baber/WOPTO huggingface dataset:
Patent CZ-282363-B6 (CZ)
Title: Plaster with active component for controlled dosage and process for preparing thereof
Inventor: HOFFMANN HANS-RAINER DR
IPC: A61K31/56
Filed: 1990-10-05
Abstract: The invention relates to a drug plaster for the controlled delivery of drugs to the skin, which consists of a backing layer and of a water-insoluble adhesive film which is attached thereto and is composed of an adhesive which contains polymers which are swellable in water and in which the drug is at least partially soluble, and of a protective layer which covers the adhesive film and can be detached again, which is characterised in that the adhesive is based on homo- and/or copolymers with at least one derivative of acrylic or methacrylic acid and contains, as drugs partially or completely dissolved in the adhesive, in a concentration of 0.5 to 10.0% by weight, oestrogens and their pharmaceutically acceptable derivatives alone or in combination with gestagens.
Patent CZ-279235-B6 (CZ)
Inventor: POLOUCEK EDUARD PROM CHEM
IPC: C08K9/04
Filed: 1988-11-07
Abstract: Povrchová úprava minerálních plniv pro plasty se  provádí roztoky amonných solí vyšších mastných  kyselin s 12 až 32 uhlíkovými atomy za normální  či zvýšené teploty. Z amonných solí se na  povrchu plniva vysráží nerozpustné soli mastných  kyselin, které jsou vázány k povrchu plniva  chemickými vazbami na rozdíl od známé impregnace  povrchu plniva nerozpustnými solemi mastných  kyselin. Lepší vazba impregnace se projeví  snížením indexu toku taveniny kompozitu plastu s  takto upraveným plnivem a snížením kroutícího  momentu.ŕ
Patent CZ-291621-B6 (CZ)
Title: Oxazolidinone derivative, process of its preparation its use and pharmaceutical preparation in which the derivative is comprised
Inventor: GANTE JOACHIM PROF DR
IPC: C07D401/04
Filed: 1996-05-03
Abstract: The present invention relates to an oxazolidinone derivative of the general formula I, in which R represents the group of the general formula (a) wherein n is 1 or 2, Re1 represents hydrogen, Re2 denotes OH, OA, OAr, OHet, NHOH, NHi2, NHA or NAi2, Re3 represents A-CO, ArCO, Het-CO, Het-O-CO-, Ar-O-CO, A-O-CO, Ar-SOi2 or A-SOi2, A denotes alkyl containing 1 to 6 carbon atoms, Ar represents aryl having 6 to 10 carbon atoms, diphenylmethyl or benzyl, which are optionally substituted with 1, 2 or 3 substituents being selected from the group comprising A, fluorine, chlorine, bromine, iodine, AO, -O-CHi2-O-, COOA, COOH, CFi3, OH, NOi2, CN, -O-CO-A, NHi2, NHA and NAi2, Het represents a mono- or bicyclic, saturated, unsaturated or aromatic heterocyclic group having 1 to 4 nitrogen atoms, oxygen and/or sulfur being optionally substituted with one substituent selected from the group comprising fluorine, chlorine, bromine, CFi3, A, OH, OA, CN and NOi2. The above described derivative and physiologically acceptable salts thereof inhibit binding of fibrinogen to corresponding receptors and are  therefore suitable for treating thromboses, osteoporoses, tumor diseases, apoplexy, heart infarct, ischemia, inflammations, arteriosclerosis and osteolytic diseases.
Patent CZ-281677-B6 (CZ)
Title: Auxiliary circuit controller
Inventor: MARES FRANTISEK
IPC: H01H3/00
Filed: 1995-05-30
Abstract: The equipment consists of the gate (2) of the rotary knob (1) where the gate form No.I (4) together with the gate path (8) of the arrester (6) specify the movement of the rotary knob (1). In the arresting groove (3) there is a sealing (9) with a hole and an arresting ring (11) and the arresting hole (13) which after mounting on the arresting groove (3) and arresting in the previously specified position by arresting pins (16) is located in the head (15) of the insert and passes through the arresting holes of the arresting ring (11), sealing (9) and the arresting pin (6) prevents the removal of the gate form No.II (5).<IMAGE>
Patent CZ-298655-B6 (CZ)
Title: Apparatus for registration of overvoltage pulses between a pair of elements with different electric potential
Inventor: CERNICKA JOZEF
IPC: G01R29/02
Filed: 1999-08-20
Abstract: In the present invention, there is disclosed an apparatus for registration of overvoltage pulses between a couple of elements with different electric potential comprising a connecting element (1) provided with at least one connecting conductor (5, 6) with an overvoltage pulse sensor (9) assigned thereto. Said overvoltage pulse sensor (9) includes a ferromagnetic element (10) being provided with a slot (10) accommodating a magnetic field sensor (12) that is coupled with an evaluation module (14). One of these connecting element (1) connecting conductors (5, 6) is at least partially wound round said overvoltage pulse sensor (9) ferromagnetic element (10).
Patent CZ-298063-B6 (CZ)
Title: Apparatus for introducing gobs of molten glass into a glass container forming machine of the individual section type
Inventor: CIRINCIONE RONALD A
IPC: C03B40/027
Filed: 1998-10-12
Abstract: In combination with a blank mold (18) of a glass container forming machine of the individual section type, there is disclosed an apparatus having a loading funnel (10) adapted to be positioned immediately upstream of the blank mold (18) for aligning gobs (G) of molten glass passing in sequence through the loading funnel (10) into the blank mold (18), said loading funnel (10) comprising: an upper gathering section (10a) having an outer shape in the form of an inverted frustum of a cone; and a lower shaping and orienting section (10b) whose outer shape is that of a cylinder being a portion of said loading funnel (10) and being disposed immediately above the blank mold (18). The internal diameter of the shaping and orienting section (10b) is somewhat less than the outer diameter of a gob passing therethrough, to thereby contact the gob in a substantially circumferential pattern, and the shaping and orienting section has a length that is sufficient to precisely align the longitudinal central axis of the gob (G) with a longitudinal central axis of the blank mold (18), to thereby eliminate or substantially eliminate the need to swab the interior of the blank mold (18) with a mold dopant composition.
Patent CZ-295747-B6 (CZ)
Title: Substituted benzylamines and pharmaceutical composition
Inventor: LEYSEN DIRK CASIMIR MARIA
IPC: A61K31/42
Filed: 1997-04-15
Abstract: In the present invention, there are disclosed benzylamine derivatives of the general formula I, in which Re1 and Re2, which can be the same or different are each selected from the group consisting of aryl containing 6 to 12 carbon atoms, heteroaryl having 2 to 14 carbon atoms, arylalkyl containing 6 to 12 carbon atoms in the aryl moiety and 1 to 6 carbon atoms in the alkyl moiety, heteroarylalkyl having 2 to 14 carbon atoms in the heteroaryl moiety and 1 to 6 carbon atoms in the alkyl moiety, wherein the alkyl, aryl or heteroaryl moieties can be optionally substituted and wherein heteroaryl contains one to three heteroatoms being selected from the group consisting of oxygen, sulfur and nitrogen, or one of the Re1 and Re2 groups is as defined above and the other represents hydroxy; Re3 and Re4, which can be the same or different are each selected from the group consisting of aryl containing 6 to 12 carbon atoms, heteroaryl having 2 to 14 carbon atoms, arylalkyl containing 6 to 12 carbon atoms in the aryl moiety and 1 to 6 carbon atoms in the alkyl moiety, heteroarylalkyl having 2 to 14 carbon atoms in the heteroaryl moiety and 1 to 6 carbon atoms in the alkyl moiety, wherein the alkyl, aryl or heteroaryl moieties can be optionally substituted; or one of the Re3 or Re4 groups together with one of the Re1 and Re2 groups and a nitrogen atom attached thereto form a 5- or 6-membered heterocyclic ring, Re5 represents one or several ring substituents being selected from the group consisting of halogen, a hydrogen atom, alkyl having 1 to 6 carbon atoms and alkoxy containing 1 to 6 carbon atoms; and Re6 represents a single ring substituent of the general formula A, in which the dotted lines represent an optional bond; Y denotes an oxygen atom or the group -NRe8 (wherein Re8 denotes a hydrogen atom or alkyl containing 1 to 6 carbon atoms) and Re7 represents one or several substituents being selected from the group consisting of a hydrogen atom, halogen, haloalkyl having 1 to 6 carbon atoms in the alkyl moiety, alkyl containing 1 to 6 carbon atoms and alkoxy containing 1 to 6 carbon atoms; or pharmaceutically acceptable salts or solvates  thereof. Disclosed are also pharmaceutical compositions containing the above-described derivatives as well as their use in medicine, particularly for treating depression.
Patent SK-280143-B6 (SK)
Title: Heterobicyclic compounds, method of their praparation, and pharmaceutical compositions them contaiing
Inventor: LEONARDI AMEDEO
IPC: A61K35/00
Filed: 1993-02-23
Abstract: There are disclosed compounds of general formula (I). The heteroatom X is preferably oxygen, or sulphur, imino, C1-6alkylimino group. The group W is preferably a carbonyl group, but also C=S, CH2, CH(OH). The preferred heterocyclic ring is thus a 4-oxo-4H-1-benzopyran ring. This may have a wide range of R2, R3, R6, R7 substituents. Y is a linking group, chosen from a wide range, but including -COO-, - CONH-, -O-, -SO2- and -SO2NH-. Z is an alkylene chain, and B is a complex amine. These compounds and their prodrugs, enantiomers, diastereoisomers, N-oxides and pharmaceutically acceptable salts are useful for the treatment of hypertension and urinary tract troubles associated with benign prostatic hypertrophy.
Patent SK-282058-B6 (SK)
Title: Acetic acid derivatives, method for their production, pharmaceutical preparations based on them and their use for production of medicaments
Inventor: ALIG LEO
IPC: C07C259/18
Filed: 1994-11-30
Abstract: Acetic acid derivatives of the formula <IMAGE> in which L, M, Q and T have the meaning stated in the description, can be used for the treatment or prophylaxis of diseases caused by the binding of adhesive proteins to blood platelets, and by aggregation of blood platelets and cell-cell adhesion. They are prepared by eliminating protective groups in corresponding protected compounds or by converting the cyano group into the amidino group in corresponding nitriles.
Patent SK-279003-B6 (SK)
Title: Substrate with the negative working light sensitive layer
Inventor: VESELY MICHAL
IPC: G03G7/00
Filed: 1992-07-30
Abstract: The solution described in this patent deals with the substrate covered by the light sensitive layer for photo chemical reproduction, during the chemical treatment, while this substrate is created based on the metal substrate covered by the light sensitive layer, while this layer consists of 90 up to 98 weight percent phenol formaldehyde resin or substituted phenol formaldehyde resin, of 2 up to 10 weight percent anthracene and of 0,01 up to 0,5 weight percent related to singlet sensitiser, while this light sensitive layer contains 0,05 up to 1 weight percent of organic pigment.
Patent SK-279572-B6 (SK)
Title: Biodegradable material, process for producing the same, use thereof
Inventor: SCHROETER JOHANNES
IPC: C08J3/20
Filed: 1992-12-31
Abstract: The invention relates to a biodegradable material which contains from 30 to 85 percent by weight of a biodegradable polysaccharide-based plastic, from 15 to 70 percent by weight of native starch or unmodified cellulose, and optionally conventional auxiliaries. Said biodegradable plastic is melt down at temperature ranging from the melting point of plastics to 240 degrees Celsius, simultaneously or subsequently to, starch or unmodified cellulose is added with the proviso that water content present in starch does not exceed 20 percent. Thus obtained mixture is subjected to granulation, then is moulded according to known methods, or the biodegradable plastic is dissolved in such a solvent that prevents starch dissolving, then starch is added and organosol thus obtained is moulded according to known methods.
Patent SK-278031-B6 (SK)
Title: Combine regulating circuit of hydrogenerator for constant through flow
Inventor: KLEINEDLER PETER
IPC: G05D7/06
Filed: 1990-12-27
Abstract: Combined regulating circuit controls the geometrical volume of hydrogenerator (1). Solution safeguards the constantional leading through flow in second high-pressure leading (4) by different inlet revolutions of hydrogenerator (1) and possibility of arbitrary delivery in first high-pressure leading (2) in dependence of inlet revolutions of hydrogenerator (1) and position of adjustment of mechanical-hydraulic servosystem.
Patent CZ-297025-B6 (CZ)
Title: Cylinder-type lock
Inventor: MOTTURA SERGIO
IPC: E05B19/00
Filed: 1999-05-06
Abstract: The present invention relates to a cylinder-type lock comprising a cylinder /10/ having a plurality of locking tumblers /16/, which are rotatably mounted around respective axes. The introduction of a key /3/ causes rotation of each locking tumbler /16/ to an operative position in which the tumblers enable the disengagement of a locking member /17/ carried by the cylinder /10/ from a seat /19/ formed in the stator /8/ of the lock.
Patent CZ-300620-B6 (CZ)
Title: Method for synchronizing internal clock of mobile radio terminal with local time
Inventor: ZSCHINTZSCH HANS
IPC: H04Q7/32
Filed: 2001-08-09
Abstract: In the present invention, there is disclosed a method for the synchronization of the internal clock of a mobile radio terminal device with the local time, characterized in that the mobile radio terminal device sends at time ti0 a short message (SM) that is conducted via a so-called Short Message Service Center (SMSC), and here each message is provided with a time stamp tiZ which, in turn, is indicated to the receiver of the message. The mobile radio terminal device registers the sending time ti0 of the short message(SM) as well as the time of acknowledgment ti1 of the short message and therefrom derives the time tiM=(ti1+ti0)/2, wherein tiM corresponds approximately to the point in time of the time stamp tiZ. The mobile radio terminal device extracts from the received short message (SM) the time stamp tiZ, compares it with tiM, and corrects the internal clock by the difference tiD=tiZ-tiM.
Patent CZ-303945-B6 (CZ)
Title: Closing and securing mechanism of rotary mounted door of steam sterilizer sterilizing chamber
Inventor: OSTADAL JINDRICH
IPC: A61L2/20
Filed: 2009-12-08
Abstract: In the present invention, there is disclosed a mechanism eliminating a force needful for compression of a door (2) upon its closing and sealing by distribution the closing process in several phases. The force of a sterilization chamber (1) and the door (2) compression load is distributed on the side of a closure in two points. The closing and securing mechanism of the present invention consists of the hinged door (2) attached to the sterilization chamber (1) of a steam sterilizer. Fixed components of the door (2) form a mount (14) of a guide and a mount (15) of centering, which both are provided with coaxial openings. In the guide mount (14) opening, there is slidably mounted a door pin (3) that is coupled with a distance tube (7) with a spring (12) arranged thereon. Said spring (12) preloading is defined by both, a support (17) being fixedly coupled with the door (2) a limiter (18) being fixedly coupled with the distance tube (7). At the same time, said limiter (18) functions as a stop and defines thereby axial movement of the distance tube (7).
Patent CZ-305452-B6 (CZ)
Title: Pendant for coin accommodation
Inventor: GAŠPÁR ZDENĚK
IPC: A44C25/00
Filed: 2014-03-11
Abstract: The present invention relates to a pendant for placing a coin in a peripheral groove thereof, wherein the pendant consists of two flanges (1, 2) with identical contours and coaxial openings (3, 4) for showing the coin, wherein the first flange (1) is provided with axially projecting hollow cylinder (6) that is provided on its outer wall with a thread for screwing into internal thread of a cylindrical cavity performed in the second flange (2), whereby the diameter (R1) of each opening (3, 4) in the flanges (1, 2) is smaller than the inside diameter (R) of the hollow cylinder (6). At the same time, each flange (1, 2) is provided on its circumference with a connecting opening (8), and in screwed up state said connecting openings (8) are coaxial.
Patent CZ-305420-B6 (CZ)
Title: Electricity generation plant with the use of steam-gas mixture
Inventor: VILIMEC LADISLAV
IPC: F01K27/00
Filed: 2014-09-29
Abstract: A steam turbine with a second current generator is connected in a steam piping within a circuit of a plant with a combustion chamber (1), a gas turbine (7) a mixer (10) and a steam-gas heater (6), wherein said steam turbine inlet faces the combustion chamber (1) while the outlet thereof faces the mixer (10). Preferably, at least one steam superheater (17) is connected in front of the steam turbine (14) inside the combustion chamber (1). Optionally, a bleeding piping (16) is connected to the steam piping, between the combustion chamber (1) and the mixer (10).
Patent CZ-307497-B6 (CZ)
Title: An air gun
Inventor: Rotrekl Michal
IPC: F41B11/70
Filed: 2017-10-06
Abstract: An air gun with a barrel (1) provided with a bore (2), wherein the bore (2) is connected to the supply channel (3) of the compressed medium. The supply channel (3) is terminated by an annular distributor space (4) arranged around the axis of the barrel (1), wherein the distribution channels (5) connected to the barrel (1) bore (2) extend from the annular distributor space (4) towards the axis of the barrel (1)
Patent CZ-308129-B6 (CZ)
Title: Electric railway vehicle for handling spent nuclear fuel envelope
Inventor: HALADA PAVEL
IPC: G21F5/14
Filed: 2018-10-26
Abstract: The electric railway vehicle (1) for handling a package of burnt nuclear fuel is used as a container for handling the spent fuel (5) of burnt nuclear fuel, and its main part is a railway chassis (2), lifting mechanism (3) and leading mechanism (4). To insert the spent nuclear fuel set (5), of the burnt nuclear fuel two pairs of opposing support and guide pins (6) are used which are part of the spent nuclear fuel set (5), the lower pair guide it into the tube (10) by guide surfaces (8) and guide grooves (7) and the upper pair for handling with an external handling device.
Patent CZ-309716-B6 (CZ)
Title: A preparation for treating degenerative damage to the retina
Inventor: BAUER PETR
IPC: A61K35/12
Filed: 2019-12-12
Abstract: The invention relates to a therapeutic preparation consisting of stem cells and a buffered aqueous solution containing trehalose or sucrose for intravitreal administration and is intended for the invasive treatment of degenerative diseases of the human eye, especially pathological changes on the retina. The preparation according to the invention contains 7 to 13 x 106 purified expanded mesenchymal stem cells per ml of the preparation, the pharmaceutical solution contains cations K+, Mg2+ Na+ and anions Cl-, PO43- and/or HPO42- and/or H2PO4-, SO42- and further contains 0.18 to 0.22 mol of trehalose or sucrose per litre of pharmaceutical solution, the pH of the pharmaceutical solution is 7.1 to 7.6 and the total osmolarity of the pharmaceutical solution is 200 to 400 mosmol/L.
Patent CZ-309885-B6 (CZ)
Title: Triterpenes with inhibitory activity on the Hedgehog signalling pathway for the use in the treatment of cancer
Inventor: URBAN MILAN
IPC: C07J63/00
Filed: 2022-06-21
Abstract: The subject of the presented solution are terpenoid derivatives of the general formula I, in which,------ is a single or double bond; A, X, Y and Z are independently selected from the group consisting of CH, C, N, NH, O, S; wherein at least one of A, X, Y, Z is O or S; R1 is selected from the group consisting of -CH2OH, -CH2O(CH2)nCH3, -CH2OC(O)(CH2)nCH3, -COOH, ‑COO(CH2)nCH3 and -COO(CH2)Ph, -COOCH2OC(O)CH3, where independently n = 0 to 5; and pharmaceutically acceptable salts thereof. Terpenoid derivatives of formula I significantly inhibit the Hedgehog cell signalling pathway and are useful for the treatment of cancer diseases.
Patent CZ-298223-B6 (CZ)
Title: Bias estimating method for a target tracking system
Inventor: SVIESTINS EGILS
IPC: G01S15/86
Filed: 1998-10-26
Abstract: In the present invention, there is disclosed a bias estimating method for a target tracking system, comprising the steps of: collecting target tracks (T) and associated measurements (M) from said target tracking system; calculating estimates of bias parameters (b) based on said target tracks (T) and measurements (M) associated therewith; providing said target tracking system with said calculated estimates of the bias parameters (b), characterized in that the calculating step comprises the steps of: generating an error function, comprising at least two terms, where a first term is dependent of at least the magnitude of the discrepancy between measurements and a measuring model, where the measuring model is a model function of an unknown target position and unknown bias parameters, and where a second term is dependent of at least predetermined evaluations of the a priori statistical distributions of the bias errors (15) and said unknown bias parameters; and minimising said error function with respect to said bias parameters as well as said target position. The process of the invention repeatedly generates estimates for sensor bias errors (b) by minimising a function, given on one hand by the magnitude of the discrepancy between measurements (M) and a measuring model, where the measuring model is a function of the unknown target location and unknown bias parameters, and on the other by the bias parameters and their predetermined statistical distributions (15). In a preferred embodiment of the present invention, the minimising step is performed by linearising components of the function around an approximate target position (normally obtained from the tracker (10)) and around nominal (typically zero) bias errors, and the function is subsequently minimised with respect to target positions as well as to the bias parameters (b). In addition, possible time dependence of the bias parameters is modelled by the incorporation of process noise.
Patent CZ-294045-B6 (CZ)
Title: Mechanism for tightening belts of belt gearbox
Inventor: SLAMA PAVEL ING
IPC: F16H7/10
Filed: 2000-05-09
Abstract: In the present invention, there is disclosed a mechanism for tightening belts of a belt gearbox intended particularly for drive of spindles of machine tools, machine centers and automatic machine tools, with a transmission box mounted on a machine tool headstock, wherein the mechanism comprises a tightening screw (9) and a T-square (10) fastened on a transmission box (3). In the transmission box (3), there is mounted on a pin-type lugs (11) a pivoted lever (12) with a tightening pulley (13) bearing in working position on a V-shaped belt (7, 8) connecting a drive pulley (4) and a driven pulley (6). Said pivoted lever (12) is provided on the side turned away from the V-shaped belt (7, 8) with bearing surfaces (121). Press-away screws (14) are arranged opposite to the bearing surfaces (121) in the transmission box (3).
Patent CZ-295289-B6 (CZ)
Title: Filter candle
Inventor: HAHN ADOLF
IPC: B01D29/33
Filed: 2002-03-15
Abstract: The present invention relates to a filter candle for a precoated filter for filtering and/or stabilizing fluids, especially beer. The inventive filter candle comprises a tubular filter body (2) that is configured from a spirally wound wire (17), with gaps (11) being provided between the wire (17) windings for allowing the fluid to pass. The surface (20) of the wound wire (17) that rests against the exterior of the filter body (2) is inclined by an angle alpha relative to the longitudinal axis of the filter candle (1). Said wire cross section is substantially triangular and narrowed inwardly, whereby the triangle base line lies on outer side of the filter body (2) to thereby enabling radial stepping of the adjacent edges of the surfaces (20) of the wire (17) coils following each another.