baber/WOPTO huggingface dataset:
Patent CS-271489-B2 (CS)
Title: Method of alkylsulphonamidophenethylamines' sulphonamidoderivatives production
Inventor: CROSS PETER EDWARD DR
IPC: C07D333/66
Filed: 1988-05-23
Abstract: The method of production of sulfonamide derivates of alkyl sulfonamide phenethylamines is of a general formula I, where alk is C1-4-alkyl, R<1> is C1-4-alkyl and Het is the rest of the formula E, F or G, in which R<2> is hydrogen, methyl or ethyl, X is oxygen, sulphur or the rest of NR<4>, where R<4> is hydrogen or methyl and their pharmaceutically utilizable salts, characteristic by the fact that a compound of the general formula B, where R<a> is an amino group or the rest NHSO2alk and Het is the rest of the formula E, F or G; which can instead of -NHSO2alk configuration contain also an amino group providing that in the starting substance molecule there is at least one amino group is let to react with the C1-4-alkansulfonylchloride or -bromide or with an anhydride of C1-4-alkan-sulphonic acid. Finally the product of the general formula I is converted to salt. The produced compounds are efficient as anti-arrhythmic active substances and can be used in pharmaceuticals.<IMAGE>
Patent CS-212236-B2 (CS)
Title: Device against the density differences of the fabric by the start in the loom
Inventor: DEBORDE ALBERT H
IPC: D03D49/04
Filed: 1979-07-16
Abstract: A weaving loom is equipped with a system for controlling oscillation of a warp yarn support roller in which a first rotary cam actuates an oscillating first lever connected to a first arm integral with a first shaft on which the roller is mounted. The first shaft rests, through the intermediary of raising members, in bearings supported by second levers pivoting about a fixed pivot and connected, through the intermediary of pivoted connecting rods, to the third and fourth levers which are keyed to a second shaft and subject to urging by at least one spring. The system includes a fifth lever keyed to the second shaft and a second rotary cam actuating an oscillating sixth lever pivotably connected to a second arm which is alongside the fifth lever and is freely mounted on the second shaft. A fixed first hook is mounted on the second arm and a pivotable second hook is mounted on the fifth lever. An electromagnet holds the second hook clear of the first hook except when the loom is being started. In this event the second cam causes the second arm to pivot downwards about the second shaft so that the first hook pushes the second hook downwards causing the fifth lever to pivot downwards and rotate the second shaft. This rotation throws the connecting rods which pivot the second levers which move the support roller transversely to warp yarn passing thereover to increase tension in the yarn.
Patent JP-H0784726-B2 (JP)
IPC: E01F9/04
Filed: 1987-01-12
Abstract: Pavement marking (I) comprises ceramic microspheres (II) held by a binder (III), (II) being solid transparent non-vitreous microspheres with at least one crystalline phase comprising at least one metal oxide other than TiO2 (although a small amt. of this may be present), and having particle size up to 125 microns. A similar compsn. is also claimed, in which the microspheres are of fully dense silica, up to 125 microns. Coating compsns. having these constitutions are also claimed. Pref. the binder consists of paint or thermoplastic resin.
Patent JP-3103979-B2 (JP)
IPC: G01M11/02
Filed: 1987-01-17
Granted: 2000-10-30
Abstract: A method for evaluating the in vivo ability of a contact lens to become or remain wet includes the steps of supporting the subject's head to determine a fixed orientation of the lens, illuminating the lens with coherent light, imaging the pre-lens tear film in a manner to form an interference pattern, recording in a time sequence manner the image formed thereby, and determining the tear film thickness by correlating the interference bands of the recorded image. The classical contact angle is derived, and other measures, such as the time interval from blink until the onset of tear film breakup, or the time until the film evaporates, and the initial or average film thickness are derived. In addition, the nature and evolution of localized dry spots may be directly observed, clarifying the causes of tear film breakdown on worn contact lenses. The invention enables wetting characteristics to be evaluated as they are affected by lens material, lens aging and lens soiling, as well as the evaluation of solvents, additives and cleaners, for their effects on wetting characteristics.Apparatus for performing the method includes means for supporting the head so as to determine a fixed location of the contact lens (8), a coherent light source (9), and a camera (19) focused at the pre-lens film from a position to image light from the source specularly reflected from the front and rear surfaces of the tear film. A film motion analyzer (50) provides numerical coordinates of interference bands, and a microprocessor (60) analyses the coordinates to provide a quantitative measure of lens position or wetting characteristics.
Patent AU-556922-B2 (AU)
Title: Pyridobenzodiazepinone derivatives
Inventor: SCHMIDT GUNTER
IPC: C07D471/04
Filed: 1983-02-08
Granted: 1986-11-27
Abstract: This invention relates to compounds of the formula    <IMAGE>  (I) wherein R is (1-methyl-4-piperidinyl)methyl, (1-methyl-1,2,5,6-tetrahydro-4-pyridinyl)methyl, 1-methyl-1,2,5,6-tetrahydro-4-pyridinyl, (1-methyl-4-piperidinylidene)methyl, 2,3-dehydro-8-methyl-8-azabicyclo[3.2.1]oct-3-yl methyl, endo-8-methyl-8-azabicyclo[3.2.1]oct-3-yl-methyl, or exo-8-methyl-8-azabicyclo[3.2.1]oct-3-yl-methyl, each of which may optionally have one or two methyl substituents on the six-membered heterocyclic ring, and non-toxic, pharmacologically acceptable acid addition salts thereof. The compounds as well as their salts are useful as anti-ulcerogenics.
Patent AU-571434-B2 (AU)
Title: Ethers and oxime ethers of alkylaminoalcohols
Inventor: LECLERC GERARD
IPC: A61K31/13
Filed: 1983-02-18
Granted: 1988-04-21
Abstract: Glaucoma can be treated by the application to the eye of a physiologically active amount of a compound of the formula   <IMAGE> in which: each of R3 and R4 is selected from hydrogen, and alkyl, alkenyl and cycloalkyl radicals, or R3 and R4 together with the carbon between them are a cycloalkylidene radical, R2 is a lower alkyl radical, and the salts thereof with pharmaceutically acceptable acids, in an opthamologically accepted carrier therefor, which when liquid and an isotonic agent is present can have the form of an eye lotion. The 1-N-tert.-butylamino derivatives of 3-(cyclopropyl-methyl-ketone-oximino)-propan-2-ol, 3-(dicyclopropyl-ketone-oximino)-propan-2-ol, and 3-(3,3,5-trimethylcyclohexane-1-ketone-oximino)-propan-2-ol are novel compounds within such formula specifically useful for such treatment.
Patent AU-554716-B2 (AU)
Title: Tubular die for the continuous casting of a thin-walled tube from cast iron
Inventor: BELLOCCI RIO
IPC: B22D11/00
Filed: 1983-03-01
Granted: 1986-08-28
Abstract: The die (6) comprises a thick cylindrical body (7) which is surrounded by a cooling jacket (15) clamped against the pouring basin (2) and in contact with the latter in a plane (P). The body (7) is extended in the casting orifice (4) by a composite head (17) comprising a thin inner annular lip (22), whereof the inner surface extends that of the body (7) and a ring (24) of refractory material fitted between the lip, the body and the casting orifice. The (hot) lip (22) is connected to the body (7) in the plane (P), so that the ring (24) rejoins it also in this plane and that the flow of heat (f1) passing from the casting orifice to the cooling jacket must skirt around this ring.
Patent AU-774148-B2 (AU)
Title: System for repairing bituminous wearing courses
Inventor: GOODHART JONATHAN LUKE HENRY
IPC: C09D195/00
Filed: 1999-11-25
Granted: 2004-06-17
Abstract: The invention provides a method for repairing a damaged area of a bituminous wearing course. The method comprises heating the damaged area, applying a liquid to the damaged area that rejuvenates damaged bitumen, adding new material to the damaged area in an amount required to level the area, and compacting the new material. The invention also provides a new composition for rejuvenating damaged bitumen. The composition may comprise an emulsifier, a heavy paraffinic distillate solvent extract, a heavy naphthenic distillate solvent extract and water.
Patent AU-780142-B2 (AU)
Title: Compositions and methods for treating conditions responsive to estrogen
Inventor: THOMPSON DAVID DUANE
IPC: A61K31/4035
Filed: 2001-01-11
Granted: 2005-03-03
Abstract: This invention relates to methods, pharmaceutical compositions and kits useful in treating conditions responsive to estrogen by the administration of estrogen agonists / antagonists. Conditions responsive to the compositions and methods include rheumatoid arthritis, colon cancer, tissue wounds, skin wrinkles and cataracts. The compositions are comprised of an estrogen agonist / antagonist and a pharmaceutically acceptable vehicle, carrier or diluent. The compositions and methods of treatment are effective while substantially reducing the concomitant liability of adverse effects associated with estrogen administration. <IMAGE>
Patent AU-742021-B2 (AU)
Title: Hair colorant preparation
Inventor: HOFFKES HORST
IPC: A61K8/64
Filed: 1998-11-28
Granted: 2001-12-13
Abstract: The invention relates to a hair colorant comprised of a flowable, aqueous preparation of oxidation colorant intermediate products (A) and a flowable, aqueous oxidation agent preparation (B) which are mixed in a weight ratio A:B=1:2 to 2:1 to produce a gel-forming coloring batch immediately before applying on the hair. As supporting components in the oxidation colorant preparation, the hair colorant comprises 3.0 to 15 wt. % of a saturated or unsaturated, linear or branched alcohol with 8 to 36 C-atoms, 0.1 to 20 wt. % of a low-molecular water-soluble alcohol, 0.1 to 15 wt. % of a liquid fatty acid with 16 to 22 C-atoms in the form of a water-soluble soap, 0.1 to 20 wt. % of an addition product of 1 to 5 mole ethylene oxide on a linear fatty alcohol with 8 to 22 C-atoms and/or 0.1 to 15 wt. % of an optional alkoxylated amine. The oxidation agent preparation (B) preferably comprises 3 to 12 wt. % hydrogen peroxide, 0.1 to 5 wt. % of a water-soluble, synthetic tenside and 1 to 5 wt. % of a dispersed acrylic acid polymerizate or copolymerizate and/or methacrylic acid polymerizate or copolymerizate.
Patent AU-640565-B2 (AU)
Title: Polyamines useful as antagonists of excitatory amino acid neurotransmitters
IPC: A01N43/38
Filed: 1992-04-30
Granted: 1993-08-26
Abstract: A substantially pure compound, derived from the venom of Agelenopsis aperta spider, of the formula <CHEM>  wherein each R is the same and is H or OH. The polyamines of this invention and the salts thereof antagonize excitatory amino acid neurotransmitters, which neurotransmitters affect cells of various organisms, and are useful in antagonizing said neurotransmitters, per se, in the treatment of excitatory amino acid neurotransmitter mediated diseases and conditions and in the control of invertebrate pests.
Patent AU-553793-B2 (AU)
Title: Electrolytic cell with plurality of electrode units
Inventor: LOHRBERG KARL
IPC: C25B9/19
Filed: 1983-06-24
Granted: 1986-07-24
Abstract: In an electrolytic cell having a membrane and vertical electrodes composed of a plurality of units, a. the electrode having one polarity is horizontally divided into a plurality of units, b. the electrode having the opposite polarity is vertically divided into a plurality of units, and c. the units of at least one of the two electrodes are adapted to be displaced by spring elements. Spacers are suitably provided between the units of that electrode which is not contacted by the membrane.
Patent AU-777150-B2 (AU)
Title: Intraocular lens implanter
Inventor: HJERTMAN BIRGER
IPC: A61F9/007
Filed: 2000-11-29
Granted: 2004-10-07
Abstract: A device for deforming and ejecting a deformable intraocular lens for insertion into a small incision in an eye, the device comprising a) a housing, b) a lens transporting duct in a front part of the housing defining a duct axis, the duct having a front end with a cross-section adapted to the lens in deformed state with small maximum dimensions transversal to the duct axis, a rear lens-receiving end with a cross-section adapted for the lens in un-deformed state, or less deformed state, than at the front end, with larger maximum dimensions lateral to the duct axis than at the front end and an intermediate convergent duct part between the front and rear ends with a varying cross-section shape, having decreasing maximum dimensions lateral to the duct axis when moving from rear to front in the duct and c) a plunger operative to displace the lens in the duct at least in the forward direction. According to various aspects of the invention part of the duct has the overall shape of a crescent, the plunger is re-shapeable between different height to width ratios, the device has fixing structures for preventing lens rotation and the plunger is driven with a preprogrammed movement pattern. The invention also includes methods corresponding to the operational steps of the devices.
Patent AU-701672-B2 (AU)
Title: Testicular prosthesis and method of manufacturing and filling
Inventor: PETRICK TIMOTHY B
IPC: A61F2/02
Filed: 1995-03-03
Granted: 1999-02-04
Abstract: Testicular prosthesis and method of manufacturing wherein the testicular prosthesis has a saline or other biologically safe fluid filled silicone elastomer shell which includes a self-sealing injection site for filling the prosthesis and a tab for suturing the testicular prosthesis into position in the scrotum. A method of filling and a method of identifying and serialization is also provided.
Patent AU-761937-B2 (AU)
Title: Apparatus and method for a custom soft-solid hearing aid
Inventor: JUNEAU ROGER P
IPC: C12Q1/34
Filed: 1998-12-18
Granted: 2003-06-12
Abstract: A hearing aid instrument of the in-the-ear type (and preferably CIC) provides a receptacle with electronic hearing aid components mounted thereto. The receptacle has a cavity for holding electronic components (eg. battery, microphone, amplifier). A soft polymeric body is preliminarily formed by encapsulating a plurality of the electronic hearing aid component shaped inserts. The body is soft and is shaped to conform to the ear canal of the user. After forming, the insert is removed to provide an insert cavity that can carry electronic components. The soft polymeric body and encapsulated electronic hearing aid components define a soft structure compliant to the ear canal during use and that is substantially solid and free of void spaces between at least some of the components and the ear canal. This combination of soft compliant structure and encapsulated electronic hearing aid components addresses problems of peripheral leakage, poor fit, pivotal displacement that occurs with jaw motion and internal cross talk of components housed in prior art hollow type hearing aids.
Patent AU-563905-B2 (AU)
Title: Spreading volume of traffic over different control channels
Inventor: GRAUEL CHRISTOPHER
IPC: H04B7/26
Filed: 1983-12-15
Granted: 1987-07-23
Abstract: A cellular radio system in which the mobile radio stations in the zone of any base radio station assign themselves to the control channels allocated to that base station so as to evenly spread the volume of traffic over such control channels. The base station transmits on each control channel a channel group code signifying the range of group code numbers allocated to that particular control channel. Each mobile station stores its identifying group code number, scans the group code numbers of all control channels, and assigns itself to the control channel having a channel group code which includes its group code number. The spread of traffic over the various control channels can be changed by the base radio station simply by changing the channel group codes of the various control channels, without addressing specific commands to the mobile radio station.
Patent AU-562142-B2 (AU)
Title: Line marking apparatus
Inventor: WILSON J B S MILLIGAN R J LOUG
IPC: E01C23/16
Filed: 1983-11-30
Granted: 1987-05-28
Abstract: PCT No. PCT/AU83/00175 Sec. 371 Date Nov. 30, 1984 Sec. 102(e) Date Nov. 30, 1984 PCT Filed Nov. 30, 1983 PCT Pub. No. WO84/02150 PCT Pub. Date Jun. 7, 1984.Pavement line marking apparatus adapted to detect old line markings on a pavement surface and to repaint such markings or alternatively to paint new line markings to a desired pattern, the apparatus comprising a support beam (11) with a marking detection element (80) arranged at one end such that any old line markings are detectable thereby, upon movement of the detection element 80 over the desired pavement surface, paint applicator means (75,76) arranged mounted from the support boom rearwardly from the marking detection element (80) for movement transversely of the direction of movement of the support boom (11) along the desired pavement surface, and control means actuable in response to a signal from the marking detection element to move said paint applicator means to a position over the old line markings and to operate the paint applicator means to deposit paint along the old line markings on the pavement surface.
Patent AU-670248-B2 (AU)
Title: A waste combustor apparatus
Inventor: JONG JOHANNES DE
IPC: F23G5/027
Filed: 1992-10-09
Granted: 1996-07-11
Abstract: Apparatus for utilising the energy of waste matte comprises respective gasification and combustion chambers (2, 3) connected by an intermediate chamber (4), an entry (5) for ambient combustion air into at least the intermediate chamber (4), and means (6) to cool an inner and external wall of the apparatus and heat the ambient combustion air for passage to the entry (5). <IMAGE>
Patent AU-657038-B2 (AU)
Title: Surface hardened biocompatible metallic medical implants
Inventor: DAVIDSON JAMES A
IPC: A61F2/24
Filed: 1993-02-04
Granted: 1995-02-23
Abstract: This invention provides surface hardened, abrasion resistant high strength, biocompatible metal medical implants, in particular, titanium alloy implants which do not include any elements which have been shown or suggested as having short term or long term potential adverse effect from a standpoint of biocompatibility. Further, the invention provides methods of strengthening and hardening the surfaces of other titanium, zirconium, and cobalt-based alloy implants with small concentrations of a metal solute such as zirconium, yttrium, tantalum, aluminum, silicon, chromium, or thorium via internal oxidation or nitridation. Alternatively, nitrogen, oxygen, or carbon can be diffused directly into the surface of the implants by interstitial hardening to further increase the surface abrasion resistance of these internally oxidized or internally nitridized implant metal or metal alloys.
Patent AU-585837-B2 (AU)
Title: Base coat applicator
Inventor: HAHN ROGER
IPC: B05C13/02
Filed: 1984-08-22
Granted: 1989-06-29
Abstract: @ A base coat applicator utilizing an in-feed chute which provides supply of cans which are mounted on mandrels for application of base coat material by applicator wheels. The mandrels are rotated so that surface speed of the cans matches the applicator wheel speed to prevent smearing. Independent control of the inventory production speed of the base coat applicator machine and the applicator wheels allows any desired num<sub>-</sub> ber of base coat layers to be applied to the cans. Two applicator wheels are used to reduce surface speeds to prevent misting and slinging of base coat material from the applicator wheels and can surfaces. The applicator assembly is automatically withdrawn when the supply of cans is not present and can be manually withdrawn by the operator to prevent application of base coat material to cans or empty mandrels. Disk transfer unit is utilized to transfer the coated cans to a deco pin chain.
Patent AU-691340-B2 (AU)
Title: Anthracycline derivatives
Inventor: SUARATO ANTONINO
IPC: A61P25/00
Filed: 1995-09-05
Granted: 1998-05-14
Abstract: PCT No. PCT/EP95/03480 Sec. 371 Date May 6, 1996 Sec. 102(e) Date May 6, 1996 PCT Filed Sep. 5, 1995 PCT Pub. No. WO96/07665 PCT Pub. Date Mar. 14, 1996The present invention provides the new use in the manufacture of a medicament for use in the treatment of amyloidosis of an anthracycline of formula A: wherein R1, R2, R3 and X are appropriate substituents. Novel compounds of the formula A, processes for their production and pharmaceutical compositions containing them are also described.
Patent AU-578917-B2 (AU)
Title: Unitary armed suture mounting board
Inventor: ROSHDY CONSTANCE ELIZABETH
IPC: A61B17/06
Filed: 1984-11-27
Granted: 1988-11-10
Abstract: The invention provides an element for holding a needled suture comprising a suture strand having at least one end attached to a needle and having a first portion of said suture strand remote from the end attached to said needle and a second portion of said suture strand intermediate between said first portion and the end attached to said needle, said element comprising a unitary piece of soft, flexible polymeric foam and said element further comprising (a), a first retaining means for retaining said needle; (b) a second retaining means remote from said first retaining means for retaining said first portion of said suture strand; and (c) securing means remote from said first and second retaining means for frictionally engaging said second portion of said suture strand when said strand is extended relatively tautly from said first retaining means to said securing means to said second retaining means. The invention also provides a suture package which utilizes the above-described element.
Patent AU-573294-B2 (AU)
Title: 11-beta-arylestradienes
Inventor: ROHDE RALPH
IPC: C07J43/00
Filed: 1984-12-20
Granted: 1988-06-02
Abstract: 11 beta -Arylestradienes of general Formula I are disclosed <IMAGE>  (I)  wherein R2 is a hydrogen atom, a methyl group, or an ethyl group, R3 is a hydrogen atom or an acyl group, R1 and A-B have various meanings, which possess antigestagen and antimineralocorticoid activity.
Patent AU-577736-B2 (AU)
Title: Randomly interstratified clays
Inventor: NADEAU PAUL HENRY
IPC: C01B33/26
Filed: 1985-02-18
Granted: 1988-09-29
Abstract: Randomly interstratified clay is synthesised by:(i) saturating (replacing all the exchangeable cations of) a first clay with alkali metal ions (preferably Na<sup>-</sup> or Li<sup>+</sup>), removing any excess alkali metal ions, and forming the saturated clay into a suspension containing no suspended particles exceeding 10<sup>-7</sup>m equivalent spherical diameter,(ii) saturating a second clay with alkali metal ions (preferably Na<sup>+</sup> or Li-), removing any excess alkali metal ions, and forming the saturated clay into a suspension containing no suspended particles exceeding 10<sup>-7</sup>m equivalent spherical diameter,(iii) mixing the suspensions from (i) and (ii) to form a mixed suspension, and(iv) sedimenting and optionally drying the mixed suspension, the sediment being the synthetic randomly interstratified clay.A wider range of synthetic clay compositions is thereby made available for use as catalysts, sorbents etc.
Patent AU-764973-B2 (AU)
Title: Apparatus for soccer training
Inventor: KILLION DARRYL
IPC: A63B69/00
Filed: 1999-05-06
Granted: 2003-09-04
Abstract: A sports ball is held in a novel manner within a cradle having multiple arms encircling the ball and attached by Velcro TM  to a set of strips attached to a flexible tether line fastened to a person's waist. The ball is able to be kicked or punched and return to the striker in each cycle.