baber/WOPTO huggingface dataset:
Patent UA-73152-C2 (UA)
Title: Condensed azepins as agonists of vasopressin
IPC: C07D495/04
Filed: 2001-01-04
Abstract: This invention provides novel compounds according to general formula (1) wherein A is a bicyclic or tricyclic azepine derivative, V1 and V2 are both H, OMe or F, or one of V1 and V2 is Br, Cl, F, OH, OMe, OBn, OPh, O-acyl, N3, NH2, NHBn or NH-acyl and the other is H, or V1 and V2 together are =O, -O(CH2)pO- or -S(CH2)pS-; W1 is either O or S; X1 and X2 are both H, or together are =O or =S; Y is OR5 or NR6R7; R1, R2, R3 and R4 are independently selected from H, lower alkyl, lower alkyloxy, F, Cl and Br; R5 is selected from H and lower alkyl; R6 and R7 are independently selected from H and lower alkyl, or together are -(CH2)n-; n = 3, 4, 5, 6; and p is 2 or 3. The compounds are agonists at the vasopressin V2 receptor and are useful as antidiuretics and procoagulants. The invention further comprises pharmaceutical compositions incorporating these vasopressin agonists, which compositions are particularly useful in the treatment of central diabetes insipidus, nocturnal enuresis and nocturia.
Patent UA-77157-C2 (UA)
Title: Polypeptide anti-egfrviii scfvs with improved cytotoxicity and output, molecule of nucleic acid, that codes the indicated polypeptide, and method of cell destructure with using of this polypeptide
IPC: A61K47/48
Filed: 2001-02-23
Abstract: The invention provides antibodies for mutant form of the epidermal receptor growth factor known as EGFRvIII. This mutant is found only or, primarily, on the surface of hlyoblastomic cells, on cells of the mamma carcinoma, ovary, lungs. Antibodies that provided by the invention, have high affinnity for EGFRvIII and form the immunotoxins with 38 kD by the fragment of the A Pseudomonas exotoksine , in which the domain I, with higher cytotoxicity and output was deleted, than antibodyies that known from a level of technique, including scFv, that is marking as MR1. In particular, the invention provides antibody designated as MR1-1, that has mutations in CDR3 VH and VL of circuits for providing theantibodies with especially improved cytotoxicity. The invention provides also the additional antibodyies, in which MR1 mutated into 2 VH or VL, or to both, for the best, than for starting MR1 antibody, binding with EGFRvIII.
Patent UA-79983-C2 (UA)
Title: Telescopc support of external fixation apparatus
Inventor: KOSTIUK ANATOLII NYKYFOROVYCH
IPC: A61B17/66
Filed: 2005-03-18
Abstract: The invention relates to orthopedics and traumatology. The telescopic support of external fixation apparatus comprises fixed component, in which one end rigidly anchors the core, and movable component, arranged on the core and connected to it with the opportunity of linear shift and hrigidly anchored relatively to angular displacements. The screw, entered into it by its one end, its connected with a threading bushing disposed in the core with the opportunity of inline offset, and opposite one comprises handwheel, fixed to movable component with the opportunity of rotation around its axis. Fixed component and core comprise through threaded hole for hold-down screw in a place of their connection. The supporting element allows to perform dosed or manual compression and distraction of bones without additional mechanical facilities. The duration of compression and distraction processes is shortened, and the preparation for surgery is simplified.
Patent UA-90448-C2 (UA)
Title: Method for manufacturing electrodes with a low contact resistance for batteries and capacitors with a double electric layer
Inventor: MALETIN YURII ANDRIIOVYCH
IPC: H01M4/02
Filed: 2005-06-25
Abstract: A manufacturing method for electrodes having a low contact resistance for batteries and capacitors with double electric layer relates to electric engineering, in particular to manufacturing electrodes with low contact resistance for batteries and capacitors with double electric layer between electrode material and metal current collector that may be used in pulse current sources. A set problem is achieved by manufacturing electrodes with comprise a metallic current collector and a polarization electrode. Particles of high conductive carbon material are fused into a surface of the metallic current collector maid of metal foil. Particles of carbon material having high conductivity, for example graphite, are fused into in metal foil of current collector using spark and arc methods. The technical result is decreasing of electrode contact resistance that provides high operating parameters of energy-storage apparatus, as well as simplicity and low price.
Patent UA-78651-C2 (UA)
Title: Protective method for carbonaceous products or half-finished products from corrosion
Inventor: SYVOHRYVOV YURII HAVRYLOVYCH
IPC: C25B11/00
Filed: 2005-12-12
Abstract: A protective method for carbonaceous products or half-finished products from corrosion at high temperatures involves impregnation in the impregnation furnace by immersion of them into the impregnation melt on the base of derivatives of phosphoric acid and phosphor containing salts of alkaline metals, formation of vaporous atmosphere, at that the vaporous atmosphere is formed from the evaporation products of impregnation melt of the impregnation furnace, and half-finished products or products which are subjected to impregnation are maintained in it, before their immersion into the impregnation melt, and the maintaining of half-finished products or products in the vaporous atmosphere is carried out in the additional chamber, which is connected to the impregnation furnace with air channels, through which from the impregnation furnace to the chamber the evaporation products of impregnation melt are supplied, at that before the supplying of the evaporation products of impregnation melt into the additional chamber, the half-finished products or products which are subjected to impregnation are disposed among the cooled in it impregnated half-finished products or products.
Patent UA-82015-C2 (UA)
Title: Device for transporting and cleaning tuberous roots
Inventor: BULHAKOV VOLODYMYR MYKHAILOVYCH
IPC: A01D33/08
Filed: 2006-10-10
Abstract: A device for transporting and cleaning tuberous roots consists of a frame, a feed conveyer, a baffle brush, a cleaner, as well as of an unloading conveyer, arranged in series, is proposed. The cleaner is made as a cleaning unit installed as an inclined one. The rollers of the cleaning unit, which are arranged longitudinally, from above comprise an activator as two drive spherical disks arranged at the same distances, at angle to the cleaning surface of the unit and at the same time at angle to each other. The disks form a gap between each other and have counter-rotational movement.
Patent UA-86076-C2 (UA)
Title: Process for the preparation of composite organo-mineral fertilizer and the process for the treatment of seeds and plant vegetative mass by composite organo-mineral fertilizer
Inventor: DULNIEV PETRO HEORHIIOVYCH
IPC: C05D9/00
Filed: 2007-01-31
Abstract: A process for the preparation of composite organo-mineral fertilizer in which carbamide, vermicompost, milk whey, phytohormone, humate of alkali metal or ammonium, potassium nitrate, potassium phosphate, ammonium phosphate, mixture of polyoxyethylene glycols and microelements are mixed, and the treatment process of seeds and plant vegetative mass by composite organo-mineral fertilizer.
Patent UA-91685-C2 (UA)
Title: Apparatus (variants) and process for cooling and de-steaming hot evaporated calcined stucco
Inventor: BOLIND MICHAEL L
IPC: F25D23/12
Filed: 2005-05-19
Abstract: The present invention is an apparatus and process for cooling and de-steaming hot calcined stucco used in the production of gypsum boards or bagged plaster. The apparatus is fluid bed stucco cooler and comprises a cooler housing having a plenum having a stucco inlet and stucco outlet. The stucco cooler includes a rotating disk in the plenum. The rotating disk includes nozzle for spraying fluid, and is attached to a rotable shaft extending from the side of the cooler also includes a fluidization pad and agitator to help to mix the air and the stucco powder to insure fluidization, prevent channeling, and prevent the stucco powder from building up on the various components. The air also forces steam from the hot calcined stucco out through an air outlet located at the top of the stucco cooler, thereby de-steaming the stucco. The stucco flows through the plenum and passes over the cooling coils, thereby cooling the stucco as it reaches the stucco outlet.
Patent UA-92909-C2 (UA)
Title: Method for managing machine for manufacturing tobacco products
Inventor: DRAGHETTI FIORENZO
IPC: A24C5/00
Filed: 2006-04-18
Abstract: A method of managing a machine for manufacturing tobacco products (2) includes the steps of monitoring the operation of single devices and/or units making up the machine (3; 4), and supplying error signals (48) to a master control unit (46) to indicate faults or malfunctions in any of the devices; on receiving an error signal (48), the control unit (46) responds automatically by stopping the machine (3; 4), activating a step in which obstructions are removed and foreign matter cleared from the faulty or malfunctioning device, and finally, with normal operating conditions restored, restarting the machine (3; 4).
Patent UA-83453-C2 (UA)
Title: Unit for transporting and cleaning tuberous roots
Inventor: BULHAKOV VOLODYMYR MYKHAILOVYCH
IPC: A01D33/08
Filed: 2007-12-19
Abstract: A unit for transporting and cleaning tuberous roots consists of a frame, a feed conveyer, a baffle brush, a cleaner and also of an unloading conveyer. The cleaner is made as a single-hollow hyperboloid connected to a rotary actuator made by round concentric rods arranged with gaps to each other. The lower outlet of the hyperboloid has inside a hollow projection of a conical shape with the upper plane which is also formed by round radial rods arranged with gaps to each other, above which on the upper plane thereof a double-blade beater is disposed, it is placed at the end of a projecting driving shaft arranged in the lower part. In the upper part inside the cleaner a driving activator as two elastic blades fixed at the end of the projecting driving shaft arranged from above is mounted. Under the lower outlet of the single-hollow hyperboloid an immovable accumulator of a conical shape internal surface thereof has on the conical part console short elastic fingers fixed is brought.
Patent UA-93906-C2 (UA)
Title: Modified foamable and foamed materials and a method of obtaining thereof
Inventor: STACHURA DARIUSZ
IPC: C08J9/12
Filed: 2007-05-07
Abstract: The present invention relates to modified foamable and foamed materials which, in addition to polystyrene, carbonic acid diamide and stilbene derivatives, contain also a dispersion stabilizer in the form of carboxymethylcellulose sodium; a dispersing agent in the form of a water solution of cationic surface-active agent, an endogenous and exogeneous fires inhibitor in the form of di-nitrosopentamethylenetetramine and a solution of water silicic acid sol. The present invention also relates to a method of obtaining foamable and foamed materials, in particular polystyrene which the method reduces considerably, amongst other things, the risk of exposure to chemicals emitted during the processes of pyrolysis of these materials.
Patent UA-89932-C2 (UA)
Title: Method for healing injuries on trees
Inventor: DULNIEV PETRO HEORHIIOVYCH
IPC: A01N3/00
Filed: 2009-05-25
Abstract: The invention relates to agriculture, especially to horticulture, in particular to a method for repair of injuries on trees with a garden paste which improves regenerative processes while repairing injuries up to 49% as against sampling.
Patent UA-95328-C2 (UA)
Title: Method for coating metal substrate and coated substrate
Inventor: MCMURDIE NEIL D
IPC: C09D5/08
Filed: 2007-10-12
Abstract: Disclosed are methods for coating a metal substrate with a yttrium-containing coating, including ferrous substrates, such as cold roiled steel and electrogalvanized steel. Also disclosed are coated substrates produced thereby.
Patent UA-94141-C2 (UA)
Title: Method for protecting oilseed rape, herbicidal composition for protecting oilseed rape and method for controlling weeds
Inventor: LOCKETT JOHN
IPC: A01N47/22
Filed: 2007-12-20
Abstract: The invention provides use of, or a method of using, a composition comprising phenmedipham as a herbicide in the protection of oilseed rape. Compositions comprising phenmedipham are also provided.
Patent UA-91474-C2 (UA)
Title: method for treatment of metal sheets
Inventor: HANENBERG LOTHAR
IPC: B21B1/46
Filed: 2008-02-05
Abstract: The invention relates to a method for the treatment of metal sheets that are rolled in a roll stand to their final dimensions, subsequently cooled online, straightened, and heat-treated for homogenization and influencing the microstnicture. According to the invention, in order to improve the heat treatment options online, the heat treatment occurs online but decoupled from the prior cooling and straightening processes, for which purpose, taking into account the speed of the metal sheet as it exits the final machining station located upstream, the point in time at which the heat treatment begins is selected such that the metal sheet has completely left said final machining station before the metal sheet is subjected to heat treatment.
Patent UA-96650-C2 (UA)
Title: Push-pull balanced current amplifier
Inventor: AZAROV OLEKSII DMYTROVYCH
IPC: H03K5/22
Filed: 2010-02-25
Abstract: A pull-push balanced current amplifier relates to pulse technique and can be used in analog-to-digital converters and digital instruments. The current amplifier comprises first and second current sources, a feedback resistor, positive and negative buses, zero bus and six transistors. In addition, first and second current compensators, bi-directional current reflector, first and second current switchers are incorporated. All said elements are interconnected in an appropriate manner. In the amplifier operation accuracy is increased due to fitting coefficients of current amplification of upper and low stages of amplifier cascades, also linearity improves due to automation of DC balancing process of amplification stages operation points that extends area of utilizations in different devices of pulse and computation engineering.
Patent UA-98372-C2 (UA)
Title: Process for titanium trifluoride production
Inventor: PRETORIUS GERARD
IPC: C01G23/02
Filed: 2008-12-29
Abstract: A method for the production of titanium trifluoride from a titanium-containing material includes the steps of producing a fluoride solution of Ti(IV) from the titanium-containing material and reducing the Ti(IV) in the solution with a transition metal or an alloy of the transition metal. The transition metal is selected from manganese, iron, cobalt, nickel and zinc. An ammonium containing salt and either ammonia or ammonium fluoride are added to the resulting solution containing Ti(III) to produce a precipitate, and the precipitate is pyrolysed to produce titanium trifluoride.
Patent UA-101010-C2 (UA)
Title: 6.7-dialkoxy ouinazoline derivatives useful for treatment of cancer related disorders
Inventor: JYOTHI PRASAD RAMANADHAM
IPC: C07D239/94
Filed: 2008-01-18
Abstract: In view of the great potential the quinazoline class of compounds offer, we started the synthesis and screening of a large number of new chemical entities with novel structural features. It has been surprisingly and unexpectedly found that quinazolines having 3-ethynyl anilino group at the 4th position and specifically substituted alkoxy groups in the 6 and 7 positions, impart much enhanced and special anti-proliferative properties when compared to other prominent members of the quinazoline class of drugs. Also, surprisingly the compounds of this invention are much less toxic and the safety profile is exceedingly beneficial for therapeutic applications. The novel chemical entities described in this invention are designated by the general structure (I) and have not been synthesized earlier nor investigated for their therapeutic benefits and safety profile. Compound (I) is NRC-2694, when structure (A)., (I), (A)
Patent UA-99757-C2 (UA)
Title: Method (variants) and apparatus (variants) for supporting data transmission in multi-carrier communication system
Inventor: ZHANG DANLU
IPC: H04W72/00
Filed: 2009-02-27
Abstract: Techniques for supporting data transmission on multiple carriers in a wireless communication system are described, A user equipment (UE) may determine available transmit power for data transmission on multiple carriers. The UE may distribute the available transmit power Lo multiple carriers (e.g., using uniform power distribution, greedy filling, water filling, etc.) to obtain allocated transmit power for data for each carrier. The UE may send at least one resource request with information indicative of the allocated transmit power for each of the multiple carriers to a Node B. The UE may receive at least one resource grant with information indicative of granted transmit power for each of at least one carrier, which may be all or a subset of the multiple carriers. The UE may send data on the at least one carrier and may limit its transmit power for each carrier to the granted transmit power for that carrier.
Patent UA-97210-C2 (UA)
Title: Method for switching without any interruption between winding taps on a tap-changing transformer
Inventor: BRUECKL OLIVER
IPC: H03K17/68
Filed: 2008-08-27
Abstract: The invention relates to a method for switching without any interruption between two winding taps (tap n, tap n+1) of a tap-changing transformer, wherein each of the two winding taps is connected to the common load output line via in each case one mechanical switch (D) and a series circuit, arranged in series thereto, comprising two IGBTs (I, I) which are switched in opposite directions.
Patent UA-101066-C2 (UA)
Title: Process for electrokinetic decontamination of solid porous medium
Inventor: CUER FREDERIC
IPC: E04G23/02
Filed: 2009-10-01
Abstract: The invention relates to a process for the electrokinetic decontamination of a porous solid medium, which comprises: a) the extraction of the contaminating species present in this solid medium into an electrolyte that is in the form of an essentially inorganic gel, this extraction being obtained by applying an electrical current between two electrodes positioned at the surface of and/or within the solid medium, the contact of at least one of these electrodes with said solid medium being provided by a layer of said gel, b) the drying of the gel containing the contaminating species thus extracted until a dry residue is obtained which breaks up, and c) the elimination of the dry residue thus obtained from said solid medium. Applications: decontamination of materials having a cement matrix, especially in the context of dismantling military or industrial, in particular nuclear, installations or of rehabilitating installations liable to have been contaminated by environmentally hazardous or radiological chemical species; remediation of geological soils, sediments and sludges.
Patent UA-110193-C2 (UA)
Inventor: LEIFELD SABINE
IPC: B65D83/04
Filed: 2009-11-14
Abstract: Група винаходів характеризує картридж та дозатор лікарських засобів, а також застосування згаданих елементів. Відповідно до першого аспекту винаходу картридж (900), який вставляється у дозатор (1) лікарських засобів для порцій (Т) лікарського засобу з твердої речовини й виконаний з ресивером для розміщення порцій (Т) лікарського засобу, при цьому картридж (900) має роз'єднувальний пристрій (910), який виконаний для видачі заданих порцій (Т) лікарського засобу, і який містить виконаний з можливістю переміщення пристрій (940) для відділення заданої порції (Т) лікарського засобу з ресивера й для видачі з дозатора (1) лікарських засобів, при цьому роз'єднувальний пристрій (910) виконаний для встановлення кінематичного зв'язку з передбаченим у дозаторі (1) лікарських засобів пристроєм (14, 220, 224, 226; 15, 210, 230) керування для роз'єднувального пристрою (910), і при цьому порції лікарського засобу (Т) при роз'єднанні, а також їх видачі або ж звільненні з дозатора, не доторкаються до дозатора або його деталей. Другий аспект винаходу також стосується дозатора (1) лікарських засобів для порцій (Т) лікарського засобу з твердої речовини, який виконаний для розміщення змінного картриджа (900), при цьому картридж (900) має ресивер для порцій (Т) лікарського засобу, а також роз'єднувальний пристрій для видачі заданих порцій (Т) лікарського засобу, при цьому дозатор (1) лікарських засобів має щонайменше один пристрій (14, 220, 224, 226; 15, 210, 230) керування для роз'єднувального пристрою (910), а також засоби для встановлення кінематичного зв'язку між щонайменше одним пристроєм керування і виконаним із можливістю переміщення пристроєм (940) на роз'єднувальному пристрої (910) й сл
Patent UA-107706-C2 (UA)
Inventor: BRUNCKO MILAN
IPC: C07D471/04
Filed: 2010-11-22
Abstract: Розкриті сполуки, які інгібують активність антиапоптичних Bcl-2-білків, композиції, що містять такі сполуки, і способи лікування захворювань, у процесі яких експресується антиапоптичний Bcl-2-білок.
Patent UA-110236-C2 (UA)
Inventor: MAGDINA ROMAN
IPC: C09D7/63
Filed: 2012-07-02
Abstract: Вогнестійкий матеріал для покриттів ADINA. Вогнестійкий матеріал для покриттів ADINA, що містить поліфосфат амонію в кількості від 5 до 50 % мас./мас., пентаеритрит - в кількості від 6 до 33 % мас./мас., меламін - в кількості від 4 до 22 % мас./мас., зв'язуюче на основі дисперсії полівінілакрилату - в кількості від 10 до 16,3 % мас./мас., пластифікатор на основі діізононілфталату - в кількості від 2,3 до 3,5 % мас./мас., тальк - в кількості від 3 до 10 % мас./мас., стабілізатор (консервант) на основі 4-хлор-3-метилфенолу - в кількості від 0,15 до 0,25 % мас./мас. і воду - в кількості від 13,5 до 17 % мас./мас.
Patent UA-111761-C2 (UA)
Title: 2',4'-дифтор-2'-метилзаміщені нуклеозидні похідні як інгібітори реплікації phk вірусу гепатиту c
IPC: C07H19/06
Filed: 2012-12-17
Abstract: Даний винахід стосується сполук Формули І:I.Також розкриті фармацевтичні композиції, що містять сполуки Формули І, способи застосування сполук Формули І та/або композицій, що містять сполуки Формули І, для лікування ВГС.
Patent UA-112578-C2 (UA)
Title: Амортизаційно-поглинаючий пристрій
IPC: F16F15/02
Filed: 2014-10-31
Abstract: Винахід належить до деталей машин і підйомно-транспортних машин. Амортизаційно-поглинаючий пристрій містить корпус, в якому з можливістю переміщення встановлений поршень зі штоком, який сполучений з корпусом пружно-демпфуючими елементами, якими є канати. Кожен з останніх закріплений одним кінцем у корпусі, а іншим - у поршні, один із кінців кожного каната закріплений жорстко, а інший - рухомо, та має можливість повороту за рахунок кінематичного зв'язку між рухомо закріпленим кінцем каната та елементом амортизаційно-поглинаючого пристрою, в якому жорстко закріплений протилежний кінець каната. Технічним результатом є підвищення надійності та демпфуючої здатності.
Patent UA-115880-C2 (UA)
Title: Herbicidal compostions comprising 4-amino-3-chloro-5-fluoro-6-(4-chloro-2-fluoro-3-methoxyphenyl) pyridine-2-carboxylic acid or a derivative thereof and bromobutide, daimuron, oxaziclomefone or pyributicarb
Inventor: YERKES CARLA N
IPC: A01P13/00
Filed: 2013-07-19
Abstract: Provided herein are synergistic hurbicidal compositions containing (a) a compound of formula (I): or an agriculturally acceptable salt or ester thereof and (b) bromobutide, daimuron, oxaziclomefone or pyributicarb, or an agriculturally acceptable salt thereof. The compositions and methods provide control of undesirable vegetation, e.g., in direct-seeded, water-seeded and trans-planted rice, cereals, wheat, barley, oats, rye, sorghum, corn or maize, sugarcane, sunflower, oilseed rape, canola, sugar beet, soy-bean, cotton, pineapple, pastures, grasslands, rangelands, fallowland, turf, tree and vine orchards, aquatics, plantation crops, vegetables, industrial vegetation management (IVM) or rights of way (ROW).