baber/WOPTO huggingface dataset:
Patent CR-6436-A (CR)
Title: Inhibidores de la receptacion de monoaminas para el tratamiento de trastornos del snc
Inventor: MARK LEONARD ELLIOTT
IPC: C07D265/30
Filed: 2001-08-08
Abstract: Se refiere a compuestos que son útiles y presentan actividad como inhibidores de la recaptación de la serotonina, norepinefrina y dopamina, a sus sales farmacéuticamente aceptables, y a su uson en el tratamiento de trastornos del sistema nervioso central y otros trastornos.
Patent GB-562570-A (GB)
Title: Variable speed transmission gear
IPC: F16H33/08
Filed: 1943-01-01
Abstract: 562,570. Variable-speed gearing. DEMOCRATIS, A., KAMMER, G. S., and REILLY, C. O. C. Jan. 1, 1943, No. 48. [Class 80 (ii)] In an automatic infinitely variable torque converter a mass caused to revolve by the driving effort is rotatable about two alternative pivot axes so related to the driven'shaft that during half of each revolution in relation to the driven shaft the mass rotates about an axis spaced from the centre of the shaft and the centrifugal force of the mass tends to pull the pivot round the shaft in one direction and during the remainder of each revolution the mass rotates about an axis at or near the centre of the shaft so as to avoid producing a torque in the opposite direction. As shown an eccentric 2b is fixed to the driven shaft 1 and is surrounded by an eccentric 3b of equal eccentricity. A strap 4b round the eccentric 3b carries a mass 5b which is dragged round by a link 6 pivoted to a driving flywheel 21. A spider 8b freely mounted on the driven shaft 1 carries an eccentric 11b mounted on a pin 12b fixed to the eccentric 3b. The eccentric 11b is acted on by a spring 9 the other end of which is connected to the spider 8b. The position of the pin 12b in relation to the eccentrics 3b, 11b, is such that rotation of the eccentric 3b relatively to the shaft 1 in the driving direction is prevented when the centre of the eccentric 3b co-incides with the axis of the shaft 1. Preferably a plurality of units as above are arranged in balanced formation around the driven shaft as shown in Fig. 1.
Patent GB-211649-A (GB)
Title: Improvements in loose leaf binders
IPC: B42F13/04
Filed: 1923-01-01
Abstract: 211,649. Schade, J. Jan. 1, 1023. Clamping - devices; post files. - In a loose-leaf binder having clamping - bars connected by extensible tubular posts each comprising a fixed section 18, a telescoping section 19, and a flexible member 11 connected to the section 18 and guided through the section 19, the clamping-bars are separated or drawn together by pulling or pressing the flexible members. The latter are operated by a screw device wholly enclosed in one clamping-bar, so as to permit interchangeability. This device comprises a pair of grooved bars 8 forming a runway for the member 11, connecting-rods 13, and a pair of nuts 14 adjusted by a right and left-handed screw 15. The sections 19, which may be extended by auxiliary units, is secured to the bar 2 by screws 20, and the sections 18 are held in openings in the runway 10 by spring catches 21. The member 11, composed preferably of pivoted links, is supported rigidly by the sides of the runway 10, the posts 18, and guides 23. Clamping-bars.-The clamping-bars comprise two flanged members 1, 2 provided with ears to which similar ears on the covers are hinged by pintles.
Patent HK-2792-A (HK)
Title: Thiadiazole antiviral agents
Inventor: RIEDER BRENT JEFFREY
IPC: A61K31/415
Filed: 1992-01-02
Abstract: (1) 1,3,4-Thiadiazole-2-cyanamide and derivs. of formula (I) and their salts are new. In (I), R1 = H; R2 = CN; or R1+R2 = =C(SR6)NH2 or =C(NH2)2; R6 = 1-4C alkyl, cyano-(1-4C)alkyl or pyridyl-(1-4C)alkyl. (2) In vitro antiviral method for protecting mammalian cells in culture comprises adding to the culture a cpd. (I) in which either (A) R1 = H; R2 = CN or =CH-NHR3; or R1+R2 = =C(NH2)2 or =CR5-NHR3(1); R3 = COOR4; R3(1) = H or COOR4; R4 = 1-10C alkyl, 2-10C alkenyl or Ph, each opt. substd.; R5 = H or SR6; R6 = 1-4C alkyl, cyano-(1-4C)alkyl or pyridyl-(1-4C)alkyl; or (B) as defined for (A) except that R1+R2 = =CR5NHR31 only; and R3, R31 = H or COOR4.
Patent IS-4627-A (IS)
Inventor: BAILEY CAROLE ANN
IPC: C07D211/60
Filed: 1997-12-04
Abstract: Compositions which increase the bioavailability of proteinase inhibitors are disclosed. The compositions include a pharmaceutically acceptable carrier comprising monoglycerides of medium chain-fatty acids.
Patent IS-5355-A (IS)
Inventor: BRYANS JUSTIN STEPHEN
IPC: C07C229/32
Filed: 2000-01-21
Abstract: This invention is novel processes for the stereoselective preparation of gabapentin analogues.
Patent IS-6319-A (IS)
Inventor: NICKEL BERND
IPC: A61K31/4439
Filed: 2002-03-21
Abstract: The invention relates to the use of N-substituted indol-3- glyoxylamides of general formula 1 for treating tumors, in particular, in cases of drug resistance and metastatic carcinoma, and as angiogenesis inhibitors having distinctly fewer side effects, in particular, distinctly lower neurotoxicity. The invention also relates to medicaments containing the inventive compounds.
Patent IS-8025-A (IS)
Inventor: SPADONE THOMAS
IPC: B22D7/00
Filed: 2005-09-14
Abstract: Mold (1) for fabrication of an ingot by cooling and solidification of a mass of molten metal includes a wall (2) and an opening (3). The wall defines a bottom (4) and an inner surface (5) of which a part (S), the cooling surface, is able to evacuate all or part of the thermal energy released by the mass of metal during cooling and solidification. The wall incorporates at least one shaped element (6,7,8) to form at least one locking element, a stacking element or a handling element on the ingot. The cooling surface includes at least one element with a flat surface (Si) forming all or part of the bottom of the mould. At least one point (C) exists on a plane (Pi) tangent to each surface such that all the right segments (D) connect all points (R)of the cooling surface to the point (C) passing uniquely to the inside of the mold and the total area of the element(s) of the surface (Si) is at least equal to 10 % of the cooling surface. An independent claim is also included for the fabrication of a metal ingot using this mold.
Patent CR-10467-A (CR)
Title: Profarmacos de penem
Inventor: BRIGHTY KATHERINE ELIZABETH
IPC: A61K31/431
Filed: 2008-11-27
Abstract: Profarmacos de sulopenem con biodisponibilidad por via oral, por ejemplo, y sus solvatos e hidratos, su preparacion, su formulacion y su uso para tratar y prevenir la infeccion en mamiferos tales como seres humanos. Este resumen no limita la invencion.
Patent CR-10722-A (CR)
Title: Compuestos heterociclicos y su uso como inhibidores de la glucogeno sintetasa quinasa 3
Inventor: TURNER SEAN COLM
IPC: A61K31/4709
Filed: 2009-04-17
Abstract: Un compuesto heterociclico de formula general (I) y su uso y su preparacion, metodos para prepararlo, composiciones que contienen al menos uno de dichos compuestos, y metodos de tratamiento donde se usa al menos un compuesto. En particular, los compuestos de formula general (i) son utiles para inhibir la glucogeno sintetasa quinasa 3 (GSK-3).
Patent CR-11443-A (CR)
Title: Productos quimioterapeuticos cristalinos
Inventor: ROZEMA MICHAEL J
IPC: A61K31/423
Filed: 2010-05-19
Abstract: Forma cristalina 1 de N-[4-(3-amino-1H-indazol-4-il)fenil]-N'-(2-fluoro-5-metilfenil)urea, maneras para elaborarla, formulaciones que comprenden a la misma y elaboradas con la misma y metodos de tratamiento de pacientes que padecen una enfermedad para usarla.
Patent DK-78989-A (DK)
Inventor: RICHAUD FRANCOIS
IPC: C12N15/09
Filed: 1989-02-21
Abstract: The invention relates to a method for the integration of a chosen gene or a specified DNA sequence into a DNA sequence such as a bacterial chromosome or episome, wherein: a) the chosen gene or chosen DNA sequence is cloned inside a transposon, stripped of its arms, outside the essential portions of the transposon, b) the transposon is integrated into the DNA sequence, such as the chromosome or episome of the bacterium, as well as to the bacterial strains obtained by carrying out this method. <IMAGE>
Patent GB-316847-A (GB)
Title: Improvements in the manufacture and production of complex metal compounds of azo dyestuffs
IPC: C09B45/16
Filed: 1928-07-24
Abstract: 316,847. Johnson, J. Y., (I. G. Farbenindustrie Akt.-Ges.). July 24, 1928. Divided on and addition to 310,343. Samples furnished. Azo dyes, soluble metal compounds of. - Azo dyestuffs containing chromium or copper analogous to the dyestuffs containing chromium of the parent Specification are obtained by treating with compounds of chromium or copper o-oxyazo dyes produced by coupling diazotized o-amincphenols substituted by two or more negative groups with 1 : 3-phenylenediamine-4-sulphonic acid. In an example the dyestuff picramic acid # 1:3- phenylenediamine-4-sulphonic acid is heated under pressure for 3 hrs. at 120‹ C. with hydrated chromium oxide and formic acid; the product dyes leather violet-brown shades very fast to light, and dyes wool deeper brown shades fast to washing and milling. Reference has been directed by the Comptroller to Specifications 26460/12, 1611/15, 15127/15, and 15456/15.
Patent GB-1443391-A (GB)
Title: Method of forming waterproof and decorative membrane on wall  surface of building structure
IPC: B05D5/00
Filed: 1975-04-28
Abstract: 1443391 Coated wall surfaces S SAMURA 28 April 1975 00189/74 Heading B2E A waterproof decorative membrane with a textured pattern is formed on the structure of a wall surface by mixing a polyurethane, polysulphide or silicone elastic material with a curing agent to a viscosity of between 25000 and 200000 cps measured with a Brookfield rotational viscosimeter using a rotor No. 7 at 10 rpm and at 20‹C under thixotropy index range between 0.5 and 0.9 measured with a Brookfield rotational viscosimeter using a rotor No. 7 at 20‹C the thixotropy index being defined as being equal to and spraying the mixed material on to a vertical wall surface in a thickness of at least 0.5 mm with a spray gun to form a non-textured pattern. The pattern may be a crater, orange peel or glaciate pattern. The elastic material may comprise 100 parts of liquid polysulphide, 30-80 parts of filler, 10-20 parts of pigment, 5-25 parts plasticiser and 0-2 parts of thixotropic agent and 0-20 parts of solvent. The curing agent may be 7 to 9 parts of PbO curing agent, 0-10 parts of plasticiser, 0-10 parts of filler and 0-5 parts of retardant. The polyurethane elastic material may contain 100 parts of polyurethane prepolymer with 3.7 mol percent of NCO, and a curing agent may be 40-80 parts of diamine solution in polyol or 40-95 parts of polyol only, from 90-100 parts of filler, 10-20 parts of pigment, 0-20 parts of plasticiser, 0-2 parts of thixotropic agent and 0-50 parts of solvent. To obtain a surface having a socalled glaciate type the polyurethane contains 5 mol percent of NCO. Other suitable compositions are also specified.
Patent GB-1213852-A (GB)
Title: Variable geometry antennae
IPC: H01Q19/10
Filed: 1968-01-02
Abstract: 1,213,852. Aerials. THOMSON-CSF. 2 Jan., 1968 [9 Jan., 1967; 16 May, 1967], No. 333/68. Heading H4A. An aerial having a collapsible reflector comprises two circular supports 1, 2, Fig. 2, to which are fixed at their respective ends two crossed assemblies of wires 3, 3<SP>1</SP>. When the circular supports are spaced apart in their operative positions, the two assemblies of wires lie along the surface of an hyperboloid of revolution. Radiating elements A 1 , A 2  . . . An are mounted in a circle approximately coinciding with the locus of the focus of a parabola which is osculatory to the generating hyperbola at its apex. A group of adjacent elements is energized, with suitable phase and amplitude differences between them, and scanning is obtained by stepping around the circle. The aerial is applicable to a spin-stabilized communcations satellite, as it is stowable for launching and provides means for counter-rotating a radio beam, to maintain it pointing towards an earth station. The individual wires of the systems 3, 3<SP>1</SP> may be provided with tensioning springs at their ends, outside the supports 1, 2 (Fig. 7, not shown), and the said supports may carry, respectively, a central piston 16, Fig. 8, and a co-operating cylinder 15. The piston is moved from an inner retracted position to an outer expanded position by gas pressure or other means and is locked in the latter position by a spring-loaded plunger 18 which enters a recess in the cylinder. In a second embodiment (Fig. 4, not shown), two concentric hyperboloids of revolution are provided between two circular supports. The inner hyperboloid is formed by two crossed assemblies of wiers, whilst the outer hyperboloid is formed by one assembly of wires. In this way, linearly polarized waves from the radiating elements may be transformed on reflection into circularly polarized waves. Means are described for compensating for the effect of the varying spacing between the wires of the outer hyperboloid, from the equatorial plane to the circular supports, by suitable choice of the parameters of the hyperboloids. In another embodiment (Fig. 6a, not shown) a single truncated hyperboloidal reflector is used, and in others (Figs. 6b, 6c, not shown) two or more coaxial hyperboloid reflectors are used.
Patent GB-1391232-A (GB)
Title: Key ejecting lock
IPC: E05B63/00
Filed: 1973-01-03
Abstract: 1391232 Key ejecting lock ILLINOIS TOOL WORKS INC 3 Jan 1973 [4 Jan 1972] 413/73 Heading E2A A key ejecting lock comprises a body 12, a latch means rotatably mounted within the body in fixed axial relationship therewith and having a keyway, and a spring urged key ejecting means mounted in the latch means for ejecting the key should it be left in the lock. The latch means comprises a barrel 14 having a latch or bolt 16 snap fastened thereto by resilient legs 130. The barrel 14 carries at its forward end two plate tumblers 70 which are held in position by a cover 84 which clips onto the barrel 14. Only one plate tumbler may be provided. The key ejecting means comprises a portion 110 moving co-axially of the barrel through apertures 78 in the tumblers 70 and an offset portion 112 moving in a slot 104 in the barrel. The rear end of the body 12 is formed with resilient portions 36 which clip into a groove 100 in the barrel 14 to provide the aforesaid fixed axial relationship therebetween. The body 12 is also provided with a workpiece engaging flange 34 and a clip 46 co-operating with one of two grooves 44 in the body 12 is provided to hold the body in the workpiece. A bezel 48 may be provided for the cover 84. The lock is disclosed as being mounted on a freezer chest (Figs. 1 and 3, not shown) with the parts thereof being of a poor heat conducting lubricious plastics material.
Patent GB-939986-A (GB)
Title: Improvements in men's wearing apparel
IPC: A41B9/02
Filed: 1962-01-04
Abstract: 939,986. Undergarments. STEDMAN MANUFACTURING CO. Jan. 4, 1962 [Jan. 4, 1961], No. 417/62. Class 141. A man's brief is provided with a knitted cotton gusset portion 13 and a knitted fabric pouch bounded by an arcuate elastic tape 9 and supported by inelastic vertical tapes 10, 11, 12. The pouch portion may be formed from cloth covered rubber fibres in which case an inelastic strip is also provided between the pouch and gusset portion 13, to prevent the fibres unravelling.
Patent GB-231929-A (GB)
Title: Improvements in friction clutches
IPC: F16D13/71
Filed: 1924-01-07
Abstract: 231,929. Girling, A. H. G. Jan. 7, 1924. Clutches, friction.-A primary spring clutching-force of constant magnitude is augmented or opposed by a secondary force acting through levers, wedges, or the like and varying automatically with the torque, the ratio of force to torque being manually controlled by varying the angle of the lever, slope of the wedge, &c. A lever D is pivoted at about its centre on a lug F in a casing A secured to the driving-shaft and is engaged by one ball end of a link E, of which the other end engages a lug G on a clutch plate B turning with the casing A. Springs I act to clamp the clutch disc C on the driven shaft between the parts B, A. A spring J and a handoperated rod H control the inclination of the lever D, which in a position parallel ,to the plate B is ineffective, but when out of parallelism automatically either increases or decreases the pressure between the clutch plates with increase of load. At the limit of adjustment of the control rod H, the lever D may engage a lug K on the plate B to disengage the clutch. When the driven plate C overruns the casing A or the direction of drive is reversed, the lug K strikes a lug L on the casing and the springs I alone maintain the clutch contact. In the modification shown in Fig. 2, the thrust of the lever D is applied to a curved face on the lug G, with any point on which it may be brought into engagement. In the form shown in Fig. 3, the lever D is of bell-crank form and is pivoted to both parts A, B, the adjustable control-rod H acting as an abutment between the lug F and the lever D.
Patent GB-1137292-A (GB)
Title: Method of preparing isocyanic acid and stabilizing the same
IPC: C01C3/20
Filed: 1966-01-05
Abstract: 1,137,292. Isocyanic acid. STAUFFER CHEMICAL CO. 5 Jan., 1966 [18 Jan, 1965], No. 524/66. Heading C1A. Stabilized isocyanic acid is produced by contacting carbamoyl chloride with a Lewis base, the basicity of which is sufficient to abstract hydrogen chloride from the carbamoyl chloride, but not sufficient to cause trimerization of the so-formed isocyanic acid. The weak Lewis base may be an ether (e.g. diethylether), a polyether (e.g. a dialkoxyalkane such as 1,2-dimethyoxethane), a polymeric ether (e.g. a polyoxyethylene resin), a thioether (e.g. as a dialkylsulphide such as diemthyl-sulphide, diethylsulphide or di-n-propyl sulphide) and substituted amides (e.g. an N,N-dialkyl amide such as N,N-dimethylacetamide). The carbamoyl chloride may be generated just before use by reacting phosgene with ammonia in a heated reaction zone and collecting the carbamoyl chloride in a water cooled receiver.
Patent GB-238452-A (GB)
Title: Improvements in or relating to reinforced concrete linings for window and door openings in hollow or cavity walls of houses and other buildings
IPC: E06B1/24
Filed: 1925-01-08
Abstract: 238,452. Robertson, L. Jan. 8, 1925. Girders.-Lintels consist of slabs i which have tongued and grooved or dowelled connection with upright slabs g and are provided with ribs m for engaging the cavity c of the wall and fillets e on the opposite side for the reception of the door or window frame. Metal-reinforcing members j may project into the cavity c, a concrete filling k being provided.
Patent GB-429850-A (GB)
Title: Improvements in ornamental fabric
IPC: D03D15/00
Filed: 1934-01-08
Abstract: 429,850. Ornamental fabrics. FRANK ASSOCIATES, Inc., 35, West 39th Street, New York, U.S.A.-(Assignees of Frank, M. J. ; 595, West End Avenue, New York, U.S.A.) Jan 8, 1934, No. 694. Convention date, Feb. 1, 1933. [Class 142 (iv)] The base comprises weft threads 1 interwoven with warp threads 2 and also but more loosely with warp threads 3, ornamental ribbons R of lustrous cellulosic material preferably transparent being interwoven with the wefts and formed into projecting loops. The edges of the ribbons R just overlay the edges of the threads 3. Ribbons R of different colours may be used. The threads 1, 2, 3 may be natural or artificial silk or cotton. The fabric may be used for millinery and trimmings.
Patent GB-735727-A (GB)
Title: An improved fastener
IPC: F16B5/12
Filed: 1953-01-09
Abstract: 735,727. Stud and socket fasteners. FERNTOL PATENTS, Ltd., and FERNBERG, E. B. Jan. 8, 1954 [Jan. 9, 1953], No. 766/53. Class 44. A fastener comprises a single strip of spring material having the central portion of its length bowed to a head 18 of C-shape, each of its arms such as 13 on either side of the head being formed with a notch 16 or 17 in the edge, and with its free end such as 11 pointed. As shown each of the arms is notched on each side and the fastener is intended to fasten an ornamental beading 21 to a panel 19, the notches engaging the periphery of an aperture 22. The beading clips over the head 18 and a fabric trimming 20 which is pierced by the pointed ends of the fastener can be positioned between the beading and the panel.
Patent GB-676461-A (GB)
Title: Improvements connected with reciprocated liquid-spraying pumps
Inventor: LUDFORD LESLIE BRENTNALL
IPC: A01M7/00
Filed: 1950-01-12
Abstract: 676,461. Reciprocating pumps. FOUR OAKS SPRAYING MACHINE CO., Ltd. Feb. 19, 1951 [Jan. 12, 1950], No. 790/50. Class 102 (i) A reciprocating pump has a liquid agitator 9 pivoted on its outlet pipe 3, and oscillated by the piston 4 through a rod 12 and slotted arm 11. The piston is operated by a lever 5 pivoted on a link 6. A stand pipe 2 is provided.
Patent GB-764115-A (GB)
Title: Improvements relating to the washing and after-treatment of threads of regenerated celloulose
IPC: D01D10/04
Filed: 1955-01-11
Abstract: <PICT:0764115/IV(a)/1> <PICT:0764115/IV(a)/2> <PICT:0764115/IV(a)/3> <PICT:0764115/IV(a)/4> Washing and after - treatment of groups of parallel regenerated cellulose threads is effected by leading the groups of threads downwardly and upwardly over pairs of rollers arranged in an upper and a lower series pairs, the upper and lower series being in staggered relationship so that the descending threads follow a substantially vertical path and pass through troughs containing the washing or treating liquid, leaving the troughs through small apertures so as to entrain a thin sheath of the liquid. All the rollers or only the upper rollers of each pair may be driven. As shown in Figs. 1-3, the threads pass over pairs of rollers 1, 2 and on their downward run pass through troughs 3 containing the washing or treating liquid, leaving the bottom of the trough through a series of apertures 7.  The trough may be made in two parts, one part 9 being fixed and having the apertures 7 formed therein as a series of notches, the other part 10 being pivotally mounted so that it can be swung clear to facilitate threading up. The part 10 is clamped in its operative position, gasket 8 making the trough liquid-tight.  Comb-guides 6 may be used to keep threads separated on the upward run.  Lower rollers 2 may dip into a bath 5 of the washing or treating liquid.  In a modification, Fig. 4, the trough may be of the section shown, the threads running through a series of notches 4 and entraining liquid which is maintained in an overflowing condition in the trough.
Patent GB-1219802-A (GB)
Title: Improvements in and relating to sheet material
Inventor: SPILLER LESTER LASZLO
IPC: D21H17/28
Filed: 1968-01-05
Abstract: 1,219,802. Papermaking; electrostatic deposition. RANSBURG ELECTRO-COATING CORP. 5 Jan., 1968 [5 Jan., 1967], No. 889/68. Headings D1L, D2A and D2B. Fibrous cellulosic sheet material, e.g. paperboard or newsprint, as a wet web is sized by electrostatically charging atomized droplets of a slurry of ungelatinized granular starch, to deposit the particles on the wet web, dewatering and heating to assist gelatinization. The starch may be modified to reduce its gelatinization temperature, e.g. by surface hydroxyethylation. The liquid of the slurry is preferably water, but this may be replaced wholly or in part by glycols or polyglycols; glycerine and pentaerythritol can be added. The slurry may also contain surfactants, pigments, fillers, latices of styrene-butadiene copoloymers or emulsions of polyvinyl chloride. As shown, the slurry is circulated through conduits 22 to spray guns 23 above a web P of paper between the first and second wet presses of a paper machine. A valve in each spray gun is controlled through a control tube 24. The slurry is forced out of the guns by the pressure in the conduit, atomized and electrostatically charged by an electrode (33, Fig. 2 not shown). The web is effectively earthed and so the slurry is deposited at 25. Alternatively, it may be deposited on the wire side at 26, between the press and drier sections, between first and second drier sections or even before the couch, or both sides may be treated. The invention may also be used with cylinder or other machines. Very small amounts of starch can be applied uniformly by this technique.