室（２４）はその間に流れを生ぜしめるため連通せしめられる。
Patent JP-2002510990-A (JP)
Title: ゴルフボール用の新規な２重コア
IPC: A63B37/04
Filed: 1998-03-27
Abstract: (57)【要約】
本発明は、２重コア構成要素、内側カバー層(14)、および外側カバー層(16)を備えるゴルフボール(5)を目標とする。２重コア(10)は、熱硬化材料、熱可塑性材料、またはそれらの組み合わせから形成される、内部球状中心構成要素を備える。２重コア(10)はまた、熱硬化材料、熱可塑性材料、またはそれらの組み合わせから形成された中心構成要素の周囲に配置されたコア層を備える。内側カバー層（14）は、高酸性アイオノマーまたはアイオノマーブレンドからなる。外側カバー層(16)は、軟質の、極めて低い弾性率のアイオノマーまたはアイオノマーブレンド、もしくは、ポリウレタン、ポリエステル、またはポリエステルアミドのような非アイオノマー熱可塑性エラストマーからなる。本発明のゴルフボール(5)は、２重コア(10)を包囲する外側コア層を更に備え得る。結果として生じる本発明の多層型ゴルフボール(5)は、公知の多層ゴルフボールと比較した場合に、プレイ可能性または耐久性を犠牲にすることなく、向上した距離を提供する。
Patent JP-2000516189-A (JP)
Title: 永久磁石付きエレベータ同期モータを制御する電気駆動回路のパラメータ決定方法
IPC: H02P6/08
Filed: 1998-04-03
Abstract: (57)【要約】
永久磁石付きエレベータ同期モータを制御する電気駆動回路のパラメータ決定方法。この電気駆動回路の動作を制御するコンピュータには、エレベータを記述し設定可能なパラメータを含む制御モデルが設けられる。エレベータシャフトに設置されたエレベータカーは、エレベータの各重量の間の平衡の差によって生ずる動作状態におかれ、同期モータの端子に接続された２つの負荷を用いて、エレベータカーが一定の走行状態にあるとき、同期モータの回転速度、起電力および同期リアクタンスを測定し、また固定子抵抗を別な測定によって測定する。エレベータを記述する制御モデルをこれらの測定から算出し、形成する。
Patent JP-2001522501-A (JP)
Title: スレーブ群インターフェース装置を介して周辺機器をバスにインターフェースする方法
IPC: G06F13/38
Filed: 1999-02-04
Abstract: (57)【要約】
複数の周辺機器が、スレーブ群インターフェース装置を介してバスにインターフェースされる。これが、クロック信号、選択信号を含む制御信号及び更に情報ビットの伝送を可能にする。特に、上記装置は周辺機器読み取りデータを適宜のビット重要度レベルにしたがってオアする。書き込み制御信号がない場合、全ての周辺機器書き込みデータは重要でないレベルに維持される。周辺機器から受信される種々の制御信号は、縮小されたバス制御信号に並列に圧縮される。
Patent JP-2001521627-A (JP)
Title: サーモクロミックゲームピース
IPC: G01R31/385
Filed: 1998-04-15
Abstract: (57)【要約】
サーモクロミックゲームもしくは賞またはメッセージインジケータは、第２の導電基板に結合された第２の熱反応型ディスプレイを有する第１の導電基板に結合された通常のサーモクロミックまたは感熱型バッテリーテスターを含む。あるいは、本発明の熱反応型ゲームピースもしくは賞またはメッセージインジケータは、導電基板に結合された通常のサーモクロミックまたは感熱型バッテリーテスターを、導電基板の延長部と組み合わせる。サーモクロミックゲームもしくは賞またはメッセージインジケータは、賞が勝ち取られたかどうかを伝える言語メッセージまたはアイコンを表示するために使用され得る。さらに、サーモクロミックゲームもしくは賞またはメッセージインジケータは、所望の言語メッセージまたはアイコンを表示するために使用され得る。
Patent JP-2002504897-A (JP)
Title: ３−（ピロリジン−３−イル）−１，３，４−オキサジアゾール−２（３ｈ）−オン誘導体および５−ｈｔ４リガンドとしての使用
IPC: A61K31/454
Filed: 1998-05-04
Abstract: (57)【要約】
本発明は、一般式（Ｉ）［式中、Ｒ 1 は水素またはアルキルもしくはシクロアルキルメチル基を表し、Ｘ 1 は水素もしくはハロゲンまたはアルコキシ基を表すか、またはＯＲ 1 およびＸ 1 は一緒に式−ＯＣＨ 2 Ｏ−、−Ｏ（ＣＨ 2 ） 2 −、−Ｏ（ＣＨ 2 ） 3 −、−Ｏ（ＣＨ 2 ） 2 Ｏ−または−Ｏ（ＣＨ 2 ） 3 Ｏ−で表される基を表し、Ｘ 2 は水素原子、アミノ基または一般式−ＮＨＣＯ 2 Ｒ−［式中、Ｒはアルキルまたはフェニルアルキル基を表す］で表される基を表し、Ｘ 3 は水素またはハロゲンを表し、Ｒ 2 は水素またはアルキル、フェニルアルキルもしくは［（４−ジメチルアミノ）ピペリジン−１−イルカルボニル］アルキル基を表す］で表される化合物に関する。本発明は治療に適用可能である。この化合物を、中枢神経系、胃腸系、心臓血管系または泌尿系において５−ＨＴ４受容体が関与する障害の処置または防止に使用することができる。
Patent JP-2002500574-A (JP)
Title: ミクロメカニカルデバイスを製造する方法と装置
IPC: H01L21/308
Filed: 1999-03-16
Abstract: (57)【要約】
ミクロメカニカルデバイスを製造する方法を開示する。この方法は、（ａ）マスク（２）を有する基板を、該マスクの開口部を通じて、所望の深さまでエッチングして、基板（１）内に、側壁（４）と底面（５）を有する深溝（６）を形成し、（ｂ）前記基板とマスクとの露出表面上に、保護物質（７）層を蒸着し、（ｃ）保護物質（７）を前記底面（５）から選択的に除去し、（ｄ）フッ素含有エッチング剤を使用して、前記底面（５）をエッチングする、各ステップから成る。前記方法によって製造されるミクロメカニカルデバイス、および該ミクロメカニカルデバイスを製造する装置をも開示する。
Patent MX-149813-A (MX)
Inventor: WILKINSON RICHARD L
IPC: G11B7/26
Filed: 1981-08-11
Abstract: In a method of forming a video disc or a digital sound recording disc for example, a uniform layer of a predetermined thickness has to be applied to a substrate, and according to the invention, the layer material is applied in the form of a liquid with a known viscosity and the disc is rotated at a first velocity to spread the liquid and then the disc is rotated at a higher velocity to dry the liquid at least partly, to be in the form of a coating having a thickness which is dependent upon the viscosity of the liquid and the higher velocity at which the substrate is rotated. The method may be used is preparing a glass or other substrate for the application of a photoresist layer, or it may be used in the application of the photoresist layer, or in the application of a developer for developing an exposed photoresist layer.
Patent NZ-218020-A (NZ)
Title: Pharmaceutical compositions containing radiosensitising amounts of cobalt (iii) or iron (iii) co-ordination compounds
Inventor: ABRAMS M J
IPC: A61K33/24
Filed: 1986-10-21
Abstract: The present invention relates to radiosensitization and, more particularly, to rendering hypoxic cells more sensitive to being killed by X-rays or other forms of irradiation. In particular, the invention is directed to a pharmaceutical composition containing a radio-sensitizing amount of Co (III) or Fe (III) coordination compound selected from the group consisting of: 
 
  (1) compounds having the formula:
 [CoNnX6-n]<Y> (1)
 where n has a value of 3 or 4;
 N is an uncharged nitrogen donor atom that is contained in a ligand;
 X represents an anionic ligand; and
 Y represents the charge on the complex; 
  (2) compounds having the formula:
 (CoA2X<1>D)<Y @> (2)
 where A represents a bidentate or tetradentate negative ligand containing N or O donor atoms:
 X<1> and D represent the same or different monodentate ligands; and
 Y<1> represents a positive or negative charge on the complex; 
  (3) compounds having the formula:
 [CoZ3] (3)
 where Z represents a chelating mononegative ligand; and 
  (4) Compounds of the formula:
 [Fe TT<1>]<+> (4)
 where T and T<1>, which may be the same or different, represent mono-negative tridentate ligands. 
 
<??>The invention also includes a method for rendering hypoxic cells more sensitive to irradiation which comprises subjecting the cells to treatment using the Co (III) or Fe (III) coordination compounds defined above.
Patent NZ-218126-A (NZ)
Title: Recovery of lignin from solution
Inventor: LORA J H
IPC: D21C3/20
Filed: 1986-10-30
Abstract: Lignin is precipitated in high yields and at high rates from a black liquor produced by pulping wood at high temperatures and pressures with an aqueous lower aliphatic alcohol solvent. The lignin is precipitated by diluting the black liquor with water and an acid to form a solution with a pH of less than 3, an alcohol content of less than 30% by volume and a temperature of less than 75 DEG C. The precipitated lignin, when subsequently dried, is in the form of a powder which requires little or no crushing to convert it into a fine uniform size suitable for use without further significant processing.
Patent NZ-221565-A (NZ)
Title: Container sealing panel for use with plastic screw cap has curled edge
Inventor: MOLONEY JOHN J
IPC: B65D41/34
Filed: 1987-08-25
Abstract: A closure panel (48) for a composite closure which is formed of a corrosive metal and while the metal of the closure panel (48) is coated on both edges, in the formation thereof a raw edge (42) develops. In lieu of a straight peripheral flange (34) terminating in such raw edge (42), the peripheral flange (34) has been modified to terminate in a curl (50) with the raw edge (42) being protected by the curl (50).
Patent NZ-232144-A (NZ)
Title: Treating pre-menstral syndrome by administering melatonin and optionally progestogen
Inventor: COHEN MICHAEL
IPC: A61K31/58
Filed: 1990-01-17
Abstract: A method of alleviating climacterial menopausal and post-menopausal symptoms in females comprises administering an effective amount of a composition comprising melatonin and at least one estrogen and/or at least one androgen.
Patent NZ-268868-A (NZ)
Title: Determining meat quality of live animals by infrared imaging
Inventor: JONES STEPHEN D MORGAN
IPC: G01N33/12
Filed: 1994-06-30
Abstract: The invention provides methods of detecting poor meat quality in live animals using infrared thermography. In cattle, animals whose thermographs are predominantly outside the test temperature range, 28 DEG -32 DEG +/-2 DEG  C., are rejected as having a high probability of producing poor meat quality. In swine, the test temperature range is 24 DEG -26 DEG +/-2 DEG  C.
Patent NZ-287734-A (NZ)
Title: Preparation of n-phosphonomethylamino carboxylic acids using dialkyl phosphite
Inventor: CHENG BRIAN KAI-MING
IPC: C07F9/38
Filed: 1995-05-26
Abstract: A process for preparing N-hydroxyalkylaminomethylphosphonic acid or salts thereof which comprises contacting an alkanolamine, formaldehyde and a dialkyl phosphite in the presence of an alcohol under suitable reaction conditions to produce a reaction mixture, and hydrolyzing the reaction mixture under acidic or basic conditions. In one embodiment, the N-hydroxyalkylaminomethylphosphonic acid or salts thereof is catalytically oxidized to produce an N-phosphonomethylaminocarboxylic acid or salts thereof.
Patent NZ-302967-A (NZ)
Title: Process for preparing aza cyclohexapeptide derivatives
Inventor: BELYK KEVIN M
IPC: A61P31/12
Filed: 1996-02-06
Abstract: There is disclosed a novel process for preparing aza cyclohexapeptides of the formula (I) where all variables are defined herein.
Patent NZ-322401-A (NZ)
Title: Integrin-linked kinase, its inhibitors and methods of medical treatment using these inhibitors, gene therapy, and pseudo-substrate inhibitors
Inventor: DEDHAR SHOUKAT
IPC: A61P35/02
Filed: 1996-11-19
Abstract: This application relates to an isolated and purified serine/threonine kinase which is an integrin-linked kinase, designated "ILK".  ILK can be used to modulate cell growth, modulate cell adhesion, modulate cell migration and modulate cell invasion.  Inhibitors of ILK activity include (1) screens aimed at DNA, RNA or structural components of ILK, (2) pseudo-substrate inhibitors, such as a peptide which mimics a substrate sequence for ILK, and (3) drugs which specifically inhibit ILK activity.  The diseases treated by these inhibitors include cancer, leukemia, solid tumors, chronic inflammatory disease, arthritis, osteoporosis and cardiovascular disease.  Diagnostics of ILK activity include DNA-based reagents derived from the nucleotide sequence of ILK and antibodies against ILK screen biopsy-derived samples of amplified ILK DNA, or increased expression of ILK mRNA or protein.  Assays which screen drugs which specifically inhibit ILK activity are also included.
Patent NZ-332568-A (NZ)
Title: Recombinant antigens useful for the serodiagnosis of neosporosis
Inventor: LALLY NICOLA C
IPC: G01N33/569
Filed: 1997-04-15
Abstract: The specification describes antigens for the detection of antibodies to Neospora parasites and as such is  suitable for the diagnosis of neosporosis. Recombinant antigens may be produced by expression of DNA sequences derived from Neospora caninum. Both antigens are capable of detecting antibody responses in animals experimentally inoculated with N. caninum but show no evidence of cross-reactivity with serum from animals inoculated with closely related parasites such as Toxoplasma gondii or Sarcocystis species.
Patent NZ-334690-A (NZ)
Title: Substituted amino acid ester derivatives useful for inhibiting beta-amyloid peptide release and/or synthesis
Inventor: DROSTE JAMES J
IPC: C07K5/08
Filed: 1997-11-21
Abstract: A substituted amino acid ester derivative of formula (I) or a pharmaceutically acceptable salt thereof is used to inhibiting b-amyloid peptide release and/or its synthesis in a cell or is used to prevent the onset of Alzheimer's disease in a patient at risk of developing Alzheimer's disease wherein: R1 is optionally substituted alkyl, alkenyl, or alkynyl or is cycloalkyl, cycloalkenyl, aryl, heteroaryl or heterocyclic; R2 is hydrogen, optionally substituted alkyl, alkenyl or alkynyl or is cycloalkyl, aryl, heteroaryl or heterocyclic; each R3 is independently hydrogen or methyl or R3 together with R4 can be fused to form a cyclic structure of from 3 to 8 atoms which is optionally fused with an aryl or heteroaryl group; each R4 is independently hydrogen, optionally substituted alkyl, alkenyl, or alkynyl, or is aryl, cycloalkyl, cycloalkenyl, heteroaryl or heterocyclic; each R5 is hydrogen or methyl or together with R4 forms a cycloalkyl group of from 3 to 6 carbon atoms; X is -C(O)Y, -C(S)Y or -CR6R6Y'; Y is optionally substituted alkyl provided that the substitution does not include a-haloalkyl, a-diazoalkyl, a-OC(O)alkyl or a-OC(O)aryl or is cycloalkyl, optionally substituted alkoxy or thioalkoxy, hydroxy, aryl, heteroaryl, heterocyclic, NR'R", -NHSO2-R8, -NR9NR10R10 or NR9[C(O)O]zR10; each R6 is independently hydrogen, optionally substituted alkyl, cycloalkyl, aryl, heteroaryl or heterocyclic; Y' is hydroxyl, amino, thiol, optionally substituted alkoxy or thioalkoxy, -OC(O)R7, -S-SR7, -S-SC(O)R7; R7 is optionally substituted alkyl, cycloalkyl, aryl, heteroaryl or heterocyclic; X' is hydrogen, hydroxy, or fluoro; X" is hydrogen, hydroxy or fluoro, or X' and X" together form an oxo group; Z is a bond covalently linking R to -CX'Xn-, oxygen or sulphur; n is 1 or 2; z is 0 or 1 and R', R", R8, R9, R10 are as defined in the specification limited by the provisos listed in the specification.
Patent NZ-500667-A (NZ)
Title: Stirling refrigeration engine with oil sealing
Inventor: KOMATSUBARA TAKEO
IPC: B01F27/94
Filed: 1999-10-28
Abstract: There is disclosed a stirring device (1) in which oil rising is prevented, and an adverse influence onto oil sealing bellows (53,58) by a pressure rise accompanying the temperature rise of the crank chamber (26) is prevented. The oil sealing bellows (53,58) are disposed between a space in a housing (25,26) and compression and expansion cylinders, and a buffer tank (59,60) provided with the pressure adjusting bellows (61,62) is disposed between a space on the back surface side of the compression and expansion pistons (69,70) and the space in the housing (25,26), so that the pressure rise in the housing and the pressure fluctuation of the space are absorbed.
Patent NZ-501755-A (NZ)
Title: Use of fumaric acid derivatives for treatment of an auto-immune disease
Inventor: JOSHI RAJENDRA KUMAR
IPC: H01M6/16
Filed: 1998-04-01
Abstract: The use of one or several compounds selected from the group of sodium, potassium, calcium, magnesium, zinc and iron salts of fumeric acid monoalkyl esters of formula (1), optionally in combination with dialkyl fumerate of formula (2) wherein; A is a bivalent cation from the series containing Ca, Mg, Zn, or Fe or a monovalent cation from the series consisting of potassium or sodium respectively, and n denotes the numeral 1 or 2 depending on the type of cation, or one or several of the compounds from the series consisting of alkyl hydrogen fumerates formula (3), optionally in combination with dialkyl fumerate of formula (4), in pharmaceutical compositions. The compositions is useful in treating auto-immune diseases selected from the group consisting of polyarthritis, multiple sclerosis, graft-versus-host reactions, juvenile diabetes, Hashimoto tyroiditis, Grave's diseases, systemic Lupus erythaematodes (SLE), Sjogren's Syndrome, pernicious anaemia and chronic active (lupoid) hepatitis.
Patent NZ-504930-A (NZ)
Title: S-oxide and S-dioxide tetrahydrothiopyran phenyloxazolidinones and assay for determining inhibitory activity of oxazolidinones
Inventor: POEL TONI-JO
IPC: C07D263/20
Filed: 1998-11-23
Abstract: Described are compounds of formula (I) and formula (II) useful as antimicrobial agents wherein R1 is methyl, ethyl, cyclopropyl, or dichloromethyl; R2 and R3 are independently hydrogen or fluoro; R4 is ethyl or dichloromethyl.  Also described is an assay for determining the inhibitory activity of oxazolidinones to human monoamine oxidase.
Patent NZ-504986-A (NZ)
Title: Erythromycin and azalide derivatives and pharmaceutical compositions thereof, useful as antibacterial agents and antoprotozoa agents
Inventor: DIRLAM JOHN PHILIP
IPC: A61P31/04
Filed: 1998-12-21
Abstract: The invention relates to novel erythromycin analogs and azalides,  particularly ones with novel  C-13  substituents, and   to  pharmaceutically  acceptable  salts  thereof.  The compounds  of this invention are antibacterial  agents  that may   be  used  to  treat  various  bacterial  and  protozoa infections.  The  invention also relates  to  pharmaceutical compositions  containing such compounds and  to  methods  of treating  bacterial  protozoa  infections  by  administering such  compounds. The invention also relates  to  methods  of preparing  such  compounds and to  intermediates  useful  in such preparation.
Patent NZ-507095-A (NZ)
Title: Security screen and extrusion therefor
Inventor: BOND BRIAN PETER
IPC: E06B9/52
Filed: 2000-09-25
Abstract: A screen construction for a door frame or window frame, comprising a substantially rigid mesh (13) having a substantially rigid folded back portion (43) formed along the edge thereof at an acute angle and a frame (15) prescribing a border and support for the mesh (13).  The frame has a recess (31) formed therein into which the folded back portion (43) and mesh proximal thereto (13) is received.  The recess (31) has formed integrally therewith a means to interfere (35) with the exposed edge of the folded back portion (43) to retain the folded back portion (43) in the recess (31).  The means to interfere is formed integrally with the frame (15).  The folded back portion (43) and the mesh proximal thereto (13) is under compression when being inserted in the recess (31).
Patent NZ-512135-A (NZ)
Title: Alpha-methylbenzyl-containing thiourea inhibitors of herpes viruses containing a phenylenediamine group
Inventor: CURRAN KEVIN JOSEPH
IPC: C07D407/12
Filed: 1999-12-06
Abstract: Compounds having formula (I) that is useful in the treatment of diseases associated with herpes viruses including human cytomegalovirus, herpes simplex viruses, Epstein-Barr virus, varicella-zoster virus, human herpesviruses-6 and-7, and Kaposi herpesvirus is disclosed, wherein R1-R5 are independently selected from hydrogen, alkyl of 1 to 6 carbon atoms, alkenyl of 2 to 6 carbon atoms, alkynyl of 2 to 6 carbon atoms, perhaloalkyl of 1 to 6 carbon atoms, cycloalkyl of 3 to 10 carbon atoms, heterocycloalkyl of 3 to 10 carbon members, aryl, heteroaryl, halogen,-CN,- NO2,-CO2R6,-COR6,-OR6,-SR6,-SOR6,-SO2R6,-CONR7R8,- NR6N(R7R8),-N(R7R8) or W-Y-(CH2)n-Z provided that at least one of R1-R5 is not hydrogen; or R2 and R3, or R3 and R4, taken together to form a 3 to 7 membered heterocycloalkyl or 3 to 7 membered heteroaryl; R6 and R7 are independently hydrogen, alkyl of 1 to 6 carbon atoms, perhaloalkyl of 1 to 6 carbon atoms, or aryl; R8 is hydrogen, alkyl of 1 to 6 carbon atoms, perhaloalkyl of 1 to 6 carbon atoms, cycloalkyl of 3 to 10 carbon atoms, heterocycloalkyl of 3 to 10 members, aryl or heteroaryl, or R7 and R8, taken together may form a 3 to 7 membered heterocycloalkyl; W is O, NR6, or is absent; Y is -(CO)- or-(CO2)-, or is absent; Z is alkyl of 1 to 4 carbon atoms,-CN,-CO2R6, COR6,- CONR7R8,-OCOR6; G is phenyl optionally substituted with one or more substituents selected from alkyl of 1 to 6 carbon atoms, alkenyl of 2 to 6 carbon atoms, alkynyl of 2 to 6 carbon atoms, perhaloalkyl of 1 to 6 carbon atoms, cycloalkyl of 3 to 10 carbon atoms, heterocycloalkyl of 3 to 10 carbon members, aryl, heteroaryl, halogen,-CN,-NO2,-CO, R6,-COR6,- OR6,-SR6, -SOR6, -SO2R6, -CONR7R8, -NR6N(R7R8), -N(R7R8) or W-Y- (CH,),-Z or G is quinolyl, isoquinolyl or benzofuranyl; X is (CH)J; J is alkyl of 1 to 6 carbon atoms, cycloalkyl of 3 to 7 carbon atoms, phenyl or benzyl; and n is an integer from 1 to 6.
Patent NZ-513136-A (NZ)
Title: Method for obtaining an oil that is rich in hydroxyoctadecadienoic fatty acids (HODE) or the esters thereof from a mixture containing linoleic or linolenic acid or the esters thereof, and compositions thereof containing 9-HODE
Inventor: ROMBI MAX
IPC: A23L33/20
Filed: 2000-01-28
Abstract: A process for obtaining an oil that is enriched in hydroxyoctadecadienoic (HODE) fatty acid or esters thereof from an oily mixture containing linoleic acid or esters thereof, wherein a controlled oxidation of linoleic acid and/or linolenic acid is carried out in the presence of an oxidation catalyst, the oxidation being stopped when the total content of HODE is greater than 5% and/or the content of 9-hydroxy-10,12-octadecadienoic acid (9-HODE) is greater than 1.5%, and in that the hydroperoxides formed during the oxidation reaction are reduced with a reducing agent.  Also covered is the use of said oil in the preparation of a medicament for the treatment of obesity.