baber/WOPTO huggingface dataset:
Patent CZ-289043-B6 (CZ)
Title: Pharmaceutical preparation for treating diabetes mellitus type II
Inventor: KOLTERMAN ORVILLE G
IPC: A61K38/22
Filed: 1996-06-07
Abstract: In the present invention there is described the use of amylin agonist for preparing a pharmaceutical preparation intended for treating non-insulin-dependent diabetic individual of the type II and for reducing glucose level in blood of this individual.
Patent CZ-286525-B6 (CZ)
Title: Safety belt wind-up mechanism
Inventor: EBNER RALF
IPC: B60R22/46
Filed: 1997-03-19
Abstract: The invented safety belt (14) wind-up mechanism has a belt tightening mechanism that is engaged through the mediation of a first connecting mechanism with a belt reel (12), further a box (10), the belt reel (12) blocking automatic device being dependent on the vehicle and/or the safety belt (14), and a second connecting mechanism producing a force flow between the box (10) and the belt reel (12) after the safety belt (14) is tightened and during motion of the belt reel (12) in the direction of the safety belt (14) release. The first connecting mechanism is connected on the side of the force output and the second connecting mechanism is connected on the side of the force input with a first end of a torsion rod (30) whose other end is attached to the belt reel (12).
Patent CZ-283290-B6 (CZ)
Title: Process of stereoselective preparation of beta-phenylisoserine derivative and intermediate therefor
Inventor: DENIS JEAN-NOEL
IPC: C07C233/83
Filed: 1993-10-04
Abstract: PCT No. PCT/FR93/00966 Sec. 371 Date Apr. 5, 1995 Sec. 102(e) Date Apr. 5, 1995 PCT Filed Oct. 4, 1993 PCT Pub. No. WO94/07847 PCT Pub. Date Apr. 14, 1994This invention relates to a method of stereoselective preparation of a derivative of  beta -phenylisoserine of formula (I) by the action of an N-carbonyl-benzylimine of formula (II) on an optically active amide of a protected hydroxyacetic acid of formula (III), followed by hydrolysis of the product obtained. In formula (I), (II) or (III), R is an optionally substituted phenyl radical or R1-O, Ar is an optionally substituted aryl radical and G1 is a hydroxy function protection grouping. The product of formula (I) is particularly useful in preparing taxol and Taxotere which have remarkable antitumor properties.    <IMAGE>  (I)  ArCHNCOR (II)   <IMAGE>  (III)
Patent CZ-283312-B6 (CZ)
Title: Stabilized oxidation bath for metal treatment
Inventor: SVEHLA PAVEL RNDR CSC
IPC: C23C22/63
Filed: 1991-06-28
Abstract: This bath contains 0.05 to 0.5 moles/l of peroxodisulphate of an alkaline metal or ammonium, 0.1 to 2 moles/l of hydroxide of an alkaline metal or their mixture, 0.01 to 1 moles/l of sulphate or the chloride of an alkaline metal, up to 1 mole/l of the carbonate of an alkaline metal, and 0.001 to 0.5 moles/l of at least one substance from the group which includes fluoride or phosphate or diphosphate or the hexametaphosphate of an alkaline metal or ammonium or urea or amine, urea, and primary, secondary or tertiary amine.
Patent CS-276007-B6 (CS)
Inventor: MATULA JAN ING
IPC: F15B15/22
Filed: 1989-04-03
Abstract: Mezi obě větve (31,32) spojovacího
potrubí ( 3 ), je za hydrogenerátorem (1)
vřazen alespoň jeden hydrostatický
zámek (4), jehož přívod (311) řídicího
tlaku je připojen k té z větvi
(31,32) spojovacího potrubí (3), jejíž
průtok není tímto hydrostatickým
zámkem (4) blokován. Je určeno pro
uzavřený hydraulický obvod pojezdu
důlního dobývacího stroje pracujícího
v úklonu.
Patent CS-276551-B6 (CS)
Inventor: HUDEK LUBOMIR ING
IPC: C03B23/06
Filed: 1990-06-29
Abstract: ■Tvarovaci mechanismus je namontován v jed- ·
né pracovní stanici pracovního otočného
stolu (1) krokovacího karuselového stroje
nesoucího v zásobnících skleněné tyče (3)
zahřáté na jednom konci na tvarovaci teplotu
skla. Tvarovaci mechanismus má nejméně
dvě tvarovaci formy ¢10), které jsou radiálně
orientovány vůči obvodu pracovního otočného
stolu (1) a jsou horizontálně suvné
a výkyvně pohyblivé prostřednictvím výkyvné
páky (9). Tvarování skleněného ouška
tvarovaci formou (10) zabezpečuje tvarovapí
kladka (14) umístěná na jednom konci
kyvného pantografu (17), jehož druhý konec
nese přední kopírovací kladku (22) a zadní
kopírovací kladku (24), které sledují
tvar přední kopírovací šablony (23) a vratné
kopírovací šablony (25). Při držení vytvarovaného,
ale ještě nezchladlého skleněného
ouška zajišťuje přítlak přední kopírovací
kladky (22) a zadní kopírovací
kladky (24) k přední kopírovací šabloně
(23) a k vratné kopírovací šabloně (25)
přítlaková pružina (29) přes zdvihátko
(30) dosedající na smykací kámen (26
Patent CZ-277990-B6 (CZ)
Title: Process for continuous separation of acetone oxime from inorganic components in an aqueous solution
Inventor: GIRETH ROBERT ING
IPC: C07C249/14
Filed: 1989-07-03
Abstract: Solution is dealing with the process of continual separation of acetonoxim in the mixture with aqueous solution of ammonium sulfate and acetone.  Separation is processed in packing column where is from the side of the column sprayed the mixture of acetonoxim, aqueous solution of ammonium sulfate and acetone. From the head of column is yielded isotropic mixture acetonoxim, water and acetone and from the bottom of the column through the heater is flowing the mixture of ammonium sulfate.  Steams with the content to 0,11 molar fraction of acetonoxim are anorganic component free. Acetonoxim separated by this method is usable at the preparation of hydroxylamin salts eventually after condensation as aqueous solution in organic synthesis.
Patent CS-277043-B6 (CS)
Title: Machine for performing gradual working operations on a footwear extreme portions
Inventor: BROWN TERENCE JOHN
IPC: A43D37/00
Filed: 1989-07-19
Abstract: Two embodiments of the invention are described, namely a machine for performing an adhesive-applying operation progressively along marginal portions of the bottoms of lasted shoes and a machine for performing a roughing operation progressively along side wall portions of lasted shoes, each machine comprising a tool holder (670) for supporting a tool (20) for operating along three axes (X-, Y- and Z-axes) upon a workpiece surface, e.g. marginal portions of a shoe bottom. In addition the tool holder (670) is capable of pivoting in two directions, widthwise and lengthwise of the shoe bottom, about a point (P), but without displacement of said point in relation to the shoe support by reason of such pivotal movement. The movement along the various axes and the pivotal movement are all controlled by n.c. motors, e.g. stepping motors ((84), (144), (122), 698, 700), and operator-actuatable means is provided for enabling the path of such tool, including such pivotal movement, to be digitised under operator control.
Patent CZ-278555-B6 (CZ)
Title: Cast-iron mould for metal continuous casting
Inventor: HORNSCHEMEYER WOLFGANG
IPC: B22D11/043
Filed: 1986-07-21
Abstract: The mould comprises a backing frame (3) and an assembly of individual mould wall plates defining the casting cavity. A mould wall plate (7) comprises two complementary parts (8, 9) one of which (8) affords a surface (11) of the casting cavity (F) whilst the other (9) is shaped to mate with the frame (3). The parts (8,9) mate along an interface (10) at which coolant-conducting passages (13) are provided. Seals (16) may be provided at the interface (10) or a copper foil may be provided between the two parts (8, 9), especially if these are of different materials e.g. copper and steel. <IMAGE>
Patent CS-275615-B6 (CS)
Inventor: HONSA JAN
IPC: B28C9/04
Filed: 1987-08-28
Abstract: Řešeni ae týká zateplená betonárky, určené
pro výrobu betonových 8měai, která Je
sestavena z kontejnerů. Vynález řeší jednoduchou
montáž a demontáž 1 minimální náklady
na dopravu zateplená betonárky. Zateplená
demontovatelná betonárka se zásobníkem
na kamenivo vytápěným zasunutými topnými
vložkami sestavená z dolního kontejneru
(1), horního zadního kontejneru (2) a
horního předního kontejneru (3). V dolním
kontejneru (1) je vestavšná dolní Část zásobníku
na kamenivo a uzávěry, pod kterými
je zavššena váha na kamenivo a dolní část
skipové dráhy. Na plošlnš nad nádrži na vodu
Je uložen pneumatický agregát, čerpadlo
na vodu a nádrže na přísady s dávkovači.
Horni zadní kontejner (2) tvoři horni část
zásobníku na kamenivo a rozdělovačem frakci
v horni části. V zadní etšnš a částečně ve
střeše je výřez pro šikmý dopravník zakrytý
poklopem. V přední stěně jeou dvířka pro
vatup do zásobníku na kamenivo. Horni přední
kontejner (3) je rozdělen na dvě části.
V horní čáati je upevněna násypka na cement.
V dolní části je uložena míchačka na beton
a váha na cement. Kolem míchačky na beton
a podál zadní stěny Jeou ochozy se zábradlím
(6). Může být využita ve stavebním strojírenství.
Patent CZ-278143-B6 (CZ)
Title: Linking of two multi-axled bogies into set of rail-vehicle bogies
Inventor: AHLBORN GUNTER
IPC: B61F5/30
Filed: 1989-11-21
Abstract: The invention relates to the connection of two running gears with multiple axles to a group of running gears for railway vehicles with low-lying loading bridge (10), the running gears having at least two wheel sets (4) of small wheel base and a running gear frame, comprising side cheeks (1) and transverse beams (2) between two axles in each case, the wheel sets (4), being fixed in the running gear frame by means of axle bearings (3) and each running gear being connected to the loading bridge without king pins, merely by means of in each case a laminated bearing spring (6), lying longitudinally at the side in front of each side cheek (1), and a link suspension. The object of the invention was to combine running gears of the type mentioned at the beginning into groups of running gears and to arrange them underneath the vehicle frame or the loading bridge (10) in such a way that the exact turning angle of each running gear and of each group of running gears when travelling around a bend is ensured without enforcement and that an exact axle load balancing of the running gears of each group of running gears is ensured. This object is achieved by the running gears of each group of running gears being connected to one another by a connecting beam arranged in the longitudinal centre of the running gears and mounted on them in a jointed manner, the connecting beam (13) being arranged centrally with play between guide brackets (14) of the loading bridge (10). In this arrangement, the facing ends of each laminated bearing spring (6) of the running gears of each group of running gears are connected to each other via their links by a compensating lever, which is mounted on a bracket of the weighing bridge. <IMAGE>
Patent CS-276085-B6 (CS)
Inventor: RYSANEK VLADIMIR PROF ING DRSC
IPC: H04M1/53
Filed: 1990-12-28
Abstract: Je řešeno zařízení, které při nepřitom- '
nosti obsluhy sepne náhradní obvod, chovající
se jako obsluha a umožňuje uvést
v činnost i případná další napojená zařízení.
Telefonní linka (1) je připojena
přes spínač (2) k jednomu konci prvního
kondenzátoru (3). Druhý konec prvního
kondenzátoru (3) je připojen ke společnému
bodu katody a anody první a druhé diody
(4) a (5), které jsou zapojeny jako
napěťový zdvojovač. Paralelně k tomuto
napěťovému zdvojovači je připojen druhý
kondenzátor (6), jehož společný bod s katodou
druhé diody (5) je přes doutnavku
(7) připojen na řiditelný rezistor (8).
Posuvný kontakt řiditelného rezistoru
(8) je připojen k cívce relé (9). První
spínací kontakt (10) relé (9) je připojen
přes rezistor (12) ke společnému bodu
spínače (2) a prvního kondenzátoru (3).
Relé (9) může mít další spínací kontakty
(ll), k nimž jsou připojena další pomocná
el< "rická zařízení.
Patent CZ-283324-B6 (CZ)
Title: Pump with reciprocating motion
Inventor: CLOCKEMANN RALPH
IPC: F03C99/00
Filed: 1993-10-22
Abstract: PCT No. PCT/AU93/00547 Sec. 371 Date Apr. 21, 1995 Sec. 102(e) Date Apr. 21, 1995 PCT Filed Oct. 22, 1993 PCT Pub. No. WO94/10452 PCT Pub. Date May 11, 1994An engine for driving a piston arrangement for pumping water from an inlet to an outlet at a higher level is disclosed. The engine includes a hollow housing having an inlet and an outlet between which liquid passes, the housing at least partly enclosing a chamber through which the liquid flows from the inlet to the outlet. A movable wall is mounted in the housing and partly defines the chamber. A valve is provided to open and close the outlet so that when it closes, liquid in the chamber is suddenly decelerated producing an increase in pressure in the chamber to force the wall to move to a direction so as to increase the volume of the chamber. After an initial increase in the pressure, the water relaxes and the pressure decreases to such an extent that a spring will open the valve and the spring returns the wall to the position of decreased volume in the chamber. Thus, the wall is caused to reciprocate under the influence of pressure of the liquid increasing and decreasing as the valve is opened and shut.
Patent CZ-295983-B6 (CZ)
Title: Cosmetic composition and skin care method
Inventor: GRANGER STEWART PATON
IPC: A61K8/34
Filed: 1997-09-18
Abstract: In the present invention, there is disclosed a cosmetic composition comprising: (a) from 0.001 to 10 percent of a compound selected from the group consisting of retinol, retinyl ester and mixtures thereof; (b) from 0.001 to 50 percent of a compound which at 100 micron concentration inhibits at least 20 of LRAT or ARAT catalyzed retinol esterification as measured by an in vitro microsomal assay; wherein the compound is selected from derivatives of cyclic unsaturated hydrocarbons and wetting agents, hydroxy ethyl imidazoline derivatives of fatty acids; and (c) a cosmetically acceptable vehicle. Disclosed is also a cosmetic method of conditioning skin wherein the method comprises applying topically to skin the above-described composition.
Patent CZ-292509-B6 (CZ)
Title: Xanthine derivatives, process of their preparation and medicaments containing them
Inventor: GEBERT ULRICH DR
IPC: C07D473/04
Filed: 1997-06-05
Abstract: In the present invention there are disclosed xanthine derivatives of the general formula I, in which 1) the symbols Re1 and Re3 represent each an alkynol residue of the general formula Ia or Ib, Re2 represents alkyl containing 1 to 5 carbon atoms, cycloalkyl containing 3 to 6 carbon atoms or cycloalkylalkyl containing 4 to 6 carbon atoms in the cycloalkyl moiety, Re4 denotes hydrogen or alkyl containing 1 to 3 carbon atoms, Re5, Re6 and Re7 are each hydrogen, alkyl containing 1 to 6 carbon atoms, cycloalkyl having 3 to 6 carbon atoms, cycloalkylalkyl containing 4 to 8 carbon atoms in the cycloalkyl moiety, arylalkyl having 1 or 2 carbon atoms in the alkyl moiety and the aryl moiety being derived from benzene or naphthalene, or trialkylsilyl having 1 to 4 carbon atoms in the alkyl, or Re5 and Re6 together with a nitrogen atom to which they are attached  form an optionally substituted four- or seven-membered   saturated ring that can optionally contain another heteroatom, A represents alkylene having 1 to 6 carbon atoms, and Ze- denotes anion of a physiologically acceptable acid, or 2) one of the Re1 and Re3 residues represents an alkynol  residue of the general formula Ia or Ib and the another of the Re3 and Re1 residues denotes hydrogen or Re8, wherein Re8 represents alkyl containing 1 to 6 carbon atoms, cycloalkyl having 3 to 6 carbon atoms or cycloalkylalkyl containing 4 to 8 carbon atoms in the cycloalkyl moiety. These derivatives are suitable for preparing medicaments intended for treating cerebrovascular diseases exhibiting ischemia-conditioned extinction of nerve cells.
Patent CZ-282400-B6 (CZ)
Inventor: KOCH KEVIN
IPC: C07D407/12
Filed: 1992-11-13
Abstract: Jsou popsány benzpyranové sloučeniny obecného vzorce I, ve kterém znamená A kyslík, CH.sub.2.n., síru, NH nebo N(C.sub.1.n.-C.sub.6.n.)alkyl; n je 0 , 1 nebo 2; R.sup.1.n. je zbytek na poloze b nebo vzorce (E); R.sup.2.n., R.sup.8.n.,R.sup.9.n. a R.sup.10.n. představují vodík nebo každý nezávisle představuje jeden nebo libovolné dva z následujících významů:fluo'r, chlo'r, alkylová skupina, alkoxyskupina, perfluoralkylový skupina perfluoralkoxyskupina, alkylthioskupina, alkylsulfinyl a alkylsulfonyl; R.sup.3.n. představuje -(CH.sub.2.n.).sub.q.n.CHR.sup.11.n.R.sup.12.n., -(CH.sub.2.n.).sub.q.n.R.sup.12.n., -O(CH.sub.2.n.).sub.p.n.CHR.sup.11.n.R.sup.12.n. nebo -O(CH.sub.2.n.).sub.p.n.R.sup.12.n.; p je 0, 1 nebo 2; a q je 0, 1, 2 nebo 3; R.sup.4.n. představuje karboxyskupinu, tetrazolylovou skupinu nebo skupinu R.sup.13.n.SO.sub.2.n.NHCO; R.sup.11.n. znamená vodík, alkyl nebo R.sup.8.n.-substituovanou fenylovou skupinu, kde R.sup.8.n. má uvedený význam; R.sup.12.n. a R.sup.13.n. předstŕ
Patent CZ-291927-B6 (CZ)
Title: Method for the production of bristle goods
Inventor: WEIHRAUCH GEORG
IPC: A46D3/04
Filed: 1997-04-17
Abstract: Brushes with a bristle carrier (4, 16, 20) and a bristle facing of individual, vertical plastic bristles (4, 16, 20) are manufactured in that the individual bristles 4, 16, 20) with their fastening-side ends (14) at the front are introduced into in each case one hole (13) of a hole template (7), whose hole diameter is slightly larger than that of a single bristle (4, 16, 20) and whose hole pattern corresponds to the positioning of the bristles (4, 16, 20) within the bristle (4, 16, 20) facing or part thereof, to such an extent that their fastening-side ends (14) project roughly to the same extent at the opposite side of the hole template (7). The bristles (4, 16, 20) are subsequently fixed against axial and radial displacement in the hole template (7), at least on the fastening-side surface of the bristle (4, 16, 20) carrier (15) is prepared a bed (3) of liquid, curable material, the liquid material flows round the bristles (4, 16, 20) with their fastening-side ends (14) immersed in the bed (3) and subsequently the bed (3) is cured.
Patent CZ-296590-B6 (CZ)
Title: Locking device
Inventor: LERCHNER LEONHARD
IPC: E05B49/00
Filed: 1999-02-18
Abstract: The present invention relates to a locking device comprising at least one key (22) and a locking cylinder (10) having at least one cylinder core (11, 12) with a key groove mounted in a rotating manner in a cylinder armored housing (2). The locking device is further provided with a locking element (21) which in its locked position prevents the cylinder core (11, 12) from being rotated by means of the key (22) and in its release position allows for the cylinder core (11, 12) to be rotated by means of said key (22). The invention further provides for an actuator (19) which blocks the locking element (21) in the locked position and releases it in the release position, as well as an electronic code generator (42) in the key (22) and an electronic code evaluator (37), which controls the actuator(19). The locking cylinder (10) has a cylinder armor-plate (1) comprising an amour-plate (1) housing (2) covering the cylinder armored housing (2) and an amour-plate disk (6) mounted therein in a rotating manner and having a key (22) insertion slot (7) which is flush with the key groove of the cylinder core (11, 12). The locking element (21) and the actuator (19) are arranged in the armor plate housing(2). In its locked position, the locking element (21) engages the armor-plate disk (6) such as to prevent rotation and releases it in the release position.
Patent CZ-286153-B6 (CZ)
Title: Concrete with demanded amount of grains with size not exceeding 0.25 mm
Inventor: PAVLICA JIRI
IPC: C04B18/12
Filed: 1998-11-19
Abstract: The proposed concrete with demanded amount of grains with size not exceeding 0.25 mm of all components contained in such concrete contains in addition to fraction of coarse aggregates a an aggregate fraction 0-4 from at least  two different sources, from which the aggregate fraction 0-4 of the first source contains 0.1 to 10 percent by weight grains with size up to 0.5 mm and 80 to 88 percent by weight grains with size exceeding 0.5 mm and the aggregate fraction 0-4 of the second source contains 5 to 30 percent by weight fine grains with size up to 0.25 mm and 15 to 60 percent by weight grains with size up to 0.5 mm and 40 to 85 percent by weight grains with size above 0.5 mm, whereby within the range of dosing 150 to 450 kg cement per one cubic meter of concrete the both sources mutual ratio ranges between 5 : 95 to 95 : 5 percent by weight.
Patent SK-280161-B6 (SK)
Title: Substitued pipecolinic acid derivatives and pharmaceutical preparation them containing and their use
Inventor: ANDERSON PAUL C
IPC: C07D403/12
Filed: 1993-03-12
Abstract: Disclosed herein are derivatives of pipecolinic acid of formula (1) wherein X is a terminal group, for exemple, an aryloxycarbonyl, an alkanoyl or an optionally mono- or disubstituted carbamoyl; B is absent or an amino acid residue, for example, Val or Asn; R1 is hydrogen or a ring substituent, for example, fluoro or methyl; R2 is alkyl; and Y is a ring substituent, for example, phenoxy, 2-pyridinylmethoxy, phenylthio or 2-pyridinylthio. The compounds inhibit the activity of human immunodeficiency virus (HIV) protease and interfere with HIV induced cytopathogenic effects in human cells. These properties render the compounds useful for combating HIV infections.
Patent SK-279905-B6 (SK)
Title: Process for the preparation of adipic acid
Inventor: DENIS PHILIPPE
IPC: B01J23/46
Filed: 1992-09-30
Abstract: The subject of the invention is a process for the preparation of adipic acid by reaction of water and carbon monoxide with at least one pentenic acid, in the presence of an iridium-based catalyst and of at least iodinated promoter, at a high temperature, under a pressure greater than atmospheric pressure, in at least one solvent chosen from the group consisting of saturated aliphatic or cycloaliphatic hydrocarbons and their halogenated derivatives, aromatic hydrocarbons and their halogenated derivatives, and aliphatic, aromatic or mixed ethers, the I/Ir atomic ratio being less than 20.
Patent CZ-299568-B6 (CZ)
Title: Solar cell with a solar collector and accumulation elements
Inventor: FENT GIUSEPPE
IPC: F24J2/04
Filed: 1999-04-20
Abstract: In the present invention, there is disclosed a solar cell (1) comprising a honeycomb structure (5), which is situated behind a rear-ventilated glass pane (2) and which exhibits durable storage properties. The solar cell (1) characterizes a solar energy yield (v') by an arrangement, which selects for an angle of incidence. Said solar energy yield does not lead to overheating in the room interior (R) also when the sun is at a high position. A thermal time constant is obtained by means of heat insulations (11, 12) and storage elements (13), which are vapor permeable and connected in succession. Said time constant guarantees comfortable temperatures in the interior (R) of the house also in the case of low supplementary heating. The solar cell (1) considerably reduces heat requirements and can be optimally adapted to a wide range of local climate relationships, whereby emission of heat by the storage elements (13) takes place with maximum delay of at least four hours.
Patent CZ-307116-B6 (CZ)
Title: Amorphous ritonavir, methods for its preparation, its use, and a pharmaceutical composition comprising it
Inventor: BAUER JOHN F
IPC: C07D417/12
Filed: 1999-07-19
Abstract: The present invention relates to substantially pure amorphous ritonavir and a process for the preparation thereof. The invention also relates to a process for the praparation of the substantially pure ritonavir crystalline polymorph Form I.