baber/WOPTO huggingface dataset:
Patent PT-1519939-E (PT)
Title: N-aryl diazaspiracyclic compounds and methods of preparation and use thereof
Inventor: BHATTI BALWINDER S
IPC: A61P25/28
Filed: 2003-06-27
Abstract: Compounds, pharmaceutical compositions including the compounds, and methods of preparation and use thereof are disclosed. The compounds are bridged analogues of N-heteroaryl diazaspirocyclic compounds, or prodrugs or metabolites of these compounds. The aryl group can be a five or six-membered heterocyclic ring (heteroaryl). The compounds and compositions can be used to treat and/or prevent a wide variety of conditions or disorders, particularly those disorders characterized by dysfunction of nicotinic cholinergic neurotransmission, including disorders involving neuromodulation of neurotransmitter release, such as dopamine release. CNS disorders, which are characterized by an alteration in normal neurotransmitter release, are another example of disorders that can be treated and/or prevented. The compounds and compositions can also be used to alleviate pain. The compounds can (i) alter the number of nicotinic cholinergic receptors in the brain of the patient, (ii) exhibit neuroprotective effects and (iii) when employed in effective amounts, not result in appreciable side effects (e.g. side effects such as significant increases in blood pressure and heart rate, significant negative effects upon the gastrointestinal tract, and significant effects upon skeletal muscle).
Patent PT-1558707-E (PT)
Title: Gas generator grate
Inventor: SAARES TIMO
IPC: C10J3/42
Filed: 2003-10-21
Abstract: A grate for a gas generator ( 7 ) adapted to operate in the gasifier of the gas generator so as to provide support to solid fuel fed thereon such as wood chips, peat, bark and hog fuel from forest harvesting and the like refuse fuel, the cross sections of the gasifier and thus also its grate being substantially circular in shape and the grate being equipped with substantially circular slots ( 9 ) having the same center point but a varying radius, whereby the circular slots are formed between the annular grate rings ( 3 ), and the grate having placed thereon a mass of balls ( 2 ) with a diameter larger than the width of the grate slots. The invention is implemented by way of mounting below the grate a member ( 4 ) that is rotatable about the center axis of the grate and is equipped with projections ( 6 ), at least some of which extending upward through the circular grate slots ( 9 ) to a level higher than the top level of the grate.
Patent PT-1665494-E (PT)
Title: Method for operating or controlling a wind turbine and method for providing primary control power by means of wind turbines
Inventor: FORTMANN JENS
IPC: F03D7/04
Filed: 2004-09-03
Abstract: Operating method for at least a wind turbine with a rotor and an electricity generator coupled to the rotor for output of electrical power to an energy distribution network. Power output is controlled with a control arrangement that ensures the turbine operates in its working range, whereby dependent on a change in a network operating parameter, the turbine is controlled so that it outputs more power to the network than would occur during its normal steady-state operation. An independent claim is made for a method for operating a wind turbine in which the turbine rotor is operated at a speed above its normal steady-state speed in order to supply, at least temporarily, extra power to an electricity distribution grid.
Patent PT-1541146-E (PT)
Title: Zolpidem hemitartrate solvate
Inventor: LEONOV DAVID
IPC: A61P43/00
Filed: 2001-04-24
Abstract: The present invention provides for novel polymorphs of zolpidem hemitartrate and the preparation of the polymorphs.
Patent PT-1657005-E (PT)
Title: Method of manufacturing a sheet metal profile
Inventor: KRONSTEINER RAINER
IPC: B21D5/08
Filed: 2005-09-16
Abstract: Production of profiled metal strip with flanges (6, 7) which are connected to the remainder of the profile by radii (8) and which has reinforcing ribs (4', 5') comprises embossing the edges of a metal strip to form the ribs. The radii and the flanges are then produced by roll forming.
Patent PT-1591953-E (PT)
Title: System and method for decoding digital encoded images
Inventor: ALASIA ALFRED V
IPC: G06T1/00
Filed: 2005-04-25
Abstract: A method is presented for decoding an encoded image produced from a primary image and at least one secondary image using at least one encoding parameter. The encoded image is formed so that when the encoded image is printed, the secondary image is not discernible to a viewer without an optical decoding device having characteristics corresponding to the at least one encoding parameter. The method comprises obtaining a digital version of the encoded image, determining the at least one encoding parameter, and constructing a decoded image from the digital encoded image using at least one of the encoding parameters in the encoding parameter set.
Patent PT-1926373-E (PT)
Title: Use of cni-sl formulations for controlling white fly
Inventor: THIELERT WOLFGANG
IPC: A01N25/00
Filed: 2006-08-26
Abstract: Method of controlling eggs and nymphal stages of whitefly by the spray application of agrochemical formulations containing at least one insecticide from the series of the neonicotinyls, at least one fatty alcohol ethoxylate of the formula (I), at least one solvent from the group consisting of dimethyl sulphoxide, N-methylpyrrolidone and butyrolactone, and, if appropriate, additives.
Patent PT-2061636-E (PT)
Title: Cleaver having a crush-forged crank
Inventor: DROESE JOACHIM
IPC: B21D53/64
Filed: 2007-07-20
Abstract: The present invention relates to a cleaver (8) having a crush-forged crank (6). In order to provide a cleaver having an improved manageability and surface feel, thereby preventing any possible injuries during the use of the cleaver, the invention proposes that the crank according to the invention extends from the handle (4) in the direction of the cutting edge (11) along the blade and/or edge surface (5) on the handle side.
Patent PT-697866-E (PT)
Inventor: SAMUELS GLENN JAY
IPC: A61K31/535
Filed: 1994-05-10
Abstract: Mycophenolate mofetil and mycophenolic acid can be conveniently manufactured into high dose oral formulations by the hot melt filling of a supercooled mycophenolate mofetil or mycophenolic acid liquid into a pharmaceutical dosage form. High dose oral pharmaceutical formulations and manufacturing methods therefor are disclosed.
Patent PT-884052-E (PT)
Inventor: SHIMURA TAKESADA
IPC: A61L27/22
Filed: 1996-11-14
Abstract: A cartilage and bone morphogenetic repairing material which contains a bone morphogenetic protein and a polyoxyethylene-p-olyoxypropylene glycol. In particular, it is preferable that a molecular weight of a polypropylene glycol, i.e., a component of said polyoxyethylene-polyoxypropylene glycol, being in the range of about 1,500-4,000 and a weight ratio of ethylene oxide being in the range of 40-80%/molecule, and a concentration of said polyoxyethylene-polyoxypropylene glycol in an aqueous solution being about 10-50%. It may be applied in a cartilage and bone morphogenetic method requiring no surgical operation and which comprises a bone morphogenetic protein and a carrier having a high bio-absorption, a good affinity to the bone morphogenetic protein and capable of temperature dependent gel-sol reversible transition. It is convenient to apply locally to the site of bone fracture or bone defect with efficient treatment effect. <IMAGE>
Patent PT-845263-E (PT)
Inventor: MARCHI EGIDIO
IPC: A61K9/66
Filed: 1997-10-17
Abstract: The invention refers to capsules made by soft or hard gelatine containing as active principle the antiinflammatory drug known as diclofenac (INN) or the sodium, potassium or hydroxyethylpyrrolidine salts thereof dissolved in a solvent selected from polyethylene glycols, C8-C10 saturated polyglycosylated glycerides, diethylene glycol monoethylether and mixtures thereof.
Patent PT-991428-E (PT)
Inventor: RAJAGOPALAN RAGHAVAN
IPC: C07D417/14
Filed: 1997-05-09
Abstract: This invention provides functional dyes of the general formula:    <IMAGE>  1   <IMAGE>   wherein R1, R2, and R5 may be the same or different and are selected from the group consisting of hydrogen, C1-C10 allkyl, C1-C10 alkoxyl, hydroxyl, C1-C10 hydroxyalkyl, C1-C10 alkoxyalkyl, C1-C10 aryl, carboxyl, C1-C10 carboxylalkyl, halogen, nitro, C1-C10 alkoxycarbonyl, mercapto, C1-C10 mercaptoalkyl, C1-C10 alkylthio, sulfonate, and -(CH2)m-N(R6)(R7) wherein R6 and R7 are independently hydrogen or C1-C10 alkyl, C1-C10 acyl, and R6 and R7 are capable of forming 5, 6, or 7 membered rings which may optionally be substituted with -O-, -NR8, or -S-; R3 and R4 may be the same or different and are selected from the group consisting of C1-C10 alkyl, C1-C10 hydroxyalkyl, C1-C10 alkoxyalkyl, C1-C10 aryl, C1-C10 carboxylalkyl, C1-C10 alkyl sulfonate, mercapto alkyl and -(CH2)mN(R6)(R7); W1 and W2 may be the same or different and are selected from the group consisting of -S-, -O-, -Se-, -Te-, -NR8 and C(R9)(R10); and m is about 0-10; R8 is hydrogen, C1-C10 alkyl, C1-C10 alkoxy, C1-C10 mercaptoalkyl, hydroxyl, C1-C10 hydroxyalkyl, C1-C10 alkoxyalkyl, C1-C10 aryl, C1-C10 carboxylalkyl, C1-C10 alkoxycarbonyl, C1-C10 alkylthio, and -(CH2)m-N(R6)(R7); R9 and R10 are independently hydrogen, C1-C10 alkyl, C1-C10 alkoxyl, C1-C10 hydroxyalkyl, C1-C10 alkoxyalkyl, C1-C10 carboxyalkyl, C1-C10 alkoxycarbonyl, and -(CH2)m-N(R6)(R7); and A or B may be the same or different and are selected from the group consisting of -(CH2)m, -C(R9)(R10), -(CH2)m-N(R6)(R7), -O-, -S-, or -NR8.
Patent PT-989850-E (PT)
Inventor: OERTEL WOLFGANG H
IPC: A61K31/425
Filed: 1998-01-16
Abstract: The present invention provides the use of pramipexole in the treatment of restless legs syndrome.
Patent PT-962044-E (PT)
Inventor: LAMP KARL J
IPC: H02K49/04
Filed: 1998-02-20
Abstract: An adjustable coupler has a group of magnet rotors with permanent magnets separated by air gaps from non-ferrous conductor elements presented by a group of conductor rotors. The air gaps are adjusted by axial movement of one of the groups relative to the other to vary the slip of the coupler and control the load speed under varying load conditions. <IMAGE>
Patent PT-929926-E (PT)
Title: Method and apparatus for supplying contactless power
Inventor: MEINS JURGEN G
IPC: H02M7/48
Filed: 1998-08-07
Abstract: A method and apparatus for supplying contactless power. Electrical power is transferred from a power source to a load through a primary energy converter that can be connected to the power source, through a primary inductive loop connected to the primary energy converter and a secondary pickup coil magnetically coupled to the primary inductive loop, and then to a secondary energy converter. The power factor for the transfer of electrical energy is one. Multiple loads can receive power from the power source and, where the loads are located in zones, collisions between the loads can be prevented.
Patent PT-1048089-E (PT)
Inventor: FERREIRA ANTONIO L DE M
IPC: H01M50/494
Filed: 1998-10-14
Abstract: The invention concerns an absorbing separator for lead-acid storage cells regulated by a valve, comprising a first glass fibre layer, a second glass fibre layer and a synthetic resin strip inserted between the first and second layers.
Patent PT-1149167-E (PT)
Inventor: SCHREIBER MICHAEL
IPC: C07K14/16
Filed: 1999-12-03
Abstract: The present invention relates to a pharmaceutical composition or a vaccine which comprises a mixture of viral protein molecules which are sequence variants of a single viral protein or of part of same. The invention furthermore relates inter alia to a DNA vaccine which codes for a mixture of structurally different virus proteins, the vaccine containing a mixture of sequence variants of a viral DNA molecule or of part of same which code for sequence variants of a viral protein or part. According to a preferred version of the invention, the viral proteins are sequence variants of the GP120 protein of the human immunodeficiency virus (HIV) which differ from each another in their amino acid sequence in the region of the V2 loop and/or of the V3 loop. The invention furthermore relates to the preparation of the virus vaccines including the intermediate stages or constructs, preparation processes and uses connected with them.
Patent SG-24487-G (SG)
Title: Embossed panty liner
IPC: A61F13/511
Filed: 1987-03-09
Abstract: A thin absorbent undergarment liner is provided which exhibits a clear, aesthetically pleasing embossed pattern on the body facing surface thereof while still maintaining the longitudinal edges soft and comfortable. The liner is provided to have areas of deep depressions on the body facing surface and shallow impressions on the longitudinal edges.
Patent SG-57689-G (SG)
Title: Method and apparatus for measuring the strength of a radio frequency signal
IPC: H04B/
Filed: 1989-08-25
Abstract: A method and apparatus for measuring the strength of a radio frequency (RF) signal subject to Rayleigh fading. The strength of the RF signal is sampled two or more times during a predetermined time interval and the sampled signal strength having the largest magnitude is selected. The selected signal strength is a reasonably accurate measure of the signal strength since the true average strength of a Rayleigh fading signal is close to its peak signal strength. The inventive method and apparatus is particularly well adapted for use in a scanning receiver located in a base station radio (111, 121, 131) of a cellular radiotelephone communications system. The scanning receiver includes an antenna selector (102) for selecting one of a plurality of sector antennas, an RF signal receiver (104) tunable to a plurality of different RF signal frequencies, an analog-to-digital converter (106) for converting RF signal strength samples to a binary data signal and a microprocessor (114) together with peripheral devices (108, 110, 112, 116, 118, 120) for controlling the operation of the antenna selector (102), RF signal receiver (104) and analog-to-digital converter (106).
Patent IE-780037-L (IE)
Title: IMIDAZO [1,2-a] QUINOXALINES
IPC: A61P31/04
Filed: 1978-01-06
Abstract: A 1-(2-acylaminophenyl)imidazole of formula: <IMAGE> wherein R2 is hydrogen or a radical bonded to the nitrogen by a carbon to nitrogen linkage and selected from the group consisting of aliphatic, cycloaliphatic, phenyl, substituted phenyl, fused bicyclic aryl, and monocyclic aryl substituted aliphatic groups.
[US4160097A]
Patent IE-44583-L (IE)
Title: Indication of signal pulse length
IPC: G01R19/165
Filed: 1977-01-20
Abstract: 1507652 Pulse duration discriminator TELEFONAKTIEBOLAGET L M ERICSSON 17 Jan 1977 [23 Jan 1976] 01815/77 Heading H3T A circuit blocks input pulses shorter than a predetermined length by detecting whether a pulse derived from a monostable circuit triggered by the input pulse terminates before the end of the input pulse. In Fig. 2, delay circuits DE1, DE2 compensate for gate propagation delays, such that the positive edges of the input signal and the positive edge of the monostable SSE2 output arrive simultaneously at AND2, and similarly for the EXCLUSIVE-OR EOR. The leading edge of an interfering pulse DP shorter than the monostable period T, will cause SSE2 to give an output, but the trailing edge applied to AND2 will inhibit SSE2 output before the end of the monostable period T. Thus for short pulses, inputs of the same sense will always be applied to EOR, which will remain at logic 0. A wanted pulse, of longer duration than T, will cause SSE2 to give an output for time T, after which it goes to logic 0. As the input is still at logic 1, AND 2 changes state and the inputs to EOR are different, thus giving an output pulse 15. A second embodiment Fig. 3 comprises a monostable ME having a CLEAR input C and a Master-Slave flip-flop comprising an AND gate AND3 and a J-K flip-flop FF. A trailing edge applied to C inhibits the monostable output. Input B of AND3 only responds to transitions and as shown only responds to negative edges. The leading edge of a wanted input pulse will cause AND3 to provide a short pulse RP which will set the flip-flop FF to provide an output IS, and the trailing edge of the input pulse will reset FF.
[SE7600714A]
Patent IE-39344-L (IE)
Title: 7ó-alkoxy cephalosporanates and corresponding¹penicillanates
IPC: A61P31/04
Filed: 1974-03-14
Abstract: 1439898 Alkoxy-substituted cephalosporins and penicillins SMITHKLINE CORP 12 March 1974 [15 March 1973] 10871/74 Heading C2C A compound of the formula wherein R is hydrogen or acyl; R<SP>1</SP> is C 1-6 alkyl; Z is R<SP>2</SP> is hydrogen, or an easily removable ester protecting group; and A is a non-interfering group, is prepared (a) when R is H, by treating a compound of the formula wherein R<SP>3</SP> is C 1-6 alkyl, with a C 1-6 alkyl alcohol in the presence of a mercuric or silver ion in a compatible solvent at a temperature and for a length of time to cause substitution without decomposition, or (b) when R is acyl, treating a compound of the formula with a C 1-6 alkyl alcohol in the presence of a silver ion in a compatible solvent at a temperature and for a length of time to cause substitution without significant decomposition. Preparation of intermediates is described as follows: t-butyl 7#-benzylideneamino-desacetoxycephalosporanate is reacted with methyl methanethiosulphate and NaH to give t-butyl 7# - benzylideneamine - 7α - methylthiodesacetoxycephalosporanate which is treated with HC1 to form t-butyl 7#-amino-7α-methylthiodesacetoxycephalosporanate and its HCl salt; t-butyl 7#-aminocephalosporanate and benzaldehyde are reacted to form t-butyl 7#- benzylideneaminocephalosporanate which is reacted as above to form t-butyl 7#-benzylideneamino - 7α - methylthiocephalosporanate which is converted to t-butyl 7#-amino-7α- methylthiocephalosporanate; benzyl 6#- aminopenicillanate is similarly converted to benzyl 6# - benzylideneaminopenicillanate; benzyl 6# - benzylideneamino - 6α - methylthiopenicillanate; benzyl 6# - amino - 6α- methylthiopenicillanate and its p-toluenesulphonic acid salt.
[GB1439898A]
Patent IE-33092-L (IE)
Title: Piperidine derivatives
IPC: C07D213/26
Filed: 1969-05-15
Abstract: 1,203,149. Piperidine derivatives. IMPERIAL CHEMICAL INDUSTRIES Ltd. 13 May, 1969 [10 June, 1968], No. 27502/68. Heading C2C. [Also in Division A5] Novel compounds of Formula I wherein R<SP>1</SP> is H, alkyl or aryl and X is a substituted or unsubstituted aryl radical and their acid addition salts are prepared by the reduction of the corresponding pyridine derivative or of an acid addition salt or quaternary N-benzyl salt of said pyridine derivative. Intermediates isolated are the starting materials for the above reaction which are prepared by the reaction of a compound X-O-Na with a corresponding halo-methyl-pyridine derivative (which is prepared by reaction of the corresponding hydroxymethyl derivative with thionyl chloride). The said hydroxymethyl derivatives are prepared by reduction of the appropriate keto derivatives.
[GB1203149A]
Patent IE-840691-L (IE)
Title: Antibiotic l.17046.
IPC: C07K9/00
Filed: 1984-03-21
Abstract: The present invention is directed to a new antibiotic substance arbitrarily denominated antibiotic L 17046. This antibiotic substance is obtained from the known antibiotic substance called teicoplanin (formerly teichomycin) by chemical treatment.The new compound possesses antimicrobial activity especially against gram-positive bacteria.
Patent FI-821196-L (FI)
Inventor: KAELBERER HEINZ
IPC: A22C13/00
Filed: 1982-04-05
Abstract: A process and apparatus for coating the interior of a fiber-reinforced tube formed of cellulose hydrate in which a tube filled with a coating liquid is passed through a special conveying and pumping device which also serves to replenish the coating liquid. Above the level of the coating liquid, the tube is inflated with a support gas and is gradually flattened. The flattened tube then travels through a metering device made up of wipers in the form of doctor blades or rollers, which retain the major quantity of the coating liquid which is present on the inside surface of the tubing so that a thin, uniform film of the coating liquid is formed. The tubing is thereafter dried to remove the volatile constituents of the coating liquid, and is subsequently wound up.
Patent IE-861542-L (IE)
Title: Hybrid interferons
IPC: A61K38/21
Filed: 1986-06-10
Abstract: Novel hybrid interferons are produced which are derived from lymphoblastoid interferons a-2 and a-3 belonging to the interferon aB and αD groups, respectively. The novel hybrid interferons possess valuable antiviral and antiproliferative properties.
Patent IE-41642-L (IE)
Title: Noise reducing material.
IPC: F02B77/13
Filed: 1975-07-25
Abstract: 1451707 Laminates BRITISH URALITE Ltd 8 July 1975 [26 July 1974] 33185/74 Heading B5N [Also in Divisions C3 F1 and F2] A noise reducing material for application to the surface of a machine component that is prone to vibrate, to reduce machine noise, consists of a laminate comprising a metallic sheet which is from 0À4 to 2 mm. thick and has a density of at least 7 gm./c.c., and, adhesively bonded to each face of the sheet, a layer of substantially non-porous reinforced thermoplastic material comprising a matrix of pliant thermoplastic material reinforced with fibrous material in the form of staple fibres forming a disperse phase in the matrix. The metallic sheet may be formed of lead. Specified materials for the matrix are asphaltic bitumen, vinyl chloride polymers and low density polyethylene, the fibres being preferably of asbestos although metal fibres or synthetic fibres may be used. In a preferred embodiment, each layer of fibre reinforced thermoplastic material comprises one or more sheets reinforced with asbestos fibres, the asbestos reinforcement in each layer being in the form of laminµ of asbestos fibres, each lamina extending parallel to the plane of the sheet, such sheets being formed for example by forming a dispersion of short asbestos fibres and bitumen in water and building up the desired sheet thickness from a plurality of layers of the dispersion, e.g. by use of a board machine. Fillers, e.g. finely divided mineral fillers such as talc or finely divided metal particles may be included in the layer of thermoplastic material. Layers of other material for additional sound deadening, decoration or protection from environmental attack may be included in the laminate, e.g. layers of felt and/or foamed plastics and/or glass fibre may form an internal or external layer of the laminate. When the laminate is to be applied to an internal combustion engine, the exposed surface thereof may be treated with an oilresistant paint, e.g. an epoxy resin or polyamide; an elastomeric material, e.g. a polysulphide rubber may be applied, e.g. by dipping as an external layer. The layers of the laminate are bonded by an adhesive, e.g. a polymeric adhesive such as a rubber-based adhesive which may be applied by spray, roller coating or brush coating and may be continuous or discontinuous. Consolidation of the laminate is effected by calendering.
[GB1451707A]