baber/WOPTO huggingface dataset:
Patent IL-99345-A0 (IL)
Title: 6-or 7-(2-imino-2-imidazolidine)-1,4-benzoxazines as alpha adrenergic agents
IPC: A61P27/02
Filed: 1991-08-29
Abstract: Compounds having  alpha  adrenergic activity and useful for the treatment of glaucoma, renal and gastrointestinal disorders and vasoconstictors have the formula  <IMAGE>  where R1 is independently H, or lower alkyl or 1 to 6 carbons; R2 is independently H, or lower alkyl of 1 to 6 carbons or the two R2 symbols jointly represent a carbonyl oxygen; R3 is H, lower alkyl of one to 6 carbons, O, OH and OR7 where R7 is lower alkyl of 1 to 6 carbons, or R3 is COH or COR8 where R8 is lower alkyl of 1 to 6 carbons; R4 and R5 independently is H, Br, Cl, or lower alkyl of 1 to 6 carbons, lower alkenyl or lower alkynyl with the proviso that when the R2 groups symbolize a carbonyl oxygen then R4 and R5 both cannot be hydrogen; R6 is hydrogen, Br, Cl, or lower alkyl of 1 to 6 carbons, lower alkenyl or lower alkynyl, and the R5 and the (2-imidazoline-2-yl)amino substituents are connected mutually exclusively to the 6 and 7 positions of the 1,4-benzoxazine nucleus.
Patent IL-99434-A0 (IL)
Title: 3-(1h-indazol-3-yl)-4-pyridinamines,a process and intermediates for their preparation and pharmaceutical compositions containing them
IPC: C07D213/73
Filed: 1991-09-06
Abstract: This Invention relates to 4-(1H-indazol-3-yl)-4-pyridinamines of the formula I <CHEM> where R1 is hydrogen, loweralkyl, arylalkyl or acyl; R2 is hydrogen, loweralkyl or arylalkyl; R3 is hydrogen, loweralkyl or aryl and X is hydrogen, halogen, nitro or amino, or the pharmaceutically acceptable addition salts thereof, and where applicable, the geometric and optical isomers and racemic mixtures thereof. The compounds of this invention are useful as analgesics and as topical antiinflammatory agents for the treatment of various dermatoses. The invention relates further to intermediates of the formula II <CHEM> where R1, R2 and R3 have the above meaning, which have also analgesic activity, as well as to processes for the preparation of compounds of both formulae.
Patent IL-99633-A0 (IL)
Title: Elevating and lowering apparatus
IPC: A62B1/06
Filed: 1991-10-02
Abstract: The rope lifting and lowering apparatus has a base plate (1) to which a rope lowering pulley (2) mounted in a freely rotating manner and having a pawl stop is fastened. A toothed ring (7) is fastened to the side of the rope lowering pulley facing the base plate. The teeth (7a) of the toothed ring (7) interact with a pawl (9) in such a way that in the free-wheeling direction the pawl is lifted and in the locking direction the pawl clamps the toothed ring or the rope lowering pulley in position. The pawl is let into the base plate. <IMAGE>
Patent AU-PM589894-A0 (AU)
Title: Metal strip casting
IPC: B22D27/08
Filed: 1994-05-27
Abstract: A method and an apparatus of continuously casting metal strip (20) is disclosed. A casting pool (30) of molten metal is formed in contact with a moving casting surface such that metal solidifies from the pool (30) onto the moving casting surface. In addition, sound waves are applied to the casting pool of molten metal to induce relative vibratory movement between the molten metal of the casting pool (30) and the casting surface.
Patent IL-111400-A0 (IL)
Title: Pharmaceutical compositions containing metroprolol and methods for the preparation thereof
IPC: A61K9/20
Filed: 1994-10-25
Abstract: A sustained release oral solid dosage form of metoprolol pharmaceutical formulation includes a sustained release excipient including a gelling agent, an inert pharmaceutical diluent, a cationic cross-linking agent, and metoprolol provides release of metoprolol for at least about 24 hours. In certain embodiments, the sustained release formulation further includes a hydrophobic material.
Patent IL-112583-A0 (IL)
Title: Oral delivery of chemically modified proteins
IPC: A61K38/21
Filed: 1995-02-08
Abstract: Provided are compositions and methods for oral delivery of chemically modified proteins, including chemically modified G-CSF and chemically modified consensus interferon. Uptake from the intestine to the bloodstream is demonstrated for pegylated G-CSF and pegylated consensus interferon. <IMAGE>
Patent IL-124593-A0 (IL)
Title: Substituted aryl or heteroarylamides having retinoid-like biological activity
IPC: C07D/
Filed: 1996-11-19
Abstract: Compounds of the formula wherein the symbols have the meaning described in the specification, have retinoid-like biological activity.
Patent IL-131964-A0 (IL)
Title: A process for preparing phosphodiester compounds
IPC: C07F9/09
Filed: 1998-01-27
Abstract: A process for preparing a phosphodiester of the formula: is described that involves (1) reaction of a first alcohol with phosphorous trichloride to form a phosphorodichlorodite, (2) reaction of the phosphorodichlorodite with an amine to form a phosphorodiamidite, (3) reaction with a second alcohol (which may be the same as the first alcohol) to form a phosphoramidite diester, and finally, (4) hydrolysis and oxidation of the phosphoramidite to form the phosphodiester. R and R1 may represent aliphatic, aromatic, heterocyclic, peptidic, peptoid, deoxyribo- or ribonucleotidic or nucleosidic, or organic chelating moieties.
Patent IL-132098-A0 (IL)
Title: Controlled free radical polymerization process
IPC: C08F293/00
Filed: 1998-03-31
Abstract: A polymerization process for the preparation of (meth)acrylate containing homopolymers or block copolymers comprises heating a mixture of a free radical initiator, a stable free radical agent, and a polymerizable monomer compound to form a thermoplastic resin or resins with a narrow polydispersity. The stable free radical agent is a piperazinone or morpholone based nitroxide or any adducts thereof.
Patent IL-134617-A0 (IL)
Title: Application of substances on a package
IPC: B65B61/26
Filed: 1998-08-20
Abstract: The present invention relates to a process for producing a packaging system (4) comprising a first step, the packaging system comprising a hollow body (4), the first step consisting in applying a first substance onto a selected surface area of the packaging system by use of first application means (5), the selected surface area and the hollow body (4) being both in motion relative to the first application means (5) and the selected surface area being solely in contact with the first substance during the first step. The process also comprises a second step which consists in applying a second substance onto the selected surface area by use of second application means after completion of the first step, the selected surface area and the hollow body being both in motion relative to the second application means and the selected surface area being solely in contact with the second substance during the second step, the process taking place at a continuous line speed.
Patent IL-152239-A0 (IL)
Title: Endoventricular device for the treatment and correction of cardiomyopathies
IPC: A61L31/00
Filed: 2001-03-28
Abstract: The invention consists in a device that concerns the optimization of the cardiac geometry in patients with heart failure. The device comprises one or more elastic elements in the radial direction towards the inside of the ventricle, the element being equipped with means for attaching it to the internal wall of the ventricle.
Patent IL-160102-A0 (IL)
Title: Electric motor comprising a cooling system
IPC: H02K1/20
Filed: 2002-05-10
Abstract: An electric motor, e.g., a linear motor, includes a cooling system, which may permit the dissipation of heat from the primary part of the electric motor in a simple but effective manner. The iron core and the coils may be surrounded by a potting compound that stabilizes one of the coils and the electrical leads of the latter so that channels are formed in the gaps of the iron core. A coolant, e.g., air, flows from a first flow chamber through the channels into a second flow chamber. The direct contact with the iron core, potting compound, and optionally with the regions of the coils that are not filled with compound produces effective cooling action, without having to forego advantages of stability provided by an encapsulated primary part.
Patent IL-160915-A0 (IL)
Title: Indolizines inhibiting kinase proteins
IPC: A61K31/4985
Filed: 2002-09-17
Abstract: The present invention concerns compounds of general formula (I): in which the substituents are as described herein.
Patent IL-162706-A0 (IL)
Title: Confocal imaging equipment in particular for endoscope
IPC: G02B21/00
Filed: 2002-12-20
Abstract: Equipment includes an image guide ( 1 ) consisting of flexible optical fibers with: on the proximal end side: a source ( 2 ), angular scanning elements ( 3 ), injection elements ( 4 ) in one of the fibers, elements for splitting ( 5 ) the illuminating beam and the backscattered signal, elements for spatial filtering ( 6 ), elements for detecting ( 7 ) the signal, electronic elements ( 8 ) for controlling, analyzing and digital processing of the detected signal and display; and on the distal end side: an optical head ( 9 ) for focusing the illuminating beam exiting from the illuminated fiber. The scanning elements include a resonant line mirror (M 1 ) and a galvanometric field mirror (M 2 ) with a variable frequency and two afocal optical systems adapted to conjugate the two mirrors (M 1 , M 2 ) firstly in the field mirror (M 2 ) and the injection elements ( 4 ) in the image guide in a second step.
Patent IL-166689-A0 (IL)
Title: A portable beverage preparation device and system
IPC: A23L1/00
Filed: 2005-02-03
Abstract: A portable beverage preparation device and system for making brews, mixes, and potions on demand by selectively introducing and mixing predetermined quantities of at least one stored, edible, beverage preparation confined in at least one sealed chamber into a portable beverage container containing a predetermined volume of a potable base liquid and having a dispenser means for introducing the at least one beverage preparation into the potable base liquid; wherein the drink container and the at least one sealed chamber are in close physical proximity to each other and separated by at least one thin membrane which, when inwardly perforated by the dispenser means, introduces the at least one beverage preparation into the base liquid. The system of the invention further provides a brewing element and a portable heating unit, the heater element of which fits into the beverage container for heating the liquid.
Patent IL-182764-A0 (IL)
Title: Methods for treating obesity and obesity related diseases and disorders
Filed: 2007-04-23
Abstract: Methods for treating obesity or obesity related disorders are disclosed. These methods include the use of anti-obesity agents directed to the forebrain in combination with anti-obesity agents directed to the hindbrain.
Patent IL-206596-A0 (IL)
Title: Composition for treating sterile inflammation
IPC: A61K35/30
Filed: 2010-06-24
Abstract: Biological medical means for treating sterile inflammatory diseases are disclosed. The invention relates to the use of L-arginine-hydrochloride (Arg) or lysine (Lys) and L-leucine (Leu) for the manufacture of a pharmaceutical composition for treating or preventing sterile inflammation. The composition further comprises trace elements chromium (Cr), tin (Sn), selenium (Se), strontium (Sr), vanadium (V), wolfram (W) and folic acid. The pharmaceutical composition can further comprise zinc (Zn) and or manganese (Mn) as well as central nervous system (CNS) lipids. Sterile inflammations are related to disorder such as fibromyalgia, Crohn's disease, psoriasis and rheuma.
Patent RO-129986-A0 (RO)
Title: Gambling game based on undrawn lottery numbers
Inventor: RĂDUŢ CĂTĂLIN FLORIAN
IPC: G07C15/00
Filed: 2014-07-09
Abstract: The invention relates to a gambling game based on numbers and/or lottery elements which are not drawn after the lottery official drawing, carried out by one or more national or private lotteries or carried out instantly, practicable in casinos or in specially arranged rooms, on the internet or as society game. According to the invention, the game consists of a game ticket that the gambler fills in with combinations of 6 numbers out of 49, the winning combinations consisting of any of some undrawn numbers and/or elements (1), undrawn numbers and/or elements (2) belonging to certain rows of elements, undrawn and drawn numbers and/or elements (3) and undrawn elements (4) belonging to certain rows of elements and undrawn or drawn elements.
Patent RO-130293-A0 (RO)
Title: Method for the ecological reconstruction of waste and/or ash heaps
Inventor: COMAN ALEXANDRU
IPC: C05G3/00
Filed: 2014-08-08
Abstract: The invention relates to a method for ecological reconstruction of waste and/or ash heaps resulting after the extraction and processing of coal, and the combustion thereof, respectively. According to the invention, the method consists in the revegetation of heaps by the cultivation of the perennial plant Miscanthus, the year following the plantation, the stems being chopped on the spot and left on the heap for covering, fixing and enriching the soil with organic matter, and starting with the second year, the stems of Miscanthus are harvested and exploited as fuel, either as such or in combination with the processed coal.
Patent AP-2001002352-A0 (AP)
Title: A device comprising a chamber and a piston.
Inventor: VAN DER BLOM NICOLAAS
IPC: F01C5/00
Filed: 1999-04-22
Abstract: The object of the invention is to provide a reliable and inexpensive combination of a chamber and a piston to be used in any device where such a combination is needed so that it complies with specific demands towards the operation force for e.G. pumps, specifically manually operated pumps. By a device comprising a chamber and a piston positioned inside the chamber said chamber and said piston relatively movable to each other in a predetermined direction of movement between a first position and a second position of which the cross-section of the chamber in a plane perpendicular to the direction of movement is larger at the first position than at the second position, the change in the cross section of the chamber is essentially continuous between the first position and the second position and the cross-section of the piston in a plane perpendicular to the direction of movement is arranged to adapt itselft to the cross-section of the chamber. It is further possible that the piston has a fixed geometrical shape, that the wall of the chamber has different sizes of cross-sections in the direction of the movement and is arranged to adapt itself to the piston. Moreover, both the piston and the wall of the chamber can adapt itself to each other.
Patent AP-2003002840-A0 (AP)
Title: Pyridine matrix metalloproteinase inhibitors
Inventor: BARVIAN NICOLE CHANTEL
IPC: C07D213/82
Filed: 2002-02-04
Abstract: Selective MMP-13 inhibitors are pyridine derivatives of the formula (I) or a pharmaceulically acceptable sail thereof, wherein: R1 and R2 independently are hydrogen, halo, hydroxy, C,-C6 alkyl, CrC6 alkoxy. C2-C6 alkenyl, C:-Cb alkynyl, NO;, NR'R1, CM, or CF3; K is indepcndenily O or S; A and B independently are OR4 or NRJKS; R4 and R5 independently are H, C,-C6 alkyl, C3-C6 alkenyl, C2-C6 alkynyl, (CM2)n aryl, (CU2)n cycloalkyl, (CH2),, heteroaryl, or R4 and R5 when taken together with the nitrogen to which they are attached complete a 3- to 8-mernbered ring containing carbon atoms and optionally containing a heteroatom selected from O, S, or NH, and optionally substituted or unsubsiiimed; n is 0 to 6.
Patent MA-37099-A1 (MA)
Title: Procédé de traitement des molécules émergeants et récalcitrants (pestisides, produits périmés chimiques) par le phosphate dopé à l'oxyde de titane (tio2), à l'aide d'un réacteur fonctionnant à l'énergie solaire.
Inventor: CHERKAOUI RACHID
IPC: C02F1/30
Filed: 2014-06-03
Abstract: L’invention concerne un procédé dedégradation des pesticidespar le phosphate dopé avec le titane, comprenant les étapes suivantes : - on enlève les impuretés qui existent au phosphate brut par un tamis: l'analyse granulométrique - on lave le phosphate avec l’eau distillée, suivi d’une filtration dans les conditions normales et on le sèche. - on prétraite le flux liquide par déshuilage suivi d’une décantation de particules discrètes - on clarifie le flux par élimination des matières en suspension en mettant ledit flux en contact avec le phosphate dopé - on poste-traite le flux liquide par une décantation secondaire à l’aval du procédé l’invention concerne aussi un dispositif pour la mise en œuvre dudit procédé.
Patent UY-23648-A1 (UY)
Title: Puerto alternativo propulsor de energia
IPC: F03B13/26
Filed: 1993-09-17
Abstract: La presente invención se refiere a la construcción sobre los Bancos del Río de la Plata, de escolleras con formas de flechas; paralelas entre sí por el lado del cateto mayor y que este y que estén surtidas por canales de intersección con el canal mayor cercano; este canal permite a los barcos del exterior el derivar su rumbo y recalar entre las banquinas de amarre. Dichas escolleras bordean una pileta de contención de las aguas de abatimiento; las que drenan a popa por tunos munidos de cisternas (y unidas las piletas por vaso comunicante) y las dársenas artificiales pueden contar con elevadores de granos y rieles con montaje de puente; tipo empleadas en Coquimbo, Chile y que permiten a zorras "devauvilles" portar el grano hasta volcarlo sobre las sentinas de los graneleros en carga. La electricidad producida se ysa en principio para abastecer necesidades de alije y carga; etc.
Patent UY-24556-A1 (UY)
Title: Comprimidos con alto contenido de famciclovir
Inventor: JOHN GREENWAY
IPC: A61K47/26
Filed: 1997-05-16
Abstract: Un comprimido farmacéutico en el que el famciclovir es el ingrediente activo y en el porcentaje en peso de famciclovir en el comprimido es del 85% o mayor.
Patent UY-27785-A1 (UY)
Title: Nueva composición farmacéutica
Inventor: BAILLY JACQUES
Filed: 2003-04-28
Abstract: La presente invención, se refiere a composiciones y procedimientos para el tratamiento de la obesidad. De una forma más particular, la invención, se refiere a una composición que comprende un inhibidor de lipasa, y konjac o glucomanan.
Patent AT-522234-A1 (AT)
Title: Verfahren und Vorrichtung zum Geraderichten von Draht oder Bandmaterial
IPC: B21F1/02
Filed: 2019-02-28
Abstract: Verfahren zum Geraderichten von Draht oder Bandmaterial mittels einer Dressurvorrichtung mit an gegenüberliegenden Seiten des durchlaufenden Materials ( 1) versetzt angreifenden Richtrollen (3, 4, 6, 10), von denen einige abhängig von einem Modell, das anhand von Eingangsdaten des Materials und bei dessen Durchlauf durch die Dressurvorrichtung ermittelten Daten des Drahtes und der Dressurvorrichtung stochastisch ermittelt worden ist, automatisch so angestellt werden, dass die Anforderungen an die Geradheit erfüllt werden, wobei die Stellung mindestens einer Richtrolle laufend adaptiert wird aufgrund der genannten, beim Durchlauf durch die Dressurvorrichtung erfassten Daten, welche für die erzielte Geradheit repräsentativ sind, wobei (i) die Größe und Richtung der an den Richtrollen angreifenden Kräfte an den Richtrollen selbst und/oder (ii) die Temperatur des Materials vor und nach dem Durchgang durch die Anordnung der Richtrollen und/oder (iii) die Position des Materials im Anschluss an jede der Richtrollen gemessen und die erhaltenen Messwerte in das die Anstellung der anstellbaren Richtrollen steuernde Modell eingegeben werden.
Patent CH-713389-A1 (CH)
Title: Système de liaison d'un arbre à une pièce.
Inventor: ALEXANDRE BUFFET
IPC: G04B13/02
Filed: 2017-01-27
Abstract: L’invention concerne un système de liaison pour pièce d’horlogerie comprenant: un arbre (2) sur lequel est destiné à être monté un composant (1) d’une pièce d’horlogerie, ledit arbre (2) présentant une première structure d’arrêt axial (23), et une structure d’arrêt en rotation (20), présentant une géométrie permettant d’assurer un arrêt en rotation, un élément d’arrêt axial (3) doté d’une ouverture (30) conformée pour permettre, dans au moins une position angulaire dudit élément d’arrêt axial (3) par rapport à l’arbre (2), un engagement en translation sur l’arbre (2) et le passage de la première structure d’arrêt axial (23), et un appui sur ladite première structure d’arrêt axial (23) dans au moins une autre position angulaire, dite position d’arrêt, un élément de maintien radial (4), agencé pour coopérer solidairement avec l’élément d’arrêt et doté d’une ouverture (40) conformée pour coopérer avec la structure d’arrêt en rotation (20) dudit arbre (2) pour empêcher une rotation de l’élément de maintien autour dudit arbre (2).
Patent DZ-2551-A1 (DZ)
Inventor: CROCKER LOUIS
IPC: C07D413/06
Filed: 1998-07-01
Granted: 2003-08-15
Abstract: This invention is concerned with a novel polymorphic form of the compound 2-(R)-(1-(R) -(3,5-bis(trifluoromethyl) -phenyl)-ethoxy)-3-(S)-(4-fluoro) phenyl-4-(3-5 (-oxo-1H,4H-1,2,4-triazolo) methylmorpholine which is a tachykinin receptor antagonist useful in the treatment or prevention of disorders of the central nervous system, inflammatory diseases, pain or migraine, asthma, and emesis. The instant polymorphic form has advantages over the other known forms of 2-(R)-(1-(R) -(3,5-bis(trifluoromethyl) -phenyl)ethoxy)-3-(S )-(4-fluoro) phenyl-4-(3-5 (-oxo-1H,4H-1,2,4-triazolo) methylmorpholine in terms of thermodynamic stability and suitability for inclusion in pharmaceutical formulations.
Patent ES-172507-A1 (ES)
Title: Mejoras introducidas en las bombas rotativas
Filed: 1946-02-09
Abstract: Mejoras introducidas en las bombas rotativas que comprenden en combinación un cuerpo que tiene una cavidad cilíndrica y una cámara de válvulas formada en ella extendiéndose esta cámara tangencialmente a dicha cavidad siendo la totalidad de la cámara de válvulas parte de dicha cavidad y comunicando directamente con ella una entrada formada en dicho cuerpo una salida formada en dicho cuerpo en el mismo lado de la cavidad cilíndrica que la entrad y en el lado opuesto de dicha cámara de válvulas con respecto a la entrada un rotor excéntricamente sostenido en el cuerpo para mantener una porción de la periferia del mismo en contacto deslizante con la periferia de dicha cavidad de cuerpo medios que constituyen una válvula situada en dicha cámara de válvulas en alineación virtual con la entrad estando la entrada la salida la cámara de válvulas y la válvula situadas unas junto a otras teniendo dicha válvula un vástago alargado y una porción que se extiende transversal mente a dicho vástago y una superficie considerablemente ancha en contacto de deslizamiento con una superficie considerablemente ancha de la cámara de válvulas que se extiende transversalmente al eje de la entrada y teniendo otra superficie considerablemente ancha que se desliza sobre la periferia del rotor y un pivote montado en la entrada en el lado de la misma apartado del paso del fluido de salida en la bomba y que sostiene el extremo exterior del vástago.
Patent ES-176784-A1 (ES)
Title: PERFECCIONAMIENTOS INTRODUCIDOS EN LAS PLUMAS ESTILOGRáFICAS
Filed: 1947-02-12
Abstract: Perfeccionamientos introducidos en las plumas estilográficas de escritura seca caracterizados por el hecho de que el órgano escribiente de la pluma está constituido por una bolita giratoria constantemente en contacto con una tinta especial contenida en un depósito prácticamente inagotable estando previstos medios para hacer independiente el pulsador de la lámina que lleva el pestillo de guía en la sola dirección de la rotación; medios que sirven también para la unión axil del pulsador al conjunto escribiente y medios para deshacer el bloqueo del pestillo que fija el pulsador y el conjunto escribiente en posición de escritura.