baber/WOPTO huggingface dataset:
Patent RS-51237-B (RS)
Inventor: LIU CHUAN-FA
IPC: C07K19/00
Filed: 1999-10-22
Abstract: Jedinjenje koje se vezuje na mpl receptor, a ima strukturu TMP1-(L1)n-TMP2gde su TMP1 i TMP2, svaki nezavisno, odabrani iz grupe središnih jedinjenja sa strukturama odabranim od grupa koje čine:a) X2-X3-X4-X5-X6-X7-X8-X9-X10 gde,X2   je odabran iz grupe koju čine Glu, Lys i Val;       X3   je odabran iz grupe koju čine Gly i Ala; X4   je Pro;X5   je odabran iz grupe koju čine Thr i Ser; X6   je odabran iz grupe koju čine Leu, lie, Val, Ala i Phe; X7   je odabran iz grupe koju čine Arg i Lys;  X8   je odabran iz grupe koju čine Gln, Asn i Glu;X9   je odabran iz grupe koju čine Trp, Tyr, Cys, Ala i Phe;X10  je odabran iz grupe koju čine Leu, lle, Val, Ala, Phe, Met i Lys;b) X2-X3-X4-X5-X6-X7-X8-X9-X10 gde,X2   je odabran iz grupe koju čine Glu, Asp, Lys i Val;X3   je Ala;X4   je Pro;X5   je odabran iz grupe koju čine Thr i Ser;X6   je odabran iz grupe koju čine Leu, lle, Val, Ala i Phe;X7   je odabran iz grupe koju čine Arg i Lys;X8je odabran iz grupe koju čine Gln, Asn i Glu;X9   je odabran iz grupe koju čine Trp, Tyr, Cys, Ala i Phe;X10 je odabran iz grupe koju čine Leu, lle, Val, Ala, Phe, Met i Lys;c) X2-X3-X4-X5-X6-X7-X8-X9-X10gde,X2   je odabran iz grupe koju čine Glu, Asp, Lys i Val;X3   je odabran iz grupe koju čine Gly i Ala;X4   je Pro;X5   je Ser;X6   je odabran iz grupe koju čine Leu, lle, Val, Ala i Phe;X7   je odabran iz grupe koju čine Arg i Lys;X8   je odabran iz grupe koju čine Gln, Asn i Glu;X9   je odabran iz grupe koju čine Trp, Tyr, Cys, Ala i Phe;X10 je odabran iz grupe koju čine Leu, lle, Val, Ala, Phe, Met i Lys;d) X2-X3-X4-X5-X6-X7-X8-X9-X10gde,X2  je odabran iz grupe koju čine Glu, Asp, Lys i Val;X3  je odabran iz grupe koju čine Gly i Ala;X4  je Pro;X5  je odabran iz grupe koju čine Thr i Ser;X6  je odabran iz grupe koju čine lle, Val, Ala i Phe;X7  je odabran iz grupe koju čine Arg i Lys;X8  je odabran iz grupe koju čine Gln, Asn i Glu;X9  je odabran iz grupe koju čine Trp, Tyr, Cys, Ala i Phe;X10 je odabran iz grupe koju čine Leu, lle, Val, Ala, Phe, Met i Lys;e) X2-X3-X4-X5-X6-X7-X8-X9-X10gde,X2  je odabran iz grupe koju čine Glu, Asp, Lys i Val;X3  je odabran iz grupe koju čine Gly i Ala;X4  je Pro;X5  je odabran iz grupe koju čine Thr i Ser;X6  je odabran iz grupe koju čine Leu, lle, Val, Ala i Phe;X7  je Lys;X8  je odabran iz grupe koju čine Gin, Asn i Glu;X9  je odabran iz grupe koju čine Trp, Tyr, Cys, Ala i Phe;X10 je odabran iz grupe koju čine Leu, lle, Val, Ala, Phe, Met i Lys;f) X2-X3-X4-X5-X6-X7-X8-X9-X10 gde,X2  je odabran iz grupe koju čine Glu, Asp, Lys i Val;X3  je odabran iz grupe koju čine Gly i Ala;X4  je Pro;X5  je odabran iz grupe koju čine Thr i Ser;X6je odabran iz grupe koju čine Leu, lle, Val, Ala i Ph
Patent YU-44714-B (YU)
Title: Process for obtaining disymmetrical esther derivatives of 1,4-dihydropyridin-3,5-dicarbonic acid
Inventor: ROBIN J
IPC: C07D491/10
Filed: 1988-03-09
Abstract: The present invention relates to novel asymmetrical esters derived from 1,4-dihydrophyridine-3,5-dicarboxylic acid, of the formula: <IMAGE>  (I)  in which: R1 represents a C1-C4 alkyl group, R2 represents a C1-C4 alkyl group, a benzyl group, a benzoyl group or a phenyl group optionally substituted by one or more C1-C4 alkoxy, C1-C4 alkyl, cyano, nitro, hydroxyl or trifluoromethyl groups or by one or more halogen atoms, and R3 and R4, which are identical or different, each represent the hydrogen atom, a nitro group or a chlorine atom, their optical isomers and diastereoisomers and also the corresponding addition salts. These novel esters are useful in therapy, especially as antihypertensives.
Patent RS-50843-B (RS)
Inventor: GOULET SYLVIE
IPC: A61K31/4436
Filed: 2002-07-18
Abstract: Enantiomer, dijastereoizomer ili tautomer jedinjenja predstavljenog formulom II:pri čemu:R1 izabran iz grupe koja se sastoji od: H, (C1-6alkila eventualno supstituisanog sa:- halogenom, OR11, SR11 ili N(R12)2, pri čemu R11 i svaki R12 jeste nezavisno H, (C1-6)a1kil, (C3-7)cikloalkil, (C1-6)alkil- (C3-7)cikloalkil, (C1-6)alkil-aril ili (C1-6) alkil-Het, a pomenuti aril ili Het su eventualno supstituisani sa R10; ili su oba R12 međusobno kovalentno vezana i sa azotom za koji su vezani obrazuju 5, 6 ili 7 - člani zasićeni heterocikl;R2 je izabran između: halogena, R21, OR21, SR21, COOR21, SO2N(R22)2 N(R22)2, CON(R22)2, NR22C(O)R22 ili NR22C(O)NR22, pri čemu R21 i svaki R22 jeste nezavisno H, (C1-6 alkil, haloalkil, (C2-6)alkenil, (C3-7)cikloalkil, (C2-6)alkinil, (C5-7)cikloalkenil, 6 ili 10 - člani aril ili Het, a pomenuti R21 i R22 su eventualno supstituisani sa R20;ili su oba R22 međusobno vezana tako da obrazuju 5, 6 ili 7 - člani zasićeni heterocikl sa azotom za koji su vezani;R3 izabran između (C1-6) alkila, haloalkila, (C3-7)cikloalkila, (C5-7)cikloalkenila, (C6-10) bicikloalkila, (C6-10)bicikloalkenila, 6 - ili 10 - članog arila, Het, (C1-6)alkil - arila ili (C1-6)alkil -Het,a pomenuti alkil, cikloalkil, cikloalkenil, bicikloalkil, bicikloalkenil, aril, Het, alkil - aril i alkil - Het su eventualno supstituisani sa od 1 do 4 supstituenta izabrana između: halogena, ilia) (C1-6) alkila eventualno supstituisanog sa:- OR31 ili SR31, pri čemu R31 jeste H, (C1-6alkil), (C3-7)cikloalkil, (C1-6)alkil - (C3-7) cikloalkil, aril, Het (C1-6 alkil - aril ili (C1-6) alkil - Het; ili- N(R32)2, pri čemu svaki R32 jeste nezavisno H, (C1-6) alkil, (C3-7) cikloalkil, (C1-6) alkil - (C3-7) cikloalkil, aril, Het, (C1-6) alkil - aril ili (C1-6) alkil - Het; ili su oba R32 međusobno kovalentno vezana i sa azotom za koji su vezani obrazuju 5, 6 ili 7 -člani zasićeni heterocikl;b) OR33, pri čemu R33 jeste H, (C1-6)alkil, (C3-7)cikloalkil ili (C1-6) alkil - (C3-7) cikloalkil, aril, Het, (C1-6) alkil - aril ili (C1-6) alkil - Het;c) SR34, pri čemu R34 jeste H, (C1-6)alkil, (C3-7)cikloalkil, ili (C1-6)alkil - (C3-7) cikloalkil, aril, Het, (C1-6) alkil – aril ili (C1-6) alkil - Het; id) N(R35)2, pri čemu svaki R35 jeste nezavisno H, (C1-6) alkil, (C3-7) cikloalkil, (C1-6) alkil - (C3-7)cikloalkil, aril, Het, (C1-6)alkil - aril ili (C1-6)alkil - Het; ili su oba R35 međusobno kovalentno vezana i sa azotom za koji su vezani obrazuju 5, 6 ili 7 - člani zasićeni heterocikl;K jeste N ili CR4, pri čemu R4 jeste H, halogen, (C1-6) alkil, haloalkil, (C3-7) cikloalkil ili (C1-6) alkil - (C3-7) cikloalkil; ili R4 jeste OR41 ili SR41, COR41 ili NR41COR41, pri čemu svaki R41 jeste nezavisno H, (C1-6)alkil, (C3-7)cikloalkil ili (C1-6alkil- (C3-7)cikloalkil; ili R4 jeste NR42R43, pri čem
Patent ZA-81882-B (ZA)
Title: Television set with supervisory functions of alarming burglary and safe watching distance
Inventor: HO CHI CHEN
IPC: G08B13/00
Filed: 1981-02-10
Abstract: A supervisory assembly incorporates a sensing means operatively associated with a TV set, so that one of the options available to the user is that when the sensing means detects someone it responds by altering the TV output. For example it may blank the screen, cut the TV power supply, or use the TV to make an alarm noise. 
<??>The sensing means has a detecting device (1), the output of which passes through a signal processing circuit (2) so as to operate a switch element (4). The switch element can operate a TV control means (6), to affect the TV output. Other, conventional, alarms (5,7) may also be operated by the switch element (4). 
<??>The assembly has use as a burglar alarm, and also for warning that someone is closer to the TV than a safe watching distance. In the latter case it is useful if the assembly's response is delayed slightly, so as to prevent it from giving the alarm when e.g. someone changes TV channel. 
<??>The sensing means may operate by emitting a signal (eg. ultrasonic) and detecting any reflection of it.
Patent ZA-91392-B (ZA)
Title: Di-and tetra-fluoro analogs of squalene as inhibitors of squalene epoxidase
Inventor: JARVI ESA TERO
IPC: A61K31/045
Filed: 1991-01-18
Abstract: This invention relates to certain novel di- and tetra-fluoro analogs of squalene and to their methods of use in lowering plasma cholesterol and in inhibiting squalene epoxidase in patients in need thereof.
Patent AT-407038-B (AT)
Title: Process and apparatus for washing contaminated screenings
IPC: C02F1/00
Filed: 1997-07-07
Granted: 2000-11-27
Abstract: The invention relates to a process for washing contaminated screenings, in particular in sewage treatment plants. It is especially characterized in that, by means of a combined linear and rotary movement, the contaminants are removed from solids or solid components introduced with feed of water. The invention further relates to an apparatus for carrying out the process. <IMAGE>
Patent AT-401242-B (AT)
Title: Apparatus for producing spacer frames for panes of insulating glass from hollow sectional strips
IPC: B21D53/74
Filed: 1992-07-16
Granted: 1996-07-25
Abstract: In an apparatus for bending hollow sectional strips into spacer frames for panes of insulating glass which has a sloping supporting wall 1, at the bottom edge 8 of which at least one bending head 2 is provided, a conveyor track 20 for feeding in hollow sectional strips to be bent into spacer frames and an apparatus 40 for transferring hollow sectional strips from the conveyor track 20 into supports 7 in the region of the lower edge 8 of the supporting wall 1 are provided behind the supporting wall 1. As a result, the space behind the supporting wall 1 is used and the front side of the apparatus remains free so that it can be entered without danger by an operator and deposition space is saved. <IMAGE>
Patent AT-389668-B (AT)
Title: Auxiliary device for a portable drill or the like
Inventor: PURSCHKE NORBERT
IPC: B25F5/02
Filed: 1986-12-01
Granted: 1990-01-10
Abstract: A device for making wall cutouts for retrofitting hollow wall boxes of an electric installation. The device is driven by a drive device, such as a drill, and has a hollow drill as its working tool. In this connection, this drive device is assigned a connectable auxiliary device 60 which has a connecting part 61 and a spring- loaded insertion body 72 which can be introduced into a wall cutout which has already been made. The centre of rotation of the insertion body 72 has a distance from the centre point of the actual working tool of the device which corresponds to the standard distance of the centre points of installation devices of an installation device combination. The device has an elongate connecting part 61 which has, at one of its ends, a detachable clamp 62, 63, 64, 65 which can be fastened on the standard fastening receiver of the drill and, at its other end, a receiving bush 67. Arranged in the latter is the rear end of a connecting rod 68 for the insertion body 72. <IMAGE>
Patent AT-395480-B (AT)
Inventor: MALNIG HELMUT W DIPL ING
IPC: F42C19/08
Filed: 1985-12-09
Granted: 1993-01-25
Abstract: The object of the invention is to ensure symmetrical detonation of an explosive charge even when the detonation is initiated with a direction change. The electrical detonator 1 is located in a small, thin tube 2. During detonation, the peripheral tearing of the small tube 2 is passed to the relay charge 6, and is deflected through 90 degree by it. The relay charge is located in a blank 7 which has a shutter 7a towards the booster charge 10. Since the blank 7 is dimensioned such that the detonation wave reaches the shutter 7a before the collapse of the blank, the booster charge 10 (and subsequently the explosive charge) is detonated precisely symmetrically, namely only in the region of the shutter 7a. <IMAGE>
Patent CH-624821-B (CH)
Inventor: TAKE HIROSHI
IPC: G02F1/155
Filed: 1978-06-29
Abstract: An additional electrode is provided for developing a secondary electrochromic phenomenon on a counter electrode apart from the major electrochromic phenomenon which is developed between one or more display electrodes and the counter electrode. Current flows from an additional electrode to the counter electrode in developing the secondary electrochromic phenomenon. Coloration of the counter electrode, where the magnitude of an overvoltage of the counter electrode is small is stabilized to thereby enhance electronic properties of the electrochromic display. The material of the additional electrode is selected from metals having an appropriate ionization tendency with respect to an electrolyte, such as Mg, Al, Zn, Cr, Fe, Ni, Sn, and Pb, or a combination thereof. Otherwise, the material of the additional electrode is selected to be an inert material with respect to the electrolyte such as Ag, Au, Pt, Pd, In2O3, and SnO2 or a combination thereof. The combination which is composed of both the appropriate ionization tendency metals and the inert metals can be available for the additional electrode. The electrochromic display can be controlled under one of several groups of driving techniques consisting of a potentiostatic driving, a constant current driving, and a constant voltage driving method.
Patent DK-158156-B (DK)
Inventor: KASTENING BERTEL
IPC: C23F1/00
Filed: 1981-08-20
Abstract: In addition to catalyzing the reoxidization of spent alkaline etching agent, the suspension of activated carbon powder in the etching solution also increases the speed of etching when the etching solution is recirculated in the etching of printed circuit boards. The ammonium sulfate etching solution is set to a pH of about 9 by the addition of ammonia gas. In the recirculation of the etching solution, a part of the solution can be freed by filtration from suspended carbon particles and passed through the cathode and anode chambers of an electrolysis cell for the recovery of the etched metal by deposition on the cathode. The activated carbon powder for this purpose is calcined before use, at a temperature of between 900 DEG and 1200 DEG  C. in vacuum or in an atmosphere that is inert, reducing, or only slightly oxidizing as in the case of an atmosphere containing carbon dioxide, water vapor or both, in a concentration that does not appreciably oxidize the carbon particles.
Patent DK-162974-B (DK)
Inventor: BICHOT BERNARD
IPC: B31C1/00
Filed: 1985-09-05
Abstract: In the manufacture of insulating shells formed by a felt of mineral fibers wound around a mandrel, main pressing elements intervene as soon as the winding begins and remain in contact with the surface of the shell during the entire winding phase. Auxiliary pressing elements intervent only when the shell, during shaping, has reached a given outside diameter of, for example, 200 mm. The process applies particularly to the insulation of conduits of small and average outside diameters.
Patent FI-79625-B (FI)
Inventor: FANCHER PHILIP DANIEL
IPC: G08B13/24
Filed: 1983-04-06
Granted: 1989-09-29
Abstract: An article surveillance system employs a label or tag containing a non-linear impedance element, such as a semi-conductor diode, connected to a metal antenna loop configured to pick up two distinct radio frequency transmissions displaced on either side of a selected center frequency. The non-linear impedance element connects opposing sides of a closed loop section at one end of the antenna to form a tuned tank circuit having a resonant frequency twice that of the selected center frequency. A first transmitter generates a tone modulated radio frequency displaced on one side of the center frequency, and a second transmitter generates a continuous wave radio frequency displaced from the center frequency on the other side. Both transmitter signals are fed separately to respective radiating antennae located adjacent to a surveillance area. The antennae are chosen to produce circularly polarized transmission of both frequencies within the surveillance area. The two different frequencies picked up by the transponder antenna are mixed by the non-linear impedance causing the tank circuit to resonate at a single higher frequency equal to their sum, which is double the center frequency; that resonant frequency is reradiated to be picked up by a receiver antenna or antennae suitably placed with respect to the surveillance zone to be detected by a very narrow band receiver responsive to the sum frequency. The modulating tone signal is derived from the received signal to produce a gradually increasing charge that is compared against a preselected threshold level to trigger an alarm for a fixed interval only when the detected signal is of a sufficient strength and duration.
Patent FI-95044-B (FI)
Inventor: HARDER ABRAHAM
IPC: C12P1/00
Filed: 1987-07-13
Granted: 1995-08-31
Abstract: Immobilized water-insoluble biocatalysts in particulate form comprise living cells, particularly yeast, dispersed in a cross-linked gelling agent. An enzyme, particularly amyloglucosidase, may be co-immobilized in the particles. These particles are prepared by suspending the living cells in an aqueous solution of a gelling agent, dispersing this suspension in a water immiscible organic liquid to form a suspension in the liquid of aqueous particles comprising the living cells and gelling agent, gelling the gel and cross-linking the gelling agent. It is found that when living cells such as microbial cells and especially yeast are immobilized in this way, that surprisingly, not only is their viability retained, but the ability of yeast cells to produce ethanol under continuous fermentation conditions is significantly improved. Specific strains of Saccharomyces cerevisiae, suitable for immobilization in this way, are described.
Patent FI-87931-B (FI)
Inventor: ROSELLE BRIAN JOSEPH
IPC: C11D3/395
Filed: 1988-03-04
Granted: 1992-11-30
Abstract: Detergent compositions suitable for use in automatic dishwashing machines are disclosed. The compositions contain detergency builder materials, a chlorine bleach component, an optional low-foaming, bleach-stable surfactant and a relatively water-soluble stilbene dye which is color-stable with respect to said chlorine bleach component and which does not stain dishes etc.
Patent FI-80092-B (FI)
Title: Procedure for creating an endless process belt and endless process belt
Inventor: VUORIO SEPPO
IPC: F16G3/02
Filed: 1988-05-26
Granted: 1989-12-29
Abstract: To produce an endless process belt (1), a spiral wire (3) is attached to each end of a piece (2) of process belt woven in the usual way. The spiral wires (3) and the piece (2) of the process belt woven in the usual way are joined together by cutting finger-like projections in the edge of each piece (2, 3) that pass between one another, preferably in the shape of a triangle, and the pieces (2, 3) are fixed to one another by being filled at the edges and in nearby areas with binding material (6), that can be glue, resin, plastic or another material suitable for the purpose. From the process belt piece (2) equipped with spiral wires (3) at either end and woven in the usual way, an endless process belt (1) is formed by joining the spiral wires (3) using a normal spiral wire connection. In order to keep the process belt's (1) permeability largely unchanged, the spiral wires (3) can be filled out with different filler wires and similar.<IMAGE>
Patent FI-96258-B (FI)
Inventor: MORRISON DAVID GEOFFREY
IPC: H04N7/30
Filed: 1989-03-02
Granted: 1996-02-15
Abstract: Values, such as a set of coefficients in a transform-based video coder are to be transmitted sequentially in any one of a number of possible preset orders. The order to be selected is the one that results in the largest number of consecutive zeros (or low values) at the end of the sequence. Values are supplied (in an arbitrary sequence) with addresses, in parallel to a bank of assessment sections - one for each preset order - each of which translates the addresses into addresses representing a position in the respective order and records the highest for which the associated value is non-zero. The outputs of the sections are than compared to identify the lowest, and hence the optimum order of transmission.
Patent FI-108002-B (FI)
Inventor: SCHUBERT PAUL FREDERICK
IPC: C07C11/113
Filed: 1991-12-05
Granted: 2001-11-15
Abstract: Catalyst supports, catalyst systems, methods for the preparation thereof, and dimerization process therewith are provided catalyst supports are extruded from a thick paste of potassium carbonate and water catalyst systems comprise at least one elemental alkali metal deposited on the catalyst support. Optionally, the catalyst system further comprises at least one promoter.
Patent FI-87746-B (FI)
Title: Process for directing the cracking of a log and a log
Inventor: SAARELAINEN REINO
IPC: B27M3/00
Filed: 1991-12-13
Granted: 1992-11-13
Abstract: The invention relates to a process for directing the cracking of a log 18 such that the log is provided with a guide recess 19 running in its longitudinal direction and standing essentially vertically to its surface. According to the invention, the guide recess 19 is arranged in the log as periodic short recesses 19a which lie on the same straight line at a distance apart. <IMAGE>
Patent FI-98434-B (FI)
Inventor: ZIMMERMAN WALTER
IPC: A46B3/18
Filed: 1992-07-09
Granted: 1997-03-14
Abstract: An interproximal brush comprises a handle having an end portion provided with a transverse hole communicating with a longitudinal groove for receiving the elongated stem of an interproximal brush. The handle further has a cylindrical boss formed on the lower surface thereof through which the transverse hole extends, and the brush stem is retained securely in the longitudinal groove on closure of a cap, which is pivotably attached to the end portion.
Patent FI-109796-B (FI)
Inventor: HOLTON ROBERT A
IPC: C07D409/12
Filed: 1994-03-22
Granted: 2002-10-15
Abstract: A metal alkoxide having the following formula:   <IMAGE> (1)  wherein T1 is hydrogen or a hydroxy protecting group, Z is -OT2, or -OCOCH3, T2 is hydrogen or a hydroxy protecting group, and M is selected from the group comprising Group IA, IIA and transition metals are useful in the preparation of biologically active derivatives of baccatin III and 10-deacetyl baccatin III.
Patent FI-106205-B (FI)
Inventor: BRU-MAGNIEZ NICOLE
IPC: A61K31/7042
Filed: 1994-07-06
Granted: 2000-12-15
Abstract: PCT No. PCT/FR92/01241 Sec. 371 Date Jun. 29, 1994 Sec. 102(e) Date Jun. 29, 1994 PCT Filed Dec. 29, 1992 PCT Pub. No. WO93/14102 PCT Pub. Date Jul. 22, 1993.The present invention relates to the derivatives of the formula    <IMAGE>  Formula (I)  and their addition salts, and to their use in therapeutics, especially as analgesics and as antihypertensives.
Patent FI-110714-B (FI)
Title: Ventilation pipe extension arrangement - has pipes joined end to end and orientated in same direction, and linked to duct supplying fresh air into room inside building
Inventor: GROENLUND CHRISTER
IPC: F24F13/32
Filed: 1998-01-15
Granted: 2003-03-14
Abstract: Ventilation pipes (35,36) connected to a duct supplying fresh air into a room are joined together end to end orientated in the same direction.
Patent HU-191596-B (HU)
Title: Process for producing pharmaceutical composition
Inventor: PANDIT NEVEDITA
IPC: A61K47/00
Filed: 1984-03-15
Abstract: Water-soluble dispersions of chlorthalidone are prepared by a process comprising: (a) forming a solution comprising a water soluble pharmaceutically acceptable polymeric carrier and a C1-C4 alkanol,  (b) dissolving chlorthalidone in the solution thus formed, and  (c) removing the C1-C4 alkanol from the solution by evaporation, the amount of said carrier being effective to suppress substantially the formation of the alkyl ether by-product from the reaction of chlorthalidone with the C1-C4 alkanol. A preferred water soluble carrier is polyvinylpyrrolidon and a preferred C1-C4 alkanol is methanol.