baber/WOPTO huggingface dataset:
Patent CZ-20002818-A3 (CZ)
Title: Synthetic taxol analogs and process of their preparation
Inventor: VANEK TOMAS RNDR CSC
IPC: A61K31/337
Filed: 2000-08-02
Abstract: In the present invention, there are disclosed taxol synthetic analogs of the general formula II, in which x is 1 or 2 and Y represents COCHi2Cl or COCHi2Br, Ac denotes an acetyl group and Bz represents a benzoyl group. These compounds are prepared so that taxol of the general formula I is treated with a modified amino acid of the general formula III in a solvent such as dichloromethane or  dimethylformamide in the presence of coupling agents and tertiary amines and dimethyl aminopyridine.
Patent CZ-20021010-A3 (CZ)
Title: Novel quinazoline compounds and pharmaceutical preparations in which they are comprised
Inventor: MORTLOCK ANDREW AUSTEN
IPC: C07D239/88
Filed: 2000-09-18
Abstract: The use of a compound of formula (I) or a salt, ester or amide thereof; where X is O, or S, S(O) or S(O)2, NH or NR<8> where R<8> is hydrogen or C1-6alkyl; R<a> is a 3-quinoline group or a group of sub-formula (i) where R<5>, R<6> and R<7> are various specific organic groups, in the preparation of a medicament for use in the inhibition of aurora 2 kinase. Novel compounds of formula (I) and pharmaceutical compositions useful in the treatment of cancer are also described and claimed.
Patent CZ-20021675-A3 (CZ)
Title: Beam of high-temperature superconducting rotor coil and the coil carrying method
Inventor: WANG YU
IPC: H02K9/19
Filed: 2002-05-14
Abstract: A rotor for a synchronous machine is disclosed comprising: a rotor core (22); a super-conducting coil winding (34) extending around at least a portion of the rotor core, said coil winding having a coil end section (54) adjacent an end (56) of said rotor core, and a coil support (58) bracing said end section and being thermally isolated from said rotor core. <IMAGE>
Patent CZ-20022628-A3 (CZ)
Title: Substituted piperidines, process of their preparation and pharmaceutical preparation in which the compounds are comprised
Inventor: RUDOLF KLAUS
IPC: A61K31/496
Filed: 2000-12-22
Abstract: The invention relates to substituted piperdines of general formula (I) in which A<1>, A<2>, R, R<1> and R<2> are defined as in Claim No. 1, to their tautomers, diastereomers, enantiomers, mixtures, and to their salts, in particular, their physiologically compatible salts with inorganic or organic acids or bases, which comprise valuable pharmacological properties, in particular, CGRP-antagonistic properties. The invention also relates to medicaments containing these compounds, to their use and to methods for the production thereof.
Patent CZ-20022826-A3 (CZ)
Title: Pluraflavins and derivatives thereof, process for their preparation and use thereof
Inventor: VERTESY LASZLO
IPC: A61P11/00
Filed: 2001-02-15
Abstract: The invention relates to a compound of formula (I) wherein R1 is a sugar; R2 is -CH2-O-(R7)m, R7 representing a sugar, or R2 is -COOH; R3 is an epoxide-comprising group, C1-C6-alkyl or C2-C6-alkenyl, unsubstituted or substituted by at least one OH; R5 is H, C1-C6-alkyl, C2-C6-alkenyl or C2-C6-alkynyl; R4, R6, R8 and R10 independently of one another are H,C1-C6-alkyl, C2-C6-alkenyl, C2-C6-Alkynyl, -X2H, or -X2R12, or R4 and R6 together and/or R8 and R10 together are =X2; X2 is O, NH, N-C1-C6-alkyl, N-C2-C6-alkenyl, N-C2-C6-alkynyl or S; R12 is C1-C6-Alkenyl, C2-C6-alkynyl, C2-C6-alkynyl, aryl or acyl; and m and n are 1 or 2; and its physiologically acceptable salts. The compounds are obtainable from a culture of the microorganism Actinomycetales species HAG 003959, DSM 12931, by fermentation. Accordingly, the invention relates to a process for their preparation and to the use of the compounds as pharmaceuticals, for example as anti-tumor agents.
Patent CZ-20023306-A3 (CZ)
Title: Electric machine
Inventor: SADARANGANI CHANDUR
IPC: F02B1/12
Filed: 2001-04-06
Abstract: An electrical machine with at least a machine unit. The machine unit includes a stator, which includes a plurality of magnetic flux conductors and an electric conductor forming a winding extending in a substantially closed winding path through each magnetic flux conductor, and a movable element, which includes permanent magnet elements movable in a reciprocating movement in relation to the stator along a movement path. The winding path includes a first current carrying portion, which extends substantially in parallel with the movement path. Each magnetic flux conductor is arranged to form, together with one of the permanent magnet elements, a closed magnetic flux circuit extending around the current carrying portion. The magnetic flux conductors are arranged in an alternating order with respect to the direction of the magnetic flux in relation to the permanent magnet elements in the respective magnetic flux circuit.
Patent CZ-20031479-A3 (CZ)
Title: Sealing ring
Inventor: STADLER ROLF
IPC: F16J15/3284
Filed: 2002-06-14
Abstract: The invention relates to a sealing ring comprising a bearing ring (1), which is connected to a lip ring (2) made of an elastomer material.  Said bearing ring (1) is made from a reinforced fibrous material or wood.
Patent CZ-20031981-A3 (CZ)
Title: Bone implant, in particular, an inter-vertebral implant
Inventor: MATHYS ROBERT JR
IPC: A61F2/44
Filed: 2001-01-30
Abstract: The inter-vertebral implant is made from a radiation-transparent material and embodied as an annular hollow body (1). Said implant comprises a sleeve (6) in the form of a hollow cylindrical section, comprising a front (9), a rear (10) and two lateral sections (11) and defines a cylindrical axis (7). The hollow body (1) is divided by two intermediate walls (3), running essentially parallel to the cylinder axis (7) and connecting the front section (9) with the rear section (10) of the sleeve. The surface (2) of the bone implant comprises a surface roughness of at least 2  mu m. This surface roughness permits the newly growing bone a better fixation to the implant, in other words a better bone integration.
Patent CZ-20033331-A3 (CZ)
Title: Integrated memory controller circuit for fiber optics transceiver
Inventor: ARONSON LEWIS B
IPC: H01S5/042
Filed: 2002-02-04
Abstract: A controller (110) for controlling a transceiver having a laser transmitter and a photodiode receiver. The controller includes memory (120, 122, 128) for storing information related to the transceiver, and analog to digital conversion circuitry (127) for receiving a plurality of analog signals from the laser transmitter and photodiode receiver, converting the received analog signals into digital values, and storing the digital values in predefined locations within the memory. Comparison logic (131) compares one or more of these digital values with limit values, generates flag values based on the comparisons, and stores the flag values in predefined locations within the memory. Control circuitry (123-1, 123-2) in the controller controls the operation of the laser transmitter in accordance with one or more values stored in the memory. A serial interface (121) is provided to enable a host device to read from and write to locations within the memory. Excluding a small number of binary input and output signals, all control and monitoring functions of the transceiver are mapped to unique memory mapped locations within the controller. A plurality of the control functions and a plurality of the monitoring functions of the controller are exercised by a host computer by accessing corresponding memory mapped locations within the controller.
Patent CZ-200897-A3 (CZ)
Inventor: HRABAL FRANTISEK
IPC: B60C23/00
Filed: 2008-02-21
Abstract: Vynález se týká zarízení pro úpravu tlaku v pneumatikách, sestávajícího z komory (K) s tvarovou pametí a ventilu (V). Ventil (V) je trícestný, se vstupy propojenými s vnejším okolím (O) a vnitrním prostorem (P) pneumatiky, pricemž jeden vstup (V1) je opatren ventilem (JV), další vstup (V2) je pripojen k jednomu konci tvarové komory (K) a poslední vstup (V3) je propojen s uzavíracím prvkem (R).
Patent DD-235795-A3 (DD)
Title: Verfahren zur herstellung von vinylacetat aus acetylen und essigsaeure
Inventor: ADLER ROLAND
IPC: C07C69/15
Filed: 1980-08-01
Abstract: Vinylacetat wird aus Acetylen und Essigsaeure in der Dampfphase in Gegenwart fester, relativ rasch alternder Vinylacetatkatalysatoren in gekuehlten Lamellen- oder Rohrbuendelreaktoren, denen nach neuen Erkenntnissen adiabat betriebene Katalysatorschichten vorgeschaltet sind, bei geringfuegigem Ueberdruck hergestellt. Das Ziel der Erfindung besteht darin, die Bedingungen herauszufinden, bei denen das verschaltete System im gesamten Betriebszyklus reaktionstechnisch stabil betrieben werden kann, ohne dass man zwischen beiden Reaktoren Umsaetze bestimmen muss. Erfindungsgemaess wird dieses durch die Vorgabe von maximal zulaessigen Temperaturen in Abhaengigkeit von Aktivitaetszustand des Katalysators und eine separate Steuerung des gekuehlten und adiabaten Reaktors geloest. Dabei ist es wichtig, zunaechst die Kuehlmitteltemperatur im gekuehlten Reaktor und nach Erreichung des stationaeren Zustandes die Gaseintrittstemperatur im adiabaten Vorreaktor zu erhoehen. Dieses Verfahren ist fuer jede Katalysatorqualitaet anwendbar, wenn fuer die Einfuellmasse der adiabaten Katalysatorschuettschicht die angegebenen Vorgaben beachtet werden. Es ist ausserdem moeglich, im adiabaten Vorreaktor Katalysatoren geminderter Qualitaet, wie beispielsweise regenerierte Katalysatoren, ohne Produktionseinbussen einzusetzen.
Patent DD-218785-A3 (DD)
Title: Anordnung zur sicherung der achsmittigen lage von dampfturbinengehaeusen
Inventor: BUHR WALTER
IPC: F01D25/26
Filed: 1982-12-13
Abstract: DIE ERFINDUNG BETRIFFT EINE ANORDNUNG FUER DAMPFTURBINEN ZUR SICHERUNG DER ACHSMITTIGKEIT DES TURBINENGEHAEUSES GEGENUEBER DEN LAGERUNGEN, BEI DENEN DAS TURBINENGEHAEUSES GEGENUEBER DEN LAGERUNGEN, BEI DENEN DAS TURBINENGEHAEUSE AM BENACHBARTEN LAGERGEHAEUSE MITTELS EINER VORGESEHENEN DREIFACHFUEHRUNG RADIAL WAERMEBEWEGLICH BEFESTIGT IST. AUFGABE IST ES, UNTER BEIBEHALTUNG DER DREIFACHFUEHRUNG EINE ACHSMITTIGE LAGESICHERUNG ZU ENTWICKELN, DIE MIT EINFACHEN MITTELN EINE BEGRENZUNG DER ASYMMETRISCHEN VERSCHIEBBARKEIT VON TURBINENGEHAEUSE UND LAGERUNG, INSBESONDERE IN DER HORIZONTALEBENE, ERMOEGLICHT UND DIE SICH SOWOHL FUER DEN EINSATZ AN NEUBAUANLAGEN WIE AUCH FUER NACHRUESTUNGEN EIGNET. ERREICHT WIRD DAS DURCH VERTIKAL UND BEIDERSEITIG ODER EINSEITIG DER ACHSE DER TURBINENWELLE ANGEORDNETE BEGRENZUNGSELEMENTE, DIE IN DER TRENNEBENE DER ANLAGEFLAECHEN VON TURBINENGEHAEUSE UND LAGERGEHAEUSE ZUSAETZLICH ZUR DREIFACHFUEHRUNG VORGESEHEN SIND. DIE BEGRENZUNGSELEMENTE WEISEN EIN SEITLICHES SPIEL VON EINER GROESSE AUF, DAS IM DURCHWAERMTEN BETRIEBSZUSTAND DES AGGREGATS, DURCH AUF ENTGEGENGESETZTEN SEITEN DER ANLAGEFLAECHEN STATTFINDENDES SCHULTERARTIGES ANLIEGEN, KOMPENSIERBAR IST.
Patent DD-270821-A3 (DD)
Title: Fahrzeugfenster fuer notausstieg
Inventor: WEICHERT HORST
IPC: B61D25/00
Filed: 1987-06-12
Abstract: Die Erfindung betrifft ein Fenster fuer Notausstieg bei Schienenfahrzeugen, welches in Havariesituationen benutzt werden kann. Die Aufgabe wird dadurch geloest, dass ein Festfenster mit ueblichem Fensterdruckrahmen einen zweiteiligen Fensterrahmen besitzt, der in seinen unteren Fuegeflaechen formschluessig gehalten wird und im oberen Fensterrahmenteil durch Riegelmechanismen zusammengehalten und ueber eine Riegelschiene mit Riegelbolzen durch Bedienelemente ent- und verriegelt werden kann. Fig. 1
Patent DD-276984-A3 (DD)
Title: Keramische Gemenge auf der Basis von Ton und Glas
Inventor: SCHMIDT VOLKER
Filed: 1987-09-28
Abstract: Keramische Gemenge zum Versintern bei niedrigen Temperaturen. Die Erfindung wird in der keramischen Industrie fuer Erzeugnisse der Fein- und Grobkeramik angewendet. Das erfindungsgemaesse Gemenge enthaelt einheimische Tone und Natrium-Calcium-Silicatglas in Form von industriellem Abfallglaspulver oder durch Mahlung von Sekundaerglas erhaltenem Pulver mit einer maximalen Korngroesse von 100 mm. Aus dem Gemenge sind bei Brenntemperaturen unter 1 300 K feste Keramiken herstellbar.
Patent DD-274140-A3 (DD)
Title: Verfahren zur bandnachlaufkontrolle an foerderbandanlagen
Inventor: SCHWABL ROLF
IPC: B65G43/08
Filed: 1987-10-29
Abstract: Die Erfindung betrifft ein Verfahren zum Messen des Nachlaufens von Foerderbaendern, wenn diese durch eine automatische Sicherheitseinrichtung, z. B. Metallnachweiseinrichtung, abgeschalten werden. Erfindungsgemaess wird die Aufgabe der Schaffung einer Messeinrichtung dadurch geloest, dass die Umdrehung einer Bandtrommel vom Ausloesen durch das Metallspuergeraet bis zum Stillstand des Bandes mittels an der Bandtrommel angeordneten Metallelementen, die durch einen Initiator erfasst und durch eine Auswerteinheit gezaehlt und angezeigt werden, gemessen wird.
Patent EP-1031344-A3 (EP)
Inventor: HALLORAN DANIEL JOSEPH
IPC: C09K23/54
Filed: 2000-01-10
Abstract: Methods of forming microemulsions are disclosed
which involve mixing an oil and water with a surfactant
(S1) and a co-surfactant (S2). The oil, preferably a
cyclic siloxane, is added to a solution of the surfactant
(S1) and water. A two-phase system containing the
siloxane results. The two-phase system is then titrated
with co-surfactant (S2) until a clear isotropic
microemulsion results. An emulsion polymerization
catalyst is added to the clear isotropic microemulsion
and polymerization of the cyclic siloxane is initiated.
The polymerization is allowed to advance until the
reaction is complete or a desired degree of
polymerization (DP) has been obtained. Microemulsions of
high molecular weight silicone polymers with low
polydispersity are produced.
Patent EP-1034785-A3 (EP)
Inventor: HOUGHTON MICHAEL
IPC: C07K14/18
Filed: 1990-03-16
Abstract: A pharmaceutical composition comprising a hepatitis C virus (HCV)
antisense polynucleotide which is selectively hybridizable for the sense strand
of the genome of an HCV, wherein the polynucleotide comprises a
contiguous sequence of at least 8 nucleotides complementary to the sense
strand of the genome of an HCV and a pharmaceutically acceptable excipient,
wherein HCV is characterized by:
   (i) a positive stranded RNA genome;   (ii) said genome comprising an open reading frame (ORF)
encoding a polyprotein; and   (iii) said polyprotein is encoded by an HCV genome wherein the
HCV genome has an homology at the polypeptide level of at
least 40% to the 169 amino acid sequence shown in Figure 11.
Patent EP-1093157-A3 (EP)
Inventor: SHINOZAKI HIROYUKI
IPC: H01L21/312
Filed: 2000-10-13
Abstract: A substrate processing method and apparatus capable
of uniformly supplying a processing liquid to a substrate
surface in substrate processing such as development
processing without exerting an influence on the physical
properties of the processing liquid and without damaging
the substrate. A rotating blade is disposed above the
horizontally placed substrate so as to face the substrate.
The processing liquid is supplied to the surface of the
substrate, and the rotating blade is rotated while being
kept out of contact with the processing liquid to induce a
gas current. The gas current forms a mass of processing
liquid having an internal circulating current on the
substrate surface below the rotating blade.
Patent EP-1099624-A3 (EP)
Inventor: SCHAEFER WILHELM DR
IPC: B63H23/06
Filed: 2000-11-02
Abstract: The ship's drive has a single motor-gearbox with an axle offset for driving a propeller shaft (7) with a propeller (5) positioned by bearings, whereby the gearbox (2) is rigidly connected to the drive (1), an integral pressure bearing for taking up and transferring propeller thrust and a clutch (3) for connecting or disconnecting the drive. The drive and the gearbox are separately elastically supported on the ship's base plate (6) via an elastic support and via bearings containing elastic elements (13) respectively. The elastic elements are integrated into a separate bearing block rigidly attached to the ship's base and are connected to foot straps laterally formed on the gearbox.
Patent EP-1069355-A3 (EP)
Inventor: KERGER LEON
IPC: F16K17/38
Filed: 2000-06-22
Abstract: Soupape de sûreté pour réservoir de gaz sous pression comprenant
un bouchon (24) en matière fusible destiné à fondre à une température
prédéterminée pour libérer le gaz sous pression hors du réservoir et éviter
des risques d'explosion. Le bouchon fusible (24) est soumis à l'action d'un
piston coulissant (14) à action différentielle destiné à réduire au moins une
partie de l'effet de la pression du gaz sur le bouchon fusible (24) pour
éviter que le bouchon ne fonde à une température inférieure à la température
prédéterminée sous l'effet de la pression.
Patent EP-1026550-A3 (EP)
Inventor: DEN BOEF ARIE JEFFREY
IPC: G03F7/20
Filed: 2000-02-02
Abstract: In a lithographic projection apparatus, an interferometric alignment system
provides an alignment signal for reproducibly registering a reticle 10 with a wafer 12. The
radiation from a laser 50, which is the illumination source for the interferometer, is
modulated by a phase modulator 52 to eliminate spurious noise from the alignment signal.
Patent EP-1038664-A3 (EP)
Inventor: KATAYAMA KAZUTAKA
IPC: C08L77/00
Filed: 2000-03-20
Abstract: A conductive polyamide resin composition including 6 to 15
phr of conductive carbon black and 0.3 to 5 phr of a coupling agent
has excellent conductivity and resistance to sour gasoline,
thereby being useful as an inner tube material for a tube.
Patent EP-1061231-A3 (EP)
Inventor: MARSHALL MIKE E
IPC: E21B33/06
Filed: 2000-06-13
Abstract: A stripper/packer (14) for sealing against tubing being moved
therethrough includes sealing elements (176) which are urged against a tubing (22)
being moved into or removed from a wellbore to isolate the pressure in the
wellbore. The sealing elements (176) are comprised of a non-pliable material,
preferably an ultra-high molecular weight (UHMW) plastic. The sealing elements
(176) are urged into sealing engagement with the tubing (22) so that as the tubing
passes therethrough, the wellbore pressure is isolated. The sealing elements (176)
may be used in stripper/packers which apply pressure laterally to cause the sealing
elements to engage the sides of the tubing, or in stripper/packers that apply
pressure to the top and bottom of the sealing element to cause the element to
compress and seal around the tubing.
Patent EP-1073099-A3 (EP)
Inventor: CHAUDHRY SAMIR
IPC: H01L21/02
Filed: 2000-07-17
Abstract: A method of making a capacitor includes the steps of
forming an interconnection line above a substrate,
depositing a first dielectric layer on the interconnection
line, and etching a via in the first dielectric layer. The
via has a tapered width which increases in a direction
toward the substrate. Further, the method includes filling
the via with a conductive metal to form a metal plug, and
etching a trench in the first dielectric layer around an
upper portion of the metal plug. The metal plug has a
tapered width which secures it into the dielectric layer.
A second dielectric layer is deposited adjacent the metal
plug and an upper electrode is deposited on the second
dielectric layer. Preferably, a lower electrode is
deposited to line the trench and contact the metal plug.
Patent EP-1070587-A3 (EP)
Inventor: TSURUOKA YUJI
IPC: B41J2/05
Filed: 2000-07-18
Abstract: A printing apparatus and printing method for
improving printing speed in multi-pass printing without
increasing the capacity of a printer power source while
utilizing a conventional printhead. A plurality of
printing elements (86001 to 86192) of the printhead is
divided into a plurality of blocks (83); different
blocks are selected from the plurality of blocks for
each scan of the multi-pass printing; printing elements
included in the selected block are time-divisionally
driven (Fig. 10); and moving speed of the carriage is
increased in accordance with the number of times of
scans in multi-pass printing. In multi-pass printing,
for instance, in a case where the number of blocks
selected for each scan of multi-pass printing is one
half of the total number of blocks, the moving speed of
the carriage is doubled, thereby achieving high-quality
image printing while maintaining high speed of the
printing.
Patent EP-1075940-A3 (EP)
Inventor: NAGATA TORU
IPC: B29C65/02
Filed: 2000-08-11
Abstract: A laminating method for forming a laminated layer
in the form of a transparent film on the surface of
image on a printed object (P) by forming a laminated
portion by overlapping with the printed object a member
for laminating use (2) provided with a laminating layer on
heat resistive base material comprises the steps of
transferring the laminated layer to the surface of
image on a printed object (P) for laminating; and peeling
off from the heat resistive base material of the member
for laminating use the rear edge portion of the printed
object having the surface of image laminated with the
transferred laminating layer of the member for
laminating use by exerting active force on the rear
edge of the printed object in the carrying direction
having laminated thereon the laminating layer of the
member for laminating use (2). The laminating method thus
arranged, only the needed portion of the laminating
layer on the heat resistive base material is
transferred to the surface of image on the printed
object. Then, the portion of the laminating layer
transferred to the printed object (P) and the portion
remaining on the heat resistive base material are
reliably separated efficiently, hence making it
unnecessary to cut further the printed object and the
member for laminating use to obtain a predetermined
shape. Thus, no wasteful cut pieces are created.
Patent EP-1078821-A3 (EP)
Inventor: BYMA GEORGE
IPC: B60R13/08
Filed: 2000-08-25
Abstract: An automotive interior trim product (12), for example a
headliner, and method of producing such a product. The
product (12) comprising an energy management element (18)
which is adapted to be secured to an automotive interior to
provide an energy management function. The energy
management element (18) is fabricated from a material
comprising an array of fused or bonded tube-like members
(6), and comprises a one-piece unitary structure with zones
of differing physical properties. The zones of differing
physical properties provide different levels of energy
management which are matched to the requirements of the
interior. The differing physical properties and so
differing levels of energy management in the different
zones being produced by moulding (G,H) of the unitary
element (18). Alternatively and/or in addition within the
fused array (18) differing types of tube-like members (6)
may be used in the differing zones. Such differing types of
tubes (6a,6b) may have different wall (24) thicknesses
(t a ,t b ), different diameters/dimensions (d d ,d e ).
Patent EP-1111895-A3 (EP)
Inventor: MCCLENNON ROBERT SCOTT
IPC: H04L12/10
Filed: 2000-12-18
Abstract: A data traffic predictor for a modem, and a method for
power management in a modem, are described. The data traffic
predictor includes a data traffic monitor, a periodicity
detector and a power mode controller. The data traffic monitor
monitors incoming data to the modem. If the periodicity
detector determines if the data is substantially periodic, which
indicates that the data traffic is isochronous, the power mode
controller changes the modem power mode to quiescent power mode
operating at a minimum data rate to permit the isochronous data
traffic to be carried. The apparatus and method of the present
invention permit low level control of a modem's power mode, and
permit the use of a quiescent power mode running at a reduced
data rate, without sacrificing quick recovery time to a full on
power mode when required.
Patent EP-1136702-A3 (EP)
Title: Pressurised water supply
Inventor: RUOFF MICHAEL
IPC: F15B11/16
Filed: 2001-03-01
Abstract: The pump (2) is controlled by a variable speed motor (1) according to a central control unit (17) which also controls a pressure limiting valve (5), overflow throttle valve (7) and a shut off valve (6). Spray gun outlets (15,16) have shut off valves (8-10) and pressure control valves (11-13) also controlled by the unit when any are switched on or off and the pressure is held at the supply line (4).