baber/WOPTO huggingface dataset:
Patent EA-017471-B1 (EA)
Title: Phenylpropionamide compounds and the use thereof
Inventor: ZHOU XIAOMING
IPC: A61K45/06
Filed: 2007-10-31
Abstract: The invention relates to phenylpropionamide compounds of Formula (I): and pharmaceutically acceptable salts, prodrugs, and solvates thereof, wherein A, B, R, R, R, Rand Rare defined as set forth in the specification. The invention is also directed to the use of compounds of Formula (I) to treat, prevent or ameliorate a disorder responsive to the activation of opioid receptors, particularly [mu]-opioid receptors. Compounds of the present invention are especially useful for treating pain.
Patent EA-019853-B1 (EA)
Title: 1-(pyridin-3-yl)-3-methylaminomethyl-5-phenylsulfonylpyrazol derivatives
Inventor: NISHIDA HARUYUKI
IPC: A61K31/4439
Filed: 2010-03-25
Abstract: Disclosed is a compound having an excellent inhibitory activity on the secretion of an acid and exhibiting an antiulcer activity and others. The compound is represented by the formulawhere Rrepresents a fluorine atom, Rrepresents (i) a methyl group or (ii) a cyano group, and Rrepresents a hydrogen atom, or a salt thereof.
Patent EA-024155-B1 (EA)
Title: Antipsychotic injectable depot composition
Inventor: GUTIERRO ADURIZ IBON
IPC: A61K47/34
Filed: 2011-05-31
Abstract: The present invention is directed to compositions for injectable in-situ forming biodegradable implants for extended release that can be used to deliver an antipsychotic drug such as risperidone and to provide therapeutic plasma levels thereof from the first day. The composition is an injectable depot composition, comprising a drug which is risperidone and/or 9-OH-risperidone; at least one biocompatible copolymer which is a copolymer based on lactic and glycolic acid having a monomer ratio of lactic to glycolic acid in the range from 50:50 to 75:25, and at least one water-miscible solvent with a dipole moment about 3.9-4.3 D, wherein the viscosity of the solution comprising the polymer and the solvent is between 0.5 and 3.0 Pa∙s and the solvent/drug mass ratio is between 10 and 4, and wherein the drug/polymer mass ratio is between 25 and 35% expressed as the weight percentage of the drug with respect of the drug plus polymer, the particle size distribution of the drug is as follows: less than 10% particles smaller than 10 microns, less than 10% particles larger than 225 microns, and a d0.5 value in the range of 60-130 microns. Once the composition contacts the body fluids, the polymer matrix hardens retaining the drug, forming a solid or semisolid implant that releases the drug in a continuous manner. Therapeutic plasma levels of the drug can be achieved since the first day up to at least 14 days or more.
Patent EA-029003-B1 (EA)
Title: Agrochemical organic crystal with a micelle coating and process for coating said crystal
Inventor: MULQUEEN PATRICK JOSEPH
IPC: C09D153/00
Filed: 2012-07-03
Abstract: The present invention relates to a process for coating an agrochemical organic crystal with micelles comprising an AB block copolymer. The process comprises treating the agrochemical organic crystal with an apolar liquid containing the micelles. Said AB block copolymer comprises: (i) a first hydrophobic block A selected from the group consisting of a homopolymer of an acrylate or alkylacrylate monomer; a copolymer comprising two or three different monomers selected from acrylate or alkylacrylate monomers; a homopolymer of a styrenic derivative; a copolymer comprising two different monomers selected from styrenic derivatives; and a random, alternating, gradient or block copolymer comprising monomers selected from acrylate monomers, alkylacrylate monomers and styrenic derivatives; and (ii) either a second hydrophobic block B or a hydrophilic block B having a different affinity than the block A for the liquid medium in which the AB copolymers are dispersed such that micelles are formed. The present invention also relates to an agrochemical organic crystal with a micelle coating coated by the process according to the invention.
Patent EA-026033-B1 (EA)
Title: Insecticidal water-in-oil (w/o) formulation
Inventor: KIJLSTRA JOHAN
IPC: A01N25/20
Filed: 2013-05-14
Abstract: The invention relates to an insecticidal water-in-oil (W/O) formulation, comprising at least one insecticidal active ingredient and at least one burning salt, and the production of said formulation. The formulation according to the invention is suitable in particular for treating suitable carrier materials, in particular paper carriers, in an economical single-step process by means of conventional application methods. The present invention further relates to insecticidal products that can smolder, which are produced by treating a carrier material with the formulation according to the invention.
Patent EA-029710-B1 (EA)
Title: Blast furnace and method for operating a blast furnace
Inventor: KUEHL OLAF
IPC: C21B7/00
Filed: 2014-06-05
Abstract: The present invention is directed to a blast furnace and a method for operating a blast furnace which are able to reduce the COproduction and reduce the amount of applied additives and heating material when compared to presently known metallurgical plants. This problem is solved by a process for metal production of metal ores comprising the following steps: reducing a metal ore, particularly a metal oxide; producing furnace gas containing COin a blast furnace shaft; discharging said furnace gas from the blast furnace shaft; directing at least a portion of the furnace gas directly or indirectly into a COconverter and reducing the COcontained in the furnace gas into CO in the COconverter; directing at least a portion of the CO from the COconverter into the blast furnace shaft. Besides solving the above mentioned problem, the method also produces CO as a gaseous reduction agent which may be easily introduced into the blast furnace shaft. A blast furnace for extracting metal that operates in accordance with the above mentioned process comprises a blast-furnace shaft having a first furnace gas outlet and at least one CO inlet; a COconverter, which has a COconverter entry and a COconverter gas inlet for gases containing COand which is suitable for reducing COto CO; wherein the first furnace gas outlet is connected directly or indirectly to the COconverter gas inlet; and wherein the COconverter has at least one first CO outlet for discharging a first part of the CO produced in the COconverter, said first CO outlet being connected directly or indirectly to the blast-furnace shaft.
Patent EA-031802-B1 (EA)
Title: Drug delivery system
Inventor: VERHOEVEN WILLY J H
IPC: A61K31/569
Filed: 2014-12-08
Abstract: Described herein is an intra-vaginal drug delivery system comprising (i) a core comprising a first ethylene-vinylacetate copolymer and etonogestrel, wherein etonogestrel is dissolved in the ethylene-vinylacetate copolymer, and (ii) a skin surrounding the core comprising an ethylene-vinylacetate copolymer, wherein etonogestrel is less permeable in the second ethylene-vinylacetate copolymer than the first ethylene-vinylacetate copolymer, and 17beta-estradiol in solid form, wherein 17beta-estradiol is loaded in a portion of the skin.
Patent EA-034154-B1 (EA)
Title: Method of determining pore diameter of porous objects
Inventor: Charnaya Elena Vladimirovna
IPC: G01N24/08
Filed: 2017-12-21
Abstract: The claimed invention relates to a method of determining an average pore diameter of a porous object, the method comprising: (A) entering liquid gallium or one of the alloys in a liquid state selected from the group consisting of gallium indium (Ga-In), gallium-tin (Ga-Sn) and gallium-indium-tin (Ga-In-Sn) into said porous object; (B) measuring the nuclear magnetic resonance spectrum on the gallium nuclei in liquid gallium or in one of the alloys in the liquid state selected from the group consisting of gallium indium (Ga-In), gallium-tin (Ga-Sn) and gallium-indium-tin (Ga-In-Sn) in said object with the Knight Shift determination (K) from the NMR spectrum obtained; (C) measuring the nuclear magnetic resonance spectrum on the gallium nuclei in liquid gallium or in one of the alloys in the liquid state selected from the group consisting of gallium indium (Ga-In), gallium-tin (Ga-Sn) and gallium-indium-tin (Ga-In-Sn) with the Knight Shift determination (K) from the NMR spectrum obtained; (D) determining the average pore diameter of said porous object according to the formula d=-dln[(K-K)/αK], wherein α takes the meanings from 0.01 to 0.3, dtakes the meanings from 1 to 7 nm. The technical results of the present invention consist is reduced measurement and analysis time, increased accuracy of pore size determination, reduced energy costs, increased overall safety of the method.
Patent EA-033038-B1 (EA)
Title: Liquid crystal panel and manufacturing method therefor
Inventor: WU CHUAN
IPC: G02F1/1339
Filed: 2014-12-12
Abstract: A liquid crystal panel and a manufacturing method therefor are provided. The liquid crystal panel comprises an array substrate provided with thin film transistors; a color filter substrate provided with primary photo-spacers and secondary photo-spacers. The primary photo-spacers are disposed opposite the thin film transistors. The stage differences between the secondary photo-spacers and the primary photo-spacers decrease from the middle of the panel to boundaries thereof. The area between the two substrates is filled with liquid crystal and the substrates are then sealed. Provided is a design that utilizes the stage differences between the primary photo-spacers and the secondary photo-spacers being gradually changed, so that the decline of optical quality due to the fact that box thickness in different areas is uneven is prevented.
Patent EA-033757-B1 (EA)
Title: Methods of precipitating polymer and deactivated organometallic catalyst in an olefin oligomerization reaction
Inventor: ZILBERSHTEIN TIMUR MIKHAILOVICH
IPC: C07C7/12
Filed: 2014-12-23
Abstract: A method of precipitating polymer and deactivated organometallic catalyst in an olefin oligomerization reaction is provided. The method includes providing an effluent stream from an olefin oligomerization reaction. The effluent stream can include a polymer and an organometallic catalyst. The method can further include introducing sorbent particles into the effluent stream. The sorbent particles can include a deactivating agent. The deactivating agent can be water, an alcohol, an amine, an amino alcohol, or a combination thereof. At least about 10% of the sorbent particles can have a particle size in a range from 10 and 60 μm. The method can further include cooling the effluent stream, thereby precipitating polymer and deactivated organometallic catalyst from the effluent stream to provide a precipitate that includes sorbent, polymer and deactivated catalyst.
Patent EA-033569-B1 (EA)
Title: Method of digital data transfer
Inventor: GULAJ ANATOLY VLADIMIROVICH
IPC: H04L12/70
Filed: 2017-12-08
Abstract: The invention relates to the field of digital communication and control devices, and it may find use in constructing highly-effective intellectual systems with remote transfer of data streams. Utilization of the device allows to create a high reliability system for multi-channel transfer of digital data, avoid laying multiple highly expensive cable lines or allocating sufficient number of valuable radio frequencies carved out of the extremely deficit radio frequency spectrum. The method for data transfer is based on forming a Hadamard matrix at the transmitting side of the line, its dimension corresponding to the number of data sources, and the elements of its strings representing the values of orthogonal Walsh functions, attributing each such function to specific information source. Then, next bits with the same numbers are picked from each initial data package, converted into time-coded representations using the abovementioned orthogonal Wash functions and the data part of the bit frame is filled with such coded representations. After that an error-tolerant block code is superimposed by forming the control part of the bit frame, both parts of the bit frame flagged and/or attributed with "start-stop" signals and then the data are sent down the communication line. Once the adornments are removed at the receiving end of the line, the data and control parts of the bit frame are checked for correctness, adjusted, if necessary, and the bit values of individual data packages are restored using the abovementioned Wash functions and the newly formed data packages are transferred to the data user.
Patent EA-036703-B1 (EA)
Title: Temperature-control device for a battery system
Inventor: KREISEL PHILLIP
IPC: H01M10/643
Filed: 2016-10-18
Abstract: The invention relates to a temperature-control device (1) for a battery system, at least comprising a cuboid-shaped hollow body (2) having at least one connection device (3) for supplying and at least one connection device (4) for discharging a separately temperature-controlled fluid, a plurality of regularly arranged and identical openings (7) extending from a first body surface (5) to a second body surface (6), wherein a cylindrical battery cell (8) is accommodated by each opening (7), such that a fluid-tight fluid chamber is formed. The hollow body (2) extends below an output of a cell head (11) and a cell base (12) over a height h from >20 to <100% of the total height H of the battery system.
Patent EA-038691-B1 (EA)
Title: Apparatus for delivery of therapeutic agents
Inventor: HANNAMAN ANDREW W
Filed: 2017-03-28
Abstract: Methods and an apparatus for the reproducible, consistent and efficacious delivery of a therapeutic agent to a subject. The invention provides an apparatus for the controlled administration of the therapeutic agent through an orifice to a subject, a plurality of penetrating electrodes arranged with a predetermined spatial relationship relative to the orifice, and an electrical signal generator operatively connected to the electrodes.
Patent EA-037488-B1 (EA)
Title: Benzazepine derivative, preparation method, pharmaceutical composition and use thereof
Inventor: GAO DAXIN
IPC: A61P37/00
Filed: 2017-05-04
Abstract: Disclosed are a benzazepine derivative, a preparation method, a pharmaceutical composition and the use thereof. The compound as shown in formula (I) of the present invention, and a stable isotope derivative or a pharmaceutically acceptable salt thereof have the following structure. The benzazepine derivative of the present invention has a good regulation effect on the TLR family and the related signalling pathway, and in particular, has a very good regulation effect on TLR8, can effectively treat, relieve and/or prevent various diseases mediated by the TLR family and the TLR-related signalling pathway, and in particular, can effectively treat, relieve and/or prevent various diseases mediated by TLR8, such as cancers, autoimmune diseases, infections, inflammations, transplantation rejections, graft-versus-host diseases, etc.
Patent EA-038284-B1 (EA)
Title: Power-variable motor and intelligent controller
Inventor: ZHANG SHIXING
IPC: H02K3/28
Filed: 2017-07-05
Abstract: Disclosed are a power-variable motor and an intelligent controller therefor. The motor is mainly composed of a rotor, a stator, a shell, a stator winding and a terminal. The stator winding is formed by the same stator core being inserted into a plurality of series windings. Various series nodes of the stator winding, respectively serving as a supply terminal with various different powers, are respectively led out individually. The various series windings of the stator respectively control, by means of the intelligent controller, the connection and disconnection of a plurality of shift switches. The soft-start and soft-stop of the motor can be realised, and a load is automatically tracked to regulate the power of the winding during operation, so as to obtain a power-saving effect.
Patent ES-2171140-B1 (ES)
Title: Articulo absorbente desechable con ajuste de cintura mejorado.
Inventor: CORONA CARLOS ALBERTO
IPC: A61F13/15
Filed: 2000-12-15
Granted: 2003-12-16
Abstract: Artículo absorbente desechable con ajuste de cintura mejorado. La presente invención se refiere a un pañal desechable para bebés o para adultos incontinentes en el cual se logra un ajuste integral del mismo hacia el cuerpo del usuario mediante el uso de un cinturón elástico de ajuste en la parte de cintura trasera del pañal, constituido por una zona elástica que abarca toda la anchura de esta parte de cintura trasera y por las cintas de sujeción, que son una prolongación de esta zona elástica, de forma que al jalar las cintas para colocar el pañal en el usuario, se tensiona el elástico y se logra un verdadero ajuste del producto hacia el usuario. Este cinturón elástico de ajuste es ideal para utilizarse en artículos que no tienen cintura elástica por la parte frontal, aunque se puede utilizar aún cuando el producto contenga la misma.
Patent ES-2192455-B1 (ES)
Title: Sistema de regulacion de energia electrica de alta eficiencia y calidad de onda.
Inventor: SANZ BADIA MARIANO
IPC: G05F5/02
Filed: 2001-06-29
Granted: 2004-08-01
Abstract: Sistema de regulación de energía eléctrica de alta eficiencia y calidad de onda, del tipo de los utilizados en la conversión y regulación de energía eléctrica, caracterizado porque está formada por una configuración de conmutadores estáticos de gran potencia previstos para su bloqueo por inversión de tensión, tales como diodos y tiristores, con componentes conmutadores de pequeña potencia de bloqueo rápido por señal, previstos para su funcionamiento a gran frecuencia con técnicas PWM tales como lgbf''s, Bjt''s, Mosfet''s, interconectados por una unidad de almacenamiento, y un sistema electrónico de control de dichas configuraciones, permitiendo la presencia de la doble configuración de pequeña potencia controlar el flujo de energía en las dos direcciones, optimizando las condiciones de funcionamiento en el generador o motor y la calidad de onda y suministro en la red, regulando simultáneamente el flujo de energía eléctrica con altas prestaciones en la calidad de onda, así como la velocidad para cualquier tipo de generador o motor conectados a la red a través de dicho sistema, y la mejora del suministro eléctrico entre tramos de la red eléctrica interconectados por este sistema.
Patent ES-2188418-B1 (ES)
Title: Metodo para analisis y test funcional de circuito digitales de gran dimension mediante emuladores hardware.
Inventor: AGUIRRE ECHANOVE MIGUEL
IPC: G06F11/26
Filed: 2001-11-29
Granted: 2004-11-16
Abstract: Método para análisis y test funcional de circuito digitales de gran dimensión mediante emuladores HARDWARE. Parte de un número indefinido de eventos o condiciones (1), (1'')... (1n ), respectivos circuitos detectores (2), (2'')... (2n), actuantes en combinación con un detector de flanco (3), que recibe información del pad externo de reactivación (4), y con la colaboración de un pad externo (5) de control, del sistema, es posible vigilar tanto eventos deterministas como eventos temporales, concretamente vigilar una condición determinista en tiempo de ejecución, vigilar una condición temporal en tiempo de ejecución, generar una señal o bandera que registre el evento, cualquiera que sea su naturaleza, congelar el circuito para facilitar su análisis desde un sistema gráfico o similar, y comunicar al sistema que se ha producido un evento e identificar cuál de los eventos programados se ha producido.
Patent ES-2193885-B1 (ES)
Title: Puntero para gaita.
Inventor: MENENDEZ SUAREZ MIGUEL ANGEL
IPC: G10D9/00
Filed: 2002-04-22
Granted: 2005-03-01
Abstract: Puntero para gaita que consiste en un cuerpo de material rígido provisto de perforaciones no equidistantes (2), que presenta una perforación (3) con un rebaje o avellanado, y presentando interiormente, conos internos mecanizados.
Patent ES-2224795-B1 (ES)
Title: Muerte celular programada como sistema de contencion biologica.
Inventor: CAMACHO PAEZ ANA G
IPC: C07K14/32
Filed: 2002-07-03
Granted: 2006-05-16
Abstract: Muerte celular programada como sistema de contención biológica. La presente invención se refiere a unas construcciones genéticas que portan genes que codifican una citotoxina, péptido citotóxico {ds} y su antídoto {ep}. Esta invención también se refiere al uso de las construcciones para la transformación de microorganismos utilizados en procesos biotecnológicos que requieran un sistema activo de contención biológica, para eliminar microorganismos genéticamente modificados liberados para la mejora de cultivos, protección de plantas y cosechas, limpieza medioambiental, etc.
Patent ES-2246135-B1 (ES)
Title: Particulas de microgel polimerico con glucosa oxidasa inmovilizada y su uso como biosensor de glucosa.
Inventor: LOPEZ RUIZ BEATRIZ
IPC: G01N27/30
Filed: 2004-04-02
Granted: 2006-11-01
Abstract: Partículas de microgel polimérico con glucosa oxidasa inmovilizada y su uso como biosensor de glucosa. La presente invención se refiere al diseño de un biosensor para la determinación de glucosa basado en un procedimiento para la inmovilización de la enzima glucosa oxidasa en microgeles poliméricos que consigue mantener la actividad enzimática constante durante largos períodos de tiempo. Comprende el diseño de un biosensor amperométrico de glucosa formado por un electrodo de platino sobre cuya superficie se inmoviliza la capa enzimática que consta de glucosa oxidasa atrapada dentro de microgeles de poli (ácido acrílico/acrilamida), que consiste en las siguientes etapas: - Preparación de la emulsión concentrada acuosa/oleosa con el enzima, monómeros, agente entrecruzante, agente iniciador y tensioactivo. - Polimerización de la emulsión concentrada a temperatura controlada. - Recuperación del producto mediante la separación de fases por centrifugación. - Conservación de las partículas de microgel, refrigeradas a 4ºC. - Preparación del biosensor. Como transductor se utiliza un electrodo de disco de platino. Sobre su superficie se incorporan las micropartículas con glucosa oxidasa en su interior y se fijan mediante una membrana de diálisis. La medida de glucosa se realiza en una celda amperométrica de tres electrodos: como electrodo de trabajo el biosensor, como electrodo de referencia uno de plata cloruro de plata y como electrodo auxiliar uno de platino. La medida se realiza a +0,6 V vs. AgCl/Ag. La corriente obtenida está directamente relacionada con la concentración de glucosa en la muestra.
Patent ES-2253111-B1 (ES)
Title: Mejoras introducidas en la patente de invencion 200402619 referente a un sistema de limpieza automatica para sanitarios.
Inventor: LOSTAL GRASA FRANCISCO JAV
IPC: E03D9/00
Filed: 2004-11-05
Granted: 2007-07-16
Abstract: Mejoras introducidas en la patente de invención 200402619 referente a un sistema de limpieza automática para sanitarios con una carpa que cubre el sanitario y un sistema de rociadores, en las cuales la carpa se constituye mediante una persiana de lamas impermeables y resistentes a la corrosión, enrollable en un alojamiento previsto en la pared o suelo, y guiada por guías laterales provistas en paredes o mamparas laterales enfrentados que flanquean el sanitario. En el suelo se dispone una rejilla bajo la cual se dispone la zona técnica así como unos rociadores dirigidos hacia la parte exterior del sanitario. En el interior de la zona cubierta se proveen rociadores dirigidos hacia la carpa o cubierta en orden a eliminar proyecciones de residuos sobre las mismas durante la limpieza.
Patent ES-2310062-B1 (ES)
Inventor: RODRIGUEZ AGUIRRE JOSE FRANCISCO
IPC: A61K39/00
Filed: 2005-07-15
Granted: 2009-11-13
Abstract: The chimeric empty viral-like particles derived from the infectious bursal disease virus (IBDV) are formed by the assembly of fusion proteins comprising a region A consisting of an IBDV pVP2 protein or a "1-n" fragment of said IBDV pVP2, wherein "n" is an integer comprised between 441 and 501, bound to a region B consisting of a heterologous polypeptide comprising a polypeptide of interest, such as a polypeptide useful for prophylactic, therapeutic or diagnostic purposes.