baber/WOPTO huggingface dataset:
Patent SK-47794-A3 (SK)
Title: Chinolyl-dihydropyridinecarboxylic acid esters, method of their production, medicines containing these matters, method of their production and using of these compounds
Inventor: STOLTEFUSS JURGEN
IPC: C07D401/04
Filed: 1994-04-26
Abstract: The invention relates to novel 4-quinolyldihydropyridine esters of the general formula (I) <IMAGE>  in which  R1 to R6 have the meaning given in the description, processes for their preparation and their use in medicaments, in particular in compositions for the treatment of cardiovascular disorders.
Patent SK-54298-A3 (SK)
Title: (-)-cis-6(s)-phenyl-5(r)[4-(2-pyrrolidin-1-ylethoxy)phenyl]- -5,6,7,8-tetrahydronaphthalen-2-ol d-tartrate
Inventor: CHIU CHARLES K
IPC: C07D295/092
Filed: 1996-10-04
Abstract: Disclosed is a process for the preparation of (-)cis-6(S)- phenyl-5(R)-[4-(2-pyrrolidin-1-ylethoxy)phenyl]-5,6,7,8- tetrahydronaphthalen-2-ol D-tartrate, wherein 1) racemic or partly optically enriched cis-6(S)-phenyl-5(R)-[4-(2- pyrrolidin-1-ylethoxy)phenyl]-5,6,7,8-tetrahydronaphthalen-2-ol is diluted in a boiling aqueous ethanol solution forming the first solution; 2) to the first solution equimol amount of D-tartaric acid diluted in aqueous ethanol solution is added, forming the second solution; 3) second solution is cooled; and 4) product formed in 3) is gathered. Disclosed are also pharmaceutical preparations based on this compound.
Patent SK-55795-A3 (SK)
Title: Method for preparing taxane derivatives
Inventor: DENIS JEAN-NOEL
IPC: C07D413/12
Filed: 1993-10-28
Abstract: A method for preparing taxane derivatives of general formula (I) by esterifying protected baccatine III or protected 10-deacetyl baccatin III with an acid of general formula (II). In general formulae (I) and (II), Ar is an aryl radical; R1 and R2 which are the same or different, are a hydrogen atom, an alkyl, phenylalkyl, phenyl, alkoxyphenyl or dialkoxyphenyl radical, or R1 and R2, together with the carbon atom to which they are attached, form a 4-7 membered ring; R3 is an acetyl radical or a hydroxy function protective grouping, and R4 is a hydroxy function protective grouping; R is a phenyl radical or a radical of formula R5-O- wherein R5- is an alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, phenyl or saturated or unsaturated nitrogenous heterocylcyl radical. The products of general formula (I) are particularly useful for preparing taxol, Taxotere and analogues thereof having remarkable antitumor properties.
Patent CH-608325G-A3 (CH)
Title: Wristwatch and method of encasing this watch
IPC: G04B37/02
Filed: 1975-05-05
Abstract: The watch includes no movable piece but comprises an electronic module and a light-emitting diode or liquid-crystal display device, which are housed in a casing. With a view to increasing the reliability of the watch, all of the space left free in the casing by the module and the display device is filled with a dielectric liquid which is chemically stable and inert with respect to materials with which it is in contact.
Patent CZ-823286-A3 (CZ)
Inventor: FANCOVIC KAROL ING CSC
IPC: C07C51/34
Filed: 1986-11-13
Abstract: Monokarboxylové kyseliny Ci - C21 sa pripravujú ozonizá*
ciou alkenických surovin obsahujúcich dva až dvadsaťdva
uhlíkových atómov v molekule, v prostředí monokarboxylových
kyselin Ct - C21 cez peroxidické medziprodukty,
1 1 ktoré sa oxidačně rozkládajú a izolujú destiláciou, alebo
rektifikáciou s výhodou za zníženého tlaku. Monokarboxy*
lově kyseliny Ci - C21 sa před izoláciou rozdelia na časť,
»
ktorá sa použije na rozpustenie alkénov C2 - C22 a postupuje
ako násada do ďaíšieho cyklu spracovania, a časť ktorá
představuje produkt a postupuje do ďeíiaceho procesu. Spóf
sob je možné kontinualizovaf. Vynález má široké uplatne-
?' nie aj pře přípravu iných derivátov monokarboxylových
kyselin z rózných aj substituovaných alkénov.
Patent CZ-101296-A3 (CZ)
Title: Massaging machine for foodstuff articles
Inventor: SUHNER WALTER
IPC: A22C9/00
Filed: 1996-04-05
Abstract: Foodstuff products, particularly for salted meat products, are treated in a massage tumbler comprising a driven drum (2) and flight sections (8) for moving the pieces of meat in the drum. An insert (10) is provided in the drum for additional movement and pref. consists of a member fitted rigidly in the drum w.r.t. the axis of rotation having \- one projecting arm (26). Pref. the arm has a rod-shaped section (27) and a plate-shaped section (28). The arm may be in the form of a knife and may be detachably fastened on one end to a drum suspension (17) and on the other end to the drum cover of an aperture (6).
Patent CZ-173695-A3 (CZ)
Title: Cystatin containing oral and eatable preparations against dental decay
Inventor: REVIS GEORGE JOE
IPC: A23L2/66
Filed: 1993-12-13
Abstract: The present invention relates to oral and edible compositions intended to provide an anticaries benefit. The primary active ingredient in these compositions is a protein selected from the group consisting of cystatin S, cystatin SA, cystatin SN and mixtures thereof which are salivary proteins. Also included are fragments of the proteins which may be used in place of the total proteins.
Patent CZ-183497-A3 (CZ)
Title: Thiazolidinone compounds, process of their preparation and pharmaceutical composition containing thereof
Inventor: ISHIHARA SADAO
IPC: C07D413/04
Filed: 1995-12-13
Abstract: Thiazolidinone compounds having the general formula: <CHEM> Äwherein W represents a sulfur atom or an oxygen atom, and X represents a group having the formula: -N(R<1>)-; or   X represents a sulfur atom or an oxygen atom, and W represents a group having the formula: -N(R<1>)-; R<1> represents a hydrogen atom, an alkyl group or a substituted alkyl group; R<2> and R<3> may be the same or different and each represents a hydrogen atom, an alkyl group, a substituted alkyl group, an aryl group or a 5- or 6-membered aromatic heterocyclic group; R<4> represents a hydrogen atom, an alkyl group or a substituted C1-C4 alkyl group; R<5> represents a substituted cycloalkyl group optionally containing a nitrogen atom Äsaid substituent is essentially a group having the formula: -B-ONO2 (wherein B represents a single bond or an alkylene group) and optionally an alkyl groupÜ; and A represents a single bond or an alkylene group; Ü or pharmacologically acceptable salts thereof.  ÄEffectÜ   The compounds have an excellent anti-angina pectoris action and are useful as a therapeutic or preventing agent for angina pectoris.
Patent CZ-186996-A3 (CZ)
Title: Method of selective provocation of methionine insufficiency for malignant cells of mammals
Inventor: NOBORI TSUTOMU
IPC: A61K47/48
Filed: 1994-12-22
Abstract: An improved method for chemotherapy of mammalian malignant cells which have an absolute requirement for methionine but lack methylthioadenosine phosphorylase (MTAse). The method comprises detection of MTAse negative cells in a mammal, administration of methionine  gamma -lyase in sufficient amounts to reduce the volume of MTAse negative cells in the mammal, and co-administration of methylthioadenosine in amounts sufficient to ensure the continued availability of methionine to the mammal's non-malignant cells. Means for detection of MTAse negative cells are provided. Means for production and use of recombinant chemotherapeutic agents are also provided.
Patent CZ-200836-A3 (CZ)
Inventor: HAMAMATSU TOYOHIRO
IPC: G02B5/02
Filed: 2008-01-23
Abstract: Desticka rozptylující svetlo (3) podle tohoto vynálezu zahrnuje základní vrstvu (8), která je zhotovena z pryskyricné kompozice obsahující cástecky rozptylující svetlo ve množství 0,1 hmotnostních dílu až 5 hmotnostních dílu na 100 hmotnostních dílupropylenového polymeru, a povrchovou vrstvu (9), která je nanesena na jednom nebo na obou površích základní vrstvy (8) tak, že s nimi tvorí jeden celek, pricemž tato povrchová vrstva (9) je zhotovenaz pryskyricné kompozice obsahující cástecky se stredním prumerem cástecek stanoveným z integrovaného objemu 10 až 200 .mi.m ve množství 5 až 50 hmotnostních dílu na 100 hmotnostních dílu propylenového polymeru. Desticka rozptylující svetlo je lehká,má dostatecnou pevnost a není deformována teplem nebo vzdušnou vlhkostí, má dostatecnou tvrdost povrchu a má také vynikající odolnost proti poškrábání.
Patent CZ-201535-A3 (CZ)
Inventor: ŽVÁTORA PAVEL
IPC: C07B57/00
Filed: 2015-01-21
Abstract: Způsob provedení isolace a čištění bedaquilinu (Ia) ze směsi stereoizomerů 6-bromo-2-methoxy-chinolin-3-yl)-4-dimetylamino-2-(1-naftyl)-1-fenyl-butan-2-olu značených I-rac, kde se jedná o směs stereoizomerů vzorců Ia, Ib, a II-rac, kde se jedná o směs stereoizomerů vzorců IIa, IIb, s libovolných poměrem jednotlivých složek směsi vyznačující se tím, že je výše uvedená směs rozpuštěna společně s deriváty 1,3 propandiol hydrogen fosfátu vzorce IV, kde R1, R2, R3 značí nezávisle na sobě vodík, halogen, alkyl C1-C6, aryl, naftyl, fenyl, a s výhodou halogenovaný či libovolně substituovaný fenyl, a vzniklá sůl je krystalizována.
Patent CZ-238095-A3 (CZ)
Title: Perforated plastic foil, process of its production, apparatus for making the same and absorption article employing said foil
Inventor: MORRIS YANG CHUNG-YUN
IPC: B32B7/02
Filed: 1995-09-14
Abstract: An apertured plastic film (10) having a plurality of wales (12), a plurality of sloped side walls (14) extending from the wales (12) and a plurality of clusters of irregular micro-holes (18) defined by a network of fiber-like elements (20), each cluster of irregular micro-holes (18) being connected between at least two of the sloped side walls (14). The film also has a plurality of rows of undulating ribs (22) having the network of wales (12) connected to opposite sides of the ribs (22) and extending in a transverse direction from the ribs (22). The films of the invention are useful as covering materials for absorbent products such as diapers, wound dressings and sanitary napkins. <IMAGE>
Patent CZ-245098-A3 (CZ)
Title: Hand-operated device for transferring film from supporting foil to base
Inventor: MANUSCH CHRISTOPH
IPC: B05C17/00
Filed: 1997-01-27
Abstract: PCT No. PCT/EP97/00352 Sec. 371 Date Feb. 24, 1999 Sec. 102(e) Date Feb. 24, 1999 PCT Filed Jan. 27, 1997 PCT Pub. No. WO97/29036 PCT Pub. Date Aug. 14, 1997A hand-held device for transferring a film from a carrier tape to a substrate includes an applicator with an end projecting from a housing around which the carrier tape coming from a supply roll is guided to a take-up spool and on which contact surfaces are provided for the "pull" and "push" operating modes of the device, the carrier tape being pressed against the substrate by the contact surfaces for the purpose of transferring the film. The applicator contains two application toes which are separated from one another by an empty space and each of which carries one of the two contact surfaces.
Patent CZ-282897-A3 (CZ)
Title: N-benzylazolium derivatives
Inventor: ICHIHARA SHIGEYASU
IPC: C07D405/06
Filed: 1997-09-08
Abstract: N-Benzylazolium derivatives of the general formula (I), wherein Q is the remainder of an azole compound of the formula II  possessing antifungal activity; Z is nitrogen or methine; R1 and R2 are each independently a hydrogen atom or a group -OY [in which Y is a group easily hydrolyzable under physiological condition]; R3 and R4 are each independently a hydrogen or halogen atom, lower alkyl, lower alkoxy, lower alkylthio, (lower alkylcarbonyl)thiomethyl, carboxy or methoxycarbonyl; and X- is a pharmaceutically acceptable anion, as well as salts, hydrates or solvates of the compounds of the general formula (I) have antiftngal properties.
Patent CZ-324895-A3 (CZ)
Title: Antitumor preparation
Inventor: BICHER HAIM I
IPC: A61K33/243
Filed: 1994-05-27
Abstract: Anti-cancer compositions containing chiral monosaccharides and methods of their use are disclosed herein. The compositions, exhibiting cytostatic and cytotoxic properties with regard to neoplastic cells are formulated using the L-isomeric form of monosaccharides. A preferred embodiment of the invention employs the L-isomeric form of glucose with a pharmaceutically acceptable carrier. The compositions may be used alone or as an adjunct to other forms of cancer therapy. They are useful in combination with all major forms of cancer therapy including surgery, biological and chemical therapies, radiation therapy, and hyperthermia. In addition to increasing the mortality rate of neoplastic cells, these compositions can reduce the metastatic potential of the tumor, and slow the growth of the malignancy.
Patent CZ-9903757-A3 (CZ)
Title: Novel Bacillus strain for controlling diseases of plants and Diabrotica undecimpunctata chrysomel
Inventor: HEINS SHERRY DARLENE
IPC: A01N63/50
Filed: 1998-05-08
Abstract: The present invention relates to a novel antibiotic-producing and metabolite-producing Bacillus subtilis strain that exhibits insecticidal, antifungal and antibacterial activity. The supernatant of this novel strain contains effective insecticidal, antifungal and antibacterial agents. Also included in the invention is a solvent extractable, small molecular weight (<10,000 daltons) corn rootworm-active metabolite produced in the supernatant. Also included in the invention are methods of protecting or treating plants from fungal and bacterial infections and corn rootworm infestations comprising the step of applying to the plant an effective amount of the antibiotic/metabolite-producing novel Bacillus subtilis strain, the antibiotic/metabolite produced by the novel Bacillus subtilis strain or a combination thereof, optionally further comprising another antibiotic-producing bacterial strain and/or a chemical pesticide. The invention also includes methods of preventing or treating fungal and bacterial infections using whole broth cultures or supernatants obtained from cultures of the novel Bacillus subtilis strain alone or in combination with chemical pesticides and/or other biocontrol agents. The invention also includes novel antifungal and antibacterial compounds designated agrastatins and a novel combination comprising an A-type iturin, a plipastatin, a surfactin and an agrastatin. Methods of treating or protecting plants from fungal and bacterial infections and corn rootworm infestations comprising administering the novel agrastatins and the novel combination comprising an A-type iturin, a plipastatin, a surfactin and an agrastatin are provided.
Patent CZ-424199-A3 (CZ)
Title: Fungicidal mixtures
Inventor: SCHELBERGER KLAUS
IPC: C07C251/48
Filed: 1998-05-13
Abstract: A fungicidal mixture comprisesa) a phenyl benzyl ether derivative of the formula I.a, I.b or I.c, and/or a carbamate of the formula Idwhere X is CH or N, n is 0, 1 or 2 and R is halogen, C1-C4-alkyl or C1-C4-haloalkyl, it being possible for the radicals R to be different if n is 2, or a salt or adduct thereof,and(b) a N-acetonylbenzamide of the formula II where:R1 and R3 independently of one another are each halogen or C1-C4-alkyl;R2 is cyano, C1-C4-alkyl, C2-C4-alkenyl, C2-C4-alkynyl or C1-C4-alkoxy;R4 is hydrogen or C1-C4-alkyl;R5 is C2-C4-alkyl;R6 is thiocyano, isothiocyano or halogen,or a salt or adduct thereof,in a synergistically effective amount.
Patent CZ-452499-A3 (CZ)
Title: Absorptive interlabial preparation
Inventor: OSBORN THOMAS W III
IPC: A61F13/20
Filed: 1998-06-15
Abstract: An absorbent interlabial device worn by female wearers for catamenial purposes, incontinence protection, or both, is disclosed. The absorbent interlabial device of the present invention includes a liquid pervious topsheet, a liquid impervious backsheet, and an absorbent core positioned between the two. The length of the device is between about 60 mm and about 130 mm. The width is between about 25 mm and 50 mm. The device has an axis of preferred bending along its longitudinal centerline. When folded along the axis and inserted into the wearer's interlabial space, the topsheet maintains contact with the walls of the wearer's labia. A method of using a system of feminine hygiene products is also disclosed. The system includes the use of an absorbent interlabial device in combination with a sanitary napkin. The absorbent interlabial device of the present invention may also be used in combination with an absorbent tampon. The absorbent interlabial device may be packaged in a common package with a sanitary napkin or a tampon as a feminine hygiene kit.
Patent ES-8800956-A3 (ES)
Title: Benzoyl D-ribofuranosyl triazole carboxamide prepn.
IPC: A61K31/70
Filed: 1987-01-09
Abstract: 1-(5-O-benzoyl beta-D-ribofuranosyl) 1,2,4-triazole 3-carboxamide for pharmacological use for its anti-viral activity, is made by amidation of the methyl ester of 1-(2,3,5-tri-O-benzoyl beta-D-ribofuracosyl)1,2,4-triazole 3-carboxylic acid, by treatment in a solvent, e.g. methanol, satd. with anhydrous ammonia. The prod. is evaporated to dryness and recrystallised from a medium e.g. aq. ethanol.
Patent SK-327992-A3 (SK)
Title: Method of manufacture of magnetic steel belt top casted
Inventor: BAVAY JEAN-CLAUDE
IPC: B22D11/06
Filed: 1992-10-30
Abstract: Process for manufacturing a magnetic steel strip which has a thickness of less than 5 mm and contains, in composition by weight, more than 2 % of silicon, less than 0.1 % of carbon and elements which inhibit secondary recrystallisation in an appropriate quantity, the remainder being iron, obtained by direct casting on a cylinder or between two cylinders (5, 6), which process is characterised in that a crystallisation structure is created, comprising {110} <001> oriented grains as a skin, that is to say at the surface of the quenching zone, due to the abrupt cooling of the steel in contact with the roll(s) (5, 6), the surface temperature of which is lower than 400 DEG C. The steel strip consists of two zones (8, 9) at the side of the middle zone (7).
Patent SK-329292-A3 (SK)
Title: Covered goods wagon or container
Inventor: ALTMANN HELMUT
IPC: B61D3/18
Filed: 1992-06-19
Abstract: The goods wagon or container has a lower loading floor (2) on whose longitudinal sides a plurality of columns (3) are attached. Perpendicular guides (10) with flanges (15) which protrude in the longitudinal direction of the goods wagon or container are constructed on the columns (3) and engage in pairs over one perpendicular edge (16) each of lower side wall parts (11) and upper side wall parts (7). The lower side wall parts (11) are attached to the columns (3) via the guides (10). The upper side wall parts (7) are permanently connected to a roof (6) and are guided in the guides (10) so that they can be vertically adjusted together with the roof (6). The upper and lower side wall parts (7, 11) of each side wall (5) are arranged in every position of the roof (6) at least approximately in a common perpendicular plane and when the roof (6) is raised they clear an opening (12) in the same plane. Therefore, the loading space of the goods wagon or container is well ventilated and accessible to natural light when the roof (5) is raised. Additional openings (12') which are constructed between the loading floor (2) and the lower side wall parts (11) and are closed with slides (14) when the roof (6) is lowered, open when the roof (6) is raised by virtue of the fact that said roof is connected to the slides (14) by means of a linkage (13).
Patent SK-792021-A3 (SK)
Inventor: IĽKOVIČ SERGEJ
IPC: G01D3/00
Filed: 2021-10-29
Abstract: Opísaný je modulárny merací systém, ktorý pozostáva z modulu centrálnej jednotky a senzorických a aktuátorových jednotiek. Každá senzorická/aktuátorová jednotka obsahuje senzor/aktuátor a mikrokontrolér a komunikuje s modulom centrálnej jednotky. Na ovládanie a nastavenie zariadenia sa využíva PC, tablet alebo smartfón, ktorý sa prostredníctvom Wi-Fi technológie pripája na modul centrálnej jednotky a využíva sa na nastavenie a spustenie merania a následné zobrazenie nameraných údajov. Senzorická a aktuátorová jednotka modulárneho meracieho systému zabezpečuje posielanie nameraných hodnôt do/z modulu centrálnej jednotky, zabezpečuje jeho pripojenie do systému, manažuje rozsahy a pracuje s viacerými meranými veličinami a aktuátormi.
Patent BE-1000845-A3 (BE)
Title: Plaque pare-feu, et paroi coupe-feu fabriquee a partir de telles plaques.
Inventor: PAUL HANS-GUNTER
IPC: C04B26/12
Filed: 1987-12-15
Granted: 1989-04-18
Abstract: Une plaque pare-feu renferme de 10 % à 14% en volume d'un liant organique, de 40% à 60% en volume de microstructures minérales creuses, et de 26% à 50% en volume d'hydroxyde d'aluminium. La paroi coupe-feu est fabriquée par collage ou par appareillage cimenté de telles plaques.
Patent BE-1006736-A3 (BE)
Title: Polyamide compound
Inventor: FLIPPO PETER
IPC: C08K5/3492
Filed: 1993-02-05
Granted: 1994-11-29
Abstract: The invention relates to a flame extinguishing, non -dripping polyamidecompound, that comprises polyamides and additives whereby the compound, withregard to the total compound, has a 1-40 weight percent melamine cyanurateand 0.01-5.0 weight percent powder form polytetrafluroethylene as additives.Preferably this compound does not contain any inorganic fibres or fillers.The polyamide compound complies with the VO classification in accordancewith UL94.
Patent BE-1010628-A3 (BE)
Title: Method for improvement of the action of a catalyst and catalytic reactor with improved functioning
IPC: B01J19/24
Filed: 1996-09-17
Granted: 1998-11-03
Abstract: Method for the improvement of the action of a catalyst of the type that comprises one or more elements that are formed by a substrate that forms channels or passages, a specific feature being that low frequency sound waves are distributed in the channels (9) or passages for the catalyst elements (8). To this end, a catalytic reactor built in accordance with the invention contains at least one source (10) of low frequency waves.<IMAGE>
Patent BE-1010933-A3 (BE)
Title: Samenstelling voor het behandelen en voorkomen van comedovorming.
IPC: A61K8/92
Filed: 1997-02-18
Granted: 1999-03-02
Abstract: De uitvinding betreft een samenstelling voor het behandelen en voorkomen van comedovorming, welke samenstelling een gel en linolzuur bevat waarbij het linolzuur aanwezig is als linolzuur bevattende saffloerolie. De samenstelling bevat bij voorkeur 5 - 20 gew. % saffloerolie en 2,5 - 20 gew. % linolzuur. De uitvinding betreft eveneens een werkwijze voor het bereiden van genoemde samenstelling en het gebruik van genoemde samenstelling voor cosmetische toepassingen.