baber/WOPTO huggingface dataset:
Patent UA-80120-C2 (UA)
Title: Glucocorticoid mimetics, pharmaceutical composition based thereon
Inventor: BEKKALI YOUNES
IPC: C07C49/577
Filed: 2003-03-21
Abstract: Compounds of Formula (IA) and Formula (IB) wherein R1, R2, R3, R4, R5 and R6 are as defined herein for Formula (IA) or Formula (IB), or a tautomer, prodrug, solvate, or salt thereof; pharmaceutical compositions containing such compounds, and methods of modulating the glucocorticoid receptor function and methods of treating disease-states or conditions mediated by the glucocorticoid receptor function or characterized by inflammatory, allergic, or proliferative processes in a patient using these compounds.
Patent UA-79464-C2 (UA)
Title: Substituted indoles, methods for their production and method for treating disorders mediated by prostaglandin d2
Inventor: BONNERT ROGER
IPC: A61K31/405
Filed: 2003-05-27
Abstract: The present invention relates to substituted indoles of formula (I) useful as pharmaceutical compounds for treating respiratory disorders. , (I)
Patent DE-2538372-C3 (DE)
IPC: H02K37/12
Filed: 1975-08-28
Granted: 1978-06-08
Abstract: A pulse motor comprising a rotor having at least two magnetization axes extending parallel to a shaft of the rotor and angularly spaced apart at a uniform interval, the direction of magnetization of each magnetization axis being opposite to that of the adjacent magnetization axis; a pair of upper stators extending above the rotor and defining two upper gaps between them, said upper gaps being adapted to face respective unlike polarity poles on the upper side of the rotor; a pair of lower stators extending below the rotor and defining two lower gaps between them, said lower gaps being adapted to face respective unlike polarity poles on the lower side of the rotor; and at least one drive coil for magnetizing the upper and lower pair stators alternately to opposite polarities such that the polarity of one of the upper pair stators and one of the lower pair stators is opposite to the polarity of the other upper and lower stators.
Patent DE-2705930-C3 (DE)
IPC: B60K/
Filed: 1977-02-10
Granted: 1981-08-27
Abstract: An automatic multiratio drive transmission having an automatic shift control system with a speed and throttle position pressure controlled shift valve controlling shifts between the highest drive ratio and the next lower drive ratio. When the shift valve is in the lower drive ratio position, a normal speed pressure signal increasing with increasing speed acting on the shift valve overcomes an opposing bias force controlled by throttle pressure to upshift the shift valve to the higher drive ratio position at increasing upshift speeds for increased throttle positions and provides an upshift hysteresis force decreasing with increasing throttle positions to prevent shift cycling as the highest ratio is established in a short time period and after a longer time delay period reduces the normal speed related governor pressure in an amount equal to the upshift hysteresis force at full throttle so that the downshift speed is the same as the upshift speed at the full throttle position.
Patent DE-3036165-C3 (DE)
IPC: G04B19/04
Filed: 1980-09-25
Granted: 1982-03-18
Abstract: Instead of conventional hands, an hour disc and a minute disc are provided. The hands are represented by markers vaporized upon the undersides of the discs. The discs are pivoted on an arbor anchored in the watch glass. This arbor is hollow, and inserted in the free end thereof is a rivet-shaped retaining part which keeps the discs from slipping off the arbor. Each disc is toothed at its circumference. The teeth of the minute disc engage a gear wheel having a pinion which meshes with the teeth of the hour disc. This wheel and pinion are mounted on an arbor, one end of which is anchored in the watch glass. A retaining ring prevents the wheel from becoming detached from the arbor. This gear wheel likewise engages a pinion of another gear wheel mounted on an arbor. One end of this arbor is also anchored in the watch glass. A pinion of a stepping motor meshes with the teeth of the further gear wheel. The yoke of the stepping motor is rigidly connected to the watch glass by means of bolts which likewise have one end anchored in the watch glass. A shaft bearing the pinion and the rotor of the stepping motor is pivoted at one end in a recess in the watch glass. Because all the parts necessary for driving the discs, as well as the discs themselves, are either fixed to the watch glass or pivoted about arbors anchored in the watch glass, plates can be dispensed with, so that manufacture of the timepiece is considerably simplified.
Patent DE-19781742-C5 (DE)
Title: Nachweis von Schmutzstoffen in der Luft
Inventor: KNOX RONALD
IPC: G08B17/107
Filed: 1997-05-02
Granted: 2016-05-19
Abstract: Rauchmelder, umfassend eine Detektorkammer, einen Einlaß zum Einleiten eines zu messenden Luftstroms in die Kammer, einen Auslaß für den Luftstrom aus der Kammer, Einrichtungen für die Erzeugung eines Lichtstrahls innerhalb der Kammer, einen Streulichtdetektor, der auf die Gegenwart von Streulicht innerhalb einer Zone der Kammer infolge der Gegenwart von Rauchteilchen innerhalb des zu messenden Luftstroms in der Zone anspricht, einen Lichtabsorber an einem Ende der Kammer, das von der Lichtquelle entfernt ist, zur Aufnahme und Absorbtion des Strahls nach dem Durchgang durch die Kammer, eine erste Kollimatorscheibe zum Kollimieren des Strahls und eine zweite Kollimatorscheibe hinter der ersten Kollimatorscheibe, wobei die zweite Kollimatorscheibe eine Öffnung mit einer solchen Größe aufweist, dass der durch die erste Kollimatorscheibe kollimierte Strahl durch die Öffnung in der Kollimatorscheibe tritt, ohne den Rand der Öffnung zu berühren, wobei die Öffnung der zweiten Kollimatorscheibe größer als die Öffnung der ersten Kollimatorscheibe ist und die zweite Kollimatorscheibe dazu dient, Lichtschimmer abzufangen, die vom Rand der ersten Kollimatorscheibe stammen, und dadurch Störlicht in der Zone, in der der Nachweis der Lichtstreuung stattfindet, zu reduzieren und der Rauchmelder noch eine weitere Kollimatorscheibe umfasst, die sich hinter der zweiten Kollimatorscheibe befindet und eine Öffnung hat, die größer ist als die Öffnung der zweiten Kollimatorscheibe, so dass der durch die Öffnung in der zweiten Kollimatorscheibe hindurch tretende Strahl auch durch die Öffnung in der weiteren ...
Patent DE-60022050-C5 (DE)
Inventor: VAN WAGENEN C
IPC: C07D241/44
Filed: 2000-06-02
Granted: 2007-10-11
Abstract: The present invention provides compounds, and pharmaceutical compositions containing those compounds, that are active at metabotropic glutamate receptors. The compounds are useful for treating neurological diseases and disorders. Methods of preparing the compounds also are disclosed.
Patent RU-2323235-C9 (RU)
Title: Composition for preparing foam plastic
Inventor: KONONOV MIKHAIL VLADIMIROVICH
IPC: C08L9/02
Filed: 2006-10-19
Granted: 2008-07-10
Abstract: FIELD: chemistry of polymers, chemical technology. 
     SUBSTANCE: composition for preparing foam plastic comprises the following components, mas. p. p.: soluble phenol-formaldehyde resin (novolacs), 20-40; phenol (resol) resin, 60-80; nitrile rubber, 20-40; blowing agent, 3-7; foam regulating agent, 1-20. As a foam regulator, products of processing alkylphenols with ethylene oxide can be used. Composition can comprise sulfur in the amount 0.2-0.5 mas. p. Invention provides preparing heat-stable, impact-strength foam materials not causing corrosion of nonferrous metals (copper, silver and their alloys) in direct contact and showing working capacity up to temperature 150°C. These materials can be used as heat-stable, vibration-proof materials in radiotechnical articles and articles having electric contacts made of nonferrous metals and alloys. 
     EFFECT: improved and valuable properties of composition. 
     3 cl, 2 tbl, 3 ex
Patent RU-2514672-C9 (RU)
Title: Рекомбинантная клетка, продуцирующая 2-гидроксиизомасляную кислоту
Inventor: RAJNEKE LIV
IPC: C12P7/42
Filed: 2009-04-28
Granted: 2014-10-20
Abstract: Изобретение относится к рекомбинантной клетке Ralstonia eutropha, предназначенной для получения 2-гидроксиизомасляной кислоты. Клетка трансформирована плазмидой с последовательностью SEQ ID NO:2. Клетка, несущая указанную плазмиду, продуцирует 2-гидроксиизомасляную кислоту в концентрации до 0,72 ммоль/кг. 4 ил., 4 пр.
Patent DK-6383-D0 (DK)
Inventor: MALBRANCQ JEAN-MICHEL
IPC: A61M1/34
Filed: 1983-01-10
Abstract: Apparatus/process for the withdrawal and return of liquid materials from a donor source, comprising means for withdrawing whole blood from a mammalian donor; a membranous blood filtration cell which includes a membrane separator/filter, a compartment downstream therefrom for receiving a blood plasma fraction and a compartment upstream thereof for receiving a blood cellular component fraction; conduit means for communicating the withdrawal means and an inlet end of the upstream compartment; a collection vessel; conduit means for communicating an outlet end of said upstream compartment and said collection vessel; means for determining the volume of liquid material withdrawn from the donor source during a withdrawal stage; means for back-filtering and returning liquid material from said collection vessel to the donor source; a second collection vessel; and conduit means for communicating an outlet end of the downstream compartment and the second collection vessel.
Patent DK-79985-D0 (DK)
Inventor: HOLDER ANTHONY ARTHUR
IPC: C12N15/30
Filed: 1985-02-21
Abstract: The present invention relates to the cloning of the P.195 gene of Plasmodium falciparum, its use in expressing the P.195 protein and the use of P.195 in vaccines for the treatment or prophylaxis of malaria.
Patent DK-90687-D0 (DK)
Inventor: WAUTIER HENRI
IPC: C01G25/02
Filed: 1987-02-23
Abstract: Process for the manufacture of vitreous metal oxides in which a metal alcoholate derived from an alcohol, the pka of which is less than 15.74, is hydrolysed with an aqueous medium, the pH of which is greater than 1.5. The process is applied especially to the manufacture of vitreous zirconium oxide.
Patent DK-134789-D0 (DK)
Inventor: CURTISS ALAN CLARKSON
IPC: A61K9/22
Filed: 1989-03-20
Abstract: A method for enhancing the unrolling of an active agent-containing matrix device, including a laminate device, in an aqueous use environment, said device being constrained in a rolled configuration prior to placement in said environment, comprising coating one side of the device with an elastomer prior to constraining it in a rolled configuration; and the devices so treated.
Patent DK-162887-D0 (DK)
Inventor: FREUND BERNHARD
IPC: A61J3/06
Filed: 1987-03-31
Abstract: The invention relates to a brick made of pellets with delayed and controlled release of the active ingredient in a meltable matrix consisting of a pharmacologically tolerated binder.
Patent DK-166986-D0 (DK)
Inventor: BOESTEN WILHELMUS HUBERTUS JOS
IPC: C12P41/00
Filed: 1986-04-11
Abstract: The invention relates to a process for racemizing an optically active N-benzylidene amino-acid amide, characterized in that a solution of the N-benzylidene amino-acid amide is mixed in a water-miscible organic solvent with at least 0.05 mole strong base per litre solution.The invention further relates to a process for preparing an L-amino acid by enzymatic separation of the corresponding DL-amino-acid amide with an enzyme preparation from Pseudomonas putida, in which process also unconverted D-amino-acid amide is left behind in solution, characterized in that benzaldehyde is added to the solution, during which addition a precipitate of D-N-benzylidene amino-acid amide is being formed, this precipitate is subsequently, after being separated off, dissolved in an acetone-water mixture, 0.08-0.15 mole KOH/litre solution is subsequently added, the resulting solution is stirred for 1-20 hours at 20-60 ¤C, sulphuric acid is then added until the pH of the solution is 5 and the resulting sulphuric acid salt of the DL-amino-acid amide is finally, after isolation at pH 8-10, converted into the DL-amino-acid amide and this DL-amino-acid amide is used again.
Patent DK-185087-D0 (DK)
Inventor: KOENIG WOLFGANG
IPC: C12Q1/34
Filed: 1987-04-10
Abstract: Chromophoric peptides of the formula
 DIS-D-Ala-Pro-R
 in which R is Gly-OH or NH2 and DIS is 5-dimethylamino-naphthalene-1-sulphonyl, their preparation, and their use for detecting peptidylglycine- alpha -amidating monooxygenase.
Patent DK-313389-D0 (DK)
Inventor: EBNER GUIDO
IPC: A01K29/00
Filed: 1989-06-23
Abstract: A novel method is described, which, on the basis of the short-term application of electrostatic fields, results in lasting beneficial and desirable properties in fish, which are otherwise achievable only with a substantial additional effort, if at all. As a result of the simplicity of the measures constituting the method according to the invention and the significant results, the culture of fish, particularly of edible fish but also of ornamental fish, is genuinely revolutionised. <IMAGE>
Patent DK-329187-D0 (DK)
Inventor: MUTERSPAUGH MAX WARD
IPC: H03D7/12
Filed: 1987-06-26
Abstract: A mixer for mixing first and second signals for providing a difference signal comprises a mixing transistor (200). The first and second signals are applied between the base and emitter electrodes of the transistor. A non-linear impedance (212) is coupled in series with the emitter electrode. Spurious signal components are reduced in amplitude compared with the difference signal.
Patent DK-363385-D0 (DK)
Inventor: BUDDE KLAUS
IPC: H05K3/46
Filed: 1985-08-09
Abstract: Linear fluorooligomers having at least two reactive end groups per polymer molecule are incorporated into radiation sensitive polymer systems which have improved continuous temperature resistance and low dielectric constant. The polymer systems can be applied as lacquers. Preferably perfluorated poly-ethers and perfluorated alkanes are used as starting compounds. The polymeric product is usable as a coating for the production of printed multi-layer wirings and economises on through-bores and additional copper intermeidate layers. A further field of application exists in the field of integrated semiconductor ciruits in VLSI-technology for the production of negative photo-resists.
Patent HU-901222-D0 (HU)
Title: Process for transmitting signals
Inventor: EDLER BERND
IPC: G10L19/022
Filed: 1990-01-26
Abstract: PCT No. PCT/EP90/00143 Sec. 371 Date Oct. 1, 1990 Sec. 102(e) Date Oct. 1, 1990 PCT Filed Jan. 26, 1990 PCT Pub. No. WO90/09063 PCT Pub. Date Aug. 9, 1990.Transmitting a signal wherein the signals is segmented by means of windows into successive overlapping blocks, the partial signals contained in the blocks are converted by transformation into a spectrum, with the spectra then being coded, transmitted, decoded after transmission and converted back into partial signals by retransformation. Finally, the blocks containing the partial signals are joined in an overlapping manner, with the overlapping regions of the blocks being weighted such that the resultant of the window functions in the respective overlapped regions equals one. To 2.2. In order to avoid interferences in adjacent blocks upon changes in the signal amplitude, the length of the window functions is selected as a function of signal amplitude changes. The method is suitable for the treatment of audio and video signals which are subjected to data reduction during transmission.
Patent HU-903008-D0 (HU)
Title: Improved process for the preparation of 3,5,6-trichloro-pyridin-2-ol
Inventor: R GARTH PEWS
IPC: B01J23/72
Filed: 1990-05-11
Abstract: A process for the preparation of 3,5,6-trichloropyridin-2-ol from trichloroacetyl chloride and acrylonitrile is improved by separately conducting the individual addition, cyclization and aromatization steps. By separating these steps, water and HCl, which are by-products of the latter steps, can be precluded from interfering with the earlier steps. The individual process steps have also been improved.
Patent NO-872507-D0 (NO)
Inventor: DREYER CHRISTIAN
IPC: F27B13/02
Filed: 1987-06-16
Abstract: The invention concerns an improvement in a suction or blowing pipe for a furnace having partition chambers intended for the firing of carbonaceous blocks. The pipe comprises a main body (3) provided with a plurality of nozzles (10) to which tubular nipples (2) are connected in a number equal to the number or partitions (5) forming the chambers of the furnace. Each of the nipples is connected to a transverse furnace wall (9) or a partition (5) by a taphole (8) disposed in the upper part of the wall or partition. The improvement comprises forming each nipple by at least two tubular elements disposed in series, a first element (15) provided in its upper part (15A) with a first flat flange (18) adapted to cooperate in jointed relationship and in respect of rotation with a flat flange (19) located in the lower part of a nozzle (10), and in its lower part (15C) with a second flat flange (27) which is parallel to the first flat flange (18), and a second element (16) provided in its upper part (16A) with a third flat flange (26) which cooperates in jointed relationship and in respect of rotation with the second flange (27). The first and second elements have over at least part of their height an axis inclined by an angle  alpha  with respect to the axis 23 which is perpendicular to the plane of the flanges.
Patent NO-894063-D0 (NO)
Inventor: FAIREY NORMAN REGINALD
IPC: B01J38/00
Filed: 1989-10-11
Abstract: A fabric knitted from a precious metal fibre, especially platinum or palladium or alloys thereof, offers advantages as a catalyst gauze, for example in ammonia oxidation. A method for knitting at high weights involves the co-feeding of a supplementary fibre with the metal fibre.
Patent NO-903297-D0 (NO)
Inventor: MERVAL JEAN-PAUL
IPC: C09D5/03
Filed: 1990-07-25
Abstract: Thermoplastic compositions in the form of powder based on polyamide and/or polyetheresteramide and containing epoxy/sulphonamide resins. The invention also relates to a number of processes for obtaining these powders and to their use for the coating of metal substrates not requiring any adhesion primer.
Patent NO-904666-D0 (NO)
Inventor: FRIARY RICHARD J
IPC: A61K31/42
Filed: 1990-10-26
Abstract: Fused polycyclic heterocyclic compounds of the generalized formula,   <CHEM> their use as PAF-antagonists, antihistamines and/or antiinflammatory agents, methods of manufacture and pharmaceutical compositions incorporating said compounds are disclosed.
Patent NO-911137-D0 (NO)
Inventor: SCHMID GERHARD
IPC: C12N15/12
Filed: 1991-03-21
Abstract: A process for obtaining hirudin derivatives from E. coli secretor mutants in which   (1) a recombinant vector on which the gene coding for a hirudin derivative is located directly behind a DNA section which codes for a bacterial signal peptide is constructed, (2) a E. coli secretor mutant is transformed with the recombinant vector constructed in step (1),   (3) the transformed cells are cultivated in a medium and   (4) the hirudin derivative is obtained from the medium, and a recombinant vector which contains one or more copies of a gene construct which codes for a protein consisting of a bacterial signal peptide and a hirudin derivative, and a hirudin derivative with the N-terminal amino-acid sequence A-Thr-Tyr-Thr-Asp in which A is Ala, Gln, His, Phe, Tyr, Glu, Ser, Asp or Asn are described.
Patent NO-912875-D0 (NO)
Inventor: MCCARTHY JAMES RAY
IPC: A61P3/06
Filed: 1991-07-23
Abstract: The present invention relates to a group of compounds which are novel substituted piperidines and which act to inhibit the synthesis of cholesterol in mammals and in fungi.
Patent NO-931181-D0 (NO)
Inventor: PIANI SILVANO
IPC: C08B37/10
Filed: 1993-03-30
Abstract: The synthesis of new semi-synthetic glycosaminoglycans is described in which one of the saccharide units characteristic of glycosaminoglycans with heparin or heparan structure, more specifically that of  alpha -L-iduronic-2-O-sulfate acid, has undergone a structural modification, entirely or in part, with transformation into  alpha -L-galacturonic acid substituted with nucleophilic radicals in position 3. These new semi-synthetic glycosaminoglycans of general formula IV <CHEM> have good pharmaceutical properties in that they may also be absorbed orally and have good anti-thrombotic activity accompanied by low risk of hemorrhage and reduced anti-coagulating activity.
Patent NO-933115-D0 (NO)
Inventor: OHNO KAZUNORI
IPC: C07D471/04
Filed: 1993-09-01
Abstract: A 3-Oxadiazolyl-5,6,7,8-tetrahydro-1,6-naphthyridine derivative of the formula (I): <CHEM> wherein Het is an oxadiazole ring, R1 is hydrogen atom, an acyl group, a lower alkyl group or a group of the formula: -CH2R1' (in which R1' is a cyclo-lower alkyl group, a lower alkenyl group, a lower alkynyl group, benzyl group, aryl group or a heteroaromatic group), R2 is a lower alkyl group, a cyclo-lower alkyl group, a lower alkenyl group, a lower alkynyl group, aryl group, a heteroaromatic group, a halogeno-lower alkyl group, a lower alkoxy-lower alkyl group, a lower alkoxy group, a lower alkenyloxy group, a phenoxy group or a lower alkylthio group, or a pharmaceutically acceptable acid addition salt thereof, is useful as benzodiazepine receptor agonist.
Patent NO-940911-D0 (NO)
Inventor: ASPEHAUG NILS
IPC: E04H12/22
Filed: 1994-03-14
Abstract: PCT No. PCT/NO95/00055 Sec. 371 Date Sep. 12, 1996 Sec. 102(e) Date Sep. 12, 1996 PCT Filed Mar. 13, 1995 PCT Pub. No. WO95/25213 PCT Pub. Date Sep. 21, 1995A foundation for masts, posts, pillars, etc., wherein the foundation has a foundation tube (3) which is lowered into a pre-drilled hole (2) in the ground (1), where the pre-drilled hole has a diameter larger than the diameter of the tube (3) and where at least the space between tube (3) and ground (1) is filled with a casting mixture (8), e.g. concrete, a tube (3) is used which is designed with perforations (4) in its lower area. The foundation tube (3) is equipped with a coating which gives the tube protection against corrosion, and possibly also an electrical insulation. The coatings can have a rough surface in order to create the best possible adhesion to the casting mixture. In order to ensure that the coated foundation tube (3) is safely lowered into the hole, it is first lined with a casing (13), which is removed during or immediately after the casting.
Patent NO-941678-D0 (NO)
Inventor: ENHSEN ALFONS
IPC: C07J9/00
Filed: 1994-05-06
Abstract: nor-Bile acid derivatives of the formula I  G1 - X - G2      I, in which G1, G2 and X have the stated meanings, processes for preparing these compounds and medicines are described. On the basis of their pharmacological action, they can be used as antihyperlipidaemic.
Patent NO-944401-D0 (NO)
Inventor: FODOR ANDREAS
IPC: E01B7/02
Filed: 1994-11-17
Abstract: Railway switch (points) with rigid rails (2) and pivotable switch blades (switch tongues) (4), at least one roller (1) with a shaft (11) being arranged in the pivoting region, the upper vertex (7) of which lies higher than the corresponding bearing surface (5), the roller (1), in the position of contact of the switch blade (4) on the rigid rail (2), bearing against the switch blade (4) below its upper vertex (7) and, outside this position, the switch blade (4) being able to be carried by rollers (1), and the roller (1) being resiliently mounted in the direction transversely to the track plane (8), the roller (1) being arranged to be adjustable both transversely and in the direction of the track plane (8), and its shaft (11) being oriented in the direction of the rigid rail (2), and the shaft ends (12) of the roller (1) being arranged to be height-adjustable in receptacles (21), and at least one receptacle (21) being holdable indirectly or directly in the direction of the rigid rail (2) via at least one distance piece (29). <IMAGE>
Patent NO-951055-D0 (NO)
Inventor: ANDRIEU VERONIQUE
IPC: A61P15/00
Filed: 1995-03-20
Abstract: A pharmaceutical prepn. form for targeted release of alfuzosine chlorohydrate is new. The prepn. form comprises a core contg. the active ingredient surrounded by a coating contg. a pH-dependently-soluble polymer.