baber/WOPTO huggingface dataset:
Patent AT-E161251-T1 (AT)
Inventor: FLYNN GARY A
IPC: C07C211/40
Filed: 1994-10-20
Granted: 1998-01-15
Abstract: The present invention relates to a novel enantiospecific process for preparing (S)-1-[2(S)-(1,3-dihydro-1,3-dioxo-isoindo-2-yl)-1-oxo-3-phenylpropyl ]-1,2,3,4-tetrahydro-2-pyridine-carboxylic acid methyl ester which is a useful intermediate in the preparation of [4S-[4 alpha , 7 alpha (R*), 12b beta ]]-7-[(1-oxo-2(S)-thio-3-phenylpropyl) amino]-1,2,3,4,6,7,8,12b-octahydro-6-oxo-pyrido[2,1-a][2]benzazepine-4-carboxylic acid and [4S-[4 alpha , 7 alpha (R*), 12b beta ]]-7-[(1-oxo-2(S)-acetylthio-3-phenylpropyl)amino]-1,2,3,4,6,7,8,12b-octahydro-6-oxo-pyrido[2,1-a][2]benzazepine-4-carboxylic acid and pharmaceutically acceptable salts thereof which is useful as an inhibitor of enkephali nase and angiotensin converting enzyme and to novel intermediates thereof.
Patent AT-E165414-T1 (AT)
Inventor: OESTERLE HELMUT
IPC: E04D3/36
Filed: 1994-12-05
Granted: 1998-05-15
Abstract: A large-surface plain washer (1) has an opening (5) for inserting a fastener. Engagement elements (1) that increase the engagement with a plate and/r web to be fastened are provided at the surface of the washer (1) that faces in the fastening direction. In addition, projecting spacers (17) shaped as tongues (26) that become effective when several washers (1) are stacked are provided at the lower side of the washer (1). The free end of these tongues (26) may be supported on the top side of the plain washer located directly underneath, so that the washers may be stacked without causing the engagement elements (13) of different washers (1) to engage each other. Individual washers (1) may thus be easily separated from a stack of washers (1), either by rotating or by moving the lowermost washer.
Patent AT-E165020-T1 (AT)
Inventor: ULLRICH JUERGEN
IPC: A63G1/12
Filed: 1995-01-31
Granted: 1998-05-15
Abstract: PCT No. PCT/EP95/00339 Sec. 371 Date Sep. 4, 1996 Sec. 102(e) Date Sep. 4, 1996 PCT Filed Jan. 31, 1995 PCT Pub. No. WO95/20426 PCT Pub. Date Aug. 3, 1995The present invention relates to a carousel for people, especially children, with a substructure that is stationary relative to the ground and that has a stator axle essentially perpendicular to the ground and a radial support star essentially parallel to the ground, and with a rotor being rotatable about the stator axle and having a turning section for carrying people. To create a carousel of this type that is easy to operate and versatile and that affords adequate safety even when used improperly, the invention proposes that the radial support star should be located on a profiled ground plate in recesses thereof that essentially conform to the shape of the radial support star, and that the radial support star or ground plate has provided thereon a central centering shoulder aligned to engage in a central receiving portion provided on the respectively other member.
Patent AT-E177944-T1 (AT)
Inventor: NORLING TOMAS
IPC: A61K9/00
Filed: 1995-06-14
Granted: 1999-04-15
Abstract: A novel drug delivery system, e.g. in the form of a solid dosage form or a liquid formulation based on a pharmaceutical multiple unit in the form of cores such as, e.g., coated cores. The pharmaceutical formulations are based on a novel principle allowing preparation of cores such as, e.g., cores in the form of pellets, i.e. substantially spheric particles which have such a mechanical strength (expressed in terms of friability) that the cores are sufficiently robust to substantially remain intact after having been subjected to coating by standard pharmaceutical procedures well known by a person skilled in the art such as, e.g., a coating process involving a fluidized bed process. A spray-drying process for the preparation of the pharmaceutical formulation is also described.
Patent AT-E174751-T1 (AT)
Inventor: VON ALLWOERDEN WILHELM
IPC: A01D43/00
Filed: 1995-09-02
Granted: 1999-01-15
Abstract: A self-propelled harvester with a harvest distributor is disclosed. A self-propelled harvester, in particular for green fodder, has a cutting device (2) for cutting the harvest, a conveyor (4) for conveying the harvest, a processing device (5.1, 5.2) for processing the harvest, a pressing device (7) for pressing the harvest into mats and a depositing device (8) for depositing the mats on the fields. In order to ensure a trouble-free passage of the harvest through the individual devices of the harvester, and to improve or increase its capacity in comparison with known state-of-the-art harvesters, the pressing device is directly arranged behind the processing device, dispensing with a dosing device.
Patent AT-E183237-T1 (AT)
Inventor: KLASEN RALF
IPC: C12N1/21
Filed: 1996-02-07
Granted: 1999-08-15
Abstract: Prodn. of 5-ketogluconate (I), comprises increasing the expression of the gluconate:NADP<+>-5-oxidoreductase (A) gene. Also new are: (1) Gluconobacter oxydans (A) gene (the 1512 bp nucleic acid sequence of which, and the 256 residue amino acid sequence encoded by it, are given in the specification), including its allelic variants; (2) gene structures and vectors contg. the gene of (1); and (3) transformed cells contg. the gene of (1), or the gene structures or vector of (2).
Patent AT-E197145-T1 (AT)
Inventor: HOECHSTETTER CRAIG S
IPC: A61K31/42
Filed: 1992-02-03
Granted: 2000-11-15
Abstract: Isoxazole derivs. of formula (I) and their acid-addn. salts and solvates are new: In (I) R = 1-4C alkyl, allyl or cyclopropylmethyl; R1 = H, 1-4C alkyl, allyl, cyclopropylmethyl or aryl(1-4C)alkyl; X = CH2 or O; y = 4-R2-5-R3-3-isoxazolyl or 3-R2-4-R3-5-isoxazolyl; R2 and R3 = H, 1-4C alkyl, 1-4C alkoxy, 1-4C alkylthio, OH, NH2, CN or Ph. Pref. x = CH2; R and R1 = 1-4C alkyl, esp. n-Pr; R2 and R3 = H.
Patent AT-E261960-T1 (AT)
Inventor: NAKAE TAKAHIKO
IPC: C07C311/29
Filed: 1996-09-27
Granted: 2004-04-15
Abstract: Sulfonamide derivatives of the formula (I) <CHEM> wherein R<1> is, inter alia, alkyl, alkoxy, hydroxy, keto, nitro, halogen, trihalomethyl, cyano, amidino and -COOR<7> (in which R<7> is hydrogen or alkyl),  n is an integer from 0 to 5; <CHEM>  is a carbocyclic ring or heterocyclic ring; <CHEM> in which R<2> and R<3> each is hydrogen, alkyl, alkoxy, halogen, trihalomethyl or phenyl, or  R<2> and R<3>, taken together, represent alkylidene, or <CHEM> in which R<2> and R<3>, taken together with the carbon atom to which they are attached represent cycloalkyl; R<4> is alkyl or alkoxy or two of R<4>, attached to the benzene nucleus at ortho positions relative to each other, taken together, represent alkylene; m is an integer from 0 to 4; and <CHEM> is optionally substituted amino or a nitrogen-containing ring, are described as new pharmaceutical compounds having inhibitory activity or elastase.
Patent AT-E230017-T1 (AT)
Inventor: BRAVO ADRIANA
IPC: C12C5/00
Filed: 1996-10-28
Granted: 2003-01-15
Abstract: The present invention is directed to a method for stabilizing the flavor of a fermented malt beverage, most particularly a beer, by the addition of an oxoaldehyde reductase enzyme, the fermented malt beverage prepared by such a method, and to the use during the brewing process of oxoaldehyde reductase enzymes from naturally occuring sources, including those produced by yeasts, to stabilize the flavor of the resulting beer product and to produce a beer having a stable flavor. The invention also relates to microorganisms, particularly yeasts, which have been specifically modified, selected, or genetically engineered to express or secrete an oxoaldehyde reductase enzyme which may be used during the brewing process to stabilize the flavor of the resulting beer product and to produce a beer having a stable flavor. The present invention also provides extracts from a naturally occuring source (e.g., yeast), or a modified yeast or extract thereof, which will provide a sufficient amount of the necessary enzymes to block, inhibit or reduce the Maillard reaction intermediates (e.g., 3-deoxyglucosone), which result in the formation of the stale flavor in fermented malt beverages. In addition, the present invention provides fermented malt beverages having enhanced flavor stability produced by these methods.
Patent AT-E266852-T1 (AT)
Inventor: AMOROSI STEFANO
IPC: G01B11/00
Filed: 1996-12-31
Granted: 2004-05-15
Abstract: The process uses information from the scan sweeps of a laser scanner, and readings with a CCD reader, to obtain a series of stipulated areas corresponding to successive cross-sections of the object as reckoned by moving the object relative to the scanner and the reader. The volume is then obtained by multiplying each of said areas by the feed distance of the object. The possibility is further contemplated of accommodating the slope angles of the scan plane and the read plane, or alternatively neglecting their effects if said angles are sufficiently small. The volume measurement may be accompanied by the reading of an optical code provided on the object. <IMAGE>
Patent AT-E216590-T1 (AT)
Inventor: WARNE NICHOLAS W
IPC: A61K47/12
Filed: 1996-02-02
Granted: 2002-05-15
Abstract: Provided by the present invention are novel compositions and methods for obtaining concentrated preparations of IL-12 and formulations of IL-12 suitable for storage and administration.
Patent AT-E200942-T1 (AT)
Inventor: LEWIN ROBERT GLYN
IPC: H01M4/86
Filed: 1996-03-18
Granted: 2001-05-15
Abstract: PCT No. PCT/GB96/00639 Sec. 371 Date Jan. 19, 1998 Sec. 102(e) Date Jan. 19, 1998 PCT Filed Mar. 18, 1996 PCT Pub. No. WO96/28856 PCT Pub. Date Sep. 19, 1996A solid oxide fuel cell and method of production are provided. The cell may have a layer of electrolyte material and a first and second electrode on either side thereof. The electrodes are separated from electrolyte by separator layers which are a mixed conductor. The fuel sell may be used in a stack.
Patent AT-E260107-T1 (AT)
Inventor: CHIPMAN STEWART
IPC: C07D487/04
Filed: 1996-06-05
Granted: 2004-03-15
Abstract: Disclosed is a method of treating osteoarthritis. The method comprises administering a therapeutic amount of debromohymenialdisine to an individual or animal with osteoarthritis. Debromohymenialdisine is able to slow the joint deterioration and cartilage degradation associated with the disease.
Patent AT-E265878-T1 (AT)
Inventor: GIERVELD JOHAN
IPC: A63C1/00
Filed: 1996-05-24
Granted: 2004-05-15
Abstract: PCT No. PCT/NL96/00209 Sec. 371 Date Mar. 12, 1998 Sec. 102(e) Date Mar. 12, 1998 PCT Filed May 24, 1996 PCT Pub. No. WO96/37269 PCT Pub. Date Nov. 28, 1996The invention relates to a frame for a sporting device for coupling to a shoe, such as a ski which is slidable or rollable by means of wheels, in particular a cross-country ski, or a skate frame for an ice-skate or roller-skate, which frame comprises: an upper sub-frame with means for coupling to a shoe to be worn by a user, a lower sub-frame which is coupled via a pivot mechanism to said upper sub-frame for pivoting in a main plane and which is provided with or adapted to be provided with a runner or wheels; and a resetting spring for urging both sub-frames toward each other. The frame according to the invention has the special feature that the sub-frames are mutually pivotable and translatable in the said main plane. A specific embodiment has the feature that the sub-frames form part of a mechanism comprising at least four mutually pivotable and/or translatable rods.
Patent AT-E227885-T1 (AT)
Inventor: SCHELLENBERGER WILHELM
IPC: H01L21/304
Filed: 1996-08-09
Granted: 2002-11-15
Abstract: A method of drying a substrate surface (1), comprising:   dipping the substrate into a liquid bath (2); separating the substrate from the liquid bath (2), whereby the liquid of the liquid bath (2) comprises an aqueous HF solution (3), the substrate surface being hydrophobic upon separation from the liquid bath, the substrate being separated from the bath at a rate that permits the bath liquid to drain from the hydrophobic surface of the substrate to produce a dry substrate; and that a gas comprising an O2/O3 mixture that forms a hydrophilic surface on the substrate is directed over the surface of the substrate (1) after separating the substrate (1) from the liquid bath.   <IMAGE>
Patent AT-E257469-T1 (AT)
Inventor: WEHRLI CHRISTOF
IPC: C07D489/00
Filed: 1997-09-26
Granted: 2004-01-15
Abstract: (Z)-1[1-(4-Methoxybenzylidene)-1,2,3,4,5,6,7,8-octahydro-isoquinolin-2-yl]alkanones of the formula  produced under specific reaction conditions in a one-pot process in an advantageous manner by a Bischler-Napieralski cyclization of N-(2-cyclohex-1-enylethyl)-2-(4-methoxyphenyl)-acetamide and subsequent lower-alkanoylation of the resulting 1-(4-methoxybenzyl)-3,4,5,6,7,8-hexahydro-isoquinoline of the formula    <IMAGE>  III  under an inert gas atmosphere and, if desired converted to dextomethorphan in a known manner.
Patent AT-E202680-T1 (AT)
Inventor: PAVELESCU LIVIU-MIHAI
IPC: A43B7/12
Filed: 1997-01-08
Granted: 2001-07-15
Abstract: PCT No. PCT/EP97/00042 Sec. 371 Date Aug. 4, 1998 Sec. 102(e) Date Aug. 4, 1998 PCT Filed Jan. 8, 1997 PCT Pub. No. WO97/24940 PCT Pub. Date Jul. 17, 1997A waterproof shoe structure including at least part of a shoe, has an outer layer, a lining including a functional layer that is waterproof but permeable to water vapor, an insole, and an outsole. The lining containing the functional layer has a lower end area that is turned in and arranged parallel to the outsole, the turned-in end area lies in a common plane with the insole and has an inner edge and an outer edge, the outer edge of the insole runs at least approximately parallel to the inner edge of the turned-in end area, and the insole is joined to the turned-in end area. The outsole is applied by adhesive over a full surface thereof at least to the turned-in end area of the functional layer of the lining, and the lower end of the upper layer is arranged substantially perpendicular to the outsole and at least in a shank area thereof is joined to a retainer arranged parallel to the outsole, and/or at least in a toe area thereof a netting of monofilaments is joined to the lower end of the outer layer. The lining inside the outer layer is arranged in a detached manner.
Patent AT-E393182-T1 (AT)
Inventor: KITAHARA SHIZUO
IPC: C08F283/01
Filed: 1997-03-07
Granted: 2008-05-15
Abstract: An unsaturated polyester (i) having a weight-average molecular weight (Mw) of 1,000-100,000 and at least two carbon-carbon unsaturated bonds in the molecule thereof obtained by esterifying an unsaturated carboxylic acid (b) with a polyester-polyol (a) obtained by subjecting a polybasic carboxylic acid containing polymerized fatty acid and/or polymerize fatty acid ester to polycondensation with a polyhydric alcohol; and an unsaturated (poly)urethane having Mw of 1,000-100,000 and at least two carbon-carbon unsaturated bonds in molecule obtained by reacting said polyester-polyol (a), polyisocyanate (d) and compound (e) having active hydrogen and polymerizable carbon-carbon unsaturated bond. Said unsaturated polyester and unsaturated (poly)urethane exhibit excellent adhesive property, heat resistance, water resistance and flexibility after being cured.
Patent AT-E198237-T1 (AT)
Inventor: SMYERS SCOTT D
IPC: H04L29/10
Filed: 1997-02-19
Granted: 2001-01-15
Abstract: An asynchronous data pipe (ADP) automatically generates transactions necessary to complete asynchronous data transfer operations for an application over a bus structure. The ADP includes a register file which is programmed and initiated by the application. The register file includes the bus speed, transaction label, transaction code, destination node identifier, destination offset address, length of each data packet, packet counter, packet counter bump field, control field and a status field. During a data transfer operation, the ADP generates the transactions necessary to complete the operation over the appropriate range of addresses, using the information in the register file as a template. The ADP increments the value in the destination offset address field for each transaction according to the length of each data packet, unless the incrementing feature has been disabled and the transactions are to take place at a fixed address. The packet counter represents the number of transactions remaining to be generated. The packet counter value is decremented after each packet of data is transferred. The application can increment the packet counter value by writing to the packet counter bump field. A multiplexer is included within a system having multiple ADPs for multiplexing the information from the ADPs onto the bus structure. A demultiplexer is included within a system having multiple ADPs for routing information from the bus structure to the appropriate ADP.
Patent AT-E208053-T1 (AT)
Inventor: ISLER DANIEL
IPC: F27B21/14
Filed: 1997-05-23
Granted: 2001-11-15
Abstract: PCT No. PCT/FR97/00902 Sec. 371 Date Nov. 16, 1998 Sec. 102(e) Date Nov. 16, 1998 PCT Filed May 23, 1997 PCT Pub. No. WO97/45761 PCT Pub. Date Dec. 4, 1997An endoscopic probe includes an inspection head attached to the end of a longitudinally flexible supporting line which connects it to an operating unit provided with means for moistening the line. The supporting line (2) is rigid under axial torsion, whilst the inspection head (1) is movable in axial rotation and is formed by a demountable assemblage of two parts: a permanent part (11), attached to the end of the supporting line by means of a rotary joint (10) and housing a miniaturized photography device (26), and an interchangeable part (12), fastened rigidly to said permanent part in the extension of the latter with the aid of a demountable joint (44) and comprising a parietal (lateral or axial) orifice provided with a wide angle ocular lens (23) followed by an optical line (25) for conveying the light energy picked up by said lens toward the photography device (26). A motor system and encoder (32 to 36) are mounted in the probe for motorizing the axial rotation of the inspection head and ensuring adjustment of its angular position in relation to the supporting line. The endoscopic probe is suitable for the visual inspection of the flues of coke ovens.
Patent AT-E216435-T1 (AT)
Inventor: PETERS CHRISTOPHER THOMAS
IPC: C22C26/00
Filed: 1997-09-01
Granted: 2002-05-15
Abstract: A method of manufacturing a metal bonded abrasive product such as a saw or drill segment or bead for a diamond wire is provided. The method includes the steps of providing a mixture of the metal, in particulate form, and the abrasive particles, cold pressing the mixture to the desired final shape at a pressure in the range 320 to 1500 MPa to produce a cold pressed product at a temperature in the range 900 to 1300 DEG  C. under conditions which inhibit degradation of the abrasive particles and the particulate metal. The product, after free sintering, will generally have a relatively high porosity, for example, a porosity of 10 to 25 percent by volume.
Patent AT-E210227-T1 (AT)
Inventor: ZUERBES ARNO DR-ING
IPC: E01C19/34
Filed: 1998-01-22
Granted: 2001-12-15
Abstract: The appliance has an integral drive (3) and a guide bracket (6) with a grip end for an operator. Mass distribution of the bracket results in vibration reduction at the bracket grip end (9). Bracket geometry and mass distribution are satisfied according to:- Hs divided by ms(lhg x lh - lv x lv) = 0.8 - 1.3 ms = mass of the guide bracket; Hs = mass moment of inertia of the bracket about an axis through the centre of gravity (10) of the bracket, which is parallel to an axis through the hinge points (8); lh = distance at right angles to tamper axis (A), between centre of gravity and axis through hinge points; lhg = distance at right angles to tamper axis, between grip end and centre of gravity; lv = distance parallel to the tamper axis, between centre of gravity and axis through hinge points. The ratio for weight distribution is approx. between 0.9 and 1.3, esp. between 1.0 and 1.15. For this purpose, the bracket has a weight.
Patent AT-E280778-T1 (AT)
Inventor: ERNI BERNHARD
IPC: C12N9/99
Filed: 1998-02-02
Granted: 2004-11-15
Abstract: The bacterial phosphotransferase system (PTS) as a drug target system catalyses the uptake and phosphorylation of carbohydrates. It is further involved in signal transduction, e.g. catabolite repression, chemotaxis, and allosteric regulation of metabolic enzymes and transporters. It is ubiquitous in bacteria but does not occur in eukaryotes. This uniqueness and the pleiotropic function make the PTS a target for the development of new antimicrobials. Assays are described that lead to the discovery of compounds which uncouple the PTS, by acting as protein histidine/cysteine phosphatases. Uncoupling of the PTS leads to inhibition of carbohydrate transport, repression of catabolite controlled genes (e.g. certain virulence genes) and depletion of phosphoenolpyruvate. Compounds from combinatorial libraries with high affinity for phosphoenolpyruvate-protein-phosphatase (Enzyme 1) serve as lead structures for the development of inhibitors and uncouplers of the PTS.
Patent AT-E219539-T1 (AT)
Inventor: KRAEMER BERTHOLD
IPC: D21F5/02
Filed: 1998-04-01
Granted: 2002-07-15
Abstract: The heat exchanger, especially for a heated roller, is operated by steam with a feed channel (7) and a channel (8) to extract the condensation. When using a heating fluid, the condensation channel (8) is used for its outflow. The feed and outlet channels lead to a valve (9) so that, under pressure in the feed channel (7), the outflow channel (8) is blocked so that only condensation and/or slip steam is fed through the outlet (18) of the outflow channel (8). On pressure in the outflow channel (8), it opens into a build-up zone (14). The feed channel (7) is linked to the valve (9) through the heating circuit of the heat exchanger, and the outflow channel (8) leads directly to the valve (9). The valve is a non-return valve (9), with a valve body (15) expanding in a slight cone shape into a feed zone in the lifting direction. It has a pot shape, with a conical pot base towards the outflow channel (8). The valve body (15) is of a plastics material with a low specific gravity, and pref. ≤ 7.85 g/cm<3>, and is resistant to corrosion. The feed zone material or its coating has the same thermal coefficient of expansion as the valve body (15). The feed zone has a limit stop (19) to define the stroke movement of the valve body (15). The dimensions of the moving parts of the valve allow their movement through the feed channel (7) for exchange and/or repair.
Patent AT-E402151-T1 (AT)
Inventor: BLEY KEITH ROGER
IPC: A61K31/41
Filed: 1998-08-26
Granted: 2008-08-15
Abstract: The invention relates to IP receptor antagonists selected from the group of compounds represented by formula <CHEM>  wherein     R<1> is a group represented by formula (A), (B) or (C): <CHEM> and other substituents as defined in the specification, and their pharmaceutically acceptable salts, crystal forms therof and pharmaceutical compositions containing them.