baber/WOPTO huggingface dataset:
Patent RU-2205831-C2 (RU)
Title: Quinazolinones inhibiting farnesyltransferase activity
Inventor: ANZHIBO PATRIK RENE
IPC: C07D405/04
Filed: 1998-04-17
Granted: 2003-06-10
Abstract: FIELD: organic chemistry, biochemistry. SUBSTANCE: invention proposes derivatives of quinazolinone of the general formula (I)   and their pharmaceutically acceptable acid-additive salts and stereochemical isomeric forms where dotted line is optionally linkage; X is oxygen atom; R 1  and R 2  each means independently hydrogen or halogen atom; R 3  and R 4  each means independently hydrogen or halogen atom; R 5  means hydrogen, halogen atom or radical of the formula -O-R 10  (a-1) or N-R 11 R 12  (a-3) where R 10 , R 11 , R 12  are hydrogen atom; R 6  means radical of the formula (b-1)   or (b-2)   where R 16  is hydrogen atom or phenyl; R 17  is hydrogen atom or C 1-6 -alkyl; R 7  is hydrogen atom or C 1-6 -alkyl under condition that dotted line is not a linkage; R 8  is hydrogen atom, C 1-6 -alkyl or Het 1 CH 2 ; R 9  is hydrogen atom;   is pyridinyl. Compounds of the general formula (I) show inhibitory effect on farnesyltransferase activity and can be used for preparing medicinal agents inhibiting proliferative diseases. Invention relates also to pharmaceutical composition based on compounds of the general formula (I) eliciting inhibitory effect on farnesyltransferase activity, to method for preparing this composition, to intermediate derivatives of quinazolinone of the general formula (IX)   and their acid-additive salts or stereochemical isomeric forms where n = 2 or 3 and R 1 , R 2 , R 3 , R 4 , R 9 , mean values indicated above, to method for preparing some compounds of the general formula (I) where R 6  is radical of the formula (b-2) and to method for preparing intermediate derivatives of quinazolinone of the general formula (IX) and their acid-additive salts or stereochemical isomeric forms. EFFECT: improved preparing method of compounds and composition, valuable medicinal and biochemical properties. 10 cl, 4 tbl, 15 ex
Patent UA-27923-C2 (UA)
Title: Steam generator
IPC: F22B37/10
Filed: 1993-08-06
Abstract: The invention relates to steam generator working on fossil fuel, with gas duct with surrounding wall formed of connected to each other with sealing pipes. The pipes in the first section of gas duct placed lower have larger inner diameter compared to the higher second part of gas duct.
Patent UA-40611-C2 (UA)
Title: immunoconjugate, method for its preparation, pharmaceutical composition
Inventor: Holtzer Wolfgang
IPC: C12N15/02
Filed: 1995-09-14
Abstract: The present invention relates to the new fusion proteins which consist of a tumor-associated targeting element preferentially a monoclonal antibody or a fragment thereof recognizing a molecule which is preferentially expressed on human tumor cells such as the human epidermal growth factor receptor (EGFR), and a biologically active ligand, selected from group consisting of chemokines, preferably from the family C-X-C. Present invention provides an immunoconjugate comprising of a monoclonal antibody or a fragment thereof directed to a tumor cell bearing an antigen epitope of the epidermal growth factor receptor (EGFR), and a chemokine, which is fused to said antibody or antibody fragment, at that chemokine is IL-8.
Patent UA-57033-C2 (UA)
Title: Chip module and a method for producing the module
Inventor: FISHER JURGEN
IPC: H01L23/12
Filed: 1997-08-21
Abstract: The present invention pertains to a chip module presenting on its inner surface (2) a contact area (3) consisting of a plurality of electro-conductive contact units (4) isolated from each other, substantially flat and including at least one semiconductor wafer (6) with one or more integrated semiconductor circuits, joined through electrical connections (8) to the units in the contact area (3). The contact units 4) in the chip module (1) consist of prefabricated mounts intended for supporting the lead frame or at least one semiconductor wafer (6), and, located on one or more opposing faces of the chip module, two or more connections turned outwards, aligned close to each other (8) and intended for the surface assembly of said chip module (1) cither on the components side (9) of an external printed circuit board or on the surface of an external board substrate (10).
Patent UA-35504-C2 (UA)
Title: lubricant composition
Inventor: ALEKSANDROV SERHII MYKOLAIOVYCH
IPC: C10M169/00
Filed: 1999-10-22
Abstract: The invention relates to lubricant compositions and can be used for the treatment of friction units of different machines and mechanisms in manufacturing processes, which purpose is modification of frictions surfaces. A lubricant composition, containing oil and powder-like abrasive filling material, at that it contains in addition thickener and wax.
Patent UA-46943-C2 (UA)
Title: Electrode for determining electric properties of surface coating of a cylindrical conductive substrate
Inventor: OPRYSHKO OLEKSII OLEKSANDROVYCH
Filed: 1999-12-08
Abstract: The proposed electrode for determining electric properties of surface coating of a cylindrical conductive substrate differs in that it is designed as an elastic conducting strip with a specified width. The strip electrode is wrapped onto the cylindrical substrate to be tested. To the free end of the strip, a weight with a specified mass is suspended.
Patent RU-2188585-C2 (RU)
Title: Method for operative treatment of vertebral arterial malformations
Inventor: SAKHARJUK A P
IPC: A61B17/11
Filed: 2000-02-22
Granted: 2002-09-10
Abstract: FIELD: medicine, vascular surgery. SUBSTANCE: the method deals with ligation of thyrocervical trunk. A part of subclavial artery is resected distally against vertebral artery deviation. An end-to-end anastomosis of subclavial artery is applied. EFFECT: improved results of operative interference.
Patent RU-2182260-C2 (RU)
Title: Method for starting nuclear rocket engines based on resonant-dynamic fission and fusion reactions
Inventor: IRDYNCHEEV L A
IPC: G21D5/06
Filed: 2000-02-29
Granted: 2002-05-10
Abstract: FIELD: nuclear rocket engines. SUBSTANCE: method involves introduction of source nuclear fusion gas or steam, or fissionable gas escaping from fissionable material into reactor core or magnetic trap until desired density is attained. Then high-energy protons are injected in reactor core for the time of fission or fusion reaction initiation; these protons revolving within reactor generate neutrons from fissionable material nuclei. Electromagnetic and magnetoacoustic waves excited due to adequate selection of energy (relativistic mass of protons) have their frequency coinciding with frequency of rotation of source fusion nuclei residing in near-axis area thereby heating them to thermonuclear temperatures. In addition, high-energy protons ionize fission and fusion nuclei with the result that they start revolving under the action of crosslinked electric and magnetic fields of magnetic trap about longitudinal axis of reactor at drift speed providing for resonant fission of fissionable material nuclei during their collision with thermal neutrons entering reactor core from moderator wherein they were produced from fast neutrons during moderation of the latter. Supply of high-energy protons is ceased upon ignition of joint fission and fusion reactions. However, their supply may be continued in case critical density of fissionable material should be additionally reduced or additional nuclear energy should be generated. EFFECT: provision for joint resonant-dynamic fission and fusion reactions due to high-energy protons accelerated to energy of hundreds of megaelectron-volts. 1 dwg, 2 tbl
Patent RU-2195707-C2 (RU)
Inventor: EZERSKIJ S V
IPC: G08B29/00
Filed: 2000-03-07
Granted: 2002-12-27
Abstract: FIELD: electrical and microprocessor engineering. SUBSTANCE: device designed for use in central alarm systems of substations equipped with digital or electrical relay protective and automatic control facilities and in various other industries has monitoring unit, voltage change recording unit, microprocessor system, and four switches connected to transformer primary windings. Information from transformer secondary winding arrives at monitoring-unit microprocessor which transmits it to central processor unit of microprocessor system which controls audio alarm relay, integrated, or any other alarm connected to information output devices of microprocessor system. Proposed device provides for detecting open circuits, deenergized or abnormal conditions of internal circuits of pulse alarm channel. Device incorporates provision of diagnosing input units and introducing data recording, display, and alarm functions for varying configuration and instant transmission of information. EFFECT: enhanced reliability and enlarged functional capabilities of device. 5 dwg
Patent RU-2217310-C2 (RU)
Title: Ручной позисторный трубосварник смыслова
Inventor: SMYSLOV I I
IPC: B29C65/18
Filed: 2000-03-20
Granted: 2003-11-27
Abstract: Изобретение относится к различным технологическим процессам, обработке пластиков, устройствам для соединения предварительно сформованных частей с нагревом, с использованием нагретого инструмента, в данном случае электронагреваемого устройства для сваривания термопластовых труб, а именно ручного трубосварника, а также к их ремонту с использованием предварительно сформованных элементов, затем соединяемых вместе с помощью ручного трубосварника. Ручной трубосварник содержит теплопроводный корпус, нагреватель с нагревательным резистором, скрепленный с корпусом с хорошим тепловым контактом, набор сменных тепловводов, электроцепь и электротеплоизолирующую рукоять с питающим кабелем. Трубный тепловвод выполнен с возможностью вдвигания в него сменного тепловвода для трубы меньшего диаметра, а муфтовый тепловвод - с возможностью надвигания на него сменного тепловвода для муфты большего внутреннего диаметра. Оба сменных тепловвода выполнены с возможностью их сопряжения с тепловводными поверхностями трубного и муфтового тепловводов. Сменные трубные тепловводы выполнены из материала с большим коэффициентом линейного расширения, чем корпус. Теплопроводный корпус выполнен с плоским пазом в средней части, в котором размещен нагреватель с позистором в качестве нагревательного резистора. Изобретение позволяет снизить расход электроэнергии, металлоемкость, имеет простую конструкцию и широкое применение. 2 з.п.ф-лы, 3 ил.
Patent RU-2197254-C2 (RU)
Inventor: MARUGIN I A
IPC: A61K35/60
Filed: 2000-04-07
Granted: 2003-01-27
Abstract: FIELD: biotechnology. SUBSTANCE: invention relates to methods of production of protamine sulfate from milts of mature fishes. Method involves raw boiling out in water, milling, treatment with acetone, drying to granules formation followed by extraction of granules with 4% sulfuric acid solution, proteins precipitation from extract by addition of alcohol twofold volume, precipitate dissolving in hot water, treatment with barium hydroxide and addition of ammonia, treatment with kieselguhr, filtration, passing filtrate through cationite in H + -form, eluate concentration, precipitation of end product, its isolation and drying. EFFECT: improved processes of extraction and filtration in granules preparing. 1 tbl
Patent RU-2190231-C2 (RU)
Title: Process of calibration of meter of amplitude modulation factor
Inventor: SHEVELENKO V D
IPC: G01R29/06
Filed: 2000-04-07
Granted: 2002-09-27
Abstract: FIELD: radio engineering, certification of reference measurement aids. SUBSTANCE: technical result of invention lies in increased accuracy of formation of amplitude-modulated signals thanks to diminished effect of instability of amplitude and frequency of modulating oscillation on value of amplitude modulation factor. Process includes formation of reference AM signals by harmonic action on element of meter with modulation frequency F m  to form AM oscillations which determines oscillation amplitude of carrier frequency f H  with subsequent measurement of maximal and minimal values of AM signal and computation of modulation factor by them. Trains of rectangular pulses of double frequency f H  are formed from harmonic oscillations of carrier frequency 2f H  which control commutator switching over resistors of scale converter which relation determines value of its gain factor at moments of transit by oscillations of carrier frequency f H  of zero values and changes by harmonic law of modulation. EFFECT: increased accuracy of formation of amplitude-modulated signals. 2 dwg
Patent RU-2210913-C2 (RU)
Inventor: GRIGOR EVA R Z
IPC: A21D13/08
Filed: 2000-04-12
Granted: 2003-08-27
Abstract: FIELD: confectionery industry and public catering. SUBSTANCE: method involves preparing soya paste, which is used as partial substitute of sugar-egg mixture for aerating in an amount of 25-30 wt% or part of flour and starch in an amount of 25-30 wt%; aerating resultant mixture until volume increases by 3.0-3.5 times; kneading dough and baking for obtaining finished product. Method allows porosity to be increased by 25-40%. EFFECT: increased biological value of biscuit semi-finished product, increased content of vitamins and mineral substances, wider range of products, improved organoleptical properties and reduced energy value of biscuit. 4 ex
Patent RU-2214008-C2 (RU)
Title: Protected memory having plurality of protection levels
Inventor: BENHAMMOU JEAN-PIERRE
IPC: G06F21/79
Filed: 1998-09-23
Granted: 2003-10-10
Abstract: FIELD: protected memories. SUBSTANCE: proposed memory that provides plurality of protection levels for application areas has first protection level area, protection code input attempt counter, plurality of application areas, each including save area, application protection area, protection code input attempt counter for application area, erase key section, and erase key input attempt counter. EFFECT: enhanced reliability of protecting memory as part of intelligent card in its multiple reuse. 1 cl, 20 dwg
Patent RU-2182286-C2 (RU)
Title: Hot-water boiler block
Inventor: POBEGALOV S A
IPC: F24H1/30
Filed: 2000-05-15
Granted: 2002-05-10
Abstract: FIELD: designed for water heating, applicable for heat supply. SUBSTANCE: the hot-water boiler block has interconnected heat-exchange panels with windows, gas-circulating cavities formed by transverse walls and gas-proof shells, and a furnace made for burning of solid and gas-liquid fuel. The furnace at burning of gas-liquid fuel is positioned in the windows of the panels and provided with a body, and at burning of solid fuel it is provided with refractory settings. Installed in the windows of the panels connected by threaded bushes are perforated catalytic water walls, and the body, transverse walls and shells may be provided with heat insulation. EFFECT: enhanced efficiency of heat exchange. 4 dwg
Patent RU-2179420-C2 (RU)
Inventor: JANOVSKIJ L M
IPC: A61K6/60
Filed: 2000-05-26
Granted: 2002-02-20
Abstract: FIELD: medicine. SUBSTANCE: method involves applying water-alcohol extraction of solved organic substances from sodium chloride hydrogen sulfide mineral water with sodium fluoride taken in known proportions. This means is used for rinsing oral cavity every second day during 10 days with following course repetition 6 months later. EFFECT: enhanced effectiveness of treatment; prevented adverse side effects. 1 tbl
Patent RU-2197182-C2 (RU)
Inventor: KOPLATADZE A M
IPC: A61B17/04
Filed: 2000-05-31
Granted: 2003-01-27
Abstract: FIELD: medicine, surgery. SUBSTANCE: a vascular stem of a hemorrhoid is sutured followed by its dissection at 3, 7 and 11 according a clock face. The wound is sutured with an uninterrupted submucous suture by capturing the wound's bottom without any puncturing of mucous membrane. Inand out-punctures are made by leaving 2 cm against the wound's edge. A suture is tightened up till the juncture of the wound's mucous edges. The method prevents complications of postoperational period, such as hemorrhage, a scar narrowing of anal canal, infecting of postoperational wound. EFFECT: higher efficiency of therapy. 4 dwg
Patent RU-2204369-C2 (RU)
Inventor: BJUZO EHRVE
IPC: A61F13/26
Filed: 1998-12-23
Granted: 2003-05-20
Abstract: FIELD: medical engineering. SUBSTANCE: device has pressure lever and elongated pushing member made as a whole. The pressure lever rotatably connected to posterior end part of the elongated pushing member and rotatably connected to external cylinder behind an opening for moving forwards the elongated pushing member in the direction of the external cylinder through the opening to push the tampon out. EFFECT: enhanced effectiveness of applicator operation; reliable tampon pushing-out. 13 cl, 5 dwg
Patent RU-2186303-C2 (RU)
Inventor: IL INYKH V V
IPC: F25B15/10
Filed: 2000-08-04
Granted: 2002-07-27
Abstract: Способ получения холода в абсорбционно-диффузионном агрегате включает выпаривание хладагента из крепкого раствора, конденсацию паров хладагента и испарение жидкого хладагента. В процессе стекания в испарителе жидкий хладагент собирают в емкость в нижней части испарителя. Из емкости посредством парлифтного насоса жидкий хладагент подают в сепаратор. Далее хладагент через гидрозатвор направляют на вход дополнительного испарителя. Использование изобретения позволит уменьшить металлоемкость и габариты холодильного агрегата. 4 з.п. ф-лы, 1 ил.
Patent RU-2220813-C2 (RU)
Inventor: KROOS JOAKHIM
IPC: B22D11/06
Filed: 1999-03-01
Granted: 2004-01-10
Abstract: FIELD: metallurgy, namely process and equipment for providing uniformness of melt metallic film, for example steel film made by continuous casting of band. SUBSTANCE: melt applied onto moving belt has thickness as uniform as possible and similar properties along band width. In order to provide uniformness of metallic film along its width, gas flow inclined by angle 0 - 80 degrees relative to normal line is guided onto surface of metallic film opposite relative to flowing direction of cast metallic film. Apparatus includes at least one row of gas nozzles arranged along width of band opposite relative to motion direction of conveyor belt. EFFECT: possibility for such change of film of melt metal before and after feeding it onto conveyor belt that to provide uniform thickness along its whole width and uniform properties of its material. 17 cl, 2 dwg, 1 ex
Patent RU-2194660-C2 (RU)
Title: Tank-container
Inventor: BURMISTROV N V
IPC: B65D88/12
Filed: 2001-03-15
Granted: 2002-12-20
Abstract: FIELD: railway, road and water transport. SUBSTANCE: invention relates to containers for storage and transportation of liquids. Proposed tank- container has cylindrical barrel with bottom plates, compartments of level metering and draining and shutoff valves, two rectangular end face frames with upper and lower crossmembers, vertical uprights with load grippers at angles, upper and lower diagonal braces connecting vertical uprights with crossmembers, adapter shells welded to bottom plates and rectangular end face frames, four support beams arranged in pairs at each side of barrel and secured on lower angles of end face frames and barrel, and contact elements. Tank-container is furnished additionally with four stops secured on barrel shell. Upper support beams are rigidly secured at one side to stops and at other side, to upper grippers of frame. Lower support beams are rigidly connected to contact elements and, respectively, to lower load grippers, angle between axis of barrel and lower support beam being 22-23 ° . Adapter shell is made in form of cylinder being rigidly connected to frame by means of support shell at one side of container. Compartments of level metering and draining device and shutoff valves are found in one unit located in lower part of barrel. Stops are made in form of brackets to inner surfaces of which upper support beams are rigidly connected. Brackets are provided with trunnions rigidly secured on one of side surfaces of brackets. Invention improves operation reliability of tank-container and prevents discharge of transported liquid into atmosphere, improves manufacturability and cuts down production expenses. EFFECT: improved reliability. 4 cl, 5 dwg
Patent RU-2220070-C2 (RU)
Inventor: ARUTJUNJAN A M
IPC: B63C7/20
Filed: 2001-04-25
Granted: 2003-12-27
Abstract: FIELD: raising sunken objects. SUBSTANCE: proposed device has two opposite gripping pins articulated together; each consists of links. Each subsequent link is connected with previous articulation and hydraulic mechanism. Besides that, device is provided with ballasting pontoons which are articulated with said links of gripping pins. EFFECT: extended functional capabilities. 4 cl, 10 dwg
Patent RU-2211814-C2 (RU)
Title: Impregnated yarns of glass fibers and cloth on their base
Inventor: LOTON EHRNEST L
IPC: C03C25/47
Filed: 1999-10-08
Granted: 2003-09-10
Abstract: FIELD: fiber yarns with coating. SUBSTANCE: yarns of fibers with coating include, at least, one fiber having layer of dried residue compatible with polymers of coating composition, at least, on a part of surface, at least, of one fiber. Coating composition compatible with polymers includes: (a) multitude of discrete and stable in size particles produced from materials selected from group consisting of organic materials, polymer materials, composite materials and their mixtures ensuring production of hollows between one fiber and, at least, one adjacent fiber, with particles having overage size of about 0.1 to about 5 mcm; (b) at least, one lubricating material; (c) at least, one polymer film-forming material, and (d) at least, one finishing agent. Invention also covers cloth including, at least, one of such yarns of fibers. EFFECT: reduced wear and brittleness of fibers in friction, provided good wettability and impregnability of coating with matrix material. 59 cl, 8 dwg, 5 tbl, 4 ex
Patent RU-2202462-C2 (RU)
Title: Method for dressing laps in two-disc lapping machine tools
Inventor: KUDASHOV V JA
IPC: B24B7/17
Filed: 2001-06-29
Granted: 2003-04-20
Abstract: FIELD: abrasive working processes, namely lapping high- accuracy plane-parallel surfaces of parts in two-disc lapping machine tools with planetary lapping mechanism. SUBSTANCE: method comprises steps of determining value H lap  and form of out-of-planeness of one of laps (usually lower lap as more comfortable); applying abrasive paste (suspension) with grain size d a  = ( 2 - 3) H lap  on lap surface and uniformly distributing it; mounting at least three dressing tools between laps uniformly along circle in such a way that their continuous surface is turned to side of convex surface of one lap and their annular surface is turned to side of concave surface of other lap; performing cyclic dressing at providing rotation of laps clockwise and counter-clockwise; measuring value of out-of-planeness between cycles; then tilting dressing tool and going on dressing; selecting outer diameter of dressing tool equal to 1.0 - 1.01 of lap width and selecting width of annular surface consisting (0.2 - 0.3) of width of working surface of lap. EFFECT: simplified dressing process, enhanced efficiency, enlarged manufacturing possibilities of method. 6 dwg
Patent RU-2244037-C2 (RU)
Inventor: KHE DA KHAJ
IPC: C22C1/08
Filed: 1999-12-16
Granted: 2005-01-10
Abstract: FIELD: powder metallurgy, in particular electric contact materials. 
     SUBSTANCE: invention relates to carbon-copper composite. Material is produced from copper powder having purity of 99.9 % and black carbon powder with particle size at most 5 µm. Copper matrix has grid structure with through pores. One part of pores contains black carbon providing microstructure with carbon constituents. Parameter according to "International standard for annealed copper" is at least 40 %; density is at least 6.0 g/cm 3 . Copper powder is purified and annealed followed by blending of carbon and copper powders, double-side pressing under 500-1600 MPa, and sintering at 960-1100 0 C. 
     EFFECT: material with increased density and conductivity and enhanced durability. 
     20 cl, 1 dwg, 7 tbl