baber/WOPTO huggingface dataset:
Patent BR-PI0902315-B1 (BR)
Title: Sensor de posicionamento à prova de fraude
Inventor: EIDI NAKAGAWA
IPC: G08B15/00
Filed: 2009-07-15
Abstract: sensor de posicionamento à prova de fraude, mais particularmente trata-se do desenvolvimento de um sensor de posicionamento (sp) composto de um dispositivo local (1) e um dispositivo remoto (2) dotados de uma inteligência programada (12), sigilosa e criptografada que o torne imune a tentativas de fraude e que permita determinar com um elevado grau de confiabilidade o posicionamento de um determinado elemento em relação a outro; algumas possíveis aplicações para este sensor de posicionamento poder ser relacionadas como sensor de abertura/fechamento de portas, sensor de posicionamento de determinado módulo lógico em um determinado gabinete que não pode ser movido sem a devida autorização.
Patent BR-PI0922028-B1 (BR)
Title: sistema de configuração e modelagem de bico de pulverização
Inventor: KEITH L CRONCE
IPC: B05C11/00
Filed: 2009-11-10
Abstract: sistema de configuração e modelagem de bico de pulverização um sistema de configuração de bico e de análise de injeção de pulverização é descrito tendo uma unidade de entrada de usuário que coleta os parâmetros de entrada de sistema de pulverização e retransmite os parâmetros coletados para uma unidade de combinação de desempenho de fluido e/ou unidade de geometria de problema para processamento subsequente. o usuário introduz parâmetros básicos de sistema, incluindo as características desejadas do fluido de pulverização, para obter configuração sugerida de sistema, incluindo tipos e quantidades de bicos de pulverização. a exatidão do tipo de bico de pulverização sugerido e da configuração é aumentada por intermédio de aproximação dos parâmetros de viscosidade e/ ou tensão de superfície do fluido de pulverização desejado com aqueles dos dados de desempenho coletados. quando um usuário já conhece o tipo de bico de pulverização desejado e os parâmetros associados de sistema, a unidade de entrada de usuário encaminha essa informação para a unidade de geometria de problema para criação de um arquivo de geometria de problema, incluindo o cálculo de distribuição de tamanho de gota e velocidade de pulverização, e modelagem de desempenho por intermédio da unidade de modelagem de fluido.
Patent EA-000348-B1 (EA)
Title: Method of lessening the risk of vertebral fractures
Inventor: KARPF DAVID B
IPC: C07F/
Filed: 1996-02-13
Abstract: 1. A method of reducing the risk of vertebral fractures in an osteoporotic female comprising administering an effective amount of alendronate or a pharmaceutically acceptable salt thereof for a period of more than two years. 2. A method according to Claim 1 wherein the alendronate is administered orally. 3. A method according to Claim 2 wherein the dose is from 2.5 mg to 50 mg daily. 4. The method according to Claim 3 wherein the alendronate is administered substantially daily for a period of at least two years. 5. The method according to Claim 3 wherein the alendronate is administered substantially daily for a period of at least three years. 6. The method according to Claim 1 wherein the female is elderly. 7. A method of reducing the severity of a fracture in patients who sustain a fracture by administering an effective amount of alendronate for a period of more than two years. 8. A method according to Claim 7 wherein the alendronate is administered orally. 9. A method according to Claim 8 wherein the dose is from 2.5 mg to 50 mg daily. 10. The method according to Claim 9 wherein the alendronate is administered substantially daily for a period of at least two years. 11. The method according to Claim 9 wherein the alendronate is administered substantially daily for a period of at least three years. 12. The method according to Claim 7 wherein the female is elderly. 13. A method of decreasing spinal deformity in osteoporotic women comprising administering an effective amount of alendronate for a period of more than two years. 14. A method according to Claim 13 wherein the alendronate is administered orally. 15. A method according to Claim 14 wherein the dose is from 2.5 mg to 50 mg daily. 16. The method according to Claim 15 wherein the alendronate is administered substantially daily for a period of at least two years. 17. The method according to Claim 15 wherein the alendronate is administered substantially daily for a period of at least three years. 18. The method according to Claim 13 wherein the female is elderly 19. A method of preventing loss of height in osteoporotic women by administering an effective amount of alendronate for a period of more than two years. 20. A method according to Claim 19 wherein the alendronate is administered orally. 21. A method according to Claim 20 wherein the dose is from 2.5 mg to 50 mg daily. 22. The method according to Claim 21 wherein the alendronate is administered substantially daily for a period of at least two years. 23. The method according to Claim 21 wherein the alendronate is administered substantially daily for a period of at least three years. 24. The method according to Claim 19 wherein the female is elderly.
Patent EA-003332-B1 (EA)
Title: A substituted triazolo-pyridazine derivative, pharmaceutical compositions made therefrom
Inventor: CARLING WILLIAM ROBERT
IPC: C07D487/04
Filed: 1999-06-15
Abstract: 1. 7-(1, 1-Dimethylethyl)-6-(2-ethyl-2H-1,2,4-triazol-3-ylmethoxy)-3-(2-fluorophenyl)-1,2,4-triazolo [4,3-b] pyridazine. 2. Polymorph A of 7-(1, 1-dimethylethyl)-6-(2-ethyl-2H-1,2,4-triazol-3-ylmethoxy)-3-(2-fluorophenyl)-1,2,4-triazolo [4,3-b] pyridazine as characterised herein. 3. A pharmaceutical composition comprising 7-(1,1dimethylethyl)-6-(2-ethyl-2H-1,2,4-triazol-3-ylmethoxy)-3-(2-fluorophenyl)1,2,4-triazolo [4,3-b] pyridazine in association with a pharmaceutically acceptable carrier. 4. The use of 7-(1,1-dimethylethyl)-6-(2-ethyl-2H-1,2,4-triazol-3ylmethoxy)-3-(2-fluorophenyl)-1,2,4-triazolo [4,3-b] pyridazine for the manufacture of a medicament for the treatment and/or prevention of anxiety. 5. A process for the preparation of 7-(1,1-dimethylethyl)-6-(2ethyl-2H-1,2,4-triazol-3-ylmethoxy)-3-(2-fluorophenyl)-1, 2, 4-triazolo [4,3-b] pyridazine, which comprises reacting a compound of formula III with the compound of formula IV:     wherein L<1> represents a suitable leaving group. 6. A process for manufacturing 7-(1, 1-dimethylethyl)-6-(2-ethyl-2H-1,2,4-triazol-3ylmethoxy)-3-(2-fluorophenyl)-1,2,4-triazolo [4,3-b] pyridazine, which comprises reacting a compound of formula XI (or tautomer thereof 1, 2, 4-triazolo [4,3-b] pyridazine-6-one) with the compound of formula XII:     wherein L<3> represents a suitable leaving group 7. A process for manufacturing 7-(1, 1-dimethylethyl)-6-(2-ethyl-2H-1,2,4-triazol-3ylmethoxy)-3-(2-fluorophenyl)-1,2,4-triazolo [4,3-b] pyridazine, which comprises reacting trimethylacetic acid with the compound of formula XIII: in the presence of silver nitrate and ammonium persulfate. 8. A process for manufacturing 7-(1, 1-dimethylethyl)-6-(2-ethyl-2H-1,2,4-triazol-3ylmethoxy)-3-(2-fluorophenyl)-1,2,4-triazolo [4,3-b] pyridazine, which comprises reacting the compound of formula XIV with the compound of formula XV: wherein M represents -B(OH)2 or -Sn(Alk)3, where Alk is C1-6 alkyl group, and L<4> represents a suitable leaving group in the presence of a catalyst based on a transition metal. 9. A process as claimed in claim 5 wherein reaction (A) is carried out in 1-methyl-2-pyrrolidinone, in the presence of sodium hydroxide, at a temperature in the region of 0 degree C. 10. A method for the treatment and/or prevention of anxiety which comprises administering to a patient in need of such treatment an effective amount of 7-(1,1-dimethylethyl)-6-(2-ethyl-2H-1,2,4-triazol-3ylmethoxy)-3-(2-fluorophenyl)-1,2,4-triazolo [4,3-b] pyridazine.
Patent EA-005674-B1 (EA)
Title: Method for the preparation of citalopram
Inventor: PETERSEN HANS
IPC: C07D307/87
Filed: 2001-05-10
Abstract: A method for the preparation of citalopram comprising reaction of a compound of formula 5-aminomethyl-1-(3-dimethylamino-propyl)-1-(4-fluoro-phenyl)-1,3-dihydro-isobenzofuran with an oxidising agent to prepare citalopram.
Patent EA-004414-B1 (EA)
Title: Locking and sealing device
Inventor: LAZHENTSEV OLEG ARKADIEVICH
IPC: E05B39/02
Filed: 2003-06-02
Abstract: 1. A locking and sealing device comprising a housing, a spring-loaded fixing element, designed in the form of at least two separate elements with a male outer conical surface corresponding to a female conical surface made in the housing, a locking element in the form of a cylindrical rod with a head at one end and other sharpened end conjugated with the cylindrical portion, characterized in that said locking and sealing device comprises a stabilizer of the fixing element arranged in the housing and designed in the form of a step disc having an axial aperture spring-loaded by said spring to provide a contact with the end of the fixing element , wherein the other end of the latter is provided with an inverse lead-in cone, and the rod has a cylindrical turning the sharpened rod end is designed as a cone and conjugated with said cylindrical portion interacting with the stabilizer. 2. The device of claim 1, characterized in that the fixing element is designed as a split bushing. 3. The device of claim 1, characterized in that the length of the rod turning exceeds the length of the fixing element. 4. The device of claim 1, characterized in that the angle of said inverse lead-in cone of the fixing element is equal to the angle of the rod cone. 5. The device of claim 1, characterized in that the female conical surface of the housing is a through surface.
Patent EA-006225-B1 (EA)
Title: Novel cyclohexyl sulphones
Inventor: CHURCHER IAN
IPC: C07D211/62
Filed: 2002-08-16
Abstract: Novel sulphones of formula I are disclosed: The compounds modulate the processing of amyloid precursor protein by gamma-secretase, and hence are useful in the treatment or prevention of Alzheimer's disease.
Patent EA-005732-B1 (EA)
Title: A cleaning efficiency testing method and apparatus therefor
Inventor: HEDSTROM STEFAN
IPC: B01D65/10
Filed: 2002-11-26
Abstract: A method and an apparatus are provided for testing the efficiency of a cleaning procedure for a filter in a filtering system. After the cleaning procedure (21) of the filter, the filter pores contain a fluid (22). The system is pressurized (23), and a decay in pressure over a predetermined time period is measured (24). Based on the pressure decay, it is determined whether or not the cleaning procedure has been effective (25); a pressure decay smaller than a predetermined threshold value indicates that the cleaning procedure has not been effective.
Patent EA-007828-B1 (EA)
Title: Cigarette having porous heat transfer tube
Inventor: DANTE HENRY M
IPC: A24D1/00
Filed: 2004-02-13
Abstract: A smoking article includes a cylinder of smoking material, a filter attached to the cylinder of smoking material, and a tube of preferably porous and/or perforated material adapted to collapse at an open end upon exposure to thermal energy and preferably extending from one end portion of the smoking material to the junction of the filter and the cylinder of smoking material. Thermal energy generated by a burning portion of the tobacco filler material within the cylinder of smoking material is transferred by convection through the open portion of the tube after the end portion of the tube has collapsed and closed by the heat from the burning portion of the tobacco.
Patent EA-010505-B1 (EA)
Title: High performance water-based drilling mud and methods of use
Inventor: PATEL ARVIND D
IPC: C09K8/04
Filed: 2004-09-01
Abstract: A water based drilling fluid for use in drilling a subterranean well through a subterranean formation that swells in the presence of water, the drilling fluid is formulated to include: an aqueous based continuous phase; a weight material; an optional shale hydration inhibition agent and a shale encapsulator. The shale encapsulator is preferably a quaternized polyvinyl alcohol having the formula (I)in which x and y have a value so that the molecular weight of the cation is in the range of about 10,000 to about 200,000 AMU; A is selected from C-Calkyl, C-Cether or C-Camide; R, R' and R" are independently selectable C-Calkyl; and Bis a charge balancing anion to the quarternary amine. The shale hydration inhibition agent and the shale encapsulator may be present in sufficient concentrations to reduce the swelling of the subterranean formation in the presence of water. Conventional additives may be included into the formulation of the drilling fluid, such conventional additives may include: fluid loss control agents, alkaline reserve and other pH control agents, bridging agents, lubricants, anti-bit balling agents, corrosion inhibition agents, surfactants and solids suspending agents as well as mixtures and combination of these and similar compounds that should be known to one of skill in the art.
Patent EA-010265-B1 (EA)
Title: Pyrimidine derivatives for use as vanilloid receptor ligands and their use in the treatment of pain
Inventor: WANG HUI-LING
IPC: C07D405/12
Filed: 2005-02-11
Abstract: Pyrimidine ethers and compositions containing them, for use as vanilloid receptor ligands for the treatment of acute, inflammatory and neuropathic pain, dental pain, general headache, migraine, cluster headache, mixed-vascular and non-vascular syndromes, tension headache, general inflammation, arthritis, rheumatic diseases, osteoarthritis, inflammatory bowel disorders, inflammatory eye disorders, inflammatory or unstable bladder disorders, psoriasis, skin complaints with inflammatory components, chronic inflammatory conditions, inflammatory pain and associated hyperalgesia and allodynia, neuropathic pain and associated hyperalgesia and allodynia, diabetic neuropathy pain, causalgia, sympathetically maintained pain, deafferentation syndromes, asthma, epithelial tissue damage or dysfunction, herpes simplex, disturbances of visceral motility at respiratory, genitourinary, gastrointestinal or vascular regions, wounds, burns, allergic skin reactions, pruritus, vitiligo, general gastrointestinal disorders, gastric ulceration, duodenal ulcers, diarrhea, gastric lesions induced by necrotising agents, hair growth, vasomotor or allergic rhinitis, bronchial disorders or bladder disorders.
Patent EA-012587-B1 (EA)
Title: Biotinylated hexadecasaccharides, preparation and use thereof
Inventor: DUCHAUSSOY PHILIPPE
IPC: A61F2/958
Filed: 2005-09-07
Abstract: The invention concerns novel biotinylated hexadecasaccharides of general formula (I) wherein: Biot is a biotin derivative; R, Rand R, represent independently of one another a C-Calkoxy or and –OSO; Rrepresents a C-Calkoxy or an –OSO, or Rconstitutes a -O-CH-bridge; Pe represents a saccharide concatenation; as well as their pharmaceutically acceptable salts, and their use as medicines.
Patent EA-017784-B1 (EA)
Title: Device for storing and dosage administration of viscous medicament
Inventor: YUKHT IGOR
IPC: A61J1/00
Filed: 2007-12-29
Abstract: The proposed device relates to medical engineering, in particular to devices for storing and dosage administration of viscous substances, ointments, pastes, oils and gels on skin. The device can be used as an individual means for administering first medical aid. The proposed device for storing and dosage administration of viscous medicament provides a controlled dosage, uniform and thickness application on injured and wounded skin surfaces, thus enhancing treatment efficiency due to a single dosing required for each pathology, causing lesser traumatism and pain reaction, quick medicament absorption. A container cover has a flat support part for a dosage administration, wherein the cover is positioned in the down part of the device to provide a direct and constant contact with the medicament in the container through a valve element having an orifice in the container body. At least the container side surface is performed transparent and the container has a control means for checking medicament volume therein, the volume control means is graduated on the transparent container side surface or quite close to it.
Patent EA-013129-B1 (EA)
Title: Storage-stable sulphonamide formulations
Inventor: SCHNABEL GERHARD
IPC: A01N47/36
Filed: 2006-08-29
Abstract: The present invention relates to solid, storage-stable, water-dispersible formulations comprising one or more active herbicidal compounds from the group of the sulphonamides and their salts, one or more carrier materials, and one or more wetting agents from the group of the naphthalenesulphonic acids and the group of the sulphosuccinic acid derivatives and also the salts of these groups. The formulations of the invention are suitable for the crop protection sector.
Patent EA-013100-B1 (EA)
Title: Surgical repair product comprising uhmwpe filaments
Inventor: OOSTEROM ROGER
IPC: A61B17/06
Filed: 2006-11-28
Abstract: The invention relates to an elongate surgical repair product comprising a cable of which bending stiffness can be lowered, which fibrous member is a heat-set cable comprising at least 50 mass% of high-performance polyethylene yarn. The product shows very high tenacity, combined with a relatively high initial bending stiffness that is significantly reduced upon bending or flexing the member, without significant dimensional change; and allows both easy and well-controlled handling and good knot tying characteristics. The invention also relates to a method of making said elongate product, wherein the heat setting is carried out at a temperature (preferably between 140 and 151°C) under elongational tension.
Patent EA-020993-B1 (EA)
Title: Communication apparatus and communication method
Inventor: AIBA TATSUSHI
IPC: H04W72/08
Filed: 2008-09-03
Abstract: Provided is a mobile communication system in which a mobile station apparatus transmits a reception quality information indicating the quality of a signal received from a base station apparatus, characterized by that the base station apparatus transmits information indicating transmission of the reception quality information not accompanied by any upstream link data, included in the upstream link data transmission permission signal, and the mobile station apparatus transmits reception quality information not accompanied by the upstream link data according to the information indicating transmission of the reception quality information not accompanied by the upstream link data. Thus, even when no upstream link data exists between the mobile station apparatus and the base station apparatus, it is possible to transmit the reception quality information having a large information amount from the mobile station apparatus and it is possible to perform transmission control flexibly corresponding to the information amount and the transmission frequency of the reception quality information transmitted from the mobile station apparatus. Thus, more effective communication control (scheduling) between the base station apparatus and the mobile station apparatus can be achieved.
Patent EA-018725-B1 (EA)
Title: Smoking article with controlled flavor release
Inventor: KARLES GEORGIOS D
IPC: A24C5/56
Filed: 2008-06-06
Abstract: Provided are smoking articles 10 with a controlled flavor release product 16. The controlled flavor release product includes a first time-release flavorant 24 and a second time-release flavorant 26. The controlled flavor release product is a film or a lip balm type formulation that is applied to the downstream end 14 of a smoking article.
Patent EA-021873-B1 (EA)
Title: Method for producing a vessel closure
Inventor: POEL-ASENDORF CHRISTIANE
IPC: C09K3/10
Filed: 2008-11-07
Abstract: The invention relates to a method for producing a vessel closure for vessels comprising an opening that is to be closed by the vessel closure, an inner diameter of more than 2 cm and surrounds a polymer-based sealing element that is arranged in the vessel closure in such a manner that is sealingly rests on the opening of the vessel in the closed state, wherein a polymer material being used becomes sufficiently free-flowing by warming and is applied to the vessel closure in the region of the sealing element that is to be produced, and optionally, is mechanically formed into the desired shape which it maintains after cooling, wherein the sealing element of the vessel closure, the inner surface of which has no free access, is formed by a stamp or extrusion, wherein the polymer comprises a polyethylene and alkene and does not comprise PVC, and wherein the sealing element has a Shore A hardness in a range from 40 to 90 and a compression set in a range from 30 to 70%;
Patent EA-017822-B1 (EA)
Title: Injection device
Inventor: JENNINGS DOUGLAS IVAN
IPC: A61M5/20
Filed: 2008-07-28
Abstract: An injection device comprises a locking-mechanism in the form of two buttons (170) located on the front end of the injection device. In an engaged position, the locking mechanism prevents removal of a cap (111) from the injection device and, in a disengaged position, prevents movement of a syringe carrier (127) holding a syringe but permits removal of the cap from the housing. This assists in preventing damage to the syringe prior to actuation of the injection device.
Patent EA-018350-B1 (EA)
Title: Process for stabilization of hydrocarbon fuels against oxidation decomposition
Inventor: ORLOVSKAYA NINA FEDOROVNA
IPC: C07C7/20
Filed: 2011-10-27
Abstract: The invention relates to organic chemistry, in particular to processes for stabilization of hydrocarbon fuels against oxidation decomposition. the invention is aimed at enhancing effectiveness of fuel stabilization 3-(1,1,2,2-tetraflouroethyl)-5-phenyl-N,N-diethyl-4-nitrozoaniline due to introduction an additional antioxidant, stipulating the increase of solubility and an antioxidant activity of the nitroozoaniline. The stabilization of the hydrocarbon fuels against oxidation decomposition is carried out by adding in their composition a solution 3-(1,1,2,2-tetraflouroethyl)-5-phenyl-N,N-diethyl-4-nitrozoaniline in hexadecane oxygenate, comprising a mixture of saturated monoatomic primary and secondary alcohols with molar ratio 3-(1,1,2,2-tetraflouroethyl)-5-phenyl-N,N-diethyl-4-nitrozoaniline and a mixture of the saturated monoatomic primary and secondary alcohols (0,5-1,5):(140-160).
Patent EA-020078-B1 (EA)
Title: Rolling drilling bit
Inventor: BUTKIN VLADIMIR DMITRIEVICH
IPC: E21B10/20
Filed: 2011-11-01
Abstract: The invention relates to rolling drilling, in particular, to a design of a rolling drilling bit for use in drilling boreholes of any direction in mining, oil and gas industry, road and channel construction, etc. A rolling drilling bit comprises a housing with nipple and vent passages, cutters of semispherical or flattened spherical shape and their support with vertical trunnions; support of each cutter is made in the form of stepped support shaft, with possibility of rotation, one end of which faces the bottom hole and has rectangular cross section and is fixed inside removable solid cutter, and the other end having the shape of cylinder or flattened cone is installed in the housing hole, and is equipped with ringless thrust ball bearing, and in the hole at the housing outlet the stepped shaft is equipped with sealing elements fixed with unsplit detachable cover attached to the bit housing. For drilling conditions of horizontal wells in mine rocks of small and medium thickness the support shaft is made at an angle of 5-15 degrees to bit axis; at that, teeth of peripheral rim of bits have dimensions which are by 1.2-1.3 times more than those of the last rim. The technical effect provides increasing service life and operating efficiency of bit; reducing manufacturing costs.