baber/WOPTO huggingface dataset:
Patent BG-107817-A (BG)
Title: Benzodiazepine derivatives as gaba a receptor modulators
Inventor: MASCIADRI RAFFAELLO
IPC: A61P43/00
Filed: 2003-05-16
Abstract: The present invention relates to compounds of formula wherein R1 is hydrogen, halogen, lower alkyl, lower alkoxy, hydroxy, cyano, trifluoromethyl, trifluoromethoxy or lower alkylthio; R2 is -C(O)O-lower alkyl, isoxazol, 1,2,4-oxadiazol-3-yl or 1,2,3-oxadiazol-5-yl, which rings may be substituted by lower alkyl, trufluoromethyl or cycloalkyl; R3 is hydrogen, lower alkyl, -(CH2)n-cycloalkyl, -(CH2)n-halogen, -(CH2)n-pyridin-4-yl, or -(CH2)n-phenyl, wherein the phenyl ring may be substituted by one or two substituents selected from the group consisting of lower alkoxy, halogen, -SO2CH3, phenyl, OCF3, nitro, CF3, -NR2, or is -(CH2)n- indolyl, optionally substituted by lower alkyl or lower alkoxy, or is pyrrolidinyl-5-oxo, -C(O)-NR2, -(CH2)n-OH, -(CH2)n-NR2 or -(CH2)n-benzo[1,3]dioxole; R is hydrogen or lower alkyl; and n is 0,1, 2 or 3; and to their pharmaceutically acceptable acid addition salts, with the exception of the following compounds: ethyl 9H-imidazo[1,5-a][1,2,4] triazolo[3,4-d][1,4]benzodiazepin-10-carboxylate, 10-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-9H-imidazol[1,5-a] [1,2,4][1,2,4]triazolo[4,3-d][1,4]benzodiazepin, ethyl, 3 fluoro-9H-imidazo[1,5-a][1,2,4]triazolo[4,3-d][1,4]benzodiazepin-1 0-carboxylate; 10-(3-cylcopropyl-1,2,4-oxadiazol-5-yl)-3 fluoro-9H-imidazo[1,5-a]-triazolo]4,3,-d][1,4] benzodiazepin, ethyl-3-chloro-9H-imidazo[1,5-a][1,2,4]-triazolo[4,3-d][1,4]benzod iazepin-10-carboxylate, and 3-chloro-10-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-9H-imidazo[1.5-a] [1,2,4]-triazolo[4.3-d][1,4]-benzodiazepin. The benzodiazepin derivatives have a good affinity to the GABA A alpha5 receptor and they are therefore useful form the treatment of diseases, related to this receptor. 19 claims
Patent BG-110502-A (BG)
Title: A metod for local hardening of rail car wheel axles
Inventor: SOKOLOV VLADIMIR
IPC: C21D1/06
Filed: 2009-10-23
Abstract: The method is applied in transportation and metallurgy in hardening railcar wheel axles. The problem of railcar wheel axles life time improvement is solved. The method is to harden one of two of the wheels through conducting electric current by rotating contact rollers which are pressed to the surface treated. Heating and hardening of the surface is performed in one or several bands. The rotation speed of the wheel during heating is from 3,5 to 15 rphr.
Patent BG-111860-A (BG)
Title: Твърдо гориво на основата на битови и промишлени отпадъци, метод за неговото получаване и използване
Inventor: YORDANOV DOBROMIR
IPC: C10L5/00
Filed: 2014-11-19
Abstract: Изобретението се отнася до твърдо гориво на основата на битови и промишлени отпадъци, метод за неговото получаване и използване. Получен е продукт на основата на механично смесване между суровините (дървени стърготини, утайка от кафе от вендинг-автомат, изсушени при 20 градуса С в продължение на 24 h) и дозиране на отпаден глицерол от производството на биодизел. Показателите на продукта са следните: влага (обща) - 2,21 %; пепел - 5,53 %; сяра на сухо гориво - 0,14 %; топлина на изгаряне (долна на сухо гориво) - 19,84 MJ/kg; топлина на изгаряне (долна на работно гориво) - 19,35 MJ/kg. Топлината на изгаряне (долна на сухо гориво) на получения продукт е с 9-10 % по-висока от топлината на изгаряне на дървесните пелети на пазара. 3 претенции
Patent BG-112999-A (BG)
Title: Preparation method for ultrafine monodisperse nanoparticles with laser pulses
Inventor: NIKOLOV ATANAS
IPC: B22F9/06
Filed: 2019-09-24
Abstract: The invention relates to a preparation method for ultrafine monodisperse nanoparticles with laser pulses in a liquid medium applicable in medicine, biomedicine, photonics and the like. According to the method for preparing ultrafine monodisperse nanoparticles with laser pulses, a silver plate is placed on the bottom of a container and is covered with a layer of double distilled water. It is set to Nd: YAG laser energy below the ablation threshold and by means of a manual mode of computer-controlled X-Y mass the silver plate is positioned under the laser beam. The position of the silver plate is chosen so that in the process of ablation the laser beam remains only on its upper surface. The silver plate is screened by laser radiation. Upon changing the energy of the Nd: YAG laser to values above the ablation threshold, the screening is removed and at the same time the computer-controlled X-Y mass is turned on. The main length (lambda = 1064 nm) of the Nd: YAG laser is used for the ablation process. When the computer-controlled X-Y mass moves according to the set parameters, on the surface of the silver plate is constituted a contour representing the ablated area. From the separated material from the silver plate during ablation in the double distilled water, there are nanoparticles of silver formed as well as a colloid solution. In order to maintain the ablation rate for a certain period of time, the laser energy density increases step-like in the ablation process from 12.0 J / cm2 to 21.0 J / cm2, after which the ablation process is terminated. The resulting colloid solution is transferred to a glass cuvette and the rotating mass is set in motion to homogenize it. A laser beam with a wavelength of 355 nm and an energy density in the range of 0.059 to 0.068 J / cm2 is directed onto the surface of the colloid solution. After a certain time, the radiation of the colloidal solution is terminated. Part of the resulting colloida solution is transferred to a quartz cuvette and its optical transmission is measured.
Patent CN-1265844-A (CN)
Title: 一种复合蔬菜营养素及其制备工艺
Inventor: FANG YUAN
IPC: A23L19/00
Filed: 2000-03-16
Abstract: 本发明属食品技术领域,是一种复合蔬菜营养素及其制备工艺。该营养素由精选的8种蔬菜经特定工艺制备而成。其营养均衡、丰富,能满足人体健康对各种营养成分的需求,是一种绿色食品。本发明产品携带、食用方便,能使不同地区、不同季节的人们均能获得有效的各种蔬菜营养成分。
Patent CN-1354051-A (CN)
Title: 低装配应力铸轧辊
Inventor: ZHANG LIHUA
IPC: B21B27/03
Filed: 2000-11-20
Abstract: 一种铸轧辊,本发明在铸轧辊两端的辊芯、辊套装配面上安装轴向销,轴向销与辊芯、辊套的联结为过盈配合,销孔在安装时配铰钻。本发明采用低装配应力铸轧辊辊芯、辊套的组合结构,使得铸轧辊辊芯、辊套热装过程变得容易;铸轧辊辊芯、辊套的装配应力大幅降低,两者的使用寿命和铸轧板坯的表面质量得到明显提高,同时改善了板形。
Patent CN-1341417-A (CN)
Title: 含头孢噻肟和他唑巴坦的注射用药物组合物配方
Inventor: TONG MINGQING
IPC: A61P31/04
Filed: 2001-06-05
Abstract: 本发明涉及一种由头孢塞肟和他唑巴坦组成的注射用药物组合物配方,头孢噻肟和他唑巴坦的优选配比为1∶1－6∶1,头孢噻肟和他唑巴坦的最佳配比为2∶1－4∶1。本发明所述的他唑巴坦包括他唑巴坦钠盐、他唑巴坦半水合物。
Patent CN-1452153-A (CN)
Title: 乐器鼓
Inventor: BELLI REMOR D
IPC: G10D13/02
Filed: 2002-08-09
Abstract: 一种改进的鼓壳结构包括第一片材层，所述第一片材层具有弹性特性；第二片材层，与所述第一片材层以偶接的方式结合；粘接材料，连接所述的第一片材层和第二片材层；其中，所述第一片材层的弹性模量施加到所述第二片材层，以能够促使形成具有变化和改进的声音吸收及发射特性的鼓壳，从而控制及提高鼓面的音色。
Patent CN-1412533-A (CN)
Inventor: ZHANG QINYAO
IPC: G01J1/46
Filed: 2002-11-20
Abstract: 一种双色线列红外焦平面探测器读出电路结构，包含波段一输入级，波段二输入级，与该两输入级一起工作的移位寄存器和外引线键压点，其特点是它由两系列开关管、光敏元、栅控管、积分电容、复位开关和源极限随器相连构成，光敏元列阵与读出电路各输入端是通过铟柱互联而实现电连接的。本发明的电路结构紧凑，二个波段的光敏元列阵工作点，对应的积分电容可分别独立设置，二个波段的响应信号分别输出，以此结构制成的读出电路具有模块形式，可以实现多模块无缝拼接，形成双色长线列红外焦平面探测器。
Patent CN-1509081-A (CN)
Inventor: YONGQIN ZENG
IPC: H04N21/258
Filed: 2002-12-20
Abstract: 本发明提出了一种在保持现有SDTV传输不改变的同时，能显著节约带宽的传送SDTV/HDTV服务的方法和系统。根据本发明的一个实施例，可实现一个用于提供HDTV信号的系统。该系统获得一个包含HD增强数据流的增强层。并将该HD增强层传送到一个服务器。用户能通过一个机顶终端访问该服务器，以通过网络系统接收HD增强层。在本发明的另一个实施例中，一个包含SD数据流的基本层也被传送到机顶终端，使所述终端将HD增强层和基本层合并成为一个HDTV输出。
Patent CN-1492829-A (CN)
Inventor: TYNI TAPIO
IPC: B66B1/20
Filed: 2002-02-19
Abstract: 用于分配登梯呼叫的电梯组控制方法，在此方法中，一个目标值被分配到电梯组的给定服务时间，并且对电梯的分配登梯呼叫使得以平均值实现服务时间的分配目标值，从而降低了电梯组的能耗。
Patent CN-1514743-A (CN)
Inventor: SPRING D J
IPC: A62C2/04
Filed: 2002-04-02
Abstract: 从气源A来的空气，可能是飞机的排放气，在空气流量控制单元(10)控制下进入系统。有机燃料从燃料容器(12或13)在燃料流量控制单元(14)控制下进入混合室(16)与空气进行混合。在第一阶段，有机燃料是来自容器(12)的氧化有机燃料，在随后阶段中，有机燃料是来自容器(13)的烃类燃料。气体和燃料混合物进入包含贵金属催化剂如铂、钯或其混合物的催化剂床(18)。发生较低温度、非燃烧反应，所得的气体混合物包含低浓度的氧气和大量的惰性气体如氮气、二氧化碳和水蒸汽。这种反应后的混合物，在B点离开系统，适于抑制和熄灭火灾，尤其适于在飞行中当检测到火灾时，用于吹洗飞机货舱的空气。温度控制单元(20)与催化剂床(18)相关联，可用来防止其在反应中过热。控制单元(24)根据系统中各个点处传感单元(22)检测的各种参数如气体，压力，温度和流量的信号做出的响应，控制空气流量控制单元(10)、燃料流量控制单元(14)和温度控制单元(20)。
Patent CN-1518147-A (CN)
Inventor: AKIRA TANAKA
IPC: H01M8/00
Filed: 2003-04-02
Abstract: 提供一种即使阴极侧构件(5)是薄而刚性小的材料，也能将面压均匀地加在阴极(2)上，降低阴极侧构件(5)和阴极(2)之间的接触电阻，提高发电能力的燃料电池。在阴极侧构件(5)和阳极侧构件(6)之间有支撑材料(7)，通过用螺钉紧固靠近该支撑材料(7)的内侧，使阴极侧构件(5)发生弯曲力矩，通过使中央部附近朝向MEA4一侧挠曲，降低阴极侧构件(5)和阴极(2)的接触电阻，提高输出。
Patent CN-1521163-A (CN)
Inventor: XU DANQIAN
IPC: C07D211/00
Filed: 2003-01-27
Abstract: 本发明涉及一种室温离子液体的制备方法。其特征是采用目标产物即室温离子液体为反应介质，以烷基吡啶卤化铵或烷基咪唑卤化铵和含氟盐为原料，制备由烷基吡啶阳离子或烷基咪唑阳离子和含氟阴离子组成的室温离子液体。该方法操作简便，反应条件温和，产品质量好，并且反应过程环境友好，是一种绿色室温离子液体的制备方法。
Patent CN-1567374-A (CN)
Title: 藉由多张低解析度影像产生高解析度影像的方法
Inventor: GAO ZHAOYANG
IPC: G06T5/50
Filed: 2003-06-16
Abstract: 本发明提供一种具有改良的高解析度逻辑并重建高解析度影像的方法。本发明的方法基于反复修正法，并且应用预测的初期插补技术、健全的影像套合、自动化的影像选择，进一步可再施以影像品质提升的后处理。根据本发明的方法，可藉由关于静态景象的序列影像快速重建高解析度影像，亦可藉由关于动态物体的序列影像快速重建高解析度影像。
Patent CN-1537274-A (CN)
Inventor: ATSUSHI TOGAWA
IPC: G06F9/52
Filed: 2003-04-17
Abstract: 一种具有记录这样一种定时的机制的处理系统，在该定时具有高紧急度的处理被启动。如果该处理系统在具有低紧急度的处理期间进入临界区，就记录和检查是否在临界区的执行期间启动具有高紧急度的处理。如果具有高紧急度的处理不被启动，则该处理系统进入临界区，如果具有高紧急度的处理被启动，则该处理系统进行控制，以推迟进入临界区，直至具有高紧急度的处理结束。在执行多个任务的环境中，最好能够执行临界区中的专有存取控制。
Patent CN-1649995-A (CN)
Inventor: TSUYOSHI YANAI
IPC: C12M3/00
Filed: 2003-08-15
Abstract: 通过一种简单的结构可减少在各处理步骤中被尘粒、细菌等的污染。使用培养容器(1)，其中密封有培养基的培养基容器(3)和能够容纳主培养容器(2)中的流体的废培养基容器(4)通过连接管线(5)和(6)与主培养容器(2)在相对于外部密封的状态下相连接，所述连接管线能够限制所述容器之间的流体流动。培养设备被如此构成，其中各容器(2、3、4)的内部容积都是可变的，并且所述培养设备设有具有用于容纳各容器(2、3、4)的凹槽的壳体，以及通过施加外部压力使容纳在凹槽中的容器收缩的压制装置。
Patent CN-1826057-A (CN)
Inventor: HARALD MEYER
IPC: A23L27/30
Filed: 2003-08-28
Abstract: 本发明描述了一种水溶液，由于存在β－环糊精作为溶解度增加剂，该溶液中的阿司帕坦高度浓缩。
Patent CN-85108240-A (CN)
IPC: C12N1/20
Filed: 1985-11-16
Abstract: 通过培养对嘧啶类似物有抵抗力及在培养基中有产生胞苷和/或脱氧胞苷能力的，缺乏胞苷脱氨酶活力的芽孢杆菌属微生物，高得率地产生胞苷和脱氧胞苷。
Patent CN-86107845-A (CN)
Title: 耐磨、配副性好的合金铸铁汽缸套
IPC: C22C37/00
Filed: 1986-11-19
Abstract: 一种耐磨、配副性好的合金铸铁汽缸套。该铸铁化学成分为：碳3.1～3.8％，硅2.1～2.6％，锰0.7～1.3％，硼0.02～0.08％，磷0.15～0.50％，硫＜0.1％，铝0.3～1.0％，其余为铁。将该铸铁制成的发动机汽缸套经离子热处理，得到耐磨性、减磨性均佳的结构，使产品的耐磨性和配副性大幅度提高。
Patent CN-1119921-A (CN)
Title: 果实的种子取出装置
Inventor: SAITO MASAYUKI
IPC: A23N4/14
Filed: 1994-11-14
Abstract: 本发明涉及从果实中取出种子的装置。用下部保持部件5和上部保持部件6夹持果实，使切入用刃部16切入到果实内，其后，使压出用刃体10向上运动将心核从果实中往上推出。
Patent CN-1230212-A (CN)
Title: 包含烷基取代萘和酯的润滑油
Inventor: KRINKER R
IPC: C10M111/02
Filed: 1997-07-10
Abstract: 一种包含烷基取代萘和酯的润滑油。
Patent CN-1242776-A (CN)
Title: 用超滤、反渗透和纳滤纯化糖类
Inventor: DEFREES S
IPC: C13B30/08
Filed: 1997-10-09
Abstract: 本发明提供了用超滤、纳滤和/或反渗透来纯化包括寡糖、核苷酸糖和相关化合物在内的糖类的方法。在寡糖酶促合成或降解后,可从不需要的污染物(如存在于反应混合物中的化合物)中纯化获得糖类。
Patent CN-1244963-A (CN)
Title: 电子设备间的连接方法和连接电缆
Inventor: TAKASHI YAMAMOTO
IPC: H01R24/44
Filed: 1998-01-26
Abstract: 本发明是一种能传送良好的低频信号并能显著改善高频信号的干扰辐射电平的连接方法及连接电缆。电子设备1a、1b之间用连接电缆4连接时,用第1外部导体3a将连接电缆的信号线2从一端至另一端的区间加以屏蔽,并将第1外部导体3a的一端连接电子设备1a的基准电位,而且用第2外部导体3b屏蔽第1外部导体3a,并将第2外部导体3b连接电子设备1b的基准电位,通过第1外部导体3a与第2外部导体3b之间的杂散电容使一个电子设备的基准电位与另一电子设备的基准电位耦合,还根据针对抑制干扰辐射的频率,调整第2外部导体3b与第1外部导体3a的对置长度。
Patent CN-1288929-A (CN)
Title: 抗渗防水剂
Inventor: QIN HONGYOU
IPC: C09K3/18
Filed: 1999-09-20
Abstract: 一种无机新型高强刚性防渗防水材料,其特点是1.5—3mm薄层即具有优良的防渗防水功能,与新旧建筑物砖石及砼结合牢固,不老化,使用简单,不污染环境,属绿色建材。根据需要,还可生产出更高强度的防渗防水材料。
Patent CN-1305393-A (CN)
Title: 回收化学和机械平整化所用水与浆料研磨剂的方法和设备
Inventor: CORLETT GARY L
IPC: B24B37/04
Filed: 1999-05-25
Abstract: 一种从含有粉碎的、悬浮固体的含水浆料中回收液体和研磨剂的方法,该法包含至少一个过滤步骤,该步骤用烧结金属膜和/或陶瓷膜并和测量比重或密度方法相连结、物理地浓缩和使研磨剂颗粒从可通过标准工业废物系统处置的液流中分离或回用上清液流的方法。该方法还用于回收固体以回用于其它的、严格性差些的用途中,由此减少或消除抛光工艺的无用的副产物。
Patent CR-20120633-A (CR)
Title: Procedimiento de para producir clinker para cemento hidràulico con baja emisiòn de c02 y alta resistencia
Inventor: RAMIREZ TOVIAS HOMERO
IPC: C04B7/02
Filed: 2012-12-12
Abstract: La presente invención se refiere al procedimiento de fabricación de un clinquer para cemento caracterizado porque este se obtiene mediante la trituración de una harina en bruto que comprende, en particular, A1203, Fe203 y SO3.
Patent CR-20120664-A (CR)
Title: Método para proteger arroz contra la infección por hongos
Inventor: STIERL REINHARD
IPC: A01N43/653
Filed: 2012-12-21
Abstract: Método para proteger arroz contra la infección porhongos nocivos, en donde se tratan los hongos, su hábitat, las plantas de arroz, sus semillas, el material de propagación vegetaldel arroz o el suelo donde el arroz está creciendo o va a crecer, conepoxiconazol y triciclazolen cantidades sinergéticamente efectivas; el uso de una composición, que comprende epoxiconazol, triciclazol y opcionalmenteun fungicida adicional disponible en el comercio, para proteger arroz contra la infección porhongos nocivos.
Patent CR-20130646-A (CR)
Title: Compuestos de pirrolidinil urea y pirrolidinil tiourea como inhibidores de cinasa trka
Inventor: ALLEN SHELLEY
IPC: A61K31/4155
Filed: 2013-12-11
Abstract: Compuestos de Fórmula I: o estereoisómeros, tautómeros o, sales o solvatos o profármacos farmacéuticamente aceptables de los mismos, donde R1, R2, Ra, Rb, Rc, Rd, X, Y, B y el Anillo C son tal como se definen en la presente, y donde el resto Y-B y el resto NH-C(=X)-NH están en la configuración trans, son inhibidores de cinasa TrkA y son útiles en el tratamiento de enfermedades que se pueden tratar con un inhibidor de cinasa TrkA tal como dolor, cáncer, inflamación, enfermedades neurodegenerativas y determinadas enfermedades infecciosas.
Patent CR-20170315-A (CR)
Title: Inhibridores bace 1 selectivos
Inventor: HEMBRE ERIK JAMES;
IPC: C07D513/04
Filed: 2016-02-17
Abstract: La presente invención proporciona un compuesto de Fórmula II: o una sal aceptable para uso farmacéutico.
Patent CR-20190179-A (CR)
Title: Anti-il-33 antibodies and uses thereof
Inventor: BENSCHOP ROBERT JAN
IPC: C07K16/24
Filed: 2017-10-24
Abstract: Antibodies which bind and neutralize human IL-33, and methods of using same, are provided, said antibodies are useful as agents for treating conditions associated with allergic disease including treating atopic dermatitis.La presente invención proporciona anticuerpos los cuales se unen y neutralizan IL-33 humano, y métodos para usar los mismos, tales anticuerpos son útiles como agentes para el tratamiento de condiciones asociadas con enfermedad alérgica que incluye tratar dermatitis atópica
Patent EC-SP045468-A (EC)
Title: Nuevas proteínas de fusión con trombomodulina dirigidas contra factores tisulares como anticoagulantes
IPC: C07K14/485
Filed: 2004-11-30
Abstract: Nuevas proteínas de fusión compuestas de una proteína direccionadora que se une al factor tisular (TF), ligadas operativamente al dominio EGF456 de la trombomodulina (TM) ya sea sola o en combinación con al menos un dominio adicional de TM seleccionado del grupo formado por el dominio hidrofóbico de la región N-terminal, el dominio EGF123, el bucle de interdominio entre EGF3 y EGF4 y el dominio rico en Ser/Thr O-glicosilado, o análogos de los mismos. La proteína de fusión se une en el sitio de una lesión e impide el inicio de una trombosis. La proteína de fusión se puede usar en el tratamiento de diversas condiciones trombóticas, incluyendo, por ejemplo, la trombosis venosa profunda, la coagulación intravascular diseminada y el síndrome coronario agudo.
Patent EC-SP099802-A (EC)
Title: SALES DEL INHIBIDOR DE JANUS CINASA (R)-3-(4-(7H-PIRROLO[2,3-d]PIRIMIDIN-4-IL)-1H-PIRAZOL-1-IL)-3- CICLOPENTILPROPANITRILO
Inventor: LI HUI YIN
IPC: A61K31/519
Filed: 2009-12-14
Abstract: La presente invención proporciona formas de sal de (R)-3-(4-(7H-pirrolo[2,3-d]pirimidin-4-il)-1H-pirazol-1-il)-3-ciclopentilpropanitrilo que son útiles en la modulación de la actividad de la cinasa Janus que incluye, por ejemplo, enfermedades relacionadas con el sistema inmunitario, trastornos de la piel, trastornos proliferativos mieloides, cáncer, y otras enfermedades.
Patent EC-SP961873-A (EC)
Title: Compuestos ciclicos inhibidores de la adhesion
Inventor: GOODMAN SIMON
IPC: A61K31/19
Filed: 1996-09-12
Abstract: La invención se refiere a nuevos ciclopéptidos de fórmula ciclo -(nArg-nGly - nAsp - nD- nE), en la que D y E independientemente representan Gly, Ala, Bala, Asn, Asp, Asp, (OR), Arg, Cha, Cys, Gln, Glu, His, Lle, Leu, Lys, Lys(Ac), Lys(AcNh2), Lys(AcSH), Met, Nal, Nle, Orn, Phe, 4-Hal, Phe, homo -Phe, Phg, Pro, Pya, Ser, Thr, Tia, Tic, Trp, Tyr, ó Val, pudiendo tratarse de derivados de estos amino ácidos; R representa alquilo de 1 a 18 tomos de C; Hal, F, Cl, Br ó L; Ac, alcanoilo de 1 a 10 tomos de C, aroilo de 7 a 11 tomos de C o arilalcanoilo de 8 a 12 tomos de C, y n significa que no hay sustituyentes o bien representa un resto de alquilo R, bencilo o un resto de arilalquilo de 7 a 18 tomos de C, unidos a la función alfa -amino del resto de amino ácido en cuestión; con la condición de que al menos uno de los restos de amino ácido presenta un sustituyente n, estndo incluidas tanto las formas D como las formas L en caso de uqe los amino ácidos y restos de amino ácidos tengan actividad óptica, y las sales inobjetables desde el punto de vista fisiológico de estos compuestos. Estos compuestos actúan como inhibidores de las integrinas y se pueden emplear en partcular para prevenir y tratar enfermedades del sistema circulatorio, enfermedades angiogénicas infecciones microbianas y para el tratamiento de tumores.
Patent EC-SP993070-A (EC)
Title: Ligandos de alta afinidad para el receptor de nociceptina orl 1
Inventor: HEY JOHN A
IPC: A61K31/43
Filed: 1999-07-26
Abstract: Nuevos compuestos de fórmula (gráfico), o una sal o solvato de los mismos, farmacéuticamente aceptable en los cuales: la linea de puntos representa un doble enlace opcional; X1 es H, alquilo, cicloalquilo, arilo, heteroarilo, heterocicloalquilo o heterociclilo benzofusionado opcionalmente sustituidos; X2 es H, -CH=, -CN, amino, alquilo o arilo opcionalmente sustituido; o X1 o X2 conjuntamente forman un grupo espiro heterociclilo opcionalmente benzofusionado. R1, R2, R3 y R4 son independientemente H o alquilo, o (R1 y R4) o (R2 y R3) o (R1 y R3) o (R2 y R4) conjuntamente pueden formar un puente alquileno de 1 a 3 átomos de carbono; Z1 es alquilo, arilo, heteroarilo, cicloalquilo o heterocicloalquilo opcionalmente sustituido o -CO2(alquilo o amino substituido) o CN, Z2 es H o Z1; Z3 es H o alquilo; o Z1, Z2 y Z3 conjuntamente con el carbon al cual están unidos forman anillos biciclicos saturados o insaturados; composiciones farmacéuticas que incluyen los mismos y el uso de dichos compuestos como inhibidores, receptores de nociceptina útiles para el tratamiento, ansiedad, tos, asma, depresión y abuso de alcohol.
Patent FI-20002441-A (FI)
Inventor: VAEAENAENEN MIKKO KALERVO
IPC: H04M1/72436
Filed: 2000-11-08
Abstract: The invention relates to an electronic short messaging and advertising method and means. In particular the invention relates to an electronic advertising method, where minimal initiative is required from the consumer. Some embodiments of the invention may also be applied to an electronic sales method. The invention may be applied for normal short messaging also. The electronic short messaging and advertising method comprises at least one subscriber terminal and uses the Internet and/or the telephony network. With the method in accordance with the invention the recipient can receive advertisements or other short messages with the shortest manipulation time possible. No navigation, browsing of inboxes, copying and/or pasting of telephone numbers needs to be done. The user is shown the message automatically, and he may delete it or receive further information on it with one single press of a dedicated key.
Patent FI-20030553-A (FI)
Inventor: UITTO VESA
IPC: E21B47/01
Filed: 2003-04-11
Abstract: The invention relates to a drill hole measuring device and a rock drilling unit equipped with the measuring device. The measuring device (1) comprises a protective element (3), inside which a sensor (6) can be transferred by means of a transfer device (4).
Patent FI-20030818-A (FI)
Title: Wireless agent application provision method for ad-hoc type short distance connection, selects and collects information and sends it to telephone over same transmission path over which requested visiting card is received
Inventor: HUHTINIEMI PASI
IPC: H04W12/06
Filed: 2003-05-30
Abstract: An application distribution unit identifies the address of an intelligent telephone on the basis of wireless connection, and determines the type of information based on the contents of a visiting card. The distribution unit selects and collects the information and sends it to the telephone over the same transmission path over which the requested visiting card is received. An independent claim is also included for software product for providing wireless agent application for ad-hoc type short distance connections.
Patent FI-20105579-A (FI)
Inventor: KUITTINEN JARNO
IPC: B60W50/14
Filed: 2010-05-25
Abstract: The invention relates to a rock drilling rig, a method for transfer drive of the rock drilling rig, and a speed controller. The rock drilling rig includes combustion-engine-free drive equipment which includes a plurality of electric components for implementation of the transfer drive. The control unit of the rock drilling rig includes load monitoring which monitors the load of the components during the transfer drive. Load monitoring allows the electric driving system to be intentionally overloaded for a period of time limited in advance. A user interface of the control unit comprises a speed controller whose control element has a first control range, where operation takes place in the rated load range, and a second control range, where operation takes place in the overload range.
Patent FI-20125629-A (FI)
Inventor: ANTILA JARKKO
IPC: G01J3/26
Filed: 2012-06-08
Abstract: The invention relates to controllable Fabry-Perot interferometers which are produced with micromechanical (MEMS) technology. The prior art interferometers have a temperature drift which causes inaccuracy and requirement for complicated packaging. According to the invention the interferometer arrangement has both an electrically tuneable interferometer and a reference interferometer on the same substrate. The temperature drift is measured with the reference interferometer and this information is used for compensating the measurement with the tuneable interferometer. The measurement accuracy and stability can thus be improved and requirements for packaging are lighter.
Patent FI-20205468-A (FI)
Title: A mounting tool
Inventor: VARTIAINEN JUSSI
IPC: E04G21/18
Filed: 2020-05-08
Abstract: The mounting tool comprises a body (10) having a general shape of a letter L with a first leg (20) and a second leg (30). The length (L1) of the first leg determines a desired spacing between two adjacent longitudinal objects to be attached to a base construction. The second leg comprising at least one first cylindrical passage (41, 42, 43, 44) passing in an inclined manner through the second leg. The first cylindrical passage guides a fastening means (50) in the angle of inclination from a side edge of the object through the longitudinal object and into the base construction in order to attach the longitudinal object to the base construction.