baber/WOPTO huggingface dataset:
Patent NZ-712540-A (NZ)
Title: Phenyl derivative having s1p2 antagonistic activity
Inventor: NAGANAWA ATSUSHI
IPC: C07D211/48
Filed: 2014-03-25
Abstract: Provided is a compound with strong human S1P2 antagonistic activity in order to develop drug products that are useful for treating S1P2 mediated disorders such as disorders that cause constriction of blood vessels, fibrosing disease, respiratory disease, and the like. The compound expressed by general formula (I) (in formula, all symbols are as described in the specification) has strong human S1P2 antagonistic activity by introducing a halogen atom or a haloalkyl group and a phenoxy group to a specific substitution site, and therefore can provide a therapeutic agent for S1P2 mediated disorders such as disorders that cause constriction of blood vessels, fibrosing disease, respiratory disease, and the like.
Patent NZ-718928-A (NZ)
Title: A flocculant dispensing system and method
Inventor: ROBERT GRAEME COULSON
IPC: C02F1/52
Filed: 2013-09-25
Abstract: A flocculant dispensing system (110) for dispensing flocculant into a pond (129) is disclosed. The flocculant dispensing system comprises a flocculant storage reservoir, a dispenser, a pump (127), and an electronic controller. The system further includes a sonic sensor (123) arranged to detect water flow rate into the pond (129). The sensor generates a control signal which is processed by the electronic controller to determine the amount of flocculant to be dispensed.
Patent NZ-728687-A (NZ)
Title: Magnetically-chambered fully automatic air gun
Inventor: MARSHALL JAMES
IPC: F41B11/00
Filed: 2015-07-27
Abstract: The present invention relates to the field of mechanical guns. Conventional mechanical guns are difficult to maintain and involve overly complex mechanical actions. Further, convention mechanical guns that use magnetic forces, merely use magnetism as an adjunct to some form of mechanical action. The presently claimed invention relates to an open chamber air gun where a round is gravity fed or magnetically fed into the open chamber and falls into the magnetic flux lines of a magnet disposed at the chamber. Due to the magnet, the round is pulled securely into the chamber and then remains momentarily held in place, blocking much of the air behind it and thus increasing the air pressure driving it. When the round moves down the barrel from the breech toward the muzzle, it quickly leaves the vicinity of the magnet and the magnetic drag ceases, after which the air pressure is free to drive the round to full velocity. High rates of fire and muzzle velocities are achieved with moderate air pressure and an action with no moving parts.
Patent NZ-729815-A (NZ)
Title: Fused heterocyclic compounds as gpr120 agonists
Inventor: SHARMA RAJIV
IPC: A61K31/4035
Filed: 2015-09-09
Abstract: The present invention relates to fused heterocyclic compound of Formula (I), a stereoisomer, a tautomer, a pharmaceutically acceptable salt, a pharmaceutically acceptable solvate, a prodrug, a polymorph, N-oxide, S-oxide, or a carboxylic acid isostere thereof; processes for their preparation; pharmaceutical compositions comprising said compounds; and their use for the treatment of the diseases or disorders mediated by GPR120 receptor. Key compounds of formula (I) include 4-(2-(2-(5-cyclopropylthiophen-2-yl)-5-fluorophenyl)benzofuran-5-yl)butanoic acid, 4-(2-(5-Fluoro-2-(5-(1-methylcyclopropyl)thiophen-2-yl)phenyl)benzofuran-5-yl)butanoic acid, 4-(2-(2-(5-Cyclopropylthiazol-2-yl)-5-fluorophenyl)benzofuran-5-yl)butanoic acid, 4-(2-(2-(5,6-Dihydro-4H-cyclopenta[d]thiazol-2-yl)-5-fluorophenyl)benzofuran-5-yl)butanoic acid, 4-(2-(5-Fluoro-2-(4,5,6,7-tetrahydrobenzo[d]thiazol-2-yl)phenyl)benzofuran-5-yl)butanoic acid, 4-(2-(5-Fluoro-2-(isoindolin-5-yl)phenyl)benzofuran-5-yl)butanoic acid, 4-(2-(2-(5,7-Dihydrofuro[3,4-b]pyridin-3-yl)-5-fluorophenyl)benzofuran-5-yl)butanoic acid and 4-(2-(2-(6,7-Dihydro-5H-cyclopenta[b]pyridin-3-yl)-5-fluorophenyl)benzofuran-5-yl)butanoic acid.
Patent NZ-730643-A (NZ)
Title: Bottle lid assembly with retractable spout
Inventor: MEBBERSON NICK
IPC: B65D47/28
Filed: 2015-09-22
Abstract: A bottle lid assembly incorporating a spout that is covered by a lid when not in use to prevent contamination of the spout and which exposes the spout to the user through the lid upon activation of mechanism by the user. The lid assembly for a bottle including a base attachable to said bottle over a mouth, a main body rotatably connected to said base, a cover configured to extend over an open upper end of the main body, the cover including an opening extending therethrough, a spout slidably held within said main body and movable along a first axis between a retracted and an extended position and a pivotable flap configured to close the opening in the cover when the spout is in the retracted position, wherein pivoting of the flap is actuated by movement of the main body. The main body including an internal spur gear wherein upon rotation of said main body the internal spur gear is engageable with the pinion to move the flap across or clear of the opening in the cover and when the internal spur gear member and pinion are not engaged the flap remains substantially stationary while the main body continues to rotate.
Patent NZ-739131-A (NZ)
Title: Methods for making a foamed adhesive containing closed cells
Inventor: LUNDE ERIK
IPC: C09J5/08
Filed: 2012-09-20
Abstract: Method for making foamed adhesive compositions suitable for use in adhesive dressings for topical application to the body, the method including providing a molten adhesive composition, combining an inert gas with the molten adhesive composition in a first mixer, mixing the molten adhesive composition comprising the inert gas in the first mixer under conditions effective to form a first foamed adhesive composition; and mixing the first foamed adhesive composition in a second mixer that includes a rotating mixing blade under conditions effective to provide a second foamed adhesive composition having a substantially homogenous distribution of closed cells containing the inert gas. An internal pressure of the first foamed adhesive composition entering the second mixer is greater than an external pressure of the second foamed adhesive composition exiting said second mixer, thereby providing a pressure differential. The pressure differential is about 115 psi or greater.
Patent NZ-750974-A (NZ)
Title: Antibody and checkpoint inhibitor combination therapy
Inventor: LAVRANOS TINA CHRISTINE
IPC: A61K39/395
Filed: 2017-09-14
Abstract: The present invention provides a combination therapy for treatment of a tumour in a subject. The combination therapy comprises administration of (i) an antibody directed against cancer stem cells and (ii) a checkpoint inhibitor.
Patent NZ-756484-A (NZ)
Title: Tuning of a kinematic relationship between members
Inventor: CHRISTOPHER JAMES ALLINGTON
IPC: B60R22/46
Filed: 2014-08-18
Abstract: A clutch or brake comprising: At least one first member in a kinematic relationship with at least one further member to form a system, the system moving within a limited range of motion and wherein the system interacts when an external energising force is imposed on the system causing the members to respond due to their kinematic and dynamic characteristics and thereby creating relative motion between the members; and at least one trigger member mechanically coupled to the at least one first member that moves with respect to the first member in response to a pre-determined system movement and, when the at least one trigger member moves, the at least one trigger member or a part thereof imposes a braking action on the system or a member or members thereof, by an interaction between the trigger member and the further member, resisting relative movement between the trigger member and the further member; wherein the speed and/or intensity of the braking action imposed by the at least one trigger member on the system or a member or members thereof is controlled by the at least one trigger member rate of movement with respect to the first member and this rate of movement is in turn governed by a magnetic flux interaction between the at least one trigger member or a part thereof and the at least one first member or a part thereof causing formation of a magnetically-induced eddy current force between the at least one trigger member or a part thereof and the at least one first member or a part thereof, the eddy current force resisting movement of the trigger member with respect to the first member.
Patent NZ-767139-A (NZ)
Title: Multicyclic compounds and methods of use thereof
Inventor: SHAO LIMING
IPC: A61P25/00
Filed: 2010-12-03
Abstract: Disclosed are cyclopenta[b]thiophene compounds of general formula (I), wherein X and Y are CH2; Z2 is C; Z3 is S; Z1 is C; R5 is hydrogen; R6 and R7 are each independently hydrogen, halo or alkyl; m is 0; n is 0; and wherein the remaining substituents are as defined herein. Representative compounds include 1-(3-methyl-5,6-dihydro-4H-cyclopenta[b]thiophen-4-yl)-N-methylmethanamine. Medicaments comprising the compounds are provided for use in treating neurological disorders such as schizophrenia, psychotic disorders, Parkinson’s psychosis, bipolar disorder, Alzheimer’s disease agitation, attention deficit disorder, attention deficit hyperactivity disorder, Tourette’s syndrome, post-traumatic stress disorder, depression, obsessive compulsive disorder, narcolepsy, substance abuse or dependency, autism and the like.
Patent PT-108887-A (PT)
Title: Material compósito à base de materiais provenientes da atividade agroindustrial, processo de produção e respetivo uso.
Inventor: ANA MARIA SANTOS LIMA
IPC: B09B3/00
Filed: 2015-10-14
Abstract: A PRESENTE DIVULGAÇÃO DIZ RESPEITO A UM MATERIAL COMPÓSITO, À BASE DE UM AGENTE LIGANTE E/OU AGLOMERANTE E DE MATERIAIS RESULTANTES DA ATIVIDADE AGROINDUSTRIAL, NOMEADAMENTE RESÍDUOS, BIORRESÍDUOS, E/OU SUBPRODUTOS AGROINDUSTRIAIS RESULTANTES DE VÁRIAS INDÚSTRIAS. ESTA DIVULGAÇÃO TAMBÉM DIZ RESPEITO AO PROCESSO DE PRODUÇÃO DO REFERIDO MATERIAL COMPÓSITO E AO RESPETIVO USO DO MESMO.
Patent PT-109231-A (PT)
Title: Equipamento de fabrico aditivo para a produção de componentes em vidro multicolor
Inventor: ARTUR JORGE DOS SANTOS MATEUS
IPC: C03B37/00
Filed: 2016-03-11
Abstract: A PRESENTE INVENÇÃO DIZ RESPEITO A UM EQUIPAMENTO DE FABRICO ADITIVO DE COMPONENTES EM VIDRO MULTICOLOR, FORNECIDO SOB A FORMA DE VARETAS (2), QUE APRESENTA UM RESERVATÓRIO DE MATERIAL (VIDRO SOB A FORMA DE VARETAS DE DIFERENTES CORES E DIÂMETROS) (1), UM ALIMENTADOR DE MATERIAL AUTOMATIZADO (3), UM ACUMULADOR DE CALOR(5), UM SISTEMA DE PROJEÇÃO DE PÓS DE VIDRO DE DIFERENTES CORES (4), UMA FONTE DE CALOR (6) E UM SISTEMA DE TROCA AUTOMATIZADO DA PLATAFORMA DE CONSTRUÇÃO (7) A QUAL É PARTE INTEGRANTE DE UM SISTEMA DE MUDANÇA DA PLATAFORMA DE CONSTRUÇÃO AUTOMÁTICO (7). OS COMPONENTES PRODUZIDOS SÃO CARACTERIZADOS POR POSSUÍREM UMA QUASE TOTAL LIBERDADE DE GEOMETRIAS E FORMAS, COMO RESULTADO DA DEPOSIÇÃO, POR EXTRUSÃO, CAMADA A CAMADA DE VIDRO DE DIFERENTES CORES. O VIDRO APRESENTA-SE SOB A FORMA DE VARETAS COM DIFERENTES CORES E DIÂMETROS. O EQUIPAMENTO, OBJETO DA PRESENTE INVENÇÃO, INCLUI UM CONJUNTO DE PELO MENOS QUATRO EIXOS CARTESIANOS (XYZW E OUTROS) MOTORIZADOS E CONTROLADOS POR UM SISTEMA DE CONTROLO, GERADOR DE TRAJETÓRIAS E SISTEMA DE MUDANÇA DA PLATAFORMA DE CONSTRUÇÃO AUTOMÁTICO (7), O QUAL SE PODE MOVIMENTA NO SENTIDO DO EIXO ZZ.
Patent RU-94017056-A (RU)
Inventor: MAZURKIN P M
IPC: A01G23/06
Filed: 1994-05-10
Abstract: FIELD: equipment for continuous, strip and local soil cultivation. SUBSTANCE: working tool has supporting-rotary device 4 with movable toothed wheel 6 and drive with drive gear, supporting plate 11 with self-rotating cutters 7 positioned in casing 9, with cutter axes being positioned at an angle with respect to axis of movable toothed wheel 6. Cutting edges of cutters 7 are offset with respect to their axes. EFFECT: increased efficiency in loosening felling area soil, clearing reclamative channels and other lands from bushes, wider operational capabilities and enhanced reliability in operation. 3 cl, 4 dwg
Patent RU-94034759-A (RU)
Inventor: BOGATYREV A E
IPC: C08J5/22
Filed: 1994-09-20
Abstract: FIELD: membrane technologies. SUBSTANCE: as compared with the prototype, the amount of resin in the offered membrane is reduced to 0.003-11.0 mas.% of the total membrane mass and left on walls of pores of the base only thin film of resin or some other hydrophylic agent with thickness of 1.0 to 10-15 monomolecular layers, for which purpose, excessive resin is pickled out by oxidizing pickling agents from membranes produced by the method described in the Application for a patent. EFFECT: higher efficiency.
Patent RU-94042056-A (RU)
Inventor: PEREZHILOV A E
IPC: E21D1/12
Filed: 1994-11-22
Abstract: FIELD: mining. SUBSTANCE: control over stage-by-stage process of forming ice-rock guard is carried out. Design volume of cold carrier is pumped through a group of wells under active mode of freezing to form individual ice-rock bodies of optimum size. Changing over the stage is carried out by switching over a group of wells of the previous stage to passive mode of freezing. Joining of individual ice-rock bodies into common ice-rock guard is carried our with predetermined term at the final stage of forming. EFFECT: increased safety in mining.
Patent RU-94042714-A (RU)
Inventor: SPRAVNIKOV E I
IPC: B61K9/06
Filed: 1994-12-02
Abstract: FIELD: railway transport; automatic car axle box heating control systems. SUBSTANCE: device can be used on cars with floor members on background of which axle boxes are inspected and on cars without floor members in axle box unit area (cars with defective bottoms, shortened base) in which axle box units are inspected on background of sky. Method of inspection comes to conversion of infrared radiation into electric heat signal with subsequent amplification of signal, limiting signal amplitude formed by getting of sky background into infrared radiation detector, setting zero potential directly before inspection of axle box unit, measuring excess of signal amplitude of axle box unit inspected on background of sky over limited amplitude of signal from sky background. Heating of axle box unit is judged by level of excess. Device has amplitude limiter whose input is connected with output of receiving capsule and output, with input of zero level detector. Amplitude limiter limits signal amplitude formed by sky background getting into infrared radiation detector. Follow-up amplitude limiter unit has limiter, series-connected amplifier, half-wave rectifier, analyzer, repeater and inverter. Inverter output is connected with control input of limiter, and amplifier output is connected with input of limiter. When inspecting axle box units on background of floor members, heat signal is not limited in amplitude limiter, and algorithm of operation of device is the same as in prototype. EFFECT: increased accuracy of determination of axle box unit heating temperature level.
Patent RU-94046285-A (RU)
Inventor: SHADKOVSKIJ STANISLAV
IPC: B22D41/24
Filed: 1993-05-27
Abstract: FIELD: foundry. SUBSTANCE: apparatus has immovable plate 8, movable plate 10 retained by carriage 9 and pouring pipe 2. Melt flow rate is controlled by sliding plate 10 relative to plate 8. Pouring pipe 2 is fixed in opposed relation with respect to movable plate 10 strictly below pouring opening 27 of plate 10, which covers pouring opening 15. Pipe 2 is fixed in above mentioned position by means of devices 31 for pushing it upward. Devices 31 are connected with carriage 9. EFFECT: increased efficiency, reduced consumption of melt, enhanced reliability in operation.
Patent RU-95101112-A (RU)
Inventor: BUSHMA V O
IPC: B23K9/173
Filed: 1995-01-26
Abstract: FIELD: welding technology; electric arc welding with stationary melting electrode. SUBSTANCE: method ensures stable welding process for lengthy articles of large thickness (in excess of 25 mm), and producing faultless weld seams. Inserted into clearance between articles to be welded together is melting electrode made in the form of a strip with dielectric coating applied to its opposite surfaces. Electrode and articles are connected to different poles of power source. Electric arc is ignited between electrode end face directed towards seam root and articles for welding. Electric arc is supplied with power from source having combined output volt-ampere characteristic. Arc is ignited at gently sloping section of output characteristic of power source with subsequent transfer within nominal welding currents to steep section of output characteristic. At location of arc from seam root at distance longer than 15-20 mm, welding is performed at slowly ascending section of output characteristic of power source. Welding electrode is connected to corresponding pole of power source at several points located at equal distance L, from each other over electrode length, and L, meets condition: L ≅ V x T, where V - welding speed, T - time required for heating material of melting electrode by welding current up to maximal preset temperature depending on temperature dependence of electrical strength of dielectric coating material. In process of arc moving relative to electrode melting front, changed smoothly or steplike is incline of gently sloping or gently ascending sections of power source output characteristic. EFFECT: high efficiency.
Patent RU-95102468-A (RU)
Inventor: GAZIZOV M G
IPC: B01D17/04
Filed: 1995-02-23
Abstract: FIELD: petroleum engineering. SUBSTANCE: part of gas-liquid stream is cut without completely closing stream. A sample is taken, which is subjected to automatically measuring water content and content of water isolated for a given time. Ratio of the latter to the total water content in emulsion is found as a measure of readiness of oil emulsion to be settled. EFFECT: provided automatic control of used demulsifiers and thereby reduced cost. 2 dwg
Patent RU-95105755-A (RU)
Inventor: MALAFEEV S I
IPC: H03F3/20
Filed: 1995-04-14
Abstract: FIELD: pulse device. SUBSTANCE: device has two resetting integrators 9 and 10 which operate in identical mode but in opposite phases. Each integrator operates in two cycles of equal duration which is equal to half of power supply period. During first half period of cycle control voltage is generated, during second one constant reference voltage is generated; sign of reference voltage is opposite to sign of control voltage. Said reference voltage is generated at output of gate 19 which transmission rate is controlled depending on voltage sign at outputs of integrators 9 and 10 in time moments which correspond to clock pulses. Output pulse is generated during second half period from its start until output voltage of integrator reaches level when comparator switches. During second half period integrators are reset to initial state. Sing-alternating sequences of control pulses for gates of bridge reversing power amplifier are generated at outputs of first and second OR gates 24 and 27. Duration of output sign-alternating pulses is varied in range from 0 for zero control signal to half of supply line period T/2 for maximal control signal. Polarity of control signal determines phase shift of output alternating voltage with respect to power supply voltage. EFFECT: increased stability to noise of pulse-width modulator which controls power amplifier. 3 dwg
Patent RU-95106289-A (RU)
Inventor: VORONOV V A
IPC: B03D1/06
Filed: 1995-04-24
Abstract: FIELD: automation of mineral concentration processes; may be used in control, regulation, monitoring of operation of flotation machine. SUBSTANCE: device has chamber of flotation machine with impeller and measuring member of air concentration in pulp. Measuring member is made in the form of two pairs of pipes located at different levels in flotation machine chamber. Ends of one pair of pipes are located in zone of aerated pulp, and ends of the other pair are located in zone of nonaerated pulp. Connected to indicated pipes are differential pressure gages whose electric leads are connected with division device connected to regulator whose output is connected with input of frequency converter connected to input of electric motor connected with impeller. EFFECT: improved conditions of flotation due to maintenance of preset aeration of pulp. 1 dwg
Patent RU-95106727-A (RU)
Inventor: AZARKOVICH A E
IPC: F42D99/00
Filed: 1995-04-26
Abstract: FIELD: excavation, explosions. SUBSTANCE: method for forming extended pits by excavation explosure includes drilling of vertical wells in lines, seating charges, setting firing pins, filling upper part of the well with stemming material, blasting circuit installation, and subsequent blasting. Borehole charge length is taken by the formula presented in the description. EFFECT: more correct size of pits.
Patent RU-95108898-A (RU)
Inventor: FILIMONOV V G
IPC: B23H7/16
Filed: 1995-05-31
Abstract: FIELD: electrophysical and electrochemical methods of treatment, production of apparatuses for protection of electrodes against short circuits during pulse-cyclical electrochemical treatment in particular. SUBSTANCE: aim is to increase reliability and to expand operational capabilities of apparatus for protection against short circuits. Aim is realized by solution of task of active and visual control after peak level of industrial electric current in conditions of its frequent interruptions in process of treatment and significant increase of absolute value of industrial current peak level to the end of treatment. To achieve the aim apparatus has two-step system of controlled peak detectors forming successively with help of control circuit current controlled signal and current reference signal with mode of its storing and also two controlled comparison devices, one of which operates in mode of tracking with running reference signal and another one operates with given reference signal in maximum current protection mode. Increased reliability of protection apparatus operation is achieved due to selective registration by peak detector of reference signal level in intervals between pulses of controlled signal and pulses of selectivity of comparison devices control and also due to duplication of operation of tracking channel of protection by channel of maximum current protection. Expansion of functional capabilities is achieved due to introduction of measurements of industrial current pulses registered peak values. EFFECT: increased reliability and expanded operational capabilities of apparatus for protection against short circuits.
Patent RU-95109751-A (RU)
Inventor: AL TSHUL R A
IPC: H02M7/757
Filed: 1995-06-13
Abstract: FIELD: converter substation for power lines and D C inserts, electrified railways, electric metallurgy and chemical industry. SUBSTANCE: each arm of two-valve bridges of twelve-phase inverted self-commutated converter includes two parallel circuits. Each circuit incorporates thyristor branch with turn-off thyristors placed in series and diode branch with diodes connected in series. One circuit starts in direction of conductance with thyristor branch and the other one, with diode branch. Capacitor is placed between centers of both circuits. Thanks to such manufacture of arms commutation of current in bridges occurs gradually without overvoltages which leads to increased reliability of converter. EFFECT: increased reliability of converter. 3 dwg
Patent TW-200301811-A (TW)
Title: Application of symbol sequence analysis and temporal irreversibility to monitoring and controlling boiler flames
Inventor: DAW CHARLES STUART
IPC: B01D1/00
Filed: 2002-11-14
Abstract: The current invention provides a method and apparatus, which uses symbol sequence techniques and/or temporal irreversibility derived from chaos theory to monitor the operating state of individual burner flames on a appropriate time scale. Both the method and apparatus of the present invention may be used optimize the performance of burner flames.