baber/WOPTO huggingface dataset:
Patent FI-850829-L (FI)
Inventor: BUNDGAARD HANS
IPC: A61P43/00
Filed: 1985-02-28
Abstract: The invention relates to compounds of the general formulae Ia and Ib <IMAGE> where R1 is a group of the formula II R3-CO-A- where R3 is alkyl; mono- or poly-halogenated lower alkyl; phenyl, or substituted phenyl, or R3 is an aromatic heterocyclic 5- or 6-ring which contains one or two hetero atoms selected from a group which consists of nitrogen, oxygen and sulphur; and A is a single bond or a group of the formula IIa -O-CR6R7- where the carbon atom is connected to the nitrogen atom in the primary ring system and where R6 and R7 are identical or different and each represents hydrogen or has the same meaning as R3; or R1 is a group of the formula III R8R9N-Y- CO-A- where R8 and R9 are identical or different and each represents hydrogen or has the same meaning as R3; or R8 and R9, together with the adjacent nitrogen, form a heterocyclic 5- or 6-ring which, in addition to the nitrogen, can contain one or two further hetero atoms selected from a group which consists of nitrogen, oxygen and sulphur; Y is a single bond or a group of the formula IIIa (-CR6R7)n where n is an integer from 1 to 5 and A, R6 and R7 are defined as above; or R1 is a group of the formula IV R'3-O-CO-A where A is defined as above and R'3 has the same meaning as R3 as was defined above, with the proviso that R'3 is not ethyl when A is a bond; or R1 is a group of the formula VII R13-CO-(CH2)n- CO-A- when n and A are defined as above, and R13 is hydroxyl or a group of the formula -NR8R9 where R8 and R9 are defined as above; or R1 is a group of the formula IX (HO)2PO2-CR6R7- where R6 and R7 are defined as above; R2 is one of the groups II, III, IV and VII as were defined above, with the proviso that A is only the group IIa as was defined above; and R5 is hydrogen or has the same meaning as R2 as was defined above, and salts thereof. The compounds according to the formulae Ia and Ib are prodrugs of allopurinol and possess, inter alia, a much higher solubility in water and/or higher lypophilicity than does allopurinol.
Patent FI-852138-L (FI)
Inventor: KLAVENESS JO
IPC: A61K49/00
Filed: 1985-05-29
Abstract: There are provided NMR contrast agents comprising water-soluble paramagnetic metal chelates, preferably of Cr(III), Fe(III) or Gd (III), wherein the chelating entity is an anilide group containing organic moiety, preferably a compound of formula Iwherein R<sup>1</sup> to R<sup>5</sup> may represent hydrogen or halogen atoms, optionally halogenated alkyl or alkyoxy groups or carboxyl groups. The agents are especially suitable for use in NMR imaging of the hepatobiliary system.
Patent IE-831144-L (IE)
Title: Oligopeptide prodrugs
IPC: C07K7/04
Filed: 1983-05-17
Abstract: Prodrugs are described whose structures have a oligopeptide chain which is substituted by a nucleophilic chemotherapeutic residue at the  alpha -position. The products have increased cell membrane permeability and beneficial physico-chemical properties.
Patent IE-801485-L (IE)
Title: Unsaturated steroids
IPC: C07J13/00
Filed: 1980-07-17
Abstract: A process for preparing a DELTA 9(11)- and/or DELTA 16-unsaturated steroid comprises heating the corresponding steroid of the pregnane series substituted by 9 alpha -chloro- and/or 16 alpha -chloro- or 17 alpha -acyloxy, in an inert, aprotic high-boiling solvent at 180 DEG -350 DEG C.
[US4290963A]
Patent IE-821502-L (IE)
Title: Delta-8,9- prostanes
IPC: C07C35/06
Filed: 1982-06-24
Abstract: DELTA 8,9-Prostane derivatives of Formula I   <IMAGE>   wherein R1 is CH2OH or   <IMAGE>  wherein R2 is hydrogen, alkyl, cycloalkyl, aryl, or a heterocyclic residue; or R1 is   <IMAGE>   wherein R3 is an acid residue or R2; A is -CH2-CH2- or cis-CH=CH; B is -CH2-CH2-, trans-CH=CH- or -C 3BOND C- W is a free or functionally modified hydroxymethylene group or free or functionally modified   <IMAGE> wherein the OH-group can be in the  alpha - or  beta - position; D and E jointly are a direct bond or D is straight chain or branched alkylene or alkenylene of 1-10 carbon atoms which can optionally be substituted by fluorine atoms, and E is oxygen, sulfur, a direct bond, -C 3BOND C- or -CR6=CR7-, wherein R6 and R7 differ from each other and each is hydrogen, chlorine or alkyl; R4 is free or functionally modified hydroxy and R5 is an optionally substituted aliphatic group, cycloalkyl, optionally substituted aryl, or a heterocyclic group, and when R2 is hydrogen, physiologically compatible salts thereof with bases, have valuable pharmacological properties, e.g. luteolytic and abortifacient activities.
Patent IE-39535-L (IE)
Title: A wall construction
IPC: E06B7/14
Filed: 1973-10-15
Abstract: There is provided an improved wall construction including a vertical mullion assembly and a horizontal member assembly. Both assemblies are formed of interlocking gutter and face sections defining opposed glazing channels. The horizontal member assembly is provided with a pair of longitudinally extending screw splines. The assemblies may be joined in accordance with an improved shear pin system wherein the vertical mullion assembly is prepared for attachment of a horizontal member by drilling holes to receive the head of a shear pin and a dowel pin. The horizontal members are prepared by the insertion of a shear pin into one of the screw splines formed in the horizontal member and by the insertion of a dowel pin into the other of the screw splines formed in the horizontal member assembly. The horizontal member is then attached to the vertical by intalling the heads of the shear pin and the dowel pin into the holes previously drilled for them.
[US3797191A]
Patent IE-39957-L (IE)
Title: Steroid formulation
IPC: A61K47/10
Filed: 1973-10-22
Abstract: A steroid formulation having enhanced properties for topical application comprises 21-chloro-9 alpha -fluoro- DELTA 4-pregnene-11 beta ,16 alpha ,17 alpha -triol-3,20-dione 16,17-acetonide in a vehicle containing as major ingredients propylene glycol and water.
[US3892857A]
Patent IE-43721-L (IE)
Title: Improving animal nutrition using salinomycin
IPC: A23K20/195
Filed: 1976-09-10
Abstract: The feed additive to promote nutrient conversion and growth in ruminants and animal species with a similar physiology of the digestive system contains salinomycin, its physiologically acceptable salts and/or esters and carrier material. The feed additive can be given together with the feed or before or after feeding.
[GB1562805A]
Patent IE-892462-L (IE)
Title: Detection and treatment of infectious and inflammatory¹lesions
IPC: A61K47/48
Filed: 1989-07-28
Abstract: A polyspecific anti-leukocyte antibody conjugate for targeting foci of leukocyte accretion comprises an immunoreactive polyspecific composite of at least two different substantially monospecific antibodies or antibody fragments, conjugated to at least one imaging agent, wherein at least two of said antibodies or antibody fragments specifically bind to different leukocyte cell types. A method for targeting an imaging agent to an inflammatory or infectious lesion comprises injecting a mammal parenterally with an effective amount for targeting of the above anti-leukocyte imaging conjugate. A therapeutic anti-leukocyte conjugate for targeting foci of leukocyte accretion comprises at least one immunoreactive substantially monospecific antibody or antibody fragment which specifically binds to at least one leukocyte cell type, conjugated to a therapeutic antimicrobial agent, boron addend and/or radionuclide. A method of treatment of an infectious lesion comprises injecting a mammal parenterally with an effective amount for therapy of the above anti-leukocyte therapeutic conjugate.
Patent IE-802706-L (IE)
Title: Semiconductor manufacture
IPC: H01L23/64
Filed: 1980-12-22
Abstract: A plural layered wiring which comprises a plurality of polycrystal semiconductor layers can be improved in its magnitude of circuit integration, when one or more upper polycrystal semiconductor layers which is or are doped to a moderate impurity concentration is or are utilized as resistor elements, the lowest polycrystal semiconductor layer which is highly doped is utilized for electrodes and/or wirings for active elements, and both polycrystal layers are connected with each other by regions which are highly doped by upward diffusion of impurities contained in highly doped regions of a substrate, because this configuration entirely avoids the restriction that is imposed for the location of resistor elements arranged in the upper layers. This arrangement is realized by a specific sequential combination of steps which includes a step of upward diffusion of impurities from the highly doped regions of the substrate. An additional advantage of this method is the exclusion of a so-called non-butting process.
[US4399451A]
Patent IE-812728-L (IE)
Title: Metallizing a silicon solar cell
IPC: H01L31/0224
Filed: 1981-11-20
Abstract: A silicon solar cell is metallized with a nickel-antimony alloy to provide external contacts.
[US4342795A]
Patent IE-872903-L (IE)
Title: Device for coupling a longitudinal testpiece and a drawing¹head
IPC: G01N3/04
Filed: 1987-10-28
Abstract: The invention relates to a device for coupling a longitudinal metal specimen (1) to a tensile-testing device (4, 5), the specimen being subjected to tensile tests and comprising a flattened rectangular cross-section with two large surfaces (6, 7) and two small surfaces (8, 9). According to the invention, the end (2, 3) of the specimen has a general arrow shape such that the said two small surfaces (8, 9) are inclined towards each other there, whilst the two large surfaces remain parallel to each other, such that the said inclined surfaces are provided with sawtooth-section parallel grooves (13) extending perpendicularly to the axis of the specimen, the teeth being inclined in the same direction as the said surfaces, and such that the tensile- testing device comprises a rigid counterpiece (11) of a shape complementing that of the arrow-shaped end of the specimen (1), the length of the grooves of this counterpiece being at least equal to that of the grooves (13) on the specimen (1). <IMAGE>
[EP0267492A1]
Patent IE-892998-L (IE)
Title: Pharmaceutical composition
IPC: A61K31/34
Filed: 1989-09-19
Abstract: The invention provides a pharmaceutical composition for use in human or veterinary medicine which comprises ranitidine or a physiologically acceptable salt thereof, alginic acid or a physiologically acceptable salt thereof, and a carbonate or bicarbonate. The composition preferably comprises 1.25% to 10% w/w ranitidine hydrochloride, 5% to 35% w/w alginic acid, and 2% to 15% w/w sodium bicarbonate and is preferably in the form of a capsule or tablet. The compositions are suitable for the treatment of gastrointestinal disorders and particularly reflux oesophagitis.
[US5456918A]
Patent IE-893026-L (IE)
Title: Wired glass
IPC: B32B17/10
Filed: 1989-09-21
Abstract: A wired glass having a wire mesh formed of wires coloured to have a different visual appearance to metallic wires employed in conventional wired glass. Preferably the wire mesh has an applied decorative coating of different colour to the colour of the cores of the metallic wires forming the wire mesh. The decorative coating suitably provides the wired glass with an attractive visual appearance.
[EP0361872A1]
Patent IE-853193-L (IE)
Title: Process for fabricating a device
IPC: H01L21/306
Filed: 1985-12-17
Abstract: Process for fabricating a device, including etching of a substrate with a chlorine-containing plasma. By adjusting the AC field conditions, e.g., by grounding the environment of the substrate being etched, a significant increase in etch selectivity is achieved. By applying a similar AC field adjustment to the reaction chamber surfaces, excellent etch uniformity is achieved in conjunction with excellent selectivity.
[WO8603887A2]
Patent NO-763311-L (NO)
Inventor: TAKAHASHI S
IPC: F16G13/12
Filed: 1976-09-28
Abstract: Kj éttingledd.
Patent NO-810479-L (NO)
Inventor: KARJALAINEN ARTO JOHANNES
IPC: C07D233/64
Filed: 1981-02-12
Abstract: The invention provides compounds of the formula:wherein each of R<sub>1</sub>, R<sub>2</sub> and R<sub>3</sub>, which can be the same or different is hydrogen, chloro, bromo, fluoro, methyl, ethyl, methoxv, amino, hydroxy or nitro; R<sub>4</sub> is hydrogen or alkyl of 1 to 7 carbon atoms; X is(R<sub>5</sub> is hydrogen or hydroxy) and n is 1-4; and their non-toxic pharmaceutically acceptable acid addition salts. These compounds exhibitvaluable pharmacological activity and are useful in the treatment of mammals, especially as anti- hypertensive agents. Furthermore, some of the compounds have proved to possess diuretic, ß-blocking activity and/or antithrombotic activity. The compounds may be made by a variety of methods and may be incorporated in pharmaceutical compositions also comprising a compatible pharmaceutically acceptable carrier.
Patent NO-840953-L (NO)
Inventor: PADLY YVAN
IPC: A23B5/04
Filed: 1984-03-13
Abstract: A process for the continuous pasteurisation of eggs characterised in that liquid egg material is passed under a superatmospheric operating pressure through a first scraped surface heat exchanger to raise the temperature of the egg material to the pasteurisation temperature after which it is passed to a heated holding vessel under pressure of a sterile inert gas for a period of time which ensures pasteurisation but which is sufficiently short to ensure that substantially no coagulation occurs, and finally through a second scraped surface heat exchanger where it is cooled to a temperature below 10°C over a period of time less than 5 minutes.
Patent NO-841841-L (NO)
Inventor: MUELLER RICHARD AUGUST
IPC: C07C67/00
Filed: 1984-05-08
Abstract: This invention relates to novel compounds for preventing or retarding the degradation of elastin or other proteins and therefore preventing or retarding the disease states caused by said degradation, of the formula:  <IMAGE>  or its pharmacologically acceptable salts. The invention also relates to novel methods and intermediates for making the compounds.
Patent NO-850431-L (NO)
Title: Anordning ved varmeveksler.
Inventor: GYLLENSTEN JOERGEN
IPC: F28F1/12
Filed: 1985-02-05
Abstract: Anordning ved varmeveksler som har innbyrdes parallelle flenser (3, 4). I rommet mellom flensene bringes luft til å strømme ved hjelp av en vifte eller lignende. Karakteristisk for oppfinnelsen er det faktum at arrangementet omfatter en anordning (5) som er laget av termisk ledende materiale. Denne er konstruert til å passe inn i nevnte rom i termisk kontakt med flensene (3, 4) på begge sider og er slik konstruert at når den er plassert mellom flensene (3, 4), bevirker den en oppdeling av rommet mellom flensene i en flerhet parallelle kanaler (6a, 6b,..).
Patent NO-861102-L (NO)
Inventor: CONDOLIOS ELIE
IPC: C02F1/52
Filed: 1986-03-20
Abstract: A cloudy liquid to be clarified is inserted, after twice receiving flocculation additive, into the bottom of a belt of sludge (4a) in a clarification chamber (4) via a plurality of injectors (22) distributed over the area of said chamber. Uniform distribution of overall flow between these injectors is ensured by internal head loss. The clarified liquid is removed via an upper overflow (4b). Each injector is constituted by a flat cyclone and forms a jet which is highly diverting from its vertical axis in such a manner that the injected flowrate spreads out over an expansion zone belonging to said injector and meeting the expansion zones of adjacent injectors. Further, these jets set up swirling motion which prevents the formation of a layer of sludge having insufficient permeability. The sludge formed in the chamber (4) is directed via a central well (7) towards a secondary clarification sludge (3) situated beneath said chamber and supplying both clarified liquid and dense sludge.
Patent NO-863009-L (NO)
Inventor: KOLTS JOHN HENRY
IPC: C07C4/06
Filed: 1986-07-25
Abstract: Compositions of matter, including: A mixture of at least one oxide of manganese and at least one oxide of a Lanthanum Series metal, preferably lanthanum or cerium, or at leaat one oxide of niobium. The above compositions are particularly useful as catalytic compositions for the conversion of C<sub>3</sub> and C<sub>4</sub> hydrocarbons to less saturated hydrocarbons, particularly ethylene and propylene and preferably ethylene. The life of the catalyst for the selective production of ethylene is extended by carrying out the reaction in the presence of steam. The steam substantially increases the active life of the catalytic composition, before regeneration is necessary, as well as significantly increasing the selectivity to ethylene. Limiting the amount of "bound" or "fixed" sulfur in the catalytic composition also improves the catalyst.
Patent NO-865160-L (NO)
Inventor: COUCHOUD JEAN-JACQUES
IPC: C08L77/02
Filed: 1986-12-18
Abstract: 1. Thermoplastic alloys consisting essentially of 30 to 94.8 parts by weight of polyamide, of 0.2 to 65 parts by weight of polyetheramide and of 5 to 50 parts of a thermoplastic elastomer, the sum of these three constituents having to be equal to 100.
Patent NO-880177-L (NO)
Inventor: MADSEN FREDE
IPC: F16L41/08
Filed: 1988-01-18
Abstract: A pipe connecting piece for drainage pipes consists of a main part (1) and at least one branch part (2) connected thereto so that the pipe connecting piece is essentially T-shaped. The main part (1)is provided with an opening (3), disposed in the wall, which is bounded at the circumference by a part of the wall of the main part which is bent outwards in the form of a collar (4). The branch part (2) fits into said collar and is secured therein by means of a number of inwardly directed bulges (5) disposed in the circumferential wall of the collar (4) and the wall section of the branch part (2) fitted therein. The pipe connecting piece easy to manufacture without expensive tools and without use of glue joints.
Patent NO-882477-L (NO)
Inventor: CONFORTO PETER MICHAEL
IPC: B65B/
Filed: 1988-06-03
Abstract: A blank for forming a wrap-around carton is delivered to a moving support carriage which is moved to a station where the moving carriage receives a predetermined number of articles to be packaged. The carriage, with the articles resting on the bottom portion of the blank, is moved downstream while cams actuate tucker fingers which pivot up to fold the tuck flaps of the blank toward each other, causing the end and side panels to be elevated. Another cam actuates a pusher bar which pivots up to push the articles. The carton blank and the articles are thus positively moved through subsequent flap folding and gluing stations, avoiding the problems which can arise due to the use of separate means for moving the articles and the carton blank. A cam operated hinged plate is used to segregate the leading articles at the entry to the machine.
Patent NO-893208-L (NO)
Inventor: GRAVITT BILLY B
IPC: C04B/
Filed: 1989-08-09
Abstract: A hydraulic cement is formed from a Class C fly ash and an alkali metal activator. Mortar and concrete compositions can be prepared with this hydraulic cement. The cement is particularly useful in producing mortar and concrete compositions that achieve high strengths in a short time.
Patent NO-900907-L (NO)
Inventor: WATANABE NAOTAKA
IPC: D21H17/45
Filed: 1990-02-26
Abstract: Disclosed are a papermaking method of preparing a paper having a reinforced strength wherein a polymer latex is added to a paper stock in an amount of from 2.5 to 30 % by weight. The polymer latex is prepared by neutralizing a seed polymer with an acid or a salt or by quaternizing it with a quaternizing agent. The surfaces of the emulsion grains are highly densely cationated. The seed polymer is formed by adding a monomer as represented by the following formula (I) or a mixture of the monomer (I) and copolymerizable ethylenic unsaturated monomer(s) (II) to a seed latex of a carboxyl-modified synthetic rubber latex or synthetic resin emulsion and polymerizing them: <CHEM>  R1 represents H or CH3;  R2 represents an alkylene group having from 2 to 5 carbon atoms; R3 and R4 each represent H or an alkyl group having from 1 to 5 carbon atoms;  A represents   - @-O- or   -@-NH-; and R1, R3 and R4 and so selected that the monomer is hardly soluble or insoluble in water.   The paper has a noticeably improved paper-strength.
Patent NO-910956-L (NO)
Inventor: NEUWIRTH ROBERT
IPC: A61F7/12
Filed: 1991-03-11
Abstract: A method and apparatus for effecting necrosis of a tissue lining of a mammalian body cavity, particularly a uterine endometrium (27), by introducing an applicator comprising a distendable bladder (5) connected to a catheter into the uterus, distending the bladder (5) by introducing a non-toxic fluid under pressure, heating the fluid by means (44) located internal to the bladder (5) to a temperature of 190 DEG  to 215 DEG F and preferably 210 DEG F for a period of 4 to 12 minutes and preferably 6 minutes and regulating said apparatus by means (30) located external to the uterus, thereby cauterizing substantially the entirety of the tissue lining, particularly the endometrium (27). <IMAGE>
Patent NO-913811-L (NO)
Inventor: BERMES RUDOLF
IPC: C09B29/045
Filed: 1991-09-27
Abstract: Aqueous solutions containing, each percentage being based on the weight of the aqueous solution, a) from 5 to 20% by weight of the dye of the formula  <IMAGE>   (calculated as free acid) where cat(+) is a mixture of cations comprising from 5 to 50 mol % of lithium ions, from 5 to 40 mol % of diethanolammonium ions and from 20 to 90 mol % of triethanolammonium ions, and b) from 0 to 15% of urea, are useful for dyeing paper stock.
Patent NO-914610-L (NO)
Title: Girpumpe for et maalesystem for vaeske uttoemming
Inventor: ASLIN DAVID J
IPC: F04C2/08
Filed: 1991-11-25
Abstract: Det er beskrevet en girpujnpe (20) for bruk l et målesystem for væskeuttømming med et par karbongrafitt-' sliteplater (69, 70), for å øke pumpens vakuum eller sugehøyde egenskaper. Sllteplatene (69, 70) er plassert på motsatte sider av pumpens (20) sylindriske tannhjul (55, 56) og er fjærbelastet mot sidene til tannhjulene (55, 56) for å redusere den indre pumpeklaringen. FJærkraften frembringes av en elastisk o-ring (71a) plassert mellom en overflate til pumpehuset (50) og en av sitteplatene (69, 70). Tannhjulene (55, 56) er anordnet for begrenset bevegelse, slik at presset på en av sliteplatene (69, 70) .overføres via tannhjulene (55, 56) til den andre sitteplaten (70). Girpumpen (20) drives gjennom et reduksjonsglr (22) med en reversibel elektrisk motor (21). Anvendelse av girpumpen (20) sikrer en nøyaktig måling av væskemengden som tilføres fra systemet.
Patent NO-920401-L (NO)
Inventor: FLECHE GUY
IPC: C08K5/09
Filed: 1992-01-30
Abstract: Thermoformable composition characterised in that it contains at least one starchy compound and at least one salt of a hydroxycarboxylic acid.
Patent NO-924258-L (NO)
Inventor: ECKER DAVID J
IPC: C12N15/113
Filed: 1992-11-05
Abstract: Methods for modulating the expression of the HIV +E,uns tat+EE  gene are disclosed comprising contacting tat RNA with oligonucleotide or oligonucleotide analog which can bind with at least a portions of the RNA. In accordance with the preferred embodiments, oligonucleotides or oligonucleotide analogs are designed to bind to portions of the tat RNA which are of significance to the expression of the gene coding for said RNA. In accordance with a preferred embodiment, methods of treatment of human immunodeficiency virus are disclosed.
Patent NO-931396-L (NO)
Inventor: JACOBS III WILLIAM
IPC: C09D5/46
Filed: 1993-04-15
Abstract: Glycoluril based amino resin powder coating compositions have improved flow out and viscosity characteristics when a rheology improving additive selected from alkali metal oxides, alkali metal hydroxides, alkali metal carbonates, alkaline earth metal carbonates, alkaline earth metal oxides, alkaline earth metal hydroxides, aluminum oxides, aluminum hydroxides, aluminum carbonates, zinc salts of long chain fatty acids, aluminum salts of long chain fatty acids, monoamines, diamines, or mixtures thereof are added.