baber/WOPTO huggingface dataset:
Patent CO-5601020-A2 (CO)
Title: Compuestos ox-azabiciclicos
Inventor: GAUDILLIERE BERNARD
IPC: C07D471/04
Filed: 2004-08-25
Abstract: 1.- Un compuesto seleccionado de aquellos de la fórmula (I):caracterizado porque:? X1, X2 y X3, independientemente uno de otro, representan un átomo de nitrógeno o un grupo -CR3 en donde R3 representa un grupo seleccionado de hidrógeno, alquilo (de C1-C6), amino, monoalquilamino (de C1-C6), dialquilamino (de C1-C6), hidroxi, alcoxi (de C1-C6) y halógeno, con la condición de que no más de dos de los grupos X1, X2 y X3 simultáneamente representen un átomo de nitrógeno,? G1 representa un grupo seleccionado de aquellos de lasfórmulas (i/a) e (i/b): en donde:- el átomo de carbono con el número 2 está unido al grupo N-R1 del anillo,- R4 y R5, idénticos o diferentes, independientemente uno de otro, representan un grupo seleccionado de hidrógeno, alquilo (de C1-C6), arilo, arilalquilo (de C1-C6), cicloalquilo, cicloalquilalquilo (de C1-C6), heteroarilo, heteroarilalquilo (de C1-C6), heterocicloalquilo, y heterocicloalquilalquilo (de C1-C6),- R4 representa un grupo seleccionado de: hidrógeno, trifluorometilo, OR7, NR7R8, en donde R7 y R8, idénticos o diferentes independientemente uno de otro, representan hidrógeno o alquilo (de C1-C6), alquilo (de C1-C6), alquenilo (de C2-C6), alquinilo (de C2-C6), arilo, arilalquilo (de C1-C6), cicloalquilalquilo (de C1-C6), heteroarilo, heteroarilalquilo (de C1-C6), heterocicloalquilo, y heterocicloalquilalquilo (de C1-C6), estos grupos son optativamente sustituidos por uno o más grupos, que pueden ser idénticos o diferentes independientemente uno de otro, seleccionados de halógeno, amino, monoalquilamino (de C1-C6), dialquilamino (de C1-C6), cada grupo alquilo es idéntico o diferente independientemente uno de otro, ...
Patent CO-5570701-A2 (CO)
Title: Activadores de ppar
Inventor: DUGGER ROBERT WAYNE
IPC: A61K31/4545
Filed: 2005-05-19
Abstract: 1.- Un compuesto de Fórmula I un isómero del mismo, un profármaco de dicho compuesto o isómero, o una sal farmacéuticamente aceptable de dicho compuesto, isómero o profármaco;en el que m y n son, cada uno independientemente, uno o dos;V e Y son, cada uno independientemente, a) metileno, o b) carbonilo;F y G son, cada uno independientemente, a) hidrógeno, b) halo, c) alquilo (C1-C4) sustituido opcionalmente con de uno a nueve átomos de flúor, d) cicloalquilo (C3-C6); e) hidroxi, f) alcoxi (C1-C4) o g) alquiltio (C1-C4);X es a) -Z o b) -B-C(R1R2)-Z;B es a) oxi, b) tio, c) sulfinilo,d) sulfonilo, e) metileno, o f) -N(H)-;Z es a) -C(O)OH, b) -C(O)O-alquilo (C1-C4), c) -C(O)O-alquil (C0-C4)arilo, d) -C(O)-NH2, e) hidroxiaminocarbonilo, f) tetrazolilo, g) tetrazolilaminocarbonilo, h) 4,5-dihidro-5-oxo-1,2,4-oxadiazol-3-ilo, i) 3-oxoisoxazolidin-4-il-aminocarbonilo, j) -C(O)N(H)SO2R4, o k) -NHSO2R4; en el que R4 es a) alquilo (C1-C6), b) amino o c) mono-N o di-N,N-alquil (C1-C6) amino, estando los sustituyentes alquilo (C1-C6) en R4 opcionalmente e independientemente sustituidos con de uno a nueve átomos de flúor;R1 es a) H, b) alquilo (C1-C4) o c) cicloalquilo (C3-C6);R2 es a) H, b) cicloalquilo (C3-C6) o c) una cadena de carbono de uno a cuatro miembros, lineal o ramificada, total o parcialmente saturada o totalmente insaturada; en la que el(los) carbono(s) de la cadena de carbono pueden reemplazarse con uno o dos heteroátomos seleccionados independientemente entre oxígeno y azufre; y en la que el azufre está opcionalmente mono o disustituido con oxo;en la que el(los) carbono(s) de la cadena de carbono de R2 están opcionalmente sustituidos independientemente como sigue: a) el(los) carbono(s) están opcionalmente mono, di o trisustituidos independientemente con halo, b) el(los) carbono(s) están opcionalmente monosustituidos con hidroxi o alcoxi (C1-C4), y c) el (los) carbono(s) están opcionalmente monosustituidos con oxo; y en la que el(los) carbono(s) de la cadena de carbono de R2 están opcionalmente monosustituidos con Q;en la que Q es un anillo de tres a ocho miembros, parcial o totalmente saturado o totalmente insaturado, que tiene, opcionalmente, de uno a cuatro heteroátomos seleccionados independientemente entre oxígeno, ...
Patent CO-6361969-A2 (CO)
Title: Tinta orientada magnéticamente en una capa de imprimación
Inventor: DESPLAND CLAUDE-ALAIN
IPC: B42D15/00
Filed: 2011-05-16
Abstract: Se divulga documento de seguridad (D), que tiene un sustrato (S), recubierto con al menos una primera capa de recubrimiento (P) y sobre dicha primera capa de recubrimiento (P) al menos una segunda capa de recubrimiento (I), comprendiendo dicha segunda capa de recubrimiento (i) al menos un tipo de partículas magnéticas o magnetizables (F), en el que los indicios se realizan en la capa de recubrimiento (I) mediante una orientación selectiva de las partículas magnéticas o magnetizables (F). Se divulga además un proceso de fabricación de dicho documento de seguridad.
Patent CO-6420344-A2 (CO)
Title: Derivados de triazolopiridina como inhibidores de proteínas cinasas activadas por mitogeno p38 (map)
Inventor: FINCH HARRY
IPC: C07D471/04
Filed: 2011-08-16
Abstract: La presente invención se refiere a compuestos de fórmula (I) que son inhibidores de cinasa p38 MAP, útiles como agentes anti-inflamatorios en el tratamiento de, entre otros, enfermedades del tracto respiratorio en donde; R1 es alquilo C1-C4, cicloalquilo C3-C6, fenilo el cual es opcionalmente sustituido, heteroarilo monocíclico de 5 o 6 elementos el cual es opcionalmente sustituido, o un radical de fórmula (II) en donde n es 1 o 2, y R3 y R4 son independientemente H o alquilo C1-C4, o R3 y R4 tomados junto con el nitrógeno al cual están unidos forman un anillo heterociclico de 6 elementos opcionalmente que contiene un heteroátomo adicional seleccionado de N y O; Y es -O- o - S(O)p- en donde p es 0, 1 o 2; A es un radical arileno divalente opcionalmente sustituido, o un radical heteroarileno mono- o bicíclico, o un radical cicloalquileno nt divalente C3-C6 que tiene 5 o 6 átomos de anillo, o un radical piperidinileno en donde el nitrógeno del anillo se enlaza a R2NHC(=O)W-; W es un enlace, -NH- o -C(RA) (RB), en donde RA y RB son independientemente H, metilo, etilo, amino, hidroxilo o halo; y R2 es un radical como se define en las reivindicaciones.
Patent CO-6460750-A2 (CO)
Title: Fracturamiento con miembros telescópicos y sellado del espacio anular
Inventor: RICHARD BENNETT M
IPC: E21B43/10
Filed: 2011-11-11
Abstract: Se realiza una operación de fracturamiento en un agujero abierto. Se atraviesa el espacio anular mediante miembros telescópicos que se ubican detrás de las válvulas de aislamiento. Se puede destapar un banco dado de miembros telescópicos y estos miembros telescópicos se extienden para atravesar el espacio anular y ajustar la formación en una forma sellada. El fluido de fracturamiento presurizado se puede bombear a través de los pasajes telescópicos y la porción de la formación fracturada deseada. En una formación apropiada, no se necesita aplicar concreto para mantener la integridad del pozo. En formaciones que necesitan aislamiento de espacio anular, la columna en una realización preferida puede tener un material externo que crece para sellar el espacio anular en lugar de una operación de aplicación de concreto tradicional.
Patent CO-6460735-A2 (CO)
Title: Placa de comprensión con ángulo variable
Inventor: KOAY KENNY
IPC: A61B17/80
Filed: 2012-03-14
Abstract: Una placa para huesos comprende una primer superficie y una segunda superficie en combinación con un primer agujero que se extiende por la placa para huesos desde la primera superficie hasta la segunda superficie, el agujero incluye una porción de compresión y una porción de ángulo variable, abiertas una respecto de la otra mediante un espacio de conexión. La porción de compresión incluye una superficie inclinada adaptada para acoplar una cabeza de un elemento de fijación del hueso insertado allí de modo que el elemento de fijación del hueso imparte una fuerza a la placa para huesos para moverla lateralmente con relación a una porción de hueso dentro de la cual se inserta el elemento de fijación del hueso. La porción de ángulo variable incluye una pluralidad de columnas posicionadas alrededor de una circunferencia de una pared de la porción de ángulo variable. Las columnas están separadas una de otra por una pluralidad de espacios posicionados entre pares adyacentes de columnas e incluyen una pluralidad de protrusiones que se extienden radialmente hacia adentro de esta.
Patent CO-6602112-A2 (CO)
Title: Derivados de 5.6- dhidro-2h -[1.4]oxazin-3-il amina utiles como inhibidores de la betasecretasa(bace)
Inventor: TRABANCO SUAREZ ANDRES AVELINO
IPC: C07D265/30
Filed: 2012-11-29
Abstract: La presente invención se refiere a derivados novedosos de 5,6-dihidro-2H-[1,4]oxazin-3-ilamina como inhibidores de la beta-secretasa, también conocida como enzima de escisión amiloide del sitio beta, BACE, BACE1, Asp2, o memapsina2. La invención también se refiere a composiciones farmacéuticas quecomprenden dichos compuestos, a procesos para la preparación de dichos compuestos y composiciones, y al uso de dichos compuestos y composiciones para la prevención y el tratamiento de trastornos en los cuales se encuentra involucrada la beta-secretasa, tal como la enfermedad de Alzheimer (EA), deterioro cognitivo leve, senilidad, demencia, demencia con cuerpos de Lewy,Síndrome de Down, demencia asociada con el accidente cerebro vascular, demencia asociada con la enfermedad de Parkinson y demencia asociada con beta-amiloide.
Patent CO-6620013-A2 (CO)
Title: Anticuerpos hacia gdf8 humano
Inventor: STITT TREVOR
IPC: A61K39/395
Filed: 2012-12-26
Abstract: La presente invención proporciona anticuerpos humanos o humanizados aislados o fragmentos de unión al antígeno de de los mismos que se unen de manera específica al factor8 de crecimiento y diferenciación (GDF8) y bloquean la actividad de GDF8. Los anticuerpos y fragmentos de anticuerpo de la presente invención se pueden usar en métodos terapéuticos para tratar enfermedades o trastornos que son aliviados o mejorados por la inhibición de GDF8.
Patent CO-7151512-A2 (CO)
Title: Inhibidores del nampt
Inventor: CLARK RICHARD F
IPC: C07D471/14
Filed: 2014-12-03
Abstract: VER ANEXOS
Patent EP-1026913-A2 (EP)
Inventor: PRIETO JAIME L
IPC: H04B7/185
Filed: 2000-01-13
Abstract: A mapping scheme that maps standard ATMs service classes (28) of the type
used in a wired communications network into one of a plurality of available media access
control channels (30) that allow the particular ATM service class (28) to be transmitted
efficiently over the network, such as a satellite network. The various media access
controlled channel types (30) reside in a media access control layer (24) between the
ATM layer (22) and the physical layer (26). A predetermined uplink user protocol is
assigned to each MAC channel 30 to efficiently transmit to the ATM cells on the satellite
uplink.
Patent EP-1039156-A2 (EP)
Inventor: ACHLER RAINER
IPC: F16B33/00
Filed: 2000-02-24
Abstract: The protective cap (4) for the end of a bolt (5) fastened by a nut (2) has a sealing lip (7) which is thinner than the remaining walls of the cap. The cap is made of closed-cell thermoplastic foam and is held on to the bolt by its resilience.
Patent EP-1035583-A2 (EP)
Inventor: HOMMA SOICHI
IPC: H01L23/485
Filed: 2000-03-09
Abstract: The present semiconductor element comprises a
semiconductor substrate, a wiring pad formed thereon, a layer
of barrier metal formed thereon, an intermetallic compound
Ag 3 Sn formed thereon, and a protruded electrode consisting of
low-melting metal formed thereon. In addition, a fabricating
method of a semiconductor element comprises the steps of
forming a wiring pad on a semiconductor substrate, forming a
layer of barrier metal thereon, forming a metallic layer
containing Ag thereon, forming a layer of low-melting metal
containing Sn thereon, and melting the layer of low-melting
metal containing Sn to form a protruded electrode and
simultaneously to form an intermetallic compound Ag 3 Sn at an
interface between the metallic layer containing Ag and the
layer of low-melting metal containing Sn. Thus, with Pb-free
solder, a semiconductor element of high reliability can be
obtained.
Patent EP-1037138-A2 (EP)
Inventor: TERADAIRA MITSUAKI
IPC: G06F3/12
Filed: 2000-03-17
Abstract: This invention relates to a printer, an information processing apparatus, control methods for the
printer and the information processing apparatus, and a storage medium. The printer is
connected to the information processing apparatus to receive a predetermined command and a
data stream composed of data or the like for carrying out printing and predetermined processing
corresponding to the command. In the printer, a receiver receives a data stream including a
normal command and/or a real-time command. When the data stream received by the receiver is
a real-time command data stream and when an indication device, provided to give an indication
as to whether or not the real-time command is to be executed, indicates permission for the real-time
command, a real-time processing section executes real-time processing corresponding to the
real-time command data stream. Otherwise, a normal processing section executes normal
processing corresponding to the normal command data stream without carrying out the real-time
processing.
Patent EP-1008869-A2 (EP)
Inventor: SAGAR BRIAN
IPC: C09D7/12
Filed: 1994-11-17
Abstract: There is disclosed the use, in the preparation of a liquid-based, pigment or
dye-containing retroreflective medium, of retroreflective beads or microspheres separated
from a substrate coated with an adhesive in which the beads or microspheres are partially
embedded and partially exposed with the exposed surfaces of the beads or microsphere
being coated with a reflective material.
Patent EP-1038645-A2 (EP)
Inventor: EISENBACH BERND
IPC: B27G5/02
Filed: 2000-03-27
Abstract: The method is for cutting of acute, obtuse, and right angles (30) in glass battens (5,6). A clamping device (8) has two clamping plates (11,12). The plates each engage on one profile leg forming a frame corner, in a position corresponding to the angle of that corner, and are relatively aligned and locked in that position. A finishing device (23), esp. a machine table is associated with the clamping device, and has a saw or similar cutting device. The clamping device is locked in a position defined relative to the saw. A batten is placed on each clamping plate at different vertical levels, and an angled cut is made by the saw through the battens.
Patent EP-1045332-A2 (EP)
Inventor: KAZOU OSAMU
IPC: B65H1/26
Filed: 2000-04-14
Abstract: A card cassette of the present invention comprises an
outer box (1),an inner box (2), a shutter (3) which is pivotably
provided in the inner box and is urged by a pair of shutter
springs (6), a pair of slide guide members (4), a pair of slide
springs (5) for urging the slide guide members. A pair of
pins (11) are fixed on a table on which the card cassette is
to be set. As soon as the card cassette is mounted on the
table, the pins will be inserted through a pair of pin
holes (8) of the outer box so that each pin can engage into a
notch (4a) of a slide guide member. In this way, each slide
guide member is caused to slide in a direction shown by an
arrow in the drawings against an acting force of each slide
spring. As a result, since an inclined surface (4b) of each
slide guide member is released from the shutter, the
shutter will be opened by virtue of each shutter spring.
Patent EP-1067451-A2 (EP)
Inventor: GOLDBERG DAVID
IPC: G06F3/041
Filed: 2000-07-06
Abstract: The invention relates
to a method, executed on a processor, for entering symbols into a user
interface, comprising:
   providing a surface actuated when contacted with a pointing device and
positioned in relationship to at least one selectable button;   receiving stroke information in response to a stroke made by a pointing
device on the surface of the user interface (106) and in relationship to at least one
selectable button on the user interface (106);   identifying a symbol based on the stroke information; and   providing the symbol for further processing.
Patent EP-1069358-A2 (EP)
Inventor: HIRATA ICHIRO
IPC: F16K31/06
Filed: 2000-07-12
Abstract: A solenoid-side rod 5c, a bellows-side rod 5e and a
valve 3b are formed as a valve rod 5 in the form of a
unitary structure. The valve rod 5 is connected to a
plunger 2b. The valve rod 5 is slidably supported at two
points at portions corresponding to the bellows-side rod
5e and the plunger 2b.
Patent EP-1075872-A2 (EP)
Inventor: TOMIMATSU KAZUTAKA
IPC: B03C3/38
Filed: 2000-08-09
Abstract: There are provided a dust collector and method for collecting
dust in which the rarefaction of a dielectric at the rear part of electric
field forming means is prevented, whereby the collecting efficiency
can be increased. 
     The dust collector includes charging means 1 for charging a
substance to be collected 9, such as dust and mist, contained in a
gas; spray means 2 for spraying a dielectric 10 on the substance to
be collected 9 charged by the charging means 1; electric field forming
means 3, having first and second electrodes 11 and 12 for forming a
direct current electric field, for dielectrically polarizing the
dielectric 10 sprayed by the spray means 2 by means of the direct current
electric field; and dielectric collecting means 16 for collecting the
dielectric 10 which has arrested the substance to be collected 9, the
spray means 2 being provided with grounding means 17 and 18 for
electrically grounding the dielectric 10 before being sprayed to let
a charge of the dielectric 10 escape.
Patent EP-1101654-A2 (EP)
Inventor: LENT-PHILIPPS HANS-MARTIN DR
IPC: B60Q3/04
Filed: 2000-10-20
Abstract: In order to provide easy operation quickly and reliably while driving in the dark and in a dark passenger area, the driver relies on a signal from a proximity switch (3) that switches on lighting devices (2) fitted near to an instrument panel, so that the hand performing an operation is lit up during the performance of that operation.
Patent EP-1103437-A2 (EP)
Inventor: HASELSTEINER KURT
IPC: B60T13/66
Filed: 2000-11-24
Abstract: Brake test device has a central brake testing device (1) and an auxiliary unit (10) for connection to the vehicle brakes. The vehicle is connected to the auxiliary connection via a connection (22), while the auxiliary unit is connected to the central unit via a further connection (24). The auxiliary unit includes a piston valve and solenoid for shutting of air supply to the vehicle. The auxiliary unit also includes a pressure sensor. An Independent claim is made for a method for testing rail borne vehicles which allows selection of one of three test functions: leak testing, braking and activating.
Patent EP-1028473-A2 (EP)
Inventor: BLANCHARD RICHARD A
IPC: H01L29/10
Filed: 1996-05-08
Abstract: A low-voltage high-current discrete insulated-gate field-effect
transistor which is made by a very economical process with two silicon
etches. A buried poly gate gates conduction along a trench sidewall.
The channel is provided by the residuum of an epi layer, and the
source diffusion is provided by an unmasked implant which is screened
only by various grown oxides.
Patent EP-1069596-A2 (EP)
Inventor: WESTEMEYER MANFRED
IPC: H01J61/16
Filed: 2000-07-06
Abstract: The external electrode, or antenna, can take the form of a metallic concentric or spiral winding (24) located outside, on the inner surface of the lamp outer envelope (14) or molded into the envelope. It is connected to the return electrode (20) of the discharge vessel (16)
Patent EP-1028604-A2 (EP)
Inventor: KERCHNER LYNN L
IPC: F24C7/02
Filed: 2000-01-19
Abstract: A domestic cooking or defrosting appliance including a heating region and a camera
for obtaining images of food cooking or defrosting within the heating region, wherein
the camera outputs video signals to a processor that drives a display means associated
with the appliance and/or controls the cooking or defrosting operation of the
appliance. The display means is conveniently situated on the appliance to show an
easily-viewable image of the food obtained by the camera. 
     The camera is sensitive to infra-red radiation and outputs video signals representative
of the heat of the food. The processor can therefore convert infra-red information
received from the camera into visible information to create a display on the display
means representative of the infra-red information. Such a display is preferably colour-coded
in accordance with the local temperature of the food. 
     The appliance (1) is adapted for interaction with a communications network (75) such
as the Internet by the addition of a substantially self-contained discrete
communications module (12) connectable to the communications network (75), the
communications module (12) including display means (20) and command entry
means that optionally interact with the appliance (1).
Patent EP-1085656-A2 (EP)
Inventor: DEN XIAOWEI
IPC: H03K19/096
Filed: 2000-09-18
Abstract: CMOS semiconductor dynamic logic (300) is disclosed,
comprising dynamic logic circuitry (302) and tunneling structure
circuitry (328) coupled to the dynamic logic circuitry; where
the tunneling structure circuitry is adapted to hold a node
(308) voltage stable by compensating leakage current originating
from said dynamic logic circuitry.
Patent EP-1113605-A2 (EP)
Inventor: DEARMOND CURTIN STEVEN
IPC: G10L19/00
Filed: 2000-11-13
Abstract: Identification information is extracted from a current broadcast of a piece or music
or other type of information of interest to a user, and stored in a memory or other storage
device, in response to a user command. The identification information includes sufficient
information to identify at least one deliverable information item associated with the current
broadcast, e.g., a CD or MP3 file which contains the particular piece of music. When the user
later has access to a wired or wireless network connection, the extracted identification
information is delivered over a network connection to a server which processes the delivered
information to identify the deliverable information item associated with the broadcast. The
user can then purchase the deliverable information item by appropriate interaction with the
server. The extracted identification information may be stored in a removable memory device
associated with a receiver which receives the broadcast. In this case, the removable memory
device is subsequently removed from the receiver and inserted into another device which
establishes the network connection for delivery of the identification information to the server.
Patent EP-1160072-A2 (EP)
Inventor: MIYAO MAKIJI
IPC: B29C70/22
Filed: 2000-11-16
Abstract: The present invention provides a continuous reinforcing
fiber sheet, in which reinforcing fibers are arranged at an arbitrary
angle to the main axis, well applicable to pultrusion forming
without the risk of the reinforcing fibers being dispersed, which
permits the manufacture of a long fiber reinforced plastic
structural member having a remarkably improved torsional rigidity.
The continuous reinforcing fiber sheet (1) has a continuous resin-penetrable
support sheet (2), and a reinforcing fiber layer (3) held by
the resin-penetrable support sheet (2), in which long reinforcing
fibers (4) having substantially a certain length (F) are arranged in
the longitudinal direction of the resin-penetrable support sheet (2)
at a prescribed angle (α) to the longitudinal direction of the
resin-penetrable support sheet (2).