baber/WOPTO huggingface dataset:
Patent JP-5324463-B2 (JP)
IPC: A61K31/43
Filed: 2006-12-10
Granted: 2013-10-23
Abstract: The novel positively charged pro-drugs of beta-lactam antibiotics in the general 'Structure 4' were designed. The positively charged amino group of the pro-drug not only makes the drugs soluble in water, but also bonds to the negative charge on the phosphate head group of membranes. This bonding will disturb the membrane a little bit and may make some room for the lipophilic portion of the prodrug. When the molecules of membrane move, the membrane may 'crack' a little bit due to the bonding of the prodrug. This will let the prodrug insert into the membrane. At pH 7.4, only about 99% of amino group is protonated. When the amino group is not protonated, the bonding between the amino group of the prodrug and the phosphate head group of membrane will disassociate, and the prodrug will enter the membrane completely. When the amino group of the prodrug flips to the other side of the membrane and thus become protonated, then the prodrug is pulled into the cytosol, a semiliquid concentrated aqueous solution or suspension. The results suggest that the pro-drugs diffuses through human skin, blood-brain, and blood-milk barriers hundreds times faster than do beta-lactam antibiotics. In plasma, more than 90% of these pro-drugs can change back to the parent drugs in a few minutes. The prodrugs can be used medicinally in treating beta-lactam antibiotics-treatable conditions in humans or animals. The prodrugs can be administered transdermally for any kind of medical treatments. Controlled transdermal administration systems of the prodrug enables beta-lactam antibiotics to reach constantly optimal therapeutic blood levels to increase effectiveness and reduce the side effects of beta-lactam antibiotics. Another great benefit of transdermal administration of these pro-drugs is that administering medication, especially to children or animals, will be much easier.
Patent JP-5305532-B2 (JP)
IPC: C12M1/00
Filed: 2007-12-13
Granted: 2013-10-02
Abstract: A scalable photobioreactor system for efficient production of photosynthetic microorganisms such as microalgae and cyanobacteria is described. In various embodiments, this system may include the use of extended surface area to reduce light intensity and increase photosynthetic efficiency, an external water basin to provide structure and thermal regulation at low cost, flexible plastic or composite panels that are joined together make triangular or other shapes in cross-section when partially submerged in water, use of positive gas buoyancy and pressure to maintain the structural integrity of the photobioreactor chambers and use of structure to optimize distribution of diffuse light. Other embodiments concern air tubes comprised of plastic film at the bottom of each photobioreactor chamber to provide sparging air bubbles to the chamber. The photobioreactor system design also comprises gas exchange, temperature control, air pumping, liquid pumping, filtration, media recycling and harvesting methods. For biofuels production, the photobioreactor system can comprise a separate growth photobioreactor and secondary stress reactor.
Patent JP-5244124-B2 (JP)
IPC: G06F3/06
Filed: 2008-01-03
Granted: 2013-07-24
Abstract: Embodiments of the present invention relate to an apparatus, method and computer readable medium for recovering from a failed or aborted outgoing data transfer operation from a host device to a peripheral storage device. In some embodiments, before the peripheral storage device is corrupted by the failed outgoing data transfer operation, one or more recovery data objects are stored on the host-side. After the peripheral storage device is corrupted by the failed data transfer, the host device responds to a subsequent coupling with the peripheral storage device by repairing the corrupted peripheral storage device using one or more of the host-side stored recovery data objects. Optionally, the host device also restores the outgoing aborted or failed data transfer operation.
Patent JP-5327096-B2 (JP)
IPC: F21S2/00
Filed: 2010-02-23
Granted: 2013-10-30
Abstract: A lamp with ferrule 10 includes a substrate 12 in which a solid light-emitting device 11 is implemented on one surface side thereof, a thermal radiation member 14 which is fixed to the other surface side of the substrate 12 by a fluid fixing member 13 having thermal conductivity; a light-emitting portion 15 constituted by the substrate 12 and the thermal radiation member 14; a thermally conductive support member 17 which constitutes a three-dimensional light source body 16 using a plurality of light-emitting portions 15; a thermally conductive main body 18 which is provided with the support member 17 so as to project the three-dimensional light source body 16 to the one end portion side; and a ferrule member 19 that is provided on the other end portion side of the main body 18.
Patent JP-5068834-B2 (JP)
IPC: F04D25/08
Filed: 2010-03-02
Granted: 2012-11-07
Abstract: A fan assembly for creating an air current includes a nozzle mounted on a base. The base includes an outer casing, a silencing member housed within the outer casing, an impeller housing located within the outer casing, the impeller housing having an air inlet and an air outlet, an impeller located within the impeller housing and a motor for driving the impeller about an axis to create an air flow through the impeller housing. The nozzle includes an interior passage for receiving the air flow from the air outlet of the impeller housing and a mouth through which the air flow is emitted from the fan assembly. The silencing member is located beneath the air inlet of the impeller housing and is spaced from the air inlet along said axis by a distance in the range from 5 to 60 mm.
Patent JP-5684500-B2 (JP)
IPC: C08G65/26
Filed: 2010-06-23
Granted: 2015-03-11
Abstract: The present invention provides a process for the polyoxyalkylation of a starter involving establishing oxyalkylation conditions in an oxyalkylation reactor in the presence of a double metal cyanide (DMC) catalyst, continuously introducing into the reactor at least one alkylene oxide and an acidified, ultra-low water content starter, in which the starter contains greater than 100 ppm and less than or equal to 500 ppm water, based on the weight of the starter, and recovering an oxyalkylated low molecular weight starter polyether product. The inventive process allows the production of short chain polyether polyols which have hydroxyl numbers of from greater than 250 up to 500, from hygroscopic initiators, such as glycerin, without DMC catalyst deactivation.
Patent JP-5357115-B2 (JP)
IPC: H04S5/02
Filed: 2010-07-20
Granted: 2013-12-04
Abstract: A method for optimizing the acoustic localization at at least one listening position within a listening room is disclosed. A sound field being generated by a group of loudspeakers assigned to the least at one listening position, wherein the group of loudspeakers comprises a first and at least a second loudspeaker each being supplied by an audio signal via an audio channel. The method comprises calculating filter coefficients of a phase equalization filter for at least the audio channel supplying the second loudspeaker, whereby the phase response of the phase equalization filter is designed such that a binaural phase difference on the at least one listening position or a mean binaural phase difference averaged over more than one listening positions is minimized within a predefined frequency range and applying the phase equalization filter to the respective audio channel.
Patent JP-5307097-B2 (JP)
IPC: H04W64/00
Filed: 2010-09-13
Granted: 2013-10-02
Abstract: Different types of position solutions may be used to determine the position of a mobile station (104) in a wireless communication system (101). The position solutions include terrestrial, or network (102, 103), based techniques and non-network, such as satellite (160), based techniques. An apparatus and method whereby different position solutions are selected based on a figure of merit of the different solutions in determining a position of a mobile remote unit (104).
Patent JP-5341045-B2 (JP)
IPC: F02M61/18
Filed: 2010-09-30
Granted: 2013-11-13
Abstract: <P>PROBLEM TO BE SOLVED: To provide a fuel injection valve device capable of efficiently adding a swirl to fuel in a swirl chamber.  <P>SOLUTION: A communication path is formed such that a distance between a first side surface on the radial outside where fuel rotates in a swirl adding chamber as a side surface of the communication path and a line extended in the radial direction of a center chamber is shorter than a distance between a second side surface in the radial inside where fuel rotates in the swirl adding chamber as the side surface of the communication path and a line extended in the radial direction of the center chamber.  <P>COPYRIGHT: (C)2012,JPO&INPIT
Patent JP-5341047-B2 (JP)
IPC: H05K1/18
Filed: 2010-10-12
Granted: 2013-11-13
Abstract: <P>PROBLEM TO BE SOLVED: To provide a component support substrate capable of forming resin filling portions suitable for forming fitting holes.  <P>SOLUTION: A component support substrate of the present invention includes a substrate 11, resin filling portions 22, and component support bodies 24. The substrate 11 has filling holes 21 opening at least at a first principal surface 12. The resin filling portions 22 are provided inside the filling holes 21, are formed from a material lower in hardness than the substrate 11, and have fitting holes 23 opening on the first principal surface 12 side. The component support bodies 24 are fixed by being fit into the fitting holes 23 and are capable of supporting other components at positions projecting from the fitting holes 23. End faces on the first principal surface 12 side of the resin filling portions 22 are positioned on a second principal surface 13 side with respect to the first principal surface 12.  <P>COPYRIGHT: (C)2012,JPO&INPIT
Patent JP-5362703-B2 (JP)
IPC: C07C67/14
Filed: 2008-03-19
Granted: 2013-12-11
Abstract: This invention relates to a method of producing a compound represented by the following general formula (3):   
[wherein R is a bivalent aliphatic group having a carbon number of 1-16 or a bivalent aromatic group], which comprises a step (i) of reacting a compound represented by the following general formula (1):   
with a carboxylic acid halide represented by the following general formula (2):   
[wherein R is a bivalent aliphatic group having a carbon number of 1-16 or a bivalent aromatic group and X is a halogen atom] in the presence of a basic compound to form an ester, and a step (ii) of conducting a heat treatment after the step (i) to decompose an oligomer in the ester.
Patent JP-5335004-B2 (JP)
IPC: G10L19/12
Filed: 2010-02-12
Granted: 2013-11-06
Abstract: An LSP vector quantization device able to improve the precision of quantization in vector quantization where a codebook for first stage vector quantization is switched according to the type of a feature that has a correlation with the quantization target vector. In this device, a classifier (101) selects, from a plurality of code vectors for classifying, the code vector for classifying that indicates the type of the feature that has a correlation with the quantization target vector; a switch (102) selects, from among a plurality of first codebooks, the first codebook corresponding to the abovementioned type; an error minimizing unit (105) selects, from the plurality of first code vectors constituting the selected first codebook, the first code vector closest to the quantization target vector; a matrix determining unit (106) selects, from a plurality of matrices, the matrix corresponding to the abovementioned type; and the error minimizing unit (105) uses the selected matrix to select, from a plurality of second code vectors, the one that is closest to the residual vector between the selected first code vector and the quantization target vector.
Patent JP-5136660-B2 (JP)
IPC: B60L50/16
Filed: 2011-02-02
Granted: 2013-02-06
Abstract: An output shaft is arranged to be lateral and parallel to engine input shafts and a motor input shaft. An engine side gear mechanism for transmitting a power of the engine input shafts to the output shaft is provided. A motor side gear mechanism for transmitting a power of the motor input shaft to the output shaft is provided. An input side clutch engages and disengages the engine input shafts and the motor input shaft. When the input side clutch is engaged, the power transmission between a position where the engine side gear mechanism is arranged on the engine input shafts and a position where the motor side gear mechanism is arranged on the motor input shaft is invariably possible.
Patent JP-5358616-B2 (JP)
IPC: E02B7/20
Filed: 2011-04-21
Granted: 2013-12-04
Abstract: <P>PROBLEM TO BE SOLVED: To provide an intake device for make-up water, capable of automatically adjusting an intake amount from a river corresponding to the change of a water level of an intake channel in a simple configuration without using electric control.  <P>SOLUTION: An intake device for make-up water comprises a communication passage 2 for communicating a mountain stream 103 and an intake channel 101, and an intake amount adjusting part 10 for mechanically adjusting a flow rate of water W3 flowing into the intake channel 101 through the communication passage 2 from the mountain stream 103 by a float 13 vertically moved accompanying the change of the water level of water W2 flowing through the intake channel 101. The intake amount adjusting part 10 supplies a water amount corresponding to the water level of the intake channel 101 from the mountain stream 103 to the intake channel 101 when the water level of the intake channel 101 is within a prescribed range, supplies an allowable maximum water amount from the mountain stream 103 to the intake channel 101 when the water level of the intake channel 101 is below the prescribed range, and inhibits the supply of the water W3 from the mountain stream 103 to the intake channel 101 when the water level of the intake channel 101 exceeds the prescribed range.  <P>COPYRIGHT: (C)2013,JPO&INPIT
Patent JP-4934757-B2 (JP)
IPC: H04L27/00
Filed: 2011-12-07
Granted: 2012-05-16
Abstract: <P>PROBLEM TO BE SOLVED: To avoid setting of a modulation class higher than necessary when user data which is transmitted to a communication destination device does not exist or user data to be transmitted is very small.  <P>SOLUTION: A radio communication method, which uses a radio communication apparatus selecting a modulation class according to propagation path quality, includes steps S13A, 13B for selecting a modulation class corresponding to a predetermined data amount when it is determined that a detected data amount is equal to or smaller than a predetermined data amount.  <P>COPYRIGHT: (C)2012,JPO&INPIT
Patent JP-5363560-B2 (JP)
IPC: B01D17/022
Filed: 2009-04-15
Granted: 2013-12-11
Abstract: A fuel filter system, especially for Diesel engines includes filter housing (1) having a fuel inlet (27) and a fuel outlet (29) and a dehydrating filter medium (23) between the inlet and the outlet for the fuel to pass through. The filter housing (1) has a collection chamber (35) for the water trapped by the filter medium from which collection chamber the water can be supplied to a water absorbing and evaporating device (49) via a controlled dispenser (45). The components of the evaporating steam are releasable into the environment through the evaporating steam outlet (51). The water absorbing and evaporating device (49) has a valve arrangement (59, 61) by which the evaporating water outlet (51) can be closed depending on an inadmissible amount of non-evaporated water (55) collected in the evaporating device (49).
Patent JP-5351967-B2 (JP)
IPC: B24D3/34
Filed: 2009-07-30
Granted: 2013-11-27
Abstract: A structured abrasive article comprises an at least translucent film backing and an abrasive layer disposed on the backing. The abrasive layer comprises a plurality of shaped abrasive composites. The shaped abrasive composites comprise abrasive particles dispersed in a binder. The abrasive particles consist essentially of ceria particles having an average primary particle size of less than 100 nanometers. The binder comprises a polyether acid and a reaction product of components comprising a carboxylic(meth)acrylate and a poly(meth)acrylate, and, based on a total weight of the abrasive layer, the abrasive particles are present in an amount of at least 70 percent by weight. Methods of making and using the structured abrasive article are also disclosed.
Patent JP-5267685-B2 (JP)
IPC: B60L50/16
Filed: 2010-01-29
Granted: 2013-08-21
Abstract: A vehicle control device of a vehicle that can travel with inertia without transmitting power of an engine (10) to drive wheels (WL, WR) and stops an operation of an engine (10) that generates power by fuel during an inertia travel as well as prohibits a regeneration control of a regeneration device (50) that regenerates kinetic energy during a travel, wherein when it is estimated that predetermined energy in various types of energy in a vehicle fluctuates during the inertia travel, a regeneration control prohibition state of the regeneration device (50) is released during the inertia travel.
Patent JP-5341222-B2 (JP)
IPC: H04L9/08
Filed: 2012-03-29
Granted: 2013-11-13
Abstract: Techniques for sending information without interruption during a change in ciphering configuration are described. A user equipment (UE) communicates with a wireless communication network for a call. The UE sends first information to the wireless network using a first ciphering configuration. For a change in ciphering configuration, the UE selects an activation time for a second ciphering configuration and sends a security message with the activation time. This activation time is the time at which the UE applies the second ciphering configuration to transmission sent to the wireless network. The UE thereafter sends second information (e.g., a measurement report message) using the first ciphering configuration after sending the security message and before the activation time. The UE sends third information using the second ciphering configuration after the activation time.
Patent JP-5084961-B2 (JP)
IPC: C08F212/14
Filed: 2012-03-30
Granted: 2012-11-28
Abstract: To provide a polymeric compound having superior charge-providing properties, the polymeric compound contains at least one unit represented by the following general formula (5). In the general formula (5), R1 represents a hydrogen atom or an alkyl group; R2 to R4 each represent a hydrogen atom, an alkyl group, an alkoxy group, a hydroxyl group or a halogen atom, or R3 and R4 may combine each other to form a ring; and A represents a divalent linking group.
Patent JP-5524270-B2 (JP)
IPC: C07K16/28
Filed: 2012-04-13
Granted: 2014-06-18
Abstract: Isolated monoclonal antibodies or an antigen binding portion thereof which bind to prostate specific membrane antigen in its native form occurring on the surface of tumor cells characterized in that it is linked to a label or a cytotoxic agent or constructed as a part of a bispecific antibody or a recombinant diabody.
Patent FR-2971705-B3 (FR)
Inventor: MENOUD EDMOND JEAN
IPC: A61G7/10
Filed: 2011-06-23
Granted: 2013-03-22
Abstract: The trolley has a retractable support mattress formed of a set of actuators, where the actuators are cooperated with each other for supporting a body of a patient (8). Each of the actuators includes a control valve formed of a permanent magnet. The valve is opened automatically when magnetic members i.e. gloves, approach the valve. The mattress is arranged inside a shroud (3). The shroud is provided with a suction system and a polluted air treatment unit (6). A sealed and non-magnetic flexible membrane is interposed between the patient and one of the actuators.
Patent FR-3110524-B3 (FR)
Title: Dispositif de rangement dispose sur un panneau interieur d’un vehicule
Inventor: PATIL SAGAR
IPC: B60R7/06
Filed: 2020-05-20
Granted: 2022-06-17
Abstract: DISPOSITIF DE RANGEMENT DISPOSE SUR UN PANNEAU INTERIEUR D’UN VEHICULE La présente invention est prévue pour proposer un compartiment de rangement (100) disposé sur un panneau intérieur d’un véhicule. Le compartiment de rangement (100) comprend :  - un boîtier (50) définissant un espace de rangement pour ranger des articles,  - un couvercle (110) avec une patte pivotante (112) agencée de manière pivotante afin de déplacer le couvercle (110) autour d’un axe de pivot entre une position ouverte et une position fermée,  - un élément de verrouillage agencé sur une périphérie externe (101) du boîtier (50), et  - un élément de butée (130) faisant saillie de la patte pivotante (112) du couvercle (110) de sorte que l’élément de butée (130) est adapté pour venir en butée et se mettre en prise avec l’élément de verrouillage flexible (120) pour maintenir le couvercle (110) dans la position ouverte (100a).  Figure pour l'abrégé : Figure 4
Patent DE-10241538-B3 (DE)
Title: Traffic routing system accessed via computer or mobile telephone, has user response information used for continuous updating of dynamic databank used for route planning or traffic prognosis
Inventor: WOESLER RICHARD
IPC: G07B15/06
Filed: 2002-09-05
Granted: 2004-04-22
Abstract: The routing system (1) responds to interrogation information received from a user for providing the user with a route and its associated traffic prognosis and/or a traffic prognosis for a known route, using information held in a dynamic databank (11). The user transmits a response to the routing system upon reception of the route information, used for updating the dynamic databank dependent on if and when the route is to be followed.  An Independent claim for a traffic routing method is also included.
Patent DE-10255567-B3 (DE)
Title: Probenentnahme aus tiefen Bohrungen
Inventor: MUSACK MARTIN
IPC: E21B49/08
Filed: 2002-11-28
Granted: 2004-01-22
Abstract: Die Erfindung beschreibt eine Vorrichtung, mit der Materialproben aus tiefen Bohrungen entnommen werden können.
Patent DE-10303475-B3 (DE)
Title: Maximum-Likelihood-Abschätzung der Kanalkoeffizienten und des DC-Offset in einem digitalen Basisbandsignal eines Funkempfängers mit dem SAGE-Algorithmus
Inventor: HEDDERGOTT RALF
IPC: H04L25/06
Filed: 2003-01-29
Granted: 2004-10-07
Abstract: Das vorgeschlagene iterative Verfahren berechnet simultan Maximum-Likelihood-Schätzwerte für die Kanalkoeffizienten (h¶0¶, ..., h¶L¶, THETA¶h¶) und den DC-Offset (d; THETA¶d¶) auf der Basis einer Trainingssequenz (TSC) in einem TDMA-Mobilkommunikationssystem. Der SAGE-Algorithmus führt auf zwei Rekursionsformeln, durch die die iterative Berechnung von Schätzwerten für die Kanalkoeffizienten (h¶0¶, ..., h¶L¶, THETA¶h¶) und den DC-Offset (d; THETA¶d¶) bereitgestellt wird.
Patent DE-19861413-B3 (DE)
Title: Electronic timepiece has a simple calendar with a control circuit deciding the number of days required using a permanent calendar circuit to drive a date plate
Inventor: HIGUCHI HARUHIKO
IPC: G04C3/00
Filed: 1998-12-25
Granted: 2012-06-14
Abstract: Electronic timepiece includes a month-end non-correction device for a simple calendar. The timepiece is provided with a date detection plate (71) composed of a reflection part and a non-reflection part formed on the rear surface of a date plate (70). The transition across the boundary is read by a photosensor (81) when the date plate (70) rotates and the number of days required by a control circuit (20) is decided by a permanent calendar circuit to drive a date plate means (51,52).