baber/WOPTO huggingface dataset:
Patent CS-196338-B2 (CS)
Title: Herbicide and method of producing the active constituent
Inventor: DUTRA GERARD A
IPC: A01P13/00
Filed: 1976-12-28
Abstract: Alkyl-[di(benzyl) or di(aryl)]esters of N-phosphonomethyl glycine are produced by the reaction of a dibenzyl or diaryl phosphite with an N-methylene alkyl glycinate trimer. These esters and the hydrolysis products thereof containing at least one benzyloxy or aryloxy group bonded to phosphorus are novel compounds having the formula   <IMAGE> wherein R is a member of the group consisting of phenyl, benzyl, naphthyl, biphenylyl, benzyloxyphenyl and phenyl, benzyl or naphthyl groups substituted with from 1 to 3 groups selected from the class consisting of hydroxyl, lower alkyl, lower alkoxy, lower alkylthio, trifluoromethyl, carbo (lower alkoxy), nitro, or halo; R1 is hydrogen or an R group, and R2 is a lower alkyl group or hydrogen, and the strong acid salts of the compounds wherein neither R1 or R2 is H. These compounds are useful as post-emergent herbicides.
Patent CS-219297-B2 (CS)
Title: Means for destroying the weeds and method of making the active substance
Inventor: FRATER GEORG
IPC: C07C317/18
Filed: 1980-12-11
Abstract: The invention is concerned with herbicidally active propionic acid esters of the general formula   <IMAGE> wherein R<1> represents hydrogen, C1-6 alkyl or a phenyl group, R<2> represents C1-6 alkyl, C2-6 alkenyl, C2-6 alkynyl or a phenyl group or R1 and R2 together with the carbon atom to which they are attached form a C4-10 cycloalkane ring which, if desired, can be mono-, di- or tri-substituted with C1-3 alkyl, R<3> represents a halogen atom or a trifluoromethyl or nitro group and R<4> and R<5> each represent a hydrogen or halogen atom.
Patent AU-650316-B2 (AU)
Title: Intermediates for preparing 7-(1-pyrrolidinyl) -3-quinolone- and -naphthyridone- carboxylic acid derivatives
Inventor: PETERSEN UWE
IPC: A23K20/195
Filed: 1992-01-16
Granted: 1994-06-16
Abstract: 7-(1-Pyrrolidinyl)-1,4-dihydro-4-oxo-3-quinoline-carboxylic acid and 7-(1-pyrrolidinyl)-1,4-dihydro-4-oxo-1,8-naphthyridin-3-carboxylic derivs. of formula (I), their hydrates, acid addition salts, as well as their alkali metal, alkaline earth, silver and guanidinium salts are new; X<1> = halo; X<2> = H, NH2, 1-4C alkylamino, di(1-3C alkyl)amino, OH, 1-4C alkoxy, SH, 1-4C alkylthio, arylthio or halo; R<1> = 1-4C alkyl, 2-4C alkenyl, 3-6C cycloalkyl, 2-hydroxyethyl, 2-fluoroethyl, OMe, NH2, MeNH, EtNH or Me2N; or is Ph (opt. mono- or disubstd. by F); R<2> = H, 1-4C alkyl or (5-methyl-2-oxo-1,3-dioxol-4-yl)methyl; R<3> = a gp. of formula (a): R<4> = 1-4C alkyl, aryl or 1-4C acyl; R<5> = H, 1-4C alkyl, OH or OMe; R<6> = H, 1-4C alkyl (opt. substd. by OH), aryl, heteroaryl, benzyl, 1-4C alkoxycarbonyl, 1-4C acyl, (5-methyl-2-oxo-1,3-dioxol-4-yl)methyl or 3-6C cycloalkyl; R<7> = H or 1-4C alkyl; R',R'' = H, Me or Ph; R''' = H or Me; Y = O, CH2, CH2CH2 or CH2O (where the bond to N may be via C as well as O); (Note: Y is not otherwise defined in claim 1). Z = O or S; A = N or CR<8>; R<8> = H, halo, Me, CN, NO2 or OH, or R<8>+R<1> = a bridge of type (b)-(d): Cpds. of formula (e) are excluded; R1 = 1-4C alkyl; R2,R3 = H or 1-4C alkyl; R4 = cyclopropyl, Ph, halophenyl, thienyl, opt. substd. by 1-4C alkyl or halo; R5 = halo. Also claimed is the S,S-configuration of a cpd. of formula (f) and its salts:A = CCl, CF or COMe.
Patent AU-551844-B2 (AU)
Title: Aspectic filling of a container
Inventor: SCHOLLE WILLIAM J
IPC: B65B55/10
Filed: 1983-01-26
Granted: 1986-05-15
Abstract: A device for filling containers (11) through a spout (13) on the container includes a sterile chamber (21) that has an opening (27) in a wall (23) through which the spout (13) of the container may be inserted into the chamber. A filling head (71) inside the chamber (21) can connect with the spout (13) and fill the container through the spout. A cup-shaped cap (51) inside the chamber (21) can be brought to cover the opening (27) in the wall (23) to substantially prevent the escape of a sterile gas from the chamber (21) when the spout is not in the opening. A fluid spray head (52) inside the cup-shaped cap (51) sprays fluid for sterilizing the spout before it is exposed to the sterile chamber. A pair of jaws (31) fit around the spout (13) when the spout is in the opening (27) to substantially prevent the escape of the sterile gas during the filling operation when the container cap (15) is removed.
Patent AU-768915-B2 (AU)
Title: Novel apparatus and process for preparing crystalline particles
Inventor: FERRIE ALAN RONALD
IPC: A61K31/135
Filed: 2000-11-03
Granted: 2004-01-08
Abstract: An apparatus for preparing crystalline particles of a substance suitable for inhalation therapy comprises  (i) a first reservoir 3 of said substance dissolved in a liquid solvent; (ii) a second reservoir 3 of liquid antisolvent for said substance which is miscible with the liquid solvent; (iii) a cylindrical mixing chamber 2 having first and second tangential inlet ports and an axial outlet port; (iv) means for delivering the contents of the first and second reservoirs to the mixing chamber in a stream via the first and second inlet ports respectively at independent controlled flow rate, the streams of liquid from t he i nlet a nd o utlet ports being intimately mixed in the cylindrical mixing chamber through formation of a vortex thereby causing precipitation of crystalline particles of the substance; and (vi) means 5 for collecting crystalline particles suspended in the stream of liquid discharged from the outlet port of the mixing chamber.
Patent AU-687970-B2 (AU)
Title: Process for the preparation of blocked polyisocyanates, and their use in polyurethane coating systems
Inventor: GRAS RAINER
IPC: C08G18/80
Filed: 1995-02-27
Granted: 1998-03-05
Abstract: The prodn. of totally or partly blocked polyisocyanates (I) based on a blocking agent (II) and a polyisocyanate with at least 2 free NCO gps. (III), opt. in the presence of a chain extender, is carried out as a continuous process in the absence of solvent.
Patent AU-751453-B2 (AU)
Title: Benzenesulfonamide inhibitors of PDE-IV and their therapeutic use
Inventor: CONNOR DAVID THOMAS
IPC: A61P25/28
Filed: 1998-11-04
Granted: 2002-08-15
Abstract: PCT No. PCT/US98/23482 Sec. 371 Date Feb. 7, 2000 Sec. 102(e) Date Feb. 7, 2000 PCT Filed Nov. 4, 1998 PCT Pub. No. WO99/26616 PCT Pub. Date Jun. 3, 1999The present invention provides compounds and pharmaceutical compositions thereof, and methods of using same in the treatment of diseases whose treatment benefits from the inhibition of phosphodiesterase (PDE-IV) or Tumor Necrosis Factor (TNF) including asthma, allergic diseases, rheumatoid arthritis, osteoarthritis, septic shock. The compounds provided by this invention have formula (I) wherein R1, R2, R3, R4 are as defined herein.
Patent AU-648885-B2 (AU)
Title: ATP analogues
Inventor: INGALL ANTHONY HOWARD
IPC: A61K31/708
Filed: 1992-04-02
Granted: 1994-05-05
Abstract: There are disclosed compounds of formula I, <CHEM>     wherein Q represents CR<1>R<2>,     R represents O or CR<3>R<4>,     W represents O or CH2, R<1>, R<2>, R<3> and R<4> independently represent hydrogen or halogen, X represents S(O)nR<5>, alkyl C1-6, alkoxy C1-6, acylamino C1-6, CONR<6>R<7>, NR<8>R<9>, halogen, a 5- or 6-membered S containing heterocycle, or phenyl optionally substituted by alkyl C1-6,     n represents 0, 1 or 2, R<5> represents aryl or alkyl C1-6 optionally substituted by one or more substituents selected from hydroxy, alkoxy C1-6, halogen and aryl; R<6>, R2<7>, R<8> and R<9> independently represent hydrogen or alkyl C1-6,     Y represents NH2 or alkoxy C1-6, and     Z represents an acidic moiety, in addition, when R represents CR<3>R<4>, then -Q-Z may also represent hydroxy or -OP(O)(OH)2, and pharmaceutically acceptable salts thereof, with certain provisos, for use as pharmaceuticals.
Patent AU-662135-B2 (AU)
Title: Imidazole-derivatives having agonistic or antagonistic activity on the histamine H3-receptor
Inventor: TIMMERMAN HENDRIK
IPC: C07D233/90
Filed: 1992-02-27
Granted: 1995-08-24
Abstract: The invention relates to imidazole-derivatives of general formula (a). The invention in particular relates to derivatives having agonistic or antagonistic activity on the histamine H3-receptor. The novel imidazole-derivatives are isothio urea-, guanidine- and amidine-derivatives. The invention further relates to pharmaceutical compositions comprising the novel imidazole-derivatives as well as to methods for preparing the derivatives and for preparing pharmaceutical compositions having antagonistic and agonistic activity on the histamine H3-receptor.
Patent AU-569034-B2 (AU)
Title: Zirconia ceramic materials and method of making same
Inventor: HUGHAN ROBERT RANDOLPH
IPC: C04B35/48
Filed: 1983-05-27
Granted: 1988-01-21
Abstract: A partially magnesia stabilised zirconia ceramic material is claimed having a cubic zirconia phase content of 25-70 vol.% and a MgO content of 3.0-3.65 wt.% of the ceramic. The material contains an additive metal oxide which forms an insol. zirconate that does not combine with MgO, in an amt. of 0.05-1.00 wt.%. The microstructure consists of grains of cubic ZrO2, each grain contg. pptes. of tetragonal ZrO2 transformable on application of tensile stress or heat treatment into monoclinic ZrO2. The pptes. are lenticular in shape and have an ave. length of about 150 nm in their longest dimension. Each grain contains grain matrix monoclinic ZrO2 as transformed tetragonal ZrO2 in a first specified range of monoclinic ZrO2 content. A ground surface and a polished surface of the material each contains monoclinic ZrO2 in second and third specified ranges of content, the specified ranges of content being different for ceramics to be used in different ranges. Also claimed is a method of mfg. the ZrO2. ZrO2 based materials can be provided for different temp. range uses, with appropriate combinations of the properties, thermal shock resistance, strength and wear resistance, without trying to obtain the optimum of each of these properties for use at all temps.
Patent AU-703242-B2 (AU)
Title: Film coated tablet of paracetamol and domperidone
Inventor: PRUDHOE GORDON
IPC: A61P29/00
Filed: 1995-02-27
Granted: 1999-03-25
Abstract: PCT No. PCT/EP95/00719 Sec. 371 Date Jun. 4, 1996 Sec. 102(e) Date Jun. 4, 1996 PCT Filed Feb. 27, 1995 PCT Pub. No. WO95/22974 PCT Pub. Date Aug. 31, 1995The present invention is concerned with a film coated tablet comprising as active ingredients the analgesic agent paracetamol and the antiemetic agent domperidone, and with a process of preparing such tablets.
Patent AU-760334-B2 (AU)
Title: Apparatus and method for mixing drill cuttings in a tank and transferring them therefrom
Inventor: JAGER VERNON DE
IPC: F04D7/04
Filed: 1999-12-20
Granted: 2003-05-15
Abstract: An apparatus and method for slurrying waste materials and drill cuttings. The apparatus includes a pump having a chamber an inlet opening into the bottom of the chamber, an impeller, an outlet on one side of the chamber for removal of material into a discharge line, and circumferentially spaced circulation ports in the chamber side. The impeller extends below the chamber and breaks up debris in addition to drawing material into the pump chamber. The pump may be rotated by a swivel connection and moved and manipulated in the tank by a crane arm, or it may be suspended by cable or other means. The pump stirs up a slurry by rotating the impeller, opening the circulation ports at least partially so that the material entering the bottom inlet to the chamber and being agitated by the impeller is forced out of the circulation ports. The pump can operate in the stirring mode until the material to be removed is generally homogenious, whereupon the circulation ports can be closed allowing the impeller to direct the slurry through the side outlet of the chamber into the discharge line. The stirring or slurrying mode can be combined with a discharge mode by opening the circulation ports as required to slurrify the material while it is pumped out the discharge line. An auxiliary discharge conduit may also be connected with the outlet to discharge material back into the tank to exchange upper fluid layers with lower layers.
Patent AU-617677-B2 (AU)
Title: Polyethylene glycol carbamates
Inventor: PETER HEINRICH
IPC: C07C311/00
Filed: 1988-07-22
Granted: 1991-12-05
Abstract: Compounds of the formula    <IMAGE>  (I)    <IMAGE>   in which R is alkyl having up to 4 carbon atoms, n has an average value of at least 9, X is a radical of the formula -C(=O)-(NH-SO2)m- in which m is 0 or 1 and, if m is 1, the carbonyl group may be bonded to the oxygen atom or to the nitrogen atom, and each of the radicals A1, A2 and A3, independently of the others, is hydrogen or an acyl radical, and salts of salt-forming compounds of formula I, as well as metal complexes of compounds of formula I, in which A1, A2 and A3 are hydrogen can be used as metal chelators and as auxiliaries in diagnosis.
Patent AU-563457-B2 (AU)
Title: Hand held electric power tool
Inventor: LAERE CHRISTIAAN G M VAN
IPC: B25B21/00
Filed: 1983-09-29
Granted: 1987-07-09
Abstract: An electric rotary power tool apparatus is adapted for loosening jammed or seized automobile wheel nuts or bolts and holdable by hand during operation. It comprises (1) an electric motor laid out to be driven by an electric direct current having an operational voltage of at least 8 to 30 volts and at least 20 up to 60 amperes, and comprising a stator, a rotor, first and second pole means, and a driving shaft bearing said rotor and having a rotary axis, the speed of said motor, at a nominal voltage of 12 to 24 volts ranging from 8000 to 30000 r.p.m under load;  (2) a casing in which the motor is housed;  (3) an on-off and reversing switch; (4) tool socket means being adapted for receiving a socket tool therein and comprising a driven shaft, the speed under load of which driven shaft is in the range of from 1200 to 4000 r.p.m.; (5) a speed-reducing unit comprising a gear transmission positively and drivingly connecting the said driving shaft with the driven shaft and adapted for directly and uninterruptedly transmitting torque from the driving motor shaft to the driven shaft and reducing the speed of the former to the latter shaft in a ratio of from about 7:1 to about 12:1. (6) impact-producing means comprising an impact mass separate from said motor and being associated with the tool socket means, mentioning under (4), supra, for imparting impacts to the latter means. The apparatus can also be used as a hobby tool by eliminating the impact-generating unit.
Patent AU-713768-B2 (AU)
Title: Pressure die-casting or injection machine
Inventor: COLLOT JEAN
IPC: B30B15/30
Filed: 1997-05-08
Granted: 1999-12-09
Abstract: A device for feeding a billet (2) of material into the injection chamber of an injection machine, press tool or the die of a forge press consists of a support (1) positioned in at least one heating system (14,14') and that the means to assure transfer of the billet consists of a means (3) to the move the support horizontally to take the billet from the heating position to a point vertically above the injection chamber (16). A means (4) rotates the support about its axis to cause the slug to fall under gravity into the injection chamber or press die.
Patent AU-683739-B2 (AU)
Title: Thiazolidines and oxazolidines substituted by a pyridine ring and their use as hypoglycemic agents
Inventor: OHARA YOSHIO
IPC: C07D413/14
Filed: 1995-03-27
Granted: 1997-11-20
Abstract: The present invention provides novel pyridine type thiazolidines and their salts, expressed by formula (I) (wherein X<1> is S or O; X<2> is S, O or NH; Y is CR<6>R<7>, R<6> is a hydrogen atom, a C1-C7 alkyl group or a C3-C7 cycloalkyl group, and R<7> is a hydrogen atom, a C1-C7 alkyl group or a C3-C7 cycloalkyl group or forms a bond together with R<4>), or SO2; Z is a C1-C10 alkyl group, a C2-C10 alkenyl group, a C2-C10 alkynyl group, a C3-C7 cycloalkyl group, a C3-C7 cycloalkenyl group (each of said alkyl, alkenyl, alkynyl, cycloalkyl and cycloalkenyl groups may be substituted with at most 3 of hydroxyl, oxo, C1-C7 alkyl and C1-C7 alkoxy groups), a phenyl group, a biphenyl group, an  alpha -naphthyl group, a  beta -napthyl group, a benzyl group or a heterocyclic group. The compounds have a hypoglycemic effect.
Patent AU-659859-B2 (AU)
Title: Piston dispensing apparatus
Inventor: MARTIN JAMES H
IPC: B65D83/44
Filed: 1992-06-04
Granted: 1995-06-01
Abstract: In a fluid dispenser a spring biased piston is mounted for reciprocable movement along a stem member which is moved longitudinally to actuate the dispenser. A metering chamber is located between the end of the piston and the end wall of a cylindrical chamber in which the piston is mounted, and axial passageways extending from opposite ends of the stem connect the metering chamber to a discharge location when the stem is in a discharge positon and connect the metering chamber to a fluid reservoir when the stem is in a fill position.
Patent AU-605915-B2 (AU)
Title: Process for single-step coal liquefaction
Inventor: DELBIANCO ALBERTO
IPC: C10G1/00
Filed: 1988-09-30
Granted: 1991-01-24
Abstract: A process for the single-step coal liquefaction is disclosed, which comprises reacting the same coal in an aqueous suspension with carbon monoxide in the presence of a CO-conversion catalyst selected from an alkaline hydroxide or carbonate, characterized in that the reaction is caused to take place at a temperature firstly maintained for a time of up to 20 minutes equal to a value selected within the range of from 300 to 370 DEG C, then is increased over a time comprised within the range of from 20 to 40 minutes, until a temperature value is reached, which is comprised within the range of from 420 to 450 DEG C, at which value it is kept constant for a time of up to 20 minutes.
Patent AU-763032-B2 (AU)
Title: Methods and compositions for treating disorders involving excitotoxicity
Inventor: GALDES ALPHONSE
IPC: C12N5/0793
Filed: 1999-12-03
Granted: 2003-07-10
Abstract: It is shown here that hedgehog polypeptides possess novel activities beyond phenotype specification. Using cultures derived from the embryonic day 14.5 (E14.5) rat ventral mesencephalon, we show that hedgehog is also trophic for dopaminergic neurons and other neurons which are sensitive to exotoxicity.
Patent AU-568339-B2 (AU)
Title: Wire stuffing cover
Inventor: HUGHES RICHARD LAMARR
IPC: H01R4/24
Filed: 1984-03-12
Granted: 1987-12-24
Abstract: A one-piece wire stuffing cover having a series of tubular terminal receiving sockets with wire gripping slots at front and rear faces and respective wire stuffers between the slots, lead-out openings for wires terminated by the cover being provided in the sockets rearward of the wire stuffers. The lead-out openings are provided by rebated portions in the sockets which define wire engaging shoulders extending across a rear axial end of the terminal for strain relief. The slots in the rear face diverge progressively to release the wire at the rear face during termination.
Patent AU-755404-B2 (AU)
Title: Hydrofluorination of chlorinated hydrocarbons
Inventor: WILMET VINCENT
IPC: C07C21/18
Filed: 1999-02-25
Granted: 2002-12-12
Abstract: Improved process for the catalytic hydro-fluorination of saturated or unsaturated organic compounds corresponding to the general formula CwHxClyFz (I) in which w is an integer between 1 and 6, x is an integer between 0 and (2w+1) or between 0 and (2w-1), y is an integer between 1 and (2w+1) or between 1 and (2w-1), z is an integer between 0 and (2w+1) or between 0 and (2w-1) and the sum (x+y+z) is equal to (2w+2), comprising a continuous feed of hydrogen chloride.Process for preparing 1,1,1,3,3-pentafluoropropane starting with 1,1,1,3,3-pentachloropropane, comprising two catalytic reaction steps, in which hydrogen chloride is preferably fed continuously into the reaction medium of at least one of the two reaction steps.
Patent AU-763776-B2 (AU)
Title: Portable data support with a detachable mini chip card
Inventor: HAGHIRI YAHYA
IPC: G06K19/077
Filed: 2000-02-16
Granted: 2003-07-31
Abstract: The invention relates to a portable data carrier ( 1 ) with a break-out mini smart card ( 2 ) embedded therein. The mini smart card ( 2 ) is separated from the remaining card body by a free punch ( 3 ) extending over substantial parts of the mini smart card. According to the invention, the mini smart card ( 2 ) contains another rated breaking line ( 5 ) having a different break-out direction from that of the mini smart card.
Patent AU-622155-B2 (AU)
Title: Atomized instant cooling process
Inventor: TAN DOMINGO K L
IPC: B60H1/32
Filed: 1989-03-20
Granted: 1992-04-02
Abstract: Method of instantly lowering the temperature of the passenger compartment a of vehicle using atomized bursts of alcohol-water solution.
Patent AU-690324-B2 (AU)
Title: Process for loading a protected storage zone of an information processing device, and associated device
Inventor: UGON MICHEL
IPC: G07F7/10
Filed: 1995-10-11
Granted: 1998-04-23
Abstract: The method involves writing confidential data in a protected zone (11) which belongs to a module (8) of a data processor system (1). The protected zone of memory is accessible for reading/writing by the internal processor (9) of the module, but inaccessible to at least a write action from an exterior module. The data transfer is made using an analogous protected memory zone (27) of a portable device (21) having a similar structure to that of the module. The portable device is placed in a reader (6) of the data processor. The data (K) and/or the programs (P1) are transferred from the portable device protected zone to the module protected zone.
Patent AU-729929-B2 (AU)
Title: A synthetic plant core promoter and upstream regulatory element
Inventor: BRUCE WESLEY B
IPC: C12N15/29
Filed: 1997-06-10
Granted: 2001-02-15
Abstract: Synthetic elements for enhancing expression of genes in plant cells are disclosed. These include a promoter with a "TATA to start" sequence containing 64 % or greater GC content and an upstream element incorporating several OCS binding motifs and novel flanking sequences.
Patent AU-652509-B2 (AU)
Title: Speed governor for rotational drive
Inventor: REYNOSO FRANK
IPC: F16D59/00
Filed: 1993-01-13
Granted: 1994-08-25
Abstract: A speed governor is enclosed within a generally cylindrical housing which defines an interior cylindrical surface. A rotor is rotatably supported within the enclosure of the housing and is coupled to a power coupling belt by a pulley formed in the rotor shaft. A pair of weighted arms are pivotally secured to the rotor forming a pair of centrifugal counterweights. A coil spring is commonly coupled between the counterweights to provide a drawing force urging the counterweights to a collapsed inward position. Each counterweight supports a friction pad on its outer surface facing the cylindrical surface of the governor housing.
Patent AU-757090-B2 (AU)
Title: Polarized gas accumulators and heating jackets and associated gas collection and thaw methods and polarized gas products
Inventor: DRIEHUYS BASTIAAN
IPC: F17C13/00
Filed: 1998-12-11
Granted: 2003-01-30
Abstract: Methods of collecting, thawing, and extending the useful polarized life of frozen polarized gases include heating a portion of the flow path and/or directly liquefying the frozen gas during thawing. A polarized noble gas product with an extended polarized life product is also included. Associated apparatus such as an accumulator and heating jacket for collecting, storing, and transporting polarized noble gases include a secondary flow channel which provides heat to a portion of the collection path during accumulation and during thawing.