baber/WOPTO huggingface dataset:
Patent CO-6220950-A2 (CO)
Title: Compuestos heterociclicos compuestos que los comprenden y metodos para su uso
Inventor: AUGERI DAVID J
IPC: A61K31/422
Filed: 2009-09-30
Abstract: 1.- Un compuesto de la fórmula I:o su sal o solvato farmacéuticamente aceptable, en donde:A es un heterociclo opcionalmente sustituido; R1 es OR1A, OC(O)R1A, C(O)OR1A, hidrógeno, halógeno, nitrilo, o alquilo opcionalmente sustituido, arilo, alquilarilo, arilalquilo, heteroalquilo, heterociclo, alquilheterociclo, o heterocicloalquilo; R2 es OR2A, OC(O)R2A, hidrógeno, halógeno, o alquilo opcionalmente sustituido, arilo, alquilarilo, arilalquilo, heteroalquilo, heterociclo, alquilheterociclo, o heterocicloalquilo; R3 es N(R3A)2, hidrógeno, hidroxi, o alquilo opcionalmente sustituido, arilo, alquilarilo, arilalquilo, heteroalquilo, heterociclo, alquilheterociclo, o heterocicloalquilo; y cada uno de R1A, R2A, y R3A es independientemente hidrógeno o alquilo opcionalmente sustituido, arilo, alquilarilo, arilalquilo, heteroalquilo, heterociclo, alquilheterociclo, o heterocicloalquilo. 2.- Un compuesto de la fórmula I(a):o su sal o solvato farmacéuticamente aceptable, en donde: A es un heterociclo opcionalmente sustituido;R1 es OR1A, OC(O)R1A, C(O)OR1A, hidrógeno, halógeno, nitrilo, o alquilo opcionalmente sustituido, arilo, alquilarilo, arilalquilo, heteroalquilo, heterociclo, alquilheterociclo, o heterocicloalquilo; R5 es OR5A, OC(O)R5A, N(R5B)2, NHC(O)R5B, hidrógeno, o halógeno; R6 es OR6A, OC(O)R6A, N(R6B)2, NHC(O)R6B, hidrógeno, o halógeno; R7 es OR7A, OC(O)R7A, N(R7B)2, NHC(O)R7B, hidrógeno, o halógeno; R8 es CH2OR8A, CH2OC(O)R8A, N(R8B)2, NHC(O)R8B, hidrógeno, o halógeno;cada uno de R1A, R5A, R6A, R7A, y R8A es independientemente hidrógeno o alquilo opcionalmente sustituido, arilo, alquilarilo, arilalquilo, heteroalquilo, heterociclo, alquilheterociclo, o heterocicloalquilo; y cada uno de R5B, R6B, R7B y R8B es independientemente hidrógeno o alquilo opcionalmente sustituido con uno o más grupos hidroxi o halógeno.
Patent CO-6270235-A2 (CO)
Title: Un peptido de proiselt seleccionado de un grupo acetilo n-terminal, amida y cisteine
Inventor: LEVETAN CLARESA S
IPC: A61K38/22
Filed: 2010-04-05
Abstract: Las realizaciones se refieren a péptidos Prolslet, preferentemente, HIP, que exhiben una estabilidad y eficacia aumentadas, y a los métodos para utilizarlos para tratar una patologia asociada con la funcion pancreatica alterada, incluyendo diabetes tipo 1 y 2 y sus sintomas. 1.- Un péptido Prolslet caracterizado porque comprende una modificacion de optimizacion, donde dicha modificacion de optimizacion se selecciona del grupo formado por un grupo acetilo N-terminal, un grupo amida C-terminal, y un residuo de cisteina C-terminal. 2.- El péptido de la reivindicacion 1, caracterizado porque dicha modificacion de optimizacion se selecciona del grupo formado por (i) un grupo acetilo N-terminal y un grupo amida C-terminal y, (ii) un grupo acetilo N-terminal y un residuo de cisteina C-terminal. 3.- El péptido de la reivindicacion 1, caracterizado porque dicho péptido es un péptido HIP1 modificado, un péptido HIP2 modificado, o un péptido HIP3 modificado. 4.- El péptido de la reivindicacion 1, caracterizado porque dicho péptido es un péptido humano REG3A modificado, un péptido humano REG3G modificado, un péptido humano REG1A modificado, un péptido humano REG1B modificado, un péptido humano REG4 modificado, un péptido INGAP en hamster, un péptido REG2 en hamster modificado, un péptido REG3G en hamster modificado, un péptido REG1 en rata modificado, un péptido PAP/REG3B en rata modificado, un péptido PAP3 en rata modificado, un péptido REG3G en rata modificado, péptido REG 1 en raton modificado, péptido REG2 en raton modificado, péptido REG3A en raton modificado, péptido REG3B en raton modificado, péptido REG3G en raton modificado, péptido REG3S en raton modificado, péptido REG4 en raton modificado, péptido bovino PTP modificado.
Patent CO-6300864-A2 (CO)
Title: Derivados polisustituidos de 6-heteroaril-imidazo[1,2-a]piridinas su preparacion y su aplicacion en terapeutica
Inventor: DE PERETTI DANIELLE
IPC: A61K31/437
Filed: 2010-09-20
Abstract: 1.- Compuestos de fórmula (I): en la que:R1 representa:un grupo fenilo o naftilo, un grupo heteroarilo o un grupo heterocíclico, pudiendo estar estos grupos sustituidos opcionalmente con uno o varios átomos o grupos elegidos independientemente los unos de los otros entre los átomos o grupos siguientes : halógeno, alquilo(C1-C10), haloalquilo(C1-C10), alcoxi(C1-C10), haloalcoxi(C1-C10), tioalquilo(C1-C10), -S(O)(alquilo-C1-C10), -S(O)2-alquilo(C1-C10), hidroxilo, oxo, ciano, nitro, hidroxi-alquileno(C1-C10), NRaRb-alquileno(C1-C10), alcoxi(C1-C10)-alquileno(C1-C10)-oxi, NRaRb, CONRaRb, SO2NRaAb, NRcCORd, OC(O)NRaRb, OCOalquilo(C1-C10), NRcC(O)ORe,NRcSO2Re, arilalquileno(C1-C10), arilo o heteroarilo monocíclico, estando el arilo o el heteroarilo monocíclico sustituido opcionalmente con uno o varios sustituyentes elegidos entre un halógeno, un grupo alquilo(C1-C10), haloalquilo(C1-C10), alcoxi(C1-C10), haloalcoxi(C1-C10), NRaRb, hidroxilo, oxo, nitro, ciano o OCOalquilo(C1-C10) y R1 está unido a la imidazo [1,2-a]piridina por un carbono aromático; Het representa un grupo heteroarilo monocíclico que contiene de 5 a 6 átomos entre ellos 1 a 3 heteroátomos elegidos entre N,O y S;X representa de 1 a 3 sustituyentes idénticos o diferentes el uno del otro, elegidos entre un hidrógeno, un halógeno, alquilo(C1-C10), alcoxi(C1-C10), NRaRb, nitro, ciano, pudiendo estar el alquilo(C1-C10) sustituido opcionalmente con uno o varios grupos elegidos entre un halógeno, alcoxi(C1-C10), haloalcoxi(C1-C10), NRaRb o hidroxilo;R representa en posición 3, 5, 7 u 8 de la imidazo[1,2- a]piridina de 1 a 4 sustituyentes idénticos o diferentes el uno del otro, elegidos entre un hidrógeno, un halógeno, alquilo(C1-C10), haloalquilo(C1-C10), alcoxi(C1-C10); ...
Patent CO-6341583-A2 (CO)
Title: Catalizador para la descomposición de lignina, método para la preparación de alcoholes y ácidos orgánicos, método para la preparación de productos de la descomposición de lignina, catalizador para la descomposición de hidrocarburos aromáticos, método
Inventor: ISHIBASHI TORU
IPC: B01J31/02
Filed: 2011-02-16
Abstract: 1.- Un catalizador para la descomposición de lignina que comprende una porfirina que puede mostrar su función catalítica a través de la irradiación de la misma con rayos de luz.2.- Un catalizador para la descomposición de lignina que comprende una porfirina que puede mostrar su función catalítica en una solución alcalina.3.- Un catalizador para la descomposición de lignina que comprende una porfirina que puede mostrar su función catalítica en una solución alcalina, mientras se irradia la misma con rayos de luz.4.- El catalizador para la descomposición de lignina como se establece en una cualquiera de las reivindicaciones 1 a 3, en donde la porfirina es un compuesto de tetrapirrol que lleva un grupo metilo y un grupo éster etílico o un grupo acetato (grupo ácido propiónico) sobre el anillo de porfirina.5.- El catalizador para la descomposición de lignina como se establece en una cualquiera de las reivindicaciones 1 a 3, en donde la porfirina es un compuesto de tetrapirrol que lleva cuatro grupos metilo y cuatro grupos éster etílico o grupos acetato (grupos ácido propiónico) sobre el anillo de porfirina.
Patent CO-6470827-A2 (CO)
Title: Mejora en la precisión de llenado durante la formación de una bolsa
Inventor: WEAGANT SIMON
IPC: B65B3/36
Filed: 2011-11-25
Abstract: En uno de sus aspectos, la presente invención se relaciona con un proceso para formar una bolsa flexible para empaque de líquidos. Este proceso mejora la precisión del llenado del material fluido contenido en la bolsa. Específicamente, la invención se relaciona con un proceso para mejorar la precisión de llenado de una bolsa mediante incorporar al menos un tubo vertical en un tanque de alimentación que alimenta la bolsa con material fluido que debe ser empacado. Esta invención se relaciona también con aquel aparato diseñado para mejorar la precisión en el llenado de la bolsa flexible para empacar líquidos.
Patent CO-6612256-A2 (CO)
Title: Sistema estructural por paneles para construcción de edificaciones
Inventor: VANKER JOHN LOUSI
IPC: E04B1/18
Filed: 2012-07-18
Abstract: En un aspecto, una sección de una edificación incluye columnas estructurales directamente conectadas y alineadas verticalmente. Un primera panel de cerchas estructurales se une a la primer columna estructural y un segundo panel de cerchas estructurales se une a la segundo columna estructural de tal manera que los paneles de cerchas estructurales transfieren cargas verticales vivas y muertas y cargas laterales sobre los primeros y segundos paneles de cerchas estructurales lateralmente a las primeras y segundas columnas estructurales y luego verticalmente a través de las primeras y segundas columnas estructurales.En otro aspecto, un panel integrado de cercha estructural se configura para transferir lateralmente carga vertical viva y muerta y carga lateral a una columna estructural de una edificación. El panel integrado de cercha estructural incluye una pluralidad de miembros horizontales alargados, y una pluralidad de miembros verticales alargados acoplados en forma funcional a los miembros horizontales alargados.En otro aspecto, un panel estructural para una edificación incluye miembros horizontales alargados y miembros verticales alargados acoplados en forma funcional a los miembros alargados horizontales.En otro aspecto, un método para la construcción de una edificación incluye fijar un primer panel de cercha estructural a una primera columna estructural y una segunda columna estructural verticalmente directamente a la primera columna estructural. Un segundo panel de cercha estructural se fija a la segunda columna estructural, de manera que el segundo panel cercha estructural está verticalmente por encima del primer panel de cercha estructural, de manera que la carga vertical viva y muerta y la carga lateral sean transferidas lateralmente a las primeras y segundas columnas estructurales y luego verticalmente entre las primeras y segundas columnas.
Patent EP-1031473-A2 (EP)
Inventor: JANSSEN ROBERT
IPC: B60R21/235
Filed: 2000-01-07
Abstract: The airbag consists of a material containing a large synthetic fiber component. The fibers are of a heat-fixable synthetic. The folded airbag is compressed by application of an outside force, heated by heat radiation, and heat-set while compressed. The folded airbag is positioned in a chamber with moveable wall, and the chamber is subsequently evacuated.  The appliance to carry out the procedure has a plate (10) to support the folded airbag (15), a gas-proof covering film (16), units for sealed connection of film edge to plate, an underpressure source (12) connected to the space thus defined, and a heater (14).
Patent EP-1023856-A2 (EP)
Inventor: WIEGNER GEORG
IPC: A46B15/00
Filed: 2000-01-21
Abstract: The container (1) has a compartment (2) into which a brush (6) is dipped and has an opening (3) in which sits a tapering stopper (4). The brush on a handle (7) is inserted through a hole. The handle with its end facing the brush is fixed to a container-head placed onto the opening for retaining the brush in the compartment filled with a hygienic mouth-refreshing agent. One brush is in the form of a inter-dental brush . The container forms a tooth-brush (10) handle whose end facing away from the tooth-brush head (12) is in the form of a container-top (9).
Patent EP-1030097-A2 (EP)
Inventor: SEIFERT RAINER
IPC: B29C45/16
Filed: 2000-02-02
Abstract: A method is provided for rotationally attaching a connection fitting with an opposing surface by screwing the fitting into the opposing surface by threads on an outer surface of the fitting body. The connection fitting is formed by at least one seal manufactured together with the fitting body in an injection molding process to form a multi-component plastic part in which the fitting body is made of a hard plastic component and the seal is made of a soft plastic component, wherein the components are of a kind which do not adhere to one another. The seal is secured in an axial direction on the fitting body in a form-fit manner, but during the rotational attachment step the seal is rotatable relative to the fitting body in a peripheral direction.
Patent EP-1028086-A2 (EP)
Inventor: ABONNET JAQUES
IPC: B66F9/075
Filed: 2000-02-09
Abstract: The carrier vehicle which travels over the floor, such as a forklift truck or an order picker, has two drive wheels (6,7) with steering, and a steering system used by the operative. Each drive wheel (6,7) has a drive motor. The wheels (6,7) are linked to the steering shaft (10) so that, on moving round a curve, the inner wheel on the curve is given a stronger steering movement than the other wheel, and the wheel on the inside of the curve is rotated at a slower speed than the outer wheel, according to the position of the steering unit.
Patent EP-1036919-A2 (EP)
Inventor: SCHMIDT WERNER
IPC: F01N13/02
Filed: 2000-02-28
Abstract: The engine has a regulating device with a gas line (3) for connecting to at least one combustion chamber exhaust valve. The gas line contains a setting member (9) to alter the through flow cross section of the gas line. The position of the setting member is continuously adjusted by an electronic control apparatus (13).
Patent EP-1033756-A2 (EP)
Inventor: ONOSE HIDEKATSU
IPC: H01L29/80
Filed: 2000-03-01
Abstract: In a semiconductor device such as a pn-junction diode, a Schottky diode, a JFET, a MOSFET or a MESFET, a drift layer is made of two layers, a first layer (12) and a second layer (13) having the same conductivity type as that of the first layer (12) and being disposed on said first layer (12), a termination region being formed on the surface of said second layer (13). The impurity concentration of the second layer (13) is less than half that of the first layer (12). The thickness of the second layer may moreover be made smaller than that of a main layer (14) of the device. In accordance with the above features, the field intensity is reduced at the termination region of the device. <IMAGE>
Patent EP-1045008-A2 (EP)
Inventor: PEDEMONTE RONALD DR
IPC: C09B62/503
Filed: 2000-04-06
Abstract: The present invention provides a dye mixture comprising one or more
copper complex formazan dyes conforming to the formula (1)
 
and one or more copper complex formazan dyes conforming to the
formula (2)
 
wherein R1, R2, Y1, Y2 and M are defined as given in claim 1, methods
for preparing said dye mixtures and methods for dyeing and printing
hydroxy- and/or carboxamido-containing materials using said dye
mixtures.
Patent EP-1079494-A2 (EP)
Inventor: KINOSHITA NAOKI
IPC: B60L50/16
Filed: 2000-08-25
Abstract: The present invention relates a battery control apparatus (9) controls charge/discharge
processes of a battery (8) installed in a hybrid vehicle, according to the battery temperature so as
to prevent degradation of the battery performance. The vehicle has a combustion engine (1) for
providing a driving force, an electric motor (2) for generating a drive assist force for assisting
the output of the engine, wherein the battery supplies electrical power to the motor, and, when
the drive-assist force is not required by the engine, the motor is used as a generator to charged
the battery, the apparatus is comprised by: a residual battery charge computation device (91) for
computing a level of residual battery charge in the battery; a battery temperature measuring
device for measuring a temperature of the battery; and a charge/discharge controller (92) that
operates in such a way that, when a battery temperature measured by the battery temperature
measuring device exceeds a threshold temperature, the charge/discharge controller permits only
discharging until the residual battery charge is lowered to a level defined by a first specified
value.
Patent EP-1086803-A2 (EP)
Inventor: WARBURTON-PITT STEPHEN
IPC: B31B19/84
Filed: 2000-08-29
Abstract: The combination of a bag (10) and tubes (24,26) connected thereto
for use in pharmaceutical manufacturing and for holding
health care related solutions is formed entirely of
silicone. This avoids the previous problem of the
releasing into the held fluids of plasticizers or plastic
additives contained in the PVC material making up prior
bags.
Patent EP-1070777-A2 (EP)
Inventor: ROELL FRIEDRICH
IPC: D04B1/22
Filed: 1997-04-18
Abstract: To join knitted sections together, at a flatbed knitter, the first section is knitted, with the stitches at the junction edge left hanging on the needles. At least one further section is knitted, and the needles with the hung stitches of the first section are reactivated at the join between the two sections. Preferably at least the section is a knitted tube, where initially one side is knitted, and the final row is joined with the first row of a multi-layer knit on at least two needle beds, and then separated for knitting again on two needle beds, and finally knitted together. The first section is knitted on the first needle bed, with the edges of the junction row left hanging on the needles.
Patent EP-1088984-A2 (EP)
Inventor: HUMMEL HELMUT
IPC: F02M55/00
Filed: 2000-09-29
Abstract: The system includes a pump (1) for supplying fuel. Downstream of the pump is a fuel line (7) for supplying at least part of the fuel supplied by the pump to at least one injector (10.1-10.4). A filter element (21) removes gas from the injection system. The filter element is impermeable to fuel and permeable to gas. A venting line branches from the fuel line downstream of the pump, and the filter is arranged in it.
Patent EP-1096128-A2 (EP)
Inventor: KITANI HIROYUKI
IPC: F02G5/02
Filed: 2000-10-27
Abstract: An exhaust gas released from the exhaust gas heat
exchanger (9) is conveyed into the inlet of a bend (32)
communicated to a silencer (31). The exhaust gas mixed with
the condensed water is upwardly passed as a mixture fluid
through a passage (322) and forced into a first expansion
chamber (323). The mixture fluid is separated into the
exhaust gas and the condensed water in the chamber (323)
and conveyed downwardly in a passage (324) provided with
a second expansion chamber (325). While the exhaust gas
is forced upwardly from the lower end of the silencer (31),
the condensed water is discharged downwardly. The
condensed water is conveyed in the drain passage of a waster
water trap and released to the outside.
Patent EP-1109403-A2 (EP)
Inventor: TSUNODA HIROSHI
IPC: G11B20/10
Filed: 2000-12-12
Abstract: A data recording apparatus includes a slot for receiving a memory card having a
disk, a flash memory and a controller. Each time one frame of compressed image data is
recorded to the disk, a vacant capacity value of the disk is written to the flash memory.
This vacant capacity value is read out according to an instruction given from a CPU.
When the vacant capacity of the disk is lower than the vacant capacity of a compressed
image area formed in an SDRAM, the CPU invalidates the vacant capacity of the
compressed image area in a portion exceeding the vacant capacity of the disk. This
restricts the number of frames to be picture-taken.
Patent EP-1108983-A2 (EP)
Inventor: NAGAKI KOICHI
IPC: G08G1/0969
Filed: 2000-12-14
Abstract: A navigation system is provided with: a present position
detecting device (16, 17) for detecting a present position; a first
memory device (14) for reading map data from a record medium (1)
in which the map data is recorded; a second memory device (15) of
non-volatile type, to which the map data can be written and from
which the map data can be read; a navigation controlling device (11)
for controlling a navigation operation in correspondence with the
detected present position by using the map data, and sending a
transfer command to transfer the map data from the first memory
device to the second memory device at a predetermined timing; and
a transfer interface (30) for controlling an operation of reading the
map data from the record medium by the first memory device and an
operation of transferring the map data to the second memory device,
in accordance with the sent transfer command.
Patent EP-1023881-A2 (EP)
Inventor: O'NEIL MICHAEL J
IPC: A61F2/38
Filed: 2000-01-27
Abstract: A modular joint prosthesis includes a tibial component formed of a tibial bearing
insert and a tibial plateau. The tibial bearing insert is a modular component formed of a
tibial insert body and a modular element. The tibial insert body and the modular elements
are provided in a variety of geometries and sizes to yield various types of tibial insert
bodies. The same tibial insert body may be used, for example, to form both rotatable and
non-rotatable tibial bearing inserts.
Patent EP-1030079-A2 (EP)
Inventor: NAKAMURA KENSUKE
IPC: F16H7/08
Filed: 2000-02-07
Abstract: A blade-type tensioner for chain drives which is suitable for use as
a tensioner on the timing chain of a motor vehicle engine. The present invention is
a chain tensioner particularly suited for use in confined spaces having a blade
spring element mechanically interlocked with a plastic shoe. The shoe may be of
rigid filled nylon and engages the chain to be tensioned. The spring element is
interlocked to the plastic shoe by having ends inserted into grooves formed in the
opposite ends of the shoe. The shoe is rotatably fixed to a base by way of a pin.
The groove at the fixed end of the shoe extends towards the tip of the fixed end of
the shoe past the pin attachment point. The groove at the free end of the shoe
extends toward the tip of the free end of the shoe past the point at which the free
end of the shoe bears upon a sliding surface formed on the base.
Patent EP-1056304-A2 (EP)
Inventor: ESWARA SRINIVAS
IPC: H04W16/28
Filed: 2000-05-25
Abstract: Disclosed is an apparatus for reducing the number of control signal channels required
in a wireless communication system by using a umbrella control signal to initially
communicate with an MS (mobile station) within the umbrella and to assign the MS to
a traffic frequency corresponding to one of a plurality of antenna used to cover the
area covered by said umbrella control signal. Logic is used in combination with
measured relative signal strengths to determine the position of the MS relative to the
reliable reception coverage area of each of the plurality of antennas before the
assignment is made.
Patent EP-1065863-A2 (EP)
Inventor: BARNETT RICKY
IPC: H04M1/02
Filed: 2000-06-16
Abstract: A portable radiotelephone device comprising a body having provided on one
or more exposed surface thereof one or more electrical contact means for one
or more respective electrical input/output means, wherein said one or more
electrical contact means is covered with one or more layers of electro-resistive
material, said electro-resistive material in the relaxed condition being an
electrical insulator and in the stressed state being an electrical conductor, the
arrangement being such that to effect electrical connection between any of the
one or more electrical contact means with respective one or more electrical
input/output means, respective contact means and input/output means are
mutually engaged so as to load the elasto-resistive material under
compression.
Patent EP-1094646-A2 (EP)
Inventor: CLARK TERENCE JOHN
IPC: H04L45/243
Filed: 2000-10-12
Abstract: A communication method and system for communicating between a terminal
and service provider, in which multiple communication channels are provided between
the terminal and the communication apparatus which use a multi link protocol
communication. A single communication channel is provided between the
communication apparatus and the service provider for communicating using a single
link protocol. Within the communication apparatus, communications received from the
terminal in the multi link protocol are converted to a single link protocol for
communication to the service provider. Also communications received from the service
provider in the single protocol are converted to the multi link protocol for
communication to the terminal.