Patent EP-2540164-A1 (EP)
Inventor: FUNKE CHRISTIAN DR
IPC: A01N43/56
Filed: 2004-10-30
Abstract: Composition for controlling animal pests comprises a synergistic combination of a pyrethroid and an anthranilic acid derivative (I). Composition for controlling animal pests comprises a synergistic combination of a pyrethroid and an anthranilic acid derivative of formula (I). [Image] A 1>, A 2> : O or S; X 1> : N or CR 1> 0>; R 1> : H or optionally substituted C1-C6-Alkyl, C2-C6-Alkenyl, C2-C6-Alkynyl or C3-C6-Cycloalkyl; R 2> : H, C1-C6-Alkyl, C2-C6-Alkenyl, C2-C6-Alkynyl, C3-C6-Cycloalkyl, C1C4-Alkoxy, C1-C4-Alkylamino, C2-C8-Dialkylamino, C3-C6-Cycloalkylamino, C2-C6 Alkoxycarbonyl or C1-C6-Alkylcarbonyl; R 3> : H, R 1> 1> or optionally substituted C1-C6-Alkyl, C2-C6-Alkenyl, C2-C6-Alkynyl, C3-C6-Cycloalkyl; R 2>+R3 : a ring M; R 4> : H, C1-C6-Alkyl, C2-C6-Alkenyl, C2-C6-Alkynyl, C3-C6-Cycloalkyl, C1-C6 Haloalkyl, C2-C6-Haloalkenyl, C2-C6-Haloalkynyl, C3-C6-Halocycloalkyl, Halogen, Cyano, Nitro, Hydroxy, C1-C4-Alkoxy, C1-C4-Haloalkoxy, C1-C4-Alkylthio, C1-C4-Alkylsulfinyl, C1-C4-Alkylsulfonyl, C1-C4-Haloalkylthio, C1-C4-Haloalkylsulfinyl, C1-C4-Haloalkylsulfonyl, C1-C4-Alkylamino, C2-C8-Dialkylamino, C3-C6-Cycloalkylamino, C3-C6-Trialkylsilyl or optionally substituted Phenyl, Benzyl or Phenoxy; R 5>, R 8> : H, Halogen or optionally substituted C1-C4-Alkyl, C1-C4-Haloalkyl, R 1> 2>, G, J, -OJ, -OG, -S(O) p-J, -S(O) p-G, -S(O)p-phenyl; G : a 5- or 6-membered non-aromatic carbocyclic or heterocyclic ring optionally containing 1 or 2 C(=O), SO or S(=O)Z ring members and optionally substituted; J : an optionally substituted 5- or 6-membered heteroaromatic ring; R 6> : -C(=E 1>)R 1> 9>, -LC(=E 1>) 1> 9>, C(=E 1>)LR 1> 9>, -LC(=E 1>)LR 1> 9>, -OP(=Q)(OR 1> 9>)2, -SO 2LR 1> 8> or -LSO 2LR 1> 9>; E 1> : O, S, N-R 1> 5>, N-OR 1> 5>, N-N(R 1> 5>) 2, N-S=O, N-CN or N-NO 2; R 7> : H, C1-C4-Alkyl, C1-C4-Haloalkyl, Halogen, C1-C4-Alkoxy, C1-C4 Haloalkoxy, C1-C4-Alkylthio, C1-C4-Alkylsulfinyl, C1-C4-Alkylsulfonyl, C1-C4 Haloalkylthio, C1-C4-Haloalkylsulfinyl, C1-C4-Haloalkylsulfonyl; R 9> : C1-C4-Haloalkyl, C1-C4-Haloalkoxy, C1-C4-Haloalkylsulfinyl or Halogen; R 1> 0> : H, C1-C4-Alkyl, C1-C4-Haloalkyl, Halogen, Cyano or C1-C4 Haloalkoxy; R 1> 1> : optionally mono- to trisubstituted C1-C6-Alkylthio, C1-C6-Alkylsulfenyl, C1-C6-Haloalkythio, C1-C6 Haloalkylsulfenyl, Phenylthio or Phenylsulfenyl; L : O, NR 1> 8> or S; R 1> 2> : -B(OR 1> 7>) 2, Amino, SH, Thiocyanato, C3-C8 Trialkylsilyloxy, C1-C4-Alkyldisulfide, -SF 5, -C(=E)R 1> 9>, -LC(=E)R 1> 9>, -C(=E)LR 1> 9>, -LC(=E)LR 1> 9>, -OP(=Q)(OR 1> 9>) 2, -SO 2LR 1> 9> or -LSO 2LR 1> 9>; Q : O or S; R 1> 3> : H or optionally substituted C1-C6-Alkyl, C2-C6-Alkenyl, C2-C6-Alkynyl or C3-C6 Cycloalkyl; R 1> 4> : optionally substituted C1-C20-Alkyl, C2-C20-Alkenyl, C2-C20-Alkynyl or C3-C6-Cycloalkyl; R 1> 5> : H or optionally substituted C1-C6-Haloalkyl or C1-C6-Alkyl, or N(R 1> 5>) 2 forms a ring M; R 1> 6> : C1-C12-Alkyl or C1-C12-Haloalkyl, or N(R 1> 6>) 2 forms a ring M; R 1> 7> : H or C1-C4-Alkyl, or B(OR 1> 7>) 2 is a ring in which both O atoms are connected with a chain of 2-3 C atoms, optionally substituted with 1 or 2 of methyl oder C2-C6 Alkoxycarbonyl; R 1> 8> : H, C1-C6 Alkyl or C1-C6-Haloalkyl, or N(R 1> 3>)(R 1> 8>) forms a ring M; R 1> 9> : H or optionally substituted C1-C6-Alkyl; M : an optionally substituted ring comprising an N atom, 2-6 C atoms and optionally another N, O or S atom; n : 0 or 1; p : 0, 1 or 2; when (a) R 5> : H, C1-C6-Alkyl, C1-C6-Haloalkyl, C2-C6 Haloalkenyl, C2-C6-Haloalkynyl, C1-C4-Haloalkoxy, C1-C4-Haloalkylthio or Halogen steht and (b) R 8> = H, C1-C6-Alkyl, C1-C6-Haloalkyl, C2-C6-Haloalkenyl, C2-C6 Haloalkynyl, C1-C4-Haloalkoxy, C1-C4-Haloalkylthio, Halogen, C2-C4-Alkylcarbonyl, C2-C6 Alkoxycarbonyl, C2-C6-Alkylaminocarbonyl or C3-C8 Dialkylaminocarbonyl, (c) at least one of R 6>, R 1> 1> and R 1> 2> is present and (d) R 1> 2> is not present, then R 6> or R 1> 1> is not C2-C6-Alkylcarbonyl, C2-C6 Alkoxycarbonyl, C2-C6-Alkylaminocarbonyl or C3-C8-Dialkylaminocarbonyl. Full definitions are given in the Definitions Field (Full Definitions). ACTIVITY : Insecticide; Acaricide; Nematocide. No biological data is given. MECHANISM OF ACTION : None given.