baber/WOPTO huggingface dataset:
Patent IE-39440-L (IE)
Title: Benzoyl benzoic acid derivatives
IPC: C07C313/00
Filed: 1974-05-29
Abstract: 1443714 Benzoyl-benzoic acids LEO PHARMACEUTICAL PRODUCTS Ltd AS 11 June 1974 [22 June 1973] 29875/73 Heading C2C [Also in Division A5] Novel compounds I in which R 1 represents a straight or branched C 1 -C 6 alkyl, alkenyl or alkynyl radical which may be substituted with one or more halogen atoms or halo-C 1-6 alkyl, amino, alkylated amino, acylated amino, hydroxy, etherified hydroxy, esterified hydroxy or etherified mercapto radicals, or a C 1 -C 3 alkyl radical substituted with phenyl, halophenyl, trifluoromethylphenyl, (lower alkoxy) phenyl, or with a 5- or 6-membered heterocyclic ring containing not more than two heteroatoms selected from oxygen, sulphur and nitrogen; R 2 stands for hydrogen or a straight or branched C 1 -C 6 alkyl, alkenyl, alkynyl or alkoxy radical which may be substituted with one or more halogen atoms or halo-C 1 -C 6 alkyl, amino, alkylated amino, acylated amino, hydroxy, etherified hydroxy, esterified hydroxy or etherified mercapto radicals; Ar stands for a phenyl radical which may be substituted by one or more halogen atoms, or C 1-6 alkyl, halo-C 1-6 alkyl, amino, alkylated amino, acylated alkyl, or amino, OH, etherified OH, esterified OH or etherified mercapto radicals; and Y stands for oxygen, sulphur or a methylene radical; and pharmaceutically acceptable, non-toxic salts and esters thereof, are prepared by acylation of a compound II or an ester thereof, followed, if desired by saponification of a resulting ester or esterification of a resulting acid. 4-Benzoyl-3-benzyloxy- 5 - dimethylaminoacetamidobenzoic acid is prepared by reacting a corresponding 5-chloroacetamido compound with dimethylamine. Pharmaceutical compositions having diuretic and/or saluretic activity, for oral, enteral or parenteral administration, comprise one of the above novel compounds together with a pharmaceutical carrier and, optionally, other pharmaceutically active compounds.
[GB1443714A]
Patent IE-791366-L (IE)
Title: Fosfomycin derivatives.
IPC: A61P31/04
Filed: 1979-08-08
Abstract: Bis-(2-ammonium-2-hydroxymethyl-1,3-propanediol)(2R-cis)-(3-methyloxir anyl)-phosphonate showing high bioavailability and tolerability is disclosed, as well as a method for preparing same from (2R-cis)-(3-methyloxiranyl)-phosphoric acid, or a salt thereof, and 2-amino-2-hydroxymethyl-1,3-propanediol, or a salt thereof. Pharmaceutical compositions containing the novel bis-phosphonate; useful for clinical forms of urinary and respiratory infections, are also disclosed.
[US4727065A]
Patent IE-831534-L (IE)
Title: Detergent compositions
IPC: C11D7/60
Filed: 1983-06-30
Abstract: This invention relates to bleaching compositions that provide effective and efficient surface bleaching of textiles over a wide range of bleach solution temperatures. Surface bleaching of textiles is bleaching wherein the bleaching mechanism takes place on the textile surface and, thereby, removes stains and/or soils. The bleaching compositions within the invention contain peroxygen bleaches capable of yielding hydrogen peroxide in aqueous solutions and specific bleach activators at specific molar ratios of hydrogen peroxide to bleach activator. In a highly preferred embodiment the bleaching compositions within the invention are detergent compositions.
[US4412934A]
Patent IE-34280-L (IE)
Title: Cylinder lock mechanism
IPC: E05B27/06
Filed: 1969-11-28
Abstract: A cylinder lock which comprises a core having a key slot. A key is to be inserted in the key slot and includes wide faces for receiving recesses therein. Tumblers are provided in the core adjusted by the key with the recesses. A housing receives the core and includes a flange extending radially to the core and has bores. The key slot is disposed in symmetric cross position to the flange. At least two rows of the tumblers are arranged in the flange. The tumblers have a non-round cross-section and sit non-rotatably in the bores of the flange.
[US3824818A]
Patent IE-902276-L (IE)
Title: Serpin variants
IPC: A61K38/00
Filed: 1990-06-22
Abstract: Modified antithrombin III variants are developed which contain amino acid substitutions in the region comprising amino acids 384-396. In this region one or more amino acids are replaced by the corresponding amino acid(s) grouped around the factor Xa cleavage site in factor II related to the formation of meizothrombin. These amino acid substitutions result in altered heparin-dependent inhibitory effect of the modified antithrombin III vis-à-vis the factors IIa and Xa, respectively.
[WO9100291A1]
Patent IE-832376-L (IE)
Title: Electrical connector assembly
IPC: H05K7/14
Filed: 1983-10-10
Abstract: An electrical connector assembly, comprises an assembly frame defining an aperture with bars 10, 11 on two opposite sides of the aperture, the bars 10, 11 securing between them electrical connectors 20 which are fixedly located in the aperture by means of interengaging male and female portions 101, 111 provided on the bars 10, 11 and the connectors 20, and which connectors 20 are located with respect to the plane of the aperture by at least one support rail 104 against which the connectors 20 abut. <IMAGE>
[GB2129231A]
Patent IE-812499-L (IE)
Title: Cranial drill
IPC: A61B17/00
Filed: 1981-10-23
Abstract: A completely disposable, permanently assembled drill for perforating bone structures, which includes a generally annular drill body. A primary drill member is slidably and rotatably received in the distal end of the drill body. A driver is slidably and rotatably received in the proximal end of said drill body. A pin and slot-type spring biased clutch is disposed on the confronting surfaces of the drill member and driver. The pin of the clutch projects through the triangular openings and the sidewall of the drill body so as to limit the throw of the clutch and to link the drill body and drill member together. The interaction of the pin against the triangular side of the slot in the drill body produces a component of force which tends to urge the clutch apart. When the drill is placed against the bone structure with a force sufficient to overcome the spring bias, the clutch will engage and the driver and drill member and the drill body will rotate together. The counterbore on the drill body provides a support for the drill mechanism so that the drill member may release when it penetrates the bone structure without having the remainder of the drill move in the direction toward the cranial cavity. The sleeve holds the drill body and driver together and is made of a material that degrades when subjected to sterilization.
[US4362161A]
Patent IE-43208-L (IE)
Title: Xanthine derivatives
IPC: A61K31/522
Filed: 1975-12-19
Abstract: Compounds of the formula <IMAGE> wherein R is methyl or ethyl, R1 is methyl, ethyl or <IMAGE> and R2 is methyl, ethyl, <IMAGE> <IMAGE> <IMAGE> where Alk is alkyl of 1 to 4 carbon atoms, Q is ethyl, propyl, isopropyl or 2-hydroxy-propyl, A is 3-phenoxy-2-hydroxy-propyl, where the phenyl ring is substituted in the o-position by hydroxy, methoxy, n-hexyloxy or benzyloxy, B is alkyl of 1 to 4 carbon atoms, phenyl, p-methyl-phenyl, 3-phenyl-3-hydroxy-isopropyl or A, as defined above, and N IS AN INTEGER FROM 2 TO 6, INCLUSIVE, PROVIDED, HOWEVER, THAT ONE OF R1 and R2 must be methyl or ethyl and the other has one of the other respective meanings indicated; and non-toxic, pharmacologically acceptable acid addition salts thereof. The compounds as well as the salts are useful as peripheral vasodilators.
[US3998953A]
Patent IE-842839-L (IE)
Title: Digital switching signal circuit
IPC: H03K17/687
Filed: 1984-11-05
Abstract: In a pushpull switching circuit, whose output transistors are controlled by complementary control signals, that one of the gate electrodes which carries a sec low sec signal is kept just at the threshold voltage of the output transistor to be cut off by means of a transistor (substantially) identical to the output transistors, the gate electrode and the main electrode (drain) of this transistor being interconnected. The junction (of this gate and this drain) is connected to sources (main electrodes) of two cross-coupled with gate and drain transistors, which are connected by their drain to the gate electrodes of the respective output reansistors. 
[EP0141474A2]
Patent IE-892879-L (IE)
Title: Isocyanate reactive polymers having imino/enamine¹functionality
IPC: C08G18/30
Filed: 1989-09-08
Abstract: Isocyanate-reactive prepolymers having imino/enamine functionality are made by reacting an isocyanate-terminated urethane prepolymer with compounds having imine or enamine functionality. These prepolymers are useful in reaction injection molding systems as isocyanate-reactive ingredients.
[EP0359456A1]
Patent IE-894111-L (IE)
Title: Phosphinic acid substituted steroids as inhibitors of¹steroid 5ó-reductase
IPC: A61P43/00
Filed: 1989-12-20
Abstract: Compounds of structure (I) <CHEM> in which the dotted lines indicate the optional presence of double bonds and, inter alia, R<1> is H, R<2> is H or CH3 and R<3> is H, hydroxy or acetoxy; processes for their preparation, pharmaceutical compositions containing them and their use in medicine as inhibitors of 5- alpha -reductase.
[EP0375349A1]
Patent NO-780621-L (NO)
Title: Fremgangsmaate og varmeanlegg for forbrenning av fast brensel
Inventor: STAEHLI HANS
IPC: F23K3/00
Filed: 1978-02-23
Abstract: Fremgangsmåte og varmeanlegg for forbrenning av fast brensel
Patent NO-833847-L (NO)
Inventor: HASHISH MOHAMED A
IPC: B26F3/00
Filed: 1983-10-21
Abstract: In method and apparatus for producing a coherent stream of high velocity abrasive laden liquid, the method includes allowing particles of abrasive to assume the direction and velocity of a high velocity jet (22) of liquid. The method allows concentration of particles in the centre of the flow of liquid to reduce nozzle wear and increase cutting efficiency. The apparatus includes a nozzle (21) having a converging section (26, 27) attached to a straight section (28) that is sufficiently large that the abrasive particles approach the velocity of the fluid jet before leaving the exit (29) of the nozzle.
Patent NO-850110-L (NO)
Inventor: TOUSSAINT MICHEL GEORGES
IPC: F23J15/00
Filed: 1985-01-10
Abstract: 1. A method of diluting a gas or a mixture of gases with air before discharge to atmosphere, by means of a device comprising a shaped body (20) forming a venturi which is open to the atmosphere at both ends, said gas or mixture of gases being injected under pressure at the upstream end thereof, method characterised in that said gas or mixture of gases is injected into said body in the form of a layer of annular cross-section by means of at least one set of injection tubes (21), the circular orifices (24) of which are arranged in a ring at the upstream part of said body (20) forming a venturi.
Patent NO-883342-L (NO)
Inventor: BURNOUF MYRIANA
IPC: A61K35/16
Filed: 1988-07-28
Abstract: Concentrate of thrombin-coagulable proteins, possessing a fibrinogen content of more than 70% and a sufficient amount of endogeneous factor XIII. It can be solubilised at room temperature. Its preparation involves at least one step of precipitation in the cold state with dilute ethanol and employs whole plasma as the starting material. the concentrate makes it possible, in particular, to obtain an injectable fibrinogen and a biological glue. <IMAGE>
Patent NO-884406-L (NO)
Inventor: TSUKAMOTO SHIN-ICHI
IPC: A61K31/55
Filed: 1988-10-04
Abstract: Heterocyclic spiro compounds of formula <CHEM> @ @C represents a piperidine ring of which the nitrogene atom may have substituent(s) selected from alkyl, alkanoyl and alkoxycarbonyl and/or may be connected to a ring carbon (other than the common carbon atom of the spiro structure) via an alkylene bridging group;  X represents an oxygen of sulfur atom;    Y represents a carbonyl group (- @-), a thiocarbonyl group (@@@),    a group of the formula @CH-R<5>, a group of the formula <CHEM>  or a group of the formula <CHEM>  wherein Alk is alkylene and Z<1> and Z<2> are the same or different and selected from oxygen and sulfur atoms; R<1>, R<2> and R<3> are the same of different and selected from a hydrogen atom and alkyl R<4> represents a hydrogen atom or alkyl, carboxy, alkoxycarbonyl, or alkanoyl group; R<5> represents a halogen atom or a hydroxyl, mercapto, alkoxy, alkylthio, alkanoyloxy, or alkanoylthio group; and R<6> and R<7> are the same of different and selected from a hydrogen atom and alkyl groups. The above compounds act upon muscarinic acetylcholine receptors, thereby activating the acetylcholine nervous functions in the central nervous system.
Patent NO-893322-L (NO)
Inventor: GERHARDT WOLFGANG
IPC: B01D53/14
Filed: 1989-08-18
Abstract: The present invention relates to a process for removing CO2 and possibly H2S from a gas containing CO2 and possibly H2S by means of an absorption fluid, wherein the gas containing CO2 and possibly H2S is treated in an absorption zone with the absorption fluid, the treated gas is extracted from the absorption zone, the absorption fluid laden with CO2 and possibly H2S is then regenerated by expanding the absorption fluid laden with CO2 and possibly H2S in one or more expansion stages and extracting an expansion gas at the top of the first expansion stage or, in the case of more than one expansion stages, at the top of at least one of the first to penultimate expansion stages and feeding, if desired, the partially regenerated absorption fluid obtained from the last expansion stage to a stripping zone for further regeneration, at least one acid gas stream containing the CO2 and possibly H2S being extracted from the regeneration and the regenerated absorption fluid being recycled into the absorption zone, wherein a part stream of fully or partially regenerated absorption fluid is fed to at least one of the expansion stages, from which the expansion gas is extracted, at a point above the feed of the absorption fluid which is to be expanded.
Patent NO-900420-L (NO)
Inventor: FARUK EROL ALI
IPC: C07D311/68
Filed: 1990-01-30
Abstract: A process for the preparation of a pure (3S,4R)-isomer of a compound of formula (A): <CHEM>  wherein one of R1 and R2 is hydrogen and the other is selected from the class of alkylcarbonyl, alkoxycarbonyl, alkylcarbonyloxy, alkylhydroxymethyl, nitro, cyano, chloro, trifluoromethyl, alkylsulphinyl, alkylsulphonyl, alkoxysulphinyl, alkoxysulphonyl, alkylcarbonylamino, alkoxycarbonylamino or aminosulphinyl, aminosulphonyl or aminocarbonyl, the amino moiety being optionally substituted by one or two alkyl groups, or alkylsulphinylamino, alkylsulphonyl-amino, alkoxysulphinylamino or alkoxysulphonylamino or ethylenyl terminally substituted by alkylcarbonyl, nitro or cyano, or -C(alkyl)NOH or -C(alkyl)NNH2, the alkyl groups or alkyl moieties of alkyl-containing groups having from 1 to 6 carbon atoms; one of R3 and R4 is hydrogen or alkyl having from 1 to 4 carbon atoms and the other is alkyl having from 1 to 4 carbon atoms, or R3 and R4 together are C2-5 polymethylene; R5 is hydrogen, alkyl having from 1 to 3 carbon atoms or acyl having from 1 to 8 carbon atoms; and  n is 1 or 2; in which the pyrrolidonyl or piperidonyl ring is formed by cyclising an appropriate precursor dihydrobenzopyranol compound that has already been resolved to the (3S,4R)-configuration, or a mixture in which the (3S,4R)-configuaration predominates with respect to the (3R,4S)-configuration.
Patent NO-902754-L (NO)
Inventor: BEELE JOHANNES ALFRED
IPC: F16L5/02
Filed: 1990-06-21
Abstract: A bushing (27) for the sealing passage of a cable, pipe and the like through a wall, comprising a frame (1) made of a rigid material which may be sealingly inserted in an aperture provided in the wall, as well as one or more parallelepipedal blocks (20) of a resilient material which may be composed from two identical halves, which blocks (20) in their composite state exhibit a bore adapted to the shape and dimensions of a cable to be passed through, which blocks (20) can be inserted in the frame aperture so as to be a fine fit, with the two halves of every block encasing a cable, whereby the blocks are dimensioned such that, under operating conditions of the bushing (27), the extend outwards on at least one side of the frame (1) in a direction transverse to the plane of the frame, which blocks (20) are provided with circumferential internal ribs (22) over at least a part of their length, and whereby blocks (20) whose outer faces rest against an inner wall of the frame under operating conditions of the bushing are provided with external ribs (23) over at least a part of the said outer faces.
Patent NO-903291-L (NO)
Inventor: KLEEMANN HEINZ-WERNER
IPC: C07D295/20
Filed: 1990-07-24
Abstract: The present invention relates to compounds of the formula I <IMAGE> in which A, R<2>, R<3>, R<4> and n are defined as indicated in the description, to processes for the preparation thereof, to the use thereof as medicines and to pharmaceutical compositions containing these.
Patent NO-904729-L (NO)
Inventor: BLACKBURN PETER
IPC: A01N63/50
Filed: 1990-10-31
Abstract: Broad range bacteriocin compositions are provided. The compositions can be dissolved or suspended in a suitable solvent or matrix and are more active towards a broader range of bacteria than are any of the component parts. The dissolved or suspended compositions constitute enhanced broad range bactericides. The compositions include lysostaphin and a lanthionine containing peptide bacteriocin; lysostaphin, a lanthionine containing peptide bacteriocin and a chelating agent; and lysostaphin, a lanthionine containing peptide, a chelating agent and a surfactant. Each component is present in the enhanced broad range bactericide in sufficient amount such that the bactericide is more effective against staphylococci than is lysostaphin alone and is more effective at treating and preventing a broad range of microbial infections. Methods of treating bacterial infections using said compositions and bactericides are provided.
Patent NO-911102-L (NO)
Inventor: SCHOLZ STEFAN
IPC: A61P5/00
Filed: 1991-03-19
Abstract: PCT No. PCT/EP89/01090 Sec. 371 Date Mar. 20, 1991 Sec. 102(e) Date Mar. 20, 1991 PCT Filed Sep. 20, 1989 PCT Pub. No. WO90/03385 PCT Pub. Date Apr. 5, 1990.New 11 beta -phenyl-14 beta H-steroids of general formula (I), where Z is an oxygen atom or the hydroxyimino-grouping N DIFFERENCE OH, and M and N are either jointly a second compound or L is a hydrogen atom and M is an  alpha -permanent hydroxy group and either A and B together are a second compound and D is a hydrogen atom, where R1 is a five or six-part heteroalkyl residue or a cycloalkyl, cycloalkenyl or aryl residue or A is a hydrogen atom and B and D together are a methylene bridge, where R1 besides the aforementioned residues may be a possibly substituted hydrocarbon residue with up to 10 C atoms, a possibly substituted amino group, a hydroxy or C1-8 alkoxy, mercapto or thioalkyl group, R2 is a methyl or ethyl residue, and R3/R4 represents the usual combination of substituents on the C17 atom in steroid chemistry, having antigestagenic and other properties.
Patent NO-920803-L (NO)
Inventor: HAUSER HERBERT PHILIPP
IPC: E05B9/04
Filed: 1992-02-28
Abstract: A lock cylinder (1), which can be assembled from several units, with a locking member (2) arranged in the central region and at least one locking mechanism (W) adjacent thereto, consists of a cylinder core (6) which comprises the key channel (7) and to which the tumblers (13) are allocated. A fit and turn connection is provided between a unit (3) allocated to the locking member (2) and the unit (4) containing the locking mechanism (W). <IMAGE>
Patent NO-923817-L (NO)
Inventor: BREIVIK KAARE
IPC: B63B22/02
Filed: 1992-09-30
Abstract: PCT No. PCT/NO92/00058 Sec. 371 Date Aug. 8, 1994 Sec. 102(e) Date Aug. 8, 1994 PCT Filed Mar. 30, 1992 PCT Pub. No. WO93/11035 PCT Pub. Date Jun. 10, 1993.A buoy for use in loading or unloading a flowable medium, especially oil from a vessel at sea. The buoy includes an outer member and a central member rotatably mounted in the outer member. The central member forms a passage for the flowable medium from the lower end of the buoy which is connected to a transfer line to a tube system within the vessel. The outer member is received and latched in an opening in the bottom of the vessel. The central member is connected to the tube system by a swivel means coupled to the upper end of the central member by a flexible joint which allows angular displacement about the axis of connection.
Patent NO-942260-L (NO)
IPC: A47J27/14
Filed: 1994-06-15
Abstract: A cooking apparatus (10) comprising a cooking chamber with a conveyor (52) wholly contained therein wherein food (46) is cooked by sprays (32) of hot cooking medium.
Patent NO-943163-L (NO)
Inventor: TOBEY STEPHEN W
IPC: A23L1/308
Filed: 1994-08-26
Abstract: The present invention is directed to a baked food composition comprising food ingredients and a water-soluble cellulose ether which is useful for reducing the low-density lipoprotein serum cholesterol level of an animal. Use of a specific particle-size distribution of the water-soluble cellulose ether results in compositions which are more palatable than known compositions.
Patent NO-944511-L (NO)
Title: Innretning og prosess til fremstilling av rilleblikk med planparallelle yterkantflater
Inventor: DOOSE INGOLF
IPC: B21D17/02
Filed: 1994-11-25
Abstract: Innretning til produksjon av rilleblikk med planparalelle ytterkantflater med hydraulisk eller mekanisk presse ( 1) med minst en hydraulisk- eller pneumatisk sylinder og på hver minst et øvre og et nedre pregeverktøy ( 3- 4) som på endestykkene ( 5) er utstyrt med pregeverktøyende-stykker ( 6- 7) hvor det er anbrakt integrerte hydraulisk-eller pneumatiske sylindre ( 8- 9) med konturstempler ( 10-11) som er relativbevegelig til bevegelsene av det øvre pregeverktøy ( 3). Fremgangsmåte til produksjon av rilleblikk med planparalelle yterkanttlater i . en hydraulisk eller mekanisk presse, kjennetegnet ved at åpne riller blir formet i blikk ( 15) ved at en rille blir presset i den tilsvarende ytterkantflaten ( 16) og at denne så blir tilbakeformet til blikkets ytterkantflate som før preging av rillen, mens blikket mellom pressens ( 1) øvre og nedre pregeverktøy ( 3- 4) er spent fast.
Patent NO-950242-L (NO)
Inventor: LEWIS MICHAEL E
IPC: A61K38/22
Filed: 1995-01-23
Abstract: Derivatives of K-252a are useful for treating Parkinson's disease.
Patent NO-950732-L (NO)
Inventor: HEMBERGER JURGEN
IPC: A61K39/00
Filed: 1995-02-27
Abstract: PCT No. PCT/EP94/02087 Sec. 371 Date Feb. 28, 1995 Sec. 102(e) Date Feb. 28, 1995 PCT Filed Jun. 28, 1994 PCT Pub. No. WO95/01375 PCT Pub. Date Jan. 12, 1995A protein isolated from crude extracts of Hirudo medicinalis is disclosed, which strongly inhibits the binding to collagen of platelets and their subsequent activation, which leads to platelet aggregation and thrombus formation. Additionally the protein prevents binding of von Willebrand factor to collagen. Described is a method for isolation and purification of the protein as well as its use for blocking collagen-stimulated platelet aggregation. The new protein (Brandinin) has a molweight of approximately 15 kD, binds to collagen but has no collagen-cleaving activity. The protein is useful in the prophylaxis, prevention and treatment of thrombotic diseaeses and for coating of blood-contacting materials, rendering them thromboresistant.