baber/WOPTO huggingface dataset:
Patent IL-122216-A (IL)
Title: Dolastatin derivatives as antineoplastics and their preparation
IPC: A61K38/08
Filed: 1996-06-03
Abstract: Peptides of the formula R1R2N - CHX - CO -A-B-D-E-(F)t-K where R1 is methyl, ethyl, or isopropyl; R2 is hydrogen, methyl, or ethyl; R1-N-R2 together may be a pyrrolidine ring; A is a valyl, isoleucyl, leucyl, 2-tert- butylglycyl, 2-ethylglycyl, norleucyl or norvalyl residue; B is a N-methyl-valyl, leucyl, -isoleucyl, -norvalyl, -norleucyl -2-tert-butylglycyl, -3-tert-butylalanyl, or 2-ethylglycyl residue; D is a prolyl, 3,4-dehydroprolyl, 4-fluoro-prolyl, 4,4-difluoroprolyl, azetidine-2- carbonyl, homoprolyl, 3-methylprolyl, 4-methylprolyl, 5-methylprolyl, or thiazolidine-4- carbonyl residue; E is a 3,4-dihydroprolyl, 4-fluoroprolyl, 3-methylprolyl, 4-methylprolyl, azetidine-2- carbonyl, or 4,4-difluoroprolyl residue; F is a valyl, 2-tert-butylglycyl, isoleucyl, leucyl, 2-cyclohexylglycyl, norleucyl, norvalyl, neopentylglycyl, alanyl, b-alanyl, or aminoisobutyroyl residue; X is alkyl (preferably C2-5), cyclopropyl, or cyclopentyl; t is 0 or 1; and K is alkoxy (preferably (C1-4), benzyloxy or a substituted or unsubstituted amino moiety; and the salts thereof with physiologically tolerated acids. 3629 כ" ח בשבט התשס" ב - February 10, 2002
Patent IL-123486-A (IL)
Title: Display screens incorporating loudspeakers
IPC: G03B21/56
Filed: 1996-09-02
Abstract: A display screen (32), e.g. a projection screen comprising a panel having a light reflective surface, characterised in that the screen is a distributed mode acoustic radiator loudspeaker having a transducer (9) mounted wholly and exclusively thereon to vibrate the radiator to cause it to resonate to provide an acoustic output.
Patent IL-126028-A (IL)
Title: Injection device with electronic presentation of set doses
IPC: A61M/
Filed: 1997-03-03
Abstract: An injection device has signal generators (11, 12, 13, 14) which are connected to operative elements (8, 3, 5, 4) of the device and which give off signals which represents the operative condition of the device. The signals are sent to an electronic circuit which controls a presentation of the operational condition of the device and presents operational conditions, which are defined as not allowed, as error indications by switching off the display presenting the operational condition of the device. The number of signals from each generator is counted and a number of operations exceeding a pre-set number for the signal generator in question is interpreted as representing a not allowed operational condition.
Patent IL-133394-A (IL)
Title: Process for the preparation of macrocylic chelants and the chelates thereof with paramagnetic metal ions
IPC: C07D257/02
Filed: 1998-06-03
Abstract: A process for the preparation of complexes of macrocyclic chelants with paramagnetic metal trivalent ions of formula (XII) wherein R1, R2 and Me3+ are as described in the following, comprising: a) reaction of 1,4,7,10-tetraazacyclododecane with triethyl orthoformate to give 5H,9bH-2a,4a,7,9a-octahydrotetraazacycloocta[cd]pentalene; b) carboxymethylation reaction in water; c) hydrolysis reaction in basic conditions; d) alkylation according to known methods with an epoxide in water; e) complexation according to known methods carried out in water by addition of a paramagnetic metal salt; f) purification by diafiltration, final desalting of the aqueous solution on ion exchange resins and g) crystallization or recovery.
Patent IL-141690-A (IL)
Title: Process for preparation of rasagiline and its salts
IPC: C07C209/88
Filed: 2001-02-27
Abstract: A process for the optical resolution of racemic N-benzyl-1-indanamine, characterized in that it is carried out using (R, R)-tartaric acid as the optical resolving agent, to form N-benzyl-l-indanamine (R, R)-tartrate. 1512 א' בתמוז התשס" ד - June 20, 2004
Patent IL-147732-A (IL)
Title: Aerated frozen products
IPC: A23L29/10
Filed: 2000-07-03
Abstract: A process for the production of aerated frozen products by preparing a mixture of ingredients suitable for a frozen aerated product, adding an emulsifier mixture, aerating the mix to obtain an aerated mix having an overrun of about 20% to about 250% and about 5% to about 100% for the aerated frozen ice cream and water ice, respectively, and freezing the aerated mix to produce the aerated ice cream or water ice.
Patent IL-147867-A (IL)
Title: Anti-reflection coatings and coated articles
IPC: G02B1/11
Filed: 2000-07-27
Abstract: A transparent or translucent coated article, comprising an optical substrate and one or more layers of anti-reflection material coated on at least a portion of the optical substrate, characterized in that said one or more layers having a thickness such that the article simultaneously has (i) a color, when viewed at a specified angle or angles, under a specified illumination, that is perceived to lie within a specified volume element of color space defined by the color's CIE chromaticity coordinates, and (ii) a perceived reflectance F=««S(»,¸)R(»,¸)d»d¸ that is less than or equal to 1.25F min , wherein » is wavelength, ¸ is incident angle, S(»,¸) is the human sensitivity function as a function of wavelength and incident angle, R(»,¸) is an average of p- and s-polarized reflectance, and F min  is perceived reflectance minimized within the constraints imposed by said chromaticity coordinates.
Patent IL-153239-A (IL)
Title: Stabilisation of light sensitive substances
IPC: C09K23/52
Filed: 2002-12-03
Abstract: An emulsion comprising an organic discontinuous phase which is distributed throughout a continuous aqueous phase, wherein the organic phase comprises a light sensitive active ingredient, and the emulsion is stabilised by a water soluble stabilising material in the aqueous phase, wherein the water-soluble stabilising material is a water-soluble stabilising polymer which has a plurality of hydrophilic and hydrophobic groups and is selected from partially hydrolysed polyvinyl acetate and addition copolymers formed from (i) at least one ethylenically unsaturated carboxylic acid esters and (ii) at least one ethylenically unsaturated carboxylic acid or ethylenically unsaturated carboxylic acid anhydride, and wherein the organic phase further comprises, a) an organic solvent which is a liquid at 25° C. and/or b) an organic phase stabilising material comprises hydrophobic moieties and is a material which is more soluble in the organic phase than the aqueous phase. The composition is useful for protecting light sensitive active ingredients which would otherwise in neat form decompose on exposure to light, preferably sunlight. The invention is of particular value when the light sensitive active ingredient is a pesticide, herbicide or a veterinary treatment active. Preferably the light sensitive active ingredient is a light sensitive pyrethroids. The invention also contemplates a domestic pest control formulation comprising light sensitive pesticides.
Patent IL-155702-A (IL)
Title: Piperazinylpyrazine compounds, pharmaceutical compositions comprising them and use thereof in the preparation of medicaments for the treatment of serotonin related medical conditions
IPC: A61K31/506
Filed: 2003-05-01
Abstract: A compound of the general formula (I), wherein R1, R2, X, Y and Z are as described in the specification.
Patent IL-164547-A (IL)
Title: Pharmaceutical composition comprising an androgen, a hsieh enhancer and a thickener
IPC: A61K31/56
Filed: 2004-10-13
Abstract: A pharmaceutical composition comprising: (A) an androgen; (B) a cyclic enhancer of the type used in the compositions and methods claimed by U.S. Pat. No. 5,023,252 to Hsieh; and (C) a thickening agent; including, for example, a composition in which the cyclic enhancer is a macrocyclic ester or a macrocyclic ketone; the use of the composition to treat a condition, for example, male hypogonadism, in a patient by applying the composition to the membrane of the patient; and a method for making the composition.
Patent IL-185545-A (IL)
Title: Method of preparation of pure 4-pyrrolidinophenylbenzyl ether derivatives and intermediate compounds
Filed: 2007-08-27
Abstract: The invention relates to a method for preparing enantiomerically pure 4-pyrrolidinophenylbenzyl ether derivatives of formula I: wherein R1, R21, R22, R23, R24 and n are as defined in the description and claims and to intermediates useful in the method of the invention as well as salts thereof.
Patent IL-201674-A (IL)
Title: Methods for producing proteins with predetermined post-translational modifications
Inventor: BOUT ABRAHAM
IPC: A61P25/28
Filed: 2009-10-21
Abstract: The present invention provides methods for identifying, selecting and obtaining mammalian cells that are capable of producing proteinaceous molecules comprising predetermined post-translational modifications, wherein said post-translational modifications are brought about by the mammalian cell in which the proteinaceous molecule is expressed. Preferably, said predetermined post-translational modifications comprise glycosylation. The invention further provides methods for obtaining and producing proteinaceous molecules, using mammalian cells obtainable by a method of the present invention. Preferably said proteinaceous molecules comprise erythropoietin (EPO), since the effect of (recombinant) EPO depends heavily on the glycosylation pattern of the oligosaccharides present on the protein. Mammalian cells that have been obtained on the basis of their ability to produce proteins and/or post-translational modifications that are indicative for a predetermined post-translational modification that is desired are also provided. Preferably, said mammalian cells have neural characteristics and properties such that significant amounts of recombinant proteins can be produced that harbor 'neural- or brain-type' properties
Patent IL-205533-A (IL)
Title: Partial solvent stripping process for recovering brominated butadiene polymers from solution
IPC: C08C/
Filed: 2010-05-04
Abstract: Brominated butadiene polymers are recovered from a bromination reaction solution by partially stripping the solvent to form a concentrated solution or slurry, and then recovering the brominated butadiene polymer from the concentrated solution or slurry. The process allows for a simplified, effective an economical recovery of the brominated butadiene polymer. Brominated butadiene polymers recovered in this manner are often very thermally stable.
Patent JP-S5625635-A (JP)
Title: Apparatus for indicating clogging of air filter used in air conditioner
Inventor: SHIMIZU KEIICHIROU
IPC: F24F13/28
Filed: 1979-08-08
Abstract: PURPOSE:To detect and indicate the clogging of a filter used in an air conditioner correctly, by providing in the main circuit of a motor connected to a fan a relay which is set into operation depending on the value of current passed in said main circuit, and setting the relay into operation when the value of current is varied due to clogging of the air filter. CONSTITUTION:When a push button switch 12 for starting air blowing operation is closed and then another push bottom switch 13 for starting heating or cooling operation of the air conditioner is also closed, current is passed through the coil of electromagnetic switches 52F, 52C and their contacts are closed, so that a fan motor FM and a compressor motor CM are set into operation. As the air filter 6 is clogged along with operation of the air conditioner, resistance to air flow through the air filter 6 is increased and load of the fan motor FM is lowered. Therefore, when the current is lowered to a certain value, overload relay 11 is set into operation and its contact is closed, thereby setting a buzzer 14 into operation. By the operation of the buzzer 14, it is known that the air filter 6 is clogged to such an extent requiring its cleaning.
Patent JP-H11281241-A (JP)
Title: Low-temperature show case
Inventor: HAYASHI HIROSHIGE
IPC: F25D23/06
Filed: 1998-03-27
Abstract: PROBLEM TO BE SOLVED: To suppress the inclination of a side plate, by equipping a side plate with a cut for avoiding a spacer inserted into the center of a groove when the bottom of the side plate is set in the groove opened at the top of a heat insulating wall. SOLUTION: A storage room 6 is demarcated in the space surrounded by a heat insulating wall 5 and side walls 10 and 10, and transparent glass 7 is set to the top of the front wall 5A (rear wall) of the heat insulating wall 5 to enable a customer to see through the interior of the storage room 6. A machine room is constituted at the lower part of a heat insulating box 2, and a compressor, a condenser, etc., constituting the freezing cycle of a cooler are installed. The chill cooled with a cooler is circulated within the storage room 6 so as to cool it to a specified freezing temperature. A groove which opens in longitudinal direction is made integrally at the center in the width direction of a breaker. A cut is made in a roughly trapezoidal shape at the center in the longitudinal direction of the bottom of the side plate 51.  The cut avoids the spacer, corresponding to the spacer within the groove, and the projection can be inserted to the inner part before and behind the spacer.
Patent JP-S60243606-A (JP)
Title: Thin film optical element
Inventor: MIYAWAKI MAMORU
IPC: G02B6/122
Filed: 1984-05-17
Abstract: PURPOSE:To obtain an optically functional element having high threshold value of optical damage without decreasing deflection efficiency by setting the absorption peak of the infrared spectrum of OH group due to the proton of an optical waveguide layer to a specified range of the wave number. CONSTITUTION:Laser light 6 is conducted from a grating optical coupler 3 to an optical waveguide layer 2 formed by the thermal diffusion of Ti and proton on an x-plate or y-plate LiNbO3 crystal substrate 1 so as to result an absorption peak of infrared absorption spectrum of OH group due to proton to be in a range between 3,480-3,503cm<-1> wave number. The waveguided light is diffracted by a phase lattice by impressing a voltage to a comb-shaped electrode 11 for the electrooptic effect, and is taken out to the outside from a grating optical coupler 4. In this case, a high diffraction efficiency as high as 90% is obtd. by impressing 6V voltage on the electrode 11.
Patent JP-S59227027-A (JP)
Title: Magnetic recording medium
Inventor: HOSAKA AKIHIKO
IPC: C09D127/04
Filed: 1983-06-07
Abstract: PURPOSE:To improve an electromagnetic conversion characteristic, especially a high-output property, an S/N characteristic, and a physical characteristic by composing a binder in magnetic paint of polyurethane, vinyl chloride-vinylidene chloride, and cellulose nitrate resins in a specified ratio. CONSTITUTION:The binder is characteristically composed of 30-64wt% polyurethane resin, 10-45wt% vinyl chloride-vinylidene chloride resin, and 15- 40wt% cellulose nitrate resin. The polyurethane resin is usually the reaction product of diisocyanates and a compd. such as glycol having hydroxy groups, and the compd. having terminal OH groups is especially preferable ''Denka Vinyl 1,000W and 1,000WK'' manufactured by the Denki Kagaku Kogyo Company can be used as the vinyl chloride-vinylidene chloride resin. The cellulose nitrate is the nitrate ester of cellulose and is also called nitrocellulose. When any of the three components is beyond said specified range, one of the characteristics indispensable to the magnetic recording medium is damaged.
Patent JP-H11246769-A (JP)
Title: Preparation of organosilicon polymer emulsion
Inventor: MORITA YOSHIJI
IPC: C08L83/05
Filed: 1998-03-27
Abstract: PROBLEM TO BE SOLVED: To provide a preparation process of an organosilicon polymer emulsion having a small particle size and a high stability, wherein an organosilicon polymer having a siloxane bond and a silalkylene bond are emulsified in water. SOLUTION: A diorganopolysiloxane having silicon atom-bonded hydrogen atoms only at both ends of the molecular chain and a diorganopolysiloxane having silicon atom-bonded alkenyl groups only at both ends of the molecular chain are addition polymerized in water in emulsified states using a hydrosilation catalyst. Preferably, an emulsion prepared by emulsifying in water a liquid catalyst which comprises a platinum-alkenyl siloxane complex as the main component is used as the hydrosilation catalyst.
Patent JP-S5528523-A (JP)
Title: Signal charge input system for charge transfer element
Inventor: IIDA TETSUYA
IPC: H03H7/30
Filed: 1978-08-17
Abstract: PURPOSE: To cut off the charge transfer element with the fixed external DC voltage at all times by detecting previously the difference of the interanl potential under the 1st and 2nd gates and using the voltage to correct the external DC voltage.  
     CONSTITUTION: With supply of the pulse to charge supply source 2, the potential features VSH at the high level of the pulse and VSL at the low level respectively. At the part of gate G 1 , the level of potential V 1  is decided by DC bias VIB and input signal source 4; while the level of potential V 2  is decided with output voltage VADJ of DC voltage shift circuit 5 each. With supply of the pulse to gate G 3  from pulse supply source 6, the potential features VSH and VSL with the high and low levels of the pulse respectively. The charge amount transferred into the the CCD is proportional to voltage VADJ and then cut off at the low level. Voltage VADJ is not  constant and varied with dispersion of the manufacture time of the element. In  this connection, the potential difference is detected previously under gates G 1  and  G 2 , and external DC voltage VIN is corrected with the difference voltage to secure  the CCD cut-off state. 
     COPYRIGHT: (C)1980,JPO&Japio
Patent JP-H02279583-A (JP)
Title: Method for growing single crystal
Inventor: KUWANO YASUHIKO
IPC: C30B15/18
Filed: 1989-04-19
Abstract: PURPOSE:To grow the single crystal from a melt without contg. a flux by using a system for directly heating a crucible for heating in order to melt materials by a high frequency induction current at the time of pulling-up and growing the beta-BaB2O4 single crystal. CONSTITUTION:The solidified matter of beta-BaB2O4 is melted and packed into a platinum crucible 1. The raw materials in the crucible 1 are gradually melted by a high frequency coil 2 without overheating the crucible 1 to form the raw material melt 3 which is then subjected to an ordinary pulling-up by using a seed crystal 6 to grow the beta-BaB2O4 (beta-barium borate) single crystal. The good quality product which is large in size and contains impurities at a lower ratio is obtd. in the growing time of 1/5 to 1/10 the growing time of the conventional flux-growing method.
Patent JP-H02278385-A (JP)
Title: Picture processing circuit
Inventor: TERAI HIROYUKI
IPC: G06T7/00
Filed: 1989-04-19
Abstract: PURPOSE:To obtain a mean density value by supplementing a circuit which accumulates successively one line of data read out in a horizontal direction and the circuit which inputs a read in density value to the shift register of the portion of the number of picture elements in the horizontal direction and sums the output of the shift register and the density value in succession. CONSTITUTION:The picture processing circuit is constituted as including a horizontal picture cumulative memory 5 which stores an accumulated result signal (g) in each address designated by an address signal (h), a second adder 8 which is initialized by a clear signal (k) and adds the density signal (c) and a shift data signal (j) and outputs a second added value signal (i), the shift register 9 which delays the added value signal (i) by one horizontal line portion and sends the shift data signal (j) toward the adder 8 and has the same number of stages as the number of the picture elements in the horizontal direction of a digital picture, and a vertical picture cumulative memory 10 which stores the added value signal (i) in each address designated by an address signal (l). The cumulative density value of every horizontal line of the digital picture is stored in the vertical picture cumulative memory 10, and the data of a lower order bit is cut optionally. Thus, the mean horizontal density value can be obtained.
Patent JP-H04309672-A (JP)
Title: Air-tight and heat insulating underfloor structure for bathroom or the like
Inventor: ISHIKAWA OSAMU
IPC: F24F7/10
Filed: 1991-04-05
Abstract: PURPOSE:To obtain the air-tight and heat-insulating underfloor structure for bathroom or the like with the simple structure having high insulating property to improve the heat insulation efficiency of a bathroom and prevent cooling of the floor of the bathroom or the like. CONSTITUTION:The underfloor of a bathroom or the like 1 is formed into a closed space 5, and a suction port 11 communicated with this closed space 5 is provided in a toilet B. In a bathroom A, a clearance 15 is provided between a wall panel 13 and a bath unit 14 so as to be communicated with the closed space 5. The conditioned air inside of a building, which is conditioned at a predetermined temperature, is led from the toilet B into the closed space 5, and furthermore, the conditioned air is led from this closed space 5 to the clearance 15 inside of the bathroom A, and furthermore, it is exhausted to the outside.
Patent JP-H08269914-A (JP)
Title: Anchor cap with spiral reinforcement for bridge
Inventor: ARITA MASAHIRO
IPC: E01D19/04
Filed: 1995-03-30
Abstract: PURPOSE: To provide an anchor cap with a spiral reinforcement for a bridge which is simple in structure, and can be certainly arranged, connected and fixed at a central position between the anchor cap and the spiral reinforcement by a simple work process. CONSTITUTION: In an anchor cap with a spiral reinforcement for a bridge composed of a circular spiral reinforcement 2 and an anchor cap 12 arranged in the spiral reinforcement 2, projection parts 17, 18 extending in the axial direction of the spiral reinforcement 2 are formed protrusively toward the spiral reinforcement 2 in the anchor cap 12. A connecting jig which arranges the anchor cap 12 at a fixed position in the spiral reinforcement 2 by an engagement with the projection parts 17, 18, and connects and fixes it to the spiral reinforcement 2 is provided between the anchor cap 12 and the spiral reinforcement 2.
Patent JP-S5626660-A (JP)
Title: Molten metal cooling vessel of superior electromagnetic rabbling performance for molten metal
Inventor: HIDEMIYAMURA HIROSHI
IPC: B22D11/043
Filed: 1979-08-07
Abstract: PURPOSE:To perform superior electromagnetic rabbling by segmenting the wall of a molten metal cooling vessel provided with an electromagnetic induction device on the outside circumference of the vessel in the thickness direction and forming a minute clearance communicating the segments. CONSTITUTION:A cooling vessel 1 is formed by thermoconductive material such as, for example, Cu, and has a lower opening. This is segmented in the thickness direction of the vessel wall and a minute clearance 3 of a suitable length communicated at one or both ends with the end edge 2 of the vessel is provided along the wall. Because of this, there is the effect of dispersing the clearances that are produced between the vessel wall and frozen shell and become the hindrance for heat transfer. When a thick-walled steel plate (20mm.) is used and electromagnetic rabbling frequency of 60Hz is used, the rabbling thrust of 5-9 times higher than that of conventional methods is obtainable.