baber/WOPTO huggingface dataset:
Patent IE-35418-L (IE)
Title: Substituted azetidinones
IPC: C07D205/09
Filed: 1971-07-01
Abstract: 1315995 Azetidinone derivatives YEDA RESEARCH & DEVELOPMENT CO Ltd 22 June 1971 [31 July 1970] 37057/70 Heading C2C Azetidin-2-ones having a thioether substituent in the 4-position and a halogen, azido or dicarboxylic acid imido group in the 3-position, and especially novel compounds of formula where X is halogen, azido or dicarboxylic acid imido, R is optionally substituted alkyl or aralkyl, R<SP>1</SP> is optionally substituted alkoxy or aralkoxy, R<SP>2</SP> and R<SP>3</SP> are H or optionally substituted alkyl, aralkoxy or alkylthioalkyl, and Y and Z are each H or together represent a bond joining the carbons to which they are attached, are prepared by reacting a thioimidate derivative of an α-amino acid with XCHCOHal under anhydrous conditions in the presence of a tertiary base. X=Cl may subsequently be converted to X=azido by means of NaN 3 . Compounds of formula where R<SP>4</SP> is -CH(CH 3 ) 2 , -CH 2 OCH 2 C 6 H 5 , -CH 2 CH 2 SCH 3 and -C(CH 3 ) 2 SCH 3 are prepared by reacting appropriate amino acid esters with HCSOC 2 H 5 . is obtained from HC(NH)OC 2 H 5 and the corresponding amino acid ester. Starting materials of formula where: R<SP>5</SP>=CH 3 , R<SP>4</SP>=-CH(CH 3 ) 2 ; R<SP>5</SP>= C 6 H 5 CH 2 -, R<SP>4</SP> =-CH(CH 3 ) 2 ; R<SP>5</SP> = CH 3 , R<SP>4</SP>=-CH 2 OCH 2 C 6 H 5 ; R<SP>5</SP> = CH 3 , R<SP>4</SP>= -CH 2 CH 2 SCH 3 ; R<SP>5</SP>=4-NO 2 -C 6 H 4 CH 2 -, R<SP>4</SP>=-CH 2 CH 2 SCH 3 ; and R<SP>5</SP>=CH 3 , R<SP>4</SP> = -C(CH 3 ) 2 SCH 3 are prepared by reacting R<SP>5</SP>Hal with HC(S)NHCHR<SP>4</SP>COOCH 3 ; where R<SP>5</SP>= CH 3 OOCCH 2 CH 2 - and R<SP>4</SP>=-CH(CH 3 ) 2 and -CH 2 OCH 2 C 6 H 5 by reacting with the compounds in which R<SP>5</SP> = CH 3 or with C 2 H 5 OCH = NCH(COOCH 3 )CH(CH 3 ) 2 . CH 3 SCH = NC(COOCH 3 ) = C(CH 3 ) 2 is prepared from and CH 3 I in the presence of NaH. Phthaloylglycylvaline methyl ester is obtained as a by-product of the reaction between phthaloylglycylchloride and when R<SP>5</SP> is CH 3 - or C 6 H 5 CH 2 -.
[GB1315995A]
Patent IE-850915-L (IE)
Title: Enhancing bitterness of beer
IPC: C12C3/10
Filed: 1985-04-11
Abstract: A method of enhancing the bitterness of beer by oxidation of beta -acids obtained from a carbon dioxide extract of hops and introducing the resulting hulupone, preferably at least partially purified, into the beer. The extract contains also alpha -acids which are isomerized, separated from the beta -acids, and introduced into the beer. The result is a high yield of bitterness-producing material for use in the brewing process.
[US4717580A]
Patent IE-840982-L (IE)
Title: Piroxicam salt deposited on a pharmaceutical carrier
IPC: C07D417/12
Filed: 1984-04-19
Abstract: A process has been developed for preparing the sodium, the monoethanolamine and the diethanolamine salts of piroxicam, in which the salt is deposited on a pharmaceutically-acceptable carrier. The compositions so obtained are useful for preparing pharmaceutical dosage forms of piroxicam, from which piroxicam is rapidly absorbed from the gastrointestinal tract after oral administration to mammals. These latter dosage forms are particularly suitable when it is desired to use piroxicam as an analgesic agent, where rapid onset of action is necessary.
Patent FI-820005-L (FI)
Inventor: LINDAHL JONAS ARNE INGVAR
IPC: D21C9/02
Filed: 1982-01-04
Abstract: To provide a cleaner pulp and to obtain a higher chemical recovery during washing of chemically cooked and optionally defibrated cellulose pulp, the partially washed pulp is subjected to a mild mechanical treatment e.g. in a device (10) adapted for high-consistency treatment and provided with screwsrotating relative to each other, said treatment taking place between at least one pair of conventional washing stages (4,14).
Patent FI-853758-L (FI)
Inventor: BOURQUE RENE
IPC: A63C1/02
Filed: 1985-09-30
Abstract: 57 A skate comprises a boot and an ice skate blade (24) with fixed molded plastics support (22). The molded plastics support (22) includes a boot receiving means (26) having the outline of the sole of the boot and having a ridge (28) adapted to be fixed to the base of the boot. The support (22) may be fixed to the boot by way of a suitable adhesive, and the boot receiving portion (26) of the support replaces the sole of the boot.
Patent IE-34447-L (IE)
Title: Hauling underwater ropes
IPC: A01K73/12
Filed: 1970-08-07
Abstract: 1290769 Fishing nets RAPP FABRIKKER A/S 10 Aug 1970 [13 Aug 1969] 38497/70 Heading A1A [Also in Division B8] One end 17 of a purse seine fishing line is frictionally hauled in against the reaction of the other end 16 of such line by a winch unit 6 suspended in a submerged position in the water by a cable 3 extending from a boat 1, the seine line portion 20 passing out of the winch unit 6 being hauled up by a winch unit 22 on the boat. The unit 6 comprises a pair of drums 8 around which the line is looped several times and which are driven by an hydraulic motor 7 supplied from a pump 10 on the boat, through lines 14, the drums 8 including pawl and ratchet mechanisms 26 normally preventing pay out of the seine line. The hauling capacity of the winch unit 6 is variable in relation to the tension applied to the line portion 20 departing therefrom. The unit 6 and its associated fishing gear is raised to the surface by the cable 3 actuated by a winch 2, but alternatively the winch 22 and seine line portion 20 may be used for such raising operation. In the embodiment of Fig. 2 (not shown) the submerged winch unit is used for hauling a scraper along the sea bed, the hauling force being reacted against an anchor line attached to the winch unit. The submerged winch unit in both the above embodiments may utilise a single drum as shown in Fig. 3 (not shown).
[GB1290769A]
Patent IE-851533-L (IE)
Title: Longitudinal cutting of a tubular fibrous product
IPC: B26D3/00
Filed: 1985-06-20
Abstract: Method for longitudinal cutting of a wall of a fibrous tubular product in a step shaped profile. The apparatus comprises two parallel main blades which form radial cuts into the wall, slightly displaced from each other. One cut is made radially inward from the outer surface; and the other cut is made radially outward from the inner surface. Each cut extends toward the center of the shell wall to a depth approximately one half the thickness of the shell wall. A third cut is made within the shell wall perpendicular to and joining the other two cuts. These three cuts form a smooth step shaped cut through the wall and facilitate installation of the shell around conduit while minimizing heat loss and mechanical stresses within the wall.
[US4781089A]
Patent IE-811572-L (IE)
Title: Production of ice confection products.
IPC: A23P1/12
Filed: 1981-07-13
Abstract: A process for preparing an ice confection or other foodstuff with projecting and relatively recessed relief features of its outer surface, characterised by extruding the ice confection or other extrudable edible material from a rotating extrusion nozzle having a cross-section with an assymmetrical configuration with respect to the rotation axis, with the extruded material passing from the nozzle immediately into an unconfined space and on to an elongate travelling conveyor which does not share the rotational motion of the extrusion nozzle, thereby to lay down on the conveyor an extended spirally-formed extrudate with projecting and relatively recessed relief features derived from its extrusion through the nozzle of assymmetrical configuration.
Patent IE-34832-L (IE)
Title: Thiepin derivatives
IPC: C07D209/00
Filed: 1970-12-22
Abstract: Thiepine derivs of formula (I) (where one of X and Y is S and the other is a single direct bond and R1 is H, allyl, or 1-4C alkyl) and their acid addition salts which are useful for teating tension and agitation states of psychic or muscular origin, are claimed. Processes for preparing these cpds. are also claimed
[FR2081394A1]
Patent IE-45657-L (IE)
Title: Fungicidal compositions
IPC: A01N37/34
Filed: 1977-08-16
Abstract: For the treatment of fungal infections of cultivated plants, a composition based on 2,4,5,6-tetrachloro-1,3-dicyanobenzene and a pyrimidinemethanol compound of formula (I) <IMAGE> in which X represents chlorine or fluorine, is used. The weight ratio of pyrimidinemethanol to 2,4,5,6-tetrachloro-1,3-dicyanobenzene is preferably between 1:400 and 1.6:1. Application for destroying Puccinia recondita in cereals and Pseudoperonospora cubensis of cucurbitaceous plants. The composition exhibits a synergistic effect of the constituents.
[GB1581527A]
Patent IE-881937-L (IE)
Title: Preparation of antibiotic furmifungin
IPC: A61K31/20
Filed: 1988-06-24
Abstract: Fumifungin, a compound of the formula  <IMAGE>  can be isolated from the culture broth of fungus culture No. Y-83,0405 (DSM 4152), and has bactericidal and fungicidal properties.
Patent IE-38636-L (IE)
Title: Cyclopenta[e]-1,3-oxazine-2,4-diones.
IPC: C07C55/02
Filed: 1973-12-12
Abstract: 2, 3, 4, 5, 6, 7-HEXAHYDROCYCLOPENTA-[E]-1,3-OXAZINE-2,4-DIONE COMPOUNDS ARE PRODUCED BY REACTING AN ADIPIC ACID HALIDE OF THE FORMULA ORRRO PARALLEL ¦¦¦ PARALLEL X-C-CH2-C-C-C-C-X ¦¦¦ RRR wherein R is hydrogen or alkyl of up to 3 carbons; and X is halogen, preferably chlorine or bromine, WITH AN ISOCYANATE OF THE FORMULA O=C=N-R1 in which R1 is hydrocarbyl or substituted hydrocarbyl, preferably of less than 11 carbons. The process is conducted in the presence of a tertiary base, and optionally in the presence of a solvent, at a temperature of from 80 DEG to 180 DEG C., preferably at from 90 DEG to 130 DEG C.
[US3940390A]
Patent IE-46123-L (IE)
Title: Cyclopropane carboxylic acid esters.
IPC: A01N53/00
Filed: 1977-12-21
Abstract: 2,2-Dimethyl-3-vinyl-cyclopropane carboxylic acid esters of halogenated benzyl alcohols of the formula <IMAGE> in which each R independently represents F, Cl, Br or CH3 and m and n each represent 0, 1, 2, 3, 4 or 5 subject to the sum of m+n being not more than 5, with the provisos that (i) when each R represents F or Br then m and n cannot both be 0, (ii) when each R represents Cl, then m represents 0, 1, 2, 3 or 4 and n represents 1, 2, 3, 4 or 5, and (iii) when each R represents CH3, then m represents 0 and n represents 5, which possess arthropodicidal properties.
[US4183950A]
Patent IE-41982-L (IE)
Title: Floating fender
IPC: B63B59/02
Filed: 1975-12-22
Abstract: A floating rubber fender to be used for ships, platforms, locks, or the like. In order to provide a fender which will not sink when its support cables break, it has been proposed to manufacture the fenders partly of massive rubber, with the remainder thereof comprising sponge or foam rubber, such that the overall density is less than 1.0 and is therefore of floating construction. However, such fenders are not suitable for the heavy conditions of use to which they are subjected since the use of foam rubber or sponge results in decreased rigidity and tear resistance. To overcome this problem, the present invention provides a floating rubber fender consisting of a rubber body manufactured from massive rubber, the rubber body having been manufactured from a substantially synthetic rubber having a density below about 0.91. Additionally, a carbon black is utilized as a reinforcing filler, the carbon black promoting electrical conductivity and having a small particle size and a high structure. The carbon black is added in such an amount that the density of the rubber after vulcanization amounts to at most 0.97.
[CA1074990A]
Patent IE-883387-L (IE)
Title: Process for preparing 1,5-benzothiazepines
IPC: C07D281/10
Filed: 1988-11-11
Abstract: PURPOSE:To obtain the title compound which is used as a medicine, because of its hypotensive and cerebral and coronary vasodilative actions, readily in high yield, by intramolecular cyclization of a propionic acid derivative as a starting substance. CONSTITUTION:A propionic acid derivative of formula I (R<1> is lower alkyl, lower alkoxy; R<2> is H, lower alkanoyl; R<3>, R<4> are lower alkyl; one of R<5> and R<6> is lower alkyl, halogen, and the other is H) or its reactive derivative is subjected to intramolecular cyclization reaction in the presence or in the absence of a condensation agent or a deacidification agent in a solvent such as xylene with heat, preferably at 100-180 deg.C to give the compound of formula II. When a free form of the compound of formula I is used, the reaction is preferably carried out in a solvent in the presence of a condensation reagent, while an acid halide is used as a reactive derivative of the compound of formula I, the reaction is preferably effected in the presence of a deacidification agent.
[JP1128974A]
Patent NO-823064-L (NO)
Inventor: SHAW HERBERT JOHN
IPC: G01N37/00
Filed: 1982-09-09
Abstract: A fiber optic directional coupler (10) comprises a pair of bases (16), with respective longitudinal, arcuate grooves (13) formed therein on confronting faces (14) thereof, for mounting a pair of optical fibers (12) in close proximity. A portion of the cladding is removed from each of the fibers (12) to form planar facing surfaces (18) which permits the spacing between the fiber cores to be within a predetermined critical zone (34) so that guided modes of the fibers (12) interact, through their evanescent fields, to cause light to be transferred by evanescent field coupling between the fibers (12). The coupler (10) is "tuned" to a desired coupling efficiency by offsetting the planar facing surfaces (18) to increase the spacing between the fiber cores. A method of manufacture of the coupler includes procedures which permit the coupler halves to be made symmetrical. The method also permits couplers (10) having given coupling characteristics to be reproduced.
Patent NO-824161-L (NO)
Title: Energianvisende anordning for motorkjoeretoeyer.
Inventor: PASSANA JUAN FRANCISCO VALL-LL
IPC: B60R16/023
Filed: 1982-12-10
Abstract: Energianvisende anordning som under hensyn-tagen til trafikksituasjoner, kjøremåte og reiseprogram kan angi energiforbruk i et motorkjøretøy om-fatter følere som måler brennstoffstrmmen tilmotoren og motorens omdreiningstall, og ved hjelp av en mikroprosessor kan angi på en indikator for--ventede forbruk ved forskjellige trafikksituasjoner og kjøremåter, slik at freren ved innstilling av den eksisterende trafikksituasjon kan få informasjoner til den mest økonomiske videre kjøring.
Patent NO-830911-L (NO)
Title: Fremgangsmaate for klassifisering av mynter i henhold til deres mekaniske elastisitet
Inventor: MEYER PETER
IPC: G07D5/06
Filed: 1983-03-15
Abstract: remgangsmåte for å sortere gangbar mynt fra ikke-gangbar mynt ved å. bestemme den mekaniske elastisiteten i mynten. Dette blir utført ved å la mynten (1) falle i en vel-definert avstand (h) på en bjelke (2) som blir brakt til svingning. Via en gaffel (4) blir svingningene overført til et piezoelektrisk element (5), hvis elektriske signal blir forsterket, idet det forsterkede signals nivå blir bestemt (10).En blymynt gir en mindre signalamplitude enn en nyslvmynt av samme. diameter gjør.
Patent NO-841128-L (NO)
Inventor: KALVAAG JOHN BAARD
IPC: A61H1/02
Filed: 1984-03-22
Abstract: An apparatus for the treatment of patients suffering trom lumbar back ailments or the like comprises at least one float body (1) suspended from an overhead support (3.4,5,6,7), intended for suspending the patient who is partially submersed in water and subjected to loading from weights (13), preferably at the hip region. The overhead support consists of a suspension means (2) from which, by emans of straps (9), a vest (10) is suspended, adapted to fit closely about the chest region of the patient and thereby supporting the patient. The straps (9) are attached to the overhead support (2) via a yoke or crossbar (8) having a central, vertical journal that is pivotally mounted at the top (7) of the overhead support.The float body may consist of two elongated, substantially boat-shaped floats (1), and the overhead support may consist of four downwardly-depending legs (3,4,5,6) attached at the lower ends thereof to the floats (1) and rigidly attached at the upper ends thereof to a top piece (7) which is disposed centrally between the floats (1) and from which the crossbar is supported.
Patent NO-843464-L (NO)
Inventor: HOUGHTEN RICHATD A
IPC: C07K7/08
Filed: 1984-08-31
Abstract: A synthetic polypeptide having at least about 10% of the immunological activity of biologic heat-stable enterotoxin of E. coli. The synthetic polypeptide includes at least 14 amino acids in the sequence, from amino-terminus to carboxy-terminus, represented by the formula: CysCys-GluLeuCysCysTyr(Asn)ProAlaCysAla(Thr)GlyCysAsn(Tyr) wherein the amino acid in parentheses may replace the immediately preceding amino acid residue, and at least one intramolecular disulfide bond formed between the Cys residues. The Cys residues that are not part of the intramolecular disulfide bond can be replaced by other amino acid residues or be bonded to substituent moieties. The polypeptides can be a monomeric or multimeric material containing an intramolecular, intrapolypeptide and/or an intramolecular, interpolypeptide cystine disulfide bond.
Patent NO-852761-L (NO)
Inventor: STEEN HARALD B
IPC: G01N21/05
Filed: 1985-07-10
Abstract: PCT No. PCT/NO86/00050 Sec. 371 Date Mar. 5, 1987 Sec. 102(e) Date Mar. 5, 1987 PCT Filed Jul. 10, 1986 PCT Pub. No. WO87/00282 PCT Pub. Date Jan. 15, 1987.The present invention relates to a device which facilitates that biological cells and other microscopical particles, carried by a microscopial laminar fluid flow, are brought one by one across the open surface of a plane glass with a velocity which may be varied from above 30 m/sec. to below 1 cm/sec., so that the fluorescence and light scattering of the cells/particles may be measured through optics situated on each side of the plane glass. The device comprises a nozzle (1) with hydrodynamic focusing having its axis at an oblique angle to said glass surface. Furthermore, at the same time the electrical volume of the cells/particles may be determined by means of an electrode, made of inert metal, situated in the contact plane between the nozzle (1) and said glass (2) and an electrode situated in the fluid supply (8) of the nozzle (1). By retaining a constant electrolytical current between the electrode (6) and the electrode (7) the electrical volume of the cells/particles may be measured by the voltage pulses produced between the said electrodes when the cells/particles pass through the orifice.
Patent NO-854417-L (NO)
Inventor: WIEDERKEHR HANS
IPC: B24B19/02
Filed: 1985-11-06
Abstract: The grinding head has a bar-like member, on whose free end is mounted a grinding tool with a grinding wheel spindle arranged at right angles to the longitudinal axis of the bar-like member. The grinding tool is driven by means of a work gear and a driving shaft, which is driven by means of a coupling with a motor. The motor is mounted in a casing, which is shaped onto the mounting flange. The grinding head can be vertically or horizontally arranged in the grinding or milling machine. Due to the fact that the grinding tool has a larger diameter than that of the bar-like member, facing groove sides in bores can be worked in one setting, so that the complete working operation is made faster due to the few idle strokes and simultaneously precision is increased.
Patent NO-861613-L (NO)
Inventor: GERK ALVIN PHILLIP
IPC: B24D3/00
Filed: 1986-04-24
Abstract: A sol-gel process of producing durable alpha alumina-based ceramic abrasive grain from alpha alumina monohydrate is improved by the addition of a nucleating agent. Improved abrasive products containing the durable ceramic abrasive grains are also provided.
Patent NO-870372-L (NO)
Inventor: LANE KENNETH ROBERT
IPC: C03B37/025
Filed: 1987-01-29
Abstract: A heating oven (10) for processing glass material from which optical waveguide fibers are prepared is provided which comprises:(a) an elongated chamber (22) for receiving the glass material to be processed; and(b) means for heating the chamber, said means comprising an elongated susceptor (26), the longitudinal axis of the susceptor being parallel to the longitudinal axis of the chamber, an induction heating coil (38), means (58) for moving the induction heating coil along a path parallel to the longitudinal axes of the susceptor and the chamber, and means for energizing the induction heating coil (38).
Patent NO-883084-L (NO)
Inventor: GUTHRIE ROBERT WILLIAM
IPC: A61K31/47
Filed: 1988-07-08
Abstract: Compounds of the formula    <IMAGE>  I  Y is O ir S, *A is paraphenylene or *--(CH2)n--(X)m-(CH2)r--, X is O, S or -CH=CH-, n or r, independently, are integers from 0 to 3, s is an integer from 0 to 1, m is an integer from 0 to 1, provided that when m is 1, n+s must be at least 2, R1 and R2, independently, are hydrogen, lower alkyl, cycloalkyl, lower alkenyl, Het, aryl, R3, R4 and R8, independently, are hydrogen, lower alkyl, aryl, R5 and R6, independently, are hydrogen or lower alkyl, R7 is hydrogen, lower alkyl, cycloalkyl, Het-lower alkyl or aryl, Het is a monocyclic 5- or 6-membered hetero aromatic or a bicyclic heteroaromatic radical containing one or two hetero atoms selected from nitrogen, oxygen and sulfur, which radical may be substituted by lower alkyl, halogen or aryl, and the asterisk denotes the point of attachment, and when R6 and R7 are different, their enantiomers and racemic mixtures thereof, when R1 and R2 are different, their geometric isomers, and pharmaceutically acceptable acid addition salts thereof, are described. The compounds of formula I exhibit activity as platelet activating factor (PAF) antagonists and are, therefore, useful in disease states characerized by excess platelet activating factor or for the prevention and treatment of cardiovascular disease, pulmonary diseases, immunological disorders, inflammatory diseases, dermatological disorders, shock or transplant rejection.
Patent NO-894698-L (NO)
Inventor: SHUTSKE GREGORY MICHAEL
IPC: C07D498/06
Filed: 1989-11-24
Abstract: There are disclosed compounds having the formula <CHEM>  where  R1 is hydrogen, loweralkyl or arylloweralkyl; Z is hydrogen, loweralkyl, loweralkoxy, hydroxy, nitro or trifluoromethyl;  Y is O or NR2, R2 being hydrogen, loweralkyl or arylloweralkyl; and X is CH3, CHR3, C=O, C=S or CHN(CH3)2, R3 being hydrogen, loweralkyl or aryl; or a stereo isomer thereof or a pharmaceutically acceptable acid addition salt thereof, and a process for their preparation. The compounds are useful for the treatment of various memory dysfunctions characterized by decreased cholinergic function, such as Alzheimer's disease, and can therefore be applied as medicaments.
Patent NO-910091-L (NO)
Title: Fremgangsmaate for fremstilling av et fasadeelement av naturstein.
Inventor: HEGGHEIM ODDGEIR
IPC: E04F/
Filed: 1991-01-09
Abstract: Fremgangsmåte for fremstilling av en plate av naturstein, hvor natui— steinplaten påfres et limsjikt av typen "epoxy" eller tilsvarende. En plate av fiberbetong påstøpes deretter på natursteinplata. Fibrenefiberbetongen kan være av typen polyester.
Patent NO-923640-L (NO)
Inventor: WOMBWELL PAUL TERRENCE
IPC: C08K3/00
Filed: 1992-09-18
Abstract: The present invention provides an epoxy resin composition comprising an epoxy resin, at least one filler, a thixotropic agent in an amount less than that necessary to impart thixotropic properties and a polymer which dissolves in and thickens a mixture of the resin and a curing agent therefor when the mixture is heated prior to curing. The compositions are used for making moulded articles.
Patent NO-924502-L (NO)
Inventor: BJOERK ANDERS
IPC: C07D241/04
Filed: 1992-11-23
Abstract: The present invention relates to the relief or prevention of withdrawal syndrome resulting from addiction to non-opiate type drugs of abuse and/or the suppression of dependence on non-opiate type drugs of abuse by administering to a person in need thereof, an effective amount of certain diphenylbutyl-piperazine-carboxamides including 4-[4,4-bis(4-fluorophenyl)butyl]-N-ethyl-1-piperazine-carboxamide which is known as amperozide.