baber/WOPTO huggingface dataset:
Patent EC-SP11010843-A (EC)
Title: Compuestos de pirrolo-pirimidina como inhibidores de cdk
Inventor: BRAIN CHRISTOPHER THOMAS
IPC: A61K31/519
Filed: 2011-02-22
Abstract: Los compuestos que se dan a conocer se relacionan con tratamientos y terapias para trastornos asociados con la cinasa de proteína. También existe una necesidad de compuestos útiles en el tratamiento o la prevención o disminución de uno o más síntomas de cáncer, rechazo de trasplantes, y enfermedades autoinmunes. Adicionalmente, existe una necesidad de métodos para modular la actividad de las cinasas de proteína, tales como CDK1, CDK2, CDK4, CDK5, CDK6, CDK7, CDK8 y CDK9, utilizando los compuestos proporcionados en la presente.
Patent EC-SP12012083-A (EC)
Title: Pirrolidina-2-carboxamidas sustituidas
Inventor: BARTKOVITZ DAVID JOSEPH
IPC: C07D207/10
Filed: 2012-08-03
Abstract: Se proporcionan compuestos de la fórmula (consta gráfico) en la que X, Y, R1, R2, R3, R3, R4, R5, R6 y R7 tienen los significados aquí descritos y los enantiómeros y sales y ésteres farmacéuticamente aceptables de los mismos. Estos compuestos son útiles como agentes anticancerosos.
Patent EE-200000311-A (EE)
Inventor: JOHANSSON ANDERS
IPC: E04C2/08
Filed: 1998-06-26
Abstract: Panels for coffered ceilings comprising cladding panels of sheet metal or similar material and a method for mounting such panels. Each cladding panel comprises an essentially flat principal surface enclosed by longitudinally running joining sections as well as at least one longitudinally running stiffening section bent at an angle to the principal surface. The joining sections are designed so that any chosen panel can be removed simply and without the use of tools, so that a good seal is obtained between the panels, and so that it is possible to draw apart these to fit certain dimensions. In addition, the panels should hook into each other and remain sealed even if they should expand and buckle downwards due to fire or some other reason. According to the invention, this is solved by each of the joining sections of the panels being designed with a spacer section that ends in a hook-shaped section and that the spacer sections and the hook-shaped sections are designed so that they allow tightening and a certain displacement between the joining sections of close-by panels that overlap, and that the hook-shaped sections hook into each other first when the panels have been dawn apart a short distance from each other.
Patent EE-200300383-A (EE)
Inventor: RIELLO VALERIO GIORDANO
IPC: F24F1/00
Filed: 2001-03-20
Abstract: The present invention relates to an air-distribution cap which is to be fitted on top of a heating or air-conditioning unit with natural or forced convection and the function of which is to regulate both the flow-rate and the direction of the air output by the convector. In particular, the present invention relates to a cap ( 1 ) for distributing the air output by a heating or air-conditioning unit with forced convection or with natural convection, characterized in that it comprises a deflector ( 3, 103 ) having one or more vanes ( 13, 113 ), each vane being orientable so as to adopt a position in which it is inclined to the vertical so that its outer end faces towards the wall against which the unit is fitted.
Patent GB-189702410-A (GB)
Title: Improvements in Bottles, and in Stoppers and Caps therefor.
Inventor: MOORE ELISHA
Filed: 1897-01-29
Granted: 1897-05-29
Abstract: 2410. Moore, E., Moore, F., and Hay, A. W. Jan. 29. Stoppers; refilling, preventing ; stopper-keys.- Relates to stoppering bottles, so that, when once emptied, they cannot be refilled and restored to their original condition. In the form shown in Fig. 1, the neck of the bottle is contracted near the shoulder, and is closed at the contracted part by the ordinary stopper 3. Above this stopper is inserted a second stopper 6, which is locked in position by the arms 9 of the spring 8 engaging in recesses 5 in the neck. The bottle is opened by breaking the neck above the stopper 3, the neck being preferably weakened, as at 2, to facilitate breakage. In the form shown in Fig. 1<a>, the bottle is closed by an ordinary stopper 4 and by a cap 5, the cap being locked in position by the arms 10 of a bent spring engaging in notches 3 in the neck. The arms 10 are encircled by the hooked ends of a bail 12 mounted within the cap. The bottle is opened by breaking off the top of the cap at the groove 6, and drawing up the bail 12, the bail disengaging the arms 10 from the notches 3, so that the cylindrical portion of the cap and the bail can be removed to permit the withdrawal of the stopper 4.
Patent GB-189702840-A (GB)
Title: Improvements in and relating to Windows and Doors.
Inventor: KEITH DANIEL
Filed: 1897-02-03
Granted: 1898-01-29
Abstract: 2840. Keith, D. Feb. 3. Casement fasteners; latches.-The meeting-rails of double casement windows, which have to be raised slightly before being opened, have L-slotted plates screwed to them engaging with projections C' on the central vertical bar C as shown in Fig. 10. In cases when the upper and lower sashes can be connected, as shown in Fig. 11, the plate e<2> on the lower sash may have a latch e<4> engaging with a slotted plate e<5> on the window frame. In the case of hinged doors which can be raised and lowered to a limited extent for ventilating and other purposes, the latch bolt slides in a slotted striking- plate, which is also provided with two or more recesses for the lock bolt, so that the door can be latched and locked in the several positions.
Patent GB-189705294-A (GB)
Title: Improvements in and relating to Tea Kettles.
Inventor: SHARP FREDERICK
Filed: 1897-02-27
Granted: 1897-04-24
Abstract: 5294. Sharp, F., and Leigh, J. E. Feb. 27. Kettles.-A detachable shield a is provided to protect the hand from the steam escaping from the lid. Advertisements may be placed on the shield.
Patent GB-189705769-A (GB)
Title: Improvements in and relating to Pneumatic Tyres.
Inventor: JAMES WILLIAM HENRY
Filed: 1897-03-04
Granted: 1898-02-26
Abstract: 5769. James, W. H. March 4. Tyres, pneumatic.-The air tube A is formed with thickened abutting edges a', one of which is secured to the endless canvas band B, which has an edge b containing an inextensible core C. When the tyre is in position as in Fig. 1, the edges a' bear against the ring B, while the edges b of the latter engage with the recesses formed in the edges of the rim. Several modifications are described in which the band B may be attached to one or both sides of the ring, and in some cases the edges a' may interlock. In the example shown in Fig. 11, a ring B' of wedge-shaped section may be attached to the band B, which is secured to the rim by hooks c<1>.
Patent GB-189711461-A (GB)
Inventor: BURGESS CHARLES THOMAS
Filed: 1897-05-07
Granted: 1898-04-16
Abstract: 11,461. Burgess, C. T., and Burgess, W. B. May 7. Bicycles.-Relates to bicycles, the frames of which are formed from a strip of wood or other material. One end of the strip a starts from the plate e formed with the steering-socket and extends downwards and rearwards, the rearward portion being split to pass on each side of the wheel, the split parts being secured to the flanges b<1> of the bottom bracket b, and again to the brackets c which support the rear-wheel axle. The strip is then passed upwards, and forms a loop upon which is fixed the saddle-pin bracket d and is then made to lie in the hollow of the bracket b, whence it passes to the plate e. It may again be bent downwards and attached to the cup of the bracket b, whence it passes between the longitudinallydivided strips to which it is secured by the plate f so as to form a mud guard. The bracket b may be formed with bent plates b<3>, and stays g and h may also be added. The front and rear portions may be laced with wire to give increased strength, and also act as a dress guard. If the bicycle is for men, a stay may connect the upper parts of the loops. Modifications are described, in one of which an extra stay connects the steering-socket and bottom bracket and the arrangement of the frame is slightly varied, and in another both ends of the strip a are secured to the plate e and the form of the bracket b is modified.
Patent GB-189712260-A (GB)
Title: Improvements in Armoured Vessels.
Inventor: JOHNSON ELIAS MATTISON
Filed: 1897-05-18
Granted: 1897-09-25
Abstract: 12,260. Johnson, E. M. May 18. Drawings to Specification. War-ships are protected by means of two layers of armour with a space between them. The outer layer may consist of thin plates, while the inner layer may vary in thickness and has its outer surface hardened so as to break the points of projectiles which have penetrated the outer layer.
Patent GB-189721789-A (GB)
Title: An Improved Cycle Stand.
Inventor: EASEY ALFRED
Filed: 1897-09-23
Granted: 1897-12-11
Abstract: 21,789. Easey, A. Sept. 23. Stands for bicycles &c. A tube b rising from a base a contains a sliding rod e which carries at its upper end two horizontal sockets g containing sliding arms h, h<1>. The rod e may be raised in the tube b by a pivoted lever d engaging a pin d<2> moving in a slot b<1>. The rod may be fixed at any height by a pin e<2> engaging holes e<3> and resting on the top of the tube b. The rods h are adjusted in the sockets g to enable the curved ends h<1> to engage the members of the bicycle &c. frame. The cycle may be suspended by raising the rod e by means of the lever d. The ends h' and the tube b may be covered with leather &c. to prevent scratching.
Patent GB-189722702-A (GB)
Title: Improvements in Hollow Augers.
Inventor: BURDIN JOHN ROBERT
Filed: 1897-10-04
Granted: 1897-11-20
Abstract: 22,702. Burdin, J. R. Oct. 4. Augers, hollow. - Fig. 1 shows a plan, and Fig. 2 a sectional elevation of part of the tool. The end x of the spoke &c. s is turned down by a knife fixed to a jaw a which is pivoted at c to another jaw b. The jaws overlap one another at p, embrace the end x of the spoke, and are adjusted by nuts i on a curved rod g passing through lugs h, h, one pair of lugs being carried by each jaw. The jaws are attached to a brace &c. by a Y-shaped piece, the arms of which have lugs l, m for the screw c and the bolt n.
Patent GB-189724129-A (GB)
Title: Improvements in Electrical Transformers.
Filed: 1897-10-19
Granted: 1897-12-04
Abstract: 24,129. British Thomson-Houston Co., [Moody, W. S. Oct. 19. Transformers.- Relates to the ventilation or cooling and insulation of transformers intended for high voltages. The casing A is provided with openings B for the inspection of the terminals and with ledges B<1> for supporting the laminµ D. A passage E, fitted with a regulator F, is provided for allowing a current of air or other fluid to enter the chamber E<1>. whence it passes between the sections of the core to a chamber H having perforations in its casing. The primary and secondary coils P, S are so arranged that a current of air or other fluid may pass between them from the base A to a chamber beneath the cover K. In the arrangement shown in Fig. 3, the coils are placed within a casing L, so that they are isolated from the transverse ventilating-current. The primary coils N, preferably of flat wire, are wound in pairs separated by a thin insulation a. At the ends are fitted U-shaped insulating-pieces N, over which is fitted a layer of insulation c bound by tapes, s,pacing-pieces g being suitably arranged. The secondaries are arranged on the sides of the primary, from which they are thus efficiently insulated.
Patent GB-189724995-A (GB)
Title: A New Cloth.
Inventor: STRANG WILLIAM
Filed: 1897-10-28
Granted: 1898-03-05
Abstract: 24,995. Strang, W. Oct. 28. Striped fabrics.-Stripes of goffered, puckered, or crimped cloth are woven along with stripes of transparent or openwork cloth. The former stripes are produced by employing two warp beams, one tight and the other slack, and by inserting extra shots of weft, which are floated over the openwork stripes and afterwards cut off to leave these stripes clear.
Patent GB-189726841-A (GB)
Title: Improved Door Latch with Blocking Arrangement.
Inventor: GRIFFITHS THOMAS
Filed: 1897-11-17
Granted: 1898-10-01
Abstract: 26,841. Griffiths, T. Nov. 17. Latches.-The latch A, pivoted at B, is operated by a thumb lever in the usual way, the end D engaging a bevelled striking-plate on the door frame. The latch is blocked by sliding the piece E into a guide-plate, and blocking the end X of the latch, as shown by the dotted lines.
Patent GB-189801011-A (GB)
Title: Improvements in Holders or Sockets for Electric Incandescent Lamps.
Inventor: BOTT REUBEN JAMES
Filed: 1898-01-13
Granted: 1899-01-13
Abstract: 1011. Bott, R. J. Jan. 13. Incandescent lamps, holders for. A holder for a bayonetcapped lamp consists, in the form shown, of a casing 0 and a flanged insulator A connected by a screwed ring N, and carrying a detached sleeve B provided with diagonal slots, into which the pins on a lamp cap can be inserted in one movement. The sleeve is attached to the casing 0 by a tension spring D held by cross-pins which engage the insulator A and prevent rotation of the sleeve thereon. The lamp terminals bear on contact-pieces J, J<1> fixed in the insulator by screws which also hold the conducting-wires. The spring D allows the sleeve B to move away from the body of the holder when a lamp is inserted. In a modification, the spring is held compressed in a recess in the insulator by a cross-pin carried by lugs extending from the sleeve B within the holder.
Patent GB-189802640-A (GB)
Title: A Potato Gatherer and Cleaner.
Inventor: GIBBON JOHN
Filed: 1898-02-02
Granted: 1899-03-02
Abstract: 2640. Gibbon, J., and Read, T. Feb. 2. Potato diggers.-Relates to a machine for cutting the haulms and for digging and screening the potatoes. The haulm cutter consists of an axle A having four radial serrated. blades secured thereto and driven by the gearing shown from a gearwheel E secured to one of the main wheels D. B represents the digging-share suspended from the frame, and C, C an endless travelling screen formed of metal bars and driven from the wheel E.
Patent GB-189802712-A (GB)
Title: Improvements in Multiple Inkstands.
Inventor: ADAIR HENRY WILLIAM SHEFFIELD
Filed: 1898-02-02
Granted: 1898-03-19
Abstract: 2712. Adair, H. W. S. Feb. 2. Inkstands.-Relates to an arrangement for inkstands with several dipping-wheels, by which only one cover can be open at once. Fig. 2 shows the apparatus for a three-well inkstand, with one of the covers A' open. Each cover A<1>, A<2>, and A<3> is connected by a link to a sliding piece S<1>, S<2> or S<3>, having projecting pins S, S<1>, S<2>, S<3>, S<4> which actuate levers L, L<1>, L<2>, pivoted as shown, so that the raising of one lid causes the closing of all the others.
Patent GB-189803277-A (GB)
Title: An Improved Table for Use in Halls, Restaurants, and other places.
Inventor: CHRISTIE DAVID
Filed: 1898-02-09
Granted: 1898-12-10
Abstract: 3277. Christie, D. Feb. 9. Tables.-The top of a table for use in halls, restaurants, &c. consists of two leaves A hinged to a central part B supported on a leg C. Turnbuttons G keep the leaves in line, and prevent folding. The legs D are hinged at d, and are held extended by bolts with winged nuts engaging slotted plates E fixed to the leaves. Struts F hinged to the legs are held extended by hinged T-slotted bars f with which engage bolts with winged nuts on cross-bars of the legs D. Fig. 3 shows the table folded.
Patent GB-189803457-A (GB)
Title: Improvements in Boxes and Cases for Storing and Conveying Food Stuffs, such as Bottled Liquids, Fish, and the like.
Inventor: WILSON JOHN ALEXANDER
Filed: 1898-02-11
Granted: 1898-12-03
Abstract: 3457. Wilson, J. A. Feb. 11. Drawings to Specification. Packing-cases.-To facilitate cleaning, the bottoms of boxes for bottles &c., and the sides and bottoms of boxes for fish &c., are lined with tinned iron or other suitable metal. Openings are provided for cleansing.
Patent GB-189809315-A (GB)
Title: Improvements in Bicycles and the like.
Inventor: CLERICI GIULIO RUSCONI
Filed: 1898-04-22
Granted: 1899-02-25
Abstract: 9315. L a k e , H. H., [Clerici, G. R.]. April 22. Sociables; bicycles; convertibles. - Relates to means for converti n g an ordinary bicycle into a sociable. Fig. 2 shows a sectional front elevation of the sociable. A cross-bar D, carrying saddles E, E' at its ends, is fixed in the seat pillar. The cranks are replaced by arms of the form shown, each carrying a pair of pedals. The handle-bar is removed, and an arm F, Fig. 3, with or without a stay F<1>, is fixed to the head. Handle-bars G, G<1> are mounted in sockets on the ends of the arm F, and are connected to the steering-post by chains and chain-wheels H, H<1>, H<11>.
Patent GB-189810578-A (GB)
Title: Improvements in or relating to Cycle Stands.
Filed: 1898-05-09
Granted: 1899-03-11
Abstract: 10,578. Holmes &. Sons and Dix, W. J. May 9. Stands.-A cross-piece A, with hooked ends A' adapted to e-nbrace the frame as shown, is carried by a vertical rod B with feet B'. The stand keeps one wheel of the cycle off the ground. As shown, the front wheel is raised, but the stand may be tilted over so as to lift the rear wheel. The feet B' may be replaced by a cross-bar.
Patent GB-189813805-A (GB)
Title: Improvements in or relating to Pneumatic Actions for Mechanical Organs or the like.
Inventor: GAVIOLI ANSELME
Filed: 1898-06-21
Granted: 1899-05-06
Abstract: 13,805. Gavioli, A. June 21. Automatic instruments.-The invention relates to instruments operated by tune-sheets. The levers T have projections T' by which the tune-sheet actuates them, and are connected to valves l, by rods p. These valves are connected by other rods r to valves g situated in wind-chests, so that, when the valves l are closed, the valves g are opened, and vice versÔ. Both sets of valves are acted on by springs which tend to close them. When one of the levers T is raised, the corresponding valve l closes, and opens communication between one of the passages q and a passage o leading to a pneumatic which admits wind to the corresponding pipe. When the valve l opens again, the valve g closes, and the passage o is exhausted to the atmosphere. The wind-chests may be arranged in any manner, and are disposed so that dirt is prevented from reaching the valves.
Patent GB-189815714-A (GB)
Title: Improvements in Fluid Pressure Reducing Valves.
Inventor: MARTIN WILLIAM HAMILTON
Filed: 1898-07-18
Granted: 1899-05-20
Abstract: 15,714. Martin, W. H. July 18. Reducing - valves. -The valve 2, which slides between a seat 1<c> and a frame 3 the sides 3<a> of which are pressed against the seat by a spring 3<c>, is controlled by the tension of adjustable springs 8 and the fluid pressure in the outlet 1<b> on a plunger 5, the parts being connected together by a lever 7 and a link 4 as shown. The enlarged spindle or plunger 5 may be replaced by a piston working in a cylinder one end of which communicates with the valve outlet and the other end with the atmosphere, a condenser, or the like.
Patent GB-189816743-A (GB)
Title: Improvements in Keyless Locks.
Inventor: BRESLAUER EMIL
Filed: 1898-08-02
Granted: 1899-02-04
Abstract: 16,743. Breslauer, E. Aug. 2. Locks, permutation; padlocks.-The lock has a casing A with a dial on the outside. In the casing is mounted a notched wheel c, its spindle b with a pointer g being turned bya handle h. A tumbler e is pivoted in the casing, its barbed head e<1> being normally pressed into the path of the left jaw of a sliding locking-tongue d by a spring v. An adjustable spring yoke a is engaged in one of the wheel notches, so that, by correctly setting the pointer, the yoke is rotated to strike a pin p on the head e<1>, causing the latter to move exactly midway between the jaws of the tongue d, and allowing the tongue to be withdrawn from the casing and the door opened. An electric circuit k, l, m is connected to the tongue, the tumbler, and a pin n, so that, if the handle is turned too far or a premature attempt made to open the lock, an alarm is sounded. A spring tooth x may be provided to engage the tumbler head e<1> if moved too far and prevent further tampering. This tooth can only be re-set by someone on the inside. A spring f striking the teeth covers the noise made by the yoke striking the pin. A coiled spring normally moves the yoke away from the pin p. When the door is open the casing may be opened and the combination number varied by shifting the yoke. Fig. 6 shows a form to allow this to be done without opening the casing. The spindle has two oppositely-formed ratchet-wheels c, c' engaged by spring pawls r, t on arms a<1>, u<1>. The arm a<1> is frictionally mounted on the spindle, and the arm u<1> on a sleeve with an outside handle u. To open the lock, the pointer is placed at zero, and the handle u turned in the backward direction the same amount as is necessary to open the lock when the spindle is moved in the forward direction. The arm u is moved forward against a stop pin at zero rotating the spindle the required amount. When the door is open, a plunger q can be depressed into the path of the arm a<1>. To re-set the combination, the pointer is rotated backwardly till the arm a' is stopped by the depressed plunger. The pointer and spindle are then rotated to the desired opening number. The position of the plunger is preferably such that, in altering the opening number by turning the pointer backwards, the pointer always stands over the new opening number when its rotation is stopped. The zero position of the arm a<1> can also be obtained, when opening the lock without a pointer, by employing means such as are employed in stop-watches &c. to bring the indicator to zero. For instance, a snail cam on the spindle may be driven by a plunger on a spring arm connected to the arm u<1>. If desired, two or more tumblers and co-acting parts may be used. When applied to padlocks, the tongue d is formed on the end of the bow.
Patent GB-189822887-A (GB)
Title: Improvements in Arc Lamps.
Inventor: BARNIKOL-VEIT AUGUST BERNHARDT
Filed: 1898-10-31
Granted: 1899-03-04
Abstract: 22,887. B a r n i k o l - V e i t, A. B., and Riebel, A. W. Oct. 31. Arc lamps.-An escapement lamp has the gear frame N secured by pins and an angle-piece U between two links S, which are pivoted at i between two pillars B. The links S are made of copper or other material expansible by heat, and carry the armature A of the controlling-electromagnet M, so that any fall in the strength of field due to rise of temperature is compensated by the nearer approach of the armature to the pole-pieces C.