baber/WOPTO huggingface dataset:
Patent CO-5631445-A2 (CO)
Title: 7-alquenilamino-triazolopirimidinas, procedimientos para su obtencion y el uso de las mismas para controlar hongos nocivos, asi como productos que los contienen
Inventor: TORMO I BLASCO JORDI
IPC: C07D487/04
Filed: 2005-10-31
Abstract: 1.- 7-Alquenilamino-triazolopirimidinas de la fórmula I en la que los sustituyentes tienen los significados siguientes:L significan, independientemente, haIógeno, C1-C6-alquilo, C1-C6 halógenoalquilo, C1-C6-aIcoxi, amino, NHR o NR2,R es alquilo C1-C8 o alquilcarbonilo C1-C8;m es 1, 2, 3, 4 ó 5;X es halógeno, ciano, alquilo C1-C4, halógenoalquilo C1-C4 o alcoxi C1-C4;R1 es alquilo C1-C3 o haIógenoaIquilo C1-C3;R2 es hidrógeno, alquilo C1-C3 o halógenoalquilo C1-C3;R3 es alquenilo C2-C10, que puede ser no sustituido o parcial o completamente sustituido o llevar uno a tres grupos Ra;Ra es halógeno, ciano, nitro, hidroxi, alquilcarbonilo C1-C6, cicloaIquilo C3-C6, aIcoxi C1-C6, halógenoalcoxi C1-C6, aIcoxicarbonilo C1-C6, -alquitio C1-C6, alquilamino C1-C6, di -alquilamino C1-C6, aIquenilo C2-C6, alqueniloxi C2-C6, alquiniloxi C3-C6- o -cicIoaIquilo C3-C6,cuyos grupos alifáticos o alicíclicos pueden a su vez estar parcial o completamente haIogenados o lIevar uno a tres grupos Rb:Rb es halógeno, ciano, nitro, hidroxi, mercapto, amino, carboxiIo, aminocarbonilo, aminotiocarbonilo, alquilo, haloaIquilo, alquenilo, alqueniloxi, alquiniloxi, alcoxi, haIógenoaIcoxi, alquiltio, alquilamino, dialquilamino, formilo, alquilcarbonilo, alquilsulfonilo, alquilsulfoxilo, aIcoxicarbonilo, alquilcarboniloxi, alquilaminocarbonilo, dialquilaminocarbonilo, alquilaminotiocarbonilo, dialquilaminotiocarbonilo, cuyos grupos alquilo en estos radicales pueden contener 1 a 6 átomos de carbono y cuyos grupos alquenilo o alquinilo mencionados en estos radicales pueden contener 2 a 8 átomos de carbono;R4 es hidrógeno o alquilo C1-C2,R3 y R4 también pueden formar junto con el átomo de nitrógeno al que están ligados un anillo no saturados de cinco o seis miembros, qua puede llevar uno o varios sustituyentes Ra.
Patent CO-6220938-A2 (CO)
Title: Ligandos de receptor vainilloide novedosos y el uso de los mismos para la produccion de farmacos
Inventor: FRANK ROBERT
IPC: A61K31/44
Filed: 2009-10-16
Abstract: 1.- Compuesto sustituido de la fórmula general I.en la cual n es 0, 1, 2, 3, ó 4, R1 es H; F; Cl; Br; I; -SF5; -NO2; -CN; -NH2; -OH; -SH; -C(=O)-NH2; -S(=O)2-NH2; -C(=O)-NH-OH; -C(=O)-OH; -C(=O)-H; -S(=O)2-OH; -C(=NH)-NH2; -C(=NH)-NH-R9; -N=C(NH2)2; -N=C(NHR10)- (NHR11); -O-P(=O)2-O-R12; -NHR13; -NR14R15; -NH-C(= O)-R13; -OR16; -SR17; -C(= O)-NHR18; -C (= O)-NR19R20; -S(= O)2-NHR21; -S(= O)2-NR22R23 -C(= O) -OR24; -C(= O)- -R25; -S(= O)-R26; o -S(=O)2-R27 o un radical de C1-10 alifático no sustituido o al menos monosustituido, lineal o ramificado, saturado o insaturado, R2 es H; F; Cl; Br; I; -SF5; -NO2; -CN; -NH2; -OH; -SH; -C(= O)-NH2; -S(= O)2-NH2; -C(= O)-NH-OH; -C(= O)-OH; -C(= O)-H; -S(= O)2-OH; -C(= NH)-NH2; -C(= NH)-NH-R9; -N= C(NH2)2; -N=C(NHR10)-(NHR11); -O-P(=O)2-O-R12; -NHR13; -NR14R15; -NH-C(=O)-R13; -OR16, -SR17; -C(= O)-NHR18; -C(= O)-NR19R20; -S(= O)2-NHR21; -S(= O)2-NR22R23; -C(= O)-OR24; -C(= O)-R25; -S(= O)-R26; o -S(= O)2-R27 o un radical de C1-10 alifático no sustituido o al menos monosustituido, lineal o ramificado, saturado o insaturado, R3 es H; F; Cl; Br; I; -SF5; -NO2; -CN; -NH2; -OH; -SH; -C(= O)-NH2; -S(= O)2-NH2; -C(= O)-NH-OH; -C(= O)-OH; -C(= O)-H; -S(= O)2-OH; -C(= NH)-NH2; -C(= NH)-NH-R9; -N= C(NH2)2; -N=C(NHR10) - (NHR11); -O-P (= O)2-O-R12; -NHR13; -NR14R15; -NH-C (= O) -R13; -OR16; -SR17; -C(= O) -NHR18; -C (= O) -NR19R20; -S(= O)2-NHR21; -S (= O)2-NR22R23; -C(= O) -OR24; -C(= O)-R25; -S(= O)-R26; o -S(= O)2-R27 o un radical de C1-10 alifático no sustituido o al menos monosustituido, lineal o ramificado, saturado o insaturado, R4 es H; F; Cl; Br; I; -SF5; -NO2; -CN; -NH2; -OH; -SH; -C(= O)-NH2 ; -S(= O)2-NH2; -C(= O)-NH-OH; -C(= O)-OH; -C(= O)-H; -S(= O)2-OH; -C(= NH)-NH2; -C(= NH)-NH-R9; -N= C(NH2)2; -N=C(NHR10) - (NHR11); -O-P(= O)2-O-R12; -NHR13; -NR14R15; -NH-C(= O) -R13; -OR16; -SR17; -C(= O)-NHR18; -C(= O)-NR19R20; -S (= O)2 -NHR21; -S(= O)2 -NR22R23; -C(= O) -OR24; -C (= O) -R25; -S(= O) -R26, o -S(= O)2-R27 o un radical de C1-10 alifático no sustituido ...
Patent CO-6341640-A2 (CO)
Title: \\\"tratamiento de enfermedad autoinmunitaria e inflamatoria\\\"
Inventor: LEUNG STEWART
IPC: C07K16/28
Filed: 2011-02-11
Abstract: La presente invención proporciona nuevos procedimientos de tratamiento de la esclerosis múltiple y otras enfermedades auto inmunitarias o trastornos inflamatorios, y antagonistas, que incluyen proteínas de unión aisladas para su uso en los nuevos procedimientos. Se proporciona un procedimiento de tratamiento de la esclerosis múltiple que comprende la neutralización de la actividad biológica de la IL-7 mediante la unión a CD127 o a lL-7. Las proteínas de unión aisladas también pueden neutralizar la actividad biológica de la TSLP.
Patent CO-6450611-A2 (CO)
Title: Uso de delta-tocoferil-carbohidrato como agente despigmentante
Inventor: POIGNY STEPHANE
IPC: A61K8/34
Filed: 2011-10-31
Abstract: La presente invención divulga preparaciones cosméticas y dermatológicas para el tratamiento de cambios cosméticos o dermatológicos de la piel. Las composiciones se caracterizan por contener un vehículo dermocosméticamente aceptable y delta-tocoferil-carbohidrato. Las composiciones reivindicadas resultan particularmente útiles para tratar afecciones referentes a hiperpigmentación, en una forma localizada tal como por ejemplo lunares o pecas, o en una forma más generalizada, tales como para grandes áreas de la piel.
Patent CO-6480926-A2 (CO)
Title: Comprimidos de ibuprofeno de sodio y procedimientos de fabricación de composiciones farmaceúticas que incluyen ibuprofeno de sodio
Inventor: SEYER JEFFREY J
IPC: A61K9/20
Filed: 2011-12-22
Abstract: Se describen composiciones de ibuprofeno de sodio y procedimientos de fabricación de comprimidos y comprimidos oblongos que comprenden ibuprofeno de sodio. La formulación es ventajosa porque permite la formación de comprimidos que tienen bajo contenido de sodio y proporciona además comprimidos que exhiben estabilidad física mejorada, alta dureza de comprimido y afta resistencia, unido a excelentes características de disolución y de biodisponibilidad. Las formulaciones y procesos son además ventajosos porque pueden producirse en grandes cantidades sin un número inaceptable de comprimidos defectuosos.
Patent CO-6612263-A2 (CO)
Title: Método y sistema para operar un motor de encendido por compresión con combustibles primarios que contienen alcohol
Inventor: DUWIG CHRISTOPHE
IPC: C10L1/02
Filed: 2012-09-26
Abstract: La presente solicitud de se refiere a un método para operar un motor de encendido por compresión con combustible que contiene éter obtenido mediante la conversión a bordo de un combustible primario que contiene alcohol, que comprende las siguientes etapas: (a) retirar el combustible primario que contiene alcohol de un tanque de combustible y presurizar el combustible primario a una presión final de inyección en el motor; (b) introducir el combustible primario, presurizado en un reactor de deshidratación catalítica; (c) en el reactor, deshidratar catalíticamente el combustible primario, presurizado al combustible que contiene éter mediante el contacto con un catalizador de deshidratación de alcohol; y (d) retirar el combustible que contiene éter del reactor e inyectar el combustible que contiene éter en el motor.Adicionalmente, la invención proporciona un sistema para la operación de un motor de encendido por compresión con combustible que contiene éter, que comprende un motor de encendido por compresión; un tanque de combustible adaptado para almacenar un combustible primario que contiene alcohol; una bomba de alta presión para presurizar el combustible primario; por lo menos un reactor de deshidratación adaptado para recibir el combustible primario, presurizado y que comprende dentro de una cubierta de presión común un intercambiador de calor, y un lecho de catalizador corriente abajo con un catalizador de deshidratación de alcohol; y por lo menos un tubo de conexión que une la salida del reactor de deshidratación con uno o más inyectores.
Patent EP-1026481-A2 (EP)
Inventor: KNEPPER MARKUS
IPC: G01F1/075
Filed: 2000-01-24
Abstract: The arrangement has a sub-housing (2) for connection to the pipeline (21), a meter mechanism housing (3) with a meter mechanism (4), a display element (6) if appropriate and a separate auxiliary housing (7) for a sampling module (8) combined to form a unit with the meter mechanism housing. The auxiliary housing for the sampling module can be inserted into a recess in the meter mechanism housing.
Patent EP-1038595-A2 (EP)
Inventor: CLAIRADIN XAVIER
IPC: G02B6/36
Filed: 2000-03-16
Abstract: A system is provided for cleaning the end (80a)
of a ferrule (80) of a fiber optic connector (74) mounted
on a backplane (86) of a chassis (88) adapted for receiving
a printed circuit board (90) having a mating connector
mateable with the fiber optic connector. A dummy circuit
board (98) is receivable by the chassis (88) to replace the
actual printed circuit board. A cleaner (14) is mounted on
the dummy circuit board (98) for cleaning the end (80a) of
the ferrule (80) of the fiber optic connector (74) when the
dummy circuit board (98) is received by the chassis (88).
Patent EP-1043110-A2 (EP)
Inventor: YAMAMOTO TAKAHIRO
IPC: H05K3/00
Filed: 2000-03-30
Abstract: A plurality of feedthrough holes are efficiently
formed on the present invention by splitting a laser beam
emitted from a laser source (1) into plural laser beams (2)
by allowing the beam to pass through a diffraction grating
(3), followed by simultaneously forming a plurality of the
feedthrough holes on the ceramic green sheet (10) by
irradiating the ceramic green sheet (10) with the split
laser beam.
Patent EP-1050420-A2 (EP)
Inventor: HERPEL THOMAS DR
IPC: B60H1/00
Filed: 2000-04-06
Abstract: Die Erfindung betrifft ein Verfahren zur Regelung der Verdampfertemperatur einer Fahrzeugklimaanlage mit einem Verdampfer, einem Kompressor, einem Kondensator und einem Expansionsorgan, bei dem die Verdampfertemperatur in Abhängigkeit von Betriebsbedingungen eingestellt wird. Eine Verdampfertemperaturregelung im Zusammenhang mit einer Verbrauchs- und einer Komfortoptimierung zu erreichen, wird dadurch gelöst, daß ein erster Verdampfertemperaturwert (TV_F)bezüglich einer gewünschten Luftfeuchte kontinuierlich ermittelt wird, daß ein zweiter Verdampfertemperaturwert (TV_P) zur Sicherstellung einer ausreichenden Kühlleistung kontinuierlich ermittelt wird und daß als einzustellende Verdampfertemperatur (TV) der Kleinste der beiden Temperaturwerten ausgewählt wird. <IMAGE>
Patent EP-1081325-A2 (EP)
Inventor: GUHL JAMES C
IPC: E06B3/30
Filed: 2000-06-14
Abstract: A method for assembling a window is described including forming a lineal member
having a cross-sectional profile, where the profile includes a sash portion and a
frame portion, cutting the lineal member into lengths sized for forming the window,
and joining the lengths of the lineal member to form a shape of the window. The
sash portions form a sash and the frame portions form a frame. Then the sash is
separated from the frame.
Patent EP-1077444-A2 (EP)
Inventor: BLALOCK TRAVIS N
IPC: H05B44/00
Filed: 2000-06-28
Abstract: An on-chip system and method for calibrating an illumination
source (12a) includes a photo-detector (11a) and intensity sense and
control circuitry (50) resident on an integrated circuit (14). The integrated
circuit (14) is illuminated by an illumination source (12a), which impinges
upon the photo-detector (11a). The intensity sense and control circuitry
(50) receives the measured intensity value of the illumination source (12a)
and compares the measured intensity to a predetermined value (68)
representing the desired intensity. Subject to a range of operation (69),
the intensity sense and control circuitry (50) adjusts the intensity of the
illumination source (12a) based upon the difference between the measured
illumination intensity and the desired illumination intensity.
Patent EP-1086716-A2 (EP)
Inventor: JALDE FREDRIK
IPC: A61M16/20
Filed: 2000-08-01
Abstract: A feedback controller (1) for regulating respiratory gas in a
mechanical breathing aid system (2,3,4) comprises comparator
means (9) for periodically generating in a current breathing
cycle an error signal (10) representing the difference
between a value (7) of a gas parameter measured for gas
within the system and a target value (8) of the gas
parameter; and a control signal generator (11) for processing
the error signal (10) in accordance with a control function
to generate a control signal (12) usable in the regulation of
the respiratory gas and having a variable value integral gain
means (20) providing an input to an integrator element 21.
Adaption means (19) is arranged to determine for the current
breathing cycle an extreme value of the periodically
generated error signal (10) and to vary the value of the
integral gain used in the gain means (20) for a next
breathing cycle dependent on a rate of change of the value of
the extreme error signal with value of the integral gain.
Patent EP-1160440-A2 (EP)
Inventor: DOUYAMA YOSHIAKI
IPC: F02M17/40
Filed: 2000-11-06
Abstract: A carburetor body including a cylindrical bore, a frusto-conical
stepped shoulder portion, a valve chamber and an outlet passage which are
coaxially provided and sequentially reduced in the inner diameter inwardly from
an end wall face thereof. A plastic retainer and a metal collar are interference
fitted into the cylindrical bore. The fuel regulating needle valve includes a screw
shaft portion, an unthreaded stem portion and a valve tip which are sequentially
reduced in the outer diameter from a head of the fuel regulating needle valve
toward the valve tip. The threaded shaft portion is screwed into a threaded bore
formed in the metal collar, and at the same time, screwed into an axial bore formed
in the plastic retainer while cutting thread grooves. The unthreaded stem portion
projects from a distal end cylindrical portion of the plastic retainer into the valve
chamber, and the valve tip projects from the valve chamber into the outlet passage.
Patent EP-1108938-A2 (EP)
Inventor: SAUSNER ANDREAS
IPC: F16L13/16
Filed: 2000-11-20
Abstract: The invention proposes a connection between tubing (2) and hose (16) which can be easily and inexpensively produced, requires little installation space and results in favorable hydraulic properties. The connection is realized by means of a connecting piece (8) that is integrally formed onto the tubing (2). <IMAGE>
Patent EP-1126179-A2 (EP)
Inventor: SAPUTO RICHARD A
IPC: F04D17/16
Filed: 2000-07-10
Abstract: An electric air pump having multiple impellers parallel
mounted on the same motor shaft and typically employed for
providing a source of low pressure, high volume air for
charging inflatable devices. The multiple impellers provide
improved motor efficiency in heat dissipation and air volume
delivery when compared to a single impeller motor operating at
the same RPM, and exhibits a near zero True Indicator Reading
(TIR). In its most fundamental embodiment, the electric air
pump having multiple impellers exhibits a construction
including an outer housing having an air intake port and an air
exhaust port. An electric motor is mounted within the outer
housing and includes a rotating output shaft. A plurality of
air impellers each parallel mounted on the rotating output
shaft is employed for drawing a volume of air through the air
intake port and across the electric motor. An air compressor
chamber is positioned between the electric motor and the air
impellers for collecting the air while the air impellers
compress and exhaust the air through the air exhaust port for
providing a supply of pressurized air.
Patent EP-1024014-A2 (EP)
Inventor: FORD THOMAS DAVID REID
IPC: B41J11/00
Filed: 2000-01-28
Abstract: An ink jet printer mechanism is disclosed in which a print
receiving medium is supported in a clamp (18) in a
printing station (16) and a print head (41) is traversed
through the printing station. A service station (23) for
the print head is provided adjacent the printing station
and the print head is traversed to the service station
between printing operations. The service station includes
a carriage (25) which is movable by a drive motor (28) to
bring capping and wiping elements (30, 29) into engagement
with the print head. A mechanical linkage (33) from the
carriage opens the clamp when the capping element is
aligned for engagement with the print head.
Patent EP-1087348-A2 (EP)
Inventor: NICKERSON JOHN M
IPC: G07F19/00
Filed: 2000-03-15
Abstract: A method and machine for preparing and dispensing documents
relating to financial transactions. The machine contains an ink jet printer for
printing the documents and a bar code reader mounted for movement with the
print head of the printer for reading bar codes on each document before or
during printing. The machine includes a control unit having personal computer
architecture including a CPU, memories and input/output devices. One of the
devices is a modem allowing communication with a remote supervisory
location. Operation of the machine is controlled from the remote supervisory
location, which provides periodic authorization to continue to prepare and
dispense documents in response to transaction reports transmitted from the
machine to the remote supervisory location. A wide variety of documents can
be prepared and dispensed under control of software in the control unit.
Patent EP-1039600-A2 (EP)
Inventor: GOTO TAKENORI
IPC: H01S5/223
Filed: 2000-03-22
Abstract: An n-contact layer, an n-cladding layer, an MQW active
layer, and a p-first cladding layer are formed in this order
on a sapphire substrate. An n-current blocking layer having
a striped opening is formed on the p-first cladding layer.
The width of the striped opening gradually increases from W2
to W1 as the depth thereof decreases from a lower layer to
an upper layer in the current blocking layer. A p-second
cladding layer is formed on the n-current blocking layer and
on the p-first cladding layer inside the striped opening. The
p-second cladding layer comprises a lower layer having the
width W2 at its lower end and an upper layer having a width
W1 lager than the width W2. Embodiments comprise nitride based
semiconductors such as GaN.
Patent EP-1107068-A2 (EP)
Inventor: LOOPSTRA ERIK ROELOF
IPC: G03F7/20
Filed: 2000-11-22
Abstract: In a lithographic projection apparatus the positions and/or orientations of
reflective optical elements is dynamically controlled. The position of a reflective optical
element such as a mirror in an illumination or projection system is first measured using an
absolute position sensor mounted on a reference frame and thereafter measured by a
relative position sensor also mounted on said reference frame. The position of the element
is controlled in accordance with the measured position, e.g. to maintain it stationary in
spite of vibrations that might otherwise disturb it. The absolute sensor may be a capacitive
or inductive sensor and the relative sensor may be an interferometer.
Patent EP-1101695-A2 (EP)
Inventor: EUGSTER URS
IPC: B63C9/04
Filed: 2000-11-02
Abstract: The inflatable raft or boat has a bearing base body formed from at least two banana shaped buoyant bodies, so that the base body has an easily maneuverable boat or canoe shape. The buoyant bodies consist of two wall elements (14, 15) of waterproofed fabric, joined to each other by an airtight weld along a peripheral seam (11).
Patent EP-1277050-A2 (EP)
Inventor: GIBSON BRADFORD W
IPC: G16B15/20
Filed: 2000-05-26
Abstract: La présente invention concerne un procédé rapide et efficace qui permet de déterminer la conformation tridimensionnelle d'une protéine. Le procédé selon l'invention comprend les étapes suivantes: 1) on établit des limites de distance physique, par exemple en formant des réticulations chimiques intramoléculaires d'une taille connue entre des restes d'une protéine; 2) on enrichit le nombre de molécules ayant des réticulations chimiques intramoléculaires dans le groupe de réaction, par exemple au moyen d'une séparation fondée sur la taille pour éliminer les protéines ayant des liaisons intermoléculaires; 3) on expose le groupe de réaction enrichi à une protéase qui coupe la protéine au niveau de sites spécifiques pour produire des fragments peptidiques; 4) on mesure la taille des fragments peptidiques pour déterminer les sites de liaison ayant une certaine relation spatiale dans la protéine; et 5) on interprète les données produites pour déterminer le géométrie spatiale et la structure de la protéine sur la base de la relation spatiale déduite des sites de liaison. Ces information sont de préférence analysées à l'aide d'un système informatique, qui peut être utilisé pour générer et/ou analyser des limites de distance entre des acides aminés.
Patent EP-1328882-A2 (EP)
Inventor: OZZIE RAYMOND E
IPC: H04L12/18
Filed: 2000-06-28
Abstract: A communications manager provides communication services for an activity-based collaboration system, in which data change requests comprising deltas are communicated over a network between network-capable devices. The communications manager is operable on a local network capable device for sending locally-generated deltas over the network to at least one remote network-capable device and for receiving remotely-generated deltas over the network from the at least one remote network-capable device. The communications manager can send the deltas via unicasting, multicasting, or broadcasting techniques. The communications manager is responsive to network connection status information indicating that the remote network-capable device is connected to the network for sending the local deltas directly to an address for the remote network-capable device. A presence mechanism maintains and distributes, on request, the network connection status information, which it acquires from each of the network-capable devices. The communications manager is also responsive to the network connection status information indicating that the remote network-capable device is disconnected from the network for sending the local deltas to an address of a relay. The relay stores deltas until the relay is notified that the remote network-capable device has reconnected to the network, and then the relay sends the deltas to the reconnected remote network-capable device.
Patent EP-1192660-A2 (EP)
Inventor: FINK LUTZ
IPC: H01J31/49
Filed: 2000-06-13
Abstract: A semiconductor sensor for direct detection of electrons has a pixel structure in which a capacitance is designed to each pixel that stores a charge and converts the charge into a readable voltage. A conductive layer substantially covers the pixel structure. The conductive layer includes pixel surface coatings, each of which cover an individual pixel. Each pixel surface coating is separated from each adjoining pixel surface coating by a gap. A second conductive layer covers a surface of the gap. An insulation insulates the pixel surface coating from the second conductive layer. The conductive layers may be metal or other conductive, light impervious materials. The second conductive layer may include a capacitor electrode.
Patent EP-1222285-A2 (EP)
Inventor: PRITCHARD DAVID IDRIS
IPC: A61K38/00
Filed: 2000-10-20
Abstract: An isolated protein, for use in treatment of wounds, is characterized in that it is secreted by the organism Lucilia sericata and it exhibits proteolytic activity against FITC-casein at a pH of 8.0 to 8.5. The protein exhibits proteolytic activity against Tosyl-Gly-Pro-Arg-AMC but not against Suc-Ala-Ala-Phe-AMC, and its proteolytic activity against FITC-casein and Tosyl-Gly-Pro-Arg-AMC is inhibited by the serine proteinase inhibitors PMSF and AMPSF. The protein is also bound by immobilized aminobenzamidine.