baber/WOPTO huggingface dataset:
Patent CZ-292169-B6 (CZ)
Title: Acyclic nucleoside derivatives, process of their preparation and pharmaceutical compositions in which they are comprised
Inventor: ENGELHARDT PER
IPC: C07D473/18
Filed: 1997-02-14
Abstract: In the present invention there are disclosed acyclic nucleoside derivatives of the general formula I, in which one of the Ri1 and Ri2 substituents represents the group -C(O)CH(CH(CHi3)i2)NHi2 or the group -C(O)CH(CH(CHi3)CHi2CHi3)NHi2 and the other of the Ri1 a Ri2 substituents represents  -C(O)alkyl having 3 to 21 carbon atoms or a monounsaturated alkenyl, being optionally substituted with  one to five groups that are selected from the group comprising a hydroxyl group, alkyl containing 1 to 6 carbon atoms, alkoxy containing 1 to 6 carbon atoms, alkoxyalkyl containing 1 to 6 carbon atoms in both the alkoxy and alkyl moieties, alkanoyl containing 1 to 6 carbon atoms, an amino group, a halogen atom, a cyano group, an azido group, an oxo group, a mercapto group and a nitro group, and Ri3 represents an OH group or a hydrogen atom; as well as pharmaceutically acceptable salts thereof that are effective as antiviral agents against herpes and retroviral infections. These agents exhibit increased biological availability. Further claimed are pharmaceutical compositions containing the compound of the general formula I, their use, and process of their preparation.
Patent CZ-289069-B6 (CZ)
Title: Medicament for treating incontinence
Inventor: THOR KARL BRUCE
IPC: A61P13/02
Filed: 1994-11-23
Abstract: The present invention relates to the use of 3-aryloxypropanamine derivative or a pharmaceutically acceptable acid addition salt thereof for preparing a pharmaceutical preparation intended for treating urine incontinence.
Patent SK-281329-B6 (SK)
Inventor: KEPPLINGER WERNER
IPC: C21B13/00
Filed: 1993-10-21
Abstract: Spôsob výroby spočíva v tom, že v tavnom splyňovacom pásme (I až IV) vytvorený redukčný plyn sa sčasti privádza do redukčného pásma priamo - a to bez čistenia - na vytvorenie vírivej vrstvy (18) a z ďalšej časti vytvorenej väčšími časticami pevnej látky sa privádza po čistení v horúcej cyklóne (25) redukčného pásma do lôžka vytvoreného v jeho spodnej časti. V zodpovedajúcom zariadení plynové potrubie (17) na redukčný plyn ústi prvým odbočovacím potrubím cez zariadenie (25) na čistenie plynu do spodnej oblasti redukčného reaktora (8) a z plynového potrubia (17) pred zariadením na čistenie plynu vychádza druhé odbočovacie potrubie, ktoré ústi do vyššie ležiacej oblasti redukčného reaktora (8).ŕ
Patent SK-279989-B6 (SK)
Title: Method and device for the production of a composite thread
Inventor: RONCATO GIORDANO
IPC: B29C70/16
Filed: 1993-11-17
Abstract: A composite thread of glass and of organic material wherein continuous filaments of thermoplastic organic material are mixed in the form of a sheet with a bundle or sheet of glass filaments, with the speed of the thermoplastic filaments during their penetration into the bundle or sheet of glass filaments being greater than the speed of drawing of the glass filaments. The device comprises a die (1) for producing continuous glass filaments and a drawing head (7) for issuing continuous thermoplastic filaments and common means (3, 16) for assembling together the said continuous filaments and drawing the composite thread (6). The drawing head (7) is positioned next to a drum-type drawing device (11) with a variable speed and to a device (13) ensuring incorporation and integration of the said continuous thermoplastic filaments (5) into the sheet of glass filaments or into the bundle of the glass filaments (2).
Patent SK-281934-B6 (SK)
Inventor: JEGHAM SAMIR
IPC: A61K31/427
Filed: 1996-05-28
Abstract: Opísané 5-(hydroxymetyl)oxazolidin-2-óny sú substituované indazolovým, benzizoxazolovým alebo benzizotiazolovým kruhom a majú všeobecný vzorec (I), v ktorom X znamená atóm kyslíka, atóm síry alebo skupinu NR, kde R znamená atóm vodíka alebo priamu alebo rozvetvenú alkylovú skupinu obsahujúcu 1 až 4 atómy uhlíka, R1 znamená atóm vodíka alebo metylovú skupinu a R2 znamená buď i) skupinu R3O, v ktorej R3 znamená atóm vodíka alebo benzylovú skupinu prípadne substituovanú atómom halogénu alebo nitroskupinou alebo metyléndioxyskupinou, alebo metoxyetylovú, butylovú, 4,4,4-trifluórbutylovú, 4,4,4-trifluór-3-hydroxybutylovú alebo 4,4,4-trifluórbut-2-enylovú skupinu, alebo ii) skupinu -CH=CH-R4 alebo skupinu -CH2-CH2-R4, v ktorej R4 znamená atóm vodíka alebo fenylovú, 3,3,3-trifluórpropylovú alebo 3,3,3-trifluór-2-hydroxypropylovú skupinu. Opísaný je tiež spôsob prípravy uvedených zlúčenín a ich použitie v medicíne.ŕ
Patent SK-279886-B6 (SK)
Title: Body structure for railway vehicles
Inventor: HANNI ROLAND
IPC: B62D31/02
Filed: 1991-07-04
Abstract: The wagon body structure comprises a superstructure (2) with extruded profiles, releasably connected to one another by mechanical means and consisting of an aluminium alloy, and a substructure (1). The substructure (1) consists of longitudinal supports (3, 4) and transverse supports (5), which are releasably connected to one another and to the superstructure (2) by means of screwable corner connectors (13, 24, 25), and consist of an extruded aluminium alloy. The longitudinal supports (3, 4) and at least some of the transverse supports (5) of the substructure (1) and posts (6) and upper flanges (7) of the superstructure (2) have on at least one side two undercut longitudinal grooves (12, 15) for receiving nuts, preferably rotatable clamping plates, or clamping straps. In combination with the superstructure (2), said substructure (1) is of inherently stable construction.
Patent SK-278559-B6 (SK)
Title: A method of continual production of block polymer of propylene and ethylene
Inventor: CHIBA HIROMASA
IPC: C08F210/06
Filed: 1986-11-17
Abstract: This patent describes the continual procedure closed to the production of a propylene and ethylene block co-polymer with the well balanced features, something like the shock resistance, workability, and so on, while a good gain is reached, and two polymerisation stages together with catalyst are applied, to control the space arrangement of the result polymer containing a hard component with titan content and organic aluminium compound, while in the first stage, two or more polymerisation vessels are supplied by polypropylene and they are ordered sequentially, however 60 up to 95 weight percent of the total final product is created, in the second stage glycoether is added to reaction mixture produced in the first polymerisation stage and two or more polymerisation vessels are supplied with ethylene and the (ethylene + propylene) ratio is 0,1 up to 1,0; while 5 up to 40 weight percent closed to all of the polymerisation product quantity is created.
Patent CZ-303597-B6 (CZ)
Title: Device for exposing polymeric and damp-proof materials to radon
Inventor: JIRANEK MARTIN
IPC: G01N33/38
Filed: 2011-12-13
Abstract: In the present invention, there is disclosed a device formed by an exposing chamber (1) made of a non-corroding material having radon diffusion coefficient lower than 1.10e-12 .me2/s provided with a tightly closable lid (2). S removable structure (3) for attachment of samples (4) is disposed below the lid (2) and parallel therewith. The area above the samples (4) is connected to the space below the samples (4) through the mediation of two circuits. A source circuit is formed by a first closable and regulating valve (5.1) having its outlet into an exposure chamber (1) via the lid (2) and interconnected via a first through-flow pump (7.1) and a first radon source (6) with a second closable and regulating valve (5.2) being lead out into the exposure chamber (1) in the space below the samples (4). In case of manual monitoring, the measuring circuit is formed by a first closable valve (10.1) for taking samples of air in order to determine radon volume activity within a self-contained measuring device, wherein said first closable valve (10.1) is lead out into the exposure chamber (1) via the lid (2). In case of automatic monitoring of the radon volume activity, the first closable valve (10.1) is connected via a radon continuous monitor (8) and via a second through-flow pump (7.2) with a second closable valve (10.2) being lead out into the exposure chamber (1) in the space below the samples (4).
Patent CZ-304174-B6 (CZ)
Title: Composition for gradual release of nicotinic acid and/or nicotinamide
Inventor: HROMADKA ROBERT
IPC: A61K9/51
Filed: 2012-12-19
Abstract: In the present invention, there is disclosed a composition consisting of biologically degradable nanofibers and/or microfibers of one or more polymers being selected from the group consisting of cellulose or chitosan or polyvinyl alcohol or gelatin or collagen or hyaluronic acid or polylactic acid or chemical derivatives of these polymers, whereby the nanofibers and/or microfibers also contain 2 to 90 percent by weight of nicotinic acid and/or nicotinamide. The diameter of the biologically degradable nanofibers and/or microfibers is in the range of 40 to 1500 nm and the nanofibers and/or microfibers are usually cross linked. There is also disclosed the use of the above-described composition in drug forms, food supplements or functional foodstuffs.
Patent CZ-309798-B6 (CZ)
Title: A method of preparation of biological medicinal product based on perinatal tissue, a powdered material and its use
Inventor: Forostyak Serhiy
IPC: A61K35/51
Filed: 2022-03-15
Abstract: Name of the invention: A method of preparation of biological medicinal product based on perinatal tissueThe solution submitted provides a method of preparing a biological medicinal product based on perinatal tissue, which includes the following steps:a) cleaning of the input perinatal tissue and optionally its resection into parts whose dimension does not exceed 50 mm in any direction; wherein the tissue is allowed to dry for at least 15 minutes after cleaning;b) cryogenic grinding of the perinatal tissue in resealable surgical steel capsules with surgical steel grinding balls;c) homogenization of the ground perinatal tissue using an ultrasonic homogenizer;d) filling of the ground and homogenized perinatal tissue into the primary packaging while constantly stirring;e) lyophilization of the ground and homogenized perinatal tissue in the primary package;f) sterilization of the lyophilized ground and homogenized perinatal tissue in the primary package using gamma radiation at a dose of 5 to 20 kGy;wherein the entire process is carried out without the presence of antibiotics and antifungals.
Patent SK-283899-B6 (SK)
Title: Improved process for antiparasitic agent
Inventor: WALSHE NIGEL DEREK ARTHUR
IPC: C07H19/01
Filed: 1998-07-23
Abstract: An improved process for the preparation of the antiparasitic compound 25-cyclohexyl-22,23-dihydro-5-hydroxyiminoavermectin B1 monosaccharide from doramectine and intermediates therefor and crystalline solvates thereof.
Patent SK-284793-B6 (SK)
Title: Jacketed projectile with a hard core
Inventor: HUG CARL
IPC: F42B12/80
Filed: 1998-08-24
Abstract: Jacketed projectile (100), comprising a tungsten carbide hard core (5) on the front side and a centered, interlocking soft-core (8) placed on the hard core (5). A closed air space (6) is located between the front area (5a) of the hard core (5) and the tip of the projectile (4). This projectile configuration provides a very high penetration potential and good dynamic and ballistic properties, enabling the inventive projectiles in so far that are suitable for shooters at ball firing, for police snipers, especially to hit targets located behind a glass.
Patent SK-286216-B6 (SK)
Title: A screening arrangement
Inventor: RITZ ANDERS
IPC: E06B9/00
Filed: 1999-11-11
Abstract: The screening arrangement comprises a flexible length of screening material, a tubular rod (13), along which one end of the length is fastened, and around which the length can be wound, and a driving device for moving the length towards or away from the tubular rod. The driving device comprises an input shaft driving a driver member in driving engagement with the length. The tubular rod (13) is connected with one end of a torsion spring (35), the other end of which is connected with a drive shaft (31) driven by the input shaft in such a manner that in connection with rewinding and unwinding, the drive shaft has the same direction of rotation as the tubular rod (13).
Patent SK-287762-B6 (SK)
Title: Use of aplidine in preparation of pharmaceutical composition for treating cancer
Inventor: FAIRCLOTH GLYNN THOMAS
IPC: A61P35/00
Filed: 2000-11-15
Abstract: It is described the use of aplidine in the preparation of a pharmaceutical composition for treating cancer, which aplidine is in the form of an intravenous infusion. Next it is described the use of aplidine in combination with a skeletal muscle protector, which is preferably carnitine, for treating cancer.
Patent SK-285372-B6 (SK)
Title: Method of producing cyclene
Inventor: PLATZEK JOHANNES
IPC: C07D257/02
Filed: 1999-11-17
Abstract: Process for the production of cyclene characterized in that in a single-pot process, triethylenetetramine is reacted with 40 % glyoxal at 20 °C to 80 °C in a polar protic solvent within 4 to 40 hours; after the solvent has been removed the intermediary tricyclic compound that is thus formed is alkylated to the two secondary amine-nitrogen's atoms with a 1,2-difunctionalized alkylating agent X(CH2)2X, in which X stands for a nucleofuge group, in a polar aprotic solvent, optionally in the presence of an auxiliary base within 2 to 24 hours; after the solvent has been removed the thus obtained condensation product is treated with hydrazine hydrate in a polar protic solvent at a pH of 3 to 6 within 12 to 48 hours at reflux temperature; then the cyclene is released from the cyclene salt by adding a base and after the reaction solution is evaporated to the dry state, is it isolated.
Patent CZ-299117-B6 (CZ)
Title: Two-component product based on phenolic resin
Inventor: WEBER FRANCK
IPC: C09K17/36
Filed: 2000-11-24
Abstract: In the present invention, there is disclosed a two-component product based on phenolic resin comprising resol-based resin and sulfonic acid-based catalyst being intended for soil consolidation by injection. The present invention is characterized in that the invented two-component product contains as ingredients a surfactant or a combination of surfactants, resorcin, novolac resin or sulfonated novolac resin and/or a dispersion of preliminary crosslinked resol. These ingredients are added to the resinous component or to catalytic component.
Patent CZ-291644-B6 (CZ)
Title: Orientation and navigation system
Inventor: SEDLAR VLADIMIR ING
IPC: G01C21/04
Filed: 2001-06-12
Abstract: The present invention relates to orientation and navigation method comprising creation of a set of geographic maps and this set is stored in a preset computer. Based on sign-on data communication of a user mobile terminal to mutually interconnected data base stations, a geographic position of the user mobile terminal is determined, and/or based on the communication of the user geographic position a corresponding map is selected according to place where the user of the mobile terminal is located. Subsequently, based on the request of mobile terminal user for the object to be searched and given in the form of a data signal caught by the network of the base stations from the mobile terminal with a viewer, a visible stationary object is determined from the user view, and its position with respect to the mobile terminal is calculated. The mobile terminal user is then requested to take the mobile terminal antenna bearing to said visible object and a data reply in the form of an oriented cardinal point rose, respectively an arrow showing the direction toward the object to be searched is created, whereby said arrow forms with the mobile terminal display, respectively the mobile terminal antenna an angle corresponding to the angle formed between the visible object and the object to be searched. From the user view the visible stationary object can be the sun, the moon, a church tower, or other objects that can be easily identified by the user. The proposed orientation and navigation system comprises a mobile terminal (2) with a viewer and mutually interconnected data base stations (1) that are connected through the mediation of a backbone network (3) with a central (4) decoding all the data and divides them into voice data and solely data. The central (4) is interconnected via an access gate (5) with a preset computer (6). The preset computer (6) comprises a first block (7) for determining geographical position of the user of a mobile terminal (2) with a viewer, a second block (8) for calculating the position of a visible stationary object as viewed by the user, a third block (9) containing geographical maps and a fourth block (10). Based on data of the first block (7), the second block (8) the third block (9) and the mobile terminal (2), the fourth block (10) makes a data reply to a data signal received from the mobile terminal in the form of an oriented cardinal point rose, respectively an arrow displayed on the mobile terminal (2) display and showing the direction toward the object to be searched.
Patent CZ-305763-B6 (CZ)
Title: Capacitor powder
Inventor: REICHERT KARLHEINZ
IPC: H01G9/052
Filed: 2001-06-08
Abstract: The present invention relates to a vanadium-containing niobium-based powder, process for its preparation, anode obtainable from such a powder and a capacitor with anode obtained from the niobium-based powder and with capacitance that is independent on overvoltage.
Patent CZ-298566-B6 (CZ)
Title: Aerodynamic device wing with swirl grooves
Inventor: VACEK JAN
IPC: F03D80/00
Filed: 2003-08-15
Abstract: The present invention relates to a wing (1) having at least on its one side (3, 4) a recessed groove (2) with a profile consisting of exponential spiral (13) that passes in a circular bow (14) back to the wing (1) surface. One or several of said grooves (2) are situated predominantly in the first third of the wing (1) depth between the leading edge (5) and trailing edge (6) thereof. The grooves (2), forming a sharp edge (12) with the wing (1) surface, are usually straight and parallel to the leading edge (5). However, they can be beveled (7) or curved (8) in the direction to the trailing edge (6) at the wing (1) ends. Practical application of the present invention is in the construction of wings and propellers of airplanes, rotor blades of helicopters, wind turbine blades, ventilation device blades and generally to achieve smooth, circumfluence of aerodynamic bodies, i.e. without premature breakaway of streamlines from convex portions of their surfaces.
Patent SK-288187-B6 (SK)
Title: Method for attachment the balloon, especially by impessing, equipment for thereof
Inventor: MALCHO ZDENKO
IPC: B41F17/30
Filed: 2009-11-26
Abstract: Described the method for attachment and removal the balloons, especially in the multicoloured printing, wherein the balloon in the working position is not inflated. Described is a device for the attachment the balloon, which includes the pushing element (6), the last (1) with the peripheral binding (2) and the tapered retaining surface (4).
Patent EP-1853428-B8 (EP)
Title: Appareil d'imagerie
Inventor: SHINGYOHUCHI MITSURU
IPC: B41J2/01
Filed: 2006-03-02
Granted: 2012-04-04
Abstract: L'invention concerne un appareil d'imagerie comprenant une tête d'évacuation de liquide conçue pour évacuer le liquide d'enregistrement sous forme d'au moins une gouttelette de liquide d'enregistrement; une unité de génération de forme d'onde pilote pour générer une forme d'onde pilote comprenant au moins deux signaux pilotes compris dans une période d'impression ; une unité pilote conçue pour entrer des données de ton, pour sélectionner un signal pilote pertinent dans la forme d'onde pilote, à l'aide d'un commutateur effectuant une communication marche/arrêt selon les données de ton, et pour appliquer le signal pilote sélectionné à la tête d'évacuation de liquide; et une unité de transmission conçue pour transmettre les données de ton à l'unité pilote, plusieurs fois pendant une période d'impression, ces données de ton étant configurées à une pluralité de bits par canal.
Patent EP-1882635-B8 (EP)
Inventor: DENNIS WAYNE RICE
IPC: G16H70/40
Filed: 2003-08-06
Granted: 2010-06-16
Abstract: Computer assisted systems, methods and mediums for filling one or more orders. One embodiment of the present invention is a system that includes an order consolidation station (215) configured to receive at least one bottle containing pills individually counted and/or at least one package containing pharmaceutical products without having been designated for any of the orders when the package was created and/or at least one literature pack optionally including patient specific information. The order consolidation station is further configured to combine automatically the received bottle and/or package and/or literature pack into a container to be sent to a recipient including, for example, mail order pharmacies, wholesalers and/or central fill dealers for subsequent distribution or sale including retailer distribution or sale. The bottle is specifically designated for the order, and the order generally includes at least one prescription for the package.
Patent BR-PI0612317-B8 (BR)
Title: benzimidazóis 2-substituídos, seu processo de preparação e composição farmacêutica
Inventor: Frédéric Marc Maurice Doublet
IPC: C07D235/30
Filed: 2006-06-20
Abstract: benzimidazóis 2-substituídos a presente invenção refere-se a inibidores de replicação de (rsv) de fórmula (i), (i) aos sais de adição e formas estereoquimicamente isoméricas desses inibidores, em que q é hidrgênio, c1-6alquila opcionalmente substituídas por um heterociclo ou q é c1-6alquila substituída tanto por -or4 quanto por um heterociclo; em que esse heterociclo é oxazolidina, tiazolidina, 1-oxo-tiomorfolinila, 1,1-dioxotiazolidina, morfolinia, tiomorfolinila, 1-oxo-tiomorfolinila, 1,1-dioxotiomorfolinila, hexaidroxazepina, hexaidro-tiazepina, 1-oxo-hexaidrotiazepina, 1,1-dioxo-hexaidrotiazepina, pirrolidina, piperidina, homopiperidina, piperazina, heterociclo este que poderá ser substituído por 1-2 substituintes; cada alq é c1-6alcanodiila; r1 e ar2 ou piperidinila, piperazinila, morfonila, tiomorfolinila, piridila, pirazinila, piridazinila, pirimidinila, furanila, tetraidrofuranila, tienila, pirrolila, tiazolila, oxazolila, imidazolila, isotiazolila, pirazolila, isoxazolila, oxadiazolila, quinilinila, quinoxalinila, benzofuranila, benzotienila, benzimidazolila, benzoxazolila, benzoxazolila, benztiazolila, piridopiridila, naftiridinila, 1h-imidazo[4,5-b]piridinila, 3h-imidazo[4,5-b]piridinila, imidazo[1,2-a]piridinila ou 2,3-diidro-1,4-dioxino[2,3-b]piridila; r3 é hidróxic1-6alquila, c1-6alcóxic1-6alquila, cianoc1-6alquila, aminocarbonil-c1-6aquila, mono- ou di(c1-6alquil)aminocarbonil-c1-6aquila, carboxil-c1-6alquila, c1-6alcoxicarbonil-c1-6alquila; r2 é hidrogênio ou c1-6alquila; r3 e r4 são hidrogênio, c1-6alquila, ar2, ar2c1-6alquila, c1-6alquilcarbonila, ar2carbonila, ar2c1-6alquilcarbonila, c1-6alquilsulfonila, aminossulfonila, ar1sulfonila, ar1c1-6alquilsulfonila, c1-6alquilóxic1-6alquila, aminoc1-6alquila, mono- ou di(c1-6alquil)aminoc1-6alquila, hidróxic1-6alquila, aminocarbonilc1-6alquila, c1-6alquiloxicarbonilc1-6aquila, hidroxicarbonilc1-6aquila, aminossulfonilc1-6alquila, het, het-c1-6alquila, het-carbonila, het-sulfonila, het-c1-6alquilsulfonila e het-c1-6alquilcarbonila; het é um heterociclo opcionalmente substituído; composições farmacêuticas que contêm compostos (i) e processos para preparação de compostos (i).
Patent BR-PI0617913-B8 (BR)
Title: sistema de fixação e artigo absorvente
Inventor: ERIC C STEINDORF
IPC: D04H3/00
Filed: 2006-10-04
Abstract: <b>sistema de fixação de espuma que inclui um modificador de superfície.<d> um sistema de fixação tendo um tecido não-tecido que inclui uma trama que é formada de uma pluralidade de fios extrudados e uma camada de espuma que inclui uma superfície tendo uma pluralidade de suportes verticais livres que são adaptados para engatar pelo menos uma parte da pluralidade de fios, pelo menos alguns dos suportes verticais livres incluindo o modificador de superfície.