baber/WOPTO huggingface dataset:
Patent IL-102793-A0 (IL)
Title: Oxocyclic urea compounds and pharmaceutical compositions containing them
IPC: C07D233/80
Filed: 1992-08-12
Abstract: The novel 4-oxocyclic ureas and the pharmaceutically- acceptable salts and esters thereof of the present invention are useful as antiarrhythmic and antifibrillatory agents and have following general structure: <CHEM> wherein  (a) X is a saturated or unsaturated, 5-, 6-, or 7-membered heterocycle or carbocycle; (b) R is selected from the group consisting of covalent bond, nil, heteroatom, carbonyl, heterocyclic ring, carbocyclic ring, alkyl, alkenyl, alkoxy, alkylamino, arylalkyl, aryloxy, acyl, acyloxy, and acylamino; (c) Y is a substituted or unsubstituted, saturated or unsaturated, 5-, 6-, or 7-membered heterocyclic ring or carbocyclic ring, or is nil;  and wherein when R is nil, X and Y are fused ring systems; and when R is a covalent bond, X and Y are ring systems linked through a covalent bond; and when Y is nil, R is a covalent bond, and X is bound to L through R;  (d) R1, R2, and R3 are independently selected from the group consisting of nil, Cl, F, Br, NH2, CF3, OH, SO3H, CH3SO2NH, COOH, alkoxy, alkyl, alkoxycarbonyl, hydroxyalkyl, carboxyalkyl, aminoalkyl, acylamino and acyloxy; (e) L is selected from the group consisting of alkylamino, alkenylamino, alkylimino, alkenylimino, and acylamino; wherein the nitrogen atom thereof is bound to the nitrogen atom at the 1-position of 4-oxocyclic urea moiety; (f) R4 is selected from the group consisting of alkyl, alkenyl, alkynyl, alkylacyl, and heteroalkyl; (g) A is a substituted or unsubstituted, saturated or unsaturated, straight-chain or branched, C1-C8 heteroalkyl; or a substituted or unsubstituted, saturated or unsaturated heterocycle having 5-, 6-, or 7-members; and A has one nitrogen atom, which is adjacent to R4; and (h) R5 is a substituted or unsubstituted C1 or C2 alkyl.
Patent IL-111844-A0 (IL)
Title: Process for the processing of thermoplastic polymers by means of the injection-moulding technique
IPC: B29K105/06
Filed: 1994-12-01
Abstract: In the case of liquid crystal polymers, on the one hand the rigid molecule chains and on the other hand possibly present fibrous reinforcing materials are aligned largely parallel to a weld line or flow line, with the result that the physical properties are lacking in the region of the weld line or flow line. It is an object of the invention to provide a possible way of preventing weld lines or flow lines from occurring in the first place. For this purpose, the liquidified material is subjected to a shearing energy from its entry into the injection mould, over at least part of the length of the workpiece. This shearing energy is produced by relative movement between two surfaces of the mould parts. <IMAGE>
Patent IL-111959-A0 (IL)
Title: Benzenesulfonamide derivatives their preparation and pharmaceutical compositions containing them
IPC: C07D409/14
Filed: 1994-12-12
Abstract: A benzenesulfonamide derivative of the formula [I]: <CHEM> wherein Ring A and Ring B are the same or different and each substituted or unsubstituted benzene ring, Q is a single bond or a group of the formula: -O-, -S-, -SO-, -SO2- or -CH2-, Y is a group of the formula: -O-, -S- or -NH-, Alk is lower alkylene group or lower alkenylene group, Z is a single bond or a group of the formula: -O- or -NH-, R is a substituted or unsubstituted aromatic heterocyclic or aryl group, R<1> is hydrogen atom, trifluoromethyl group, substituted or unsubstituted lower alkyl group, substituted or unsubstituted lower alkenyl group, mono- or di-lower alkylamino group, substituted or unsubstituted lower alkylthio group, substituted or unsubstituted lower alkoxy group, substituted or unsubstituted lower alkynyl group, aromatic heterocyclic group, substituted or unsubstituted aliphatic heterocyclic group or aryl group, provided that when Z is a single bond, R is a substituted or unsubstituted aromatic heterocyclic group, or a pharmaceutically acceptable salt thereof, and processes for preparing the same, these compounds having endothelin antagonistic activity and being useful in the prophylaxis or treatment of various diseases caused by endothelin.
Patent IL-112528-A0 (IL)
Title: 3-(2-aminoethyl)-4-[3-(trifluoromethyl) benzoyl]-3,4-dihydro-2H-1, 4-benzoxazine derivatives, process for their preparation and their therapeutic application
IPC: C07D265/36
Filed: 1995-02-02
Abstract: Benzoxazine derivs. of formula (I) and their optical isomers and acid-addn. salts are new. R1 = H, F, Cl, Me, 1-3C alkoxy or NO2; R3 = H or 1-3C alkyl; R4 = 2,3-dihydro-1H-inden-2-yl, 2,3-dihydro-1H-inden-1-yl or 1,2,3,4-tetrahydronaphthalen-1-yl; or NR3R4 = 1,2,3,4-tetrahydro- 9H-pyrido(3,4-b)indol-2-yl, 1,2,3,4-tetrahydro- 9H-pyrido(4,3-b)indol-3-yl, 4,5,6,7-tetrahydro- thieno(2,3-c)pyridin-6-yl, 4,5,6,7-tetrahydro- thieno(3,2-c)pyridin-6-yl or 2,3-dihydro-1H-isoindol-2-yl.
Patent IL-117394-A0 (IL)
Title: Process for preparing bleach activators
IPC: C07C309/42
Filed: 1996-03-07
Abstract: The synthesis of phenol sulfonate esters of alkanoyl amino acids is conducted in the presence of aqueous base to provide bleach activator compounds. Thus, the acid chloride of N-nonanoyl-6-aminocaproic acid is reacted with the sodium salt of p-phenol sulfonate in the presence of water at a pH in the range of about 9 to about 12 to yield the corresponding phenol sulfonate ester. The synthesis of the phenol sulfonate ester of the monononyl amide of adipic acid is also illustrated.
Patent IL-121432-A0 (IL)
Title: Pyrroloazepine derivatives
IPC: C07D495/20
Filed: 1996-12-02
Abstract: Disclosed is a pyrroloazepine derivative or a salt thereof. The pyrroloazepine derivative is represented by the following formula (I): <CHEM>  wherein     the ring P represented by <CHEM>  means a pyrrole ring represented by the following structure: <CHEM> in which R1 represents alkyl, cycloalkyl or the like, and R2 represents H or alkyl; the dashed line indicates the presence or absence of a bond; and, when the bond is present, Z2 is not present/and Z1 represents H but, when the bond is absent, Z1 and Z2 are both H; Z1 represents H and Z2 represents a group OR3 in which R3 represents H, alkyl, aralkyl or the like; Z1 and Z2 both represent groups SR4 in which R4 represents alkyl, aralkyl or the like; or Z1 and Z2 are combined together to represent O, a group NOR5 in which R5 represents H, alkyl or the like, or a C2-C3 alkylenedithio; A represents alkylene, alkenylene or alkynylene; and Y represents a group <CHEM> in which W represents CH, C= or N, m stands for 0 or 1, n stands for 1, 2 or 3, G represents O, S, C=O, sulfinyl, sulfonyl, alkylene, alkenylene, acetal or the like; E1 and E2 represent H or lower alkyl group; and D represents an aromatic hydrocarbon or am aromatic heterocyclic ring. The compound (I) has strong serotonin-2 receptor antagonistic action and low toxicity and less side effects, and is useful as a therapeutic for circulatory diseases such as ischemic heart diseases, cerebrovascular disturbances and peripheral circulatory disturbances.
Patent IL-132973-A0 (IL)
Title: Gasoline pump
IPC: B67D99/00
Filed: 1999-11-16
Abstract: In a gasoline pump system, means for concurrent filling of more than one car, tank or container with gasoline or other liquid petroleum products, comprising a display for guiding car drivers to a gasoline pump system having an outlet available for fueling, and a display for enabling each driver to identify the outlet used for filling his/her car, and to distinguish it from outlets used for filling other cars. A method for concurrent filling of more than one car, tank or container with gasoline or other liquid petroleum products, comprising the steps of:A. Guiding car drivers to a gasoline pump system having an outlet available for fueling; andB. Enabling each driver to identify the outlet used for filling his/her car, and to distinguish it from outlets used for filling other cars.
Patent IL-135732-A0 (IL)
Title: A method and a device for displaying at least part of the human body with a modified appearance thereof
IPC: G06T1/00
Filed: 1998-10-29
Abstract: A method and a device for displaying at least part of a person's body, for example the head (<HIL><PDAT>10</BOLD><PDAT>), with a modified appearance by providing first image data representatitve of the unmodified appearance of the body part, second image data representatitve of a modification in the appearance of the body part (<HIL><PDAT>10</BOLD><PDAT>) and position data representative of the position and spatial orientation of the body part (<HIL><PDAT>10</BOLD><PDAT>). The first and second image data are linked to produce and to display third image data representative of the modified appearance of the body part, in dependence on the position data, such that the displayed, modified appearance follows changes in the position of the body part in a dynamic manner. For linking the first and second image data a virtual image data space (<HIL><PDAT>9</BOLD><PDAT>) is created comprising an aspect or aspects (<HIL><PDAT>12</BOLD><PDAT>) of the appearance of the body part (<HIL><PDAT>10</BOLD><PDAT>) to be modified. The second image data comprise virtual image data elements (<HIL><PDAT>13</BOLD><PDAT>), and the modification of the appearance of the body part (<HIL><PDAT>10</BOLD><PDAT>) is provided by modifying the virtual image data space (<HIL><PDAT>9</BOLD><PDAT>) using virtual image data elements of the second image data, wherein the virtual image data space thus formed and the first image data not comprised thereof are linked to produce the third image data in dependence on the position data.</PTEXT>
Patent IL-143670-A0 (IL)
Title: Methods for the expression of active protein-immunoglobulin fusions, active protein-immunoglobulin fusions obtained thereby and pharmaceutical compositions containing the same
IPC: C12N1/19
Filed: 1999-12-16
Abstract: Methods for high level expression of active lymphotoxin-² receptor immunoglogulin chimeric proteins and their purification.
Patent IL-150135-A0 (IL)
Title: Integrated aqua-ammonia chiller/heater
IPC: F25B15/00
Filed: 2001-01-03
Abstract: An aqua-ammonia chiller/heater apparatus is modified to provide a condenser and absorber refrigerant by-pass during a heater mode.
Patent IL-155472-A0 (IL)
Title: Printed media production
IPC: B41J2/01
Filed: 2001-10-19
Abstract: An inkjet nozzle assembly includes: a nozzle chamber having a floor and a roof spaced apart from the floor, the roof having a displaceable portion defining an ejection port; and an actuator for displacing the displaceable portion of the roof towards the floor. Displacement of the displaceable portion of the roof alters a volume of the nozzle chamber such that when the volume is altered, fluid is ejected from the ejection port.
Patent IL-164652-A0 (IL)
Title: Method of treating arrhythmias comprising administration of an A1 adenosine agonist with a beta blocker, calcium channel blocker or a cardiac glycoside
IPC: A61K31/7076
Filed: 2004-10-18
Abstract: Methods are provided for treating arrhythmia in a manner that minimizes undesirable side effects, comprising administration of a therapeutically effective minimal dose of an A1 adenosine receptor agonist with a therapeutically effective minimal dose of a beta blocker, calcium channel blocker, or a cardiac glycoside.
Patent IL-185626-A0 (IL)
Title: Sublingual coated tablet
Filed: 2007-08-30
Abstract: The present invention relates to a fentanyl coated tablet and to the method for the preparation thereof.
Patent IL-210144-A0 (IL)
Title: Surface covering device
Filed: 2010-12-21
Abstract: The invention relates to a device for covering a surface such as a swimming pool, a sports field, a glazed surface, a vehicle body, including: (a) a drum rotatingly mounted and capable of winding or unwinding a cover, said drum being mounted on longitudinal translation mechanisms including rails provided on either side of said surface; (b) an attachment system for said cover at one transverse end of the surface to be covered so that the translation and the rotation of the drum results in the winding/unwinding of the cover above the surface to be covered; (c) a system for continuously locking the longitudinal edges of the cover onto said rails that is progressively fitted during the unwinding operation.
Patent RO-125286-A0 (RO)
Title: Decorative box creating images similar to holographic images
Inventor: COJAN DAN
IPC: C03C27/12
Filed: 2009-10-30
Abstract: The invention relates to a decorative box creating images similar to the holographic images, with multiple functions, which may carry out spatial images in the shape of a globe and sphere-shaped projections, meant to be used as wall application, table top, decoration included into the furniture, into the wall or stoneware tiles, floor tile, external and internal light sign board, decorative object and/or advertising object etc. According to the invention, the box is carried out in the shape of a housing (1) or as a frame (8) wherein there is introduced a logo (2) or an object (2") which is desired to be represented in spatial image by means of some lens (5, 5"), the box including, in the order of the arrangement therein, the logo (2) or the object (2") around which there are placed some lights (4, 4'), preferably electroluminiscent diodes arranged in rows, above which the lens (5, 5") will be placed, and above said lens a preferably secured glass (7) is placed for protecting the same, while, when using the box as a floor tile, between the bottom cover of the housing (1) and the secured glass (7, 7") for the protection of the Fresnel lens (5) some shock damping elements and, possibly, a decorative element (6) with a central cut-out capable of hiding from view said shock damping elements and lights (4) are additionally inserted.
Patent RO-126736-A0 (RO)
Title: Fungal elicitor-producing botrytis cinerea strains, product for immunization of strawberry plants against grey mould and application methods
Inventor: MATEI SORIN
IPC: A01H15/00
Filed: 2010-12-08
Abstract: The invention relates to a composition of a product meant to immunize the strawberry plants against three novel virulent strains of Botrytis cinerea and to the methods for the application of this composition in the preventive treatment of grey mould in strawberry plant. The Botrytis cinerea strain, BcS1 presents greyish-white wool-like colonies with rare black sclerotes on Czapek medium, grey colonies with numerous black sclerotes on PDA medium, long septated brown conidiofores with intercalar or apical branching, non-septated hyaline smooth conidia. The Botryris cinerea strain BcP2 presents dense wool-like dark grey colonies with numerous black sclerotes, tall, thin, brown septated conidiofores with intercalar branching, non-septated hyaline smooth conidia. The Botrytis cinerea strain, BcF7 presents initially hyaline colonies light coloured in the centre, wool-like with developed black sclerotes in a moderate number, tall, thin, brown septated irregularly branched conidiofores with apical and intercalar conidial ends, non-septated light brown conidia with prominent hilum. The product claimed by the invention contains total soluble proteins 1.06...22.67 mg/l, total reducing glucides 1.98...19.39 mg/l, total flavonoids 0.01...0.4485 μ g/l, total polyphenols 39.42...336.51 mg/l, pectin lyase 0.637...0.513 U/ml, kitinase 0.423...0.627 U/ml, cellulase 0.012...1.98 U/ml, carboxymethylcellulose 0.018...0.940 U/ml, β-1,3 glucanase 1.109...7.092 U/ml, total content of amino acids 456.19...467.79 mmol/100 ml.
Patent RO-133531-A0 (RO)
Title: Voltage step-up micro-convertor device and method for carrying out the same
Inventor: SURDUCAN VASILE
IPC: H02M3/338
Filed: 2018-08-14
Abstract: The invention relates to a voltage step-up micro-convertor device meant for conversion of low-power pulsed electric energy, in the range of μW - mW, and reduced input voltage, of 20 mV...1.5 V, obtained by collecting energy with output values of 2V...5V. According to the invention, the device consists of an asymmetric autoresonant oscillator (1) comprising a voltage step-up transformer (101) with a primary coil (101a) and a secondary coil (101b) and a number of FET transistors (102) coupled in parallel and so connected as to provide a positive reaction between the primary and secondary coil of the transformer, the oscillator (1) being supplied through a constant current generator which comprises an accumulation capacitor (201), a coil (202) and a smoothing capacitor (203) and having output voltages which are rectified with a diode (110), charging a back-up accumulator (3), and with other diodes (108, 109) charging a load accumulator (4), the current charging the two accumulators (3 and 4) being limited by adjustment of autoresonant oscillation by pulse width modulation PWM, due to some resistors (112, 113) and to a capacitor (114) polarizing the grids of the FET transistors (102) from the rectified voltage obtained from the transformer secondary coil.
Patent RO-135761-A0 (RO)
Title: Eco-friendly internal combustion engine
Inventor: PASCU NICOLAE
IPC: H02N11/00
Filed: 2021-12-30
Abstract: The invention relates to an environmentally friendly internal combustion engine. According to the invention, the engine, uses some mixing and explosion chambers (1), using explosive gases in an eco-friendly power plant and for burning and exploding the air mixture, which can be also compressed air, liquefied combustible gases, natural gas, methane gas, petroleum gas, gases resulting from organic waste gasification and any other gases of the alkene family which, by combustion, produces heat, water and carbon dioxide and for sending the blow of explosion which also contains water vapor and carbon dioxide in a water jet forming device (18) at pressures that can be of the order of hundreds of bar, located at the surface of a water tank (27), and from here, through a pipe (32), the jet of water with carbon dioxide under pressure reaches an injector (22) equipped with a deflector (24) which does not allow the dispersion of the jet and, optionally, with a flow regulator needle valve (23) which directs it onto some blades (21) of the rotor which is fixed on an output shaft (25) which can be coupled to the gearbox of various types of equipment or to an electric power generator which is located above the water tank and whose housing (26) partially closes the tank (27) in which a pump (29) for draining the water with carbon dioxide in the storm sewer system or directly into rivers or marine water.
Patent AP-2004002986-A0 (AP)
Title: Use of biologically active HIV-1 TAT, fragments or derivatives thereof, to target and/or to activate antigen-presenting cells, and/or to deliver cargo molecules for preventive or therapeutic vaccination and/or to treat other diseases
Inventor: ENSOLI BARBARA
IPC: A61P27/06
Filed: 2002-07-26
Abstract: The present invention concerns a method for prophylactic and/or therapeutic vaccination and/or treatment and/or diagnosis of HTWAIDS, other infectious diseases, inflammatory and angiogenic diseases and tumours which utilizes a biologically active HTV-1 Tat protein, fragments or derivates thereof, as a module with one or more of the following features: antigen, adjuvant and targeting-delivery system to specific antigen-presenting cells including dendritic cells, endothelial cells and macrophages. In particular, it is claimed that Tat can be used only in its biologically active form as an antigen combined with one or more other antigens, to prime or to boost protective immune responses against itself as well as other antigens and/or to selectively deliver these antigen(s) as well as active compounds to dendritic cells, endothelial cells and macrophages, due to its capability of targeting these A PC and of activating their maturation and functions and of increasing Th-1 type immune responses as an adjuvant. Therefore, due to these characteristics and to the distribution of these cells in the body (during physiological and pathological disorders), biologically active Tat, fragments or derivates thereof containing the ROD region, can be used for preventive, therapeutic and/or diagnostic purposes for HTV/AIDS, other infectious diseases, inflammatory and angiogenic diseases and tumors.
Patent CU-22479-A1 (CU)
Title: Surfactante pulmonar natural porcino
Inventor: ALFONSO LORENZO WILMA DE LA CARIDAD
Filed: 1994-12-29
Abstract: El objeto de la invención es un surfactante natural de uso terapéutico obtenido por extracción orgánica de surfactante pulmonar porcino, así como su método de obtención. El surfactante en cuestión contiene de un 90%, a un 95% de fosfolipidos, de 0.5 a 1.3% de proteínas hidrofobas, que incluyen las proteínas hidrófobas SPB y SPC, más del 40% de fosfatidilcolina disaturada y más del 8% de fosfatidilinositol con respecto a fosfolipidos. Más del 75% de la composición de ácidos grasos de la fosfaritidilcolina corresponde a ácido palmítico. El contenido total de los fosfolipidos aniónicos (fosfatidilglicerol + fosfatidilinositol) es mayor de 12% respecto a fosfolípidos. Los acilglicéridos representan más de un 3% con respecto a fosfolípidos, con predominio de triglicéridos. Una de sus formas farmacéuticas es un liofilizado estable de 2 a 8 sC que se reconstituye al momento de su uso. El producto recontituido presenta una tensión superficial mínima inferior a 5 din/cm a 5 min o con menor tiempo de pulsaciones para concentraciones de 10 y de 5 mg/mL para un 50% de compresión del área a 37 sC en el surfactómetro de burbuja pulsátil. La aplicación del surfactante por vía endotraqueal en dosis de 100 mg/kg de peso resultó efectiva en el síndrome de dificultad respiratoria del neonato. La utilización de dosis menores de 200 mg de fosfolipidos totales causó un incremento estable de la PaO2 y de la relación PaO2/FiO2 en pacientes con distrés respiratorio del adulto, en dosis repetidas de 3 a 9 aplicaciones.
Patent CU-21831-A1 (CU)
Title: Herramienta de percusión
Inventor: KULAGIN RIM ASMANOVICH
IPC: E21C27/00
Filed: 1985-12-19
Abstract: Comprende una caja que aloja un golpeador movible y está conectada a un cilindro mecánico en el cual está colocada una espiga golpeadora con un mecanismo sujetador y un impulsor en forma de una prensa hidráulica. La herramienta de percusión está provista de un dispositivo de control que tiene un medio de válvula para controlar un medio de distribución. El medio de válvula de carrete tiene una envoltura y delimita dos cámaras interconectadas a través de un medio obturador . Una cámara comunica constantemente con una tubería de descarga , y la otra cámara se pone periódicamente en comunicación con el espacio del cilindro hidráulico.
Patent LU-72503-A1 (LU)
IPC: H04R1/26
Filed: 1975-05-16
Abstract: 1499407 Loud-speaker systems; resonators CBS Inc 28 April 1975 [20 May 1974] 17471/75 Headings H4J and H4X A loud-speaker 312 is mounted on a rotatable baffle 310 having unequal horizontal edges in a generally open sided upper compartment which is formed above a closed lower compartment having a second speaker 306 mounted on one side face thereof, the speaker 306 being for a frequency range below that of the speaker 312. Further speakers 314, 316 for higher frequency ranges are also provided. Speakers 312, 314 in conjunction with respective portions of the baffle 310 form dipole radiators. The respective frequency ranges of speakers 312, 314 may be 200-1000 Hz and 1000-5000 Hz respectively, the speakers 306 and 316 dealing with the ranges below 200 Hz and above 5000 Hz respectively. The baffle may be pivoted within a frame arranged to pivot about a horizontal axis so as to provide for both displacement about a vertical and a horizontal axis (Fig. 7, not shown). The speakers are of the moving coil type but it is mentioned that capacitor or electret type speakers may be used, especially for the speakers 312, 314.