baber/WOPTO huggingface dataset:
Patent AU-6839100-A (AU)
Title: Bis-sulfonamides
Inventor: BOLLI MARTIN
IPC: C07D239/69
Filed: 2000-08-16
Abstract: Sulfonamide compounds (I) and their salts, diastereomers, racemates and meso-forms, are new. Sulfonamide compounds of formula (I) and their salts, diastereomers, racemates and meso-forms, are new. [Image] R 1aryl, aryl-lower alkyl, aryl-lower alkenyl, heteroaryl or heteroaryl-lower alkyl; R 2lower alkyl, CF 3, lower alkoxy-lower alkyl, lower alkenyl, lower alkynyl, aryl, aryl-lower alkyl, aryl-lower alkenyl, heterocyclyl, heterocyclyl-lower alkyl, heteroaryl, heteroaryl-lower alkyl, cycloalkyl or cycloalkyl-lower alkyl; R 3phenyl (optionally substituted by 1-3 lower alkyl, lower alkenyl, lower alkynyl, lower alkoxy, amino, lower alkylamino, amino-lower alkyl, CF 3, OCF 3, halo, lower alkylthio, OH, hydroxy-lower alkyl, CN, carboxyl, lower alkanoyl or formyl), benzofuranyl, aryl or heteroaryl; R 4H, halo, CF 3, lower alkyl, lower alkylamino, lower alkoxy, lower alkylsulfono, lower alkylsulfinyl, lower alkylthio, lower alkylthio-lower alkyl, hydroxy-lower alkyl, lower alkyl-oxy-lower alkyl, hydroxy-lower alkyl-oxy-lower alkyl, hydroxy-lower alkylamino, lower-alkylamino-lower alkyl, amino, di(lower alkyl)amino, [N-(hydroxy-lower alkyl)-N-(lower alkyl) amino], aryl, arylamino, aryl-lower alkylamino, arylthio, aryl-lower alkylthio, aryloxy, aryl-lower alkyloxy, aryl-lower alkyl, arylsulfinyl, heteroaryl, heteroaryloxy, heteroaryl-lower alkyloxy, heteroaryl-amino, heteroaryl-lower alkylamino, heteroarylthio, heteroaryl-lower alkylthio, heteroaryl-lower alkyl, heteroaryl-sulfinyl, heterocyclyl, heterocyclyloxy, heterocyclyl-lower alkyloxy, heterocyclyl-amino, heterocyclyl-lower alkylamino, heterocyclylthio, heterocyclyl-lower alkylthio, heterocyclyl-lower alkyl or heterocyclyl-sulfinyl; R 6H, lower alkyl, cycloalkyl, heterocyclyl, heteroaryl, aryl, cycloalkyl-lower alkyl, heterocyclyl-lower alkyl, heteroaryl-lower alkyl, aryl-lower alkyl, lower alkoxy-lower alkyl, lower alkylthio-lower alkyl, lower alkylamino-lower alkyl, lower alkenyl or lower alkynyl; n : 2-5; and X : O, S, NH, CH 2 or bond. An independent claim is also included for the preparation of (I). ACTIVITY : Antimigraine; hypotensive; cardiant; vasotropic; antianginal; cytostatic; antiasthmatic; antiinflammatory; nephrotropic; cerebroprotective; nootropic; hemostatic; antiarteriosclerotic; antiulcer; auditory; opthalmological; antibacterial; antisickling; antidiabetic; immunosuppressant. MECHANISM OF ACTION : Endothelin ET A and ET B antagonist. Competitive binding assays were carried out on CHO cells expressing human recombinant ET A or ET B receptors. p-t-butyl-N-[6-(3-(2-thiophenesulfonamido)propoxy)-5-(o-methoxyphenoxy)-2-(2-cyclopropyl)-4-pyrimidinyl]benzenesulfonamide (Id) gave IC 50's of 14.8 and 1.86 nM respectively for ET A and ET B inhibition.
Patent AU-6953291-A (AU)
Title: Method and apparatus for electronic control of terry loom
Inventor: HERRIN EUGENE JAMES
IPC: D03D39/22
Filed: 1990-10-15
Abstract: A terry loom having a negative pile warp let-off motor is electronically controlled to produce terry having uniform pile-to-ground warp ratio. The negative pile warp let-off motor is controlled to dispense pile warp yarn at a rate which yields the desired pile-to-ground warp ratio regardless of the tension on the pile warp yarn. The desired rate of pile warp let-off may be provided to the loom controller as a known quantity or may be calculated by the loom controller based upon the known desired pile-to-ground warp ratio and a measured or preset ground warp let-off rate. The desired pile warp let-off rate is compared to the actual pile let-off rate, and a signal is generated based upon deviations between actual and desired pile warp let-off rates, to control the pile warp let-off motor. Simplified control with uniform pile-to-ground warp ratio is thereby provided.
Patent AU-7038491-A (AU)
Title: Apparatus and method for detecting effects indicating physical state of health and fitness
Inventor: EGELY GYORGY
IPC: A63H33/40
Filed: 1990-12-17
Abstract: An apparatus for demonstrating and measuring physical effects being in connection with the general state of health and fitness of human beings, comprising a rotor (3) arranged rotatably on a frame (11), of the mass of 0.1 and 2.0 g, more accurately 0.3 to 0.8 g, with at least one marking (19) on the edge being suitable for reading number of turns, wherein magnetic permeability is less than 50, furtheron optionally the rotor (3) and the frame (11) are connected to each other by a spring means.
Patent AU-7336894-A (AU)
Title: Container content removal device
Inventor: MICHELSON GARY KARLIN
IPC: B65D77/30
Filed: 1994-07-25
Abstract: A container assembly (20) includes a central connecting member (30) that extends to an attached support plate (40) at the bottom of the container. After opening the top of the container, lifting the connecting member results in the contents of the container being pulled up by the support plate for ease of use. The assembly is particularly useful for materials having a thick consistency such as dog food, cat food or spackling paste which are difficult to remove from their containers. In the preferred embodiment, the support plated includes openings (42) to drain any liquid from the contents of the container as the contents are being lifted from the container. <IMAGE>
Patent AU-7504494-A (AU)
Title: Wellbore fluid
Inventor: SAWDON CHRISTOPHER ALAN
IPC: C09K8/34
Filed: 1994-08-30
Abstract: PCT No. PCT/GB94/01878 Sec. 371 Date Jan. 31, 1995 Sec. 102(e) Date Jan. 31, 1995 PCT Filed Aug. 30, 1994 PCT Pub. No. WO95/06695 PCT Pub. Date Mar. 9, 1995There is disclosed a biodegradable wellbore fluid having a continuous oil phase comprising an n-alk-1-ene having from 12 to 20 carbon atoms or a linear polyunsaturated olefin having one of the double bonds in the 1-position and having from 12 to 22 carbon atoms, or a mixture thereof.
Patent AU-7623294-A (AU)
Title: A method and apparatus for non-invasively deriving and indicating of dynamic characteristics of the human and animal intracranial media
Inventor: RAGAUSKAS ARMINAS
IPC: A61B8/04
Filed: 1994-08-24
Abstract: An ultrasonic non-invasive technique is descried for deriving the time dependencies of characteristics of certain regions in the intracranium medium. Precise measurements of the transit travel times of acoustic pulses are made and processed to extract variable portions indicative of, for example, the pulsatility due to cardiac pulses of a basal artery or a cerebroventricle or the variation in the pressure of brain tissue, as well as changes in the cross-sectional dimension of the basal artery and ventricle. In one technique, the transit time variations attributable to cardiac pulses are extracted by processing higher harmonics in the frequency domain. Frequency and phase detection techniques are described.
Patent AU-7676691-A (AU)
Title: Protein partner screening assays and uses thereof
Inventor: KINGSTON ROBERT E
IPC: G01N33/68
Filed: 1991-03-26
Abstract: A rapid, simple and inexpensive method to screen and classify proteins as partners of heterodimeric proteins is described which utilizes fusion protein constructs containing a DNA binding domain and a dimerization domain from a different protein. According to the method of the invention, heterodimer formation is detected by the ability of the protein partner to displace homodimer formation, and thus reveal a phenotypic change in a bacterial host which was dependent upon maintenance of the homodimer configuration. The method of the invention may be used to identify compounds of interest which inhibit such heterodimer formation, and especially to identify compounds which prevent heterodimer formation and activation of oncogenic transcriptional regulatory proteins.
Patent AU-7724696-A (AU)
Title: Bioactive composite material for repair of hard and soft tissues
Inventor: BONFIELD WILLIAM
IPC: A61L27/44
Filed: 1996-11-08
Abstract: Composites suitable for use as prostheses for attachment to soft tissues, such as cartilage, tendons, skin, tympanic membrane and gingiva, as well as to cancellous or trabecular bone, are based on combination of a polyolefinic binder with certain bioactive glass materials. The composites bond actively with soft tissues and are readily formulated achieve mechanical properties comparable to those of the soft tissue of interest.
Patent AU-7928587-A (AU)
Title: Glass batch feeder
Inventor: GOODE HENRY CLAUDE
IPC: C03B5/14
Filed: 1987-10-01
Abstract: A pulverulent batch stream is fed into a liquefying vessel by means of an angled feed tube so as to direct the stream tangentially onto side wall portions. The tube may be rotated so as to change the location onto which the batch stream is impinged.
Patent AU-8024494-A (AU)
Title: One-pot process for the preparation of 3-quinolonecarboxylic acid derivatives
IPC: C07D471/04
Filed: 1994-12-06
Abstract: The present invention relates to a one-pot process for the preparation of 7-heterocyclyl-substituted 3-quinolonecarboxylic acid derivatives. They have a strong antimicrobial action and include active compounds such as ofloxacin, ciprofloxacin or enrofloxacin.
Patent AU-8388791-A (AU)
Title: Heteroarylmethylbenzenes
Inventor: LANG MARC
IPC: C07D263/32
Filed: 1991-09-13
Abstract: Compounds of formula I    <IMAGE>  (I)  wherein Z, X, R, R0, R1, R2 and R3 are as defined in the description, have valuable pharmaceutical properties and are effective especially against tumors. They are prepared in a manner known per se.
Patent AU-9194198-A (AU)
Title: Method for requesting and transferring information in a digital audio broadcasting system
Inventor: REBHAN RICHARD
IPC: H04H60/23
Filed: 1998-09-14
Abstract: A method for transferring information from an information provider (100) to an information consumer (190) in a secure manner by means of a digital broadcasting (140) system and a secondary bidirectional transfer network (130). The secondary bidirectional transfer network is used for transfer of crypto keys to the information consumer. The secondary bidirectional transfer network can also be used to provide the information consumer with checksums and provide a means for the information consumer to request resending of corrupted transferred information. <IMAGE>
Patent AU-9265498-A (AU)
Title: T-cell membrane protein (tirc7), peptides and antibodies derived therefrom and uses thereof
Inventor: UTKU NALAN
IPC: G01N33/68
Filed: 1998-08-28
Abstract: The present invention discloses a T cell immune response cDNA 7 (TIRC7) encoding a T-cell transmembrane protein as well as peptides and polypeptides derived therefrom and antibodies recognizing said (poly)peptides. Also disclosed is the use thereof for the preparation of pharmaceutical compositions for use in organ transplantation, for the treatment of autoimmune, allergic or infectious diseases, or for treatment of tumors. Furthermore, methods for modulating (antigen-specific) T cell unresponsiveness inducing maintaining or reversing T cell unresponsiveness by inhibiting or stimulating an (unresponsive) T cell through the novel TIRC7 membrane protein are encompassed herein.
Patent AU-9508798-A (AU)
Title: Closed, one-handed blood sampling system
Inventor: SWENDSON DAVID L
IPC: A61M5/31
Filed: 1998-09-24
Abstract: A one-handed blood sampling reservoir for an infusion line having a configuration which allows discard fluid to be drawn into the reservoir and then returned to the patient in two squeezing motions. Both drawing and returning steps are performed by squeezing two of a plurality of finger grips provided on the reservoir. The reservoir may include a bracket which enables one-handed operation in either a hand-held or a pole-mounted configurations. In the alternative, the reservoir and finger grips may be formed by telescoped inner and outer housings without a bracket. The reservoir desirably includes a syringe-like body forming a chamber and a plunger/piston assembly reciprocal therein to vary the volume of the chamber. A narrow gap is provided in the chamber open to both inlet and outlet ports when the piston is fully seated to ensure a consistent and minimum flush volume in the chamber. The piston may be spring-loaded against the syringe body to simplify manufacturing by reducing the number of close toleranced parts required. The reservoir is preferably placed within an infusion line having a pressure transducer therein, and the spring loaded piston may be adjustable to vary the dynamic response of the fluid pressure system.
Patent BE-903730-A (BE)
Title: Screw-type water pump - has inclined cylindrical rotor guide which is non-cylindrical at discharge point
IPC: F04B19/12
Filed: 1985-11-28
Abstract: The screw-type pump for lifting liquid has a rotor working in an inclined cylindrical guide. - Before and at the discharge point the guide (V1) is non-cylindrical, while the rotor blades can be at an angle other than 90 deg. to its axis. A plate can be fitted between the central rotor tube (B) and each blade.
Patent BE-904151-A (BE)
Title: Dispositif de mesure de la temperature d'un bain metallique.
IPC: G01K1/12
Filed: 1986-01-31
Abstract: Le dispositif se compose d'un conduit extérieur monté dans une paroie d'un récipient métallurgique, et d'un conduit extérieur. Le conduit intérieur contient deux corps réfractaires successifs; le premier de ces corps est perméable aux gaz et le second présente une chambre dans laquelle est logé un moyen de mesure de la température du bain, et éventuellement un moyen de mesure de la température de solidification de ce bain.
Patent BG-95237-A (BG)
Title: Kit of tyre casing and wheel rim
Inventor: KUKENSKI PETAR P
IPC: B60B25/22
Filed: 1991-09-30
Abstract: The kit finds application in motor industry. It has a high lateral stability, small mass of the tyre casing, and low bending strains in the side parts, this decreasing the heating too. The wheel rim can be with or without a chamber, and it has a trapezium-shaped cross section. There is failure moving ensured. The tyre casing has an arched protector (1) with reinforcing layers (2). The side parts (5) are straight, and they form an angle of 90o to 15Oo, and in case of low pressure they take a wavy shape, situated outside the wheel rim. Safegarding is realized by resting of the inside surface of the protector (1) against the ring (14). The pit edges (8) are safeguarded against ejection, since their fixing does not depend on the pressure in the chamber.
Patent BR-0000775-A (BR)
Title: Processo de obtenção de um produto paraadubação agrìcola e alimentação animal, atravésdo uso do bagaço da cana-de-açúcar
Inventor: SILVA PAULO CESAR
IPC: C05F5/00
Filed: 2000-03-17
Abstract: "PROCESSO DE OBTENçãO DE UM PRODUTO PARAADUBAçãO AGRìCOLA E ALIMENTAçãO ANIMAL, ATRAVéSDO USO DO BAGAçO DA CANA-DE-AçúCAR". Compreendidopor um processo para tornar o bagaço da cana-de-açúcardesidratado ou não, hidrolisado ou não e balanceado ou não,como forragem em instalações de confinamentos de animais ouaves, para receber a incidência e a influência dos dejetos destesanimais ou aves, sobre o bagaço da cana-de-açúcar, durante operíodo de confinamento, e principalmente para receber ainfluência da umidade e da amonização que ocorre naturalmentenestes resíduos, conhecidos como celulose hemicelulose e lignina,para uma incorporação e homogeneização, direcionada à geraçãode um único componente, formado pelo bagaço decana-de-açúcar, e os dejetos de animais ou aves confinados, e aseguir se necessário for, a um processo de aeração controlada,sob condições umidade e tempo direcionados conhecida comocompostagem para a obtenção de uma melhor performance destaforragem composta, quando voltados à alimentação animal eadubação agrícola.
Patent BR-0005710-A (BR)
Title: Construção de mangueira tendo núcleo interno de nbr hidrogenada
Inventor: AINSWORTH CAROL LYNN
IPC: F02M37/00
Filed: 2000-12-04
Abstract: "CONSTRUçãO DE MANGUEIRA TENDO NúCLEO INTERNO DE NBR HIDROGENADA" Uma construção de mangueira que é particularmente adequada para uso com combustível diesel. A mangueira compreende: (a) um núcleo interno de uma camada de borracha que contém borracha de acrilonitrila - butadieno hidrogenada; (b) uma camada de material de reforço sob tensão disposto diretamente contra o núcleo interno; e (c) uma cobertura elastomérica.
Patent BR-0007422-A (BR)
Title: Controlador manual para conexão com um aparelho para a execução de um programa
Inventor: OGATA HIROKI
IPC: A63F13/92
Filed: 2000-11-10
Abstract: "CONTROLADOR MANUAL PARA CONEXãO COM UM APARELHO PARA A EXECUçãO DE UM PROGRAMA". Um controlador manual (16A) possui um corpo principal (104A) e um par de pegas (106A, 108A) montadas de forma destacável no corpo principal (104A). As pegas (106A, 108A) são feitas a partir de uma resina sintética de memória de formato e podem ser deformados em um formato que seja complementar às palmas do usuário do controlador manual.
Patent BR-0009426-A (BR)
Inventor: LINK JAMES
IPC: C07D295/26
Filed: 2000-04-03
Abstract: The present invention relates to cinnamide compounds of formula (I), in which at least one of R1 to R5 is a "cis-cinnamide" (a) or a "trans-cinnamide" (b) and the other variables are as defined in the claims, that are useful for treating inflammatory and immune diseases, to pharmaceutical compositions containing these compounds and to methods of inhibiting inflammation or suppressing immune response in a mammal. <CHEM>
Patent BR-0012832-A (BR)
Title: Processo para preparação de produtos alimentìcios de batata frita e de tiras de batata frita à base de milho e tiras de batata frita à base de milho pré-fritas congeladas
Inventor: MATTSON PETER H
IPC: A23L7/10
Filed: 2000-07-28
Abstract: "PROCESSO PARA A PREPARAçãO DE PRODUTOS ALIMENTìCIOS DE BATATA FRITA E DE TIRAS DE BATATA FRITA à BASE DE MILHO E TIRAS DE BATATA FRITA à BASE DE MILHO PRé-FRITAS CONGELADAS". São proporcionadas tiras de batata frita à base de milho e um processo de preparação relacionado à estas, onde as tiras são produzidas a partir de uma massa de farinha à base de milho. A massa de farinha à base de milho compreende uma matriz de alimento milho e farinha de milho de diferentes tamanhos de grânulos ou partículas, misturada com água e opcionais constituintes aromatizantes e temperos para formar uma massa de farinha relativamente espessa possuindo uma textura adequada para extrusão e corte para formar tiras alongadas possuindo um tamanho e forma de conformidade geralmente com a da convencional batata frita à base de batata. As tiras de massa de farinha de milho formadas e cortadas podem ser pré-fritas em óleo quente, e em seguida congeladas. As tiras de milho congeladas são subseq³entemente terminadas de preparar para o consumo, preferivelmente através de um acabamento por fritura em óleo quente. As tiras de milho terminadas de preparar possuem um paladar de aperitivo de milho em combinação com uma textura definida por uma superfície externa encrespada encasulando um interior úmido e revestido da massa de farinha.
Patent BR-0013796-A (BR)
Inventor: PAVLICEVIC MILORAD
IPC: F27B1/10
Filed: 2000-09-05
Abstract: Device for the direct reduction of iron oxides of the type with a gravitational load, comprising a reactor defining, in its upper part, at least a zone inside which the reduction reaction occurs, means (14, 15) to introduce the load through a mouth (12) of the reactor, means (18, 17, 19) to introduce a current of gas into at least one section of the reactor in correspondence with the reduction zone, outlet means (13) of the reduced material from the bottom of the reactor, and means (20) to discharge the exhaust fumes, said reactor (10) including at least a first upper zone (10a) of heating, pre-reduction and final reduction, with a taper diverging downwards, and a second lower zone (10b) of carburization and cooling, with a taper converging downwards.
Patent BR-0013966-A (BR)
Title: Compostos espiroeterocìclicos úteis como inibidores reversìveis de proteases de cisteìna
Inventor: EMMANUEL MICHEL JOSE
IPC: C07D207/14
Filed: 2000-08-28
Abstract: "COMPOSTOS ESPIROETEROCìCLICOS úTEIS COMO INIBIDORES REVERSìVEIS DE PROTEASES DE CISTEìNA". Divulgados são novos compostos inibitórios reversíveis da catepsina S, K, F, L e B das fórmulas (I), (II), (Ia) e (Ib) também definidos aqui. Os compostos são úteis para tratar doenças autoimunes. Também divulgados são os processos para preparar tais novos compostos.
Patent BR-0016268-A (BR)
Title: Processo, bem como, dispositivo para a simulação de uma propagação brusca da chama
Inventor: SPIEGEL JAKOB
IPC: G09B9/00
Filed: 2000-12-08
Abstract: "PROCESSO, BEM COMO, DISPOSITIVO PARA A SIMULAçãO DE UMA PROPAGAçãO BRUSCA DA CHAMA". A invenção refere-se a um processo para a simulação de uma propagação brusca da chama em uma instalação de treinamento de corpo de bombeiros, com uma câmara de combustão para, pelo menos, um outro local de incêndio, na qual um gás é conduzido próximo ao teto da câmara de combustão e é aceso, sendo que após uma mistura com oxigênio o gás é liberado na câmara de combustão, como uma mistura combustível de gás e oxigênio e, então, é acesa. Além disso, a invenção refere-se a um dispositivo que pode ser empregado para este processo, com um dispositivo de alimentação de gás e oxigênio na região do teto da câmara de combustão, da qual flui uma mistura de gás e oxigênio para a câmara de combustão e, pelo menos, para um dispositivo de ignição.
Patent BR-0016666-A (BR)
Title: Métodos para melhorar a estabilidade da viscosidade quando da armazenagem de uma composição amaciante de tecido e para tratar tecidos, composição amaciante de tecidos, e, uso de um derivado de açucar oleoso
Inventor: BRIGGS ADAM MATTHEW
IPC: C11D1/62
Filed: 2000-12-05
Abstract: "MéTODOS PARA MELHORAR A ESTABILIDADE DA VISCOSIDADE QUANDO DA ARMAZENAGEM DE UMA COMPOSIçãO AMACIANTE DE TECIDO E PARA TRATAR TECIDOS, COMPOSIçãO AMACIANTE DE TECIDOS, E, USO DE UM DERIVADO DE AçúCAR OLEOSO". A invenção provê um método para melhorar a estabilidade da viscosidade quando da armazenagem de uma composição amaciante de tecidos compreendendo (a) 0,5 a 30%, em peso, de pelo menos um composto amaciante de tecido de amónio quaternário ligado a éster, (b) perfume, e (c) um tensoativo não iónico alcoxilado, pela inclusão, na composição, de pelo menos um derivado de açúcar oleoso em uma relação em peso de composto amaciante para derivados de açúcar na faixa de 30:1 a 1:1. Também são providos uma composição amaciante de tecidos produzida pelo método da invenção, um método de tratamento de tecido por aplicação, ao mesmo, da referida composição, e o uso de um derivado de açúcar oleoso particular para prover estabilidade da viscosidade a 37<198>C uma composição amaciante de tecidos compreendendo 0,5% a 30%, em peso, de pelo menos um composto amaciante de tecidos de amónio quaternário ligado a éster, um perfume e um tensoativo não iónicos alcoxilado.
Patent BR-0016863-A (BR)
Title: Aparelhos para conectar sub redes de distribuição de dados e usuários com sub redes de distribuição de dados e que compreende um módulo de comunicação de dados, chassis, módulo de aplicação de processamento de dados e processos para conectar usuários sobre sub redes de distribuição de dados e sub redes de distribuição de dados com múltiplos chassis e para comutar o fluxo de dados entre módulos de comunicação de dados
Inventor: NIKOLICH PAUL E
IPC: H04Q11/04
Filed: 2000-12-28
Abstract: "APARELHOS PARA CONECTAR SUB REDES DE DISTRIBUIçãO DE DADOS E USUáRIOS COM SUB REDES DE DISTRIBUIçãO DE DADOS E QUE COMPREENDE UM MóDULO DE COMUNICAçãO DE DADOS, CHASSIS, MóDULO DE APLICAçãO DE PROCESSAMENTO DE DADOS E PROCESSOS PARA CONECTAR USUáRIOS SOBRE SUB REDES DE DISTRIBUIçãO DE DADOS E SUB REDES DE DISTRIBUIçãO DE DADOS COM MúLTIPLOS CHASSIS E PARA COMUTAR O FLUXO DE DADOS ENTRE MóDULOS DE COMUNICAçãO DE DADOS". Um sistema e processo para diretamente e flexivelmente comutar conexões de fluxos de pacote de dados entre nós de um sistema e rede de processamento de dados de banda larga. O sistema atua como um único comutador IP (Protocolo de Internet).