baber/WOPTO huggingface dataset:
Patent ZA-893140-B (ZA)
Title: Substituted 1-(1h-imidazol-4-yl)alkyl-benzamides
Inventor: COSSEMENT ERIC
IPC: C07D233/64
Filed: 1989-04-27
Abstract: New substituted 1-(1H-imidazol-4-yl)alkyl-benzamides and their salts, processes for the preparation thereof and pharmaceutical compositions. These compounds have the formula  <IMAGE>  wherein R1, R2=hydrogen or C1-C4-alkyl, R3=hydrogen, amino, hydroxyl, C1-C4-alkyl or C1-C4-hydroxyalkyl, R4=hydrogen or C1-C4-alkyl, or R3R4N=pyrrolidino, piperidino or morpholino, R5 and R6=hydrogen, hydroxyl, C1-C4-alkyl or C1-C4-alkoxy, at least one of R5 and R6 being other than hydrogen. These compounds are prepared either by reacting a nitrogen compound with an alkyl 1-(1H-imidazol-4-yl)alkyl-benzoate or with a 1-(1H-imidazol-4-yl)alkyl-benzoic acid, or by hydrolyzing in an acid medium a 2-hydroxy-3-[1-(1H-imidazol-4-yl)alkyl]-benzonitrile. The compounds have anti-ischemic and  alpha 2-adrenoceptor agonist activities.
Patent ZA-894145-B (ZA)
Title: Serotonin antagonists
Inventor: BEEDLE EDWARD EARL
IPC: A61K31/44
Filed: 1989-06-01
Abstract: This invention provides a method of selectively antagonizing the 5-HT1 receptor in mammals by administering aryloxypropanolamines. Novel aryloxypropanolamines are also claimed.
Patent ZA-906307-B (ZA)
Title: 4-substituted 18beta-(cyclopropyloxy)androst-5-en-3beta-ol and related compounds useful as c17-20lyase inhibitors
Inventor: ANGELASTRO MICHAEL RICHARD
IPC: A61K31/56
Filed: 1990-08-09
Abstract: This invention is directed to 4-substituted 17 beta -(cyclopropyloxy)androst-5-en-3 beta -ols and related compounds and also to a method for using such compounds in the treatment of androgen-dependent disorders. The ethers are prepared by using the Simmons-Smith reaction and an appropriate vinyl ether.
Patent ZA-921369-B (ZA)
Title: Novel poly-iodinated compounds, process for their preparation, contrast medium containing them.
Inventor: DUGAST-ZRIHEN MARYSE
IPC: C07C/
Filed: 1992-02-25
Abstract: The subject of the invention is new polyiodinated compounds of general formula: <IMAGE> in which R1, R2, R3, R4, R5, R6, R7, R8, R9 and R10, which are identical to or different from each other, are chosen from an iodine atom, a group of formula <IMAGE>  and a group of formula <IMAGE> with the proviso that at least two groups from R1, R2, R3, R4, R5, R6, R7, R8, R9 and R10 represent an iodine atom, which can be used in contrast agents for radiography. Another subject of the invention is a process for the preparation of these compounds as well as a contrast agent containing them.
Patent ZA-921404-B (ZA)
Title: Cycloolefin(co)polymers with a narrow molecular weight distribution and a process for the preparation thereof
Inventor: BREKNER MICHAEL-JOACHIM
IPC: C08F32/08
Filed: 1992-02-26
Abstract: Polymers of polycyclic olefins, such as, for example, norbornene or tetracyclododecene, or copolymers of polycyclic olefins with cycloolefins and/or 1-olefins, having a very narrow molecular weight distribution are obtained without ring opening by polymerisation in which a catalyst is used which comprises an aluminoxane and a stereorigid, chiral metallocene compound of an element from group IVb to VIb, and in which the reaction is terminated at the point when the molecular weight distribution Mw/Mn of the resultant polymer is < 2.
Patent ZA-924219-B (ZA)
Title: Direct-current arc furnace plant
Inventor: STENKVIST SVEN-EINAR
IPC: F27B3/08
Filed: 1992-06-10
Abstract: In direct-current arc furnace the arc is deflected in a direction away from the current supply means (19) through the action of the high-current lines (18) extending under the furnace vessel. This leads to the thermal overloading of a part of the furnace vessel walls. If the high-current lines (18a) are for the major part laid in a plane above the furnace bottom, on or below the furnace platform (20), and are taken downwards to the connection fittings (10) on the furnace bottom only on the side of the furnace vessel (1) opposite the current supply means, the arc will again burn symmetrically.
Patent ZA-931250-B (ZA)
Title: Compounds which can be used in contrast products for radiography
Inventor: BENNANI FATIMA-ZARHA
IPC: C07D207/12
Filed: 1993-02-23
Abstract: The subject of the invention is polyiodinated non-ionic compounds of general formula: <IMAGE>  in which:     R1 represents a group chosen from <IMAGE>     R2 represents a group chosen from -COR1 and <IMAGE>     These compounds are useful in contrast agents for radiography.
Patent ZA-935829-B (ZA)
Title: Method for combating insects and agents for combating insects.
Inventor: BERTRAM HEINZ-JUERGEN
IPC: A01N37/02
Filed: 1993-08-11
Abstract: The present invention relates to the novel use of butyric acid and of butyric acid in the form of a mixture with other substances as an attractant in the control of insects, and to insect-control devices and compositions which contain butyric acid and butyric acid in the form of a mixture with other substances as an attractant for insects.
Patent ZA-942957-B (ZA)
Title: Blow molded plastic container including handgrip
Inventor: VALYI EMERY L
IPC: B65D1/00
Filed: 1994-04-28
Abstract: A blow molded plastic container (40) including a supporting member (50) in the hollow space of the container extending completely across the hollow space and integral with the inside wall face of the body portion of the container at two spaced locations thereof to support the inside wall face. The body portion defines regions that comprise at least two adjoining lobes (60) which form a handgrip, at least one of said lobes including segments (53) deformed under internal pressure into the configuration (55) of said handgrip. <IMAGE>   <IMAGE>
Patent ZA-959613-B (ZA)
Title: System for monitoring a continuous manufacturing process
Inventor: RUDT ROBERT J
IPC: G06T7/20
Filed: 1995-11-13
Abstract: This invention relates to a system for monitoring a process which includes a plurality of monitoring means such as video camera which collects data relative to the process. The collected data is converted into a digital format and the digitized data stored in digital data storage device such that as new data is stored earlier stored data is removed to maintain about the same volume of stored data. The system also includes a control such as a computer which communicates with the digital data storage device. In the event of a deviation from a process parameter, the control is adapted to extract and display the digitized data corresponding to the deviation.
Patent ZA-961364-B (ZA)
Title: 1-Aryl-2-acylamino-ethane compounds
Inventor: GERSPACHER MARC
IPC: C07D211/44
Filed: 1996-02-21
Abstract: PCT No. PCT/EP96/00555 Sec. 371 Date Aug. 21, 1997 Sec. 102(e) Date Aug. 21, 1997 PCT Filed Feb. 9, 1996 PCT Pub. No. WO96/26183 PCT Pub. Date Aug. 29, 19961-Aryl-2-acylaminoethane compounds of formula I wherein R1-R4, X and Am are as defined in the description, have valuable pharmaceutical properties and are especially effective as NK-1 antagonists.
Patent ZA-971231-B (ZA)
Title: Quinazoline derivatives.
Inventor: BARKER ANDREW JOHN
IPC: C07D409/12
Filed: 1997-02-13
Abstract: The invention concerns quinazoline derivatives of the formula I wherein X<SUP>1 </SUP>is a direct link or a group such as CO, C(R<SUP>2</SUP>)<SUB>2 </SUB>and CH(OR<SUP>2</SUP>); wherein Q<SUP>1 </SUP>is phenyl, naphthyl or a 5- or 6-membered heteroaryl moiety and Q<SUP>1 </SUP>optionally bears up to 3 substituents; wherein m is 1 or 2 and each R<SUP>1 </SUP>may be a group such as hydrogen, halogeno and trifluoromethyl; and wherein Q<SUP>2 </SUP>may be phenyl or a 9- or 10-membered bicyclic heterocyclic moiety and Q<SUP>2 </SUP>optionally bears up to 3 substituents; or a pharmaceutically-acceptable salt thereof; processes for their preparation, pharmaceutical compositions containing them and the use of their receptor tyrosine kinase inhibitory properties in the treatment of proliferative disease such as cancer.
Patent ZA-973822-B (ZA)
Title: Hand-held smoker's device for sidestream smoke control.
Inventor: BOWEN LARRY
IPC: A24F13/08
Filed: 1997-05-02
Abstract: PCT No. PCT/CA97/00297 Sec. 371 Date Sep. 26, 1999 Sec. 102(e) Date Sep. 26, 1999 PCT Filed May 2, 1997 PCT Pub. No. WO97/41744 PCT Pub. Date Nov. 13, 1997A cigarette combustion unit for the use in a hand-held cigarette smoke filtering device for filtering sidestream smoke emitted from a cigarette burning in the unit comprising: i) an elongate closed combustion chamber for a burning cigarette, a lower wall portion of the combustion chamber at least having an air porous portion to permit air to enter the combustion chamber, ii) a cigarette holder in an end of the combustion chamber for holding a cigarette in the combustion chamber with its burning end spaced from chamber interior wall surfaces, and iii) a sidestream smoke outlet in the end above the cigarette holder.
Patent ZA-986330-B (ZA)
Title: Medicaments comprising at least one substituted derivative of polyhydroxyalkypyrazines new derivatives and their preparation.
Inventor: BOUCHARD HERVE
IPC: A61K31/495
Filed: 1998-07-16
Abstract: Provided herein are novel polyhydroxyalkylpyrazine derivatives useful in treating and preventing a plethora of diseases including diabetes, having a general formula ofwherein Rc1 represents the chain (II) -CH(OR4)CH(OR3)CH(OR2)CH2OR1 and either Rc2 represents a hydrogen atom and either Rc3 represents the chain (III)-CH2CH(OR6)CH(OR7)CH2OR8 or Rc2 represents the chain (IV)-CH(OR5)CH(OR6)CH(OR7)CH2OR8 or chain (III) -CH2CH(OR6)CH(OR7)CH2OR8 and Rc3 represents a hydrogen atom, and 1 to 8 substituents R1, R2, R3, R4, R5, R6, R7, R8, identical or different, represent a radical independently selected among the radicals a) -COR9, b) -COOR10, c) -CR11R12OCOR13, d) -CR11R12OR13, e) -CONR14R15, and f) one or more pairs of the substituents R1, R2, R3, R4, R6, R7, R8, consecutive or separated by one of the other substituents R2, R3, R6, R7 can also form a group: -C(O)-; the other substituents R1, R2, R3, R4, R6, R7, R8 are hydrogen atoms.
Patent GB-2433813-B (GB)
Title: Distributed processing system
Inventor: ANDERSON ROBERT W
IPC: G06F9/50
Filed: 2005-10-06
Granted: 2009-07-08
Abstract: A distributed object execution system delegates the allocation and control of computing tasks to intelligent agent applications running on computing resources. User applications can invoke object methods associated with an application interface of the distributed object execution system. The system converts this method invocation into an available computing job with at least one computing tasks. The agents assess computing resources capabilities to perform available computing tasks. Based on these assessments, agents request jobs from a job server, which in turn assigns computing tasks to computing resources based on the job requests received. An agent instantiates a replica of the object and invokes a corresponding method on an associated computing resource. Upon completion of the invoked method, the user application is notified and provided with any method results. While an agent and associated computing resource is processing a method invocation, the user application can perform other activities.
Patent GB-2044596-B (GB)
Title: Method and apparatus for expanding tobacco
IPC: A24B3/18
Filed: 1980-02-12
Granted: 1983-11-30
Abstract: Tobacco containing solid carbon dioxide is fed into an expansion chamber (14) in which it is expanded by hot gas; the solid carbon dioxide thereby being sublimed and moisture and organic material in the tobacco being volatalised. The gas and expanded tobacco enter a separator (15) from which the tobacco is discharged through a rotary valve (17). Gas is withdrawn from the separator (15), a portion of it vented, and the remainder heated by heater (27) and then returned to the expansion chamber (14). In order substantially to preclude air flowing through the rotary valve (17) into the separator (15) the pressures below and above the rotary valve are equalised. Alternatively, some of the gas withdrawn from the chamber (15) my be used to isolate the valve (17) from the atmosphere. By precluding air flow into the separator (15) the tobacco may be expanded without using steam (other than that evolved from the tobacco) or excessive temperatures.
Patent GB-2043029-B (GB)
Title: Device for loading and unloading lift truck
IPC: B66F9/12
Filed: 1979-08-17
Granted: 1982-10-20
Abstract: The present invention discloses a load lifting unit for a lift truck, and more particularly, an improved structure of a load lifting unit for a counterbalance type lift truck. In the invention, to increase the loading capacity and longitudinal stability of the lift truck as well as to improve the forward view from the lift truck, two lift cylinders (7) are separately disposed on the sides of a pair of upright assemblies (1) of the load lifting unit, respectively, to provide a space (17) between the upright assemblies for allowing a lift member (4) to be lifted and lowered within the space and for allowing actuating means of various operations attachments engaged with the lift member to be accommodatedly arranged within the space.
Patent GB-2089085-B (GB)
Title: Transport system with vehicle spacing control means
IPC: G05D1/02
Filed: 1981-10-22
Granted: 1984-08-30
Abstract: PCT No. PCT/CH81/00114 Sec. 371 Date Jun. 14, 1982 Sec. 102(e) Date Jun. 14, 1982 PCT Filed Oct. 16, 1981.The equipment for maintaining the spacing of track-bound vehicles (1) shall prevent collisions of the vehicles (1). For this, light emitters radiating rearwardly and laterally in desired directions are provided at the rear on the vehicles (1) and light receivers receiving from in front and from the sides in desired directions are provided at the front on the vehicles (1). A drive control reduces the speed of a vehicle (1) with increasing received light intensity, i.e. with decreasing spacing from the vehicle (1) travelling immediately ahead. The equipment is usable for floor conveying plants with vehicles (1) travelling at small spacings one behind the other. An embodiment of the equipment is suitable for vehicles (1) travelling forwardly and rearwardly. A further embodiment of the equipment is suitable for vehicles (1) on neighboring travel paths. Special measures are provided for compensation of the influences of ambient light.
Patent GB-2113320-B (GB)
Title: Bearing housing
Inventor: LUNDGREN BENGT
IPC: F16C23/08
Filed: 1983-01-14
Granted: 1985-07-17
Abstract: The invention relates to a bearing housing (1) for supporting a bearing (2) in a bearing seat arranged in the housing. In order to provide a rigid, strong, lightweight and inexpensive bearing housing, the housing has the shape of a tube with a mainly rectangular cross section. The axis (3) of a bearing mounted in the housing extends mainly perpendicular to two housing walls (4) facing each other and the bearing is enclosed by the housing.
Patent GB-2164491-B (GB)
Title: Semiconductor devices
Inventor: SCOVELL PETER DENIS
IPC: H01L23/52
Filed: 1984-09-14
Granted: 1988-04-07
Abstract: 57 In order to prevent diffusion of silicon from under a titanium disilicide interconnect (1) and into an overlying aluminium layer (6), the disilicide is selectively nitrided at the points where interconnection between the disilicide and aluminium is required via holes (4) in a silicon dioxide layer (3). The titanium nitride contacts (5) thus formed in a truly self-aligned manner provide a good barrier to silicon diffusion whilst having an acceptable low resistivity.
Patent GB-2260623-B (GB)
Title: Improvements in or relating to calendars
Inventor: RUSHTON BRIAN DAVID
IPC: B42D15/04
Filed: 1991-10-15
Granted: 1994-12-07
Abstract: A calendar which comprises a plurality of leaves. Each leaf comprises an upper date displaying portion (14) and a lower detachable portion (16). The leaves are held together at the upper portions, and the calendar is mountable on a suitable support member by the upper portions for the purpose of display. When the lower portion has been detached, it can be used as a greetings card. <IMAGE>
Patent GB-2298306-B (GB)
Title: Array type recording system
Inventor: MIZUNO MASAHIRO
IPC: G06F11/10
Filed: 1993-10-05
Granted: 1997-03-05
Abstract: A read unit 400 which governs reading of data and a write unit 500 which governs writing of data are located separately in a RAID unit 300 which controls array type magnetic disk units. To read data from magnetic disk units 800, a control circuit 600 uses the read unit 400 to read data through an HDD control unit 700. To write data, the control circuit 600 uses the write unit 500 to write data into the magnetic disk units 800. Since the read unit and write unit are provided separately, processing performance improves. A tasking means 340 is provided for accessing a number of media in the array which selects the next task to be performed by reading an interrupt vector 344, the individual bits being set upon completion of a corresponding disk access.
Patent GB-2331523-B (GB)
Title: Vaccine production of the bacillus anthracis protective antigen
Inventor: BAILLIE LESLIE WILLIAM JAMES
IPC: C12N15/31
Filed: 1997-08-26
Granted: 2000-10-18
Abstract: Methods of preparing recombinant Bacillus anthracis protective antigen or a variant or fragment thereof for use in vaccines is disclosed. The protein is expressed in a recombinant microorganism which comprises a sequence which encodes PA or said variant or fragment thereof wherein either (i) a gene of the microorganism which encodes a catabolic repressor protein and/or AbrB is inactivated, and/or (ii) wherein a region of the PA sequence which can act as a catabolic repressor binding site and/or an AbrB binding site is inactivated. Useful quantities of protein are obtainable from these organisms.
Patent GB-2341659-B (GB)
Title: Valve control mechanism and engines containing same
Inventor: WALTERS CHRISTOPHER PAULET MEL
IPC: F01L1/14
Filed: 1999-10-29
Granted: 2002-03-27
Abstract: A valve control mechanism is disclosed which permits either or both of (a) axial displacement of the camshaft of an internal combustion engine, and (b) phasing of the camshaft (and hence of the valve operation)-i.e. an advance/retard function. The mechanism preferably includes a piston housed within a cylinder, this arrangement itself being mounted within a front end camshaft pulley. The piston is under hydraulic control, preferably governed by a microprocessor. A mechanical coupling between the piston and the camshaft translates the axial movement of the piston into one or both of axial displacement of the camshaft and relative advancement/retardation of its rotation.
Patent GB-2340240-B (GB)
Title: Relative height gauge
Inventor: HENDERSON STEPHEN CARL
IPC: G01B13/14
Filed: 1998-06-24
Granted: 2001-03-21
Abstract: A gauge for monitoring the relative height of two points comprises a generally tubular conduit extending from a first end thereof via a first limb thereof to a monitoring position spaced from the first end and via a second limb of the conduit from the monitoring position to a second end of the conduit in the region of its first end, two immiscible fluids of different densities, each in one of the first and second limbs with a mutual interface within the region of the monitoring position, means to vary the relative vertical positions of the monitoring position on the one hand and the first and second conduit ends on the other, and a pressure comparator to compare the pressures of the fluids at the conduit ends.
Patent HU-217616-B (HU)
Title: Heteroaryl-8-aza-bicyclo-[3.2.1]octanes and method for producing them
Inventor: FINK DAVID M
IPC: A61P25/18
Filed: 1992-02-03
Abstract: This invention relates to compounds of the formula <CHEM>  where     X is -O-, -S- or -NH-;     Y is hydrogen, halogen and loweralkoxy;     p is 1 or 2;     n is 2, 3 or 4; R is hydrogen, loweralkyl, loweralkoxy, hydroxy, halogen, amino, loweralkylamino, nitro, loweralkylthio, trifluoromethoxy, cyano, trifluoromethyl, <CHEM>  where aryl is <CHEM> R1 is hydrogen, loweralkyl, loweralkoxy, halogen, hydroxy, carboxyl, loweralkylamino, nitro, loweralkylthio, cyano, and trifluoromethyl; m is 1 or 2; a pharmaceutically acceptable acid addition salt thereof and, where applicable the geometric and optical isomers and racemic mixtures thereof. The compounds and compositions of this invention are useful as antipsychotic agents and as inhibitors of the reuptake of serotonin.
Patent HU-213231-B (HU)
Title: Process for preparing a dihydro benzofurane derivative, and antitumor preparations containing it
Inventor: BODER GEORGE BERNARD
IPC: C07D307/79
Filed: 1993-02-03
Abstract: This invention provides the use of N-[[(3,4-dichlorophenyl)amino]carbonyl]-2,3-dihydrobenzofuran-5-sulfon amide, and pharmaceutically acceptable salts thereof, in the treatment of susceptible neoplasms in mammals. This invention further provides the novel aforementioned compound and its pharmaceutical formulations.
Patent HU-219279-B (HU)
Inventor: IKEMOTO HISASHI
IPC: A63B41/08
Filed: 1995-10-03
Abstract: A találmány tárgya labda  labdajátékokhoz,  amely  tartalmaz  egy  bőrköpenyréteget (5) (külsőt), amit több bőrszeletnek  (2)  egy  fonallalvaló összevarrásával állítanak elő, és ez a bőr köpenyréteg  (5)  gömbalakú. Tartalmaz továbbá egy elasztomerből készült gumibelsőt (6), amiüreges és gömb alakú, a bőr köpenyréteg belsejében van  elhelyezve,  alevegőnek a gumibelsőbe  (6)  való  bevezetése  végett  szeleppel  vanellátva, amelyen át a gumibelsőt (6) levegővel megtöltik. A fonal  egyönzsugorodó fonal (9), amely varrás  után  zsugorítókezelést  kap.  Azeljárás során kialakítanak egy üreges,  gömb  alakú  gumibelsőt,  többbőrszeletet gömb alakúvá varrnak össze egy önzsugorodó  fonallal,  ígybőr köpenyréteget alakítanak ki,  és  a  belsőt  a  bőr  köpenyrétegbeteszik, majd az önzsugorodó fonalat hővel zsugorítják. ŕ
Patent HU-219730-B (HU)
Inventor: HEIDINGER HARTMUT
IPC: F17C1/00
Filed: 1997-03-17
Abstract: A találmány tárgya nyomástartó tartály gázok, elsősorbanszobahőmérsékleten és légköri nyomáson gáz alakú szénhidrogének,például metán, etán, propán, bután, izobután tárolására. A nyomástartótartálynak lényegében henger alakú és közvetve és/vagy közvetlenül egytámaszközegre, például betonra (14) felfekvő, és a gázok számárabevezetésekkel és elvezetésekkel a felső végrészen, előnyösen egyközös be- és elvezetéssel ellátott fém tömítőhéja (12) van. Atömítőhéj (12) által képzett nyomástartó tartály a talajban lényegébenfüggőlegesen van elhelyezve. A henger alakú fém tömítőhéj (12)átmérőjének és maximális kiterjedésének aránya legalább 1:100, előnyösmódon legalább 1:500, és a tömítőhéj (12) alsó része oldhatatlan,merev módon, előnyösen betonnal (33) van lezárva. ŕ
Patent HU-220352-B (HU)
Inventor: ALVAREZ ERIC
IPC: E05C9/18
Filed: 1997-04-04
Abstract: A találmány csukló vagy záró típusú vasalati szerkezeti elemrevonatkozik, különösen egy ütközőre ablakhoz vagy ajtóhoz, amelynek atokszerkezete és/vagy a nyíló szárnya profilok (2), nevezetesenalumínium- vagy PVC profilok összeállításával van kialakítva, és aprofil (2) magában foglal egy mélyedésben (3) elhelyezkedő „T” alakúhornyot (4), ugyanakkor az említett, vasalati szerkezeti elem (1)magában foglal egy széles részt (11) a „T” alakú horonyban (4) valórögzítésre alkalmas rögzítőszerkezettel (12) felszerelve, és ez arögzítőszerkezet (12) olyan beakasztószerkezettel (18) vankiegészítve, amely a profil (2) mélyedésében (3) elhelyezkedőbeakasztó- szélhez (19) kapcsolódik. A beakasztószerkezetet (18) aszéles résszel (11) párhuzamos és egy arra merőlegesen kiterjedő ésennek a széles résznek (11) a hátsó szélén (26) lévő nyúlvány (25)szabad szélén kialakított visszahajtás (24) képezi, és a vasalati elem(1) felszerelt helyeztében a visszahajtás (24) a beakasztószél (19)alatt – „P” síkban –, párhuzamosan a „T” alakú horony (4) fenekével(5), a horonnyal (4) ellentétes irányban helyezkedik el. ŕ