baber/WOPTO huggingface dataset:
Patent PH-22336-A (PH)
Title: A reactive derivative of 2,3-dioxapiperazine derivative
Inventor: SAIKAWA ISAMU
IPC: C07D499/46
Filed: 1976-11-15
Abstract: 1508064 N-Piperazinocarbonyl-amino acid derivatives TOYAMA CHEMICAL CO Ltd 28 April 1975 [13 Aug 1974 28 Oct 1974 17 Feb 1975] 15360/77 Divided out of 1508062 Heading C2C Novel compounds I and salts and carboxyl derivatives thereof (R is an amino acid residue; R<SP>2</SP> and R<SP>3</SP> are H or alkyl and R<SP>2</SP> and R<SP>3</SP> are both linked to the same carbon atom; and A is H or an optionally substituted alkyl, alkenyl, aryl or aralkyl group) are prepared by reaction of a compound II NH 2 RCOOR<SP>1</SP> (III) (R<SP>1</SP> is H or a cation) with a reactive derivative of a compound IV
Patent PH-21295-A (PH)
Title: Octahydroindolizine compounds useful as analgesics
Inventor: JOEL CARMOSIN RICHARD
IPC: A61K31/495
Filed: 1986-01-08
Abstract: Octahydroindolizidines of the formula (I):where A is a 3-7 carbon or hetero-containing ring, R' is a substituent and x is 0-3. Also, pharmaceutical composition for treating pain and methods for synthesis and use as well as novel intermediates in the synthesis.
Patent PH-27420-A (PH)
Title: Pharmaceutically active combination composition comprising as components a as plasminogen activator and as component b herein
Inventor: HEIM JUTTA
IPC: A61K38/00
Filed: 1989-09-19
Abstract: There is provided a pharmaceutical composition comprising as component A a plasminogen activator and as component B hirudin together with a pharmaceutically acceptable carrier. The pharmaceutical composition can be used for the prophylaxis and therapy of thrombosis or diseases caused by thrombosis.
Patent TR-24115-A (TR)
IPC: C07D273/04
Filed: 1988-12-02
Abstract: Compounds of the general formula I   <IMAGE> (I)  in which A denotes a radical of the formula A1, A2 or A3    <IMAGE> (A1)  <IMAGE> (A2) <IMAGE> (A3)  R1 to R3 in each case independently of one another denote hydrogen or halogen, the radicals R4 in each case independently of one another denote halogen, (C1-C3)halogenoalkyl or nitro, R5 denotes (C1-C5)alkyl, which can be halogenated, X denotes oxygen or sulfur, n denotes a number from 0 to 2 and m denotes a number from 1 to 4 with the proviso that (R4)m does not by itself denote halogen or by itself denote nitro, and where A=A1, salts thereof which can be used in agriculture, have advantageous acaricidal and insecticidal properties. Processes for the preparation of the compounds of the formula I are furthermore described.
Patent UY-31971-A (UY)
Title: Derivados de piridino-piridinonas, su preparación y su aplicación en terapéutica
Inventor: MCCORT GARY
IPC: A61P35/00
Filed: 2009-07-08
Abstract: La invención se refiere a los derivados de piridino-piridinonas, de fórmula general (I): en la que R1, R2, R3, R4, R5, R6, R7, V, W, Y, Z, m son tales como se han definido en la descripción.  Procedimiento de preparación y aplicación en terapéutica.
Patent UY-32160-A (UY)
Title: Particulas inhalables que comprenden tiotropio
Inventor: KARIM AMIGHI
IPC: A61K31/445
Filed: 2009-10-02
Abstract: La presente invención se refiere a partículas inhalables que comprenden una forma amorfa de tiotropio estabilizada con un agente estabilizante. Se refiere a las particulas inhalables que comprenden una forma amorfa de tiotropio estabilizada con un agente estabilizante mezclado con uno o más exipientes gruesos de un tamaño medio de partícula de 15 250 um. También se refiere a una composición farmacéutica que comprende las partículas inhalables de la invención, a su procedimiento para su preparación y a su uso para la preparación de un medicamento para el tratamiento del asma o de la enfermedad pulmonar obstruciva crónica (EPOC).
Patent UY-35252-A (UY)
Title: MÉTODOS PARA INTRODUCIR dsRNA EN SEMILLAS DE PLANTAS PARA MODULAR LA EXPRESIÓN GENÉTICA
Inventor: AVNIEL AMIR
IPC: A01H5/00
Filed: 2013-12-30
Abstract: Se da a conocer un método para introducir en una semilla una molécula disparadora de polinucleótido exógeno no transcribible, por ejemplo dsRNA.  El método comprende poner en contacto la semilla con la molécula disparadora de polinucleótido exógeno no transcribible, por ejemplo dsRNA, bajo condiciones que permiten la penetración en la semilla de la molécula disparadora de polinucleótido exógeno no transcribible, por ejemplo dsRNA, de esa manera, introduciendo la molécula disparadora de polinucleótido exógeno no transcribible, por ejemplo dsRNA, en la semilla.
Patent UY-35693-A (UY)
Title: Pirazolo[1,5-a]piridin-3-carboxamidas sustituidas y su uso
Inventor: TOBIAS MARQUARDT DR
IPC: C07D491/048
Filed: 2014-08-05
Abstract: La presente solicitud se refiere a novedosas pirazolo[1,5-a]piridin-3-carboxamidas, a procedimientos para su preparación, a su uso solas o en combinación para el tratamiento y/o la profilaxis de enfermedades, y a su uso para producir medicamentos pa ra el tratamiento y/o la profilaxis de enfermedades, especialmente para el tratamiento y/o la profilaxis de trastornos cardiovasculares.
Patent UY-37339-A (UY)
Title: Formas de sal de 4-ciano-n-(2-(4,4-dimetilciclohex-1-en-1-il)-6-(2,2,6,6-tetrametiltetrahidro-2h-piran-4-il)piridin-3-il)-1himidazol-2-carboxamida y composiciones que las contienen
Inventor: NAGY E FAWZY
IPC: C07D405/14
Filed: 2017-07-19
Abstract: La presente descripción trata formas de sal de 4-ciano-N-[2-(4,4-dimetilciclohex-1-en-1-il)-6-(2,2,6,6-tetrametiltetrahidro-2H-piran-4-il)piridin-3-il]-1H-imidazol-2-carboxamida.
Patent UY-37366-A (UY)
Title: Inhibidores de diacilglicerol aciltransferasa 2
Inventor: LEE ESTHER CHENG YIN
IPC: C07D409/14
Filed: 2017-08-17
Abstract: En la presente se d escriben compuestos de Fórmula I que inhiben la actividad de la diacilglicerol aciltransferasa 2 (DGAT2) y sus u so s en e l tratamiento de enfermedades enlazadas a los mismos en animales
Patent UY-38164-A (UY)
Title: Composiciones agroquímicas sólidas
Inventor: SHROFF JAIDEV RAJNIKANT
IPC: C07C69/712
Filed: 2019-03-28
Abstract: La presente invención se relaciona con composiciones herbicidas sólidas. Particularmente, la presente invención se relaciona con composiciones herbicidas sólidas que comprenden uno o más herbicidas electrolíticos, uno o más de otros herbicidas y una base para controlar las malas hierbas.
Patent YU-42690-A (YU)
Title: Podrivac
Inventor: BUDIMIR BATURAN
Filed: 1990-03-05
Abstract: PODRIVAČ, pronalazak se odnosi na troredni podrivač koji se sastoji od grede (1) kvadratnog preseka na kojoj su obezbedjene tri tačke za trozglobu vezu sa traktorom. Na gredu (1) su vijcima (9) namontirane konzole na medjusobnom razmaku koji se može regulisati u granicama od 300 - 1000 mm. U konzolu nož (3) vezan preko dve osovinice (11) od kojih donja služi kao sigurnosna. Na prednjem delu nosača (3) oslanja se sečivo (6) koje je izradjeno od materijala otpornog na habanje i zamenljivo je. Na donjem kraju noža (3) montirana je sa 4 vijka peta (7), a na kojoj je pod odgovarajućim uglom postavljena podrivna ploča (5), dok je na zadnjem kraju pete kuće krtičar (8). Kod jednorednog podrivača konstrukcija se sastoji iz grede (1) sa trozglobom vezom, sa kojom je vezana u okretnim tačkama konzola (2), na koju je vijcima montiran nož (3), stopa (4), podrivna ploča (5), sečivo (6), peta (7) i krtičar (8). Gornji deo grede (1) i konzola (2) spojeni su hidro-cilindrom (), okretnim zglobom (osovinica) tako da se hidro-cilindrom može menjati geometrija u toku rada.
Patent YU-57294-A (YU)
Title: Intermedijeri u sintezi doramektina i postupak za njihovu sintezu
Inventor: CRAWFORD T C
IPC: A61K31/7042
Filed: 1994-10-04
Abstract: Opisani su intermedijeri i postupak za dobijanje doramektina, jedinjenja formule (I), polusintetički iz sporednog proizvoda u fermentacionom postupku koji takođe daje jedinjenje formule (I). Intermedijeri dobijeni postupkom prema ovom pronalasku su takođe korisni kao antiparazitska sredstva. Postupak prema ovom pronalasku koristi kontinualno ubrizgavanje reakciono inertnog gasa koji se ubrizgava tokom faze pirolize, što dovodi do značajnog poboljšanja celokupnog prinosa ovog prevođenja.
Patent YU-75583-A (YU)
Title: Device for the manufacture of fibres from a thermoplastic material
Inventor: BATTIGELLI J
IPC: D01D13/00
Filed: 1983-03-31
Abstract: 1. Apparatus for producing fibres from a thermoplastics material and comprising a centrifuge (10) revolving about a substantially vertical axis (22), means for driving the said centrifuge with a rotary motion, means of conveying a stream (24) of material molten to the drawable condition into the centrifuge and carrying it onto the inner surface of the peripheral wall of the said centrifuge, a large number of orifices (40) in the peripheral wall through which the molten material passes to form filaments (41), end means of drawing the said filaments (41) into fibres, said means comprising an internal combustion burner delivering an annular gaseous jet adjacent to the outer part of the said peripheral wall which is directed downwardly, the said annular gaseous jet being at an elevated temperature contributing to maintaining the filaments of material under drawable conditions for a period of time sufficient for drawing, characterised in that the diameter of the centrifuge is between 550 and 1500 mm and in that the centrifuge is driven with a rotary movement under conditions in which its periphery is subject to a centrifugal acceleration comprised between 4000 and 20,000 m/s2.
Patent YU-83790-A (YU)
Title: Naprava za porazdeljevanje prašnate trdne snovi v plinski suspenziji na napredujočo podlago
Inventor: VINCENT SAUVINET
Filed: 1990-04-26
Abstract: Izum se nanaša na napravo za porazdeljevanje prašnatega produkta na podlago. Naprava ima dve steni (4), ki razmejujeta kot rezilo zasnovano votlino (5), katera konvergira proti podlagi, komoro (10) za vbrizgavanje plina, zaprto s ploščo (11), ki je predrta z množico izlivov (12) za vbrizgavanje plina pod tlakom, kateri inducira okoliški zrak v votlino (5) v bistvu vzporedno s steno (4) votline (5), ki je letem sosednja, in ki homogenizira zmes prašnatega produkta in plina ter jo pospešuje v smeri podlage, s čemer tvori na njej zvezno tanko plast.
Patent YU-85981-A (YU)
Title: Process for producing polypptides similar to human fibroblast interferon
Inventor: FIERS W C
IPC: C12R1/645
Filed: 1981-04-01
Abstract: A DNA sequence consisting of the DNA inserts of G-pBR322(Pst)/HFIF1, G-pBR322(Pst)/HFIF3, G-pBR322 (Pst)/HFIF-6, G-pBR322(Pst)/HFIF7, DNA sequences which hybridize to any of the foregoing DNA inserts and DNA sequences, from whatever source obtained, including natural, synthetic or semi-synthetic sources, related by mutation, including single or multiple, base substitutions, deletions, insertions and inversions to any of the foregoing DNA sequences or inserts.
Patent BE-898627-A (BE)
Title: Gouttiere ou encadrement d'etancheite extrude pour carrosseries d'automobiles et tete d'extrusion pour sa realisation
IPC: B29C48/30
Filed: 1984-01-06
Abstract: Encadrement d'étanchéité (1) destiné à etre applique sur le bord (6) d'une ouverture ou d'un élément de fermeture de la carrosserie (5) d'un véhicule à moteur. Il comprend une section d'ancrage (2) en matière élastomère et une section d'étanchéité tubulaire (4) également en matière élastomère coextrudée avec la section d'ancrage (2). Dans les parties destinées à etre appliquées aux parties en forme de coin du bord (6) ou aux parties du bord (6) proches d'obstacles, la section (4) est incurvée par rapport à la section d'ancrage (2) et y est raccordée le long d'une ligne courbe (L).
Patent BE-905156-A (BE)
Title: Fermeture tubulaire perdue pour trous de forage.
Inventor: OTTO-ERNST GLAESMANN
IPC: E21B33/127
Filed: 1986-07-23
Abstract: Dispositif tubulaire perdu pour la fermeture de trous de forages destiné à l'injection de fluides appropriés comme par exemple pour l'injection de résine synthétique, principalement pour renforcer les terrains, ce dispositif étant principalement constitué d'un tube de remplissage (1) équipé à son extrémité d'une soupape anti-retour (5) formant sécurité anti-retour, ainsi que d'un élément flexible (2) en matériau élastique entourant le tube de remplissage. Ce dispositif est caractérisé en ce que l'ouverture (9) à l'interieur du tube de remplissage (1) est prévue avec une soupape suplémentaire (31).
Patent BE-906103-A (BE)
Title: Procede perfectionne pour preparer du dichloro-1,2 ethane par chloration de gaz contenant de l'ethylene.
IPC: B01J23/75
Filed: 1986-12-30
Abstract: Il est possible de diminuer beaucoup la formation de produits de chloration oxygénés de l'éthylène dans l'oxychloration de l'éthylène en deux étapes si,dans la seconde étape, on fait passer les gaz usés provenant de la réaction de la première étape, après leur avoir ajouté du chlore sous une pression de 1 à 7 bar et à une température de 100 à 300 degrés C, à des débits spatiaux de 100 à 50000 h-1, sur des catalyseurs constitués de supports sur lesquels ont été déposés des chlorures et/ou des oxydes de manganèse, de nickel et/ou de cobalt.
Patent CA-1079895-A (CA)
Inventor: BORMAN WILLEM F H
IPC: C08G63/00
Filed: 1974-02-05
Granted: 1980-06-17
Abstract: ABSTRACT OF THE DISCLOSURE             Poly(alkylene terephthalates) are prepared by an improved process which provides high molecular weight, in a shortened reaction time, without excessive loss of the diol reactant to side reactions.  In the process an excess of the diol reactant is heated with a mixture of the corresponding dialkyl terephthalates and from 5 to 95 mole % of terephthalic acid, based on the mixture.
Patent CA-1043267-A (CA)
Inventor: SPARK IAN J
IPC: F02B75/02
Filed: 1974-07-02
Granted: 1978-11-28
Abstract: ABSTRACT OF THE DISCLOSURE           An everted orbital displacer is formed having a plurality of working cavities defined by an internal peripheral surface of an orbiting piston, an external peripheral wall of a stationary internal housing located within the orbiting piston, opposed stationary end plates, and vanes sliding in slots in the internal housing and substantially radial grooves in the end plates.  If the piston is double sided, a normal orbital displacer may be formed with its working cavities located on the outer periphery of the piston and the combination of the two displacers used as a two stage compressor, pump or motor or as the basis of a two stroke or four stroke internal combustion engine, the advantages of an orbital displacer of compactness, efficiency and balance being further enhanced by the combination unit.
Patent CA-1044577-A (CA)
Inventor: STEIN KARL-ULRICH
IPC: H01L21/314
Filed: 1974-08-30
Granted: 1978-12-19
Abstract: Abstract Process for compensating for the presence of boundary charges in semiconductor layers which are grown on a monocrystalline insulating substrate including the stop of introducing doping atoms into the region of the boundary charges.  The doping atoms can be introduced before any semiconductor has been deposit?? after a thin layer of the semiconductor has been epitaxially grown on the substrate, or after all of the epitaxial layer has been grown.
Patent CA-1063523-A (CA)
Inventor: ERIKSSON ERIK S
IPC: B01D33/00
Filed: 1974-12-16
Granted: 1979-10-02
Abstract: ABSTRACT OF THE DISCLOSURE           Apparatus for separating liquid from a fibrous suspension comprises a hollow container having an inlet and an outlet.  A hollow filter element enclosing a filtrate-receiving space is rotatably mounted in the container such that an annular suspension-receiving space is defined between the walls of the filter element and the container.  A discharge mechanism permits liquid filtrate to be discharged from the filtrate-receiving space at a rate sufficient to reduce the pressure in the space relative to the pressure in the suspension-receiving space so that liquid in the fibrous suspension flows through the filter element into the filtrate-receiving space, leaving a concentrated fibrous suspension in the annular space surrounding the filter element.  The annular suspension-receiving space communicates with the inlet and the outlet of the con-tainer and has a radial width that diminishes from a point adja-cent the inlet circumferentially about the container toward the outlet.  The radial width of the suspension receiving space abruptly increases adjacent the outlet of the container so that the pressure in the portion of the suspension-receiving space adjacent the outlet is reduced relative to the pressure in the filtrate-receiving space.  The pressure differential causes a back flow of filtrate through the filter element to wash fibers from the surface of the element and facilitate the discharge of the concentrated suspension from the container.
Patent CA-1043243-A (CA)
Inventor: ICHIZAWA YOSHIYUKI
IPC: B29C65/78
Filed: 1975-06-02
Granted: 1978-11-28
Abstract: ABSTRACT OF THE DISCLOSURE An automatic shaping machine for continuously shaping a plastic film constructed of at least one layer into sleeves, having pinch rollers feeding the film continuously along a definite direction, a semitubing means and a tubing means provided along the film feed line to shape the film into tubular configuration around a longitudinal axis, and a cutter means provided ahead of said pinch rollers to cut the tube at a fixed length.
Patent CA-1058610-A (CA)
Inventor: PHILLIPPS GORDON H
IPC: C07J5/00
Filed: 1975-07-30
Granted: 1979-07-17
Abstract: ABSTRACT OF THE DISCLOSURE          The specification describes compounds of the general formula:-                  (I) [wherein X represents a .beta.-hydroxy or keto group, Y represents a fluorine or chlorine atom, R1 represents a hydrogen atom or an alkyl group containing 1 - 3 carbon atoms, R2 represents a group of formula -(CH2)nNR3R4 (wherein n is 1, 2 or 3 and R3 and R4, which may be the same or different, each represents an alkyl group containing 1 - 4 carbon atoms or R3 and R4 together with the adjacent nitrogen atom form a saturated substituted or unsubstituted monocyclic 4 to 7 membered, heterocyclic ring, which may, if desired, further contain a sulphur or oxygen atom or another nitrogen atom) or R2 represents a substituted or unsubstituted monocyclic, 6-membered nitrogen-containing heterocyclic ring attached to the adjacent carbonyl group via a carbon atom of the ring, and --- represents a single or double bond] and their acid addition salts.  The compounds described in the specification have both topical and systemic anti-inflammatory activity, an especially preferred compound being 9.alpha.-fluoro-11.beta.-hydroxy_ 16.beta.-methyl-21-morpholinoacetoxy-17-propionyloxy-prregna-1,4-diene-3,20-dione.  The specification also describes a process for preparing the above compounds as well as pharmaceutical compositions containing such compounds.
Patent CA-1053878-A (CA)
Inventor: HOKANSON ALLAN E
IPC: B01D53/77
Filed: 1975-08-22
Granted: 1979-05-08
Abstract: PROCESS FOR REMOVING CONTAMINANTS     FROM HOT WASTE GAS STREAMS            Abstract of the Disclosure A process for removing sulfur dioxide and other con-taminants from a hot waste gas stream in which the waste gas stream is cooled to a temperature below 100°F and then passed in sequence through two separate absorption zones utilizing as the absorbent a recirculated aqueous solution of ammonium sulfite-bisulfite salts.  Heat is continuously withdrawn from the recirculated salt solution in each zone.  The absorbent solution in the first zone has an initial pH of from 6 to 7.2 and a salt concentration of from 1 to 20% by weight.  The absorbent solution in the second zone has an initial pH of from 5.2 to 6.5 and a salt concentration, lower than said first zone of, from 0.1 to 5% by weight.  The process provides for the efficient absorption and substantial removal of SO2, SO3 and particulate contaminants and for the economic recovery and use of heat from stack gases of a variety of industrial and commercial operations.
Patent CA-1039860-A (CA)
Inventor: UMAN MYRON F
IPC: H01J27/00
Filed: 1975-10-27
Granted: 1978-10-03
Abstract: DOUBLE CHAMBER ION SOURCE                      ABSTRACT OF THE DISCLOSURE                The ion source is comprised of two discharge chambers one of which is provided with a filament and an aperture leading into the other chamber which in turn has an extraction orifice. A low voltage arc dis-charge is operated in an inert gas atmosphere in the filament chamber while an arc of higher voltage is operated in the second ionization chamber which contains a vapor which will give the desired dopant ion species. The entire source is immersed in an axial magnetic field parallel to a line connecting the filament, the aperture between the two chambers and the extraction orifice.
Patent CA-1047160-A (CA)
Title: Variable angle support apparatus
Inventor: WILD CHARLES E
IPC: H01Q1/12
Filed: 1975-12-10
Granted: 1979-01-23
Abstract: PATENT APPLICATION          ON VARIABLE ANGLE SUPPORT APPARATUS                 BY CHARLES E. WILD                      ABSTRACT OF THE DISCLOSURE An adjustable support apparatus adapted primarily for antennas wherein most of the load is carried by pivotal rigid structural members and the drive members are subjected to a much smaller force.  An embodiment is also described illustrating self-erection principles.
Patent CA-1038004-A (CA)
Inventor: REPLIN HENRY
IPC: B60B35/18
Filed: 1975-12-30
Granted: 1978-09-05
Abstract: ABSTRACT OF THE DISCLOSURE           Method and device for aiding and enhancing rotational movement of a member journaled with another member by biassing one of the members to an offset position relative to the other member with the offset being unstable and tending to aid rotation as a restorative force.  Particularly, a bearing device having inner and outer members which are interfaced and supported in the portion of the bearing closest to the direction from which the load is imposed and in which roller members sequentially and substantially continuously offset the inner member during rota-tion to maintain an offset having a constant orientation relati-ve to the load applied through the bearing device.
Patent CA-1040131-A (CA)
Title: Switching device for switching a transversely aligned cigarette flow in plants for directly feeding cigarettes comprising a compensating device for compensating unbalances in the output of manufacturing and packeting machines
Inventor: ENZO SERAGNOLI
IPC: A24C5/35
Filed: 1976-01-21
Granted: 1978-10-10
Abstract: ABSTRACT OF THE DISCLOSURE         The present invention provides a switching device for switching a transversely aligned cigarette flow in a plants for directly feeding cigarettes from manufacturing machines to a packaging machine and having a compensating device for compen-sating output imbalances between the manufacturing and packeting machines, in which a conveyor which removes or withdraws the cig-arettes from the manufacturing machines branches in a branching zone, one branch leading to a grouping hopper arranged to feed a wrapping line of the packeting machine and another branch lead-ing to an inlet of the compensating device, said switching device comprising a pair of arm elements removably supported at the branching zone of said cigarette feeding conveyor, end portions of said elements being shaped so as to define a guide surface which is a part of a corresponding switching path and is respect-ively located on both sides of said cigarettes on said conveyor, said arm elements co-operating with removable driving members connected to a control means monitored by said packeting machine.
Patent CA-1090936-A (CA)
Inventor: KRAFT PAUL
IPC: C08F220/00
Filed: 1976-02-09
Granted: 1980-12-02
Abstract: AQUEOUS POLYVINYL CHLORIDE CONTAINING COATING COMPOSITIONS          Abstract of the Disclosure Polyvinyl chloride containing emulsion copolymer coating compositions are formed by using any convention-al emulsion polymerization procedure, said copolymers comprising about 30% to about 47% by weight polyvinyl chloride, about 50% to about 60% of at least one C1 to C8 alkyl acrylate or methacrylate, and about 3% to about 10 of acrylic or methacrylic acid.