baber/WOPTO huggingface dataset:
Patent NO-179002-B (NO)
Inventor: LANG FLORIAN
IPC: C07C323/65
Filed: 1993-02-12
Abstract: Ortho-substituted benzoylguanidines of the formula I <IMAGE>  where: R(1) is equal to halogen, alkyl, -X-R(6), where X is equal to O, S, NR(7) or Y-ZO and R(6) is equal to H, (cyclo)(halo)alkyl(methyl), -CnH2n-phenyl, R(3) is equal to H, -X-R(6), R(2) and R(4) are equal to R(11)-SO1-2-, (di)-alkyl-N-SO2-, or one of the two radicals R(2) or R(4) is equal to hydrogen or is defined as R(1), R(5) is equal to H, methyl, F, Cl, methoxy,  and their pharmaceutically acceptable salts.  They are obtained by a process in which compounds of the formula II <IMAGE> in which R(1) to R(5) have the meaning mentioned and L represents a leaving group which can be easily substituted nucleophilically, are reacted with guanidine. The compounds I are used for producing a medicament for the treatment and the prophylaxis of heart-rhythm disorders and ischaemically induced damage, as well as for producing a medicament for the inhibition of cell proliferation.
Patent SE-330883-B (SE)
Inventor: HOCKS P
IPC: C07J75/00
Filed: 1967-01-27
Abstract: 1,172,273. Steroids. SCHERING A.G. 16 Jan., 1967 [29 Jan., 1966], No. 2136/67. Heading C2U. Novel compounds of the general formula in which R 1  represents a hydrogen atom, an alkyl group containing 1-4 carbon atoms or an acyl group of an organic carboxylic acid, R 2  represents a hydrogen atom or a hydroxyl group, Z represents a hydrogen atom or a methyl group, Y represents an alkyl or alkynyl group containing at least 3 carbon atoms which may be substituted or represents an ethynyl group, C 7 =C 8  represents a single or double carbon-carbon bond and #A represents the A- ring of a steroid nucleus and which may contain at least one additional substituent attached to the steroid nucleus that is inert towards a Grignard reagent of the formula YMgX in which X represents Cl, Br, or I, and in which the hydrogen atom in the 5-position, the methyl group in the 21-position and the OR 1 -substituent in the 22-position each has the α- or #- configuration, are obtained by treating the corresponding 6-keto-20-formyl compound of the pregnane series with a Grignard reagent of the formula YMgX, and in the resulting compound, if desired, selectively hydrogenating any unsaturated carbon-carbon bond present in the group represented by Y, and/or, if desired, saponifying any acyloxy group(s) and/or eliminating any ether group(s), or esterifying or etherifying any hydroxyl group(s) other than a 14α-hydroxyl group, and/or, if desired, when R 2  represents a hydrogen atom in the resulting compound, introducing by a known method a hydroxyl group in the 14α-position.
Patent SE-311761-B (SE)
Inventor: BRILANT J
IPC: E21B47/10
Filed: 1961-06-01
Abstract: 964,714. Testing ground permeability in situ. SOLETANCHE. May 9, 1961 [June 1, 1960], No. 16843/61. Heading G1S. Apparatus for testing the permeability of ground in situ comprises a bell 5 supported within a bore-hole by a ball 6 closing an aperture at the top of the bell when cable 4 is in tension, the cable passing over a graduated pulley 3 and carrying a counterweight p which balances the weight of the bell when the latter is totally immersed in water (all the air having escaped during immersion when the cable is slack), a further counterweight P being then attachable to cable 4 to raise the water-filled bell, on release of a holding stud 8, by a predetermined height. Water enters the borehole at a measured rate and the rising movement of the bell causes pulley 3 to rotate at a rate which is a function of the permeability of the ground at the base of the borehole.
Patent SE-313762-B (SE)
Inventor: GODET J
IPC: A24C5/354
Filed: 1965-06-08
Abstract: 1,114,719. Filling containers with cigarettes and other rod-shaped articles. SERVICE D'EXPLOITATION INDUSTRIELLE DES TABACS ET DES ALLUMETTES. 8 June, 1965 [9 June, 1964], No. 24086/65. Heading B8C. Cigars or similar shaped objects fed continuously by a conveyer 1 (Fig. 1) are batched by a hopper 4, 5, the input to which is cut off at fixed intervals while the hopper releases its contents to a plate 8 which is lowered within a compartment 6 of. a container. In the form described, the container is then moved by a conveyer (15) (Fig. 3, not shown) through the width of one compartment so that the operation may be repeated in the next compartment. A time-controlled photo-electric cell 7 controls the downward movement of the plate 8. The compartments in the conveyer 1 may each receive more than one article. The feed to the hopper may be closed by sliding a pair of rods 3 (Fig. 1, and Fig. 2, not shown) over the top of the hopper. The rods 3 may be propelled by lugs on the conveyer 1, and may be subsequently retracted by springs; alternatively, the rods may be driven from a cam. The articles are released from the hopper by pivoting flaps 5. The compartments in the containers may be formed by partitions (14) (Fig. 3) mounted on a removable front cover (13). The bottom of each compartment is formed by spaced rails (16), (17) (Fig. 2) which rest on guides 20.
Patent YU-46108-B (YU)
Inventor: STRAESSLE M
IPC: F16B7/18
Filed: 1988-05-24
Abstract: A connecting element for a scaffolding framework rod has a bolt 141 rotatably mounted on one end of the rod, and a guide sleeve 151 with an axial through-bore into which a section of the bolt extends. The bolt is connected to a screw insert 161 guided by a pin 171 which rides in a slot 152 of the sleeve, and a spring 172 urges the guide sleeve against a sleeve insert 130, 121 mounted on the end of the rod.
Patent ZA-845434-B (ZA)
Title: Complexable heterogeneous oligosaccharides and alpha-hydosanes having therapeutical activity,process for their preparation and related pharmaceutical compositions
Inventor: BALDACCI MASSIMO
IPC: C08B37/00
Filed: 1984-07-13
Abstract: Complexable heterogeneous oligosaccharides and pure alpha-hydosanes, namely not contaminated from other macromolecules (mucopolysaccharides, proteins, nucleic acids, etc.) of a defined molecular weight, are produced starting from a mixture of mucopolysaccharides obtained starting from bovine or swine mucosa through a process comprising a precipitation with organic solvents, a further purification by means of specific enzymes and chromatographic separation by gel filtration. Heterogeneous oligosaccharides are obtained which can be complexed with metals, being thus able to promote the pharmacological effect of the metal thanks to the greater permeability towards the complexes of the membrane of the cells of the absorbing mucosa and of the cells of the target tissue. There are also obtained pure alpha-hydosanes having a well defined molecular weight range capable of providing several pharmacological activities, more particularly an activating effect of the anti-thrombine III, a potentiating effect of the tissutal activator and a fibrine depolymerizing effect have been found for some of them, whereas for some others an effect on the factor Xa/PTT ratio has been revealed and lastly for still others a lipasemic and anti-coagulating activity has been found.
Patent ZA-846083-B (ZA)
Title: Industrial-scale process for the production of polyols by fermentation of sugars
Inventor: TROOSTENBERGH JEAN-CLAUDE DE
IPC: C12R1/645
Filed: 1984-08-06
Abstract: An industrial process for producing polyols comprises subjecting sugars to aerobic fermentation using Moniliella tomentosa var pollinis in a fermentation medium containing a water-soluble or water-dispersible polymer which is capable of retaining the cells in the fermentation medium. The process is especially suitable for the industrial production of erythritol and/or ribitol. The process overcomes the disadvantage shared by prior proposals wherein cells are lost from the fermentation media through being carried away by the foam produced during fermentation.
Patent ZA-914578-B (ZA)
Title: Device for mounting and dismounting shaft-furnace tymps
Inventor: BONANI NICOLAS
IPC: C21B7/16
Filed: 1991-06-14
Abstract: The installation comprises a gripper (44) with retractable claws (40) which are engageable through the tuyere (26) and manoeuvring means which run through the gripper and are manoeuvrable from the outside for deploying or retracting the claws (40) radially in relation to the axis of the tuyere (26). The gripper (44) and its manoeuvring means are supported by a yoke (30) designed to be adapted to the external edge of the vault (24) and to be associated with a conventional pneumatic bolt-firing tool which is capable of being adapted to the outside of the yoke (30) either on extensions of the claws (40) or on the manoeuvring means in order to exert via its rotation and its support on the yoke (30) a traction force on the claws of the gripper. 
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Patent ZA-924753-B (ZA)
Title: Ampholyte terpolymers providing superior conditioning properties in shampoos and other hair care products
Inventor: CHEN SHIH-RUEY THOMAS
IPC: C08F299/02
Filed: 1992-06-26
Abstract: Ampholyte terpolymer conditioning additives for hair care products are disclosed which improve wet and dry hair combability, especially detangling and reduced static flyaway, sheen, and fixative properties, especially curl retention. The ampholyte terpolymers may have a weight average molecular weight of from about 10 thousand to 10 million, and comprise (a) from at least 1 to as much as 95 weight percent of the nonionic monomer acrylamide (AM), (b) from at least 5 to as much as 80 weight percent of the cationic monomer dimethyldiallylammonium chloride (DMDAAC), and (c) from at least 1 to as much as 75 weight percent of the anionic monomer 2-acrylamido-2-methylpropane sulfonic acid (AMPSA), with optionally up to 50% of said anionic monomer AMPSA being replaced with the anionic monomer acrylic acid (AA). The ampholyte terpolymers are added to hair care product formulations in amounts ranging from 0.1-10% by weight. They are particularly compatible with anionic surfactant shampoos, providing clear formulations without the loss of conditioning properties described above.
Patent ZA-946507-B (ZA)
Title: Ortho-substituted benzoylguanidines process for their preparation their use as pharmaceutical of diagnostic and pharmaceutical containing them
Inventor: WEICHERT ANDREAS
IPC: C07C237/34
Filed: 1994-08-26
Abstract: There are described ortho-substituted benzoylguanidines of the formula I <IMAGE>  in which:   R(1) is H, Hal, CN, NO2, (cyclo)alkyl, (O)(S)[NR(5)](CH2)b-(CF2)c-CF3,   R(5) is H, (C1-C4)-alkyl, -CdH2dR(6),   R(6) is cycloalkyl, (bi)phenyl(yl), naphthyl,  or   R(1) is -SR(10), -OR(10), -CR(10)R(11)R(12),   R(10) is -CfH2f-(C3-C8)-cycloalkyl, -(C1-C9)-heteroaryl or phenyl, R(11) and R(12) are defined as R(10) or are hydrogen, (C1-C4)-alkyl,  or   R(1) is naphthyl, (bi)phenyl(yl), (C1-C9)-heteroaryl,  or R(1) is -SR(13), -OR(13), -NHR(13), -NR(13)R(14), -CHR(13)R(15), -C[R(15)R(16)]OH, -C IDENTICAL CR(18), -C[R(19)]=CR(18), -[CR(20)R(21)]k-(CO)-[CR(22)R(23)R(24)]l,   R(13) and R(14) are -(CH2)g-(CHOH)h-(CH2)l-(CHOH)j-R(17),   R(17) is hydrogen, methyl, -(CH2)g-O-(CH2-CH2O)h-R(24), R(15) and R(16) are hydrogen, alkyl or, together with the carbon atom carrying them, cycloalkyl,   R(18) is phenyl, heteroaryl, (cyclo)alkyl,   R(19), R(20), R(21), R(22) and R(23) are hydrogen, methyl,   R(24) is H, (cyclo)alkyl, -CmH2m-R(18),   R(2) and R(3) are defined as R(1),   R(4) is alkyl, Hal, CN, -(CH2)n-(CF2)o-CF3,  and their pharmaceutically tolerable salts. Compounds I have no unwanted salidiuretic properties, but very good antiarrhythmic properties. They are outstandingly suitable as antiarrhythmic medicaments having a cardioprotective component for infarct prophylaxis and infarct treatment and for the treatment of angina pectoris, where they also preventively inhibit or greatly decrease the pathophysiological processes in the formation of ischaemically induced damage. Because of their protective actions against pathological hypoxic and ischaemic situations, the compounds of the formula I according to the invention, as a result of inhibition of the cellular Na<+>/H<+> exchange mechanism, can be used as medicaments for the treatment of all acute or chronic damage caused by ischaemia or illnesses primarily or secondarily induced thereby.
Patent ZA-953629-B (ZA)
Title: Soluble polypeptidic fragments of lag-3 protein method of production thereof therapeutic composition anti-idiotype antibodies
Inventor: FAURE FLORENCE
IPC: C07K16/42
Filed: 1995-05-05
Abstract: Soluble polypeptide fraction consisting of all or part of one at least one of the four immunoglobulin-type extracellular LAG-3 protein domains (amino acids 1-159, 160-230, 240-330 and 331-412 of the SEQ ID NO:1 sequence) or consisting of one peptide sequence derived from these domains by replacement, addition or deletion of one or more amino acids. The fraction of the invention has a specificity at least equal to that of LAG-3 in relation to its ligand.
Patent CH-617310-B (CH)
Inventor: WILD DANIEL
IPC: G04B37/08
Filed: 1977-09-07
Abstract: The tube (5) through which passes the control rod (6) enters notches made in the middle (1) and in the rim (2a) of the back (2), which notches are chamfered at (9) and at (8), respectively. An O-ring seal (10) is housed in an annular space accommodated between the chamfered parts (8 and 9) and a shoulder (5a) of the tube (5), the face of which facing the seal (10) is frustoconical at (11). <IMAGE>
Patent GB-2359621-B (GB)
Title: Photoelectric smoke detector, and smoke detection section assembly
Inventor: YAMANO NAOTO
IPC: H05K1/02
Filed: 2000-10-31
Granted: 2004-04-21
Abstract: A photoelectric smoke detector includes a smoke detecting section defining a smoke detecting space, a light emission section holder having a light-emission element disposed in the smoke detecting section, and a light receiving section holder having a light-receiving element disposed in the smoke detecting section. The light-receiving element receives light which has been emitted from the light-emission element and is scattered by smoke flowing in the smoke detecting space. A hybrid circuit board has an integrated circuit mounted thereon and is housed in the light receiving section holder. The integrated circuit including the light-receiving element and at least a received-light signal amplifying circuit. The hybrid circuit board is arranged so that the light-receiving surface of the light-receiving element is directed toward the smoke detecting space.
Patent GB-2385523-B (GB)
Title: Descent apparatus
Inventor: BYRNE RONAN ANTHONY
IPC: A62B1/10
Filed: 2002-02-25
Granted: 2004-01-07
Abstract: A portable descent apparatus ( 1 ) for use in effecting the controlled descent of a body from an elevated location, for example a multi-storey building, comprises in combination a support frame ( 2 ) having a substantially planar base ( 3 ) and upright supporting end brackets ( 4,5 ), a fixed shaft ( 6 ) extending between said end brackets, a rotatable drum ( 7 ) coaxially mounted on said shaft and having means for attachment of one end of a flexible cable ( 17 ) thereto, the drum ( 7 ) having fixed to one end thereof a manually or remotely controllable calliper-operated disc brake assembly and to the other end thereof a gear driven descent speed controller comprising a toothed annular member ( 13 ) meshing with a pinion ( 19 ) driving a centrifugal brake assembly ( 12 ), the flexible cable ( 17 ) having one end attached to said drum and the other end ( 16 ) thereof having anchoring means for attaching the cable to a fixed position ( 18 ), and a first handle means ( 15 ) attached to the support frame ( 2 ) adjacent to said disc brake assembly and provided with means ( 11 ) for manually or remotely controlling the braking effect of the disc brake assembly, and a second handle means ( 14 ) attached to the support frame ( 2 ) adjacent to said descent speed controller, the arrangement being such that in use the apparatus may be held using the two handle means ( 14,15 ) with the planar base ( 3 ) positioned against the descending body.
Patent GB-2400271-B (GB)
Title: Dynamic resource allocation in packet data transfer
Inventor: COOPER DAVID EDWARD
IPC: H04W24/10
Filed: 2003-04-02
Granted: 2005-03-02
Abstract: A method for control of packet data transmissions in a TDMA wireless network to provide for additional choices in the allocation of communication channels. Measurement and recovery periods are re-assigned to avoid conflicts in operating conditions. The re-assignments for the GPRS system may be reduced to a simple formula. <IMAGE>
Patent GB-2402198-B (GB)
Title: Resilient damping friction wedge
Inventor: HEWITT PAUL
IPC: B61F5/34
Filed: 2004-05-26
Granted: 2005-10-19
Abstract: A friction damping arrangement for a railway vehicle comprises first and second relatively moveable vehicle components (14,16), a friction wedge (18) having a surface (37) arranged to co-operate with a surface of the second vehicle component (16), and resiliently urged towards the first vehicle component (14), and a resiliently deformable component (48), located between the first vehicle component (14) and the friction wedge (18), the resiliently deformable component (48) being deformable to allow relative movement between the first vehicle component (14) and the friction wedge (18).
Patent GB-2460304-B (GB)
Title: Secure storage device
Inventor: SHAW NORMAN
IPC: G06F21/78
Filed: 2008-10-17
Granted: 2013-02-20
Abstract: A communication and security device for a portable computer is disclosed including a housing, a connector provided on the housing for physical connection to the portable computer, a computer interface coupled to the connector for communicating data with the portable computer, a wireless modem coupled to the computer interface for communicating data between the portable computer and a remote device via a wireless network, a regulator operable to regulate power in the communication and storage device, and a processor coupled to control the regulator, the processor coupled to the wireless modem and arranged to process at least one security command received by the wireless modem to control the regulator in response to the received command.
Patent GB-2457847-B (GB)
Title: A resource allocation method and a method for transmitting/receiving resource allocation information in mobile communication system
Inventor: LEE DAE WON
IPC: H04W72/04
Filed: 2008-03-19
Granted: 2011-08-10
Abstract: A resource allocation method and a method for transmitting resource allocation information in a mobile communication system are disclosed. That is, a LVRB (PRBs) and a DVRB which are the units of a scheduling resource are defined and a resource allocation method and a method for transmitting resource allocation information using the same are disclosed. In the LVRB, a part -bitmap scheduling method using a LVRB set is suggested and a method for constructing resource allocation information using the same is suggested. In the DVRB, a method for defining the DVRB using PRBs in a subframe is suggested and a method for constructing resource allocation information using the same when scheduling is performed using the DVRB constructed by the defined method is suggested.; In order to prevent interference and collision from occurring due to the complete matching of the DVRBs in respective cells, a method using different DVRBs in the respective cells is suggested.
Patent GB-2002631-B (GB)
Title: Phospholipid compositions
IPC: A61K35/12
Filed: 1978-07-18
Granted: 1982-03-10
Abstract: Phospholipid compositions are obtained from ground. homogenised animal organs by a four stage process. in the first stage the organs are soaked in acetone to sever bonds between phospholipids and other substances present in the organ. In the second stage, the organs are refluxed in acetone to remove extraneous matter such as proteins and amino acids. In the third stage, the phospholipids are extracted with ethanol. The acetone solutions, which may contain small amounts of entrained phospholipids, and the ethanol solution are all evaporated to dryness and the residues are taken up in diethyl ether. In the fourth stage the phospholipids are precipitated by addition of acetone. The phospholipid compositions obtained are of sufficient purity for pharmaceutical use.
Patent GB-2119957-B (GB)
Title: Annealed polyvinyl alcohol contact lens
Inventor: LEE PING I
IPC: B29D11/00
Filed: 1983-04-26
Granted: 1985-10-09
Abstract: Optically clear soft contact lenses of aqueous swollen solid polyvinyl alcohol having a weight average molecular weight of at least 6,000, having been annealed under crystallinity promoting conditions to a crystallinity degree of 0.195 to 0.7 to effectively increase the elastic modulus of the swollen lenses, and optionally subsequently crosslinked, and methods of preparation and the use thereof are disclosed. The lenses are characterized by their relatively high oxygen transmissibility, sufficient to meet the needs of the human cornea, high optical clarity, improved hot water resistance and superior mechanical properties. The lens may be tinted with dyes and pigments.
Patent GB-2188227-B (GB)
Title: Disposable diaper having an improved side closure
Inventor: TOUSSANT JOHN WILLIAM
IPC: A61F13/15
Filed: 1987-03-20
Granted: 1989-11-15
Abstract: A disposable diaper having an improved side closure is disclosed. The disposable diaper is provided with an outer fastening means (54) and an inner fastening means (60). The outer fastening means (54) maintains the waist portions of the diaper in an overlapping configuration while the inner fastening means reduces shifting of the overlapping portions.
Patent GB-2245494-B (GB)
Title: Herbicidal agents based on a combination of metamitron/ethofumesate/phenmedipham/desmedipham
Inventor: WIESCHOLLEK RAPHAEL
IPC: A01N25/14
Filed: 1991-07-02
Granted: 1994-05-25
Abstract: The invention relates to novel ready-for-use formulations of the known herbicidal active substances metamitron (I) + ethofumesate (II) +  (A) phenmedipham (III) or  (B) phenmedipham (III) and desmedipham (IV) or  (C) desmidipham (IV), preferably solid formulations such as water-dispersible powders (WP) or water-dispersible granules (WG), the ratio by weight of the active substances (I):(II):(III) or (IV) being (1):(0.05 to 1):(0.05 to 1), that of the active substances (I):(II):(III):(IV) being (1):(0.05 to 1):(0.05 to 1):(0.05 to 1), and the total active substance content in each case being between 20 and 75% by weight, and to their use as herbicides, in particular as selective herbicides in beet.
Patent GB-2274826-B (GB)
Title: An apparatus for escalading
Inventor: JEPHCOTT DAVID LYNTON
IPC: E06C7/16
Filed: 1993-02-05
Granted: 1997-03-26
Abstract: The disclosure relates to an apparatus for escalading, comprising:       at least a first, generally upwardly extending frame member; an operator support means (18) secured to the first frame member and moveable in a generally vertical direction; a load support means (22) secured to the first or a frame member and moveable in a vertical and horizontal directions; a bracing member (14a,14b) .secured to the frame member and extending outwardly therefrom; and floor- or ground-engaging means (24) secured to the first or a frame member and the bracing member respectively, the arrangement being such that, when the apparatus stands with the floor- or ground-engaging means on a level surface, the mass of the apparatus and any loads supported thereon acts within a plane interconnecting the floor- or ground-engaging means regardless of the positions of the operator support means and the load support means, characterised in that the apparatus includes three generally upwardly extending, generally parallel frame members (11a,11b,11e) interconnected by respective further frame members (12a,12b) and defining two or more generally upwardly extending, parallel planes, the operator support means (18) being constrained to move generally vertically in one of the planes and the load support means (22) being constrained to move selectively generally vertically and horizontally in the other plane.