baber/WOPTO huggingface dataset:
Patent NZ-597983-A (NZ)
Title: Tricyclic heterocyclic compounds as phosphoinositide 3-kinase inhibitors
Inventor: SHUTTLEWORTH STEPHEN JOSEPH
IPC: A61K31/519
Filed: 2010-08-19
Abstract: 597983 Disclosed are compounds of formula (I) or pharmaceutically acceptable salts thereof, wherein: W is O, NH, N(C1-C10 alkyl) or S; each X is independently CH or N; R1 is a 5 to 7- membered saturated or unsaturated, optionally substituted heterocycle containing at least 1 heteroatom selected from N or O; R2 is (LQ)m Y; and each R3 is independently H, C1-C10 alkyl, aryl or heteroaryl, are found to be inhibitors of PI3K-p110 delta. Compounds of the disclosure include: 8-Azetidin-1-ylmethyl-2-(1H-indol-4-yl)-4-morpholin-4-ylpyrido[3’,2’:4,5]furo[3,2-d]pyrimidine Cyclopropyl-[2-(1H-indol-4-yl)-4-morpholin-4-ylpyrido[3’,2’:4,5]furo[3,2-d]pyrimidin-8-ylmethyl]-methyl-amine 3-{ 4-[2-(1H-Indol-4-yl)-4-morpholin-4-yl-pyrido[3’,2’:4,5]furo[3,2-d]pyrimidin-8-ylmethyl]-piperazin-1-yl} -propionitrile And 8-(4-Fluoro-piperidin-1-ylmethyl)-2-(1H-indol-4-yl)-4-morpholin-4-yl-pyrido[3’,2’:4,5]furo[3,2-d]pyrimidine
Patent NZ-599305-A (NZ)
Title: Powder inhaler
Inventor: KAEMPER MARKUS
IPC: A61M15/00
Filed: 2010-09-30
Abstract: The disclosure relates to an inhaler for inhaling powdery pharmaceuticals from capsules, comprising - a bottom part (6) - a plate (3) received in the bottom part (6), and a mounting (18) introduced in the bottom part (6), - a mouth piece (2) that can be latched to the bottom part (6) on the plate (3), - a cover (1) that covers the mouth piece (2) in a closed position and latches by means of a closure element (14), wherein the bottom part (6) and the cover (1) are rotatably connected to each other by an axis (4), and - an actuating member (7, 10), which can be set in motion from a position of rest and in the process cooperates with at least one needle (8, 11) that can pierce the mounting (18), said needle being located in a needle holder of the inner actuating member (10).; An exchange tube (22) can be inserted in the mounting (18) as a discharge channel, the tube comprising a capsule chamber (21) with the capsule.
Patent NZ-599705-A (NZ)
Title: Process for the preparation of calcobutrol
Inventor: TRENTMANN WILHELM
IPC: A61K49/10
Filed: 2010-11-02
Abstract: NZ 599705 The disclosure relates to a process for the preparation of the calcium complex of 10-(2,3-dihydroxy-1-(hydroxymethyl)propyl)-1,4,7,10-tetraazacyclodecane-1,4,7-triacetic acid (Calcobutrol), wherein the process comprises the steps of: (a) the gadolinium complex of 10-(2,3-dihydroxy-1-(hydroxymethyl)propyl)-1,4,7,10-tetraazacyclodecane-1,4,7-triacetic acid (Gadobutrol) is de-complexed with a de-complexing agent, wherein the de-complexing agent is an oxalate ion source or a phosphate ion source and the pH before adding the de-complexing agent is higher than 2, (b) the precipitated gadolinium salt is removed, (c) the free ligand in the solution resulting from step (b) is bound to an acidic ion exchange resin, (d) said resin is eluted with an aqueous alkaline solution, (e) the eluate is treated with acidic ion exchange resin, and (f) the ligand is complexed with Ca2+ ions and crystallised.
Patent NZ-619990-A (NZ)
Title: Animal supplements and compositions containing soluble monensin and methods therefor
Inventor: GAWLAK JON THOMAS
IPC: A23K20/195
Filed: 2012-07-26
Abstract: An animal feed supplement in solution form, comprises monensin present in the supplement in a concentration of 5% to about 40% (weight/weight) of the solution, and a solvent selected from mixtures of at least two of benzyl alcohol, oleic acid, propylene glycol, vitamin E, ethanol, glyceryl mono- and di-caprylate with the solvent being present in the supplement in a concentration of about 60% to 95% (weight/weight) of the solution. A food composition comprising the above described animal feed supplement and an animal feed. The above described animal food composition is useful for preventing or treating of coccidiosis in an animal for example a bovine or a goat.
Patent NZ-621597-A (NZ)
Title: Triazolopyridine compounds as pde10a inhibitors
Inventor: FLOHR ALEXANDER
IPC: C07D471/04
Filed: 2012-09-17
Abstract: Provided are triazolopyridine derivative compounds of the general formula (I), wherein the variables are as defined in the specification. Examples of the compounds include 2-Methyl-4-(pyrrolidine-1-carbonyl)-2H-pyrazole-3-carboxylic acid (2-phenyl-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-amide and 2-Methyl-4-(pyrrolidine-1-carbonyl)-2H-pyrazole-3-carboxylic acid [2-(3-methoxypyrrolidin-1-yl)-[1,2,4]triazolo[1,5-a]pyridin-6-yl]-amide. The compounds are phosphodiesterase 10A (PDE10A) inhibitors. The compounds may be useful in the treatment of cancer and neurological disorders.
Patent NZ-623906-A (NZ)
Title: Fiber optic cassette, system, and method
Inventor: OTT MICHAEL JAMES
IPC: G02B6/46
Filed: 2012-10-05
Abstract: A fiber optic cassette is disclosed. The cassette (10) has a body defining a front and an opposite rear and an enclosed interior. A cable entry location is defined in the body for a cable (12) to enter the interior of the cassette. The cable which enters at the cable entry location is attached to the cassette body and the fibers (26) are extended into the cassette body and form terminations at connectors (92). The connectors are connected to adapters (100) located at the front of the cassette. A front side of the adapters defines termination locations for cables to be connected to the fibers connected at the rear of the adapters. A cable including a jacket, a strength member, and fibers enters the cassette. The strength member is crimped to a crimp tube (70) and is mounted to the cassette body, allowing the fibers to extend past the crimp tube into the interior of the cassette body. A strain relief boot (60) is provided at the cable entry location. The cable entry location is located at the rear of the cassette body opposite to the front. The adapters along the front are arranged linearly in one embodiment and extend in a longitudinal direction parallel to the major surfaces defined by the top and the bottom of the cassette body. The cable at the cable entry location extends parallel to the longitudinal direction before entry into the cassette body. Disposed within the cassette body are cable radius limiters which provide cable management of the fibers extending from the cable entry location to the connectors at the rear of the adapters. In one embodiment, an adapter block with a plurality of adapters is formed and includes a front end, a rear end, and internal structures which allow mating with fiber optic connectors (108) at the front end, such as SC or LC style connectors. The adapter block may be removable from a remainder of the cassette. A rear of the adapter block defines a rear clip which retains a split sleeve and a hub and ferrule of a connector which terminates an interior fibre which is cheaper to terminate, or the rear end of the adapter block defines an opening for receipt of an SC or LC style connector. The cassette can be utilized in a chassis which includes a stationary mount relative to the chassis, or the cassette can be movably mounted, such as in a variety of sliding movements to allow access to a selected cassette, thereby improving access to a selected front connector attached to the cassette.
Patent NZ-701661-A (NZ)
Title: Method for the preparation of triazole compounds
Inventor: MILITZER HANS-CHRISTIAN
IPC: C07D403/14
Filed: 2013-05-06
Abstract: The present invention relates to a process for preparing 1-[6-(morpholin-4-yl)-pyrimidin-4-yl]-4-(1H-1,2,3-triazol-1-yl)-1H-pyrazol-5-ol (I - enol form) or 2-[6-(morpholin-4-yl)-pyrimidin-4-yl]-4-(1H-1,2,3-triazol-1-yl)-1,2-dihydro-3H-pyrazol-3-one (I - keto form) from 1,2,3-triazole (III), methylbromoacetate (IV-Me-Br) or ethylbromoacetate (IV-Et-Br), 4,6-dichloropyrimidine (VIII), morpholine (IX) and hydrazine (XII).
Patent NZ-717108-A (NZ)
Title: Improved process for preparing infant formula using a rotary atomizer
Inventor: VAN DEN BRENK JOEP
IPC: A23D7/00
Filed: 2014-09-11
Abstract: The present invention relates to a process for preparing a spray-dried lipid and protein component- containing composition using a rotary atomizer, which composition comprises large lipid globules, preferably coated with polar lipids, and to the compositions obtained thereby. The obtained compositions are preferably for feeding infants and young children.
Patent NZ-721749-A (NZ)
Title: Improved o-ring drill hole plug
Inventor: PHILLIPS JEFFREY BRUCE
IPC: F16L55/11
Filed: 2014-12-22
Abstract: A plug (10) for blocking off mining exploration drill holes. The plug (10) comprises an elongate body (12) of solid impervious material, and an engineered surface (14) is provided on an external circumference of the elongate body (12). The engineered surface (14) comprises an annular anchoring groove (16) having a ramp (18) extending from a maximum diameter to a minimum diameter of the engineered surface (14) in a braking direction, in which it is intended to prevent movement of the plug (10) in the drill hole. The plug (10) also comprises an O-ring (20) received in the anchoring groove (16) and having a thickness whereby it protrudes slightly above the maximum diameter of the engineered surface (14) and engages with a wall (22) of the drill hole. In use, when the plug (10) is moved in the braking direction in the drill hole, the O-ring (20) rolls up the ramp (18) and wedges between the engineered surface (14) and the wall (22) of the drill hole to provide a braking action for the plug (10) against the wall (22) of the drill hole.
Patent NZ-728709-A (NZ)
Title: Corona discharge cells
Inventor: BRAUER JOHN LIONEL
IPC: H01T19/04
Filed: 2015-07-01
Abstract: A corona discharge apparatus comprising: (a) an elongate inner electrode, (b) an elongate dielectric sleeve mounted on the inner electrode, (c) an elongate outer electrode mounted on the dielectric sleeve, and (d) at least a pair of spaced sealing members between the inner electrode and the dielectric sleeve which define an ozone-producing region over which the outer electrode extends, the ozone-producing region having an inlet end and an outlet end, wherein an outer surface of the inner electrode located within the ozone-producing region is smooth.
Patent NZ-735249-A (NZ)
Title: Tetrahydrofurane-fused aminohydrothiazine derivatives which are useful in the treatment of alzheimer’s disease
Inventor: RICHARDS SIMON JAMES
IPC: C07D513/04
Filed: 2016-04-22
Abstract: The present invention provides a compound of Formula I: or a pharmaceutically acceptable salt thereof. The compounds are inhibitors of BACE. The compounds can be useful for the treatment of Alzheimer’s disease or for preventing the progression of mild cognitive impairment to Alzheimer’s disease.
Patent NZ-738017-A (NZ)
Title: Bucket for a construction vehicle used for loading, moving, transporting, pouring or spreading bulk material
Inventor: ABGRALL ROLAND
IPC: E02F3/43
Filed: 2016-06-10
Abstract: A bucket for an industrial vehicle configured to load, move, transport, tip and spread a bulk material, the bucket comprises: two lateral panels extending on each side of a loading panel, said loading panel comprises a loading edge and an unloading edge; a support panel to support an adjuster configured to adjust a thickness of a layer of bulk material to be spread on the ground, said support panel being situated on other side of the bucket from the loading panel; an opening panel comprising a gate comprising an opening edge, the opening edge is adjacent to the unloading edge of the loading panel when the gate is in a closed position, the closed position of the gate is configured to hold back the bulk material, the opening edge moves away from the unloading edge of the loading panel to create an opening when the gate is in an open position, the opening allows the bulk material to pour out; the adjuster comprises a rotationally moveable roller situated under the bucket and configured to turn in a rotational direction of wheels of the vehicle and to rest on the ground during a spreading operation; and a fixing attachment configured to be fixed to the vehicle, the fixing attachment being housed in a vertical translationally movable space configured to allow a vertical translational movement and the fixing attachment is configured to rotationally move about an axis of rotation perpendicular to the support panel so as to turn the bucket relative to the ground.
Patent NZ-742410-A (NZ)
Title: A cavity closer
Inventor: SPAKE LUKE DUNCAN
IPC: E06B1/60
Filed: 2017-05-17
Abstract: An assembly including a cavity closer (1) and a masking flap (2), the cavity closer including: a base (6) including a plurality of apertures (3); a flat upstand portion (4), extending at 90 degrees along a first edge of the base; a ridge (5), extending from a second edge of the base; and a flexible tip extending from the ridge. The masking flap is connected to the upstand portion, ridge or base of the cavity closer, and configured below the apertures to substantially conceal the apertures of the cavity closer from view. In use, the cavity closer closes a cavity behind a cladding and there is a gap between a tip of the masking flap and the back of the cladding. The disclosed cavity closer allows any liquid to drain out through the concealed apertures, prevents vermin from entering a cavity behind cladding, and the flexible tip hides any discrepancies in cladding.
Patent NZ-780825-A (NZ)
Title: Lanthionine c-like protein 2 ligands, cells prepared therewith, and therapies using same
Inventor: BASSAGANYA-RIERA JOSEP
IPC: A61P3/10
Filed: 2020-12-18
Abstract: Provided are compounds that target the lanthionine synthetase C-like protein 2 pathway. The compounds can be used to treat a number of conditions, including autoimmune diseases, inflammatory diseases, chronic inflammatory diseases, diabetes, and infectious diseases, such as lupus, rheumatoid arthritis, type 1 diabetes, inflammatory bowel disease, viral diseases, and nonalcoholic steatohepatitis. The compounds can also be used to generate cells, such as immune cells, for treating the conditions.
Patent PT-101465-A (PT)
Title: Means for filling and sealing bags - incorporates a sealable filling valve sealed with hot melt glue under heat and pressure
Inventor: SELMIN BENITO
IPC: B65B51/00
Filed: 1994-02-25
Abstract: A bag (5) having a filling valve (V) with hot melt glue (C) disposed on the inner surfaces of said valve. An automated filling and sealing system for said bags incorporates a belt carrier (1) with guides (3), with slides (4) on which are mounted plates (5a, 5b), in such manner as to be vertically raised or lowered. After filling said bags, heated plate (5a) is lowered to soften the glue, said plate being temperature controlled by thermocouple. Said heating plate (5a) is then raised and second plate (5b), being perforated and supplied with compressed air, cools the glue and seals the valve.
Patent PT-101673-A (PT)
Title: Support system for a camera for capturing an image under special conditions
IPC: F16M11/00
Filed: 1995-03-21
Abstract: The system is based on a camera head with full correction capability horizontally and vertically, through 360 degree, which is fitted to a remote-controlled carriage which moves on rails. The entire assembly is controlled "without wires". It consists of the following: 1 - control of six or more channels, commonly used in radio-controlled modelling; 2 - compatible receiver; 3 - mechanical servos, which are also compatible, two of which are converted for continuous operation; 4 - base which rotates horizontally and vertically to support a video camera actuated via the servos; 5 - a second base intended to receive the first four equipped with an electric motor and four-wheel drive with variable speed drive connected to the receiver 2. Adaptation to a model vehicle; 6 - channels 2 m in length, in aluminium section I, joined in parallel by wooden crosspieces. The possibility of being joined end to end allows the total length of the assembly to be infinite. Optionally, the channels may be suspended, the vehicle operating inverted. The figure which illustrates the abstract relates to this situation. <IMAGE>
Patent PT-104069-A (PT)
Title: Sistema de reconversão da energia gerada em motores trifásicos assíncronos do volante de engenhos de corte de rochas ornamentais
Inventor: LOURENCO ALBERTO MANUEL LOUREI
IPC: H02K47/00
Filed: 2008-05-21
Abstract: A PRESENTE INVENÇÃO REFERE-SE A UM SISTEMA PARA RECONVERSÃO DA ENERGIA GERADA EM MOTORES TRIFÁSICOS ASSÍNCRONOS DO VOLANTE DE ENGENHOS DE CORTE DE ROCHAS ORNAMENTAIS, DE FORMA A GARANTIR A MÁXIMA EFICIÊNCIA NO CONSUMO DE ENERGIA ELÉCTRICA DO MOTOR PRINCIPAL (MOTOR DO VOLANTE), RENTABILIZANDO O SEU FUNCIONAMENTO. O PRESENTE SISTEMA É COMPOSTO POR EQUIPAMENTOS QUE AO SEREM APLICADOS A MOTORES TRIFÁSICOS ASSÍNCRONOS DE VOLANTES DE ENGENHOS DE CORTE DE ROCHAS ORNAMENTAIS PERMITEM RENTABILIZAR A ENERGIA CONSUMIDA POR ESTES MOTORES. ESTES EQUIPAMENTOS SÃO: - VARIADOR ELECTRÓNICO DE VELOCIDADE (5) (VEV), - REGENERADOR (9), - FILTRO DE ALTAS FREQUÊNCIAS (3) PARA ENTRADA DO VARIADOR ELECTRÓNICO DE VELOCIDADE (VEV), - FILTRO DE ALTAS FREQUÊNCIAS (12) PARA SAÍDA DO REGENERADOR, - FILTRO DE HARMÓNICAS OU IMPEDÂNCIA DE CHOQUE (4) PARA A ENTRADA DO VARIADOR ELECTRÓNICO DE VELOCIDADE (VEV), - FILTRO DE HARMÓNICAS OU IMPEDÂNCIA DE CHOQUE (11) PARA A SAÍDA DO REGENERADOR, - CABO DE SINCRONISMO DE REDE (10), - DÍODOS DE POTÊNCIA (8) PARA ANTI-RETORNO DA CORRENTE CONTÍNUA (DC).
Patent RU-94007124-A (RU)
Inventor: MALYSHEV V V
IPC: B64D37/30
Filed: 1994-03-02
Abstract: FIELD: aeronautical engineering; multiengined aircraft operating on cryogenic fuel. SUBSTANCE: fuel pipe lines are made without blind sections to avoid penetration of bubbles of propellant vapor into engine; cross-feed lines are excluded as well; in case of failure of engine and/or fuel pipe line, fuel from tank of defective engine is transferred to tank of serviceable engines or to tanks common for all engines through pipe lines specially provided for the purpose. EFFECT: enhanced reliability. 5 cl, 3 dwg
Patent RU-94022986-A (RU)
Inventor: KVASENKOV O I
IPC: B01D11/02
Filed: 1994-06-29
Abstract: FIELD: extraction of biological raw material by liquid extractants in food-processing industry, medicine and perfumery. SUBSTANCE: apparatus has condenser, at least one extractant, evaporator and separator, which are connected in series through manifolds with locking fittings to define closed circuit. Extractor has bubbler mounted in its lower part. Apparatus is further provided with extractant supplying device, extract collector, auxiliary manifolds with locking fittings for connecting condenser-extractor manifold with evaporator and extractor-evaporator manifold with condenser, and auxiliary manifold with adjustable locking fittings and return valves for connecting evaporator-separator manifold with bubbler. EFFECT: increased efficiency, wider operational capabilities and enhanced reliability in operation. 1 dwg
Patent RU-94027251-A (RU)
Inventor: MALIKOV N V
IPC: B60T15/60
Filed: 1994-07-18
Abstract: FIELD: railway transport; traction vehicles. SUBSTANCE: in proposed method of checking connection of control instruments to brake pneumatic system, interlocking device is used for continuously measuring absence of compressed air pressure in main line tap of brake valve in inoperative locomotive cab and presence of compressed air pressure in brake main line of operative cab and, simultaneously, disconnecting auxiliary brake valve in inoperative cab and connecting auxiliary brake valve in operative cab with auxiliary brake main line. Vehicle can be set into motion only from operative cab. EFFECT: prevention of negative influence of interlocking device onto process of brake release and charging and prevention of possibility of setting into motion the vehicle with non-charge brake main line.
Patent RU-94036001-A (RU)
Inventor: GABRIEHL NECHUSHTAN
IPC: A45C/
Filed: 1992-01-17
Abstract: FIELD: light industry. SUBSTANCE: expandable case 10 has rigid central part 20 defining at least one laterally open edge and parallel guides 28 for receiving rib 16. Guides 28 are extending in parallel with open edge of case. Case has movable side section 12,14 defining rigid rib 16 extending along its peripheral length. Rib 16 have size providing sliding engagement with guides 28. Rib is positioned in such a way that it may be selectively brought into engagement with one of guides, with none of guides extending beyond section. At least one side section may be moved relative to central part from one guide to another to receive required volume of case. EFFECT: increased convenience and wider operational capabilities. 1 dwg
Patent RU-94039279-A (RU)
Inventor: UMBERTO ZARDI
IPC: C07C29/152
Filed: 1994-10-28
Abstract: FIELD: chemical, petrochemical branches of industry. SUBSTANCE: method to modernize reactor for heterogeneous exothermal synthesis, that has outer body, in which at least one catalytic layer is located, linked with high pressure vapor generation outside boiler by nozzle for reacted gas removal and pipeline located in the nozzle and so forming ring-type air clearance. Advantage is the fact, that air clearance forms exit way for gasses stream cooled in boiler, tat allows to avoid nozzle overheating. EFFECT: method to modernize reactor allows to avoid nozzle overheating. 3 dwg
Patent RU-94042612-A (RU)
Inventor: SAITKULOV V G
IPC: G01B17/02
Filed: 1994-11-30
Abstract: FIELD: measurement technology. SUBSTANCE: invention refers to ultrasonic inspection of articles and may be used to measured flow section of pipes with internal deposits. Method involves input of ultrasonic oscillations into pipe-line along normal to outer surface and reception with the aid of two ultrasonic converters placed on diametrically opposite outer surfaces of pipe-line of ultrasonic oscillations passed through walls of pipe-line. Time of passage of ultrasonic oscillations from first converter to boundary of separation between liquid and opposite inner surface of pipe-line with deposits is measured, time of passage of ultrasonic oscillations from the other converter to boundary of separation between liquid and opposite inner surface of pipe-line with deposits is measured, time of passage of ultrasonic oscillations from one converter to the other one is measured and flow section of pipe-line is found by formula:, where D is diameter of flow section of pipe-line; tis time of passage of ultrasonic oscillations from first converter to boundary of separation between liquid and opposite inner surface of pipe-line with deposits; tis time of passage of ultrasonic oscillations from second converter to boundary of separation between liquid and opposite inner surface of pipe-line with deposits; tis time of passage of ultrasonic oscillations from one converter to other converter; C is velocity of ultrasound in liquid. EFFECT: enhanced precision of measurement of flow section of pipe-line with deposits on inner walls of pipes without interruption of process of usage of pipe-line. 1 cl, 1 dwg