baber/WOPTO huggingface dataset:
Patent EC-SP003471-A (EC)
Title: Inhibidor de metaloproteasa acido aromatico sulfohidroxamico
Inventor: FRESKOS JOHN
IPC: A61K31/00
Filed: 2000-05-12
Abstract: El presente invento está dirigido a un proceso de tratamiento que comprende la administración y observación de un inhibidor metaloproteasa sulfo ácido hidroxámico aromático en una eficiente cantidad a un mamífero anfitrión que tenga una condición asociada con una actividad patológica metaloproteasa.
Patent EC-SP003667-A (EC)
Title: Nuevos derivados de bencimidazolonas que tienen afinidad para receptores mezclados de serotonina y dopamina
Inventor: CEREDA ENZO
IPC: A61K31/496
Filed: 2000-09-20
Abstract: El presente invento se refiere a compuestos de la fórmula General I (gráfico) en la que R1, R2, R3 y R4 significan o hidroxi, con la condición de que R1, R2, R3 y R4 no pueden representar simultáneamente hidrógeno, a procedimientos para su preparación y a su uso como compuestos farmacéuticos.
Patent EC-SP972027-A (EC)
Title: Ducha electrica
Inventor: MARTINS GOMES JOAO CARLOS
Filed: 1997-02-18
Abstract: La presente patente de invención se refiere a "DUCHA ELECTRICA", o de manera más particular, a diferentes perfeccionamientos técnicos y funcionales que se lograron mediante arreglos mecánicos, eléctricos y estructurales, desarrollado especialmente con vistas a la caracterización de una ducha eléctrica compacta.
Patent EC-SP972291-A (EC)
Title: Derivados de cepalosporin piridinio (caso rn 4410/256)
Inventor: ANGEHRN PETER
IPC: A61K31/54
Filed: 1997-10-21
Abstract: Derivados de Cefalosporin piridino de la fórmula general I (gráfico), en donde R1 es hidrógeno, alquilo inferior, cicloalquilo o acetilo; X es CH o N; n es 0,1 o 2; m es 0 o 1; R2 es hidrógeno, alquilo inferior, w-hidroxi alquilo, bencilo o alquilo inferior-heterociclilo, estando el bencilo y el grupo heterociclilo insustutuido o sustituido por a lo menos uno de los grupos amino, ciano, carboxilo, hidroxilo, alquilo inferior, alcoxilo inferior o-CONR2, siendo R hidrógeno o alquilo inferior; o R2 es -CH2CON-R4R5; en donde R4, R5 son, independientemente hidrógeno, w-hidroxi-alquilo, fenilo, naftilo o heterocíclico, estando el fenilo, naftilo o heterociclilo insustituído o sustituído por a lo menos uno de los grupos de hidroxilo, opcionalmenteprotegido, halógeno, alquilo inferior opcionalmente sustituído, alcoxilo inferior opcionalmente sustituido, w-hidroxialquilo y/o ciano; o los grupos R4 y R5 forman conjuntamente un grupo de la fórmula (gráfico), con la salvedad de que m es 1, cuando el anillo de piridinio A es un piridinio-4-ilo; así como sus ésteres fácilmente hidrolizables, sales farmacéuticamente aceptables de dichos compuestos e hidratos de los compuestos de fórmula I y de sus ésteres y sales.
Patent EC-SP993257-A (EC)
Title: Antagonistas de receptores de il 8-iii
Inventor: PALOVICH MICHAEL ROBERT
IPC: A61K9/16
Filed: 1999-12-09
Abstract: Esta invención se refiere a nuevos compuestos de fórmula (I) a (VII) y sus composiciones, útiles en el tratamiento de estados de enfermedad que ocurren con medicación de la quimioquina, interleuquina-8(IL-8)
Patent EE-9800103-A (EE)
Inventor: GARRETT L SCOTT
IPC: C03B7/094
Filed: 1998-04-09
Abstract: Apparatus for forming a cased glass stream having an inner core of glass surrounded by an outer glass casing, includes (i) means for delivering core glass from a first source through a first orifice 22, (ii) means forming a second orifice 28 vertically below the first orifice with a chamber 30 surrounding the second orifice and communicating with the second orifice through a gap between the first and second orifices and (iii) means for delivering casing glass from a second source to the chamber such that glass flows by gravity through the orifices to form the cased glass stream. The first and second orifices are carried by an orifice housing assembly 44 with means for moving the assembly into seating engagement against the means for delivering core and casting glass so as to form an area seating engagement. The orifice housing assembly further includes a fluid manifold 50 mounted on the housing assembly and having inlet means for connection to a source of cooling fluid and outlet means 58 directed toward the area 59,60 of seating engagement between the assembly and the means for delivering core and casing glass for cooling the area and thereby reducing leakage of glass between the housing assembly and the means for delivering core and casing glass. Also claimed is an orifice housing assembly for an apparatus for forming a cased glass stream. Also claimed is a method of cooling the area of seating engagement between the orifice housing and the means for delivering streams of core and casing glass.
Patent FI-20000085-A (FI)
Inventor: DESAI MANOJ C
IPC: C07D205/085
Filed: 2000-01-17
Abstract: PCT No. PCT/US93/01429 Sec. 371 Date Nov. 7, 1994 Sec. 102(e) Date Nov. 7, 1994 PCT Filed Feb. 23, 1993 PCT Pub. No. WO93/23380 PCT Pub. Date Nov. 25, 1993.The invention relates to bridged aza-bicyclic derivatives of formula (I). These compounds are useful in the treatment of inflammatory and central nervous system disorders, as well as other disorders. Also disclosed are intermediates used in the synthesis of compound of formula (I).    <IMAGE>  (I)
Patent FI-20030397-A (FI)
Inventor: SALO KAJ
IPC: H04L12/26
Filed: 2003-03-17
Abstract: A method and arrangement in a telecommunications system comprising a data transmission path (8), the arrangement comprising devices (1, 21, 221 to 22n) and data being transmitted on the data transmission path between the devices in messages (4, 9) cyclically, whereby one or more of the devices (1, 221 to 22n) are arranged, during one or more first turns, respectively, to set the timing of their own cyclic traffic between cyclic traffic detected on the data transmission path; and one or more of the devices (1, 21, 221 to 22n) are arranged, during a second turn, to transmit a message not belonging to the cyclic traffic to the data transmission path on the basis of at least one determined occurrence time slot of the cyclic traffic such that the message does not collide with messages of the cyclic traffic which occur in the determined at least one occurrence time slot.
Patent FI-20061083-A (FI)
Inventor: HAKULINEN ILKKA
IPC: A47L9/14
Filed: 2006-12-07
Abstract: The invention relates to an arrangement for mounting a dust bag to a vacuum cleaner. The arrangement comprises a cylindrical mounting collar (1) mounted to the dust bag, and a cylindrical ring flange (2) supported on the vacuum cleaner and corresponding to the mounting collar, both having cylindrical mounting surfaces (3,4) that can be placed against each other for locking the mounting collar and the ring flange together so that one is within the other. In accordance with the invention, the cylindrical mounting surfaces (3,4) of the mounting collar (1) and the ring flange (2) are divided for their entire circumference into an even number of equally long surface portions, in which every other surface portion forms a locking zone (5,6) and the surface portions between the locking zones form a free zone (7,8). In this manner, when the locking zones are placed in alignment with each other, the mounting collar and the ring flange can be pressed against each other into a locked position, and when rotated from the locked position for the length of a surface portion, they become free from the locked position.
Patent FR-1193283-A (FR)
IPC: B29C65/64
Filed: 1958-03-14
Granted: 1959-11-02
Abstract: 872,852. Method of making elastic bushings. DAYCO CORPORATION. Feb. 21, 1958 [March 19, 1957], No. 5756/58. Class 108(3). A method of manufacturing resilient bushings comprises the steps of wrapping a sheet of natural or synthetic rubber 21 round an inner metal sleeve 11 to which an adhesive has been applied, curing this assembly 30 in a mould and then forcing it into an outer metal sleeve 32 or other similar aperture to form the bushing 36. The sheet of resilient material is preferably formed by cutting off lengths of rubber extruded as a flat or curved strip of a width equal to the outer circumference of the inner sleeve. The mould comprises corresponding upper and lower halves 22, 22a with openings 26, 26a in them for up to 60 assemblies 30. The surface 31 may be flat or of the opposite taper to form different shaped bushings. Details of the curing are also given.
Patent GB-1225584-A (GB)
IPC: A61K31/055
Filed: 1969-04-15
Abstract: 1,225,584. Antiviral compositions. VSESOJUZNY NAUCHNO-ISSLEDOVATELSKY KHIMIKO - FARMATSEVTICHESKY INSTITUT IMENI S. ORDZHONIKIDZE. 15 April, 1969 [18 April, 1968], No. 19109/69. Heading A5B Pharmaceutical compositions for combating virus infections comprise an ointment base and the compound 3,5,3',5'-tetrabromo-2,4,2',4'- tetrahydroxy diphenyl. Ointments are disclosed comprising 0.1, 0.25 and 1% by weight of the active compound in a soft paraffin/liquid paraffin base.
Patent GB-1227329-A (GB)
IPC: A23L27/10
Filed: 1969-08-06
Abstract: 1,227,329. Chocolate flavour extract. NESTLE'S PRODUCTS Ltd. 6 Aug., 1969 [19 Aug., 1968], No. 39295/69. Heading A2B. A water soluble chocolate extract is obtained by steam stripping aromatic constituents from a mixture of cocoa liquor, being the liquor obtained by grinding roasted and shelled cocoa beans and comprising cocoa butter and non-fat cocoa solids, and water, condensing the aromatic constituents, heating the stripped mixture to extract water-soluble constituents from the liquor, separating into a first residual sludge and a first aqueous phase containing the water-soluble constituents, and combining the aromatic constituents with the water-soluble constituents. The sludge may be mixed with further water and separated to recover more water-soluble constituents. The product may be dried to a solid.
Patent GB-1227400-A (GB)
IPC: C07C29/17
Filed: 1968-08-14
Abstract: 1,227,400. 3,7-DimethyI-7-octen-1-yn-3-ol- and 3,7-dimethyl-7-octadien-3-ol derivatives. BADISCHE ANILIN- & SODA-FABRIK A.G. l4Aug., 1968 [16 Aug., 1967], No. 38794/68. Heading C2C. [Also in Division A5] Derivatives of 3,7-dimethyl-7-octen-l-yn-3- ol and 3,7-dimethyl-7-octadien-3-ol of general formula wherein A denotes an ethenyl or an ethynyl group, R<SP>1</SP>, R<SP>2</SP>, R<SP>3</SP>, R<SP>4</SP>, R<SP>6</SP> and R6 independently denote a hydrogen atom or a methyl or ethyl group provided that at least one of R<SP>1</SP>, R<SP>3</SP> and R<SP>*</SP> denotes a methyl or ethyl group and R<SP>7</SP> denotes a hydrogen atom or the acyl radical of a monocarboxylic acid having 1-8 carbon atoms are prepared by subjecting a ketone of general formula to a conventional ethynylation or ethenylation or to a conventional ethynylation followed by partial hydrogenation, and, where R<SP>7</SP> denotes an acyl group, the carbinol obtained is acylated, the acylation and the partial hydrogenation being carried out in any sequence.
Patent GB-1227840-A (GB)
IPC: F23Q9/04
Filed: 1968-11-20
Abstract: 1,227,840. Igniting gas burners. JUNKERS & CO. G.m.b.H. 20 Nov., 1968 [25 Nov., 1967], No. 54957/68. Heading F4F. In a device for igniting and supervising gasheated appliances which comprises a burner, an igniter 13 and a thermocouple element 15 which is connected to a thermoelectric ignition safety device, the respective housings 11, 12, 14, whose axes are coplanar, for these elements form part of a one-piece carrying plate 10 having a flanged periphery 16 and at least two peripheral fixing members, while the ends of the curved tube 26 subtend an angle of 90 degrees at its centre of curvature and the outlet end 36 of this tube serves as an earth electrode for the igniter, the head 37 of the thermocouple element being arranged such that with the gas at its maximum pressure, only the point of the flame from the ignition tube strikes the head 37. As shown, the coplanar axes of the housings 11, 12, 14 are perpendicular to the plane of the carrying plate, and the outlet end of the ignition tube is surrounded by a combustion chamber 28 arranged so that edge 36 of the ignition tube is nearer to the igniter than is the corresponding edge of the combustion chamber.
Patent GB-1229369-A (GB)
IPC: A01D69/02
Filed: 1969-12-06
Abstract: 1,229,369. Lawn mowers. T. S. SIMPSON. 6 Dec., 1969, No. 63539/69. Heading A1F. A mower comprises a blade rotating in a housing 1 and driven by an electric drill supported in a drill stand 6 mounted on the housing. Height adjustment of the cutters is effected by adjustment of the drill in the stand.
Patent GB-1229801-A (GB)
IPC: H02G3/08
Filed: 1968-01-29
Abstract: 1,229,801. Mould patterns for junction boxes. BRITISH INSULATED CALLENDER'S CABLES Ltd. 28 Jan., 1969 [29 Jan., 1968], No. 4445/68. Heading B5A. [Also in Division H2] A junction box aperture is formed in a east concrete or plastics module by securing to the mould wall a two-part pattern comprising a base-plate 12 with cable and cover connection posts 18, 14, and a tapered frame 2 which has a post 6 push-fitting a nylon stud on the base 12 and slots 7 contacting the outside of posts 14 when the two parts are together. The bridge piece 3 of the frame 2 is secured to the mould wall by screws &c., the cables are laid in apertures 5 in the frame using grooved nylon sleeves 16, unused apertures being blanked off, and after pushing on the base-plate, the module is cast. Removal of the mould or shuttering withdraws the frame 2, leaving the plate 12 securely embedded in the concrete or plastics and forming the base of a junction box aperture. A cover-plate is secured by screws to the posts 14.
Patent GB-1232418-A (GB)
IPC: D21F1/48
Filed: 1968-04-11
Abstract: 1,232,418. Papermaking. WALMSLEYS (BURY) Ltd. 10 April, 1969 [11 April, 1968], No. 17459/68. Heading D2A. A foil box for a paper- or board-making machine comprises means for vibrating at least the foils independently of any movement of other parts of the machine. The vibration may be in the direction of, or transverse to the direction of papermaking, or a compound of these two motions. The inclination of the foils to the wire may be adjustable.
Patent GB-1233552-A (GB)
IPC: B65B9/02
Filed: 1967-07-11
Abstract: 1,233,552. Wrapping wallpaper rolls. REED INTERNATIONAL Ltd. 11 July, 1968 [11 July, 1967], No. 31790/67. Heading B8C. Wallpaper is wound into a roll at 1, drops at 1<SP>1</SP> on to a belt 3 along which it is pushed by a pusher 4 and down a ramp 5 into a loop 11 (at 1<SP>11</SP>) formed by two polythene webs 121 and 131 which are joined by heat-sealing at their leading edges and which are fed from reels 12 and 13 so that the roll 1<SP>11</SP> descends and the webs 12<SP>1</SP> and 13<SP>1</SP> may be sealed together (by means of a double line seal) above the roll 1<SP>11</SP> by a device 22 which cut off the wrapped roll (between the line seals) and thereby simultaneously forms a new loop 11. The webs 12<SP>1</SP> and 13<SP>1</SP> are fed from the reels 12 and 13 by rotating rollers 14 and 15 either by the winding device 2; or hydraulically or pneumatically. As the roll 1 is being wound, a member 24 is moved to the left in the Figure and acts by way of levers 25 and 27, rack 32, pinions 33 and 34, and a rack 23, on pinions on the ends of rollers 14 and 15, so that the diameter of the roll 1 determines the length of the loop. The pusher 4 is moved in direction 8, and the belt 3 in direction 9, to prevent unrolling of the roll 1<SP>1</SP>, by a common motor 21. A clamp 36 is moved by an hydraulic piston and cylinder 38 to move the webs to the electrically-heated sealing head 35 which comprises upper and lower dies. The wrapped roll drops (at 1<SP>1111</SP>) on to a conveyer which conveys it to a unit where the polythene is heat-shrunk on to the roll.
Patent GB-1238337-A (GB)
IPC: H01H33/14
Filed: 1968-08-30
Abstract: 1,238,337. Fluid blast switches. D. KIND. 30 Aug., 1968 [31 Aug., 1967], No. 41598/68. Heading H1N. An oil blast switch has a bridging contact 1 movable away from fixed contacts 3, 4 by a stream of oil flowing along the passage 5, the arcs developing between the bridging contact 1 and the fixed contacts 3, 4 being driven by the stream of oil into tubular outlet passages 8, 9 respectively. Arcing horns 10, 11 are attached to the fixed contacts 3, 4. Three series connected switches (Fig. 2, not shown) may be housed in a single insulating block 12. A modified form of contact 1 (Figs. 3a-3c, not shown) has a plurality of resilient fingers providing a plug and socket type connection with the fixed contacts and also a separate arcing contact region.
Patent GB-1239624-A (GB)
IPC: B25C1/04
Filed: 1969-05-14
Abstract: 1,239,624. Nailing machines. SPOTNAILS Inc. 14 May, 1969 [17 May, 1968], No. 24555/69. Heading B4C. A pneumatically actuated nailing machine comprises a piston 32 having at least one bore 39 and a valve 33 between annular chambers 19, 20, the chamber 19 receiving compressed air through a passage 18, and the chamber 20 through passages 21, 22 and a trigger valve 25, from an inlet chamber 16. The valve 33 is biased to its lowermost position, Fig. 3, by a spring 37, the chambers 19, 20 both containing compressed air. In this position a passage 34 in the valve 33<SP>1</SP> is open to the atmosphere through a passage 35, and the chamber 19 is shut off from the space above the piston 32. On raising the trigger valve 25, see Fig. 4 (not shown), the chamber 20 is shut off from the inlet chamber 16 and opened to the atmosphere at 27, thus allowing the air in the chamber 19 to raise the valve 33 so that the passage 34 abuts a seal 36 to close the passage 35. Further, the raising of the valve 33 allows the compressed air in the chamber 19 to force the piston 32 downwards causing the driving blade 38 to strike a nail 15. During the descent of the piston 32, compressed air flows through the bore(s) 39 and into an annular chamber 42 via an inlet 43. The trigger valve 25 is then released, allowing the chamber 20 to refill with compressed air to lower the valve 33, so that the space above the piston 32, which is resting on a collar 45, is open to the atmosphere through the passages 34, 35 and so that the chamber 19 is again sealed. Consequently the compressed air in the chamber 42 raises the piston 32 whilst air again leaks through the bore(s) 39 ensuring a gentle return of the piston. Air may be allowed to leak from between the housing and the rod 38 to remove excess compressed air from below the piston, and the chamber 42 may be of equal volume to the chamber 40 formed above the piston.
Patent GB-1250519-A (GB)
IPC: C07C59/86
Filed: 1969-05-16
Abstract: 1,250,519. Cycylodeca pentaene derivatives. SYNTEX CORP. 16 May, 1969 [3 July, 1968], No. 25102/69. Headings C2C and C2P. Novel compounds A, B, C and D in which R is H, 1-6C alkoxy or 1-8C acyloxy derived from a carboxylic acyl group; R‹ is H or 1-6C alkoxy; R<SP>1</SP> is H or 1-3C alkyl; R<SP>2</SP> is -CHO, -CH 2 R<SP>3</SP>, -COOR<SP>4</SP>, -CONH 2  or -CONHOH; R<SP>3</SP> is OH or a hydrolysable ester thereof or ether thereof; R<SP>4</SP> is H, 1-6C alkyl or alkali metal; and X is -CH 2 -, -CCl 2 - or -CF 2 - are prepared by numerous methods which are diagrammatically illustrated below wherein Ac is acyl, R<SP>5</SP> is an acid labile protecting group, x<SP>1</SP> is -CCl 2 - or -CF 2 -, Ac<SP>1</SP> is trimethylacetyl, and R<SP>11</SP> is lower alkoxy. The compounds II-XI, XVI-XXI, XXVIXXXIV and XLIII-XLVIII may all be isolated as intermediates and final products. Pharmaceutical compositions comprise a compound A, B, C or D together with a suitable carrier or diluent and may be administered orally as anti-inflammatory, analgesic and anti - pyretic agents.
Patent GB-1250772-A (GB)
IPC: B60J7/16
Filed: 1968-03-19
Abstract: 1,250,772. Convertible vehicles. DANBURY CONVERSIONS Ltd. 11 Oct., 1968 [19 March, 1968], No. 13368/68. Heading B7B. A vertically movable roof part 1 for a vehicle supports a flexible sleeve 2 which is held taut by inclined links 6, 7 hinged at 9 and held erect by sliding rings 10. The links may be resiliently telescopic.
Patent GB-1251112-A (GB)
IPC: H04Q9/14
Filed: 1969-06-30
Abstract: 1,251,112. Ripple control receivers. LANDIS & GYR. A.G. 30 June, 1969 [8 July, 1968], No. 32932/69. Heading H4R. [Also in Division G4] In a ripple control receiver Fig. 2 a readying pulse S, Fig. 1 of A.C. received over the line and detected by the tuned circuit 23 Fig. 2, comprising capacitor 24 and relay coil 25, causes contacts 34 to close for the pulse duration, supplying mains energizing current to a synchronous selector motor 27 which, when cam 28 moves off zero, self holds over contacts 31 for one selection cycle. A predetermined time after the first pulse switch 39 is positioned by cam 48 with contacts 38 and 40 made so that if a second A.C. pulse, 3 Fig. 1, is detected by circuit 23, energizing current is applied to relay 36, which holds over contacts 42, and also makes contacts 45 to enable the circuit of a tripping relay 46. Cam 48 has a projection 50 which makes contacts 40 and 41 of switch 39, and if a further pulse is received at the time this connection is made, e.g. if the second pulse was the result of noise or interference, then the relay coil is shorted and de-energized. At a later time cam 49 makes contacts 40 and 41 and this time coincides with gap, 13, Fig. 1 in a burst of pulses 9 to 16, in the selection signal for the particular receiver, and if a pulse is present at this time, indicating a non-selection of this receiver, the relay coil is again shorted to de-energize. If a pulse does not occur the relay is held and a subsequent pulse, 17 or 18 Fig. 1, when switch 44 is operated by cam disc 30, will cause energization of a tripping relay 47. The tripping relay is operated alternately on and off by successive pulses applied to its coil and the relay has contacts 46 in its operating circuit, operated by the tripping relay, so that a pulse to switch the relay " on " has to occur at the appropriate time in the cycle, e.g. when the switch contact 43 is depressed by cam 30 to be effective and is only effective if the relay is " off ", while the " off " pulse has to occur at a different time, e.g. when the contact 43 is raised, and when the relay is " on ". Modifications of the circuit are described to utilize a preselection relay with a double winding, Fig. 3 (not shown), a D.C. relay fed via a bridge rectifier Fig. 4 (not shown) or a s.c.r. to replace the relay 36 and its contacts 42 and 45, Fig. 5 (not shown).
Patent GB-1251135-A (GB)
Filed: 1969-07-11
Abstract: 1,251,135. 0-Acyl and O-sulphonyl decarbamoyl-mitomycins. KYOWA HAKKO KOGYO K.K. 11 July, 1969 [23 July, 1968; 24 July, 1968], No. 35165/69. Heading C2A. Novel 0-acyl and O-sulphonyl decarbamoylmitomycins of Formula I wherein (a) R is -COR 1  and X is -NH 2 , Y is -OCH 3  and Z is -H; or (b) R is -SO 2 R 2  and X is -NH 2  or -OCH 3 , Y is -OCH 3  or -OH and Z is -CH 3  or -COR 1 , in which groups R 1  is substituted or unsubstituted C 1 -C 5  alkyl and R 2  is C 1 -C 5  alkyl or an aromatic hydrocarbon group, are prepared by (i) subjecting a diacylated decarbamoyl mitomycin C of formula to one or two stages of hydrolysis to replace first the N-acyl group and then optionally the 0-acyl group, by hydrogen; or (ii) by treating a decarbamoyl mitomycin of formula with a sulphonating agent. The hydrolysis may be effected by treating a solution of the starting mitomycin in a watermiscible organic solvent with aqueous weak alkali (e.g. NaHCO 3 , Na 2 CO 3  or NH 4 OH) at room temperature for a period of time necessary to give the required degree of hydrolysis. The sulphonation process suitably consists of treating the starting mitomycin with sulphonyl chloride or alkyl- or aryl-sulphonyl chloride in water or organic solvent in the presence of a molar excess of a base which may also be the solvent (e.g. pyridine), at ambient temperature or below. The compounds have bacteriostatic properties.