baber/WOPTO huggingface dataset:
Patent MD-4144-B1 (MD)
Title: Process for waste-free production from humus-containing substances of a fertilizer and a biostimulant for growth and development of plants
Inventor: GLAVNENCO NICOLAE
IPC: A01C21/00
Filed: 2011-09-22
Abstract: The invention relates to the waste-free production of ecologically clean fertilizers and biostimulants for growth and development of various farm and flower crops.The process, according to the invention, comprises the following stages:a) soaking with mixing of 1 volume of humus-containing substances with 3…5 volumes of water with a temperature of 10…40°C;b) separation after sedimentation of bacterial suspension;c) addition with agitation to the suspension residue of solid caustic alkali according to calculation: 1.5… 2.0 kg of alkali per 20 L of initial volume of the humus-containing substance with spontaneous rise in the temperature of the obtained mixture to 50…80°C;d) sedimentation of alkaline hydrolyzate suspension at room temperature;e) dilution of alkaline suspension with water to the attainment of 45…50 volumes;f) acid neutralization of the obtained diluted suspension;g) combination of neutralized suspension with the bacterial suspension obtained in the stage b);h) separation from the sediment of the supernatant fluid after sedimentation of the suspension, which is a biostimulant, in which are optionally introduced auxiliary additives, such as microelements, and packed up as necessary;i) collection of the remaining sediment in the form of dense suspension and its preparation for transportation for utilization as organic fertilizer.The result is to simplify the process and increase its efficiency, the produced biostimulant being of high quality and with a broad spectrum of activity.
Patent NO-332114-B1 (NO)
Title: Anvendelse av et pyretroid eller pyretrin samt fremgangsmate for frastotning av artropoder fra varmblodige species.
Inventor: MENCKE NORBERT
IPC: A01N65/12
Filed: 2005-08-12
Abstract: Det er beskrevet anvendelse av en artropod-frastøtende komponent fra pyrefroid/pyretrinklassen i kombinasjon med en agonist av de nikotinerge acetylkolinreseptorene av arttopoder for frastøtning av arfropoder, fortrinnsvis på dyr, på en effektiv og varig måte.
Patent NO-331205-B1 (NO)
Inventor: OLSSON LARS-ERIK
IPC: A61K38/095
Filed: 2005-10-27
Abstract: The present invention relates to a novel pharmaceutical composition as a solid dosage form comprising desmopressin as a therapeutically active ingredient, and to a method for manufacturing thereof. The invention relates to a pharmaceutical composition as a solid dosage form comprising desmopressin, or a pharmaceutically acceptable salt thereof, as a therapeutically active ingredient together with a pharmaceutically acceptable excipient, diluent or carrier, or mixture thereof, wherein at least one of said excipient, diluent and carrier is a substance selected from a monosaccharide, disaccharide, oligosaccharide and a polysaccharide, wherein the said substance has an average particle size in the range of from 60 to 1 000  mu m. A method according to the present invention provides an improved production of solid dosage forms of desmopressin.
Patent NO-338615-B1 (NO)
Inventor: RILEY ANDREW DALE
IPC: F16J7/00
Filed: 2006-02-15
Abstract: A connector assembly (46) comprises a housing (60) and a tensile member (62) disposed within the housing (60). The tensile member (60) comprises first and second end portions. Each end portion sealingly engages the housing (60) to form a hydraulic chamber (72) therebetween. A first connector (64) is pivotally coupled to the first end portion. The axial position of the first connector (64) relative to the housing (60) is controlled by pressure within the hydraulic chamber (72).
Patent NO-343146-B1 (NO)
Title: Pluggsammenstilling og fremgangsmåte for en brønnhodeåpning.
Inventor: KLEPPA ERLING
IPC: E21B47/06
Filed: 2014-04-25
Abstract: Åpningspluggsammensetning for et brønnhode, omfattende et første plugglegeme (27, 73) som omfatter koplingselementer (28) som tillater det første plugglegemet å bli forseglende og utskiftbart montert i en åpning (22b) i et brønnhode (21) i en hydrokarbonbrønn. Pluggsammensetningen omfatter en spole-enhet (24) som oppviser en aksial gjennomgående kanal (32) som strekker seg mellom en første ende (24a) og en andre ende (24b) av spole-enheten, der denne spole-enheten omfatter en første flensseksjon (33) som er anbrakt ved den første enden for forseglende montering av spole-enheten til brønnhodet ved å innrette den gjennomgående kanalen med åpningen, og en andre flensseksjon (34) anbrakt ved den andre enden, et andre plugglegeme (42, 74) som omfatter koplingselementer (43) som tillater det andre plugglegemet å bli forseglende og utskiftbart montert i den gjennomgående kanalen, og en blindflens (26, 79) som er forseglende og utskiftbart montert til den andre flensseksjonen for å tillate det andre plugglegemet og det første plugglegemet å bli fjernet fra brønnhodet via den gjennomgående kanalen.
Patent PL-81385-B1 (PL)
Title: Aqueous polymer dispersion method of producing same and their use as binders in paper coatings[us3746671a]
IPC: C08F283/08
Filed: 1970-12-18
Abstract: 1328835 Vinyl acetate polymer dispersions and their preparation VIANOVA KUNSTHARZ AG 16 Dec 1970 [19 Dec 1969(2) 9 July 1970(2)] 59764/70 Heading C3P Aqueous polymer dispersions are prepared by polymerizing in aqueous medium using a redox initiator system, 70 to 95% by weight of vinyl acetate with 5 to 30% by weight of ethyl acrylate and/or a vinyl ester of a C 3-20 carboxylic acid, in the presence of an emulsifier comprising (1) an aromatic hydroxy compound containing C 6-20 straight or branched alkyl group, which has been reacted with 2-8 moles of ethylene or propylene oxide per mole of compound, and then sulphonated, and (2) an alkylated aromatic hydroxy compound as in (1), which has been reacted with 1-40 moles of ethylene or propylene oxide per mole of compound, and/or (3) a compound of the general formula in which a = 2-40, b = 6-35, and c = 2-40. The monomer mixture may additionally contain up to 5% by weight of vinyl sulphonic acid or styrene sulphonic acid or a salt thereof. Vinyl esters of C 3-20 carboxylic acids specified, are vinyl propionate, butyrate, caproate and laurate. The monomer mixture preferably comprises 80-90% by wt. of vinyl acetate and 10-20% by wt. of ethyl acrylate and/or the other vinyl ester. The aromatic hydroxy compound in emulsifiers I and II is preferably a phenol or naphthol. The emulsifier system preferably comprises 5-95% by weight of (I), and 0-95% by weight of (II) and/or 0-95% by wt. of (III), the total being 100%. The redox initiator system may contain ammonium or an alkali metal peroxydisulphate as oxidizing agent, with ammonium or an alkali metal bisulphite, sodium dithionite or ascorbic acid as reducing agent. The dispersions are used to make coating compositions by admixing pigments such as kaolin, china clay, stain white, TiO 2 , BaSO 4 and CaCO 3 , and binders such as hydrolysed starch, casein and polyvinyl alcohol. Other usual additives may also be added.
[GB1328835A]
Patent PL-116729-B1 (PL)
Title: Process for preparing novel derivatives of carboxylic acids
IPC: C07C227/18
Filed: 1970-03-16
Abstract: Tertiary amino acids. Title cpds.: (where A Nis an alkylene-amino bicyclic gp. contg. 1-3 double bonds and 5-6 members in each ring; Ph is an opt. substd. phenylene; R1 is H or lower alkyl, and R2 is H or lower alkyl, lower alkenyl, cyclo-alkyl, cycloalkenyl, lower cycloalkylalkenyl, or lower cycloalkenyl-alkenyl). They have anti-inflammatory, analgesic and antimycotic properties.
[CH577480A5]
Patent PL-157297-B1 (PL)
Title: Web cutter in particular for tar board
IPC: B26D/
Filed: 1988-03-09
Abstract: A cutting-off machine in particular for tar board characterised in that it comprises a comb cutter (1) attached to a cutter beam (2) fastened to a post (3) to which a strand (4) is fixed which is connected by means of an articulated joint to a lever (5) and the strand (4) and lever (5) are connected also by means of an articulated joint to an actuator (6).<IMAGE>
Patent PL-158018-B1 (PL)
Title: Method of heading protection against transfer of coal dust explosion
IPC: E21F/
Filed: 1988-05-11
Abstract: 1. The method for securing mine workings to prevent transfer of coal dust explosions by their neutralisation with. The method is distinctive in that it makes use of incombustible dust in the form of phosphogypsum containing in dry mass: 92-98% by weight calcium sulfate dihydrate, less than 2% by weight free silica and about 20% by weight physical water.
Patent PL-156709-B1 (PL)
Title: Method for producing chromium complex 1:2 azo dye
IPC: C09B/
Filed: 1988-05-20
Abstract: 1. Method of producing chromic-complex azo dye 1:2 with formula 1, where M and M1 are the same or different and signify hydrogen atom or colourless cation, involving obtaining from diazotized acid, 1-amino-2-hydroxy-6-nitronaphthalenesulfonic-4 and 2-naphthol of monoazotized dye with formula 2, then, after transferring obtained monoazotized dye with formula 2, and after possible isolation from the post-reaction mixture into chromic complex 1:1, by action of trivalent chromium salt, such as sulphate and/or alkaline chromium sulphate, under pressure and in acidic element at more than 100 degrees C, then subjecting obtained chromic complex 1:1 of monoazotized dye with formula 2, to reaction with monoazotized dye with formula 3, obtained by interacting diazotized 5-nitro-2-aminophenol with 2-naphthol, where reaction of creating asymmetric chromic-complex dye 1 : 2 is performed at elevated temperature with pH above 4; is characterised in that; obtained from reaction of diazotized acid 1-amino-2-hydroxy-6-nitronaphthalenesulfonic-4 with 2-naphthol, monoazotized dye with formula 2 is transferred into chromic-complex 1: 1 by action of sulphate and/or alkaline chromium sulphate used in quantity of 0.9-1.1 moles of Cr, especially 1.0-1.05 moles of Cr for 1.0 mole of monoazotized dye with formula 2, at temperature of 110-130 degrees C with pH 1.0-3.5, especially with pH 1.5-3.0, in volume of the reaction mixture.<IMAGE>
Patent PL-156375-B1 (PL)
Title: Herbicide for selectively fighting against weeds and grass in useful plant cultures
IPC: C07D249/10
Filed: 1988-09-30
Abstract: 1,5-Diphenyl-1,2,4-triazole-3-carboxylic acid derivatives of formula <IMAGE> (I)  wherein each of Ra and Rb, independently of the other, is halogen, C1-C5alkyl, C1-C5haloalkyl, C2-C5alkenyl, C2-C5alkynyl or cyano, n is zero or a number from 1 to 3 and OR is hydroxy, a phytophysiologically tolerable metal or ammonium salt radical, or an ester radical defined in the description, are capable of specifically antagonizing the phytotoxic action of herbicides. 1,5-Diphenyl-1,2,4-triazole-3-carboxylic acid derivatives of formula I and the preparation thereof, compositions containing these components as selective herbicides and the use of these two active ingredient components for controlling weeds in crops of useful plants are described.
Patent PL-161181-B1 (PL)
Title: Method of separating racemic mixture of spirohy-dantoin compounds
IPC: C07D491/107
Filed: 1989-07-25
Abstract: A novel three-step process for resolving a racemic spiro-hydantoin compound into its optical antipodes is disclosed, which involves (1) reacting said racemic compound with an optically-active asymmetric isocyanate of the formula RNCO, wherein R is (S)- or (R)-1-phenylethyl or (S)- or (R)-1-(1-naphthyl)ethyl, to form the corresponding diastereomeric ureido compound; (2) separating the resulting diastereomeric mixture into its component parts, and (3) thereafter converting the separated ureido diastereomers obtained in step (b) to the corresponding asymmetric hydantoin compounds by treatment with an alkali metal lower alkoxide (C1-C4), followed by acidification, whereupon the desired optical isomer is obtained. The final products so obtained, such as (4S)-(+)-6-fluoro-2,3-dihydro-spiro[4H-1-benzopyran-4,4 min -imidazoli dine]-2 min ,5 min -dione (sorbinil) and (5 min S)-3 min -chloro-5 min ,6 min ,7 min ,8 min -tetrahydro-spiro[i midazolidine-4,5 min -quinoline]-2,5-dione, are known to be useful in preventing or alleviating certain chronic diabetic complications. The aforementioned diastereomeric ureido intermediates are novel compounds.
Patent PL-161485-B1 (PL)
IPC: A61M25/00
Filed: 1989-11-10
Abstract: Prowadnik, zwłaszcza cewnika naczyń wieńcowych
serca, zawierający część penetrującą utworzoną
przez sprężysty rdzeń, korzystnie wygięty w kształcie
okręgu, na którym nałożona jest sprężysta osłoną połączona
z rdzeniem najego wolnym końcu i która to część
penetrująca połączona jest z częścią manewrującą zawierającą
koncentryczny korpus z usytuowanym wewnątrz
przedłużeniem rdzenią znamienny tym, że w
korpusie (1) na rdzeniu (7) ma sprężynę (3) opartą swym
końcem o ściankę koncentrycznego przesuwnego przycisku
(2) osadzonego wewnątrz korpusu (1), przy czym
przycisk (2) zaopatrzony jest w element mocujący (4) go
do rdzenia (7), a korpus zaopatrzony jest w element
mocujący osłonę (6) do korpusu (1)
Patent PL-166791-B1 (PL)
Inventor: BIENKOWSKI KAZIMIERZ
IPC: G01S11/16
Filed: 1992-01-22
Abstract: 1. Sposób pomiaru odległości przemieszczających
się obiektów względem pomocniczego obiektu,
zwłaszcza węzłowej stacji danych sieci komputerowej,
zgodnie z którym mierzy się czas, w którym
sygnał radiowy i akustyczny pokonuje drogę między
obiektem przemieszczającym się, a obiektem pomocniczym,
przez zliczanie impulsówelektrycznych, znamienny
tym, że z drugiego nadajnika radiowego (12)
obiektu przemieszczającego się (8) wysyła się, poprzez
drugą antenę nadawczą (9), sygnał radiowy (B),
a po odebraniu tego sygnału przez pierwszy odbiornik
radiowy (5), zainstalowany na obiekcie pomocniczym
(1), wysyła się sygnał akustyczny (S) przez nadajnik
sygnałów akustycznych (7), umieszczony na tym
obiekcie pomocniczym (1), i mierzy się czas od chwili
wysłania sygnału radiowego (B) do chwili odebrania
sygnału akustycznego (S).
Patent PL-167208-B1 (PL)
Inventor: HANKUS JAN
IPC: D07B1/06
Filed: 1992-12-02
Abstract: Lina stalowa wyciągowa o punktowym i
liniowym styku drutów, okrągła, okrągłosplotkowa,
współzwita lub przeciwzwita, składająca
się z co najmniej sześciu okrągłych splotek oraz
rdzenia organicznego, znamienna tym, że stosunek
średnicy drutu rdzeniowego (3) w splotce (2) do
średnicy drutów (4) pierwszej warstwy wynosi
1,065-1,075, do średnicy drutów (5) drugiej warstwy
0,575 - 0,585, do średnicy cieńszych drutów (6)
trzeciej warstwy 0,830-0,850, do średnicy grubszych
drutów (7) trzeciej warstwy 0,635 - 0,645 i do
średnicy drutów zewnętrznych (8) 0,540-0,550,
przy czym stosunek skoku zwicia drutów (4) pierwszej
warstwy do średnicy drutów tej warstwy
wynosi 27,7-28,0, a stosunek skoków zwicia drutów
(5, 6, 7, 8) wszystkich pozostałych warstw
splotki (2) do średnicy drutów zewnętrznych (8)
wynosi 55 - 56.
Patent PL-163432-B1 (PL)
Title: Method for manufacturing peptide derivatives
Inventor: ALBERT RAINER
IPC: A61P35/00
Filed: 1989-12-04
Abstract: 1. Method for producing new somatostatine peptide derivatives including a chelating group capable of creating a complex with detectable metal ion, optionally in the form of salt or in the form of a complex with detectable metal ion, which group is directly or indirectly attached to the terminal amine group, whereas the somatostatine peptide is natural somatostatine or a compound of formula 1 where A stands for a group of formula RCO, where RCO-stands for:a) an L- or D-phenylalanine residue optionally ring-substituted by F, Cl, Br, NO2, NH2, OH, C1-3 alkyl and/or C1-3 alkoxy;b) the residue of a natural or synthetic α-amino acid other than defined under a) above or of a corresponding D-amino acid, orc) a dipeptide residue in which the individual amino acid residues are the same or different and are selected from those defined under a) and/or b) above, A' stands for hydrogen, Y1 and Y2 represent together a direct bond or each of Y1 and Y2 is independently hydrogen, B stands for -Phe - optionally ring-substituted by halogen, NO2, NH2, OH, C1-3alkyl and/or C1-3 alkoxy (including pentafluoroalanine, or Β-naphthyl-Ala, C stands for (L)-Trp- or (D)-Trp-, D stands for Lys, E stands for Thr, Ser, Val, Phe, Ile or an aminoisobutyric or aminobutyric acid residue, G stands for group of formula 10 wherein R11 stands for hydrogen, C1-3 alkyl, R12 stands for hydrogen, C1-3 alkyl or a group of formula -CH(R13)-X1.<IMAGE>
Patent PL-170680-B1 (PL)
Inventor: BONIN JAN
IPC: E02D19/10
Filed: 1993-04-19
Abstract: 1. Samoczynna bariera hydrogeologiczna,
zawierająca liczne pionowe odwadniające
studnie z przewodami czerpalnymi,
znamienna tym, że składa się z licznych,
korzystniejednakowych, ustawionych wjednej
linii (X-X) prostopadłej do kierunku (P)
przepływu wód podziemnych, studni (1), z
których każda na odcinku rury nadfiltrowej
(K) ma wykonany przelewowy otwór (2),
którego górna krawędź znajduje się na określonym
poziomie (H) zwierciadła wody w
studni i do któregojestszczelnie utwierdzony
przelewowy przewód grawitacyjny (3), przebiegający
najkorzystniej równolegle do kierunku
(P) przepływu wód, przyłączony
przeciwnym końcem wolnym (4) do oddalonego
magistralnego przewodu grawitacyjnego
(5), przebiegającego najkorzystniej
równolegle do linii (X-X) usytuowania studni
(1)
Patent PL-172515-B1 (PL)
Inventor: LUNARSKI JERZY
IPC: B23P19/06
Filed: 1994-02-21
Abstract: 1. Urzadzenie elektromechaniczne do mon- tazu polaczen gwintowych zawierajace glowice robocza i jednostke napedowa, znamienne tym, ze pomiedzy glowica (1) a jednostka na- pedow a (3) zabudow any je st w ariator elektromechaniczny (2) zawierajacy mecha- nizm róznicowy (24), którego kola talerzowe (21) i (22) sa osadzone na prawej (15) i lewej (25) obejmie wariatora, satelity (23) w jarzmie (27) lozyskowanym w obejmie (28) zakonczo- nej walkiem zdawczym (29), a zlobkowany wirnik (35) z wieloselekcyjnym zamknietym uzwojeniem (36) jest osadzony w prawej i lewej obejmie wanatora. PL
Patent PL-179636-B1 (PL)
Title: Novel derivatives of taxane and pharmaceutical agents
IPC: C07D/
Filed: 1994-08-16
Abstract: The present invention concerns antitumor compounds. More particularly, the invention provides novel taxane derivatives, pharmaceutical compositions thereof, and their use as antitumor agents.
Patent PL-177841-B1 (PL)
Inventor: Staszczuk Piotr
IPC: C01F11/18
Filed: 1994-12-28
Abstract: Sposób otrzymywania adsorbentu dolomitowego polegający na obróbce termicznej
i chemicznej materiału wyjściowego, znamienny tym, że materiał wyjściowy stanowi
rozdrobniony dolomit naturalny, który wygrzewa się w temperaturze 820 - 850°C przez
okres 4-20 godzin, po czym materiał poddaje się wymywaniu przy pomocy rozpuszczalnika
zasadowego o pH = 7 - 9,5, korzystniebuforu boraksowego lub amonowego, z udziałemultradźwięków
i suszy w temperaturze 120°C w ciągu 24 godzin.
Patent PL-181527-B1 (PL)
Inventor: BUSZEWSKI BOGUSLAW
IPC: G01N31/00
Filed: 1996-12-31
Abstract: Sposób oznaczania benzoesanu benzodietylo(2,6-ksylilokarbamylometylo)amoniowego
znamienny tym, że benzoesan benzodietylo(2,6-ksylilokarbamylometylo)amoniowy
zawarty wmatrycy ciekłej lub stałej poddaje się selektywnej sorpcji w układzie kolumny filtracyjnej,
korzystnie z porowatym filtrem chemoodpornym z polipropylenu i kolumny sorpcyjnej
wypełnionej adsorbentem zawierającym chemicznie związaną fazę C-18, korzystnie
z gęstym pokryciem powierzchni nośnika krzemionkowego, a następnie desorpcji za pomocąmieszaniny
rozpuszczalników polarnych i niepolamych, po czym po ich odparowaniu,
suchą pozostałość rozpuszcza się w mieszaninie acetonitrylu i wodnego roztworu chlorku
sodu, po czym poddaje oznaczeniu ilościowemu za pomocąwysokosprawnej chromatografii
cieczowej, korzystnie z zastosowaniem kolumny analitycznej wypełnionej selektywną fazą
stacjonarną zawierającą ugrupowania N-acyloaminowe.
Patent PL-181652-B1 (PL)
Inventor: JANISZEWSKI MAREK
IPC: H01Q15/14
Filed: 1997-01-29
Abstract: Reflektor antenotty, zwłaszcza
kątowy o postaci kratownica, znamienny
tym, że jest utworzony z niemetalowych elementów
nośnych (1) usytuowanych równolegle
do siebie i metalowych elementów
odbijających (2) usytuowanych prostopadle
do elementów nośnych (1), przy czym elementy
nośne (1) są wygięte tworząc dwie
płaszczyznyusytuowane podkątem50-110°.
Patent PL-182057-B1 (PL)
Title: Novel immunotherapeutic aryl amides
Inventor: MULLER GEORGE
IPC: C07C233/47
Filed: 1995-11-20
Abstract: Novel aryl amides are inhibitors of tumor necrosis factor  alpha  and can be used to combat cachexia, endotoxic shock, and retrovirus replication. A typical embodiment is N-benzoyl-3-amino-3-(3',4'-dimethoxyphenyl)propanamide.
Patent PL-183979-B1 (PL)
Title: Apparatus for dosing volatile active ingredient
Inventor: DANCS IMRE J
IPC: B01F3/04
Filed: 1996-05-08
Abstract: A dispensing device for dispensing a volatile active ingredient from an air-transmitting substrate that forms a part of a refill assembly. The dispensing device includes a housing which has a foot (78) with an angled support surface and a horizontal support surface. The housing has an intake vent and an exit vent and an air flow path extending between them. Refill assembly support means are provided for removably supporting the refill assembly with its substrate located in the air flow path. Battery-powered fan means are provided for propelling air from the intake vent through the substrate and out the exit vent. The battery is positioned in the device sufficiently far forward that the centre of gravity of the device is above the horizontal support surface of the foot when the device is resting on the foot, and is above the angled support surface when the device is nesting on the angled surface. This makes the device stable in both an horizontal position, or in a tilted position. 
     An air-transmitting refill assembly for use with the dispensing device includes an air-transmitting substrate and a tab attached to the margin of the substrate. The tab has a brace surface facing generally away from the substrate and shaped to engage the surface of a battery being held within the battery holder of the dispensing device.
Patent PL-191576-B1 (PL)
Title: Pharmaceutic agent and method of obtaining same
Inventor: SCHUBERT HANS-PETER
IPC: C07D473/06
Filed: 1998-02-26
Abstract: A combination of the following components for simultaneous, separate or sequential administration is new: (a) an acetylcholinesterase inhibitor or compound with muscarinergic activity, (b) a compound that increases endogenous extracellular adenosine levels, and (c) a pharmaceutical carrier.
Patent PL-193297-B1 (PL)
Inventor: GROEBKE KATRIN
IPC: C07D/
Filed: 1998-12-04
Abstract: 1. Pochodne N-(karbamimidofenylo)-glicynamidu o wzorze 1, w którym E oznacza atom wodoru albo grupe OH, Q oznacza atom wodoru albo grupe alkilowa, R ozna- cza grupe arylowa, cykloalkilowa albo alkilowa, która jest podstawiona przez R 1 , R 2 i R 3 , R 1 oznacza atom wodoru, grupe COOH, grupe COO-alkilowa albo arylowa, R 2 ozna- cza atom wodoru, grupe arylowa, cykloalkilowa albo hete- roaryIowa, R 3 oznacza atom wodoru, grupe arylowa albo (w pozycji róznej od pozycji a wobec atomu azotu, z którym zwiazana jest grupa alkilowa R) grupe OH, grupe alkoksy- lowa albo ewentualnie chroniona grupe aminowa, N(Q,R) oznacza podstawiona przez grupe COOH albo przez grupe COO-alkilowa grupe pirolidynowa, piperydynowa albo 1,2,3,4-tetrahydroizochinolin-3-ylowa, trzy sposród pod- stawników X 1 do X 4 niezaleznie od siebie oznaczaja grupe C(R a ), C(R b ) albo C(R c ), a czwarty podstawnik oznacza grupe C(R d ) albo N, R a do R d niezaleznie od siebie ozna- czaja atom wodoru, grupe OH, NO 2, grupe dialkiloaminowa, atom chlorowca, grupe alkilowa, alkoksylowa, aryloksylowa, aralkiloksylowa, heteroaryloalkiloksylowa, heterocykliloalki- loksylowa, COOH, COO-alkilowa, NH-SO 2-alkilowa, NHSO 2- -arylowa, NHCO-alkilowa, NHCO-arylowa, NHCOO-alkilowa, NHCO-alkilo-NH 2, NHCO-alkilo-NH-G, aralkilo-CONH, alkilo- -O-alkilo-CONH, arylo-O-alkilo-CONH, alkilo-COOH, ……… PL PL PL PL PL PL PL