baber/WOPTO huggingface dataset:
Patent UA-81825-C2 (UA)
Title: Derivatives of fusidic acid
Inventor: DUVOLD TURE
IPC: A61P31/04
Filed: 2004-09-07
Abstract: The present invention relates to novel fusidic acid derivatives of general formula [I] wherein X represents halogen trifluoromethyl, cyano, azido, alkyl, alkenyl or aryl, wherein, said alkyl, alkenyl or aryl are optionally substituted by one or more, same or different substituents selected from the group consisting of alkyl alkenyl, aryl, alkoxy, nitro, alkylthio, halogen, azido, trifluoromethy and cyano; Y and Z both represent hydrogen, or together with the C-17/C-20 bond form a double bond between C-17 and C-20, or together are methylene and form a cyclopropane ring in combination with С-17 and C-20; A represents a bond,. O, S or S(O); В represents Calkyl Calkenyl, Cacyl, Ccycloalkylcarbonyl or benzoyl, all of which are optionally substituted with one or more substituents selected from the group consisting of halogen, hydroxy, alkoxy, aryl, heteroaryl am azido, or, if A represents a bond, В may also represent hydrogen; Q1 and ‘Q2 independently represent. -CH2-, -C(O)-, -(CHOR)-, -(CHOR)--(CHSH)-, - (NH)-, -(CHNH2)- or -(CHW)-, wherein R represent: Calkyl and W represents halogen, cyano, azido or trifluoromethyl; Q3 represents -CH2-, -C(O)- or -CHOH-; G represents hydrogen, OH or O-CO-CHtwo bonds in the pentacyclic ring being depicted with full and dotted lines to indicate that either of the two bonds may be a double bond, in which case Y is absent and Z represents hydrogen; the bond between C-l and C-2 being either a single or a double bond; and pharmaceutically acceptable salts and easily hydrolysable esters thereof, to pharmaceutical compositions comprising said derivatives, as well as to their use in therapy.(I)
Patent UA-91670-C2 (UA)
Title: Interlocking side milling cutter and cutting blade therefor (embodiments)
Inventor: NASTASENKO VALENTYN OLEKSIIOVYCH
IPC: B23C5/02
Filed: 2006-04-04
Abstract: An interlocking side milling cutter comprises a body with grooves, in which cutting blades without tool clearances are mounted. The cutting blades are installed tangentially in the grooves on the body sides and are multi-faceted with flats or cross grooves on the tops. The flats are made on the lateral surfaces of connection of the tops with a pressure angle. The flats eliminate transitional radius areas of the sides connection and form with the cutting edge formed a pressure angle at the top. The grooves are made in the range of radii of their cross-section from, which eliminates the transitional areas of interconnected pairs of lateral sides of the blade, and to, the value of which corresponds to the thickness of the cutting blade. The invention provides improvement of the cutting process by eliminating transitional radius surfaces of connection of sides at the tops of cutting blades.
Patent UA-87113-C2 (UA)
Title: Method for obtaining the suppository based on medicinal agent of placenta tissues
Inventor: SHYTOV HENNADII HAVRYLOVYCH
IPC: A61K9/02
Filed: 2006-04-11
Abstract: A process for obtaining of a suppository based on a medicinal agent provides for the stirring of the medicinal agent of placenta, which is freeze dried, with polyethylenoxide or lipid base followed by mass formation into a blister. The suppository contains the medicinal agen6, which is freeze dried in the amount of 0.07-.
Patent UA-81870-C2 (UA)
Title: Knee-joint mechanism for prosthesis of lower limb
Inventor: KIRIEIEV PAVLO MYKOLAIOVYCH
IPC: A61F2/64
Filed: 2006-09-11
Abstract: A knee-joint mechanism for the prosthesis of the lower limb contains the hinged upper and lower elements. The locking element is designed as the spring-loaded cylindrical post with the transversal axis contacting with the end-face of the flat guide block made as a whole with the upper part of the lower element. The guide block has the angular cut for enclosing the transversal axis with the negative slope in the direction of the folding of the upper and lower elements. The lower cylindrical part of the lower element is made with the collet. The design as a whole provides for the secure hinge fixation preventing the incidental actuation of the mechanism in walking thus precluding the traumas of the disabled persons.
Patent UA-89047-C2 (UA)
Title: Method for check of gas meters and device for its realization
Inventor: VOSCHYNSKYI VIKTOR STANISLAVOVYCH
IPC: G01F25/00
Filed: 2007-01-09
Abstract: Method for check of gas flow rate meters and device for its realization relate to means for measurement of gas flow rate and can be used for checking meters and flow rate meters for gas. Method for checking gas flow rate meters includes gas supply through installed in sequence checked gas flow rate meter and reference device for gas volume that perform measurement of gas passing through those flow rate, measurement of temperature and pressure of gas, reading information obtained, collection, transfer and processing of that information with determination of any point of flow rate by means of interpolation with cubic splines. Device consists of system of pipelines with two units for formation of gas flow, three reference units for gas volume and meter being checked, this is installed in sequence with standard of gas volume, temperature and pressure transformers, units for signal reading, system for collection, transfer and processing information and device as T-like pipeline for smoothening air that goes out from meter being checked pulses. Units for formation of gas flow have in their set micro-processor device that changes gas flow rate depending on information obtained by interpolation with cubic splines and that has interface connection with system for collection and processing information. Technical result is in decrease of error of measurement in broad range of characteristic and smooth change of gas flow rate with least errors and least power consumption.
Patent UA-88033-C2 (UA)
Title: Method for erection of berthing structures at weak soils
Inventor: YERMAKOV DMYTRO VLADYSLAVOVYCH
IPC: E02D7/24
Filed: 2007-06-04
Abstract: A method for erection of berthing structures on weak soils by which mounting base of the berthing structure is formed of multisection reinforced-concrete shells piles that are placed in rows in cross and long directions thereof and are deepened to the layer of compact grounds with increasing number of sections. After shell pile exceeds design height one arranges in its lower part a cement joggle. A top of the berthing structure is fixed to the base of the berthing structure with formation of a rear wall and underberthing slope. To decrease terms and to decrease material consumption at building, multisection shells piles are deepened to the bottom of water area up to the layer of compact grounds by washing out earth masses from inner cavity of each multisection shell pile through the hollow base of the lower section with water jet. The jet is formed by means of metal pipe with nozzle at the end placed to the inner cavity through which outside water is delivered under pressure with pump. The own weight of the shell pile and artificial mechanical load is used as additional vertical pressure.
Patent UA-94921-C2 (UA)
Title: 1-orthofluorophenyl substituted 1, 2, 5-thiazolidinedione derivatives as ptp-as inhibitors
Inventor: BARNES DAVID
IPC: A61K31/433
Filed: 2006-06-12
Abstract: , (I)Compounds of the formula (I) are inhibitors of protein tyrosine phosphatases (PTPases) and, thus, may be employed for the treatment of conditions mediated by PTPase activity. The compounds of the present invention may also be employed as inhibitors of other enzymes characterized with a phosphotyrosine binding region such as the SH2 domain. Accordingly, the compounds of formula (I) may be employed for prevention and/or treatment of insulin resistance associated with obesity, glucose intolerance, diabetes mellitus, hypertension and ischemic diseases of the large and small blood vessels, conditions that accompany type-2 diabetes, including hyperlipidemia, hypertriglyceridemia, atherosclerosis, vascular restenosis, irritable bowel syndrome, pancreatitis, adipose cell tumors and carcinomas such as liposarcoma, dyslipidemia, and other disorders where insulin resistance is indicated. In addition, the compounds of the present invention may be employed to treat and/or prevent cancer, osteoporosis, neurodegenerative and infectious diseases, and diseases involving inflammation and the immune system.
Patent UA-94926-C2 (UA)
Title: Process for saturation of liquid by oxygen and device for its realization
Inventor: FILIMONOV ROMAN VOLODYMYROVYCH
IPC: C02F1/72
Filed: 2008-07-07
Abstract: A process for the saturation of liquid by oxygen comprises filling of sealed tank by liquid with formation of zone of free space above the level of liquid and supply of oxygen under raised pressure into liquid from below through apertures at least one pipe, made spiral-shaped or zigzag bended in horizontal plane, and formed in the zone of free space excess of oxygen pressure, is discharged with the help of pressure release valve, besides the pressure is controlled using manometer and device for saturation of liquid by oxygen.
Patent UA-93927-C2 (UA)
Title: Method for production of non-woven fabric from fibers
Inventor: KHARKOVSKA MYROSLAVA VIKTORIVNA
IPC: D04H1/40
Filed: 2009-05-19
Abstract: A method for production of non-woven fabric made of fibers at which one performs production of fiber mix of uniform polymer fibers, bi-component polymer fibers with different melting temperature and additional fiber filler, with obtaining fibrous web, formation of layer and thermal bonding. One prepares polymer fiber and fiber of natural origin with length from 15 to . One mixes bi-component fibers suitable for thermal bonding in amount of from 15 to 25 wt. %, homogeneous polymer fibers in amount of from 25 to 65 wt. % and fibers of natural origin in amount of from 20 to 50 wt. %. One supplies fiber mix to hackling cylinders to obtain fibrous web with chaotically arranged fibers, this is laid in folds directed at angle from 15° to 90° to direction of motion of fabric in plane normal to main plane of layer that is formed, up to density from 0.15 kg/ mto 2.0 kg/ m. The layer obtained is pressed to given thickness and inclination of folds by transportation elements, heated with hot air, after that it is calendered.
Patent UA-94774-C2 (UA)
Title: Metastin derivatives and use thereof
Inventor: ASAMI TAIJI
IPC: A61K38/16
Filed: 2007-10-24
Abstract: The present invention provides stable metastin derivatives having excellent biological activities (a cancer metastasis suppressing activity, a cancer growth suppressing activity, a gonadotropic hormone secretion stimulating activity, sex hormone secretion stimulating activity, etc.). By substituting the constituent amino acids of metastin with specific amino acids, the metastin derivatives of the present invention achieve more improved blood stability, solubility, etc., reduced gelation tendency, improved pharmacokinetics, as well as exhibit an excellent cancer metastasis suppressing activity or a cancer growth suppressing activity. The melastin derivatives of the present invention also have a gonadotropic hormone secretion suppressing activity, sex hormone secretion suppressing activity, etc.
Patent UA-93016-C2 (UA)
Title: method for prognosing the progression of fibro-cystic breast disease during pregnancy
Inventor: ZHABCHENKO IRYNA ANATOLIIVNA
IPC: A61B5/15
Filed: 2009-06-24
Abstract: The invention relates to medicine, namely to obstetrics and concerns a method for prognosing the progression of fibro-cystic breast disease during pregnancy by study of estradiol concentration, insuline-like growth factor-1 and prolactin levels in pregnant women.
Patent UA-97504-C2 (UA)
Title: Method of reducing the risk of occurrence or delaying the occurrence of cancer in a subject using an anti-vegf-specific antagonist
Inventor: FERRARA NAPOLEONE
IPC: A61P35/00
Filed: 2007-12-18
Abstract: Disclosed herein are methods of treating benign, pre-cancerous, or non- metastatic tumors using an anti-VEGF-specific antagonist. Also disclosed are methods of treating a subject at risk of developing benign, pre-cancerous, or non-metastatic tumors using an anti-VEGF-specific antagonist. Also disclosed are methods of treating or preventing recurrence of a tumor using an anti-VEGF-specific antagonist as well as use of VEGF-specific antagonists in neoadjuvant and adjuvant cancer therapy.
Patent UA-98956-C2 (UA)
Title: A blocking device for electric vacuum cleaner
Inventor: KOSTECKI MARIUS
IPC: A47L9/24
Filed: 2008-03-31
Abstract: A blocking device is provided for the electric vacuum cleaner having an impurities tank (1) with an inlet opening (2) fitted with a bush (3) to air-tightly fasten the hose end (4), and a filtration receptacle (12), placed inside the impurities tank (1), fitted with a stiff plate (11) with an opening (19) which serves to fix this receptacle on the inner end of the bush (3). The blocking device has a slidable diaphragm (9) which covers the inlet opening (2) of the impurities tank (1) to make it impossible to fix the hose end (4) in the bush (3) if the plate (11) of the filtration receptacle (12) is not correctly installed on the inner end of the bush (3). The correct installing of the filtration receptacle (12) makes the diaphragm (9) move and the inlet opening (2) to be uncovered, which makes it possible to fix the hose end (4) in the bush (3) of the inlet opening (2).
Patent UA-99488-C2 (UA)
Title: Process for the preparation of treated brine from sea brine
Inventor: ANNOPOLSKYI VOLODYMYR FRIDRIKHOVYCH
IPC: C01F11/00
Filed: 2010-05-17
Abstract: A process for the preparation of treated brine from sea brine, comprising precipitation of sodium salt by means of natural evaporation, removal of stock brine, washing and solving of sodium salt with water, preliminary sulphatation of brine with component, containing sodium sulphate, further treatment of brine with lime and soda, settling of the purified brine, gathering and removal of brine purification sludge. As component, containing sodium sulphate, liquid phase is used, produced after treatment of brine purification sludge with sodium carbonate or its mixture with bicarbonate in quantity, sufficient for transformation of sludge components, containing calcium, to carbonate.
Patent UA-98381-C2 (UA)
Title: Side frame of freight bogie
Inventor: SAVCHUK OLEKSANDR VOLODYMYROVYCH
IPC: B61F5/52
Filed: 2010-09-27
Abstract: The invention relates to car building. A side frame of a freight bogie has an upper horizontal belt of closed section with cantilevers, which form axle holes, a lower belt of closed section with a support pad for a spring group, two inclined belts connecting upper and lower belts, vertical columns, process windows and a central spring hole. The latter is limited by the support pad for the spring group, upper belt and vertical columns. The frame also comprises radial transitions from the support pad to the vertical columns, inner ribs on inclined zones that are adjacent to the radial transitions, protrusions in the area of ​​contiguity of inner ribs to radial transitions, and an outer rib adjacent to the protrusions. The distance from the center of radial transition to the vertical column is less than the radius. The inner ribs adjacent to the radial transitions are connected with process windows along a tangent to their borders. The axis of each protrusion coincides with the line of intersection of the inner rib with the cylindrical surface of radial transition. The technical result is the increase of strength of the side frame in the area of the spring opening, its reliability and safety factor of fatigue resistance.
Patent UA-100597-C2 (UA)
Title: 2-hydroxy-n-(5-hydroxy-1-naphthyl)-2-(2-oxo-1,2-dihydro-3h-indole-3-ylidene)acetamide exhibiting anti-inflammatory and antimicrobial activity
Inventor: BOLOTOV VALERII VASYLIOVYCH
IPC: C07D209/34
Filed: 2011-05-10
Abstract: The invention relates to chemico-pharmaceutical field, in particular to a novel individual chemical compounds with bioactivity. Disclosed is 2-hydroxy-N-(5-hydroxy-1-naphthyl)-2-(2-oxo-1,2-dihydro-3H-indole-3-ylidene)acetamide of general formula:,exhibiting high anti-inflammatory and antimicrobial activity, which can be used as active substance in pharmaceutical preparations of different dosage forms.
Patent UA-101232-C2 (UA)
Title: Dc voltage regulator
Inventor: BAHATSKYI VALENTYN OLEKSIIOVYCH
IPC: G05F1/569
Filed: 2011-05-31
Abstract: A DC voltage regulator relates to electronic engineering and can be used for power supply of electronic devices. The DC voltage regulator with protection from overload current comprises a regulating element, resistor current-sensing device, control unit, differentiating amplifier, resistors. An electronic amplifier element is introduced, which input is connected to output of differentiating amplifier, first output is connected to second terminal of second resistor, first terminal of resistor current-sensing device, and second output of electronic amplifier element is connected to first control input of regulating element. The regulator disclosed provides elimination of dissipation power rise on regulating element at initial stages of protection circuit operation, reduction of input voltages of differentiating amplifier, enhancement of accuracy of protection operation current magnitude, simplification of the device.
Patent UA-106140-C2 (UA)
Title: Wheel set with adjustable wheels
IPC: B61F7/00
Filed: 2013-01-04
Abstract: The invention relates to railway rolling stock able to move on the lines with two different tracks. A wheel set with adjustable wheels comprises an axle, on which adjustable wheels are mounted with elongated parts of the center bosses facing each other, which are in engagement with fixed center bosses put on the axle. It also comprises a blocking sleeve, inside which the systems of compressible springs are installed and an expander sleeve having shape of a cup with a hole made in the bottom center with a thickened edge. The latter is adjacent to the surface of a conical hole located in the center of the bottom of blocking sleeve. Elongated parts of the center bosses are made in the form of sleeves rigidly connected to the wheels, on the inner surface of which splines are made engaged with the splines formed on the outer surface of the fixed center bosses. In the central part of the axle a fixed sleeve is secured, which is covered by an expander sleeve having on the outer cylindrical surface a protrusion, whose shape corresponds to the shape of annular grooves formed on the outer surface of the fixed sleeve. The expander sleeve is rigidly attached to one of the elongated parts of centre boss and another elongated part of the centre boss has grooves corresponding to the shape of the thickened edge of the expander sleeve from the inside. The systems of compressible springs are limited by the blocking and sliding sleeves. The technical result is the reduction of weight and size, skew when moving wheels, improving manufacturability.
Patent UA-105315-C2 (UA)
Title: Rye-wheat bakery product
Inventor: DOTSENKO VIKTOR FEDOROVYCH
IPC: A21D8/00
Filed: 2013-03-22
Abstract: The invention relates to rye-wheat bakery product containing rye and wheat flour, yeast, salt, the starter "Dark Ahram" and nettle powder.
Patent UA-105741-C2 (UA)
Title: Mobile maintenance device
IPC: B60P3/14
Filed: 2013-07-08
Abstract: A mobile maintenance device has a tractor trailer with a forklift on a rear suspension, a coupled trailed platform with a main unit mounted thereon with process equipment and a platform. To ensure stable and efficient operation of the process equipment at variable climatic conditions, it additionally has a tent with a gable roof, which comprises: halyards, two holes and curtains, seven windows of a film, a device for removal of exhaust gases of the tractor trailer, eight vertical folding racks, two horizontal folding racks of variable length, folders located in the upper part that form the walkways and driveways. Tent area change is determined by the formula:, where- area of a ​​mobile maintenance device,- area of machine-tractor unit,- coefficient taking into account the working zones.
Patent UA-110043-C2 (UA)
Title: Nanoscale palladium heterogeneous catalyst for performing cross-coupling reactions
Inventor: Sharanda Liudmyla Fedorivna
IPC: B01J23/44
Filed: 2013-07-16
Abstract: The invention relates to the field of organic chemistry, namely, creation of new nanoscale nonporous reusable heterogeneous palladium catalysts with a "core-carbon shell-palladium" structure, a method of their synthesis and their use in cross-coupling reactions, in particular Heck, Negishi, Suzuki, Kumada, Sonogashira reactions, where they exhibit a high catalytic activity.
Patent UA-106459-C2 (UA)
Title: Process for production of coke with high vcm content
Inventor: FAEGH AHMAD
IPC: C10L5/04
Filed: 2012-05-10
Abstract: A process and apparatus for improving the production of coke having a high volatile combustible material content are disclosed. The process may include, for example: heating a coker feedstock to a coking temperature to produce a heated coker feed-stock; contacting the heated coker feedstock with a quench medium to reduce a temperature of the heated coker feedstock and produce a quenched feedstock; feeding the quenched feedstock to a coking drum; subjecting the quenched feedstock to thermal cracking in the coking drum to (a) crack a portion of the quenched feedstock to produce a cracked vapor product, and (b) produce a coke product having a volatile combustible material (VCM) concentration in the range from about 13 % to about 50 % by weight, as measured by ASTM D3175.
Patent UA-107547-C2 (UA)
Title: A method for dna determination in the culture of lactococcus lactis subsp. cremoris in bacterial preparations and fermented foods by polymerase chain reaction
Inventor: VAKULENKO MYKOLA MYKHAILOVYCH
IPC: C12N15/09
Filed: 2013-02-25
Abstract: The invention relates to a method for DNA determination in the culture ofin bacterial preparations and fermented foods by polymerase chain reaction.
Patent UA-112330-C2 (UA)
Title: З'єднувальний пристрій для причепів самохідної робочої машини
IPC: F16C11/04
Filed: 2012-12-11
Abstract: Покращений з'єднувальний пристрій для причепа самохідної робочої машини має перший поворотний важіль (13), другий поворотний важіль (14) та третій поворотний важіль (15). Перший поворотний важіль (13) з'єднується або підключається до робочої машини приводом (18) рухомо (17). Другий поворотний важіль (14) з'єднаний з першим поворотним важелем (13) приводом (28) рухомо (27). Третій поворотний важіль (15) з'єднаний з другим поворотним важелем (14) приводом (32) рухомо (31) та підключається або з'єднується (29) з причепом. Осі повороту (27, 31) другого поворотного важеля (14) регулюються одна відносно одної по висоті.