baber/WOPTO huggingface dataset:
Patent PT-731100-E (PT)
Inventor: BRYANT HENRY UHLMAN
IPC: C07D409/00
Filed: 1996-03-06
Abstract: The present invention provides a compound of formula I <CHEM> wherein R1 is H, OH, halo, OCO(C1-C6 alkyl), OCO(aryl), OSO2(C4-C6 alkyl), OCOO(C1-C6 alkyl), OCOO(aryl), OCONH(C1-C6 alkyl), or OCON(C1-C6 alkyl)2;     R2 is aryl, C1-C6 alkyl, C3-C6 cycloalkyl, or 4-cyclohexanol;     R3 is O(CH2)2 or O(CH2)3; R4 and R5 are optionally CO(CH2)2CH3, CO(CH2)3CH3, C1-C6 alkyl, or R4 and R5 combine to form, with the nitrogen to which they are attached, piperidine, morpholine, pyrrolidine, 3-methylpyrrolidine, 3,3-dimethylpyrrolidine, 3,4-dimethylpyrrolidine, azepine, or pipecoline;     R6 is  &rdurule&  C=CH2 , &rdurule& CH(C1-C5 alkyl),  &rdurule& CH(C2-C5 alkenyl),  &rdurule& C=CH(C1-C5 alkyl), &rdurule& CH(aryl),  &rdurule& C(OH)(C1-C5 alkyl),  &rdurule& C(OH) (C2-C5 alkenyl),  &rdurule& C(OH)aryl;  and pharmaceutically acceptable salts thereof. The present invention further provides pharmaceutical compositions containing compounds of formula I, optionally containing estrogen or progestin, and the use of such compounds alone, or in combination with estrogen or progestin, for alleviating the symptoms of post-menopausal syndrome, particularly osteoporosis, cardiovascular related pathological conditions, and estrogen-dependent cancer. As used herein, the term "progestin" includes compounds having progestational activity such as, for example, progesterone, norethylnodrel, nongestrel, megestrol acetate, norethindrone, and the like. The compounds of the present invention also are useful for inhibiting uterine fibroid disease and endometriosis in women and aortal smooth muscle cell proliferation, particularly restenosis, in humans.
Patent PT-755198-E (PT)
Inventor: MANDERFELD MICHELLE MROZIK
IPC: A23L15/00
Filed: 1996-01-23
Abstract: Prodn. of a simulated egg patty comprises: (1) forming a predetermined amt. of egg yolk into a predetermined shape; (2) freezing the shaped egg yolk at < 20 deg.F for sufficient time to provide a frozen shaped egg yolk which is gel-like and retains its shape on thawing; (3) combining the frozen shaped egg yolk with a predetermined amt. of egg white; and (4) cooking the combined egg yolk and white to obtain a simulated egg patty; where the cooked egg yolk has similar mouthfeel and texture to cooked fresh egg yolk. Also claimed is a method as above which additionally comprises steps (1a) cooling the shaped egg yolk to 0-25deg.F for  5 min., and (3a) tempering the frozen shaped yolk at 0-25 deg.F for  5 min. The simulated egg patty is claimed per se. Also claimed is a simulated egg yolk, prepd. as above without addn. of egg white, and which opt. has its cholesterol level reduced prior to being formed in to a patty.
Patent PT-774962-E (PT)
Inventor: STORDY BARBARA JACQUELINE
IPC: A61K31/20
Filed: 1996-05-24
Abstract: PCT No. PCT/GB96/01256 Sec. 371 Date Feb. 28, 1997 Sec. 102(e) Date Feb. 28, 1997 PCT Filed May 24, 1996 PCT Pub. No. WO96/37200 PCT Pub. Date Nov. 28, 1996Dyslexia or inadequate night vision is treated by administering effective amounts of docosohexaenoic acid optionally in association wit other n-3 essential fatty acids and n-6 essential fatty acids.
Patent PT-839041-E (PT)
Inventor: BROQUET COLETTE
IPC: C07C257/14
Filed: 1996-07-15
Abstract: PCT No. PCT/FR96/01095 Sec. 371 Date Jan. 6, 1998 Sec. 102(e) Date Jan. 6, 1998 PCT Filed Jul. 15, 1996 PCT Pub. No. WO97/03678 PCT Pub. Date Feb. 6, 1997Cyclo-oxygenase inhibitor and amidine derivative salts, preparation methods therefor, pharmaceutical compositions containing said salts and the use thereof particularly as NO synthase and cyclo-oxygenase inhibitors, are disclosed.
Patent PT-843327-E (PT)
Inventor: PRICE RICK A
IPC: H01G4/18
Filed: 1997-11-11
Abstract: A capacitor (10) is made from a laminated structure having multiple layers of metallized, dielectric film (14) and having a solderable, metal termination (30) at each of two ends. The metal termination (30) at each of the ends is generally rectangular with a top edge (34), a bottom edge (36), and two side edges (38) and is finished so as to have a finished surface (42), which is characterized by a three-dimensional pattern of ridges (44) having solderable surfaces and grooves (46) having solderable surfaces. The ridges (44) alternate with the grooves (46) and the ridges (44) and the grooves (46) at both of the ends are parallel to the side edges (38). The three-dimensional pattern (42) facilitates reflow soldering of the capacitor (10). <IMAGE>
Patent PT-959822-E (PT)
Inventor: DELINCE PHILIPPE
IPC: A61F2/30
Filed: 1997-01-15
Abstract: A set of humeral head prostheses including a spherical head (1) and a peg (4) insertable and lockable in a matching recess (10) in the shank (7) of a humeral prosthesis designed to be sealed inside the upper portion of the humerus. All of the prostheses in one set have spherical heads (1) with the same radius of curvature but different maximum diameters.
Patent PT-944579-E (PT)
Inventor: GOSTELI JACQUES
IPC: A61K8/41
Filed: 1997-11-17
Abstract: Amine hydrofluorides of the general formula (I):In which R is a straight-chain hydrocarbon residue having 10 to 20 carbon atoms exhibit antibacterial and caries-prophylactic activity and can be prepared in high purity. The amine hydrofluorides of the formula (I) can be formulated, optionally in combination with tin fluoride, into oral hygiene compositions such as toothpastes, mouthwashes or chewable tablets.
Patent PT-935572-E (PT)
Inventor: GUIFFANT ALAIN
IPC: B65G17/40
Filed: 1997-11-04
Abstract: PCT No. PCT/FR97/01968 Sec. 371 Date Jul. 12, 1999 Sec. 102(e) Date Jul. 12, 1999 PCT Filed Nov. 4, 1997 PCT Pub. No. WO98/19942 PCT Pub. Date May 14, 1998The invention concerns a device for transferring bodies (9) supported by plates (Ai, Bi) followed in succession in a mobile curved line; the plates are grouped in successive pairs (Ai, Bi) joined by a horizontal shaft (13) enabling their mutual rotation; the adjacent plates of two successive pairs (Bi-1, Ai; Bi, Ai+1) are coupled and articulated about at least one vertical rotation axis (2); further the horizontal shaft (13) is preferably arranged such that there is a clearance between the plates (Ai, Bi) so that they can slope with respect to each other perpendicularly to said horizontal and vertical axes.
Patent PT-837910-E (PT)
Inventor: PLANCHE JEAN-PASCAL
IPC: C08K3/00
Filed: 1997-05-06
Abstract: PCT No. PCT/FR97/00812 Sec. 371 Date Apr. 20, 1998 Sec. 102(e) Date Apr. 20, 1998 PCT Filed May 6, 1997 PCT Pub. No. WO97/43342 PCT Pub. Date Nov. 20, 1997Bitumen/polymer compositions are produced by contacting, between 100 DEG  C. and 230 DEG  C., under agitation, one bitumen or a mixture of bitumens with at least one olefinic polymer bearing epoxy or COOH groupings, then by incorporating in the product, an acid additive while the whole mixture is agitated at a range between 100 DEG  C. and 230 DEG  C. for at least 10 minutes. The product, which is subjected to treatment by the acid additive may still contain one or several additional polymers, for instance of the elastomer type cross-linkable with sulphur, and even be subjected to sulphur cross-linking before treatment. The bitumen/polymer compositions are useful directly or after dilution, to form binders for carrying out surfacing operations.
Patent PT-925163-E (PT)
Inventor: PROSL JOHANNA
IPC: B23B51/10
Filed: 1997-09-03
Abstract: The invention concerns a device for deburring workpieces, in particular moulded parts and castings made of plastics, rubber or the like, said device comprising a rotatable shank (1) and linear tool elements (5, 6) which, in the axial direction, extend coaxially to the shank axis, are secured relative to the shank (1) and, as the latter rotates, can bulge out radially under the effect of centrifugal force. The device is designed such that an upper and a lower carrier (2, 3) are secured on the shank (1). The tool elements (5, 6) consist of individual threads or thread bundles whose ends are secured in the upper and lower carriers, a spring arrangement (7) being disposed concentrically with the shank (1) between the upper and lower carriers (2, 3).
Patent PT-917831-E (PT)
Inventor: DEEVI SEETHARAMA C
IPC: A24F40/46
Filed: 1993-09-10
Abstract: A removable cigarette (224') is manufactured for use in a smoking system which includes a lighter which has electrical heating means disposed in permanent cavity for delivering a flavored tobacco response to a smoker. To manufacture the cigarette a carrier web (259') is provided which has regions (261) of tobacco flavor material. Adhesive regions (261A) are applied from an adhesive applying station (327) to the surface of the carrier web (259') to form spaced regions of adhesive (261A) in between spaced regions of flavor material (261). A filter station (329) attaches filters (333,335) to the adhesive regions (261A) and a wrapping station (337) wraps the web (259') around the filters (333,335) to form a continuous rod of alternating regions of filter and tobacco flavor material. Finally, individual removable cigarettes (224') are formed by severing the continuous rod at a severing station (339).
Patent PT-1002017-E (PT)
Inventor: FISCHER HARTMUT RUDOLF
IPC: C08K3/34
Filed: 1998-08-07
Abstract: The invention relates to a nanocomposite material on the basis of a clay having a layered structure and a cation exchange capacity of from 30 to 250 milliequivalents per 100 gram, a polymeric matrix and a block copolymer or a graft copolymer, which block copolymer or graft copolymer comprises one or more first structural units (A), which are compatible with the clay, and one or more second structural units (B), which are compatible with the polymeric matrix.
Patent PT-1027028-E (PT)
Inventor: NGUYEN LY-LAN
IPC: A61K8/98
Filed: 1998-10-06
Abstract: The invention concerns a method for the permanent setting of keratin fibres and in particular hair, characterised in that it consists in: applying on the keratin fibres a composition reducing keratin, with adhesive capacity less than 15 g and a viscosity ranging between 0 and 2500 mpa's at a laminar flow rate of 100 s<SUP>-1 </SUP>and setting them; after sufficient setting time for reducing keratin, applying an oxidising composition, without intermediate rinsing of the fibres; rinsing after sufficient time for fixing the set fibres and reduced fibres in permanent setting; rinsing with water.
Patent PT-1083791-E (PT)
Inventor: LANDHAM ROWENA ROSHANTHI
IPC: A01N25/10
Filed: 1999-05-17
Abstract: The invention provides processes for producing solid, water-soluble or water-dispersible compositions comprising non film-forming materials, such as water-soluble agrochemical electrolytes, supported by film-forming polymers. The water-soluble agrochemical electrolytes can be salts of glyphosate. The processes comprise (i) preparing film-forming aqueous media containing (a) film-forming polymers; (b) water-soluble materials which are non film-forming; (c) water-miscible solvents in which the film-forming polymers are soluble and, optionally, (d) solid fillers, and thereafter (ii) drying the film-forming aqueous media to form the solid compositions. The invention also provides compositions produced by these processes.
Patent SG-58191-G (SG)
Title: Synthesis of human virus antigens by yeast
IPC: C12N1/16
Filed: 1991-07-19
Abstract: The present invention relates to synthesis of HBsAg in yeast. Yeast expression vectors comprising a yeast promoter, ADHI, have been constructed. The region of the HBV genome coding for the S-protein, excluding a possible 163 amino acid presequence, has been transferred to the yeast expression vector. Using the described yeast vector, the successful synthesis of HBsAg by yeast has been achieved. The product is antigenic (reactive with anti-HBsAg), and a substantial portion is found associated with particles identical in electron microscopic appearance to those found in the serum of HBV-infected patients and in Alexander cells but having a smaller particle size diameter. The HBsAg synthesized by yeast has identical sedimentation behavior to purified, naturally-occurring HBsAg particles purified from Alexander cells as measured by sucrose gradient sedimentation. The present invention demonstrates synthesis and assembly of a higher ordered multi-component structure resulting from expression of a heterologous DNA coding segment in a microorganism.
Patent SG-23620-G (SG)
Title: Smoking article
Inventor: SENSABAUGH ANDREW JACKSON JR
IPC: A24D1/22
Filed: 1985-09-11
Abstract: The cigarette has a carbonaceous fuel element. A separate aerosol generator has a substrate bearing an aerosol forming material. The fuel element and substrate are arranged in a conductive relationship, so that the heat-stable substrate receives conductive heat transfer throughout the burning time of the fuel element. The fuel element is less than 30mm in length, with a density of at least 5 g/cc. An insulation material can surround part of the fuel element. The insulation is resilient and at least 15 mm thick. The cigarette also has a mouthpiece.
Patent IE-34907-L (IE)
Title: Catalyst preparation.
IPC: C07D303/04
Filed: 1971-01-20
Abstract: 1332526 Oxiranes SHELL INTERNATIONALE RESEARCH MAATSCHAPPIJ NV 19 April 1971 [22 Jan 1970] 20081/71 Addition to 1249079 Heading C2C Oxiranes are produced by the oxidation of olefinic compounds with organic hydroperoxides in the presence of a catalyst comprising titanium in combination with an inorganic siliceous solid. The catalysts are those prepared by impregnating the siliceous solid with a substantially non- aqueous solution of a titanium compound in a non-basic, inert, oxygen-substituted hydrocarbon as solvent, removing solvent and calcining the impregnated solid. The catalysts may be promoted with compounds of magnesium or alkali metals. Examples describe the preparation of propylene and 1-octene oxides.
[GB1332526A]
Patent IE-870240-L (IE)
Title: Benzhydrylsulphinylacetamide
IPC: C07C317/44
Filed: 1987-01-30
Abstract: 1. Claims for the Contracting States : BE, CH, DE, FR, GB, IT, LI, LU, NL, SE (-)-Benzhydrylsulfinylacetamide. 1. Claims for the Contracting States : AT, ES, GR A method for the preparation of (-)-benzhydrylsulfinylacetamide, which comprises : 1) reacting (+-)-benzhydrylsulfinylacetic acid with (-)-alpha-methylbenzylamine to give the (-)-benzhydrylsulfinylacetate of (-)-alpha-methylbenzylamine, 2) converting the resulting (-)-benzhydrylsulfinylacetate salt of (-)-alpha-methylbenzylamine to (-)-benzhydrylsulfinylacetic acid by acid hydrolysis, and 3) subjecting the resulting (-)-benzhydrylsulfinylacetic acid to an amidation reaction with NH3 .
[EP0233106B1]
Patent IE-42477-L (IE)
Title: Polyamide compositions with improved heat stability
IPC: C08K3/16
Filed: 1976-02-12
Abstract: 1469396 Heat-stabilized polyamides RHONEPOULENC INDUSTRIES 12 Feb 1976 [14 Feb 1975] 05604/76 Heading C3R Polyamides are heat stabilized by incorporating therein (a) 0À04 to 3% (by weight) of an alkali or alkaline earth metal halide, (b) 0À001 to 2% Cu as a complexed or non-complexed organic or inorganic salt and (c) 0À1 to 5% of a C 3-20 glycol with the OH groups in the alpha and gamma positions. The polyamide may also contain other conventional adjuvants such as fillers, lubricants, other stabilizers, plasticizers, pigments, dyes or crystallization agents, e.g. glass or asbestos fibres, glass microspheres, talc, silica and mica. Various polyamides and additives (a), (b) and (c) are mentioned; in specific examples the polyamide is nylon 66 and (a) is KI, (b) is copper stearate or cuprous oxide and (c) is 2,2-dimethyl-1,3-propanediol or 2-ethyl- 1,3-hexanediol. In the examples the glycol is melted, the copper salt and KI of particle size below 100 microns are added to the melt and stirred and the mass is cooled and ground to flakes of size less than 6 mm. which are then mixed and homogenized with the nylon. (From GB1469396 A) [FR2300782A1]
Patent IE-31864-L (IE)
Title: Percussive musical instrument
IPC: G10H1/055
Filed: 1968-04-05
Abstract: 1,164,422. Electronic musical instruments. PHILIPS ELECTRONIC & ASSOCIATED INDUSTRIES Ltd. 5 April, 1968 [8 April, 1967], No. 16538/68. Heading G5J. A circuit for imitating the touch of a percussive musical instrument is arranged so that the build-up time of the note from a tone generator G is made independent of the duration of actuation of the key T. The key is mechanically coupled to a magnet M which induces a voltage pulse in an inductance L on actuation of the key. This voltage pulse is used to charge up a capacitor C through a diode D, and is also fed to the base of a transistor Tr, causing it to conduct and so ground the base of transistor O which is thereby switched off and does not pass any signal from generator G. At the end of the pulse, transistor Tr is switched off and the voltage stored in capacitor C is fed through resistor R to the base of transistor O which is hence switched on and passes a signal from generator G to associate amplifying apparatus at a level depending on the voltage across the capacitor and hence the intensity of actuation of the key. Diode D 2 and capacitor C 2 prevent " bottoming " of transistor O if the key is depressed before the voltage across the capacitor C 1 has decayed to zero. Fig. 5 (not shown) illustrates a further embodiment in which the switching transistor Tr is arranged between the capacitor to be charged and the base of the transistor O and switches on after the capacitor has charged up to allow voltage from the capacitor to switch transistor O on.
[GB1164422A]
Patent IE-850696-L (IE)
Title: Manufacture of abrasive compact
IPC: B24D3/10
Filed: 1985-03-19
Abstract: Disclosed is an improved polycrystalline compact of self-bonded diamond particles having a network of interconnected empty pores dispersed throughout. The improved porous polycrystalline diamond compact possesses enhanced oxidation resistance and comprises all of the exterior surfaces of the porous compact being enveloped with a continuous coating which is effective under metal bond fabrication conditions so that oxidation of the diamond in the compact does not exceed a threshold level whereat loss of diamond properties of the compact occurs. Metal bond fabrication conditions comprehend an atmosphere containing oxygen or water vapor. Metal coatings are preferred, especially in coating thicknesses in excess of about 30 microns.
Patent IE-34373-L (IE)
Title: Formulations of tetramisole
IPC: A61K31/425
Filed: 1970-07-08
Abstract: Aqueous injectable solutions of tetramisole which comprise tetramisole citrate, tartrate, or phosphate equivalent to at least 6 percent w/v of L-tetramisole base, the pH of the solution being adjusted to the range of from 2 to 4 by addition of tartaric, citric or phosphoric acid.
[US3670086A]
Patent FI-812501-L (FI)
Inventor: FRANZ DIETMAR
IPC: H04L12/52
Filed: 1981-08-13
Abstract: A method is disclosed for establishing connections from subscriber stations or transmission lines connected to a data exchange system to signal converters. The data exchange system receives information concerning the free state or busy state of the signal converters. For this purpose, it is provided that, having forwarded the signals with which it has been previously supplied for signal conversion, the signal converter emits a special free signal which may differ from an accompanying signal indicating the end of signal transmission and which changes the busy state signal ("1") indicative of the busy state of the signal converter directly into a free state signal ("0").
Patent FI-813222-L (FI)
Inventor: FRIEDLI PAUL
IPC: B66B1/18
Filed: 1981-10-15
Abstract: An apparatus for controlling the access of a plurality of microprocessors at a data line. The microprocessors are connected by interface components or blocks, logic switching circuits and bus drivers with two lines or conductors. An access request or demand of a processor initiates a signal change at the first line. This signal change causes the transformation of data which is specific to the processor into a delay or a priority signal, upon the occurrence of which there is accomplished a signal change of the second line. As a function thereof there appears at an input of the interface component a signal change which is indicative of the availability of the data line. Upon simultaneous occurrence of access requests or demands of a number of processors the signal change of the second line is brought about by that processor whose priority signal possesses the smallest delay. The signal change of the second line prevents the occurrence of the priority signals possessing the greater time-delays and which are correlated to the remaining processors. At these processors there thus cannot occur any signal change at the input of the related interface component or block and which indicates the availability of the data line.
Patent IE-851396-L (IE)
Title: Biodegradable amphipathic copolymers
IPC: C08G63/66
Filed: 1985-06-04
Abstract: A pharmaceutically or veterinarily acceptable amphipathic, non-cross linked linear, branched or graft block copolymer, which has a minimum weight average molelcular-weight of 1000, in which the hydrophobic component is biodegradable or hydrolytically unstable under normal physiological conditions, and the hydrophilic component may or may not be biodegradable or hydrolytically unstable under such conditions, and which copolymer is self-dispersible in water; together with mixtures of such a copolymer and a drug, which may be water-soluble or water-insoluble, which mixtures are self-dispersible in water; and processes for the manufacture of such copolymers and such mixtures.
Patent IE-901434-L (IE)
Title: Heterocyclic diones as pesticides and plant growth¹regulators
IPC: A01N43/72
Filed: 1990-04-23
Abstract: Compounds of the general formula I   A - @ - B      I  wherein  A represents the group (i) <CHEM> in which any free hydrogen may be replaced by an agriculturally acceptable substituent; and B represents an optionally substituted aryl or heteroaryl group are disclosed, as well as methods of producing such compounds, intermediates therefore, and their use as herbicides and acaricides.
Patent IE-831459-L (IE)
Title: Method and device for energy recovery by manufacturing of¹asphalt in bulk
IPC: E01C19/05
Filed: 1983-06-21
Abstract: Method and device for manufacturing of asphalt bulk masses where a substantial part of the heat energy of the furnace gases from the drying and mixing process is transferred to the bulk mass fractions before those are supplied to the drying and mixing process and where the furnace gasses by this process at the same time are cleaned for pollutions. Bulk masses are directed downwards between two parallelly arranged inclined planes (1, 5) where the lower inclined plane (1) comprising horizontally arranged downwards directed ribs (2) directing the furnace gasses to the lower side of the bulk masses and where the second inclined plane (5) comprising vertically arranged ribs (4) suctioning the cleaned furnace gases up from the bulle masses after a substantial part of the heat energy being transferred to the bulk masses. At the lower and upper ends of the inclined planes accumulations of the bulk masses (7, 11) are maintained for preventing air from the atmosphere to penetrate into the system. The bulk mass fractions thereafter are transferred to the drying and mixing process, thereby having accumulated a substantial amount of heat energy and the bitumen components being transferred with the furnace gasses, as well as other pollutions.
[WO8400377A1]
Patent IE-831516-L (IE)
Title: Fluid jet printing apparatus
IPC: B41J2/145
Filed: 1983-06-29
Abstract: The individual elements of an elongated array of fluid jet orifices are independently positioned with respect to the individual elements of a second elongated array of individual charging electrodes thus relaxing critical mechanical manufacture and assembly tolerances therebetween. The number of fluid jet orifices is substantially greater than the number of independent charging electrodes so as to permit this independent positioning and the enhanced printing resolution of the apparatus is made possible primarily by the lesser density of individual electrodes in the electrode array.
[US4550323A]