baber/WOPTO huggingface dataset:
Patent IL-136734-A (IL)
Title: Alpha-aminoamide derivatives useful as analgesic agents
IPC: A61K31/165
Filed: 2000-06-13
Abstract: The present invention relates to novel and known alpha-aminoamide compounds, to a process for their preparation, to pharmaceutical composition containing them and to their use as therapeutic agents. In particular, the compounds of the present invention are endowed with analgesic properties and are particularly useful for the treatment and alleviation of chronic and neuropathic pain. Accordingly, one object of the present invention is to provide the use of a compound of formula (I) wherein: A is a -(CH<SUB>2</SUB>)<SUB>m</SUB>-, -(CH<SUB>2</SUB>)<SUB>n</SUB>-X- or -(CH<SUB>2</SUB>)<SUB>v</SUB>-O- group wherein m is an integer of 1 to 4, n is zero or an integer of 1 to 4, X is -S- or -NH-, and v is zero or an integer of 1 to 5; s is 1 or 2; R is a furyl, thienyl, or pyridyl ring or a phenyl ring optionally substituted by one or two substituents independently chosen from halogen, cyano, C<SUB>1</SUB>-C<SUB>4 </SUB>alkyl, C<SUB>1</SUB>-C<SUB>4 </SUB>alkoxy and trifluoromethyl; R<SUB>1 </SUB>is hydrogen or C<SUB>1</SUB>-C<SUB>4 </SUB>alkyl; one of R<SUB>2 </SUB>and R<SUB>3 </SUB>is hydrogen and the other is hydrogen or C<SUB>1</SUB>-C<SUB>4 </SUB>alkyl optionally substituted by hydroxy or phenyl; or R<SUB>2 </SUB>and R<SUB>3 </SUB>taken together with the carbon atom to which they are linked form a C<SUB>3</SUB>-C<SUB>6 </SUB>cycloalkyl ring; or R<SUB>2 </SUB>and R<SUB>3 </SUB>are both methyl; R<SUB>4 </SUB>is hydrogen or C<SUB>1</SUB>-C<SUB>4 </SUB>alkyl.
Patent IL-138978-A (IL)
Title: Drive mechanism for aiming a shell launching device
IPC: F41A27/28
Filed: 2000-10-12
Abstract: The laying mechanism (10) for a fragmentation round launch tube (12) has a rapid setting for azimuth in the foundation (15), with at least two azimuth setting motors (14) acting on the carrier ring (18), parallel to the azimuth axis. At least one setting motor can be reversed into a drive in the opposite direction, to block the movement from the other motor when the carrier ring (18) has reached the azimuth setting for the launch. The static setting motors are contained within the pot-shaped foundation, with one motor (13) for elevation and a motor (14) for azimuth.
Patent IL-144641-A (IL)
Title: Phenylalaninol derivatives, pharmaceutical preparations thereof, processes for their preparation, and uses of phenylalaninol derivatives in the preparation of medicaments
IPC: C07C/
Filed: 2001-07-30
Abstract: New Phenylalaninol derivatives (I). Phenylalaninol derivatives of formula (I) are new: [Image] X : a benzamide group of formula (i), a heterocyclyl-amide group of formula (ii) or an imidazolin-3-yl-4-one group of formula (iii): [Image] R 15halo, NO 2, CN, lower alkylsulfonyl, lower alkyl, lower alkoxy, lower alkoxycarbonyl, carboxy, lower alkylaminosulfonyl, lower perfluoroalkyl, lower alkylthio, lower hydroxyalkyl, alkoxy-lower alkyl, alkylthio-lower alkyl, alkylsulfinyl-lower alkyl, alkylsulfonyl-lower alkyl, lower alkylsulfinyl, lower alkanoyl, aroyl, aryl or aryloxy; R 16H, halo, NO 2, CN, lower alkyl, OH lower perfluoroalkyl or lower alkylthio; Het : 5-6 membered heteroaryl containing 1-2 N, O or S; or 9-10 membered bicyclic heteroaryl containing 1-4 O, S or N; R 30H or lower alkyl; p : 0-1; R 18aryl or heteroaryl; R 19optionally substituted lower alkyl, aryl, heteroaryl, aralkyl or heteroaralkyl; R 20lower alkanoyl or aroyl; Y : a group of formula (iv) or (v) or a 5-6 membered heteroaryl, bonded via C and containing 1-3 O, N or S and optionally substituted by 1-2 lower alkyl, cycloalkyl, halo, CN, perfluoroalkyl or aryl, provided that at least one of the substituents is adjacent to the bonding C; [Image] a : an optional double bond; R 22, R 23H, lower alkyl, lower alkoxy, lower cycloalkyl, aryl aralkyl, NO 2, CN, lower alkylthio, lower alkylsulfinyl, lower alkylsulfonyl, lower alkanoyl, halo or perfluoro lower alkyl; provided that at least one is not H; R 24H, lower alkyl, lower alkoxy, aryl, NO 2, CN, lower alkylsulfony or halo; R 25lower alkyl, lower alkenyl (optionally fluorinated) or R 26(CH 2) e; R 26aryl, heteroaryl, N 3, CN, OH, lower alkoxy. lower alkoxycarbonyl, lower alkanoyl, lower alkylthio, lower alkylsulfonyl, lower alkylsulfinyl, perfluoro-lower alkanoyl, NO 2 or NR 28R 29; R 28H or lower alkyl; R 29H, lower alkyl, lower alkoxycarbonyl, lower alkanoyl, aroyl, perfluoro lower alkanoylamino, lower alkylsulfonyl, lower alkylaminocarbonyl or arylaminocarbonyl; or R 28 + R 294-6 membered carbocyclic ring optionally containing 1 O, N or S and optionally substituted on C by lower alkyl or halo; Q : (CH 2) fO, (CH 2) fS, (CH 2) fN(R 27), (CH 2) f or a bond; R 27H, lower alkyl, aryl, lower alkanoyl, aroyl or lower alkoxycarbonyl; e : 0-4; and f : 1-3. An independent claim is included for preparation of (I). ACTIVITY : Antirheumatic; antiarthritic; antiasthmatic; antiinflammatory; neuroprotective. MECHANISM OF ACTION : (I) inhibit the binding of vascular cell adhesion molecule-1 (VCAM1) and fibronectin to the integrin VLA-4 (not defined) on circulating lymphocytes, eosinophils, basophils and monocytes.
Patent IL-146919-A (IL)
Title: Retarding and locking device for missile projectile
Inventor: BISEROD HANS B
IPC: F15B15/19
Filed: 2001-12-04
Abstract: A retarding and locking mechanism for use between two mutually translatable bodies. A first body can be induced into motion and guided into a second body and, after a predetermined movement of the first body, the first body is subject to retardation and interlocked to the second body, such that the first and second bodies together form a unitary, integrated body. The first body has a radially outwardly directed shoulder and the second body has a radially inwardly directed shoulder corresponding to the radially outwardly directed shoulder of the first body. A compressible element is provided between the shoulders of the first and second bodies.
Patent IL-157439-A (IL)
Title: Method and apparatus for is-95b reverse link supplemental code channel frame validation and fundamental code channel rate decision improvement
IPC: H04B7/26
Filed: 2003-08-17
Abstract: The present invention provides a method and apparatus for maximizing throughput of a data call in a wireless communication system in which data is transmitted from a wireless station, such as a mobile station, on multiple assigned channels in accordance with a known transmission standard, such as IS-95B. The multiple assigned channels include a fundamental channel and at least one supplemental channel. Data is formatted into variable rate data frames and transmitted on the fundamental channel and the supplemental channel. A wireless receiver, such as a base station, receives the multiple assigned channels. The wireless receiver demodulates and decodes data frames associated with each of the multiple assigned channels. The wireless receiver determines a likely initial data rate for each demodulated and decode data frame. The wireless receiver correlates all of the likely data rates, by comparison to one another and to a relevant transmission protocol standard, to determine a maximum likelihood combination of data rates. The maximum likelihood combination of data rates includes a maximum likelihood data rate corresponding to each likely data rate. Decoded data frames are invalidated and erased when the likely data frame rates do not match corresponding maximum likelihood data rates.
Patent IL-170501-A (IL)
Title: Fusible conductive ink for use in manufacturing microfluidic analytical systems
Filed: 2005-08-25
Abstract: A fusible conductive ink for use in manufacturing microfluidic analytical systems includes micronised powder containing platinum and carbon, poly(bisphenol A-co-epichlorohydrin)-glycidyl end capped polymer, and a solvent. In addition, the ratio of micronised powder to poly(bisphenol A-co-epichlorohydrin)-glycidyl end capped polymer is in the range of 3:1 to 1:3. The fusible conductive inks can be employed in the manufacturing of microfluidic systems to form electrodes, electrically conductive traces and/or electrically conductive contact pads.
Patent IL-171546-A (IL)
Title: Oxazolidinone-quinoline derivatives and pharmaceutical compositions comprising them
IPC: A61P/
Filed: 2005-10-23
Abstract: The present invention relates to the use of compounds, in which the pharmacophores of quinolone and oxazolidinone are chemically linked together through a linker that is stable under physiological conditions, for the treatment of anthrax and other infections.
Patent IL-175195-A (IL)
Title: Thermal cushion and device comprising such a cushion
IPC: A61F7/02
Filed: 2006-04-25
Abstract: The cushion has a network of blocks formed of hollow cells (1). The cells are formed by assembling two sheets that are embossed and welded with one another along splines (6). The splines are flexible and elastic, and serve as joint between the cells. Interstices (8) delimited between the cells and the splines are filled with a deformable thermal material. A flexible and elastic envelope (7) surrounds the cells and interstices.
Patent IL-189183-A (IL)
Title: Indole derivatives, processes for their preparation, pharmaceutical compositions comprising them and their use in the manufacture of medicaments for treating diseases
IPC: A61K/
Filed: 2008-02-03
Abstract: Indole derivatives (I), are new. Indole derivatives of formula (I) and their salts are new. R a, R bH, halo, 1-6C alkyl, CF 3, CN, COR 2, OR 2 or phenyl (optionally substituted by 1-4C alkyl or CF 3); R 21-4C alkyl, CF 3 or phenyl (optionally substituted by 1-4C alkyl or CF 3); R 2H or 1-4C alkyl; R : H or 1-3C alkyl; n : 1-3; X : a bond or O, and Ar 1phenyl, naphthyl, quinolinyl, isoquinolinyl, pyridinyl, pyrazolyl, imidazolyl, isoxazolyl, thiazolyl, benzothiazolyl, 2,1,3-benzothiadiazolyl, 3,4-dihydro-1,4-benzoxazinyl, 5,6,7,8-tetrahydronaphthlaneyl, 1,2,3,4-tetrahydroquinolinyl, 1,2,3,4-tetrahydroisoquinolinyl, 1,2,3,4-tetrahydro-2-oxoquinolinyl, 3,4-dihydro-2H-benzopyranyl, indolyl, 2,3-dihydroindolyl, 2,3-dihydrobenzofuranyl, 1,3-benzodioxolyl, 1,4-benzodioxanyl or benzoxazolyl (all optionally substituted by halo, 1-6C alkyl, CF 3, CN, CO-R 2, OR 2, NH-COR 2, morpholinyl, amino or 4-morpholinosulfonyl). Independent claims are included for the preparation of (I). [Image] ACTIVITY : Antilipemic; Antidiabetic; Cardiovascular-Gen.; Antiinflammatory; Neuroprotective; Nootropic; Antiparkinsonian; Anorectic; Antiarteriosclerotic; Cardiant; Hypotensive; Antiarthritic; Antirheumatic. MECHANISM OF ACTION : Peroxisome proliferator activated receptor (PPAR) activator. In a test used to determine activation of PPAR-alpha and/or PPAR-gamma , results showed that (I) exhibited an EC 50 value of 50 nM.
Patent JP-H10293274-A (JP)
Title: Spectacles
Inventor: ONODA TETSUHISA
IPC: G02C5/00
Filed: 1997-04-17
Abstract: PROBLEM TO BE SOLVED: To provide spectacles having few secular decrease of strength while sufficiently ensuring the fixing strength even by the engagement for directly fixing a supporting member to a lens. SOLUTION: This spectacles is provided with a lens 2 and a supporting member S for supporting the lens, an engaging protrusion engaged with the lens either in the direction from the side of the lens 2 to the middle part or in the direction of lens thickness is provided and a catching member 4, engaged with the lens in the direction intersecting the engaging direction of the engaging protrusion, is engaged with the engaging protrusion. Consequently, the supporting member is fixed to the lens.
Patent JP-H09289406-A (JP)
Title: Dielectric resonator
Inventor: IIDA MUNEO
IPC: H01P7/04
Filed: 1996-04-22
Abstract: PROBLEM TO BE SOLVED: To relax conditions between resonance frequencies f1 and f2 which can be switched by the use of a variable-frequency dielectric resonator. SOLUTION: The dielectric resonator, which has an external conductor layer 204 covering the surface of a columnar dielectric except both its end surfaces and an internal conductor layer 203 covering the internal wall surface of a hole penetrating the said dielectric center part as electrodes and uses one end surface of the said dielectric as an input terminal and the other as a reflection terminal 206, is provided with a conductor layer 207 which is electrically connected to the external conductor layer 204 nearby the reflection terminal 205 in the said dielectric, and the external conductor layer 204 and internal conductor layer 203 are connected through a switch nearby the reflection terminal.
Patent JP-S5526482-A (JP)
Title: Digital display type electronic watch
Inventor: KITA KAZUNORI
IPC: G04G9/00
Filed: 1978-08-17
Abstract: PURPOSE: To make it possible to display always a desired time in an optimum display mode by performing a prescribed switching for a main time and another time.  
     CONSTITUTION: Means 3 and 4 to obtain main time information and another time information, means 9 to display digitally obtained time information, and switching set means 14 to set the display mode of means 9 to the 12 or 24 hours system by information are provided, and time-counted main time information and another time information time-counted, operated or stored can be displayed independently in the 12 hours system time dispaly and the 24 hours system time display, so that four display modes can be selected. 
     COPYRIGHT: (C)1980,JPO&Japio
Patent JP-H075023-A (JP)
Title: Packaged material weighing control method
Inventor: KAWAGUCHI MASASHI
IPC: G01G13/08
Filed: 1993-04-02
Abstract: PURPOSE:To eliminate the need for inputting data from keyboard into a microcomputer when operating an electronic weighing machine. CONSTITUTION:Each bag is marked with its volume with bar codes. When a scanner 31 reads a bar code marked on a new bag 10, a CPU 30 extracts information corresponding to the bar code information from a memory 32 by collating the bar code information with information on a memory 32, and inputs the extracted information into a controller 19, which sets its internal weight memory so that the memory agrees with the above bar code information. Thus, the weight of a material to be filled in a bag 10 automatically agrees with the bar code information.
Patent JP-H041502-A (JP)
Title: Residual quantity detector for conductive thin wire reel
Inventor: SORIOKA MIKIYUKI
IPC: G01B7/12
Filed: 1990-04-18
Abstract: PURPOSE:To automatically and accurately detect the residual quantity of the conductive thin wire on a reel by making a couple of conductive rollers abut on the conductive thin wire, and detecting a conductive or nonconductive state and detecting the residual quantity. CONSTITUTION:At the winding end part of the steel cord reel 2, and when conductive rollers 10 and 11 roll are turned on the steel cord 1, and the steel cord is left enough on the reel 2, a current flows to the cord 1, but is intermitted since the rolls rollers 10 and 11 are bounced. Then when the cord 1 is further unwound until one roller 10 leaves the cord 1, the roller 10 comes into contact with insulating paper P, so no current flows and a lamp 20 goes out. Consequently, the timing where one of the couple of rollers 10 and 11 leaves the cord 1 can accurately be detected and the residual quantity of the final winding string of the cord 1 remaining on the reel 2 can automatically and accurately be detected from the winding diameter of the reel 2 and the wire diameter of the cord 1.
Patent JP-S5626742-A (JP)
Title: Manufacture of cullet for glass fiber
Inventor: TSUNODA TAKEHIRO
IPC: C03C1/02
Filed: 1979-08-08
Abstract: PURPOSE:To ecomonically manufacture cullet to be blended into starting material for manufacturing glass fiber by cutting washed and dehydrated glass filament scraps and pulverizing the cut scraps. CONSTITUTION:Glass fiber scraps discharged from a glass fiber manufacturing process are washed to remove greige goods, stuck dust, etc., and they are allowed to stand for about 30min to be dehydrated to about 10-20wt% residual water content. The scraps are then cut to <= about 20cm length and pulverized with an impact type pulverizer such as a hammer mill to obtain glass cullet of about 10- 20mesh. The amount of water used by this method is <= about 4ton per ton of glass fiber scraps, and no glass fiber fine powder is mixed into waste water and discharged.
Patent JP-S59225786-A (JP)
Inventor: NAKAJIMA YOSHIHIRO
IPC: B07C5/36
Filed: 1983-06-06
Abstract: (57)【要約】本公報は電子出願前の出願データであるた め要約のデータは記録されません。
Patent JP-H07278528-A (JP)
Title: Polishing/abrasive material for surface cleaning
Inventor: KATSUMATA SATOSHI
IPC: B24D3/28
Filed: 1994-04-14
Abstract: PURPOSE:To obtain a polishing/abrasive material for surface cleaning consisting of a mixture of a polycyanoaryl-based resin having a recurring unit of a specific structure as a component with a polyamide-based resin, free from breakage of a material to be polished due to electron charge and excellent in polishing/ abrasive ability. CONSTITUTION:This polishing/abrasive material is composed of a mixture of (A) a polycyanoaryl ether ketone having a recurring unit of formula I as a component, preferably a polycyanoaryl ether consisting essentially of a recurring unit of formula II (Ar is aryl) or a polycyanoaryl ether ketone consisting essentially of a recurring unit of formula II and a recurring unit of formula III with (B) a polyamide-based resin (preferably nylon 6, nylon 66 or nylon 46 having 6000-60000 average molecular weight). Furthermore, the polishing/ abrasive material is preferably mixed in a ratio of 1-100 pts.wt. of the component A to 100 pts.wt. of the component B.
Patent JP-H04333630-A (JP)
Title: String material and underwater construction
Inventor: TOMITA RIKIO
IPC: D06M101/16
Filed: 1991-05-02
Abstract: PURPOSE:To provide a string material having low rigidity in netknitting process and increased rigidity after knitting a net and enabling the incorporation of an antifouling material and to provide an underwater construction having light- weight and excellent antifouling effect and capable of keeping the shape of the net. CONSTITUTION:The objective string material is composed of a core and a sheath covering the circumference of the core, wherein the core is made of a material containing a thermosetting resin and a thermoplastic resin and the sheath is made of a material containing a thermoplastic resin. The underwater construction is constructed of the string material produced by covering a core made of a material containing a thermosetting resin and a thermoplastic resin with a sheath made of a material containing a thermoplastic resin.
Patent JP-S585538-A (JP)
Title: Pitch feed device
Inventor: SHIROGANE KIYOSHI
IPC: H01H21/48
Filed: 1981-06-30
Abstract: PURPOSE:To reduce a pitch feed device to compact size and to easily adjust the pitch feed by making the center of rotation of a feed click consistent with that of a rachet and by pitch-feeding in both directions. CONSTITUTION:When a driving lever 20 is pushed down, an interlocking member 19 turns on a pivot 14 clockwise, and a feed click body 22 is moved to the left by an interlocking pin 21 to be engaged with an inward tooth 15a, thereby to apply pitch feed to a rotor 15. When the driving lever 20 is pushed up, the rotor 15 is fed by pitch in the opposite direction by a click portion 22b of the feed click body 22. The pitch feed is adjusted according to the frequency of changes of the driving lever 20.
Patent JP-H07276382-A (JP)
Title: Mold for molded piece with cylindrical core
Inventor: FUKADA MASAHIRO
IPC: B29C39/22
Filed: 1994-04-13
Abstract: PURPOSE:To obtain a mold for suppressing occurrence of a flash on the end face of a cylindrical core to substantially zero at the time of molding a molded piece with a cylindrical core. CONSTITUTION:Pins 17, 27 are erected respectively on a movable mold 16 and a stationary mold 26 to be concentrically opposed to each other. On end of a hole of a cylindrical core 2 is previously inserted and set over the pin 17. The pin 27 is fitted into the other end of the hole as the mold is closed. With the progress of the mold closing, the peripheral ends of the cylindrical core 2 are engaged and fitted with top parts 18a, 28a of bushes 18, 28. Lastly, the cylindrical core 2 is fastened by fastening ends 17a, 27a provided on the pins 17, 27. A predetermined material is injected into a cavity 3a formed around the cylindrical core 2 to be molded into a molded piece. The cylindrical core 2 is released from a fitted state by a spring 29 and an ejector rod as the mold is opened.
Patent JP-S58217543-A (JP)
Title: Fluorocarbon resin-containing coating composition
Inventor: FUJIYAMA HARUHISA
IPC: C08L27/12
Filed: 1982-06-11
Abstract: PURPOSE:To provide a baking fluorocarbon resin-contg. compsn. which is hard, does not soften when heated and has corrosion resistance, mold release characteristics, and slip properties in combination, by dispersing a fluorocarbon resin powder and low-melting glass powder in a dispersion medium. CONSTITUTION:A fluorocarbon resin such as poly(tetrafluoroethylene) and a low- melting glass such as lead borate glass are pulverized and dispersed in a dispersion medium contg. additives such as surfactant, ethylene glycol, etc. As the dispersion medium, water is generally used. 5-120pts.wt. fluorocarbon resin per 100pts.wt. low-melting glass is used. The resulting coating compsn. is applied by a conventional method, predried and baked by heating at a temp. at which the low-melting glass is molten, for example, at 370-400 deg.C to obtain the desired coating film.
Patent JP-H02278640-A (JP)
Title: Electron gun device
Inventor: WAKAMOTO IKUO
IPC: H01J29/48
Filed: 1989-04-20
Abstract: PURPOSE:To obtain an electron beam having a uniform strength in a rectangular range by forming the plant of each grid to have an angle of less than 90deg. to the vertical shaft of a filament. CONSTITUTION:The plane of each grid 5 is formed to have an angle of less than 90deg. to the vertical shaft of a filament 1, and an anode 7 is formed to protrude to the grid 5. The sectional form and beam current value of an electron beam obtained by an electron gun are set by the form of the grid 5 and the anode 7, distance between the grid 5 and a cathode 3, distance between the grid 5 and the anode 7, acceleration voltage, grid voltage, etc., and the strength of the electron beam between the facing grids 5 is almost even. An electron beam having a uniform strength in a rectangular range can thus be obtained.
Patent JP-S62260551-A (JP)
Title: Three-phase ac motor unit
Inventor: YAGI TAKAO
IPC: H02K17/12
Filed: 1986-05-02
Abstract: PURPOSE:To enable stable operation to be performed without generating torque ripple on a motor, by a method wherein a dividing section is set on a ring- formed stator core in the diameter direction, and wherein a three-phase winding is set with a single-layer winding so that the dividing section cannot be crossed, and wherein a magnetic unit ring having a loss section on the leading wire of the winding with the phase of little impendance is set. CONSTITUTION:When AC current I is permitted to flow to a leading wire 3, then magnetic flux phi is generated in an iron-ingot-formed ring 4, and ampere turn AT is generated when the space of a loss section 5 is set to be D. When the area of the loss section is set to be A and a reactance is set to be Le, then Le=D/A is shown. In this case, the same effect as that when a reactor is inserted in the leading wire of a stator winding is generated. On the equivalent circuit of reactances 9a, 9b generated on a motor 6 with arranged stator windings and a terminal 7a..., the terminal 8a of a device..., and the iron-ingot- formed ring, impedance from the viewpoint of the terminals is unbalanced, but impedance from the viewpoint of the terminal of the device can be balanced with the size of the ring 4 and the dimension of the loss section. Accordingly, torque ripple is not generated and operation can be performed.