baber/WOPTO huggingface dataset:
Patent CZ-282770-B6 (CZ)
Inventor: CHUNG JOHN Y L
IPC: C07D211/22
Filed: 1993-02-24
Abstract: Řešení se týká vysoce účinného způsobu výroby sloučenin obecného vzorce I, v němž R.sup.1.n. znamená šestičlenný nasycený nebo nenasycený heterocyklický kruh s obsahem jednoho nebo dvou atomů dusíku jako heteroatomů, nebo skupinu NR.sup.6.n., v níž R.sup.6.n. znamená atom vodíku nebo alkylový zbytek o 1 až 10 atomech uhlíku, m je celé číslo 2 až 6 a R.sup.4.n. znamená aryl, alkyl o 1 až 10 atomech uhlíku nebo aralkyl o 4 až 10 atomech uhlíku. Syntéza se provádí v šesti stupních, používá se 4-pikolinu, dále se provádí O-alkylacetyrosinového derivátu za podmínek podle Misunoby s následným zmýdelněním nethylesteru, extraktivním odstraněním vedlejších produktů, překrystalováním se získá produkt s vysokým výtěžkem.ŕ
Patent CZ-300595-B6 (CZ)
Title: Armor made of multiple layers and process for producing thereof
Inventor: MOUREAUX BEATRICE
IPC: A41D13/00
Filed: 1998-07-14
Abstract: The present invention relates to an armor made of multiple layers (30) of flexible relatively inelastic penetration-resistant material shaped to fit over a shaped area to be protected, wherein the layers (30) are held by a plurality of darts (37) in successive layers (30) of the material, each of said layers of material having at least one dart (37) and each dart (37) in a layer (30) comprising a generally V-shaped section (35) whose edges are joined to form the dart (37), with the V-shaped section (35) folded on itself and folded over to one side to form an added thickness overlaying or underlying an adjacent part of the layer (30), the darts (37) in said multiple layers being angularly offset from one another with the folded V-shaped sections (35) oriented such that said added thickness is distributed substantially evenly around said shaped area. The invention also relates to a process for producing the above-described armor, said process comprising: providing multiple layers (30) of flexible relatively inelastic penetration-resistant material to be assembled into the shaped armor, each layer (30) having fold lines (36, 38) defining at least one dart (37) comprising a generally V-shaped section of the material, the darts (37) of the different layers (30) being angularly offset from one another around at least one point (39) of convergence; joining the edges of the V-shaped sections (35) to form the dart(s) (37) in each layer (30), the layers (30) with formed darts (37) all having substantially the same peripheral shape for assembly into the shaped armor; assembling the multiple layers (30) to form the shaped part, with darts (37) of different layers (30) angularly offset to one another and with the V-shaped sections (35) of material folded in directions to distribute the added thickness substantially evenly; and attaching the shaped multiple layers (30) to form the armor.
Patent SK-286581-B6 (SK)
Title: Dolastatin 15derivatives, pharmaceutical composition containing the same and their use
Inventor: JANSSEN BERND
IPC: A61K38/00
Filed: 1998-07-07
Abstract: Compounds of the present invention include cell growth inhibitors of formula (I), wherein A, B, D, E, F, G and K are alpha-amino acid residues, and s and r are each independently 0 or 1, L is a substituted or un-substituted amino or hydrazido group. The present invention further relates to the use of said compounds for the manufacture of a medicament for use in the treatment of cancer in a mammal, mainly a human.
Patent SK-278497-B6 (SK)
Title: The control system of the electric device
Inventor: MOREAU DOMINIQUE
IPC: G01R31/56
Filed: 1989-05-19
Abstract: The control system of the electric device contains the relay switches (3) with the electromagnet (9) excited with use of the coil (7) connected to two supplying clamps, the supplying circuit of which is passing through the exchangeable functional module (48), connected with the circuit of this coil with the use of the contact pins (51, 52) from electric point of view, and these pins also assure a mechanic hold of the module (48) on the realy switch (3) box. The pins (51, 52) getting out of the transversal wall (49) of the module, on each of the isolation shell (47) of the appropriate functional module (48) and this wall is able to attach to the transversal wall (53) of the contactor (3), equipped with supplying clamps, create the outputs of the appropriate functional module (47), the input clamps of which are connected to the resources or controlling automates of the system and they are placed at the front wall (58) of the contactor (3). Each of these modules contains electric, electromechanical or electronic control elements closed to the coil circuit.
Patent CZ-296278-B6 (CZ)
Title: Integrated fume cupboard with full-area lighting
Inventor: MORAVEK PETR
IPC: E04B9/02
Filed: 2004-08-06
Abstract: In the present invention, there is disclosed an integrated fume cupboard with full-area lighting being characterized in that an inlet of fresh filtered air is arranged in the enclosed space (12) extending between the panels (8) made of transparent materials and the ceiling (13), whereby in a peripheral cover (10), there are fitted adjustable strip slot diffusers (11). Preferably, said strip slot diffusers (11) are of circular shape and rotatable, and the panels (8) of transparent materials are preferably made as heat-insulating panels with air cavity embedded therein.
Patent CZ-298287-B6 (CZ)
Title: Detoxication method of sulfide yperite by treating thereof with haloalkane dehalogenases
Inventor: PROKOP ZBYNAOEK
IPC: A62D3/02
Filed: 2005-06-03
Abstract: In the present invention, there is disclosed a method of detoxification of yperite - bis(2-chloroethyl) sulfide - by the use of a haloalkane dehalogenases or their compositions, the method of preparation of dehalogenation enzymes and of decontamination compositions which contains at least one wild type and/or modified haloalkane dehalogenase (EC 3.8.1.5) as an chemically active component. The preferred dehalogenases are DhaA from Rhodococcus rodochrous NCIMB 13064, DmbA from Mycobacterium bovis 5033/66 or LinB from Sphingomonas paucimobilis UT26. Decontamination is utilizable for detoxification of yperite from the surfaces of technical equipment, buildings, human or animal skin and environment components by the treatment of yperite with the detoxification mixture according to the present invention with the concentration of the enzyme within the range of from 1x10e-6 to 1x10e0 mol.le-1 at a temperature ranging from +10 degC to +70 degC, preferably at about +40 degC and pH value within the range of 4 to 12.
Patent CZ-306889-B6 (CZ)
Title: A method of securing machines against vibrations and a device for implementing this method
Inventor: HABANEC JIŘÍ
IPC: G01M7/02
Filed: 2011-08-26
Abstract: The method of securing machines against vibrations, in which the vibrations of the selected machine parts are sensed, these vibrations are converted into an electrical signal which is subsequently digitized, lies in the fact that the digitization is carried out with a sampling frequency in the range of 100 kHz to 10 MHz, whereupon the digital sampled signal is filtered and evaluated, and the evaluated signal controls the machine disconnection at machine vibrations higher than critical vibrations. The device for implementing this method is provided with the vibration sensor (1), whose output is connected to the input of the amplifier (2), whose output is connected, via the analogue digital converter (4) and the filter circuit, to the input of the circuit (5) of the digital signal processing, whose control output is connected to the control input of the machine switch (6) for disconnecting the machine when the critical vibration value of the machine is exceeded.
Patent CZ-304327-B6 (CZ)
Title: Means for accelerated healing injured places and for bactericidal and viral protection
Inventor: Vošta Jan
IPC: A61K9/70
Filed: 2012-12-19
Abstract: The present invention relates to a means consisting of a micro- and/or nanofibrous fabric with quaternary nitrogen grafted by radiation thereon wherein the amount of the quaternary nitrogen is in the range of about 1 to about 30 percent by weight, based on the total weight of the micro- and/or nanofibrous fabric. The means further comprises colloidal silver and/or silver added sulfadiazine and/or silver bound to a thiol functional group of bifunctional anion exchange resin in an amount of about 0.5 to about 10 percent by weight of the silver based on the total weight of the micro- and/or nanofibrous fabric. The micro- and/or nanofibrous fabric is selected from the group consisting of alcohol-based substances, polyethylene, polypropylene, polyamides, polycaprolactam, polyacrylate, polyurethane and cellulose. The quaternary nitrogen is suitably bound to alkyl hydrocarbons having 1 to 5 carbon atoms and/or fatty hydrocarbons containing 12 to 20 carbon atoms and/or a benzyl radical. The efficiency of the micro- and/or nanofibrous fabric with grafted quaternary nitrogen and containing silver can be increased by providing thereof with a microlayer of primary and/or secondary and/or tertiary amines, polyamines, and polyaminoalcohols with molecular weight in the range of 100 to 6000. The means of the present invention can further comprise antibiotics and/or pharmaceutically active substances supporting healing of wounds. The means can be used for the treatment of injured places, but also as a mouth-screen for protection against bacterial or viral diseases.
Patent CZ-307894-B6 (CZ)
Title: Compressor
Inventor: SHIMOJI MIHOKO
IPC: F04C29/02
Filed: 2014-11-25
Abstract: The compressor (80) includes a sealed container (1) with a bottom portion with an oil storage unit (1a) for the lubricating oil; an electric motor (2) consisting of a stator (21) fastened in a sealed container (1), and a rotator (22) located inside the stator (21) and coupled to the drive shaft (23); and a compression mechanism unit (3) in a sealed container (1) connected to the coolant compression shaft (23). The compressor (80) also includes a round oil separation plate (100, 200, 300, 400) in a sealed container (1) between the electric motor (2) and the compression mechanism (3), where the oil separation plate (100) , 2000, 300, 400) comprises a first part (101a) inclined to the axial direction of the drive shaft (23), and a second part (101b) inclined to the axial direction of the drive shaft (23), the first vertical part (103a) with an upper end connected to the upper end of the first inclined part (101a) and a lower end attached to the lower end of the second inclined part (101b) and a second vertical part (103b) with an upper end attached to the upper end of the second inclined part (101b), and a lower end attached to the lower end of the first inclined part (101a).
Patent CZ-309459-B6 (CZ)
Title: First aid kit for bicycle handlebars
Inventor: BOUŠKA PETR
IPC: B62K21/26
Filed: 2019-11-28
Abstract: A first aid kit for a bicycle handlebar includes a compression storage portion (2), the compression storage portion (2) defines a space adapted to store items, and an elongated retractor member (3) attached to one end of the compression storage portion (2), the other end of which compresses the storage portion (2) is equipped with a plug (4). The plug (4) can be used to fix the compression storage part (2) in the handlebars and define the clearance between the first aid kit (1) and the handlebars. A pull-in element (3), such as a string or cable, can be used to pull the compression storage part (1) into the handlebar. The first aid kit (1) may also include a fixed storage portion for additional storage space.
Patent SK-285881-B6 (SK)
Title: Method for producing concrete or mortar with vegetal aggregate
Inventor: HOHN HERIBERT
IPC: C04B28/04
Filed: 2001-08-07
Abstract: A method for producing concrete or mortar based on exclusively vegetal aggregate, mineral binding and mixing water, the vegetal aggregate having a specific weight of 80 to 160 kgm-3, as measured at a residual moisture of approximately 15 %. 4 to 14 kg of non-hydratizable, finely ground mineralizator is added for each cubic meter of the vegetal aggregate, when the concrete or mortar is mixed, instead of pre-mineralization of the vegetal aggregate. Raw calcium carbonate is advantageous as mineralizator.
Patent SK-287259-B6 (SK)
Title: N-aryl(thio)anthranilic acid amide derivatives, pharmaceutical composition containing them, their preparation and their use as VEGF receptor tyrosine kinase inhibitors
Inventor: ALTMANN KARL-HEINZ
IPC: A61K31/444
Filed: 1999-11-08
Abstract: Described are compounds of formula (I), wherein W is O; X is NH; Y is CH2 or a N-oxide or a pharmaceutically acceptable salt thereof for the preparation of a pharmaceutical product for the treatment of a neoplastic disease which responds to an inhibition of the VEGF receptor tyrosine kinase activity. The compounds of formula (I) can be used for the treatment e.g. of a neoplastic disease, such as a tumor disease, of retinopathy and age-related macular degeneration.
Patent CZ-294637-B6 (CZ)
Title: Track renewing machine
Inventor: THEURER JOSEF
IPC: E01B29/06
Filed: 2001-06-08
Abstract: The present invention relates to a machine (1) for renewing a railroad track (2)  on a ballast bed, said machine comprising a machine frame (5) extending in a longitudinal direction, undercarriages (4) for supporting the machine frame (5) on the railroad track (2), a first tie transport device (19) for receiving old sleepers ((20) and a second tie transport device (21) for laying new ties (22), the tie transport devices (19, 21) being mounted on the machine frame (5) and being spaced from each other in the longitudinal direction, and a crawler vehicle (17) and ballast bed planing apparatus (23) being arranged on the machine frame (5) between the sleeper transport devices (19, 21), the ballast bed planing apparatus (23) being rotatable by 180 degree about a vertical axis.
Patent CZ-299540-B6 (CZ)
Title: Device for bridging height difference between a floor and extensible plate of access platform
Inventor: NOVOTNY VACLAV
IPC: A61G3/02
Filed: 2001-06-15
Abstract: The present invention is characterized by a threshold (5) being rotatably connected to a floor (12). Slewing motion of said threshold (5) toward an extensible plate (4) or away therefrom is controlled by a Geneva mechanism segment (6). Motion or position of the Geneva mechanism segment (6) depends on motion, or position of a slide (2) to which the extensible plate is rotatably joined.
Patent CZ-300623-B6 (CZ)
Title: Method for cleaning upstream surface of a particulate filter and apparatus for making the same
Inventor: ZILLIOX JEAN-PHILIPPE
IPC: B01D46/42
Filed: 2001-10-12
Abstract: The present invention relates to a method for cleaning the upstream surface (14) of a particulate filter (10) of a heat engine exhaust line, the filter (10) being arranged in a casing (12) having an outlet (20) for exhaust gases. The method comprises a step that consists in circulating a liquid flux through the particulate filter (10) from its downstream surface (18) towards its upstream surface (14) viewed from the direction of exhaust gas flow in the filter. The liquid flux circulated through the particulate filter (10) has a flow rate higher than 50 liters/minute and is distributed over the main part of the downstream surface (18) of the particulate filter. The invention also relates to an apparatus for making the above-described method, which apparatus comprises means (25) for generating circulation of a liquid flux at a flow rate higher than 50 liters/minute through the particulate filter, whereby said means for generating the liquid flux circulation is adapted for distribution of the liquid flux onto the downstream surface (18) of the particulate filter (10).
Patent SK-287596-B6 (SK)
Title: Insulating glazing and method for making same
Inventor: DEMARS YVES
IPC: C03C27/06
Filed: 2001-04-11
Abstract: An insulating glazing comprising at least two glass sheets (10, 11) separated by a gas gap (12), an interlayer (2) for spacing apart the two glass sheets and having an inner surface (20) opposite the gas gap and an opposite outer surface (21), and sealing means (3) with respect to the inside of the glazing. The invention is characterised in that the interlayer (2) is in the form of a substantially flat extruded section with encloses the periphery of the glazing by being pressed by its inner surface (20) against the edges (10a, 11) of the glass sheets, and maintained fixed by securing means (4).
Patent BR-PI0108882-B8 (BR)
Title: combinação farmacêutica
Inventor: DIANA GARCIA DEL BARCO HERRERA
IPC: A61K38/18
Filed: 2001-12-17
Abstract: "combinação farmacêutica, composição farmacêutica, e, uso da dita combinação". a presente invenção diz respeito à medicina humana e, em particular, a uma combinação farmacêutica do fator de crescimento epidérmico (egf) com um peptídeo mimético do fator de liberação do hormônio do crescimento (ghrp), que é útil na prevenção e/ou restauração da lesão tecidual causada pela irrigação sangüínea deficiente de um órgão determinado, devida a diferentes condições patológicas. a mencionada combinação pode ser usada dentro da mesma composição farmacêutica ou aplicada separadamente a um mesmo paciente como parte de um tratamento único que favoreça a vitalidade celular nos órgãos quando estes sejam submetidos a perda parcial ou total no suprimento de sangue oxigenado durante um período de tempo. esta combinação também atenua a formação de espécies tóxicas e metabólitos nos referidos órgãos, o que é particularmente útil aos tecidos submetidos a prolongados períodos de isquemia. a combinação farmacêutica pode ser aplicada, além disso, para fins profiláticos, a pacientes com condições que possam conduzir à disfunção ou lesão múltipla de órgãos de várias origens, como queimaduras, politraumatismos, síndrome da angústia respiratória, neonatos hipóxicos, choque hipovolêmico, enterocolite necrotizante, assim como a pacientes submetidos a grandes intervenções cirúrgicas.
Patent BR-PI0308207-B8 (BR)
Inventor: JUNICHI MITSUYAMA
IPC: C07C323/62
Filed: 2003-03-04
Abstract: Arylamide derivatives (I) are new. Arylamide derivatives of formula (I) and their salts are new. [Image] X : optionally substituted lower alkylene or alkenylene; G 1O, S or NH; G 2C or N; R aH, halo or optionally substituted alkyl, cycloalkyl or alkoxy; R 1optionally protected or substituted amidino; R 2NR 3R 4, NR 5YNR 6R 7 or a group of formula (i); R 3H, amino protecting group, a group of formula (ii) or optionally substituted cycloalkyl or alkenyl; W : a bond or optionally substituted alkylene; Y coptionally substituted 2-4C alkylene; Y c1optionally substituted 1-4C alkylene; R 7bH, amino protecting group, a group of formula (iii) or optionally substituted alkyl, cycloalkyl or alkenyl; Z : optionally substituted lower alkylene or alkenylene; G 3O, S, NH or bond; G 5C or N; R bH, halo or optionally substituted alkyl, cycloalkyl or alkoxy; R 8para or meta to G 3 and is optionally protected or substituted amidino; R 4-R 6H, amino protecting group or optionally substituted alkyl, cycloalkyl or alkenyl; Y : optionally substituted 2-6C alkyelene or 3-6C alkenylene; R 7R 4 or (iii); Y aoptionally substituted 2-4C alkylene; Y boptionally substituted 1-4C alkylene; G 4C or N; R 7aalkyl (optionally substituted by at least one CN, NO 2, halo, sulfo, phosphoryl, lower alkenyl, lower alkoxy, heterocyclyl, cycloalkyl, lower alkylidene, SH, amidinophenylaryloxy, aryloxy, lower alkylthio, lower alkylsulfinyl, lower alkylsulfonyl, lower alkylcarbamoyl, lower alkylsulfonylamino, lower alkylaminosulfonyl, lower carboxylalkenyl, lower alkoxyimino or optionally protected hydroxyl, amino, carbamoyl, hydrocarbamoyl, aminosulfonyl, cyclic amino or lower alkylamino), (iii) or optionally substituted phenyl, cycloalkyl or alkenyl, provided that when G 1 = NH, then X = optionally substituted 3-6C alkylene or alkenylene. [Image] ACTIVITY : Fungicide. In cytotoxicity assays, 4-[2-[1-(3-[4-[amino(imino)methyl]phenoxy]propyl)-4-piperidinyl]ethoxy]benzamidine hydrochloride (Ia) had an IC 50 value for Candida albicans TIMM1623 of 0.0039 mu g/ml. MECHANISM OF ACTION : None given.
Patent BR-PI0309142-B8 (BR)
Inventor: CASTAN CATHERINE
IPC: A61K47/38
Filed: 2003-04-07
Abstract: The invention relates to liquid pharmaceutical formulations for oral administration with the modified release of active principle(s), excluding amoxicillin, said formulations consisting of suspensions of coated particles of active principles (microcapsules). According to the invention, the microcapsules constituting the disperse phase of the suspension are designed to allow the modified release of the active principle(s) according to a profile that does not change during the storage of the liquid suspension. To do this the inventors propose the selection of a specific coating composition for the microcapsules which consists of at least four components that allow these microcapsules to be stored in water without modifying their properties of modified release of the active principle, this liquid phase furthermore being saturated with active principle(s).
Patent BR-9911769-B8 (BR)
Inventor: COLIN BROWN
IPC: A61L31/04
Filed: 1999-05-13
Abstract: A method of preventing or reducing the incidence of post-operative adhesions in or associated with a body cavity, which comprises introducing into the body cavity a composition containing an aqueous solution or suspension or gel formulation containing the polysaccharide dextrin.
Patent EP-1282748-B8 (EP)
Inventor: GJEMS OLE REIDAR
IPC: E04B2/02
Filed: 2001-04-09
Granted: 2012-02-29
Abstract: The invention relates to a cogging element (11, 21) for a cogging structure with contact surfaces (12, 22) for abutment against adjacent cogging elements (11, 21) in a common plane or against a base, and lateral surfaces (13, 23) for the formation of the sides of the cogging structure. At least one end (14, 24) of the cogging element (11, 21) has bevelled end surfaces (15, 25) which form angles (16, 26) with the lateral surfaces (13, 23) and are adapted to corresponding bevelled end surfaces (25') in ends of other cogging elements (11', 21') in an intersecting plane, and the cogging element's end (14, 24) is adapted to be fastened or provided with at least one fastening element (31) in the form of a screw for fastening to a corresponding end (24, 14) of another cogging element (21, 11) in extension of the cogging element (11, 21) in the same plane. The invention also relates to a cogging structure which is composed of the cogging elements.
Patent EP-1424987-B8 (EP)
Inventor: BERGQUIST PAUL ROLAND
IPC: C11D17/04
Filed: 2002-08-30
Granted: 2006-06-07
Abstract: An article for cleansing body surfaces is provided which includes an effervescent cleansing composition capable of generating a foam upon contact with water and a pouch for housing the composition. The pouch features first and second substrates, the latter constructed of a non-woven sheet selected from meltblown, spunbond and sheet combinations thereof. Advantageously, a high loft sheet may be bonded to the non-woven sheet. Escape of effervescent gas is controlled by the second substrate thereby maintaining a billowed pouch profile.
Patent EP-1467052-B8 (EP)
Inventor: OLSSON BO
IPC: E05F15/16
Filed: 2003-04-09
Granted: 2010-09-01
Abstract: This invention relates to a guide system in an overhead sliding door (2) which comprises, a set of guide rails (3) provided on each side of a door panel. The set of guide rails describe a path for guiding said overhead sliding door. The path comprises an upper substantially horizontal section (4), a curved section (5) and a substantially vertical section (6). At least one door panel (7) having a lower door panel portion (9) is provided, said door panel (7) being interconnected via supporting runners (11). The supporting runners (11) are guided along at least part of said guide rails (3), and a lower portion of the lower door panel portion (9) is hingedly interconnected to a guide element (1) having at least two pivotally interconnected supporting runners (13a, 13b) arranged for guiding said lower door panel portion along said path. <IMAGE>