baber/WOPTO huggingface dataset:
Patent NZ-306478-A (NZ)
Title: Phenoxthylamine derivatives having high affinity for the 5-ht<sub>1a</sub> receptor, preparation thereof, use thereof as drugs, and pharmaceutical compositions containing said derivatives
Inventor: BIGG DENNIS
IPC: C07D217/26
Filed: 1997-10-03
Abstract: Phenoxyethylamine derivatives of general formula (I) having high affinity for the 5-HT1A receptor, methods for preparing same, pharmaceutical compositions containing said derivatives, and their use, in particular as gastric acid secretion inhibitors or as antiemetics, are disclosed. In general formula (I), Ar is phenyl substituted by one or more substituents; and R is a C1-10 hydrocarbon radical selected from straight or branched alkyl, alkenyl or alkynyl radicals, saturated or unsaturated mono- or polycyclic cycloalkyl, cycloalkylalkyl or alkylcycloalkyl radicals; a pyridyl or isoquinolyl radical, phenyl optionally substituted by one or more substituents, and salts thereof.
Patent NZ-326669-A (NZ)
Title: Thiopyran or pyran derivatives useful as pharmaceutical agents
Inventor: HORWELL DAVID C
IPC: A61P25/06
Filed: 1997-01-02
Abstract: A thiopyran or pyran derivative of formula (I) or a pharmaceutically acceptable salt thereof wherein: X is O, S, S(O), S(O)2, or NR1; R1 is hydrogen, alkyl, benzyl, -C(O)R2 or -CO2R3; R2 is alkyl, or optionally substituted benzyl, or phenyl; R3 is alkyl or optionally substituted benzyl and R is hydrogen or alkyl. The pharmaceutical composition thereof is useful for treating epilepsy, faintness attacks, hypokinesia, cranial disorders, neurodegenerative disorders, depression, anxiety, panic, pain, and neuropathological disorders.
Patent NZ-332962-A (NZ)
Title: Inhaler apparatus with modified surfaces for enhanced release of dry powders that are electrostatically charged
Inventor: DATTA PABITRA
IPC: A61M15/00
Filed: 1997-06-10
Abstract: The inhaler apparatus comprises interior surfaces having contact with medicament particles of a selected size range for inhalation. The interior surfaces include an interior surface of a mouthpiece and a substrate with medicament particles deposited thereon. At least one such interior surfaces is textured having indentations or raised areas defining valleys of dimension and spacings selected to decrease the area of contact between medicament particles of a selected size range and the textured surface to reduce the adherence of the medicament particles to the textured surfaces.
Patent NZ-333586-A (NZ)
Title: Anticonvulsant sulfamate derivatives, preferably topiramate, useful in treating obesity
Inventor: SHANK RICHARD P
IPC: H01R12/14
Filed: 1997-06-23
Abstract: The specification relates to a method for treating obesity using the above known compounds. The variables are depicted below: X=CH2 or O; R= H or alkyl: and R2, R3, R4 & R5 are independently H, or lower alkyl, and when X is O R2 and R3 and/or R4 and R5 together may be a methylenedioxy group.
Patent NZ-333775-A (NZ)
Title: Safety screen for a workshop machine which has a drive motor to lower the screen before the machine starts to operate
Inventor: KOENDERS ANDREAS ALBERTUS MARI
IPC: F16P3/16
Filed: 1997-07-14
Abstract: A safety device for a workshop machine contains a safety screen (26) which is equipped with powering means (32) in order to lower the screen (26) before the machine starts to operate.  The powering means contain friction rolls (5) on opposite sides of screen (26) coupled to a drive motor (32).  Screen (26) is equipped on both its top side and its bottom side with approach switching means (22-25) which, when moved, give off an electric signal to a central processing unit (30).  The central processing unit (30) is capable of controlling drive motor (32) in accordance with the signals given off by the approach switching means.
Patent NZ-333894-A (NZ)
Title: Liquid delivery device, capsule within cigarette-like paper cylinder
Inventor: POWELL NIK
IPC: A24B15/00
Filed: 1999-11-24
Abstract: liquid cigarette device comprising gelatin capsules resembling the shape of a cigarette is disclosed.
Patent NZ-334439-A (NZ)
Title: Pyrrolidinyl and pyrrolinyl ethylamine compounds as kappa-receptor agonists
Inventor: ITO FUMITAKA
IPC: C07D/
Filed: 1997-08-21
Abstract: The specification provides a compound of the following formula: and the salts thereof, wherein A is hydrogen, halo, hydroxy, Cl-C6 (preferably C1-C4) alkyl, halo C,-C6 (preferably C1-C4) alkyl, C1-C6 (preferably C1-C4) alkoxy, halo C1-C6 (preferably C1-C4) alkoxy, oxo, OY wherein Y is a hydroxy protecting group, or absent; the broken line represents an optional double bond with proviso that if the broken line is a double bond, then A is absent; Ar' is phenyl optionally substituted by one or more (preferably one to two) substituents selected from halo, hydroxy, C1-C4 alkyl, Cz-C4 alkoxy, C1-C4 alkoxy-C1-C4 alkoxy, CF3, carboxy-C1-C4 alkoxy and C1-C4 alkoxy-carbonyl-C1-C4 alkoxy; Ar2 is aryl or heteroaryl selected from phenyl, naphthyl, pyridyl, thienyl, furyl, pyrrolyl and pyrimidyl, the aryl or heteroaryl being optionally substituted by one or more (preferably one to two) substituents selected from halo, hydroxy, amino, nitro, carboxy, C1-C4 alkyl, C1-C4 alkoxy, C1-C4 alkylamino, di C1-C4 alkylamino, halo C1-C4 alkyl, C-C4 alkylthio and sulfonyl methyl; Rl is hydrogen, hydroxy, C1-C4 alkyl, C1-C4 alkoxy or OY wherein Y is a hydroxy protecting group; and R2 and R3 are independently selected from hydrogen, hydroxy, C1-C7 alkyl optionally substituted by one or more (preferably one to five) hydroxy or halo, C3-C6 cycloalkyl, C2-C6 alkenyl, C2-C6 alkynyl, C1-C7 (preferably C,-C5) alkoxy, phenyl optionally substituted by halo (preferably substituted by one or two halogen atoms), phenyl C1-C7 (preferably C1-C5) alkyl, halo substituted phenyl Cl-C7 alkyl, and (CH2)nX-R4 wherein n is one or two, X is O, NH or S and R4 is C1-C alkyl, or when Ar2 is phenyl, -Ar2-C(=O)-N(R2)- is a phthalimide group and R3 is C1-C7 alkyl, or R2 and R3, together with the nitrogen atom to which they are attached, form a pyrrolidine, piperidine or morpholine ring, optionally substituted by Cl-C3 alkyl or halo. When Ar2 is phenyl, R2R3N-C(=O)- is preferably at the meta or para position on the phenyl ring with respect to 2-(A-pyrrolydinyl)-1-Ar-ethyl-N(R)- When oxo is selected as "A" group, it is apparent that the oxygen atom should be attached to the pyrrolidinyl group through a double bond. The pyrrolidinyl and pyrrolynyl ethylamine compounds of formula (I) exhibit good kappa-receptor agonist activity, and thus are useful as an analgesic, anesthetic, anti-inflammatory or neuroprotective agent, and also useful in the treatment of arthritis, stroke or functional bowel disease such as abdominal pain.
Patent NZ-337767-A (NZ)
Title: Punch with saw tooth leading face, for perforating cementitious tiles
Inventor: DEVEREUX WILLIAM
IPC: E04B9/04
Filed: 1998-04-09
Abstract: Cementitious board or tiles are acoustically modified by the inclusion of clean edged perforations. The perforations, in the form of slits or holes, are made using a punch (10) of elongate section having a leading face (16) with a saw tooth profile along its length. The side faces (12) are corrugated with a pitch equal to that of the pitch of the saw tooth profile. The saw tooth depth is less than 2mm and the included angle of the tooth profile is between 90o and 150o.
Patent NZ-500764-A (NZ)
Title: Catalysts containing partially embedded osmium, iridium and rhodium coated with catalytically active metal useful in the preparation of carboxylic acid salts by the reaction of primary alcohols with a hydroxide base
Inventor: EBNER JERRY R
IPC: C07C59/305
Filed: 1998-05-05
Abstract: Supported catalyst useful in the preparation of carboxylic acid salts, said catalyst comprising; an alkali resistant support, a plurality of metal particles selected from the group consisting of osmium, iridium and rhodium and a coating of a catalytically active metal selected from the group of copper, cobalt, nickel, cadmium or mixtures thereof.
Patent NZ-501139-A (NZ)
Title: Visiting card with CD rom
Inventor: FISCHER GERHARD
IPC: G06K19/04
Filed: 1998-04-15
Abstract: A business card of plastic with a printed upper side with directly visually readable information, with a lower side which is provided with electronically processed data which can be optically or acoustically reproduced by a CD drive, and with means for its centered accommodation in a CD drive, characterised in that the means for the centered accommodation are projecting downwardly from the lower side such that in the condition of the business card inserted into a CD drive they at least approximately bear on the centering shoulder for Mini-CD's.
Patent NZ-507137-A (NZ)
Title: Water making apparatus
Inventor: HODGSON THOMAS CLARENCE
IPC: F24F1/02
Filed: 1999-02-25
Abstract: This apparatus (1) is directed towards the production of water from air, and in particular for the production of drinking water. The apparatus (1) includes an air intake device (2) adapted to move air into the apparatus, an evaporator (7) adapted to freeze the water contained in the air issuing from the air intake device and defrosting means (5) adapted to defrost the water frozen by the adaptor; the volume of air passing over the frosting surface of the evaporator (7); evaporator being controlled by either the air intake device or the evaporator. In an alternative form the apparatus may include an air intake device adapted to move air into the apparatus, an air temperature controller to control the temperature of the air entering the apparatus, an evaporator adapted to freeze water contained in the air issuing from the temperature controller and a defroster adapted to defrost the water frozen by the evaporator. The apparatus may be employed for removing sufficient quantities of water from the air for general household use, as well as enabling the heating of this water if desired.
Patent NZ-507631-A (NZ)
Title: Adhesive microsphere transdermal drug delivery composition comprising at least 10 weight % of a softening agent incorporated within the microspheres
Inventor: CANTOR ADAM S
IPC: A61K9/16
Filed: 1999-03-25
Abstract: A  transdermal  drug delivery  composition  comprising pressure sensitive adhesive microspheres comprising: (i)   At  least  10  weight percent  of  a  softening  agent incorporated within the microspheres, and optionally: (ii) A therapeutically effective amount of a drug. Also   described  is  a  transdermal  drug  delivery  device comprising   the   transdermal  drug  delivery   composition described above disposed upon a backing.
Patent NZ-509292-A (NZ)
Title: Process for increasing the egg production and strengthening the eggshells of poultry using a bisphosphonic composition
Inventor: BARDON THIERRY
IPC: A23K50/15
Filed: 2001-01-10
Abstract: Described is a composition for administration to poultry for strengthening the eggshells, comprising a bisphosphonic acid or salt or hydrate of the acid. This is administered to the poultry before the average age of onset of laying. The bisphosphonic compound may have the formula (I), wherein; R1 and R2 are, independently selected from the group consisting of a hydrogen atom, a halogen atom, a hydroxyl group, a group -T, and a group -XT. T is selected from the group consisting of an aliphatic saturated or unsaturated hydrocarbon-based radical, optionally substituted and/or optionally interrupted with one or more O, S, N, N-CO, CO-N, CO, SO or SO2, a saturated, unsaturated or aromatic, optionally substituted carbocyclic or heterocyclic radical, and a radical with both an aliphatic part as defined above, the radical being optionally substituted and/or optionally interrupted with one or more O, S, N, N-CO, CO-N, CO, SO or SO2, and X is selected from the group consisting of O, NH, NT, S, CO, CO-NT and NT-CO, in which T is as defined above, and a physiologically acceptable hydrate or salt of this compound.
Patent NZ-510888-A (NZ)
Title: Modified peptides as therapeutic agents
Inventor: FEIGE ULRICH
IPC: A61K38/00
Filed: 1999-10-25
Abstract: Disclosed is the fusion of Fc domains with independently randomised IL antagonist peptide sequences. Linkage to the vehicle increases the half-life of the peptide, which otherwise would be quickly degraded in vivo. The preferred vehicle is an Fc domain. The peptide is preferably selected by phage display, E. coli display, ribosome display, RNA-peptide screening, or chemical-peptide screening. Such peptides are useful as pharmacologically active agents.
Patent NZ-512620-A (NZ)
Title: Tow Bar Deflector to deflect shins of passersby away from a tow bar and/or tow ball
Inventor: SWANEPOEL WYNAND JOHANNES
IPC: B60D1/60
Filed: 2001-06-27
Abstract: The deflector is typically of delta shape and fittable between tow bar and tow ball. The deflector is shaped to deflect shins and other body parts of passersby away from the tow bar and tow ball so as to prevent injury.
Patent NZ-513583-A (NZ)
Title: Rope to float clamp
Inventor: ALLOWAY PETER CHARLES
IPC: A01K75/04
Filed: 2001-08-16
Abstract: A clamp assembly for releasably securing a line 1 (e.g. a mooring rope) to a float 2, includes a unitary clip 10, preferably made from resilient wire, having a jaw section 15 to which a saddle 14 is fixed. The saddle 14 engages with the line, clamping the line against the float. A fastener 11 holds the jaw section in clamping engagement with the line.
Patent NZ-514276-A (NZ)
Title: A toilet odour extraction system using a portion of the flush water supply pipe for the extraction of odour-laden air from the toilet bowl
Inventor: VAN NIEKERK JAN ANTONIE
IPC: E03D9/052
Filed: 2001-09-19
Abstract: A  toilet bowl odour extraction system for  extracting bad   odour  laden  air  from  a  toilet  bowl,  said  odour extraction system including a conduit and an extraction  fan configured  to direct the odour laden air from  out  of  the toilet bowl along a substantially unimpeded flow path  to  a remote location through at least a portion of a flush  water supply  pipe  from  where  it enters  the  toilet  bowl  and supplies  the  toilet  bowl with flush  water,  wherein  the system  includes an anti-siphon arrangement to  prevent  the flush  water  from  flowing into and through  an  extraction portion of the extraction system.
Patent NZ-516877-A (NZ)
Title: Interactive wagering systems and methods for recording wagering events
Inventor: MARSHALL CONNIE T
IPC: G07F17/32
Filed: 2000-06-30
Abstract: An interactive wagering application is provided that automatically prompts a user to record wagering events based on entered wagers.  The recorded wagering events may be stored in a personal archive.  The races stored in the personal archive may be listed according to information associated with the stored race, such as the track, race number, and date of the races.  The interactive wagering application may also have access to a racing video archive and allow a user to search that archive for videos of prior races based on information associated with those races.  The user may view the races from the search results or save the races in the user's personal archive.  The wagering application may be implemented using platforms based on set-top boxes, personal computers, handheld computing devices, cellular telephones, or other suitable devices.
Patent NZ-517698-A (NZ)
Title: A trench cover element
Inventor: BYRNE DAVID VINCENT
IPC: E02D29/14
Filed: 2000-09-18
Abstract: A temporary trench cover comprises a number of cover elements (1) which are of prefabricated or cast metal construction. Interlink means for interengaging like cover elements on assembly comprises a male head part (35) at one end and a female slot at an opposite end. The male part (35) engages with the female slot in such a way as to allow limited controlled relative movement between adjacent cover elements on assembly in both the horizontal and vertical planes. In this way the cover elements readily follow the contour of the ground in which the trench is dug providing an even surface over the trench and, on assembly, unauthorized removal of a cover element is prevented
Patent NZ-520908-A (NZ)
Title: High fidelity reverse transcriptases and uses thereof
Inventor: POTTER ROBERT JASON
IPC: C12N1/19
Filed: 2001-03-15
Abstract: A retroviral reverse transcriptase having RNA-dependent DNA polymerase activity which comprises at least one mutation at an amino acid position corresponding to amino acids selected from: (a) tyrosine 64 of M-MMLV reverse transcriptase; (b) arginine 116 of M-MMLV reverse transcriptase; (c) lysine 152 of M-MMLV reverse transcriptase; (d) threonine 197 of M-MMLV reverse transcriptase; (e) glutamine 190 of M-MMLV reverse transcriptase; (f) phenylalanine 309 of M-MMLV reverse transcriptase; wherein the retroviral reverse transcriptase is not derived from a human immunodeficiency virus; the reverse transcriptase with properties selected from the group consisting of: (a) increased fidelity in comparison to the corresponding wild-type enzyme; (b) reduced terminal deoxynucleotidyl transferase activity n comparison to the corresponding wild-type enzyme; and (c) reduced RNAse H activity in comparison to the corresponding wild-type enzyme; and method for producing the reverse transcriptase, for amplifying a nucleic acid molecule and for sequencing a nucleic acid molecule.
Patent NZ-526632-A (NZ)
Title: Novel acyclic nucleoside phosphonate derivatives, salts thereof and process for the preparation of the same
Inventor: CHOI JONG-RYOO
IPC: A61K31/675
Filed: 2002-01-18
Abstract: An acyclic nucleoside phosphonate derivative represented by formula (1) is disclosed. Also described is a process for preparing the compound of formula (1). Acyclic nucleoside phosphonate derivatives of formula (1) are useful for the production of pharmaceutical compositions for the treatment of hepatitis B.
Patent NZ-527306-A (NZ)
Title: Aluminium-wettable porous ceramic material
Inventor: DE NORA VITTORIO
IPC: C25C3/08
Filed: 2002-03-04
Abstract: A composite material is disclosed that may be used as an aluminium-wettable component (21,21', 41,41', 51), in particular of a cell for the electrowinning of aluminium (60), wherein the composite material comprises an openly porous or reticulated ceramic structure whose surface during use is exposed to and wetted by molten aluminium. The structure is made of ceramic material inert and resistant to molten aluminium, such as alumina, and an aluminium-wettable material that comprises metal oxide and/or partly oxidised metal, in particular of manganese, iron, cobalt, nickel, copper or zinc, which is/are reactable with molten aluminium to form a surface layer containing alumina, aluminium and metal derived from the metal oxide and/or partly oxidised metal. The ceramic structure comprises a coating of the aluminium-wettable material on the inert and resistant ceramic material, or is made of a mixture of the inert and resistant material and of the aluminium-wettable ceramic material. The aluminium-wetted component is suitable for use as a cathode (21,21'), as a sidewall (41,41') or as another component (51) which during use is exposed to molten aluminium (60) and/or electrolyte (5), or another oxidising and/or corrosive media at high temperature.
Patent NZ-527662-A (NZ)
Title: Building cladding to frame connector element with apertured web for drainage and/or ventilation
Inventor: HASTIE ANDREW JOHN
IPC: E04B1/38
Filed: 2003-08-18
Abstract: Element 1 is typically folded by folding about lines 9, 10 to form a channel. This is then used to space building elements such as cladding (not shown) from wall framing 7. Drainage and/or ventilation holes 4 are provided. In one embodiment tabs 5 and recesses 6 are formed to facilitate fastening of the element to framing 7.
Patent NZ-533030-A (NZ)
Title: Combination of a selective PDE4 inhibitor and an adrenergic beta-2 receptor agonist
Inventor: YEADON MICHAEL
IPC: A61K45/00
Filed: 2002-11-22
Abstract: A combination of a selective PDE4 inhibitor, as defined herein, and an adrenergic ss2 receptor agonist for simultaneous, sequential or separate administration by the inhaled route in the treatment of an obstructive airways or other inflammatory disease.
Patent NZ-533144-A (NZ)
Title: Method of forming an inlaid pattern in an asphalt surface using first and second templates
Inventor: WILEY PATRICK CARL
IPC: E01C19/43
Filed: 2002-12-03
Abstract: In one embodiment the method comprises the steps of providing a first template having a predetermined pattern; impressing the first template into the asphalt surface when the asphalt surface is in a pliable state to form an impression therein; removing the first template from the asphalt surface to expose the impression; providing a second template having a predetermined pattern matching the pattern of the first template; inserting the second template into the impression; and fixing the second template in position within the impression to form the inlaid pattern. The second template may consist of a preformed thermoplastic grid having a colour and/or texture contrasting with the asphalt surface. In another embodiment the second template may include a light source for illuminating the template after it has been fixed in position. A heating method is described for gradually heating large asphalt surfaces using a reciprocating bank of infrared heaters to thermally fix the thermoplastic grid in place.
Patent NZ-533360-A (NZ)
Title: Improved method for preparing 3-hydroxy-4-hydroxymethyl-pyrrolidine compounds
Inventor: LENZ DIRK HENNING
IPC: C07D261/02
Filed: 2004-06-04
Abstract: Disclosed herein is a process for preparing (3R,4R)-3-hydroxy-4-hydroxymethylpyrrolidine compound of formula (I), or (3S,4S)-3-hydroxy-4-hydroxymethylpyrrolidine compound of formula (Ia), wherein the process involves, as a key step, the enzyme-catalysed enantioselective hydrolysis of a racemic 3,4-trans-disubstituted pyrrolidinone compound of formula (II), and wherein the variables R1 & R2 are as defined in the specification.
Patent NZ-545114-A (NZ)
Title: Multi-layer tube of improved physical properties
Inventor: ADAMS KEVIN
IPC: B65H75/10
Filed: 2004-07-30
Abstract: A tube having walls of multi-layer construction, wherein the multi-layer construction includes one or more sub-layers, each sub-layer consisting of a woven polymer mesh disposed in between one or more outer layers of material selected from the group consisting of paper, poly-propylene and polyethylene, wherein the tube is formed by affixing the sub-layers to each other whilst the sub-layers are wound around a mandrel.
Patent NZ-547373-A (NZ)
Title: Lubricant compositions, their preparation and articles coated therewith
Inventor: MCGHEE DIANE
IPC: A61L2/08
Filed: 2004-10-22
Abstract: Disclosed is a lubricious composition suitable for medical devices that comprises a hydrophilic polymer, an isocyanate-terminated prepolymer, an alkylester of a carboxylic acid such as ethyl lactate and a solvent selected from tetrahydrofuran, dimethylformamide, methylene chloride, N-methyl pyrrolidone and cyclohexanone and mixtures thereof. The lubricious composition may optionally contain a pharmacological additive and/or a polymerized urethane. Also disclosed is a method of producing the lubricious composition and methods of coating a surface such as a medical device with the lubricious composition and the resulting coated medical devices.