baber/WOPTO huggingface dataset:
Patent IL-117290-A0 (IL)
Title: Preparation of n-substituted pyrazoles
IPC: C07D521/00
Filed: 1996-02-28
Abstract: PCT No. PCT/EP96/00790 Sec. 371 Date Aug. 20, 1997 Sec. 102(e) Date Aug. 20, 1997 PCT Filed Feb. 27, 1996 PCT Pub. No. WO96/27589 PCT Pub. Date Sep. 12, 1996A process for the preparation of an N-alkyl- or N-phenylalkyl-substituted pyrazole I by reacting the corresponding N-unsubstituted pyrazole II with an alcohol III of the formula R1-OH where R1 is the same alkyl or phenylalkyl group to be added to the unsubstituted nitrogen group -NH- of the pyrazole reactant. Both of the reactants, i.e. the pyrazole II and alcohol III compounds, are catalytically reacted in the liquid phase in a molar ratio of from 0.001:1 to 1:1, at temperatures of 50 DEG -400 DEG  C. and under a subatmosheric pressure of from 0.8 bar up to a superatmospheric pressure of 250 bar. The catalyst required for this liquid phase reaction is selected as being at least one or more non-heterogeneous acid catalysts, their alkyl esters or their acid anhydrides.
Patent IL-117301-A0 (IL)
Title: Method and system for displaying signals generated by an object
IPC: G01S/
Filed: 1996-02-28
Abstract: A multi-dimensional acoustic, data processing and display system arranges acoustic data in a three-dimensional matrix. The three-dimensional matrix is compressed using singular value decomposition into singular vectors and singular values. A historical database is created and maintained and is also concatenated with the three-dimensional data. This database allows reverberation and noise to be diminished and other, weaker features in the data to be enhanced. Once the data is compressed, the data can be analyzed efficiently. The singular vectors are partitioned into one or more groups on the basis of their singular values or other criteria. Certain of the compressed data elements are enhanced or diminished by modifying the singular values within each of the groups of singular vectors. Selected singular vectors are processed further by other techniques for further enhancement, detection, isolation, feature extraction and classification. The compressed and enhanced data is then expanded back into three-dimensional form for display or for other processing.
Patent IL-123579-A0 (IL)
Title: Apparatus for producing high contrast imagery
IPC: G09F9/40
Filed: 1998-03-06
Abstract: A visual display is provided comprising a plurality of pixels each of which comprises: a surface having an area less than one square millimiter comprising first and second regions having surface finishes; and a thin planar panel having first and second sides having surface finishes, wherein the panel is rotatably coupled to the surface so as to rotate between a first and a second position about an axis parallel to the surface; wherein the panel in the first position is positioned over the first region with its second side facing the first region and wherein in the second position the panel is positioned over the second region with its first side facing the second region.
Patent IL-124409-A0 (IL)
Title: Method of detecting telomerase activity
IPC: C12Q1/68
Filed: 1996-11-27
Abstract: The invention concerns a method for the detection of telomerase activity wherein(a) a sample to be tested is provided,(b) a first primer suitable as a telomerase substrate and nucleoside triphosphates are added and the reaction mixture is incubated under conditions under which a primer extension by the telomerase can take place,(c) an amplification of the extension product produced by the telomerase is carried out,(d) the amplification product produced in step (c) is immobilized on a solid phase and(e) the immobilized amplification product is detected qualitatively or/and quantitatively. Furthermore the invention concerns a suitable reagent kit for carrying out the method.
Patent IL-137600-A0 (IL)
Title: Process and device for producing cross-linked polyolefin foams
IPC: B29K105/04
Filed: 1999-02-02
Abstract: Furnaces for cross-linking and foaming polyolefin plates or foils having several successive zones associated each with a foil heating device are known. The aim of the invention is to enable cross-linked polyolefin foams to be produced in a more economical manner. According to the disclosed process, hot air flows past the polyolefin plate or foil against its transport direction. The disclosed device (24) for heating the polyolefin plate or foil (2) is arranged and designed in such a way that the hot air (25) leaving the device (24) flows parallel to the plate or foil plane (26). The device for heating the polyolefin plate or foil (2) is preferably a heating tunnel (30) which encloses the plate or foil (2).
Patent IL-139774-A0 (IL)
Title: Multiparticular pharmaceutical form with programmed and timed release and preparation method
IPC: A61P43/00
Filed: 1999-05-20
Abstract: The invention concerns a mutliparticulate pharmaceutical form with delayed and timed release for starting to make the active principle available 4 to 8 hours after said pharmaceutical form has been ingested, then for gradually releasing the totality of the active principle within the following 8 to 20 hours. The invention is characterised in that it is free of organic acid and it is in the form of medicated spheroids consisting of a neutral spherical carrier comprising a first coating based on a mixture of at least a water soluble polymer and at least a water insoluble polymer wherein are uniformly distributed particles constituting an active principle, the whole comprising a second coating based on at least two independent pH polymers, having degrees of permeability with respect to different gastric and intestinal environments, optionally at least a dependent pH polymer, at least a plasticising agent and at least an inert filler distributed in said coating.
Patent IL-145122-A0 (IL)
Title: C16 unsaturated fp-selective prostaglandin analogs
IPC: C07C405/00
Filed: 2000-02-29
Abstract: Compounds having the general structure: which are useful for the treatment of a variety of diseases and conditions, such as bone disorders.
Patent IL-149680-A0 (IL)
Title: A method for preparing lysophosphatidylethanolamine
IPC: C12P13/00
Filed: 2000-11-28
Abstract: Disclosed herein is a method for purifying the lysophosphatidylethanolamine with high purity by treating the phospholipid mixture with enzymes, followed by solvent fractionaltion without the column purification. The method of the present invention comprises hydrolyzing phospholipid mixture containing 10-99 weight % of phosphatidylethanolamine with phospholipase A2 to produce lysophospholipid; and treating the lysophospholipid with the solvent mixture comprising water and one or more organic solvents selected from the group consisting of low alcohol, hydrocarbon and alkylester to eliminate impurities except lysophosphatidylethanolamine.
Patent IL-151211-A0 (IL)
Title: Compositions useful for regulating parkin gene activity
IPC: C12N15/09
Filed: 2001-02-15
Abstract: The present invention relates to novel compounds and their uses, in particular their pharmaceutical or diagnostic uses or their use as pharmacological targets. More particularly, the present invention relates to a novel protein, referred to as PAP1, as well as to novel peptides and compounds which are capable of modulating, at least partially, the activity of parkin.
Patent IL-157964-A0 (IL)
Title: Method for the production of biologically-degradable packagings made from biaxially-drawn films
IPC: B29C55/12
Filed: 2002-04-23
Abstract: The invention relates to a method for the plastic shaping of a biaxially-drawn film, comprising at least one base layer, containing at least one polymer (I), made from at least one hydroxycarboxylic acid and >=0.2 wt %, based on the weight of the layer, of a thermoplastic polymer (II), different from polymer (I). Said film is plastically moulded by application of pneumatic and/or mechanical forces.
Patent IL-161692-A0 (IL)
Title: 14-benzodiazepine derivatives and pharmaceutical compositions containing the same
IPC: A61P19/02
Filed: 2002-11-13
Abstract: The present invention is directed to novel 1,4-benzodiazepines, pharmaceutical compositions thereof, and the use thereof as inhibitors of HDM2-p53 interactions. Compounds have Formula I: or a solvate, hydrate or pharmaceutically acceptable salt thereof; wherein: X and Y are independently -C(O)-, -CH<SUB>2</SUB>- or -C(S)-; R<SUP>1</SUP>, R<SUP>2</SUP>, R<SUP>3</SUP>, R<SUP>4</SUP>, R<SUP>7</SUP>, R<SUP>8</SUP>, R<SUP>b</SUP>, R<SUP>c</SUP>, R<SUP>d </SUP>and M are defined herein; R<SUP>5 </SUP>is hydrogen, alkyl, cycloalkyl, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted aralkyl, optionally substituted heteroaralkyl, carboxyalkyl, alkoxycarbonyl, alkoxycarbonylalkyl, aminocarbonyl, aminocarbonylalkyl, alkylaminocarbonyl or alkylaminocarbonylalkyl; R<SUP>6 </SUP>is cycloalkyl, aryl, heteroaryl, cycloalkylalkyl, aralkyl, heteroarylalkyl, or a saturated or partially unsaturated heterocycle, each of which is optionally substituted; R<SUP>9 </SUP>is cycloalkyl, aryl, heteroaryl, a saturated or partially unsaturated heterocycle, cycloalkyl(alkyl), aralkyl or heteroarylalkyl, each of which is optionally substituted; and R<SUP>10 </SUP>is -(CH<SUB>2</SUB>)<SUB>n</SUB>-CO<SUB>2</SUB>R<SUP>b</SUP>, -(CH<SUB>2</SUB>)<SUB>m</SUB>-CO<SUB>2</SUB>M, -(CH<SUB>2</SUB>)<SUB>i</SUB>-OH or -(CH<SUB>2</SUB>)<SUB>j</SUB>-CONR<SUP>c</SUP>R<SUP>d </SUP> n is 0-8, m is 0-8, i is 1-8 and j is 0-8.
Patent IL-162332-A0 (IL)
Title: Bone anchor insertion device
IPC: A61B17/56
Filed: 2002-12-06
Abstract: A bone anchor insertion device comprises a handle, a nosepiece connected to a distal end of the handle, a bone anchor connected to the nosepiece, and an actuator disposed on the handle for deploying the bone anchor, which suture is also fixed to a portion of soft tissue to be attached to a portion of bone. A suture ratchet or tensioning mechanism is disposed in the handle for tensioning suture which is associated with the bone anchor. This mechanism permits precise tensioning, while also permitting one-handed operation, thereby allowing the practitioner to use his or her other hand for other activities, such as camera operation or the like.
Patent IL-180551-A0 (IL)
Title: Use of substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines in the treatment of nausea and vomiting
IPC: A61K31/4427
Filed: 2007-01-04
Abstract: The present invention relates to the use of substituted 2-thio-3,5-dicyano-4-phenyl-6-amino-pyridines of the formula (I) wherein the terms A and R2 are herein defined, for treatment of nausea and vomiting.
Patent IL-182845-A0 (IL)
Title: Oxidation and fatigue resistant metallic coating and method for depositing the same
IPC: C23C30/00
Filed: 2003-04-28
Abstract: The present invention relates to a metallic coating to be deposited on gas turbine engine components. The metallic coating comprises up to 18 wt% cobalt, 3.0 to 18 wt% chromium, 5.0 to 15 wt% aluminum, 0.1 to 1.0 wt% yttrium, up to 0.6 wt% hafnium, up to 0.3 wt% silicon, 3.0 to 10 wt% tantalum, up to 9.0 wt% tungsten, 1.0 to 6.0 wt% rhenium, up to 10 wt% molybdenum, and the balance nickel.
Patent IL-191135-A0 (IL)
Title: Method for storing the position of a parked vehicle and navigation device arranged for that
Filed: 2008-04-29
Abstract: The present invention relates to a navigation device comprising a processor unit (11). The navigation device (10) is arranged to detect parking of a vehicle, and, when parking is detected, determine information regarding the position of the parked vehicle. Next, the information regarding the position of the parked vehicle is stored. The stored information may be reused later to find the parked vehicle.
Patent IL-196319-A0 (IL)
Title: Methods for determining a human subject's propensity to develop a vascular disorder
Filed: 2009-01-01
Abstract: Disclosed are screening methods for determining a human subject's propensity to develop a vascular disorder and/or age-related macular degeneration (AMD), therapeutic or prophylactic compounds for treating disease or inhibiting its development, and methods of treating patients to alleviate symptoms of the disease, prevent or delay its onset, or inhibit its progression. The inventions are based on the discovery that persons with a genome having a deletion of the CFHR-1 and/or CFHR-3 gene, which normally lie on human chromosome 1 between DNA encoding CFH and CFHR-4, are at reduced risk of developing AMD, and elevated risk of developing vascular disease such as aneurysm.
Patent IL-219993-A0 (IL)
Title: Intermediate in production of [2-(3,3,5,5-tetramethylcyclohexyl)phenyl] piperazine compound
Filed: 2012-05-24
Abstract: A compound represented by the general formula below or a salt thereof is a useful intermediate in the production of a [2-(3,3,5,5-tetramethylcyclohexyl)phenyl]piperazine compound that has excellent cell adhesion inhibitory effect and cell invasion inhibitory effect and therefore is useful as a therapeutic or prophylactic agent for various inflammatory diseases and autoimmune diseases induced by the adhesion and invasion of leukocytes, such as inflammatory bowel diseases (particularly ulcerative colitis or Crohn's disease), irritable bowel syndrome, rheumatoid arthritis, psoriasis, multiple sclerosis, asthma and atopic dermatitis. wherein R1 and R2 independently represent hydrogen or a protecting group for an amino group, or R1 and R2 bond together to form an optionally substituted pyrrole ring.
Patent RO-125770-A0 (RO)
Title: Process and installation for producing powders of binary aluminium-magnesium alloys meant for making metal pieces of thixotropic structure
Inventor: BINCHICIU HORIA
IPC: C04B35/622
Filed: 2010-02-01
Abstract: The invention relates to a process and an installation for continuously producing metal powders of aluminium-magnesium alloys with melting temperatures under 1000°C, meant for the production of pieces of thixotropic structure by injection moulding. According to the invention, the installation comprises a feeding mechanism (2) for wire (1) and a feeding mechanism (3) for the cored pipe (4), which lead the components of the binary alloy with variable advance speeds to an induction-heated crucible (5) which is provided at its bottom with a system of nozzles (10) wherethrough the melted alloy flows in a laminar motion on a refractory stainless steel drum (14) which rotates with a speed ranging between 600...6000 rpm, in the preforming chamber (11) protected by argon atmosphere, the melted alloy being then projected onto a deflective plate (12) at an angle adjustable between 0...45°, where it is converted into drops which, after solidification, are deposited onto the cooling collector bed (16). The claimed process consists in an adequate dosing of the quantity of 97% active Al solid wire (1), having a diameter of 2 mm, and of the quantity of Mg-cored aluminium pipe (4), having a diameter of 3.25 mm, necessary to form a melt (9) under a protective layer of cryolitic flux (8) in an induction furnace with graphite crucible (5), said melt flowing through some nozzles into the preforming chamber (11), on a drum (14) rotating with variable speed and projecting the melt jet onto a deflective plate (12) inclined under an adjustable angle (alpha), which achieves the jet dispersion into pulverous particles (15) which are then deposited onto the cooling collector bed (16) in an atmosphere of protective inert gas.
Patent RO-130104-A0 (RO)
Title: Active inclining mechanism for 3- or 4-wheeled electric vehicles
Inventor: COCIRTA THOMAS
IPC: B62D61/08
Filed: 2014-11-07
Abstract: The invention relates to an active inclining mechanism for the three- or four-wheeled electric vehicles, provided with subassemblies of individual suspension on each wheel. According to the invention, the mechanism consists of two symmetrical longitudinal arm assemblies (B and C), mounted on a central bogie (A), and, for carrying out the inclination, it uses the action of an electric or hydraulic actuation system to allow the rotation of the two longitudinal arm subassemblies (B and C) in opposite directions about some radial axial articulations (2), having the axis perpendicular on the central plane of the bogie (A), each of the two longitudinal arm subassemblies (B and C), which carry out the inclination, including a suspension system consisting of a longitudinal suspension arm proper (3) and an intermediary suspension arm (7), rotary supported on the central bogie (A), into the same double articulation (2) having the axis perpendicular on the median plane of the vehicle, and between which there is a passive suspension system consisting of a spring (8) and a damper (9), the two longitudinal arm subassemblies (B and C) being connected to one another by means of a load equalizing system, consisting of some articulations (12 and 15), some pushing rods (13) and an equalizing lever (14), articulated on the bogie (A) into a radial-axial articulation (16) and which provides the transmission of the static forces taken over by the wheels directly into the chassis of the bogie (A) and not by means of the electric servomechanisms for the inclination actuation.
Patent LU-85426-A1 (LU)
Title: N-Alkyl:iso:stearamide antistatic agent - used in detergent compsn in washing machine for textile fabrics
Inventor: BAUMAN ROBERT ANDREW
IPC: C11D1/52
Filed: 1984-06-21
Abstract: N-alkylisostearamide antistatic agent is of formula RCONHR' (I) where RCO is derived from isostearic acid, and R1 is a primary, opt. unsatd. aliphatic hydrocarbon chain of 1-18C, pref. 7-18C. (I) is used in antistatic compsn. for the machine washing of fabrics, either in combination with an anionic, nonionic or amphoteric detergent or dispersed in an absorbing substrate. (I) imparts antistaticity to fabrics without reducing the efficiency of optical brighteners and the detergency of washing compsns.
Patent MA-20450-A1 (MA)
IPC: C07D491/048
Filed: 1985-06-06
Abstract: This invention relates to 1,3 - dihydro-6-aminomethyl-7-hydroxy-furo-(3,4-c)- pyridine derivatives of the general formula I  <IMAGE>  wherein A1, A2, R1 and R2 represent various substituents, to pharmaceutically acceptable salts of such compounds, to a process for the preparation of compounds comprising reacting a 6-chloromethyl-7-benzoxy derivative of the general formula II  <IMAGE> II  with an excess of an amine derivative  <IMAGE>  in a non-polar solvent, at a temperature not exceeding 20 DEG  C., which leads to the desired substitution in position 6, followed by an acidic treatment to cleave the benzyl group and, finally to an anti-allergic composition of matter comprising, as an essential ingredient therein, an effective amount of one of these compounds together with an appropriate diluent or carrier.
Patent MA-27195-A1 (MA)
Title: Derives d'acyl-3 -carboxyphenyluree, procedes pour les preparer et leur utilisation.
Inventor: DEFOSSA ELISABETH
IPC: C07C/
Filed: 2004-10-08
Abstract: Dérivés d'acyl-3-carboxyphénylurée, procédés pour les préparer et leur utilisation. L'invention concerne des dérivés d'acyl-3-carboxyphénylurée ainsi que leurs sels tolérés physiologiquement et dérivés physiologiquement fonctionnels. L'invention concerne les composés de formule (I) dans laquelle les restes ont les significations indiquées, ainsi que leurs sels tolérés physiologiquement et procédé pour leur préparation. Les composés conviennent, par exemple, en tant qu'antidiabétiques.
Patent MA-27711-A1 (MA)
Title: Derives de pyrazolo [1,5-a] pyrimidine
Inventor: KATAOKA KENICHIRO
IPC: A61P7/00
Filed: 2005-08-12
Abstract: Les dérivés de pyrimidine de Pyrazolo [1, 5-a] représentés par la formule I et leurs sels pharmaceutiquement acceptables exposent une activité de kinase excellente. Les médicaments comprenant les composés comme des éléments actifs sont par conséquent attendus d'être utiles comme des agents thérapeutiques ou prophylactique pour le trouble initié par la protéine kinase dans laquelle il est impliqué, tel que la maladie inflammatoire, maladie auto-immune, trouble de destruction d'os, cancer et/ou croissance de tumeur.
Patent MA-27797-A1 (MA)
Inventor: ARTERO RUIZ FERNANDO
IPC: G09F3/20
Filed: 2005-11-08
Abstract: The invention relates to an improved label-bearing section of the type that is used with shelves in commercial establishments and warehouses, in order to support and protect labels containing the prices, characteristics, etc. of the products stored thereon. The invention is  characterised in that  it comprises: separate, independent anchoring elements which are used to fix same to the shelf and to determine the positioning angle of the label; and a double sheet comprising a transparent front part, which is used to house the label and which can move independently of the two anchoring elements. The main advantages offered by the invention lie in the fact that it comprises only one type of label-bearing section which can be fixed to the shelf using various inclination angles which can be eas
Patent MA-20150107-A1 (MA)
Title: Fonctionnement d'une turbine à gaz associée à une centrale à courant d'air ascendant
Inventor: LENK UWE
IPC: F03D9/00
Filed: 2013-05-06
Abstract: L'invention concerne une centrale (1) comprenant au moins une turbine à gaz (2) ainsi qu'au moins une tour (12) munie d'une unité de génération de courant (11) pour la génération d'un courant électrique par un courant d'air dynamique ascendant dans la tour (12). La turbine à gaz (2) est raccordée en communication fluidique à la tour (12) de telle manière qu'au moins une partie de l'effluent gazeux de la turbine à gaz (2) peut en fonctionnement traverser la tour (12). La turbine à gaz (2) est raccordée en communication fluidique à la tour (12) au moins en partie au moyen d'une conduite d'écoulement (13), la conduite d'écoulement (13) comportant une section d'écoulement (20) par laquelle de l'air frais peut être amené à l'effluent gazeux pour qu'il se mélange à l'effluent gazeux avant que le mélange ne soit amené à la tour (12) et/ou pendant que le mélange est amené à la tour (12).
Patent MA-40295-A1 (MA)
Title: Optimisation de l'affectation des points de stationnement des avions dans un aéroport
Inventor: Aboulmajd Badr
IPC: G06Q10/00
Filed: 2017-05-05
Abstract: Un procédé d’optimisation automatique des emplacements de stationnement des avions dans un aéroport. Nous résolvons le problème d’affectation des points de stationnement par le biais de la programmation par contrainte, en le modélisant sous forme d’un c.S.P. Nous offrons ainsi une gestion des postes de stationnement des avions, qui consiste à assigner à chaque avion à l’arrivée un poste ou une zone de stationnement compatible avec ses caractéristiques opérationnelles
Patent MA-48432-A1 (MA)
Title: Solutions aqueuses concentrées purifiées de sel de leucoindigo
Inventor: LUCIC ERWIN
IPC: D06P1/673
Filed: 2018-08-10
Abstract: La présente invention concerne une solution aqueuse de leucoindigo comprenant une amine aromatique, en particulier de l'aniline ou de l'aniline et de la n-méthylaniline, la concentration en ladite amine aromatique étant inférieure à 200 ppm, le sel de leucoindigo dans la solution se présentant sous la forme d'un sel mixte de sodium et de potassium, le rapport molaire du sodium au potassium étant situé dans la plage allant d'une valeur supérieur à 3:1 à 10:1, et de préférence, la concentration en sel étant située dans la plage allant d'une valeur supérieure à 25 à 45 % en poids, par rapport au poids total de la solution.