baber/WOPTO huggingface dataset:
Patent EP-1420029-A2 (EP)
Inventor: DUBUFFET THIERRY
IPC: C07K5/06
Filed: 2003-12-10
Abstract: Industrial production of perindopril (I) by reacting benzyl (2S,3aS,7aS)-octahydroindole-2-carboxylate (IIa) or benzyl (2S)-2-indoline-carboxylate (IIb) with N-((S)-1-ethoxycarbonyl-butyl)-(S)-alanine (III) then catalytically hydrogenating over palladium, the reaction of (IIa/b) with (III) is carried out in presence of specific coupling agent(s). Industrial production of (2S,3aS,7aS)-1-((2S)-2-((1S)-1-(ethoxycarbonyl)-butylamino)-propionyl)-octahydro-1H-indole-2-carboxylic acid (perindopril) (I) or its salt comprises: (1) reacting benzyl (2S,3aS,7aS)-octahydroindole-2-carboxylate (IIa) or benzyl (2S)-2-indoline-carboxylate (IIb) with N-((S)-1-ethoxycarbonyl-butyl)-(S)-alanine (III) in presence of a coupling agent (or coupling agent combination) (A) and optionally a base; and  (2) subjecting the product to catalytic hydrogenation in presence of palladium, optionally followed by salification. (A) is selected from: (1) (1,3-dimethylaminopropyl)-3-ethyl-carbodiimide hydrochloride (optionally in combination with 1-hydroxybenzotriazole, 1-hydroxy-7-azabenzotriazole, N-hydroxysuccinimide, 3-hydroxy-3,4-dihydro-4-oxo-1,2,3-benzotriazine or N-hydroxy-phthalimide); or (2) combinations of dicyclohexyl carbodiimide with 1-hydroxy-7-azabenzotriazole, N-hydroxysuccinimide, 3-hydroxy-3,4-dihydro-4-oxo-1,2,3-benzotriazine or N-hydroxy-phthalimide.
Patent EP-1507859-A2 (EP)
Inventor: RENNER CHRISTOPH
IPC: C07K16/40
Filed: 2003-02-12
Abstract: Chimeric antibodies, as well as fusion proteins which comprise chimeric antibodies, are disclosed. The antibodies bind to GM-CSF, CD-30, and G250 antigen. The fusion proteins include biologically active portions of tumor necrosis factor, or full length tumor necrosis factor. Expression vectors adapted for production of the antibodies, as well as methods for manufacturing these, are also disclosed.
Patent EP-1483247-A2 (EP)
Inventor: GOEHRING R RICHARD
IPC: A61P27/16
Filed: 2003-03-13
Abstract: L'invention concerne une méthode de traitement de troubles répondant au blocage des canaux à ion sodium au moyen de nouveaux composés de pyrimidine substituées par aryle de formule (I) ou d'un sel acceptable sur le plan pharmaceutique ou d'un solvate de ceux-ci. Dans la formule (I), A, R1, R2, R3 et R4 sont définis dans la description. L'invention concerne également l'utilisation des composés de formule I dans le traitement de lésions neuronales engendrées par une ischémie globale et focale, dans le traitement ou la prévention d'états neurodégénératifs, tels que la sclérose latérale amyotrophique (ALS) et dans le traitement, la prévention ou l'amélioration de douleurs aiguës ou chroniques, comme agents anti-tinnitus, comme anti-convulsifiants et comme dépresseurs antimaniaques, comme anesthésiques locaux, comme agents antiarythmiques et dans le traitement ou la prévention de neuropathie diabétique.
Patent EP-1492677-A2 (EP)
Inventor: STAUB RENE
IPC: B44F1/12
Filed: 2003-04-03
Abstract: L'invention concerne un élément de sécurité (1) découpé dans un composite à couches (1) en plastique, destiné à être collé sur un substrat (9). Une couche de réflexion (10) est intégrée entre une couche de moulage (4) et une couche de protection (7) du composite à couches (1), ladite couche de réflexion contenant des structures optiquement actives (5, 6). L'élément de sécurité (2) comporte au moins une caractéristique de sécurité dont la surface présente une macrostructure dans la couche de réflexion (10) et/ou est divisée en une première et une deuxième surface partielle (32, 33). La première surface partielle (32) présente une première structure (5), et une deuxième structure achromatique (6) est moulée dans la deuxième surface partielle (33). Les structures optiquement actives (5, 6) dévient la lumière incidente (11) dans une zone angulaire prédéfinie (e) dans le sens de la réflexion, et contiennent une information visible mais non photocopiable étant donné que les photocopieurs sont aveugles dans la zone angulaire (e).
Patent EP-1530888-A2 (EP)
Inventor: HOFFKNECHT MARC O
IPC: H05B37/02
Filed: 2003-06-19
Abstract: L'invention concerne un système et un procédé de gestion de l'énergie d'éclairage destinés à commander des accessoires d'éclairage dans un bâtiment. Le système utilise des accessoires d'éclairage, des détecteurs de lumière et de présence, des régulateurs d'éclairage personnels et une unité de gestion de l'énergie. L'unité de gestion de l'énergie reçoit des informations des détecteurs de lumière et de présence et du régulateur personnel, et détermine un réglage de luminance optimale pour chaque accessoire d'éclairage, au moyen d'un système coordonné d'objets de zones et d'accessoires. Chaque objet de zones est associé à une zone du bâtiment et chaque objet d'accessoires est associé à un accessoire d'éclairage. Chaque objet de zones veille à ce que le niveau d'éclairage d'un accessoire d'éclairage soit réglé lorsqu'une zone physique est inoccupée. Chaque objet d'accessoires met en oeuvre des détecteurs et des entrées personnelles pour déterminer un niveau de luminance désiré, et utilise un délestage des charges et une compensation de la lumière du jour pour déterminer un niveau de luminance réglé en fonction de la lumière du jour. L'unité de gestion de l'énergie détermine un réglage de luminance optimale en fonction desdits niveaux, afin de réduire au minimum l'énergie requise par les accessoires d'éclairage.
Patent EP-1534732-A2 (EP)
Inventor: WHITE MICHAEL J
IPC: C07J1/00
Filed: 2003-03-21
Abstract: The present invention provides 5-androsten-3beta-ol steroid intermediates and processes for their preparation.
Patent EP-1529334-A2 (EP)
Title: Machine electrique tournante a double excitation autorisant un defluxage modulable
Inventor: AKEMAKOU DOKOU ANTOINE
IPC: H02K21/04
Filed: 2003-08-13
Abstract: L'invention concerne une machine électrique tournante comportant un stator entourant un rotor comportant des aimants permanents d'excitation (20, 24, 26, 30) aptes à établir des flux magnétiques, et des bobinages d'excitation (22, 28), pouvant ou non être excités et engendrer des composantes de flux pouvant s'opposer aux flux engendrés dans les aimants, dans laquelle le nombre (Na) d'aimants et le nombre (Nb) de bobinages d'excitation ainsi que la disposition des bobinages et des aimants les uns par rapport aux autres forment un motif élémentaire (me), ces nombres Na d'aimants, Nb de bobinages et Nme de motifs élémentaires étant modifiables en fonction, d'une part, d'une intensité de base (Ibase) souhaitée dans la machine, cette intensité de base étant déterminée lorsque les bobinages ne sont pas excités et, d'autre part, d'une intensité de modulation (Imod) souhaitée dans la machine, cette intensité de modulation étant déterminée lorsque les bobinages sont excités.
Patent EP-1565391-A2 (EP)
Title: Holding device
Inventor: TURVEY ROBERT R
IPC: A47B88/04
Filed: 2003-11-26
Abstract: A holding device (30) includes a support surface (32) and a first holding portion integral with the support surface (32) and adapted to suspend a bag. A second holding portion is also integral with the support surface (32) and is adapted to suspend a rigid container.
Patent EP-1529271-A2 (EP)
Inventor: HAYASHI RYOJI
IPC: A63H30/04
Filed: 2003-08-08
Abstract: Un problème se pose lorsqu'on veut fabriquer un système de télécommande qui ne permette pas d'établir une combinaison émetteur-machine mobile autre que celle qui a été déterminée dans ce système, un système de télécommande qui assure une équité pour des jeux de guerre et qui soit capable de distinguer une machine mobile et un émetteur combiné dans ce système, même lorsque cette distinction ne peut être établie visuellement. Un émetteur (2) lit des informations de caractéristique (10) sur un support d'enregistrement (3) sur lequel sont enregistrées des informations de caractéristique associées à une machine mobile (1), et il émet des informations vers la machine mobile (1) sous forme de données initiales. Si les informations de caractéristique reçues coïncident avec celles (16) que cette machine mobile possède, cette machine mobile (1) est alors prête à fonctionner. Même si des données de mobilité destinées à la machine mobile (1) sont émises, cette machine mobile (1) ne pourra fonctionner tant que les données initiales contenant les informations de caractéristique (16) ne seront pas reçues. Ce système de télécommande résout ainsi le problème évoqué plus haut.
Patent EP-1576132-A2 (EP)
Title: Acides nucleiques et proteines correspondantes, 273p4b7, utilises dans le traitement et le depistage du cancer
Inventor: CHALLITA-EID PIA M
IPC: A61K39/00
Filed: 2003-08-15
Abstract: L'invention concerne un nouveau gène 273P487 et la protéine qu'il code, ainsi que ses variants. Ledit gène 273P487 présente une expression spécifique aux tissus dans un tissu adulte normal et est exprimé de manière aberrante dans les cancers listés dans le tableau I. Par conséquent, le gène 273P4B7 fournit une cible diagnostique, prognostique, prophylactique et/ou thérapeutique pour le cancer. Ledit gène 273P487 ou un de ses fragments ou la protéine qu'il code ou des variants ou un de leurs fragments peuvent être utilisés pour déclencher une réponse immunitaire humorale ou cellulaire. Selon l'invention, des anticorps ou des lymphocytes T réagissant au gène 273P4B7 peuvent être utilisés dans le cadre d'une immunisation active ou passive.
Patent EP-1539873-A2 (EP)
Inventor: ROTZINGER BRUNO
IPC: C08K5/32
Filed: 2003-09-02
Abstract: L'invention concerne de nouveaux mélanges comprenant i) un stabilisateur de traitement sélectionné dans le groupe renfermant des stabilisateurs d'hydroxylamine, de nitrone, de benzofuran-2-one et/ou un composé de formule I dans laquelle R1 désigne la formule (II), R2 représente un alkyle en C7-C3o et R3 désigne un alkyle en C1-C3o, et ii) un agent antistatique sélectionné dans le groupe renfermant une amine éthoxylée et/ou un amide éthoxylé, utilisés comme stabilisateurs permettant de protéger des matières organiques, notamment des polymères synthétiques, contre une dégradation oxydante, thermique ou induite par la lumière.
Patent EP-1556362-A2 (EP)
Title: Beta-amino heterocyclic dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
Inventor: BIFTU TESFAYE
IPC: A61K31/55
Filed: 2003-10-14
Abstract: The present invention is directed to compounds which are inhibitors of the dipeptidyl peptidase-IV enzyme ("DP-IV inhibitors") and which are useful in the treatment or prevention of diseases in which the dipeptidyl peptidase-IV enzyme is involved, such as diabetes and particularly type 2 diabetes. The invention is also directed to pharmaceutical compositions comprising these compounds and the use of these compounds and compositions in the prevention or treatment of such diseases in which the dipeptidyl peptidase-IV enzyme is involved.
Patent EP-1437245-A2 (EP)
Inventor: MATSUBARA RYO
IPC: F02D45/00
Filed: 2004-01-02
Abstract: A compressor torque estimate device is used for a variable displacement
compressor whose displacement is variable based on a compressor control
signal for estimating a compressor torque of the compressor. The compressor
torque estimate device includes a torque calculator and a corrector. The torque
calculator calculates a torque required for driving the compressor based on the
compressor control signal, thereby obtaining a calculated torque. The corrector
corrects the calculated torque by a procedure of first-order lag, thereby obtaining
a corrected torque. The corrector also estimates the corrected torque to be the
compressor torque.
Patent EP-1477649-A2 (EP)
Inventor: BUERGER FRANK
IPC: F02B31/06
Filed: 2004-02-17
Abstract: The device has a housing for a drive motor that drives a shaft of a final control element via gears, whereby at least one magnet has a functional connection to a fixed contactless switch. Two pin magnets of different polarity are arranged in fixed defined positions relative to the shaft of the final control element and functionally connected to the contactless switch, which produces a signal used to preset the motor's running direction. The device has a housing (2,3) for a drive motor (4) that drives a shaft of a final control element via gears (5), whereby at least one magnet has a functional connection to a fixed contactless switch (16), especially a Hall switch, in the housing so that by moving the magnet the contactless switch detects a pole transition and produces at least one signal for processing by a controller. Two pin magnets (11) of different polarity are arranged in fixed defined positions relative to the shaft of the final control element and functionally connected to the contactless switch, whereby the signal is used to preset the motor's running direction.
Patent EP-1455293-A2 (EP)
Inventor: MATSUURA TOSHIHIRO
IPC: G06Q10/00
Filed: 2004-03-01
Abstract: A user mobile terminal uses an in-train merchandise
purchase program to have ordering information entered. A
merchandise management terminal in the train receives that
ordering information and, if the payment method is cash payment,
transfers the ordering information to a salesperson terminal.
The merchandise management terminal discerns the payment method
from the ordering information and, if the payment method is any
othermethodthancashpayment, requests a merchandise management
server 7 for authentication and, if authentication is given,
transfers the ordering information to the salesperson terminal.
The merchandise management server, having received a notice of
sale completion from the salesperson terminal via the merchandise
management terminal, settles the account with a passenger
requiring any other payment method than cash payment.
Patent EP-1457887-A2 (EP)
Inventor: YAMAUCHI SHINICHIRO
IPC: H04L29/06
Filed: 2004-03-12
Abstract: To provide a data communication apparatus capable of launching
communication applications (1401,1402,1403) without impairing the
real-time characteristic of a communication application (1401,1402,1403)
having a high real-time characteristic in a case where plural
communication applications (1401,1402,1403) including a communication
application (1401,1402,1403) having a high real-time characteristic are present
and to be launched at the same time. 
     Priorities are assigned to data messages DM1 through DM3
to be transmitted from communication applications (1401) through
(1403), respectively, and the assigned priorities are judged upon
receipt of the data messages DM1 through DM3 transmitted from
the communication applications (1401 through 1403),
respectively, so that the data messages are transmitted to a
card (1406) in order of decreasing priorities. In this manner,
priorities are assigned to the data transmitted from the
respective communication applications (1401 through 1403), and
data from the communication applications (1401 through 1403) is
transmitted in order of decreasing priorities.
Patent EP-1577077-A2 (EP)
Inventor: HE YILIANG
IPC: B29C48/32
Filed: 2004-06-09
Abstract: This invention provides a method for manufacturing steel mesh
reinforced plastic composite pipe, which includes: the transverse steel
wires (11) are supplied to the steel mesh welding machine from the
transverse wire reels hung outside the device, a fuzzy resistance
welding technique is adopted to form the steel mesh framework by
welding the transverse steel wires onto the longitudinal steel wires (1)
coming from the longitudinal wire feeder. The formed steel mesh
framework is continuously hauled off and passes through the combining
die (9), the combining die embraces the steel mesh framework and
receives the molted thermoplastic supplied from the side face of the
combining die, the plastic and the steel mesh framework combine inside
the combining die to form the semi-finished pipe, which is hauled off
(7) through the cooling tank (6) to form the finished composite pipe.
This invention also relates to a production line for manufacturing the
composite pipe as well as a piping system formed by connecting the pipes
with joining structures.
Patent EP-1493374-A2 (EP)
Inventor: BARKER DAVID
IPC: A47L9/22
Filed: 2004-06-16
Abstract: A vacuum cleaner 2 having a housing 4 having an inlet 12 and an outlet 54 is
disclosed. Actuation of a motor 46 causes a fan to displace air out of outlet 54, and the
resulting suction upstream of the fan draws dirty air through inlet 12 and inwardly
through walls of filter unit 22. In order to clean the filter unit 22, the user lifts lid 24 by
means of gripping portion 32, and then removes filter unit 22 and dirt collection chamber
16. Because the central portion of the dirt collection chamber 16 is raised, dirt trapped
on the outer surface of filter unit 22 has a tendency to fall into trough regions 40, 42 and
avoids falling into outlet 38. If the motor 46 should accidentally be actuated when the
filter unit 22 is removed, the opening provided by opened lid 24 is nearer to outlet 38
than inlet 12, as a result of which relatively clean air from the atmosphere passes into
recess 36 in preference to dirty air from the inlet 12, thus minimising the risk of the
motor 46 being damaged by dirt.
Patent EP-1519272-A2 (EP)
Inventor: RIEGER GOTTFRIED
IPC: G06F11/30
Filed: 2004-09-28
Abstract: An input element (MST) triggers a safety-related input (ML1). First (MSM1) and second (MSM2) processing units each derive first (DSP1) and second (DSP1a) safety data packets from the safety-related input and compare these with each other. A data interface (MSD) allows one of the safety data packets to be fed into a communications channel (MK) for data packets, in the event of a match. Independent claims are also included for : (a) a mobile operating/observation device with a safety module; and (b) a human-machine interface system with a mobile operating/observation device and a central station for controlling a technical process.
Patent EP-1521263-A2 (EP)
Inventor: JUN JIN-WAN
IPC: G11B5/09
Filed: 2004-10-04
Abstract: A method of performing a retry in a data storage system, and an apparatus using the
same, includes storing information regarding retry parameters corresponding to a position on a
storage medium in response to successfully reading data from the position using the retry
parameters, reading the data from the position in a subsequent read operation according to the
stored information, and rewriting the data at the position.
Patent EP-1570754-A2 (EP)
Inventor: BONFIGLIOLI GIANCARLO
IPC: A23N1/02
Filed: 2004-11-22
Abstract: A System (1) for the extraction of the liquid component
from drupes comprising: a cylinder oil mill (2) suitable
for crushing the drupes to obtain a paste from it; a
plurality of mullers (3) for the homogenisation of the
paste coming from the cylinder oil mill (2); a decanter
(4) for the extraction of the liquid component from the
homogenised paste coming from the mullers (3), where said
plurality of mullers (3) is arranged in parallel, each
muller (3) being suitable for individually receiving the
paste coming from said cylinder oil mill (2).
Patent EP-1449706-A2 (EP)
Inventor: FOSTER THOMAS J
IPC: B60K17/346
Filed: 2004-02-03
Abstract: A common carrier assembly (114) that is particularly adapted for use in
supporting planetary gear sets (80, 82) used in a four-wheel drive vehicle
transfer case (16). The common carrier (114) includes a drive plate (140), a
differential plate (144), and a reduction plate (142). The drive plate (140)
positioned between the reduction planetary gear set (80) and the differential
planetary gear set (82). The drive plate (140) selectively engages a clutch
(118, 180) that operates to position the reduction gear set (80) in various
operation modes.
Patent EP-1493694-A2 (EP)
Inventor: GIOMETTI STEPHEN M
IPC: B65G21/20
Filed: 2004-06-10
Abstract: A machine for inspecting a transparent bottle (12) utilizes a starwheel conveyor (10) to convey non-round bottles through a number of inspection stations before releasing the bottles to an outfeed belt conveyor (24). The starwheel conveyor has a plurality of pockets (14), and as a bottle is about to be released it engages a brush guide rail (30) for rotating and properly orienting a misoriented bottle. The brush (32) of the guide rail has a front edge (36) which is concentric to the axis of the star wheel so that it will interfere with a misoriented bottle. The brush is mounted via upper (34) and lower plates which have a front edge (38) radially spaced from the front edge of the brush at the location where a misoriented non-round bottle (12) will first engage the brush. The radial spacing (S) decreases to zero as the bottle is displaced along the brush. The front edge (36) of the brush (32) is located so that the bottle will have an acceptable orientation at the location where the radial spacing is zero, i.e. where the brush edge (36) merges with the continuing concentric edge (40) of the upper (34) and lower plates.
Patent EP-1512602-A2 (EP)
Inventor: ISHIZU TAKAZUMI
IPC: B61F5/20
Filed: 2004-09-03
Abstract: The invention provides a railway car body that causes less
noise and that can be manufactured easily. The railway car
comprises a subframe (40) disposed below a floor of the car body
with a clearance therebetween, and a bogie (30) disposed below
the subframe (40) with a clearance therebetween, wherein car body
(10) and subframe (40) and/or subframe (40) and bogie (30)
are connected via a center pin (50), the center pin being movable
in the horizontal direction via a ring-shaped cushion rubber.
Patent EP-1519539-A2 (EP)
Inventor: BOOKMAN PETER
IPC: H04L29/06
Filed: 2004-09-28
Abstract: A mobility device for use in a mobility device platform allowing for secure mobile
computing is provided. In an illustrative implementation, an exemplary mobility device platform
comprises a mobility device operable to communicate with at least one computing environment
through a communications interface and wherein the mobility device is operable to process and
store secure web services, a communications network operable to communicate data and
computing applications using web services, and a mobility device management server operable to
generate, process, store, communicate and encrypt web services to the mobility device. The
mobility device may comprise a processing unit, a mobility device communications interface for
interfacing with cooperating computing environments, a memory storage unit, and an operating
system operable to execute web services and/or computing applications.
Patent EP-1544843-A2 (EP)
Inventor: MURATA TOSHIYUKI
IPC: H05B37/02
Filed: 2004-12-10
Abstract: By detecting surrounding illuminance with a reception unit (340) provided on a
display controller (300), a change in the illuminance is recognized. A microcomputer
(370) determines presence/absence of user's input operation through a terminal operating
section (330) of a display controller (300). When recognizing the input operation, the
microcomputer (370) restricts a process of calculating, with a luminance controller (360),
a luminance control value that sets the luminance of an image display (320) to the
luminance corresponding to a change in the illuminance and outputting the luminance
control value to the image display (320) until a predetermined time has elapsed even if the
illuminance has changed during the predetermined time. This prevents a situation where
a user cannot see clearly a display window due to the change in the luminance at input
operation time, thereby facilitating the input operation.