baber/WOPTO huggingface dataset:
Patent IL-69228-A0 (IL)
Title: Compounds having diuretic activity and angiotensin converting inhibitory activity,methods of the preparation thereof and pharmaceutical compositions containing the same
IPC: A61K31/34
Filed: 1983-07-14
Abstract: Novel compounds possessing both angiotensin enzyme inhibitory activity and diuretic activity are disclosed. The compounds are represented by the general formula <CHEM> in which R1, R2, R3, R4, R5 and R6 are hydrogen, alkyl, alkenyl, alkynyl, phenyl-alkyl, and cycloalkyl, and may be the same or different: n is an integer from 0 to 4 inclusive; M is alkenyl, alkynyl, cycloalkyl, cycloalkyl-alkyl, polycycloalkyl, polycycloalkyl-alkyl, aryl, aralkyl, heteroaryl, heteroaryl-alkyl, hetero-cycloalkyl, hetero-cycloalkyl-alkyl, fused aryl-cycloalkyl, fused aryl-cycloalkyl-alkyl, fused heteroaryl-cycloalkyl, fused heteroaryl-cycloalkyl-alkyl, alkoxyalkyl, alkylthioalkyl, alkylamino-alkyl, or dialkylaminoalkyl, or M and R6 taken together with the nitrogen to which M is bonded and the carbon to which R6 is bonded from a saturated unsubstituted heterocyclic group containing 3 or 4 ring carbon atoms; Y is hydroxy, alkoxy, amino, or substituted amino, aminoalkanoyl, aryloxy, aminoalkoxy, or hydroxyalkoxy; Z1 and Z2 each is a chemical bond, the group X3-(CH2)m, an amino acid group or the group X3-(CH2)m-X3 wherein X3 is oxygen, sulfur or NH and m is an integer from 0 to 4 inclusive; A and B each is the same as R1 or halogen, trifluoromethyl, OR1, NO2, NR1R2, SO2NH2, CN, SR1, SOR1, SO2R1, CONR1R2, COOR1; C is hydrogen alkyl, heteroallyl, amino, -CR1 = CR2-, <CHEM> aminoalkyl, furfurylmethylamino, aminorayl or aminobenzyl; X1 and X2 are each S, SO, SO2, NR1, O, chemical bond, (CR9R10)m, -CR9 = CR10-, and CHOH, with the proviso that at least one of X1 and X2 be (CR9R10)m, wherein R9 and R10 are each hydrogen or lower alkyl, and m is an integer from 1 to 5: Ar is a divalent arylene or heteroarylene: and R7 and R8 are
Patent IL-79851-A0 (IL)
Title: Driving device,in particular for a proportioning pump of the piston-flowmeter type
IPC: F03C1/007
Filed: 1986-08-26
Abstract: In a driving device of the piston-flowmeter type, in particular for a proportioning pump, a distributor is mounted at one end of a piston cylinder for controlling the admission and discharge of fluid within two chambers formed respectively on each side of the piston. The distributor body is provided with circular flow passages and two pairs of valve-seats in cooperating relation with two seals of a two-position tubular valve. The valve has a central bore traversed by the piston rod and coupled to a resilient bistable mechanism for reversing the state of the valve and maintaining it in either of its two positions.
Patent IL-96821-A0 (IL)
Title: 3-aminopiperidine derivatives and related nitrogen containing heterocycles
Inventor: DESAI MANOJ C
IPC: A61P29/00
Filed: 1990-12-28
Abstract: 3-Amino-2-phenylpiperidine is a valuable intermediate for the preparation of certain 3-aminopiperidine substance P antagonists. (Divisional of application no 90313680.2).
Patent IL-96907-A0 (IL)
Title: Proteins produced by human lymphocytes,a dna sequence coding for said proteins and their pharmaceutical and biological application
IPC: C07K14/705
Filed: 1991-01-08
Abstract: Proteins produced by human lymphocytes are described, particularly a protein which is expressed on their surface. DNA sequences coding these proteins and their pharmaceutical and biological uses are also described.
Patent ES-476931-A0 (ES)
Title: Improvements introduced to the object of the main patent no.472516 for: a device for decasing ceramic pieces.
IPC: B65G47/38
Filed: 1979-01-17
Abstract: The main improvement relates to the inclusion in the process of a system for returning the empty cassettes, which had not been provided in the main patent, the system for which consists of a trolley equipped with rollers capable of moving upwards which is situated at the end of the belt removing the cassettes, perpendicular to this belt and responsible for transporting them to a return belt.
Patent FI-20020240-A0 (FI)
IPC: B42C9/00
Filed: 2002-02-06
Abstract: The mechanism is assembled of four toothed wheels (11, 13, 15, 17) to be rotated with a lever (9). Only half of the outer surface of the gear (11) fitted with the lever is provided with teeth, while the adjacent wheel (15) and the wheel (17) adjacent to same are fitted with surrounding teeth. Only a quarter of the contour of the fourth wheel (13) positioned at the opposite side of the drive gear (11) is covered with teeth.  When used at an adhesive binding device the lever (9) acts on the wheels essential for a specific operation without a second lever or holding element required.
Patent FI-20031148-A0 (FI)
Inventor: MUSTALAHTI JORMA
IPC: B66B1/14
Filed: 2003-08-12
Abstract: A method and apparatus adjust the inter-car distance in a double-deck elevator provided with hoisting ropes, in which elevator the hoisting ropes move a car frame supporting the elevator cars along guide rails. The vertical inter-car distance between the elevator cars is adjusted by moving at least one of the elevator cars in relation to the car frame by pulling the elevator car to be moved upwards and lowering the elevator car to be moved downwards by an adjusting rope.
Patent FI-20090269-A0 (FI)
Inventor: LAMPINEN RIKU
IPC: B66B/
Filed: 2009-07-08
Abstract: Rope of a hoisting apparatus, more particularly of a passenger elevator, which comprises a plurality of parts (T1, T2), which continue unbroken for essentially the whole length of the rope, which parts are preferably load-bearing parts. At least one (T2) of the aforementioned parts (T1, T2) is arranged to be essentially more susceptible to breakage in relation to the number of bends than the other (T1) aforementioned parts.
Patent IL-101224-A0 (IL)
Title: Stackable plugged barrel of synthetic material
IPC: B65D1/20
Filed: 1992-03-13
Abstract: A filling and emptying bung (9) and an aerating and venting bung (10) are arranged in a protected manner in depressions (11, 12) in the lid part (4) of the barrel. The stacking surface (8) of the lid part (4) merges into two webs (17, 18) which run in the circumferential direction, include the bottom surface of the depression (11) for the filling and emptying bung (9), run with a slight gradient from the stacking surface (8) to the bottom surface of the depression (11) and, in a slightly tilted inverted position (1') of the barrel, form drainage channels (21, 22) for the residual liquid (24) which collects on the inside (27) of the lid part (4) and drains through the bung hole (15) of the filling and emptying bung (9). <IMAGE>
Patent IL-103799-A0 (IL)
Title: Improved fish production
IPC: A23K1/16
Filed: 1992-11-19
Abstract: This invention is directed to the use of the compound ractopamine for improved production of fish.
Patent IL-104893-A0 (IL)
Title: Sulphonamido-carboxamides,their preparation and pharmaceutical compositions containing them
IPC: C07C277/00
Filed: 1993-03-01
Abstract: The novel sulphonamidocarboxamides of the formula <IMAGE>  in which     X is a group of the formula X<1> or X<2>: <IMAGE>   T is CH2 or O, and A, M, Q and Y have the meaning given in the description, and hydrates or solvates thereof inhibit the platelet aggregation and clotting of fibrinogen in the plasma induced by thrombin. They are prepared by amidination of a cyclic amino group representing the group X or by C(O)Q amide formation.
Patent IL-105624-A0 (IL)
Title: Triazolinone ring formation in tert-butanol
IPC: C07D249/12
Filed: 1993-05-06
Abstract: A process for the production of aryl triazolinones of the formula <IMAGE>  wherein R is lower alkyl; X is independently halogen, lower alkyl, nitro, hydroxy, NHSO2R', -N(SO2R')2, -N(R'(SO2R' where R' is lower alkyl, and n is an integer from 0 to 3; which comprises treating, in a tert-butanol medium, an aryl hydrazine of the formula <IMAGE>  sequentially with (i) a C1-C3 aldehyde, (ii) a cyanate and weak organic acid, and (iii) a hypochlorite, a salt thereof, or a halogen.
Patent IL-114505-A0 (IL)
Title: Tapping fitting
IPC: F16L41/06
Filed: 1995-07-09
Abstract: The tapping fitting for application to a pipe (P) in order to tap a fluid conducted therethrough to an ancillary device includes a housing (2) having a rotatable blade assembly (3) threadedly received within the housing main section (20) and including a cylindrical cutting blade (32) at its inner end such that rotation of the blade assembly (3) cuts a cylindrical slug from the pipe (P) when attached thereto. The device further includes a hollow stem (4) having an inner end secured to the rotatable blade assembly (3) and an outer end for receiving a key (5) to rotate the hollow stem (4) and the blade assembly (3) from an initial retracted position to a projected position and then to a final retracted position. A seal (50) between the outer surface of the hollow stem (4) and the housing main section (20) seals the interior of the pipe (P) from the external side of the housing (2) both during and after the cutting of the cylindrical slug from the pipe (P). <IMAGE>
Patent IL-117511-A0 (IL)
Title: Apparatus and methods for controlled placement of a polymer composition into a porous web
IPC: D06B15/08
Filed: 1996-03-15
Abstract: The present invention relates to methods for the controlled placement of a curable, shear thinnable polymer composition into a porous web. The controlled placement is performed by applying tension to the porous web. The polymer composition is applied onto a surface of the web. The composition is shear thinned sufficiently to reduce its viscosity and selectively place it into the tensioned web to encapsulate at least some of the structural elements of the web, leaving most of the interstitial spaces of the porous web open. The invention also relates to methods for selectively placing the polymer composition in a substantially continuous region extending through the web so that the polymer composition fills the interstitial spaces and adheres adjacent structural elements in the region. In the areas in the web above and below the filled region, at least some of the structural elements are encapsulated and most of the interstitial spaces are open. The invention also relates to methods for the controlled placement of a polymer composition into a tensioned porous substrate having a matrix of open cells by applying a localized shear force to selectively distribute a curable, shear thinnable polymer composition within the substrate, at least partially individually lining the cell walls of at least some of the cells, and leaving most of the cells open.
Patent IL-130059-A0 (IL)
Title: 8-Azabicyclo(3.2.1)octane derivatives their preparation and their use as insecticides
IPC: C07D498/08
Filed: 1997-10-30
Abstract: The present invention provides a compound of Formula (I):wherein Ar is optionally substituted phenyl wherein the substutuents, if present, are selected from halogen atoms, cyano, alkyl, alkenyl, alkynyl, alkoxy, haloalkyl, haloalkenyl, alkylthio and alkyl amino groups; R represents hydrogen or cyano or a group selected from alkyl, aryl, heteroaryl, aralkyl, heteroarylalkyl, alkenyl, aralkenyl, alkynyl, alkoxycarbonyl, alkanesulfonyl, arenesulfonyl, alkenyloxycarbonyl, aralkyloxycarbonyl, aryloxycarbonyl, heterocyclylalkyl, carbamyl, dithiocarboxyl or XR3 (where X represents oxygen or a group NR4); R3 and R4 are, independently, hydrogen, alkyl, aryl, heteroaryl, aralkyl, heteroarylalkyl, alkenyl, aralkenyl, alkynyl, heterocyclylalkyl, alkoxycarbonyl or carboxylic acyl each of which may be optionally substituted; R1 represents hydrogen, hydroxy, alkyl, alkoxy, amino, nitro, isocyanato, acylamino, hydroxyalkyl, optionally substituted heteroaryl, alkoxyalkyl, haloalkyl, halohydroxyalkyl, aralkyloxyalkyl, acyloxyalkyl, amidoximido, sulfonyloxyalkyl, aminoalkyl, alkoxycarbonylamino, acylaminoalkyl, cyanoalkyl, imino, formyl, acyl or carboxylic acid or an ester or amide thereof, or alkenyl or alkynyl either of which is optionally substituted; or an acid addition salt, quaternary ammonium salt or N-oxide derived therefrom; an insecticidal, acaricidal or nematicidal composition comprising a compound of formula (I) and a suitable carrier or diluent therefor; and a method of combating and controlling insect, acarine or nematode pests at a locus which comprises treating the pests or the locus of the pests with an effective amount of a compound of formula (I) or a composition as hereinbefore described.
Patent IL-131600-A0 (IL)
Title: Chimeric flavivirus vaccines
IPC: C12N7/01
Filed: 1998-03-02
Abstract: A chimeric live, infectious, attenuated virus, containing a yellow fever virus, in which the nucleotide sequence for a prM-E protein is either deleted, truncated, or mutated, so that functional prM-E protein is not expressed, and integrated into the genome of the yellow fever virus, a nucleotide sequence encoding a prM-E protein of a second, different flavivirus, so that the prM-E protein of the second flavivirus is expressed.
Patent IL-148875-A0 (IL)
Title: Sulfonyl hydrazide derivatives, their preparation and pharmaceutical compositions containing them
IPC: A61K31/4439
Filed: 2000-09-28
Abstract: The present invention is related to sulfonyl hydrazide derivatives according to formula I <CHEM> with its geometrical isomers, in an optically active form as enantiomers, diastereomers, as well as in the form of racemates, as well as pharmaceutically acceptable salts thereof, wherein Ar<1> and Ar<2> are independently from each other an unsubstituted or substituted aryl or heteroaryl group,  X<1> and X<2> are independently from each other O or S; R<1>, R<2>, R<3> are independently from each other hydrogen or a C1-C6-alkyl substituent or R<1> forms a substituted or unsubstituted 5-6-membered saturated or unsaturated ring with Ar<1>; or R<2> and R<3> form a substituted or unsubstituted 5-6-membered saturated or unsaturated ring;  n is an integer from 0 to 5; G is selected from a group comprising or consisting of an unsubstituted or substituted 4-8-membered heterocycle containing at least one heteroatom, or G is a substituted or unsubstituted C1-C6-alkyl group; for use as pharmaceutically active compounds, as well as to pharmaceutical formulations containing such sulfonyl hydrazide derivatives. Said sulfonyl hydrazide derivatives are efficient modulators of the JNK pathway, they are in particular efficient inhibitors of JNK 2 and 3. The present invention is furthermore related to novel sulfonyl hydrazide derivatives as well as to methods of their preparation.
Patent IL-159528-A0 (IL)
Title: Ceramic electrostatic chuck assembly and method of making
IPC: H01L21/3065
Filed: 2002-06-10
Abstract: A sintered ceramic electrostatic chucking device (ESC) which includes a patterned electrostatic clamping electrode embedded in a ceramic body wherein the clamping electrode includes at least one strip of a sintered electrically conductive material arranged in a fine pattern. Due to the fineness of the electrode pattern employed, stresses induced during manufacture of the ESC are reduced such that the clamping electrode remains substantially planar after the sintering operation. The resulting ESC allows for improved clamping uniformity. Another ESC includes an insulating or semi-conducting body and a clamping electrode having a high resistivity and or a high lateral impedance. The electrostatic chucking device provides improved RF coupling uniformity when RF energy is coupled thorough the clamping electrode from an underlying RF electrode. The RF electrode can be a separate baseplate or it can be a part of the chuck. The ESC's may be used to support semiconductor substrates such as semiconductor wafers in plasma processing equipment.
Patent IL-163745-A0 (IL)
Title: Use of adenoviruses mutated in the va genes for cancer treatment
IPC: B60H1/34
Filed: 2003-03-25
Abstract: This invention refers to the use of an adenovirus for cancer treatment, being this adenovirus defective in its virus-associated (VA) RNAs. Said adenovirus has a mutation in the VAI or VAII gene sequence or both. This adenovirus may also have mutations in the sequences controlling expression of the VA RNAs.
Patent IL-172232-A0 (IL)
Title: Method and device for cleaning a cylinder of a printing press
IPC: B41F35/02
Filed: 2005-11-28
Abstract: A method and a device for cleaning a cylinder of a printing press-in particular of a flexographic printing press-are described wherein a layer of ink to be transferred to a web substrate to be printed-such as paper, plastic film and the like-is deposited on said cylinder ( 1 ) and wherein a fluid suitable to detach impurities from the area concerned is sent onto the surface of the cylinder ( 1 ) to be cleaned and a suction is provided to remove said impurities from the cylinder surface, said cleaning fluid being vapour.
Patent IL-173479-A0 (IL)
Title: Device for monitoring the condition of a human being
IPC: A61B5/0205
Filed: 2006-01-31
Abstract: A device for continuously monitoring one or more indicators relating to the health or comfort of a person 12 includes one or more sensing means for measuring a value of one or more desired indicators and a communicating means 13 communicating an alarm signal when the measured value is above or below a predetermined value or range of values range, wherein the device 10 is adapted to be attached to an item of clothing 14 of the person 12.
Patent IL-173730-A0 (IL)
Title: Device and method for processing a signal having a sequence of discrete values
IPC: H04N7/30
Filed: 2006-02-14
Abstract: When processing a signal having a sequence of discrete values, wherein there is a first frequency range, in which the signal has a high energy, and wherein there is a second frequency range, in which the signal has a low energy, the sequence of discrete values is first manipulated to obtain a sequence of manipulated values, so that at least one of the manipulated values is non-integer. Then the sequence of manipulated values is rounded to obtain a sequence of manipulated values. The rounding is formed to effect a spectral shaping of a generated rounding error so that a spectrally shaped rounding error has a higher energy in the first frequency range than in the second frequency range. By spectrally shaping the rounding error so that the rounding error does not have any energy either in the storage areas where there is no signal energy, an especially efficient coding is obtained particularly in connection with a lossless coding context.
Patent RO-130106-A0 (RO)
Title: Method for lifting automobiles by using an incorporated device
Inventor: FENECHIU RELU
IPC: B66F5/02
Filed: 2014-10-23
Abstract: The invention relates to a method for lifting automobiles by using incorporated hydraulically or electrically driven devices for carrying out the operations of repairing and corrective maintenance thereof. According to the invention, the lifting method is based on using two or four lifting devices incorporated into the automobile chassis, eliminating the user's physical effort as well as the accident risk or the automobile deterioration, when using the classic jacks. According to the invention, the device used for carrying out the method performs the lifting operation by means of a rod (1), dropping from the device proper (2) and which is provided, in the lower side, with a base (3) mounted by means of a ball joint (4), either directly on the rod (1) or by means of an arm (5).
Patent AP-2004003023-A0 (AP)
Title: Nicotinic acid-heterocyclyl-amides and analogous pyrimidine derivatives serving as pesticides
Inventor: SCHAPER WOLFGANG
IPC: C07D409/12
Filed: 2002-09-14
Abstract: The invention relates to amides of formula (I) and to the salts thereof, whereby the symbols and indices have the following meanings: X represents CH or N; Y represents O or S; n is 0 or1; R1 represents (C1-C4) alkyl halide; R2 and R3. Independent of one another represents hydrogen. (C1|-C4) alkyl, (C1-C4) alkyl halide or halogen; R4 represents hydrogen, (C1,-C10) alkyl, (C3-C10) cycloalkyl. (C3-C10) alkenyl or (C3-C10) alkynyl, whereby up lo three hydrogen atoms can be replaced by halogen in said alkyl, cycloalkyl, alkenyl or alkynyl groups and, in the case of fluorine, also up to the maximum number; R5 is an aliphatic hetero-cyclic containing at least one oxygen, sulfur, nitrogen and/or silicon ring atom, which is optionally substituted by one to six monovalcnt groups and which can optionally be part of a spirocyclic, condensed or bicyclic ring system. These compounds can be used for producing pesticides.
Patent IE-900028-A1 (IE)
Title: "New process for separating optical isomers of 1,4-dihydropyridine derivatives"
Inventor: PEGLION JEAN-LOUIS
IPC: C07D209/48
Filed: 1990-01-04
Abstract: New process for separating optical isomers of the compounds of general formula I: <IMAGE>  in which:   - Ar denotes a phenyl radical optionally containing one to five identical or different substituents, each denoting a halogen atom, an alkoxy radical containing from 1 to 4 carbon atoms, an alkylthio radical containing from 1 to 4 carbon atoms, a trihalomethyl radical or a methylenedioxy radical, - each of Y, Z, Y1 and Z1, which are identical or different, denotes a hydrogen atom, a linear or branched lower alkyl radical containing from 1 to 4 carbon atoms, a cyclopropyl radical, a dicyclopropylmethyl radical, a 2,2-dicyclopropylethyl radical, a 2,2-dicyclopropylethylene radical, a 3,3-dicyclopropylpropyl radical, a 3,3-dicyclopropyl-1-propylene radical, a linear or branched alkylene radical containing from 2 to 5 carbon atoms or a phenyl radical optionally substituted by a nitro radical, and   - n is equal to 1, 2 or 3.
Patent LU-88458-A1 (LU)
Inventor: ALLEGRUCCI JEAN-PIERRE
IPC: B21K7/02
Filed: 1994-02-15
Abstract: The procedure, designed to increase the height of a rail while reducing the thickness of its web (16) and foot (18), consists of machining the upper portion of the web beneath the head (14) of the rail, and heating the remainder of the web and foot to deform it by forging. The upper portion of the web is machined to its final thickness, and the lower part of the web and foot are heated by a localised induction process, with the rail head cooled at the same time.
Patent MA-19406-A1 (MA)
Inventor: MICHEL VINCENT
IPC: E06C5/36
Filed: 1982-03-05
Abstract: 1. A control device for a rotatable, extendable ladder or similar lifting arm including at least a control for raising and lowering, a control for extension and retraction and a control for rotation to the manual selection instruments for the desired movements, the activators of raising and lowering, of extension and retraction, and of rotation, said selection instruments being adapted to apply electric signals to a microprocessor control signal reader, the said microprocessor containing a memory : the maximal reach to not exceed a function of diverse selectable and predetermined parameters of use of the ladder ; a sequence of cyclic calculations of the actual reach from information given by sensors of vertical angle and extension length ; a cyclic sequence of comparison of the actual calculated reach with the maximal reach corresponding to pre-defined conditions of use and authorizing or not the movement requested ; characterized in that the said electric signals are representative of the direction of the command and the desired speed of execution of the desired movements and that the said microprocessor contains in its memory a deceleration law, for the movements of lowering and extension at least, in the predetermined terminal zones of the evolution of these movements corresponding to a certain approach to the predetermined maximal reach for the circumstances ; and cyclic comparison sequence for this approach of the control speed shown with the speed derived from the said law for each movement considered, destined to impose the said law when the control speed shown is excessive, by furnishing to the outputs of the microprocessor controlling these movements the signals representative of the control speed shown or automatically modified as a function of the said law ; said outputs being connected to the instruments of electric control proportional to the activation of the activators of the movements considered.