baber/WOPTO huggingface dataset:
Patent AU-783141-B2 (AU)
Title: Phenanthryl piperazinyl dicarboxylic acids as selective NMDA receptor modulating agents
Inventor: MONAGHAN DANIEL T
IPC: G01N33/94
Filed: 2000-12-18
Granted: 2005-09-29
Abstract: Disclosed are compounds of formula (I) wherein : L is (a) optionally substituted by replacement of one or more of the hydrogen atoms on the phenanthrene ring system by one or more groups other than hydrogen; A is CH2, SO2 or C=O; X is CO2H, PO3H2, PO2H2, PO2HR<5>, PO2HOR<5>, SO3H, SO2H, or tetrazole; and R<1>, R<2>, R<3>, R<4> and R<5> are independently selected from H, alkyl, alkenyl, alkynyl, aryl and aralkyl; or a pharmaceutically acceptable acid salt or base addition salt or an <i>in vivo</i> hydrolysable ester or amide thereof. Compounds of formula (I) are selective NMDA receptor modulating agents and, therefore, may be used to advantage <i>in vitro</i> in neuroassays and <i>in vivo</i> in the treatment of disorders of the CNS.
Patent AU-566748-B2 (AU)
Title: Aqueous coating compositions
Inventor: BROMLEY CHARLES WILLIAM ALFRED
IPC: C09D5/00
Filed: 1983-12-30
Granted: 1987-10-29
Abstract: Aqueous compositions suitable for forming on a substrate a temporary protective coating, which can subsequently be removed by treatment with an aqueous alkaline solution, comprise a sterically stabilised dispersion in an aqueous medium of particles of size range 0.1-10 µm of a polymer derived from monomers including at least one acrylic monomer and from 5% to 40%, based on the total weight of monomers, of an ethylenically unsaturated monocarboxylic acid, or an equivalent proportion of an unsaturated polycarboxylic acid.
Patent AU-658441-B2 (AU)
Title: Substituted beta-lactam compounds useful as hypocholesterolemic agents and processes for the preparation thereof
Inventor: BURNETT DUANE A
IPC: C07F7/18
Filed: 1992-07-21
Granted: 1995-04-13
Abstract: Novel compounds of the formula <CHEM>  wherein A is -CH=CH-B; -C IDENTICAL C-B; -(CH2)p-X-B, wherein p is 0-2 and X is a bond, -NH- or-S(O)0-2; optionally substituted heteroaryl or benzofused heteroaryl; -C(O)-B; or <CHEM>  wherein k is 1-2; D is B'-(CH2)mC(O)-, wherein m is 1-5; B'-(CH2)q-, wherein q is 2-6; B'-(CH2)e-Z-(CH2)r-, wherein Z is -O-, -C(O)-, phenylene, -NR8- or -S(O)0-2-, e is 0-5 and r is 1-5, provided that the sum of e and r is 1-6; B'-(alkenylene)-; B'-(alkadienylene)-; B'-(CH2)t-Z-(alkenylene), wherein t is 0-3, provided that the sum of t and the number of carbon atoms in the alkenylene chain is 2-6; B'-(CH2)f-V-(CH2)g-, wherein V is cycloalkylene, f is 1-5 and g is 0-5, provided that the sum of f and g is 1-6; B'-(CH2)t-V-(alkenylene) or B'-(alkenylene)-V-(CH2)t-, provided that the sum of t and the number of carbon atoms in the alkenylene chain is 2-6; B'-(CH2)a-Z-(CH2)b-V-(CH2)d-, wherein a, b and d are 0-6, provided that the sum of a, b and d is 0-6; T(CH2)s-, wherein T is cycloalkyl and s is 1-6; naphthylmethyl or optionally substituted heteroarylmethyl;     B is optionally substituted phenyl; B' is naphthyl, optionally substituted heteroaryl or optionally substituted phenyl; R is hydrogen, fluoro, alkyl, alkenyl, alkynyl, or B-(CH2)h-, wherein h is 0-3; R4 is optionally substituted phenyl, indanyl, benzofuranyl, tetrahydronaphthyl, pyridyl, pyrazinyl, pyrimidinyl or quinolyl; are disclosed, as well as their use as hypocholesterolemic agents; the method of using compounds of the formula II <CHEM>  wherein R20 is optionally substituted phenyl, optionally substituted naphthyl, optionally substituted heteroaryl, or optionally substituted benzofused heteroaryl,     R21, R22 and R23 are independently selected from H or R20; E, F and G are independently a bond; cycloalkylene; alkylene; alkenylene; alkynylene; a substituted alkylene, alkenylene or alkynylene chain ; an interrupted alkylene, alkenylene or alkynylene chain ; or an interrupted alkylene, alkenylene or alkynylene chain substituted by one or more substituents; or one of R21-E and R22-F is selected from the group consisting of halogeno, OH, alkoxy, -OC(O)R5, -NR10R11, -SH or -S(alkyl);     R5 is alkyl, phenyl, R14-phenyl, benzyl or R14-benzyl; R10 and R11 are independently selected from H and lower alkyl, or a pharmaceutically acceptable salt thereof, in a pharmaceutically aceptable carrier as hypocholesterolemic agents is also disclosed.
Patent AU-694229-B2 (AU)
Title: A pharmaceutical preparation comprising glucagon
Inventor: KORNFELT TROELS
IPC: A61P3/12
Filed: 1995-05-26
Granted: 1998-07-16
Abstract: The present invention relates to a pharmaceutical preparation comprising glucagon and a stabilizing amount of a pharmaceutically acceptable ampholyte, especially an amino acid or dipeptide or a mixture thereof and optionally an excipient. The preparation is stable for extended periods of time in solution at room temperature.
Patent AU-612803-B2 (AU)
Title: Method of manufacturing a mold in the form of a multiple- impression plastic plate for reproducing intaglio printing plates and plant for implementation thereof
Inventor: COLUZZI ANTONIO
IPC: B41N3/00
Filed: 1989-03-22
Granted: 1991-07-18
Abstract: To produce a multiple form for the reproduction of line-engraved intaglio printing plates, a heat-deformable plastic plate (4) which, essentially, has the dimensions of the desired line-engraved intaglio printing plate is introduced between an engraved original plate and an electrode (7) by means of a sliding frame (3) in a position corresponding to the first impression to be made and is given the first impression (23) by hot pressing in a low-pressure chamber with high-frequency heating; after cooling and the original plate, the plastic plate (4) is removal of moved into the position corresponding to the second impression (23) and provided with the same impression; these operations are repeated until the desired number and arrangement of the impressions have been produced. 
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Patent AU-762069-B2 (AU)
Title: Creativity center apparatus and method of use
Inventor: WILSON MARTIN
IPC: B43L3/00
Filed: 2000-02-04
Granted: 2003-06-19
Abstract: A creativity center includes a base portion that is connected by a hinge to a board that has opposed drawing/design surfaces on which artistic designs and markings can be made. The board can rotate with respect to the base via the hinge and can be slid with respect to the hinge such that the board can be repeatedly flipped over and slid between two opposed "use" positions with respect to the base. Thus, an opposed drawing/design surface configured in a "use" position is presented to a user each time the board is flipped over. An eraser can be located on either the base or on the hinge to automatically remove designs or markings located on the board when the board is slid through the hinge. In addition, the base can include a storage compartment for storing art supplies.
Patent AU-717507-B2 (AU)
Title: A method for the continuous casting of thin metal products, and apparatus for carrying out the same
Inventor: CAPOTOSTI ROMEO
IPC: B22D11/06
Filed: 1997-07-09
Granted: 2000-03-30
Abstract: A method for continuously casting thin metal products, the method comprising the operations of pre-heating a pair of refractory plates (7) for the lateral containment of a bath of molten metal constituted of a pair of counter-rotating rolls (1, 2) and of abutting said pair of plates (7) towards each lateral surface of the ends of said pair of rolls (1, 2), characterized in that it comprises the operations of applying a controlled elastic or elastic/plastic deformation to said pair of plates (7) at the contacting arc between the surface of the plates (7) and the peripheral portion of the ends of said rolls (1, 2), and controlling said elastic and/or elastic-plastic deformation of said pair of plates (7) during the whole casting process, so as to minimize the surface wear of the plates (7) and of the ends of the rolls (1, 2), and to guarantee the maintainment of a predetermined distance between said rolls (1, 2) and said plates (7) lower than a predetermined value, and to minimize the occurrence of leaks-of molten metal between said plates (7) and said end parts of said rolls (1, 2).
Patent AU-759124-B2 (AU)
Title: Ternary polymer blend, the film containing it, and the easy-to-open package made therewith
Inventor: LONGO EUGENIO
IPC: B32B27/32
Filed: 1999-04-09
Granted: 2003-04-03
Abstract: Object of the present invention is an extrudable blend comprising (i) a copolymer of ethylene and acrylic acid or methacrylic acid (ii) a modified EVA copolymer and (iii) a polybutylene. Included are the films comprising said blend in the sealant layer or in a layer directly adhered to the sealant layer, and the easy-to-open packages obtained therefrom.
Patent AU-712009-B2 (AU)
Title: Vacuum extrusion apparatus and method
Inventor: SADINSKI ROBERT L
IPC: B29C48/07
Filed: 1997-08-11
Granted: 1999-10-28
Abstract: An extruder projects through a bulkhead adapted to form part of a vacuum chamber, and a die is mounted on the end of the extruder within the bulkhead. The extruder projects through a gland seal which is formed in a sleeve surrounding the extruder. The seal includes a plurality of seal rings surrounding the extruder and packed in the sleeve and held in place in a preferred from by a yieldable retainer. A shaper is positioned downstream of the die and is clamped to the upstream end of the die. The shaper is mounted on tracks on a girder extending from the bulkhead clear of its periphery. The apparatus permits congruent axial movement of the extruder, die and shaper with respect to the bulkhead.
Patent AU-773590-B2 (AU)
Title: Method for detecting and modifying mismatches and mutations in nucleic acid
Inventor: GOTOH MASANORI
IPC: C12Q1/68
Filed: 2000-04-19
Granted: 2004-05-27
Abstract: An objective of this invention is to provide a method for effectively detecting mismatches or mutations in a nucleic acid using MutM protein and a method for effectively separating a nucleic acid with mismatches using MutM protein. MutM protein has been found to be able to recognize any mismatches involving cytosine in a nucleic acid. It has also been found that, using the characteristic of the MutM protein, mismatches in a double-stranded nucleic acid can be efficiently detected and a double-stranded nucleic acid with mismatches can be separated from double-stranded nucleic acid samples.
Patent AU-759600-B2 (AU)
Title: Hydrazinium nitroformate based high performance solid propellants
Inventor: LOUWERS JEROEN
IPC: C06D5/00
Filed: 1999-05-19
Granted: 2003-04-17
Abstract: The present invention is directed to a solid propellant for rocket motors, gas generators and comparable devices, comprising a cured composition of hydrazinium nitroformate and an unsaturated hydroxyl terminated hydrocarbon compound.
Patent AU-572759-B2 (AU)
Title: Device for counting and sorting coins in a coin collector
Inventor: ZIMMERMAN GERT
IPC: G07D/
Filed: 1985-05-17
Granted: 1988-05-12
Abstract: PCT No. PCT/DE85/00171 Sec. 371 Date Jan. 21, 1986 Sec. 102(e) Date Jan. 21, 1986 PCT Filed May 17, 1985 PCT Pub. No. WO85/05478 PCT Pub. Date Dec. 5, 1985.A device for counting and sorting coins belonging to a set of coins with a guideway 8 tangentially connected to a horizontal coin plate 3 is to be developed for separating foreign coins 11' through a sort-out opening 16. To this end, and behind a coin identifying device 14 and immediately in front of the sort-out opening 16, a diversion element 18 is movably arranged for the coins 11' identified as foreign or counterfeit coins by the coin identification device 14, with its front edge 35 arranged at a distance of at least the width of guide rail 17 from the guiding edge 9, with the diversion element 18 able to be triggered by the coin identification device 14. The diversion element 18, which in its active position is brought into the path of movement of coins 11, 11', diverts the coins from guiding edge 9 by at least a distance that is equal to or greater than the width of guide rail 17. In this manner, the foreign coins 11' to be separated out can drop through the sort-out opening 16. To improve the identification quality, the coin identifying device 14 comprises in addition to an optical fiber bar 31 for identifying diameters, also inductive heads 32, 33 to identification of the alloy of coins 11, 11' and/or for determining the thickness of coins 11, 11'. In addition, further components to identify the milled edge of the coins and their surface structure are arranged downstream.
Patent AU-570134-B2 (AU)
Title: Production of synthesis gas with increased h2/co ratio
Inventor: JACOMETTI JACK
IPC: C01B3/36
Filed: 1985-10-08
Granted: 1988-03-03
Abstract: Process for the production of synthesis gas with an increased H2/CO-ratio from normally gaseous hydrocarbons comprising the following steps: a) at least one normally gaseous hydrocarbon is converted into a synthesis gas comprising H2 and CO by partial oxidation with an oxygen-containing gas; b) at least one normally gaseous hydrocarbon is converted with steam into a gaseous mixture comprising H2 and CO; c) the gaseous mixture comprising H2 and CO, formed in step (b) is separated into a CO-containing stream and a H2 stream; d) the H2/CO-ratio of the synthesis gas produced in step (a) is increased by adding at least part of the H2 stream obtained in step (c) thereto.
Patent AU-580338-B2 (AU)
Title: Biologically compatible adhesive
Inventor: BLACKWELL GORDON B
IPC: A61K6/00
Filed: 1985-10-08
Granted: 1989-01-12
Abstract: A biologically compatible adhesive that is shelf stable as a single component adhesive and includes a mixture of an adhesive promoting and polymerizable monomer system having a free radical polymerizable monomer or prepolymer having ethylenic unsaturation and a phosphorus containing adhesion promoter, a free radical polymerization catalyst, . and an accelerator for the catalyst, the accelerator selected from the group consisting of sulfinic acid or salt thereof, amine or amine salt and mixtures thereof.
Patent AU-634206-B2 (AU)
Title: A process and an apparatus for die-cutting of packaging material
IPC: B31B50/25
Filed: 1990-01-17
Granted: 1993-02-18
Abstract: PCT No. PCT/SE90/00040 Sec. 371 Date Jul. 5, 1991 Sec. 102(e) Date Jul. 5, 1991 PCT Filed Jan. 17, 1990 PCT Pub. No. WO90/08018 PCT Pub. Date Jul. 26, 1990.A process and an apparatus for preventing a packaging material which is being die-cut and scored from developing cracks. A crack-reducing sheet material (17) is positioned between the cutting/scoring tools (9, 13) and the packaging material (5) to absorb impact energy from said tools and relieve the packaging material of crackproducing forces in the direction of its plane.
Patent AU-695331-B2 (AU)
Title: Process for activating polysaccharides, polysaccharides produced by this process, and use thereof
Inventor: KARSTENS TIES
IPC: C08B37/00
Filed: 1996-03-22
Granted: 1998-08-13
Abstract: PCT No. PCT/EP96/01274 Sec. 371 Date Nov. 6, 1997 Sec. 102(e) Date Nov. 6, 1997 PCT Filed Mar. 22, 1996 PCT Pub. No. WO96/30411 PCT Pub. Date Oct. 3, 1996The process for activating polysaccharides consists of contacting the polysaccharide with liquid ammonia at an initial pressure which is higher than atmospheric pressure and at a temperature of at least approximately 25 DEG  C., the amount of liquid ammonia being sufficient at least for wetting the surface of the polysaccharide starting material which is then expanded. The volume available for the polysaccharide/liquid ammonia system is enlarged in the manner of an explosion by lowering the pressure by at least 5 bar. The process is particularly suitable for activating cellulose, guar gum, starch and chitin. The process enables cellulose to be modified in a novel manner. The activated polysaccharides display higher reactivity and improved elimination of reagents during acylation, alkylation, silylation, xanthogenation and carbomoylation with largely homogeneous reaction processes.
Patent AU-526151-B2 (AU)
Title: Rate controlled directional solidification of nickel base alloys
Inventor: GIAMEI ANTHONY FRANCIS
IPC: B22D27/20
Filed: 1979-10-16
Granted: 1982-12-16
Abstract: An improved method of directional solidification is provided by varying the rate of withdrawal of a casting from the hot zone of a solidification furnace according to the sense of change of the perimeter to area ratio of the casting. The rates are varied to achieve desired microstructure and resultant properties in the casting. Also, the rate of withdrawal is varied according to controlled and predetermined relationships to cause the solidification interface to move through a transition section connecting sections of differing perimeter to area ratios in a manner which produces a desired microstructure in a first, transition, and second sections.
Patent AU-587019-B2 (AU)
Title: Television synchronizing apparatus
Inventor: WILLIS DONALD HENRY
IPC: H04N5/12
Filed: 1986-03-25
Granted: 1989-08-03
Abstract: In a synchronized digital horizontal deflection system operating at 2xf<sub>H</sub>, a first word (HDPW) is produced that is indicative of the length of one-half the period H between f<sub>H</sub> rate horizontal sync pulses (Hs). A first f<sub>H</sub> rate signal (CMa) that is synchronized to the horizontal sync pulses (Hs) is generated. The first f<sub>H</sub> rate signal (CMa) is time shifted by one-half of the period H, in accordance with the first word (HDPW) to produce a second f<sub>H</sub> rate signal (CMb). The first (CMa) and second (CMb) signals are multiplexed (in 40) for generating a horizontal deflection control signal (CMa, CMb) at 2xf<sub>H</sub> rate that controls the retrace interval timing in a deflection circuit output stage (41).
Patent AU-678803-B2 (AU)
Title: Novel colon- or ileum-specific steroid derivatives
Inventor: BRATTSAND RALPH LENNART
IPC: A61K31/58
Filed: 1993-12-17
Granted: 1997-06-12
Abstract: Novel compounds which are a glucocorticosteroid (GCS) chemically bound to a sugar, having the general formula GCS1-O-Sugar1 for colon- or ileum-specific delivery of the GCS to inflamed bowel mucosa, as well as processes for their preparation, pharmaceutical preparations containing the compounds and the use of said compounds in therapy.
Patent AU-647400-B2 (AU)
Title: Process for coating a glass surface
Inventor: BACHLI EMIL
IPC: C03C27/12
Filed: 1990-07-16
Granted: 1994-03-24
Abstract: PCT No. PCT/CH90/00172 Sec. 371 Date Mar. 18, 1991 Sec. 102(e) Date Mar. 18, 1991 PCT Filed Jul. 16, 1990 PCT Pub. No. WO91/01429 PCT Pub. Date Feb. 7, 1991.For coating the glass edge of two wall elements (2, 3) forming interspace (5) for heat insulating structural and/or light element (1), metallic adhesive layer (4) is produced with the use of a physical (PVD) or chemical (CVD) deposition of the coating material from a gas or vapor phase on one side of each wall element (2, 3). On this adhesive layer (4) barrier layer (6) protecting the latter is deposited and the barrier layer is provided with subsequent solder layer (7). These solder layers (7) are bonded with sheet (8) that edges structural and/or light element (1) on the edge in a gastight manner.
Patent AU-721461-B2 (AU)
Title: Telecommunications switching system with readily configurable supervisor control
Inventor: HEBERT MARK P
IPC: H04L12/24
Filed: 1998-02-10
Granted: 2000-07-06
Abstract: A telephone switching system comprises a plurality of switching nodes interconnected by a call-switching network. The switching nodes are also linked by a host network to one or more hosts that exercise supervisory control over the nodes. The hosts communicate directly with one or more of the nodes, termed "switching nodes", by means of virtual connections over the host network. The other switching nodes, termed "slave nodes", are assigned to host nodes. The hosts communicate indirectly with the slave nodes by way of switching nodes to which they are assigned. Communications between a host and a slave node thus comprise messages (a) over the host network between the slave node and the switching node to which the slave node is assigned and (b) by way of a virtual connection between the switching node and the host.
Patent AU-765439-B2 (AU)
Title: Synthetic analogs of ecteinascidin-743
Inventor: COREY ELIAS J
IPC: A61K31/4995
Filed: 1999-09-30
Granted: 2003-09-18
Abstract: The present invention is directed to the synthesis and characterization of compounds having the formula: wherein R1, R2, R3, R4, R5, R6, R7, R8 and R9 are each independently selected from the group consisting of H, OH, OR′, SH, SR′, SOR′, SO2R′, NO2, NH2, NHR′, N(R′)2, NHC(═O)R′ NHC(═O)R′, CN, halogen, ═O, C(═O)H, C(═O)R′, CO2H, CO2R′, C1-C12 alkyl, C2-C12 alkenyl, C2-C12 alkynyl, substituted or unsubstituted aryl, substituted or unsubstituted aralkyl, and substituted or unsubstituted heteroaromatic; wherein each of the R′ groups is independently selected from the group consisting of H, OH, NH2, NO2, SH, CN, halogen, ═O, C(═O)H, C(═O)CH3, CO2H, CO2CH3, C1-C12 alkyl, C2-C12 alkenyl, C2-C12 alkynyl, aryl, aralkyl, and heteroaromatic; wherein each dotted circle represents one, two or three optional double bonds; wherein R7 and R8 may be are joined into a carbocyclic or heterocyclic ring system; and wherein X1 and X2 are each independently defined as above for R1-R8 R1-R6 and R9, and each further includes specific preferred groups as defined herein.
Patent AU-585091-B2 (AU)
Title: Cephalosporin compounds
Inventor: ARNOULD JEAN CLAUDE
IPC: C07D501/46
Filed: 1986-11-14
Granted: 1989-06-08
Abstract: A cephalosporin derivative of the formula I:-in which X is S, O, CH<sub>2</sub> or SO,represents one of the C-7 acyl groups known in the cephalosporin art, R3 is hydrogen or methoxy, R4 is hydrogen, optionally substituted alkyl, allyl, furfuryl or benzyl, and R5 is an aromatic heterocyclic ring system which is linked via carbon, and which contains a quaternised nitrogen atom.
Patent AU-583683-B2 (AU)
Title: Yeast production of hepatitis B surface antigen
Inventor: TSCHOPP JUERG FRIEDRICH
IPC: C12N15/36
Filed: 1986-11-19
Granted: 1989-05-04
Abstract: Novel DNA constructs comprising regulatory regions plus the structural coding region for hepatitis B surface antigen (HBsAg) are disclosed. The regulatory regions employed are responsive to methanol, non-catabolite repressing carbon sources and catabolite repressing carbon sources followed by carbon source starvation. The novel constructs are incorporated into a variety of linear and circular plasmids. Such plasmids are used to transform suitable hosts and ultimately used for the production and isolation of hepatitis B surface antigen in high yields.
Patent AU-653504-B2 (AU)
Title: Oligonucleotide analogs with novel linkages
Inventor: MATTEUCCI MARK
IPC: A61K31/7052
Filed: 1990-10-24
Granted: 1994-10-06
Abstract: The instant invention is directed to oligonucleotide compounds wherein on or more phosphodiester linkages between adjacent nucleotides are replaced by a formacetal/ketal type linkage. The nucleotides of the present invention are resistant to nucleases and do not need to exhibit the diastereomerism characteristic of many other oligonucleotide compounds and thus are capable of strong hybridization to target RNA or DNA. These oligonucleotide compounds are useful in therapies which modulate gene expression using antisense or other specifically binding oligomers.