baber/WOPTO huggingface dataset:
Patent PH-31325-A (PH)
Title: Methods of increasing thrombomodulin expression.
Inventor: SCOTH CALNEK DANIEL
IPC: A61K31/38
Filed: 1994-12-19
Abstract: A method of increasing thrombomodulin expression comprising administering to a human in need of treatment an effective amount of a compound having the formula <CHEM>     wherein R<1> and R<3> are independently hydrogen, -CH3, <CHEM>  wherein Ar is optionally substituted phenyl; R<2> is selected from the group consisting of pyrrolidino, hexamethyleneamino, and piperidino; or a pharmaceutically acceptable salt of solvate thereof. Also encompassed by the invention is a method of inhibiting a thrombotic disorder or event which includes administering to a human in need thereof an effective amount of a compound of formula 1. Also encompassed by the invention is a method of increasing Protein C activation rate which includes the administration of a compound of formula 1.
Patent UY-32046-A (UY)
Title: Derivados de 2-alquil-6-cicloamino-3-(piridin-4-il)imidazoz[1,2-b]-piridazina, su preparación y su aplicación en terapéutica
Inventor: ZHONGLI GAO
IPC: A61K31/5025
Filed: 2009-08-12
Abstract: La invención se refiere a derivados de 2-alquil-6-cicloamino-3-(piridin-4-il)imidazo[1,2-b]piridazina, representados por la fórmula general (I), donde los radicales y sustituyentes son tales como se especifican en la Memoria Descriptiva y en las Reivindicaciones. Se divulgan procedimiento de preparación y su aplicación terapéutica en el tratamiento o prevención de enfermedades que implican caseína quinasa 1 épsilon y/o caseína quinasa 1 delta.
Patent UY-37313-A (UY)
Title: Bebidas refinadas en base a cereales
Inventor: WENDT TONI
IPC: C12C1/125
Filed: 2017-06-30
Abstract: La presente invención se relaciona con métodos para preparar bebidas basadas en cereales. En particular, la presente invención provee, por ejemplo, métodos para el remojado y germinación del cereal bajo aireación continua. La presente invención también provee la molienda húmeda de granos de cereal germinado y la transferencia directa del grano germinado, sin secado, a la cervecería para su procesado ulterior. Comparado con los métodos actuales, los métodos de la presente invención reducen significativamente el consumo de agua, el consumo de energía y la necesidad de transporte.
Patent UY-37361-A (UY)
Title: Sulfonilureas y compuestos relacionados y uso de estos
Inventor: Luke O’Neill
IPC: C07D307/64
Filed: 2017-08-15
Abstract: La presente invención proporciona determinadas sulfonilureas y compuestos relacionados, los cuales tienen propiedades ventajosas y presentan actividad útil en la inhibición de la activación del inflamasoma NLRP3. Dichos compuestos son útiles en el tratamiento de una amplia variedad de trastornos donde el proceso de inflamación o, más específicamente, el inflamasoma NLRP3 esté implicado como un factor clave.
Patent UY-38348-A (UY)
Title: Composición para erradicar helicobacter pylori
Inventor: KIM BONG TAE
IPC: C07H17/08
Filed: 2019-08-28
Abstract: La presente invención se refiere a una composición para erradicar Helicobacter pylori y su uso. La composición de la presente invención mantiene un pH intragástrico en un cierto nivel o más durante un cierto período de tiempo o más, maximizando así la acción de amoxicilina y claritromicina para mostrar un excelente efecto sobre la erradicación de Helicobacter pylori
Patent UY-38976-A (UY)
Title: Antagonistas de sstr5
Inventor: HE SHUWEN
IPC: C07D513/10
Filed: 2020-12-02
Abstract: Esta divulgación está orientada, al menos en parte, a los antagonistas de SSTR5 útiles para el tratamiento de afecciones o trastornos que afectan al eje intestino-cerebro. En algunas realizaciones, los antagonistas de SSTR5 son compuestos con restricción intestinal. En algunas realizaciones, la afección o el trastorno es un trastorno metabólico, tal como la diabetes, la obesidad, la esteatohepatitis no alcohólica (NASH) o un trastorno nutricional como el síndrome del intestino corto.
Patent YU-28088-A (YU)
Inventor: SCHWARZE W
IPC: C08K5/37
Filed: 1988-02-11
Abstract: Compounds of the general formula <IMAGE>  in which  R<1>, R<2> denote H; R<2> denotes benzyl, R<2>, R<3>, R<4> denote C1-C8-alkyl, allyl, C3-C8-cycloalkyl, the latter being unsubstituted or substituted by 1-3 methyl groups, 2-hydroxyethyl, 3-hydroxypropyl, 2-hydroxypropyl or R<3> and R<4> (together) denote C4-C6-alkylene, -(CH2-CHX)2Y where X is H, CH3 and Y is O, S and their oligosulphide disproportionation products, whose average statistical chain length corresponds to S4 are prepared from the corresponding N,N'-substituted diaminomercaptotriazines. The substances according to the invention are used in vulcanisable rubber mixtures as crosslinking agents without sulphur or as vulcanisation accelerators together with sulphur.
Patent YU-37982-A (YU)
Title: Method of treating a coil surface
Inventor: HUEBECKER HANS
IPC: F16B33/06
Filed: 1982-02-19
Abstract: The surfaces of threads, sealing surfaces, and other load-bearing surfaces of oil field tubes or the like are treated by blasting surfaces to increase the roughness thereof to obtain a roughness of an average depth of from 7 to 15 micrometers under utilization of corundum or silicon carbide at a grain size of from 40 micrometers to 200 micrometers; a resin varnish is deposited onto the blasted surface for curing at higher than room temperature and including molybdenum sulfide at a layer thickness of from 5 to 20 micrometers. The varnish is cured in situ by heating.
Patent YU-47692-A (YU)
Title: Podizač ašova
Inventor: JANKOVIC Z
Filed: 1992-05-05
Abstract: Pronalazak se odnosi na podizač lista ašova koji omogućuje lakše riljanje zemlje. Na ašov i njegovu dršku se postavi jednokraka poluga podizača (1) pod uglom od 90В°C, koja se pričvršćuje pomoću dve obujmice, pri čemu se prva obujmica (2) pričvršćuje na ašov iznad lista pomoću dva zavrtnja (3) sa maticama (4), a druga obujmica (5) pomoću jednog eksera (6) na dršku ašova. Podizač za ašov ili druga ručna orudja za poljoprivredu radi na principu poluge, bez obzira na način pričvršćivanja na orudje i njegovu dršku.
Patent YU-54194-A (YU)
Title: Tripeptidna antitrombotička sredstva
Inventor: GESELLCHEN D P
IPC: A61K38/00
Filed: 1994-09-13
Abstract: TRIPEPTIDNA ANTITROMBOTIČKA SREDSTVA - opisana su jedinjenja formule 1, njihove farmaceutski prihvatljive soli i solvati formule Takođe je opisan postupak za dobijanje ovih jedinjenja koji obuhvata uklanjanje amino blokirajućih grupa iz intermedijera, hromatografisanje jedinjenja na reverzno faznoj hromatografskoj koloni sa visokim pritiskom tečnosti gradijentnim eluiranjem sa gradijentom koji obuhvata organsku fazu od oko 2 zapr% do oko 10 zapr% eluenta acetonitrila u vodenoj fazi koja obuhvata sumpornu kiselinu na pH između oko 2 i oko 3; podešavanje pH vrednosti eluata na oko 4 do 6 sa vodo-nerastvornom baznom smolom, izdvajanje smole iz eluata; i, uklanjanje vode iz eluata. Opisana jedinjenja predstavljaju inhibitore trombina i korisni su antikoagulanti.
Patent YU-83492-A (YU)
Title: Reaktivno-aktivni protivoklopni podkalibarni projektil
Inventor: MIROSLAV MITROVIC
Filed: 1992-09-14
Abstract: REAKTIVNO-AKTIVNI PROTIVOKLOPNI PODKALIBARNI PROJEKTIL, prema pronalasku, ostvaruje se tako što je u komoru impulsnog raketnog motora (6) umetnuta lansirna cev (5) u koju je smešteno izbacno punjenje (11) i pirotehničko-mehanički prenosnik (8), kojim se reguliše trenutak pripaljivanja izbacnog punjenja (11). U lansirnu cev (5) ulazi stabilizator (3) podkalibarnog projektila (1). Pri lansiranju projektila, impulsni raketni motor (6) daje početno ubrzanje, a izbacno punjenje (11) vrši razdvajanje impulsnog motora (6) od podkalibarnog projektila (1) dajući mu dodatno ubrzanje. Sagorevanje celokupnog pogonskog punjenja obavlja se u cevi lansera i time rešava tehnički problem.
Patent AT-A163599-A (AT)
Inventor: MEHRABI MOHAMMAD REZA
IPC: A61K31/5575
Filed: 1999-09-24
Abstract: The invention relates to the use of alprostadil for producing a medicament for angioneogenesis.
Patent AT-A255791-A (AT)
IPC: B65G37/00
Filed: 1991-12-23
Abstract: For the transportation of sealed insulating glass sheets with glass panes (1, 1') of different sizes, a conveying device is provided which has hook-like support elements (23) with pressure jaws (4) and bearings (3) for the smaller glass pane (1) and pressure jaws (25) and bearings (26), fixed on separate conveying chains (14') and (27), for the larger glass pane (1') which projects beyond the smaller glass pane (1). The conveying chain (27) with the bearings (26) is adjustable as to height, so that the pressure jaws (4) and (25) always engage, irrespective of the projection of the larger glass pane (1'), in the region of a spacer frame between the glass panes (1, 1'). 
<IMAGE>
Patent BE-822246-A (BE)
Title: Prefabricated frame for foundation of greenhouse - has aluminium sections bolted together over anchor bolts
IPC: A01G9/14
Filed: 1974-11-14
Abstract: Prefabricated frame which forms a foundation for a light building, such as a greenhouse or conservatory. It can be used, when assembled, as a template to mark out positions of foundation bolts. Anchor bolts with bearing plates at the end are buried in the ground with their threaded portion projecting. The frame is made of separate extruded aluminium sections with rebated corners, cut to length and bolted together (16, 18) using corner plates (20). These plates serve as fixing points for the bolts. After placing the assembled frame in position over these bolts, it is levelled up and secured using locking nuts and washers (28, 30).
Patent BE-902624-A (BE)
IPC: D02J1/22
Filed: 1985-06-07
Abstract: 1. Improved process for the stretching of synthetic filaments, especially filaments on a base of polypropylene or the like, composed of two steps, each of which corresponds to a partial stretching, the first step taking place under wet conditions by means of a filament feed mill (1) and a stretching mill (2), a liquid bath (3) and submerged guide rolls (4) being provided between these two elements (1, 2), the second stretching step using the stretching mill (2) of the first step, which now functions as a feed mill for the filaments laden with liquid as a result of their passage through the said bath (3), the said filaments being conveyed towards heated means of the second stretching step (6), characterized in that the said heated means are brought to a temperature higher than the fusion temperature of the filaments in the dry state.
Patent BE-904646-A (BE)
Title: Acide 7-amino-3-propenylcephalosporanique et ses esters.
IPC: C07D501/00
Filed: 1986-04-21
Abstract: Intermédiaires nouveaux de la céphalosporine, l'acide 7 betha-amino-3-((Z) -1- propen-1-yl) -3- céphem -4- carboxylique et ses esters ayant la formule générale,dans laquelle: la configuration du groupe 3-propényle est Z, souvent considéré comme cis-; et R est de l'hydrogène ou un groupe classique protecteur de carboxy, et leurs sels d'addition d'acides et sels métalliques du composé précité dans lequel R est un atome d'hydrogène.
Patent BE-905057-A (BE)
Title: Dispositif pour connecter une extremite d'une canule de distribution d'un medicament liquide a un appareil pour relier une seringe a une fiole contenant le medicament.
Inventor: VALENTINI LUIGI
IPC: A61M5/32
Filed: 1986-07-07
Abstract: Dispositif qui, lorsque la fiole a été enlevée, peut etre logé dans l'embase de l'appareil pour que l'aiguille puisse perforer un bouchon en caoutchouc prévu dans le dispositif ; le bouchon est connecté à une extrémité d'une canule, à l'autre extrémité de laquelle est montée, par exemple, une aiguille pour effectuer une transfusion. De cette façon, le liquide peut etre déchargé de la seringue pendant que l'aiguille est incorporée dans l'appareil et protégée par lui.
Patent BE-772488-A (BE)
Title: Deodorant compsn - comprising protease and ferrous salt
Inventor: HORN E T VAN
IPC: A61L9/01
Filed: 1971-09-10
Abstract: A mixt. of a proteolytic enzyme, having an activity of 748 u/g, and a ferrous salt, esp. FeSO4, forms a synergistic deodorant compsn. suitable for use on farms or establishments raising animals or birds, e.g. in dealing with offal or excrement. It is spread at the rate of >=98 g/m2, pref. 245-735 g/m2.
Patent BE-772734-A (BE)
Title: Chloramphenicol and thiamphenicol esters
IPC: A61K/
Filed: 1971-09-17
Abstract: Chloramphenicol and thiamphenicol esters. Cpds. of formula: (where R1 is Cl or Br; R2 is H, Cl, Br, lower alkyl, Ph, phenyl-lower alkyl, R3 is Cl, Br, lower alkyl, Ph or phenyl-lower alkyl. R4 is NO2 or CH3SO2-; R5 is H or -OCCR1R2R3) are antimicrobials active against chlor(and thi)amphenicol-resistant microbes and have improved taste. They can be prepd. by reacting chloramphenicol or thiamphenicol with R1R2R3CCOX (X = halogen), pref. in presence of an H halide acceptor.
Patent CA-1051384-A (CA)
Inventor: MOREY BOOKER W
IPC: B03C1/00
Filed: 1975-03-10
Granted: 1979-03-27
Abstract: ABSTRACT OF THE DISCLOSURE   The invention provides a method of separating non-magnetic conductive metal components from a mixture of non-magnetic conductive metal components and non-magnetic non-conductive material, including the steps of: generating a travelling electromagnetic wave from a linear motor stator with a frequency from about 400 to about 800 cycles per second; passing a stream of a mixture of non-magnetic conductive metal components of a size at least about 1/4 inch and non-magnetic non-conductive material through said travelling wave along the face of the linear motor stator on a moving belt spacing the mixture from said stator, with the direction of the linear motor travelling wave generally perpendicular to the direction of the stream of mixture, inducing eddy currents in the conductive metal components of the mixture producing forces acting on the conductive metal components in the direction of the travelling wave and moving conductive metal components from the stream along paths parallel to the stator face at a velocity substantially less than the velocity of the travelling wave, and collecting the components which are moved by the forces acting in the direction of the travelling wave.  There is also provided an apparatus for carrying out the method.  The invention offers advantages in the separation of non-magnetic, conductive metals from a mix-ture containing such metals together with non-magnetic, non-conductive metals, organic materials and non-metallic inorganic materials.
Patent CA-1055115-A (CA)
Inventor: NINOMIYA TAKESHI
IPC: H02P27/02
Filed: 1975-04-15
Granted: 1979-05-22
Abstract: ABSTRACT OF THE DISCLOSURE     A novel circuit is provided for controlling an alternating current supplied to a load which includes a variable impedance element in the form of a low emitter concentration transistor which is bidirection-al, and which has a high gain. The impedance of the variable impedance element to the flow of current therethrough is substantially the same in either direction of current flow.
Patent CA-1039758-A (CA)
Inventor: RAFF RUDOLPH A V
IPC: C04B5/00
Filed: 1975-04-24
Granted: 1978-10-03
Abstract: TITLE: LIGHTWEIGHT INORGANIC MATERIAL                    Abstract of the Disclosure A lightweight inorganic material containing fly ash cenospheres, phosphoric acid and metal phosphates.  The phosphoric acid and metal phosphates are initially contained in a liquid binder solution.  When combined with fly ash cenospheres and after heating of the combined mass to a temperature below the sintering temperature of the cenospheres, a rigid, lightweight inorganic material is produced which has particular value as a construction insulating material.
Patent CA-1046125-A (CA)
Inventor: ST LOUIS ROBERT M
IPC: D06F39/12
Filed: 1975-04-18
Granted: 1979-01-09
Abstract: ABSTRACT OF THE DISCLOSURE           A knockout portion is coined in a wall of a wrapper for an appliance.  The knockout has a second position, differing from its coined position, wherein it at least grossly reseals the opening.  Tabs are provided around the perimeter of the knockout so that when the knockout is in its second position a first edge portion of the knockout is supported by at least three interleaving tabs, there being at least one tab on each of the knockout and its opening. A further tab which may be on either the knockout or the perimeter of the opening supports a second edge of the knock-out generally opposed to the first edge, and a screw passing through the tab secures the knockout in position.
Patent CA-1058144-A (CA)
Inventor: AISHIMA ITSUHO
IPC: C08F10/00
Filed: 1975-05-12
Granted: 1979-07-10
Abstract: ABSTRACT OF THE DISCLOSURE        A process for polymerizing ethylene or a mixture of ethylene and another olefin is proposed in which the polymerization can be carried out with an extremely high efficiency by using a catalyst prepared by reacting (A) a hydrocarbon-insoluble reaction product (obtained by reacting (i) a specified organomagnesium-containing, hydrocarbon-soluble complex or reaction product of (i) with (ii) a specified siloxane compound, and (iii) at least one kind of titanium or vanadium compound containing at least one halogen atom), with (B) a specified organo-aluminum compound.  Resultant polymers have a high molecular weight and a high rigidity and molecular weight and molecular weight distribution thereof can be easily controlled.
Patent CA-1041149-A (CA)
Inventor: HOWARTH ANTHONY
IPC: F16C39/06
Filed: 1975-08-13
Granted: 1978-10-24
Abstract: ABSTRACT OF THE DISCLOSURE   The invention comprises an induction motor which comprises a ring stator formed of a plurality of poles each wound with a coil and a ring rotor floating above the stator ring which when the coil is energised rotates above the stator with a small air gap and when provided with vanes operates as a pump, fluid being fed to the motor and delivered therefrom. Alternatively the rotor may be sandwiched between two ring stators.  The motor may be employed as a pump, a conveyor or for cooling gasses from a nuclear reactor and other purposes, by providing a pressure head discharged across the rotor.
Patent CA-1046580-A (CA)
Inventor: STANTON DAVID J
IPC: G05F1/56
Filed: 1975-09-25
Granted: 1979-01-16
Abstract: ABSTRACT OF THE DISCLOSURE           A condition responsive control unit adapted to be connected to a condition sensor and which has its output current controlled in a modulated fashion between two cali-brated valves.  The current is applied to a modulating condition altering means, such as a special current modulated solenoid valve, or any other type of current operated load.  Two load control circuit means are used with a common output point to control the current between the two selected load control values.
Patent CA-1041651-A (CA)
Title: Method and system for sonic well logging
Inventor: INGRAM JOHN D
IPC: G01V1/44
Filed: 1975-11-13
Granted: 1978-10-31
Abstract: METHOD AND APPARATUS FOR ACOUSTIC LOGGING            OF A BOREHOLE                           Abstract A method and apparatus are described for preferentially exciting for extracting late arrivals at low frequencies in an acoustic investigation of a borehole.  The late arrival may be the Stoneley wave whose amplitude is derived by measuring the energy in a predetermined frequency band of a waveform produced with a low frequency transmitter-receiver system.  The transmitter produces a highly damped acoustic pulse whose frequency spectrum is selected to preferentially excite a late arrival such as the Stoneley wave and/or tube wave with wavelengths which are significantly greater than the diameter of the borehole while preserving measurable earlier arrivals at higher frequencies.  A receiver system is used which provides a generally flat frequency response including low frequencies to produce waveforms of both the earlier arrivals at high frequencies and late arrivals at low frequencies with sufficient extractable amplitudes throughout a wide range of borehole and formation conditions.  A method and apparatus are described for measuring inelastic behavior of the formation as well as elastic parameters such as the shear modulus of the material comprising the circumference of the borehole wall by investigating frequency bands in the spectrum of a late arrival such as the Stoneley wave.  A display and method for generating the display are described for the investigations of the late arrival.
Patent CA-1045922-A (CA)
Inventor: CAHN ROBERT P
IPC: F01K3/06
Filed: 1975-11-27
Granted: 1979-01-09
Abstract: ABSTRACT OF THE DISCLOSURE     More efficient use of the heat output of a constant output nuclear reactor, or constant output fossil fuel furnace, and boiler in an electricity generating plant that uses a multi-stage steam turbine and employs turbine extraction steam to preheat boiler feed water, is obtained by storing, during a period of low power demand, excess thermal energy in a liquid low vapor pressure thermal energy retention material maintained at high temperature at atmospheric pressure, and then, during a period of peak power demand, reducing or terminating the extraction of turbine steam and using the stored hot energy retention material, through heat exchange flow, to perform power plant support heating functions, including boiler feed water preheat and/or turbine interstage steam. The liquid heat retention materials include low vapor pressure organic materials such as hydrocarbon oils and aromatic ethers as well as molten metals, molten metal salts and molten metal hydroxides such as sodium hydroxide or potassium hydroxide.
Patent CA-1063516-A (CA)
Inventor: IMHOF PETER R
IPC: A61K31/21
Filed: 1976-01-02
Granted: 1979-10-02
Abstract: Abstract of the Disclosure Pharmaceutical preparations for the treatment of coronary heart diseases containing as pharmacological active comp-ounds a betareceptor-blocking compound and a compound which regulates the thrombocyte function,and, optionally, an alpha-receptor-blocking agent.
Patent CA-1057262-A (CA)
Inventor: WALKER RONALD J
IPC: B60R22/40
Filed: 1976-04-14
Granted: 1979-06-26
Abstract: Abstract of the Disclosure A retractor lock and pawl saddle combination for seat belt retractors and particularly inertial retractors in which the saddle supports the pawl or lock and the saddle is deformably installed in the retractor frame dimensionally supporting and journalling the shaft of the retractor drum and having a deflective portion in support of the pawl so that as the pawl engages the ratchet wheel, a portion of the saddle flexes guidably and the pawl is carried to thrust and lock abutment against the retractor frame. The flexing portion of the saddle supports an inertial sensor such as a pendulum and the pendulum upon movement pivots the pawl to engage the ratchet wheel.  The saddle pawl and sensor are preassembled and are then sprung into place between the upstanding walls of the retractor frame.
Patent CA-1041539-A (CA)
Inventor: KIMURA TSUNEO
IPC: C07C51/00
Filed: 1976-06-25
Granted: 1978-10-31
Abstract: PROCESS FOR PRODUCING TEREPHTHALIC ACID     Abstract of Disclosure:     There is disclosed a process for producing terephthalic acid in which the reaction temperature range and the proportion of catalyst components of a cobalt compound, a manganese compound and at least one bromine compound are specifically chosen to produce a high grade terephthalic acid suitable for direct polycondensation in the production of polyester.
Patent CA-1054527-A (CA)
Inventor: MORI YOSHIHISA
IPC: H04R1/16
Filed: 1976-07-05
Granted: 1979-05-15
Abstract: ELECTRODYNAMIC TRANSDUCER WITH ANNULAR GAP IN FLUX PATH          ABSTRACT OF THE INVENTION      An electrodynamic transducer comprising a source of magnetic flux and poles that define an annular gap in the flux path to obtain a radially oriented and uniformly dis-tributed magnetic flux across the gap.  Coils are mounted on a support that pivots universally about a center con-centric with the gap.  The coils are placed on the support so that pivotal movement of the latter causes a change in flux linkage with the coils.  The coils are wound in such a manner that the electric potentials generated in dia-metrically opposite coils are added together.  There may be sets of mutually perpendicular coils.