baber/WOPTO huggingface dataset:
Patent EA-019951-B1 (EA)
Title: Pim kinase inhibitors and methods of their use
Inventor: BURGER MATTHEW
IPC: A61K31/44
Filed: 2008-03-03
Abstract: The invention relates to new compounds of formula I, stereoisomers thereof or pharmaceutically acceptable salts thereof:wherein X, X, Xand Xare independently selected from CRand N; provided that not more than two of X, X, Xand Xcan be N; Y is substituted amino or substituted or unsubstituted C-C-cycloalkyl, heterocycloalkyl or heteroaryl; Z, Zand Zare independently selected from CRand N; provided that not more than one Z, Zand Zcan be N; Rand Rare as defined in the description; to pharmaceutical compositions for the treatment of cancer containing said compounds, to a method for inhibiting kinase activity associated with oncogenesis in a human or in animal and to the use of new compounds either alone or in combination with at least one additional therapeutic agent for prevention or treatment of cancer.
Patent EA-016036-B1 (EA)
Title: Screen clamp
Inventor: CARR BRIAN S
IPC: B07B1/46
Filed: 2008-10-01
Abstract: A screen clamp (400) including a track (402) configured to secure a shaker screen (420) to a shaker and an upper retainer (404) configured to extend from an inner wall of the shaker over at least a portion of the shaker screen.
Patent EA-019763-B1 (EA)
Title: Method and computer information product for analyzing characteristics of subterranean formation
Inventor: HRUSKA MARINA M
IPC: G01V11/00
Filed: 2009-03-27
Abstract: A method of analyzing characteristics of a subterranean formation includes applying a wavelet transform to measured data or to derived data obtained from the measured data, the measured data obtained by measuring a physical property at each of a plurality of positions in a borehole that penetrates the subterranean formation; selecting one or more scales for analyzing wavelet coefficients; performing a segmentation of the data; calculating a distribution of wavelet coefficients for each scale, for one or more spatial directions of wavelet transform application, for the wavelet transform of the data and for each segment that belongs to the portion on which the wavelet transform has been calculated; and for each segment, analyzing a distribution of the data and the distribution of the wavelet coefficients for each scale in terms of their overlap with corresponding distributions of training samples to produce a geological interpretation of the subterranean formation.
Patent EA-018807-B1 (EA)
Title: Thiazolyl-pyrazolopyrimidine compounds as synthetic intermediates and related synthetic processes
Inventor: RIZZO JOHN ROBERT
IPC: C07D487/04
Filed: 2009-09-29
Abstract: The present invention relates to a synthetic intermediate of the formula (I)and its use in a synthetic process to make compounds of the formula (II)
Patent EA-023892-B1 (EA)
Title: Immunogenic proteins for human papilloma virus and methods for using the same
Inventor: WEINER DAVID B
IPC: A61P37/02
Filed: 2010-01-22
Abstract: Improved anti-HPV immunogens and nucleic acid molecules that encode them are disclosed. Immunogens disclosed include those having consensus HPV 18 E6 and E7. Pharmaceutical composition, recombinant vaccines comprising and live attenuated vaccines are disclosed as well methods of inducing an immune response in an individual against HPV are disclosed.
Patent EA-020934-B1 (EA)
Title: Concrete mixture based on limestone material
Inventor: ALIEV ALI MUSA OGLY
IPC: E01C7/02
Filed: 2011-12-19
Abstract: The claimed invention relates to technology of producing a novel road-constructing material - limestone concrete for use thereof in making layers of road and air field structures. The invention is aimed at producing modified mineral mixtures having an optimum moisture content and predetermined granulometric composition of limestone material in compaction of which grinding and uncovering of grain surface occurs thus providing conditions for natural self-cementing of limestone materials and mineral mixtures prepared basing thereon. Said natural properties of limestone materials and wastes of its production provide to achieve the required normative-strength factors and a significant economic effect in construction of road and air field structures using said materials.
Patent EA-023393-B1 (EA)
Title: Azole derivatives, methods for producing the same, intermediates, agro-horticultural agents
Inventor: ARAKI NOBUYUKI
IPC: C07D405/06
Filed: 2010-12-07
Abstract: An azole derivative according to the invention is represented by Formula (I)wherein Rdenotes a hydrogen atom, or a C-C-alkyl group, a C-C-alkenyl group or a C-C-alkynyl group, each of which is optionally substituted with nof Xsubstituents; Rdenotes a hydrogen atom, or a C-C-alkyl group, a C-C-alkenyl group or a C-C-alkynyl group, each of which is optionally substituted with nof Xsubstituents; Xis a halogen atom; Xis a halogen atom; ndenotes 0-5; ndenotes 0-5; with a proviso that Rand Rsimultaneously do not denote hydrogen atoms; n+ndenotes 1 or more; m denotes 0-5; each Y denotes a halogen atom, a C-C-alkyl group, a C-C-haloalkyl group, a C-C-alkoxy group, a C-C-haloalkoxy group, a phenyl group, a cyano group or a nitro group; A denotes a nitrogen atom or a methyne group. As a result, an azole derivative contained as an active ingredient in an agro-horticultural agent having an excellent controlling effect on diseases can be provided.
Patent EA-027789-B1 (EA)
Title: Pyrolysis equipment for coal material
Inventor: ZHU SHUCHENG
IPC: C10B53/04
Filed: 2010-09-19
Abstract: Disclosed is a pyrolysis equipment for coal material, which comprises an enclosed kiln body with an inlet and an outlet, a flame-gas heating pipeline provided inside the kiln body, coal material propulsion and pyrolysis passage formed between the flame-gas heating pipeline and an inner wall of the kiln body, coal pyrolysis gas collecting tube communicated with the coal material propulsion and pyrolysis passage and provided on the kiln. The heat generated by flame-gas heating pipeline is conducted and radiated to coal powder in the coal material propulsion and pyrolysis passage. The coal powder sufficiently absorbs the heat and is pyrolyzed into fuel gas, tar gas and coal with high heat value inside the coal material propulsion and pyrolysis passage. The pyrolyzed fuel gas and tar gas are transferred to the gas dedusting-liquifying mechanism outside the kiln through the connecting coal pyrolysis gas collecting tube for collecting, dedusting, separating and high-pressure liquefying.
Patent EA-026421-B1 (EA)
Title: Sandwich bread
Inventor: BALASANYAN NAIRA GARNIKOVNA
IPC: A21D13/00
Filed: 2013-08-15
Abstract: The invention is related to food industry, in particular, to production of bakery products, and may find application in preparation of sandwiches with various fillings. The sandwich bread has a cavity confined by thin layers, the layers have the shape of triangulars having a common apex and two common sides, one of the layers having a notch from the middle of the base opposite to the common apex in the direction of the common apex. The notch ends at a distance of 0.5-20 mm from the common apex. The range of products is broadened, convenience of the product use as well as the product quality and shelf life are improved.
Patent EA-028020-B1 (EA)
Title: Processing biomass
Inventor: MEDOFF MARSHALL
IPC: C12P7/10
Filed: 2010-05-18
Abstract: Biomass (e.g., plant biomass, animal biomass, and municipal waste biomass) is processed for use in the production of useful products, such as fuels. For example, systems can use biomass materials, such as cellulosic and/or lignocellulosic materials, to enhance the production of a product, e.g., the production of ethanol and/or butanol by fermentation.
Patent EA-031738-B1 (EA)
Title: Method and system for energy-optimized driving a motor vehicle
Inventor: ZHEBRAK LEONID MIKHAILOVICH
IPC: B60W40/12
Filed: 2014-10-31
Abstract: The invention is designed for saving energy spent by a motor vehicle, e.g., a car, when driving, among others, in the automatic mode. The technical result attained by the invention consists in minimizing the energy spent for the vehicle movement. Said technical result is attained by determining an energy-optimized movement mode – the route of the vehicle movement and control of the vehicle movement in the route while monitoring vehicle parameters and external conditions characteristics that are used for determination of energy-optimized driving. The method of energy-optimized driving a motor vehicle comprises the following steps: determining parameters of relationships of actual tractive effort, braking power, motion resistance force, force of wheels cohesion with road pavement, vehicle mass on the basis of vehicle characteristics; determination and implementation of driving the vehicle on the basis of determined relationships of parameters.
Patent EA-028023-B1 (EA)
Title: Surfactant mixture, method for producing same and use thereof, aqueous surfactant formulation, use thereof and method for producing oil using surfactant formulation
Inventor: BITTNER CHRISTIAN
IPC: C11D1/34
Filed: 2012-10-23
Abstract: The invention relates to a surfactant mixture containing, in relation to the hydrocarbon part (R)(R)-CH-CH- at least three different ionic surfactants of general formula (I)wherein R, R, A, k, X, o, Y, a, b, M have the meaning indicated in the description and the claims. The invention further relates to the use and production thereof and to aqueous surfactant formulations containing the mixtures and to a method for producing mineral oil by means of Winsor type III micro emulsion flooding, in which the aqueous surfactant formulation is forced through injection wells into a mineral oil deposit and the crude oil is removed from the deposit through production wells.
Patent EA-030870-B1 (EA)
Title: Polyester and polyurethane production methods
Inventor: UTSUNOMIYA MASARU
IPC: C08G63/78
Filed: 2013-06-03
Abstract: A method of producing a polyester by using a dicarboxylic acid component and a biomass-resource-derived diol as raw materials, allows to efficiently produce a polyester with good color tone. As the raw material diol derived from biomass resources, a diol in which the content of a cyclic carbonyl compound having a carbon atom number of 5 or 6 is from 0.01 to 12 ppm by mass, is used. By controlling the content of a cyclic carbonyl compound having a carbon atom number of 5 or 6 in the raw material diol to fall in a prescribed range, the color tone of the polyester is improved.
Patent EA-030168-B1 (EA)
Title: Method for monitoring operative conditions of thermal and/or catalytic cracking plants and related apparatus
Inventor: BUCCOLINI MARCO
IPC: G01N21/49
Filed: 2013-10-30
Abstract: The thermal conversion and/or catalytic plants, which can be found in the productive cycle of a refinery, are aimed at the utilization of the residues of the distillation of petroleum, otherwise destined for bitumen or combustible oil (products notoriously of low commercial value), so as to convert these products, in part, into lighter products of greater value. The conversion makes it possible to obtain considerable amounts of distilled products, such as gas, benzene, kerosene and diesel oil. The conversion process is carried out so as to maximize the yield of distilled products, thus lowering the overall yield of heavy residues. Adjustment of the operative parameters of the plants described above for the purpose of maximizing the yield of light products and managing the plants with controlled fouling conditions is carried out by means of methods for measuring aggregated asphaltenes and particles of carbon suspended in the bottom residue produced. The present invention proposes an improved procedure for determining the tendency of the bottom fluid to form fouling in determined plant conditions which definitively makes it possible to obtain better yields of light distillates, better control of the fouling occurring in the plant, and therefore a reduction of the associated energy consumption. In addition, the new procedure described in the patent makes it possible to determine on-line the tendency for fouling inasmuch as the analyzed sample does not require any handling.
Patent EA-030306-B1 (EA)
Title: Bilayered composite tablet formulation comprising atorvastatin, irbesartan and magnesium carbonate
Inventor: KIM YONG IL
IPC: A61K9/24
Filed: 2013-08-30
Abstract: Disclosed are a bilayered composite tablet formation comprising: (a) a first layer comprising irbesartan or a pharmaceutically acceptable salt thereof; and (b) a second layer comprising atorvastatin or a pharmaceutically acceptable salt thereof and magnesium carbonate (MgCO) in a weight ratio of 1:4 to 1:5, and a method for preparing the same. Exhibiting excellent dissolution rates and bioavailability, the bilayered composite tablet formulation is useful as a therapeutic for hypertension and hypercholesterolemia.
Patent EA-027010-B1 (EA)
Title: Retention device for liquids or free flowing substances
Inventor: MULVIHILL MICHAEL
IPC: E02B3/10
Filed: 2013-10-21
Abstract: According to the present invention there is provided a liquid retention device comprising a braced frame mountable on foundations in a plurality of locations, in which said device comprises a base section and at least one upstanding support, and in which said brace further comprises height-adjusting means for adjusting the height of said frame, and in which said device further comprises a face supported by said frame, in which said face is inclined at an angle to the at least one upstanding support, wherein said face is covered by a least one detachable mat.
Patent EA-030907-B1 (EA)
Title: Cortistatin analogues, syntheses and uses thereof
Inventor: SHAIR MATTHEW D
IPC: C07K16/26
Filed: 2014-12-24
Abstract: Provided herein are compounds of Formulaeand pharmaceutically acceptable salts or quaternary amine salts thereof, and pharmaceutical compositions thereof. The compounds are contemplated useful as therapeutics for treating a medical condition by inhibiting CDK8 and/or CDK19 kinase activity.
Patent EA-029774-B1 (EA)
Title: Compounds
Inventor: DING XIAO
IPC: A61K31/519
Filed: 2015-01-28
Abstract: The present invention relates to novel compounds that inhibit LRRK2 kinase activity, processes for their preparation, to compositions containing them and to their use in the treatment of or prevention of diseases characterized by LRRK2 kinase activity, for example Parkinson's disease, Alzheimer's disease and amyotrophic lateral sclerosis (ALS).
Patent EA-033186-B1 (EA)
Title: Bactericidal composition for use in treating citrus diseases
Inventor: SABIN ROBERT
IPC: A01N59/20
Filed: 2015-05-20
Abstract: The present invention concerns bactericidal composition for use in treating Huanglongbing (HLB) disease of citrus, citrus canker, other citrus diseases, such as Greasy Spot, Melanose and Alternaria Brown Spot, and also Xylella fastidiosa diseases of olive trees caused by bacteria, wherein said bactericidal composition comprises at least one biologically inert carrier and at least one doped component. The doped component comprises at least one fixed copper compound doped with at least one compound selected from the group consisting of iron compounds, zinc compounds and combinations thereof. The doped component has a particle size of about 0.5 nm to about 30 μm.
Patent EA-035884-B1 (EA)
Title: New hybrid agaricus bisporus mushroom strains
Inventor: RODIER ANNE
IPC: C12N1/14
Filed: 2016-01-22
Abstract: The invention relates to the field of microorganism strain development, more particularly to the development of heterokaryotic hybrids of the fungus species Agaricus bisporus. Even more particularly, the invention relates to white Agaricus bisporus hybrid strains having improved characteristics for the users (namely the growers, the processers and the consumers). These hybrids are for example the deposited strains CNCM I-4945 and I-4946, originating from a cross plan involving the deposited line CNCM I-4948. The invention relates to strains derived from these hybrids and also progenies derived from these hybrids.
Patent EA-036144-B1 (EA)
Title: Rail transport system
Inventor: WYATT STEPHEN
IPC: B61D11/00
Filed: 2017-05-05
Abstract: A rail transport system 10 has at least two load carrying bodies 12 which are arranged end to end. Mutually adjacent bodies 12 are coupled together by respective coupling systems 14. The rail transport system 10 further includes a plurality of axles 16 each provided at opposite ends with respective rail wheels 18 which support the bodies 12. A flexible liner 20 is supported by the bodies 12. The liner 20 is configured to span respective coupling systems 14. In this way the bodies 12 and the flexible liner 20 form a continuous load carrying structure 22. The continuous load carrying structure 22 is arranged so as to be able to pivot about an axis perpendicular to the axles 16 to facilitate unloading of cargo from the bodies 12.
Patent EA-037284-B1 (EA)
Title: Fluid dispenser
Inventor: BILTON SIMON LEWIS
IPC: B05B11/00
Filed: 2017-05-23
Abstract: A robust and ergonomic fluid dispenser suitable for dispensing cosmetic compositions and comprising a cylindrical outer body, an upper section having a domed applicator surface, a cylindrical lower section that forms a protective cover for a refill cartridge, a rotatable actuator collar, an axially mobile pump housing carrying a pump engine inside, the rotatable actuator collar and the axially mobile pump housing interacting by means of a cam track on one and a cam follower on the other, the pump housing being reversibly attached to the refill cartridge, the cam follower on the pump housing rising on rotation of the actuator collar in a first direction and thereby lifting the pump housing and the refill cartridge to a raised position and actuating the pump engine, the cam follower on the pump housing falling on rotation of the actuator collar in a second direction to a rest position and thereby lowering the pump housing and the refill cartridge.
Patent EA-036440-B1 (EA)
Title: Process for the production of formaldehyde-stabilised urea
Inventor: DAVISON THOMAS
IPC: C07C273/02
Filed: 2017-10-03
Abstract: An integrated process for the production of a formaldehyde-stabilised urea is described comprising the steps of: (a) generating a synthesis gas comprising hydrogen, nitrogen, carbon monoxide, carbon dioxide and steam in a synthesis gas generation unit; (b) dividing the synthesis gas into a first synthesis gas stream and a smaller second synthesis gas stream; (c) subjecting the first synthesis gas stream to one or more stages of water-gas shift in one or more water-gas shift reactors to form a shifted gas; (d) cooling the shifted gas to below the dew point and recovering condensate to form a dried shifted gas; (e) recovering carbon dioxide from the dried shifted gas in a carbon dioxide removal unit to form a carbon dioxide-depleted synthesis gas; (f) subjecting the carbon dioxide-depleted synthesis gas to a stage of methanation in one or more methanation reactors to form an ammonia synthesis gas; (g) synthesising ammonia from the ammonia synthesis gas in an ammonia production unit and recovering the ammonia; (h) reacting a portion of the ammonia and at least a portion of the recovered carbon dioxide stream in a urea production unit to form a urea stream; and (i) stabilising the urea by mixing the urea stream and a stabiliser prepared using formaldehyde to form a stabilised urea, wherein the formaldehyde is generated by steps comprising; (1) passing the second portion of synthesis gas through a scrubber to remove contaminants therefrom and form a scrubbed synthesis gas; (2) synthesising methanol from the scrubbed synthesis gas in a methanol synthesis unit, and recovering the methanol and a methanol synthesis off-gas; (3) combining the methanol synthesis off-gas with the shifted gas and (4) subjecting at least a portion of the recovered methanol to oxidation with air in a formaldehyde stabiliser production unit to produce formaldehyde.
Patent EA-039391-B1 (EA)
Title: Use of a glutarimide derivative to treat diseases related to the aberrant activity of cytokines
Inventor: NEBOLSIN VLADIMIR EVGENIEVICH
Filed: 2018-03-06
Abstract: The invention relates to medicine and concerns the treatment of diseases related to the aberrant activity of fractalkine and monocyte chemoattractant proteins 1-4 (CCL2, CCL7, CCL8, CCL13), preferably the treatment of pain, fever, pneumonia, bronchitis, bronchiolitis, alveolitis, rheumatoid arthritis, psoriasis and other diseases, using the compound 1-(2-(1H-imidazol-4-yl)ethyl)piperidine-2,6-dioneor a pharmaceutically acceptable salt or solvate thereof.
Patent EA-038699-B1 (EA)
Title: Water pipe
Inventor: HAGEN KLAUS
Filed: 2016-11-10
Abstract: A water pipe (1) with a housing (2), into which a container (3) to be filled with a liquid medium and having at least one suction connection (5) and a heating chamber (4) connected therewith serving as receptacle for a smoke medium and comprising an air inlet (6) are integrated. The heating chamber (4) comprises a receptacle (34) for a capsule (13) provided for holding a smoke medium. The receptacle (34) has a wall (35) surrounding the capsule (13) at the side and an opening (52) on its side towards the container (3) and a taper (37) and is formed at the same time as a heating element for the capsule (13).
Patent EA-039634-B1 (EA)
Title: Lens assembly for optical image stabilization and focus adjustment
Inventor: CRAEN PIERRE
Filed: 2018-06-28
Abstract: The invention relates to adjustable or tuneable lens assembly where a deformable, non-fluid lens body is sandwiched between a bendable lens cover and a back window to form a lens. The lens assembly has an actuator system with individually addressable actuators for applying force to the lens cover in direction along the optical axis to change an overall shape of the lens. The actuator system has a focus adjustment mode to adjust the optical power of the lens and an optical image stabilisation mode where the optical axis of the lens is tilted.
Patent ES-2164003-B1 (ES)
Title: Procedimiento de reconocimiento y cabina de puertas interbloqueadas con gestion automatizada.
Inventor: MANNESCHI ALESSANDRO
IPC: G07C9/00
Filed: 2000-01-05
Granted: 2003-04-01
Abstract: La invención consiste en un procedimiento de reconocimiento y en una cabina de puertas interbloqueadas dirigida por dicho procedimiento, equipada con un dispositivo de pesaje y lector biométrico (5) situado en su interior, combinada con una unidad de lógica programada (8) a la que llegan las informaciones de la persona que se presenta para atravesarla, sea por los medios de adquisición de su código de reconocimiento, sea por el dispositivo que procede a su pesaje, sea por el lector (5) que procede a la lectura de sus datos biométricos de modo que, por comparación con los correspondientes datos memorizados, la unidad de lógica programada verifica la identidad de la persona en tránsito y ordena la apertura y el cierre de las puertas (2) y (3) de la cabina (1), así como otros eventuales dispositivos.
Patent ES-2189591-B1 (ES)
Title: Sistema de dosificacion de cafe molido.
Inventor: MARCOTEGUI GONI JOSE ANGEL
IPC: A47J42/50
Filed: 2000-05-23
Granted: 2004-11-16
Abstract: Sistema de dosificación de café molido, que comprende la medición del caudal del café molido, mediante una dosificación volumétrica que incluye un rotor (3) de aspas, cuyas aspas (4) interceptan las corrientes (2) de café molido, y un dispositivo contador de vueltas (6) que facilita información a un programa cuya lógica ajustará el tiempo de funcionamiento del motor del molino, en función de la información procedente del contador de vueltas (6).