baber/WOPTO huggingface dataset:
Patent EA-016360-B1 (EA)
Title: Inhibitors of 11-beta-hydroxysteroid dehydrogenase 1, pharmaceutical composition based thereon and use thereof
Inventor: LI RENHUA
IPC: A61K31/4545
Filed: 2007-04-25
Abstract: The present invention discloses novel compounds of Formula I:possessing 11β-HSD type 1 antagonist activity, as well as methods for preparing such compounds. In another embodiment, the invention discloses pharmaceutical compositions comprising compounds of Formula I, as well of using compounds in therapy and for preparing a medicament. Besides, the present invention relates to an intermediate compound for the synthesis of said compounds of Formula I, where said intermediate compound is a compound of a structure
Patent EA-015063-B1 (EA)
Title: Locking-sealing device
Inventor: TEMBAEVA GULNARA ISAKHMETOVNA
IPC: G09F3/03
Filed: 2009-11-05
Abstract: The proposed device relates to locking and simultaneous sealing containers, railway cars, cisterns, truck bodies and other objects for transporting and/or storing goods, mainly at railway for preventing access to gods by outsiders or violators. The inventive device is aimed at broadening a range of technical means for use as a locking-sealing device, simplification and compactness of design, manufacturing process at high reliability and high rupture strength. The locking-sealing device comprises a hollow housing with two through holes, a flexible element as a wire rope, one end of which is rigidly secured in the housing, a cylindrical sleeve with inner cylindrical surface inside which a holder is arranged comprising a support with beads, a spring cooperating with the holder, and a set of washers. Three inclined grooves spaced evenly are made on the sleeve inner surface. A holder support is made as a cylinder, a side surface if which has three trapezoidal slots spaced evenly along the circle, providing beads displacement both in axial and perpendicular directions to the axis in interacting beads surface with the inclined side surfaces of the groove slots and the wire rope. The set of washers comprises a flange washer and flat spring washer, a support washer and an insert washer. The wire rope can be extracted only in case of its damage, that is repeated locking of the device is excluded.
Patent EA-017508-B1 (EA)
Title: Fast dissociating dopamine 2 receptor antagonists
Inventor: MACDONALD GREGOR JAMES
IPC: A61K31/495
Filed: 2008-02-11
Abstract: The present invention relates to 4-aryl-6-piperazin-1-yl-3-substituted-pyridazines that are fast dissociating dopamine 2 receptor antagonists, processes for preparing these compounds, pharmaceutical compositions comprising these compounds as an active ingredient. The compounds find utility as medicines for treating or preventing central nervous system disorders, for example schizophrenia, by exerting an antipsychotic effect without motor side effects.
Patent EA-017414-B1 (EA)
Title: Sludge scraper to radial settling tank
Inventor: KURYATNIKOV ALEXEJ ALEXEEVICH
IPC: B01D21/18
Filed: 2011-08-05
Abstract: The invention relates to purification of waste waters, in particular to devices for purification of radial settling tanks from sediments as solids precipitate in the process of sewage clarification. The technical result is aimed at raising efficiency, reliability, repair ability and long life operation of the scraper by using a roller bearing of OΠ 1600 type in the central support. A pedestrian frame is designed as a bridge which represents an isosceles triangle in view plan, wherein the triangle vertexes are positioned on the central support and two electric drives on the triangle base. A bogie positioned at the triangle base provides to move apart electric drive considerably thus avoiding slipping in winter time. Two scraping members of the scraper for sludge moving are arranged at an angle to each other and form an angular scraper, wherein two others are positioned one by one before the angular scraper in the direction of the frame rotation directly in a circular sludge sink. Two scrapers forming the angular scraper are made of sections, the angle between scrapers is 80-120°. The sections are hinged connected providing to clean rough surfaces of the settling tank bottom, the scrapers have limiting stops preventing bottom scraping at rubber wear.
Patent EA-025865-B1 (EA)
Title: Crystalline form of pemirolast
Inventor: PERLBERG ANETT
IPC: A61P29/00
Filed: 2010-06-15
Abstract: There is provided a hemihydrate form of the sodium salt of pemirolast.
Patent EA-028126-B1 (EA)
Title: Trigger and firing mechanism of automatic weapons
IPC: F41A19/06
Filed: 2014-02-26
Abstract: The invention relates to automatic weapons, i.e. trigger and firing mechanisms, which provide firing in the single-shot and automatic modes and in the automatic burst mode. The trigger and firing mechanism contains a trigger, a rod, a firing pin, a spring-loaded sear, a spring-loaded free rod, a spring-loaded inertia plunger with a safety lock, a rod with a spring and a fire selector. The spring-loaded sear is installed in a modular body wit attachment option; herewith a modular body is installed on pins and spring-loaded. The modular body is fitted with a separator, which prevent a shot when the breech mechanism and the safety lock are not fully closed. The technical result of the invention is the development of a hammerless trigger and firing mechanism, which provides firing in the single-shot and automatic modes and in the automatic burst mode limited to 2 rounds.
Patent EA-025908-B1 (EA)
Title: Brines for completing a wellbore
Inventor: PEREZ GREGORY PAUL
IPC: C09K8/03
Filed: 2012-10-14
Abstract: Clear, high density brine for use in wellbore completion operations in a subterranean formation for the recovery of hydrocarbons. The brine comprises an ionic compound selected from the group consisting of zinc iodide, strontium bromide, strontium iodide, cerium bromide, cerium iodide, cerium chloride, lanthanum bromide, lanthanum iodide, lanthanum chloride, and mixtures thereof. The brine may also advantageously be used as the internal phase of invert emulsion drilling fluids.
Patent EA-032648-B1 (EA)
Title: System and grinding disc for grinding with the continuous monitoring of wear of a grinding element
Inventor: HEINRICHS ROBERT EVAN
IPC: B02C17/16
Filed: 2014-05-20
Abstract: The application describes a system for the continuous monitoring of wear. The system comprises a grinding mill (100) having at least one grinding disc (106). At least one detector (141) is provided to the at least one grinding disc (106), and at least one sensor (120) is provided to the grinding mill (100) which is configured to communicate with the at least one detector (141) during operation of the grinding mill (100). In use, the at least one grinding disc (106) wears away and ultimately affects a function of the least one detector (141). The at least one sensor (120) is configured to monitor said function of the least one detector (141). When the at least one sensor (120) detects a change in the signal of the at least one detector (141), an operator is notified that maintenance or grinding disc replacement may be necessary.
Patent EA-030390-B1 (EA)
Title: Method and device for determination of individual characteristic frequency of biological object
Inventor: BARANOV VALENTIN VLADIMIROVICH
IPC: A61B5/05
Filed: 2016-03-25
Abstract: The invention relates to electronic engineering, particularly ultrahigh frequency (UHF) engineering, and may be applied to diagnostics in phytopathology and chronic diseases in a human, based on determination of response coherent to a defined frequency from a biological object when it is sensed with UHF radiation. Objective of the claimed invention is increasing accuracy in determination of characteristic frequency of biological objects and automation of biomedical examination procedure. The set objective is solved by a method, wherein electrically frequency-controlled signal in millimetre wavelength range is formed, directed onto aimed acupuncture point or biological object surface point, reflected UHF signal carrying information of amplitudes and phases of the object in frequency retuning range is received, information of skin cover or biological object impedance in aimed acupuncture points or surface is obtained, and a value of characteristic frequency of biological object is determined, according to frequency point with maximum coherence condition, reflected UHF signal phase change, and skin cover of surface impedance change. The device according to the above method comprises a sweep frequency generator that forms electrically frequency-controlled signal in millimetre wavelength range, an unidirectional coupler oriented to reflected UHF signal and connected to miniature transceiver dielectric antenna, which energises aimed acupuncture or surface point, a measuring UHF tract whereto reflected UHF signal from biological object arrives, contact terminals with converter, connected to aimed acupuncture or surface points of biological object, a processing device for measuring information that controls the generator, receives and converts into digital codes analogue signals, which bear information of amplitude and phase of reflected UHF signal, and of changing skin cover of surface impedance, and which arrive from measuring UHF tract and from contact terminals, respectively, and a computer with a display, wherein individual characteristic frequency of biological object is determined and displayed on the screen.
Patent EA-030255-B1 (EA)
Title: Plant for processing organic raw material using pyrolysis method
Inventor: LADYGIN KONSTANTIN VLADIMIROVICH
IPC: C10B53/00
Filed: 2015-07-07
Abstract: A plant for processing organic raw material using a pyrolysis method contains a reactor (1); a loading hopper (2) for solid raw material; a loading screw conveyor (3); a loading reservoir (4) for liquid raw material; a loading pump (5); a smoke exhaust (7); a smoke flue (8), an intermediate screw conveyor (20); a storage container (21) for ash residue; an unloading screw conveyor (22); a vapour-gas mixture filter (9); a heat exchange device (10); a cooling device (11); a circulation pump (12) for a cooling liquid; a gas-liquid separator (13); a gas-drying column (14); a hydraulic valve (15); a storage tank (16); a residual-water separator (17); a tank for water (18); a fuel tank (19); a nitrogen source (23); and also pipelines, and the following, which are not shown in fig. 1: a compressor for supplying air to a combustion chamber; shut-off and adjustment fittings; expansion containers and compensating containers; and an automated control system. If necessary, the plant can contain a device for flue gas purification (6); a catalytic reactor (25); and an electrical power unit (24) of a stand-alone power supply of the plant. The reactor (1) is an assembly for thermal destruction, and contains a substantially cylindrical pyrolysis chamber (107), in a lower portion of which a screw conveyor (101) is arranged, said screw conveyor providing for the supply of raw material to the pyrolysis chamber (107), the displacement of raw material along the pyrolysis chamber (107) during processing, and the removal of ash residue from the pyrolysis chamber (107). The technical result involves enabling the plant to process solid and liquid raw material, in arbitrary combinations, with a nonstandardised moisture content, and providing for increased safety of use and an extended life between overhauls, and providing a predetermined chemical and fractional composition of a liquid pyrolysis fuel and ash residue.
Patent EA-037085-B1 (EA)
Title: Stuffy nose deblocking composition having antiviral activity
Inventor: GRASSAUER ANDREAS
IPC: A61P31/16
Filed: 2016-07-12
Abstract: The invention relates to a hyperosmolar pharmaceutical composition adjusted for topical administration to the nasal cavity for stuffy nose deblocking, having activity against viral infections of the respiratory tract, characterized in that the composition comprises a non-ionic osmolality adjusting agent in combination with an ionic osmolality adjusting agent and a carrageenan component as an active antiviral ingredient, comprising a nasally compatible buffer, wherein said composition has a pH value of from 4.0 to 8.0; disodium edetate (EDTA) at a concentration of up to 2 mg/ml; not more than 1.5% w/v of said ionic osmolality adjusting agent; from 1 to 15% w/v of said non-ionic osmolality adjusting agent; from 0.05 to 1% w/v of the carrageenan component as the sole active antiviral ingredient, and said composition has a hyperosmolar osmolality value of from 500 to 1000 mOsm/kg, and to the use thereof in preparing a medicament for unblocking of a congested nose and simultaneous treatment of a viral infection of the upper respiratory tract.
Patent EA-035906-B1 (EA)
Title: Process for the epoxidation of propene
Inventor: WOELL WOLFGANG
IPC: C07D301/12
Filed: 2017-03-10
Abstract: The present invention provides a process for the epoxidation of propene by continuously reacting propene with hydrogen peroxide in a methanol solvent and in the presence of a shaped titanium silicalite catalyst in a tube bundle reactor, wherein during start-up of the reaction cooling medium is fed to a cooling jacket at the rate for full load of the reactor and with a constant entry temperature of from 20 to 50°C, methanol solvent is fed at a rate of from 50 to 100% for full load of the reactor, hydrogen peroxide is fed at a rate that starts with no more than 10% of the rate for full load and is increased continuously or stepwise to maintain a maximum temperature in the fixed bed of no more than 60°C and a difference between the maximum temperature in the fixed bed and the cooling medium entry temperature of no more than 20°C, and propene is fed at a rate of from 20 to 100% of the rate for full load, increasing the feeding rate when the molar ratio of propene to hydrogen peroxide reaches the molar ratio for full load.
Patent ES-2170649-B1 (ES)
Inventor: FOGUET AMBROS RAFAEL
IPC: A61K31/00
Filed: 2000-03-29
Granted: 2003-06-16
Abstract: The invention relates to the use of CDP-Choline or its pharmaceutically acceptable salts for the preparation of a medicinal product for the treatment of alcohol withdrawal syndrome at daily doses equivalent to 0.5-2 g of free CDP-Choline.
Patent ES-2222810-B1 (ES)
Title: Instalacion para aspiracion de humos y/o residuos del interior de vehiculos.
Inventor: MARTINEZ ENRIQUE JUAN ANTONIO
IPC: B60N3/08
Filed: 2003-07-18
Granted: 2006-03-16
Abstract: Instalación para aspiración de humos y/o residuos del interior de vehículos, caracterizada porque consta de, al menos, un conducto principal con al menos una boca de admisión, al menos una boca de escape y dos diferentes secciones (S1), (S2) en dos tramos contiguos con desnivel cero; uno o varios conductos secundarios que, derivados de dicho conducto principal, van asociados a correspondientes terminales y alcanzan diferentes puntos o zonas interiores del vehículo; y un depósito/colector, asociado a la boca de escape y con medios para su descarga, evacuación y limpieza; de modo que, con el vehículo en circulación, entra aire del ambiente a través de la boca de admisión y provoca la aspiración de humos y/o residuos que, sucesivamente a través de dichos conductos secundarios y conducto principal, alcanzan el depósito/colector por el efecto venturi generado de forma directa o indirecta. De aplicación en la industria del automóvil.
Patent ES-2232307-B1 (ES)
Title: Humidor clasificador.
Inventor: SANCHEZ PEREZ OMAR
IPC: G07F9/10
Filed: 2003-11-11
Granted: 2006-04-01
Abstract: Humidor clasificador. El humidor comprende una cámara de almacenamiento (1) de puros (2), en la que tiene lugar la conservación de éstos en las condiciones de humedad y temperatura apropiadas. Lateralmente a dicha cámara de almacenamiento (1) existe una cara de procesamiento (3) en la que tiene lugar el traslado de los puros (2), desde el exterior o compuerta de salida (9) a una zona superior de acceso a través de una compuerta de entrada (15) a dicha cámara de almacenamiento (1). El acceso y salida de esta cámara de almacenamiento, así como la entrada a la cámara de procesamiento, incluyen las respectivas compuertas de hermeticidad (15), (9) y (10) respectivamente. Los puros son pesados y analizada su textura a través de los sensores de presión (12), (18) y son analizados cromáticamente a través de la cámara de captación de imágenes (17). Un computador central (20) analiza la información sensorial y clasifica la calidad de los puros, además de detectar la posible aparición de la lasiodermay moho del tabaco. Se pueden definir diferentes modos de operación a través del teclado (4) y la pantalla de cristal líquido (5).
Patent ES-2237334-B1 (ES)
Title: Orthodontic device comprises ideal orthodontic arches, and extrabuccal dental support bases mounted to ideal hard model for patient or to robot arms , for customizing brackets
Inventor: MARTINEZ ALBAL ELOY ANTONIO
IPC: A61C7/12
Filed: 2004-01-15
Granted: 2006-10-16
Abstract: The ideal orthodontic arches (14) and extrabuccal dental support bases (31) are mounted to ideal hard model for patient or to robot arms (29), for customizing the brackets (2). The segments (49) of adhesive hardenable material are provided between the bracket and intermediate structure (2), for connecting bracket and structure in hardened state and for enabling bracket to move relative to the structure in non-hardened state. An independent claim is also included for application method of orthodontic device.
Patent ES-2297964-B1 (ES)
Title: Filtro incremental inteligente.
Inventor: CARPENO VELAYOS ANGEL
IPC: H03H17/04
Filed: 2005-03-03
Granted: 2009-08-25
Abstract: Filtro incremental inteligente. 
     Nuevo sistema de procesamiento digital de
señales en tiempo real o nueva clase de filtro IIR adaptativo,
dirigido al  modelado robusto y estable de cualquier tipo de proceso
con el fin de realizar su aplicación principalmente en el campo  del
control automático de sistemas, caracterizado porque: 
     a) La estructura del filtro para modelar o
predecir en tiempo real la dinámica instantánea de cualquier sistema
físico  mono o multivariable es un modelo lineal que utiliza valores
incrementales de los vectores de entrada y salida del  proceso. 
     b) La trayectoria guía de referencia o de
aprendizaje tiene que ser limitada y físicamente realizable con
ganancia estática  unidad, y tiene que reinicializarse
constantemente con las salidas medidas del proceso. 
     c) El nuevo algoritmo de aprendizaje se obtiene
de hacer nulo el error instantáneo de estimación entre el incremento
de  la salida del proceso y el incremento de la salida producida por
el modelo incremental del filtro.
Patent ES-2284313-B1 (ES)
Title: Dispositivo para acoplar a un reproductor bidimensional ordinario y conseguir una reproduccion estereoscopica.
Inventor: DOMINGUEZ MONTES JUAN
IPC: G02B30/30
Filed: 2005-03-31
Granted: 2008-09-16
Abstract: Dispositivo para acoplar a un reproductor bidimensional ordinario y conseguir una reproducción estereoscópica que incorpora una trama lenticular (1) capaz de desplazarse lateralmente de izquierda a derecha respecto a una superficie plana difusora (3, 4) donde se reproducen las dos imágenes componentes de un par estereoscópico y de una barrera de paralaje (2) con capacidad de desplazamiento de izquierda a derecha y de delante atrás respecto a la pantalla difusora (3, 4) según el movimiento de la cabeza del observador. La barrera de paralaje (2) está compuesta de barras de un ancho aproximadamente igual a la mitad del ancho de la lente cilíndrica componente de la trama con capacidad de desplazamiento en las direcciones transversal y longitudinal respecto de la superficie difusora (3, 4).
Patent ES-2289860-B1 (ES)
Title: Anteojo estereoscopico de espejos moviles.
Inventor: SILVA GAITAN FERNANDO
IPC: H04N13/00
Filed: 2005-05-06
Granted: 2008-12-16
Abstract: El estereoscopio consta de dos espejos antepuestos al ojo; su uso puede ser monocular o binocular. Estando los espejos paralelos entre ellos y oblicuos con relación al ojo reflejan la imagen a observar en una posición próxima a la que sería observada por la visión directa. Alterando el estado paralelo de los espejos, la figura reflejada permuta su posición espacial, pudiendo de esta forma enfocar dos imágenes en un mismo lugar en el espacio, logrando percibir las dos imágenes como una de condición tridimensional.
Patent ES-2281249-B1 (ES)
Title: Linimento analgesico antiinflamatorio.
Inventor: BENITO MENENDEZ JOSE AGUSTIN
IPC: A61K47/44
Filed: 2006-03-15
Granted: 2008-07-01
Abstract: Linimento analgésico antiinflamatorio compuesto de alcanfor, mentol, salicilato de metilo y aceite de oliva virgen o cualquier otro aceite vegetal, pudiendo sustituirse el aceite de oliva y el vegetal por petrolato líquido, indicado para patologías como artritis, artrosis, reumatismos, dolores por esfuerzos, esguinces, contusiones, dolores musculares, tendinitis, bursitis, luxaciones y golpes causados por actividad deportiva. El linimento se prepara disolviendo al Baño María el alcanfor y el mentol en una porción de aceite de oliva virgen o aceite vegetal, después de disuelto se añade el salicilato de metilo y se completa con el aceite de oliva virgen o aceite vegetal, pudiendo sustituirse los aceites por petrolato líquido.
Patent ES-2284350-B1 (ES)
Title: Metodo y sistema para el desvio de las llamadas recibidas en el terminal movil a una linea fija.
Inventor: MORALES SAMITIER EMMA
IPC: H04W36/14
Filed: 2005-09-27
Granted: 2008-09-16
Abstract: Método y sistema para el desvío de las llamadas recibidas en el terminal móvil a una línea fija, previamente configurado en una aplicación residente en el terminal móvil, dependiendo de si se encuentra dentro del rango de un determinado dispositivo bluetooth. En caso de no encontrarse dentro de dicho rango, las llamadas se reciben directamente en el terminal móvil, a través de la gestión y control de la llamada por medio del nodo de red inteligente IN.
Patent ES-2315181-B1 (ES)
Title: Metodo de obtencion por semisintesis, de derivados de podofilotoxina.
Inventor: DOMANICO HUGO RICARDO
IPC: A61K31/343
Filed: 2007-06-26
Granted: 2010-01-08
Abstract: Método de obtención por semisíntesis, de
derivados de podofilotoxina. 
     Se provee un método para obtener derivados de
podofilotoxina en donde la  reacción de epimerización se lleva a
cabo en un sólo paso de síntesis en  presencia de un solvente
orgánico, preferiblemente solventes apróticos,  cosolventes y sales
de ácidos. Particularmente, el método permite obtener 
picropodofilotoxina (PPP), epipicropodofilotoxina,
demetilpicropodofilotoxina,  demetilepipicropodofilotoxina y sus
correspondientes acetatos, con un alto  grado de pureza y sin
requerir complejos pasos de purificación.
Patent ES-2402147-B1 (ES)
Title: PROCEDIMIENTO PARA LA OBTENCIÓN DE UN SUSTRATO CON NANOCLUSTERS
DE Au FIJADOS EN SU SUPERFICIE, Y SUBSTRATO Y CATALIZADOR OBTENIDOS
MEDIANTE DICHO PROCEDIMIENTO.
Inventor: MENDOZA GOMEZ ERNESTO
IPC: B01J23/52
Filed: 2011-10-17
Granted: 2014-03-04
Abstract: Procedimiento para la obtención de un sustrato con nanoclusters de Au fijados en su superficie, y substrato y catalizador obtenidos mediante dicho procedimiento.#Procedimiento para la obtención de un sustrato con nanoclusters 10 de Au (oro) fijados en su superficie, y substrato y catalizador obtenidos mediante dicho procedimiento. El procedimiento consiste en preparar una solución que contiene en forma dispersa nanoclusters de Au y, también en forma dispersa, un sustrato cuya superficie está funcionalizada con un polielectrolito que le confiere una carga eléctrica neta, y en someter dicha solución a una agitación intensa para provocar la fijación de nanoclusters de Au en la superficie del sustrato. Se obtiene como resultado un sustrato en cuya superficie se encuentran fijados nanoclusters de Au de forma dispersa sin presentar significativamente aglomerados. La invención también se refiere a un catalizador que comprende dicho sustrato con nanoclusters 20 de Au fijados en su superficie. Este catalizador es particularmente apto para su uso en reacciones de oxidación.