baber/WOPTO huggingface dataset:
Patent JP-3030087-B2 (JP)
IPC: C07H5/02
Filed: 1992-11-13
Granted: 2000-04-10
Abstract: 2'-Deoxy-2'-fluorocoformycin and 2'-deoxy-8-epi-2'-fluorocoformycin have now been synthesized by a multistage reaction via 3,5-di-O-benzoyl-2-deoxy-2-fluoro- alpha - and - beta -D-ribofuranosyl bromide. Also 2'-deoxy-2'-epi-2'-fluorocoformycin and 2'-deoxy- 8,2'-diepi-2'-fluorocoformycin have been synthesized from 3,5-di-O-benzoyl-2-deoxy-2-fluoro- alpha -D-arabinofuranosyl bromide by a multistage reaction. These four 2'-fluorocoformycin derivatives are novel compounds and have a potent enzyme inhibiting activity against adenosine deaminase. In particular, they are useful for treating acute lymphocytic leukemia in virtue of the above activity. Other novel compounds also obtained include various intermediates useful for the synthesis of the above derivatives.
Patent JP-4001618-B2 (JP)
IPC: C07C403/20
Filed: 1992-12-18
Granted: 2007-10-31
Abstract: In accordance with the present invention, there are provided methods to modulate processes mediated by retinoid receptors, employing high affinity, high specifity ligands for such receptors. In one aspect of the present invention, there are provided ligands which are more selective for the retinoid X receptor than is retinoic acid (i.e., rexoids). In another aspect of the present invention, alternative ligands (other than retinoic acid) have been discovered which are capable of inducing retinoic acid receptor mediated processes. In yet another aspect, methods have been developed for the preparation of such retinoid receptor ligands from readily available compounds.
Patent JP-3113277-B2 (JP)
IPC: H03M3/02
Filed: 1993-01-28
Granted: 2000-11-27
Abstract: PCT No. PCT/FI93/00027 Sec. 371 Date Aug. 11, 1994 Sec. 102(e) Date Aug. 11, 1994 PCT Filed Jan. 28, 1993 PCT Pub. No. WO93/15557 PCT Pub. Date Aug. 5, 1993The invention relates to a method for cascading two or more feedforward-type sigma-delta modulators, and a modulator system comprising at least two cascaded modulators (1, 2). According to the invention, each subsequent modulator (2) in the cascade quantizes the integrated signal estimate error (e) of the preceding modulator (1), the quantized error (e') is differentiated (3) and subtracted (6) from the quantized output signal (D'') of the preceding modulator (1).
Patent JP-3459066-B2 (JP)
IPC: A61M5/315
Filed: 1993-04-21
Granted: 2003-10-20
Abstract: PCT No. PCT/AU93/00175 Sec. 371 Date Jan. 18, 1995 Sec. 102(e) Date Jan. 18, 1995 PCT Filed Apr. 21, 1993 PCT Pub. No. WO93/20872 PCT Pub. Date Oct. 28, 1993A parenteral device (10) comprising a body (12) having a forward end (26) and a rearward end (34). The forward end (26) is capable of receiving a hollow retractable needle (20) therein so as to project therefrom. The retractable needle (20) is slidable relative to the body (12) and the body (12) also includes a chamber (14) capable of receiving parenteral fluid and capable of being reduced in volume to expel fluid contained therein. The needle (20) is capable of being manually retracted within the body (12) such that the chamber (14) reduces in volume to expel fluid contained therein and such that the needle (20) is retracted to be wholly contained within the body (12).
Patent JP-3335179-B2 (JP)
IPC: F16H3/74
Filed: 1997-11-20
Granted: 2002-10-15
Abstract: The present invention relates to a continuously variable transmission constructed in such a way that it can speed-change the power inputted to an input shaft according to the load applied to an output shaft and transmit the power to the output shaft even though all the gears remain engaged, and in addition reverse operation can also be effectuated in a simple way.Reviewing the construction thereof, it is mainly composed of a speed change system, which receives power generated by an engine, changes speed and transmits it to the output shaft, a speed change controlling system which automatically adjusts the rotational ratio to correspond to the condition of the load on the output shaft, and a reverse rotation system.The present invention, comprises two (compund) gear sets in which each same element is removed from two planet gear sets; and a reverse rotation system, and the power inputted through an input element selected from the two gear sets is changed into the required speed and transmitted to the output shaft.Reviewing the operational characteristics, the present invention is constructed in such a way that the decelerated rotation smaller than the input rotation is transmitted to the impeller by utilizing an direct clutch. Therefore, it is a characteristic of the present invention that the rotational force transmitted to the impeller is alway larger than the input torque.In view of the effects, the present invention can obtain a large propulsion force, preferable performance, smooth and quiet operation, and can speed-change steplessly at the time of reverse operation.
Patent JP-3230817-B2 (JP)
IPC: G01L5/00
Filed: 1996-02-16
Granted: 2001-11-19
Abstract: A system for measuring the dynamic pressure distribution between rolls in a nip roll press comprises a roll adapted to rotatingly contact at least one other roll in a press nip, having one or more sensors thereon, for measuring the nip pressure at several locations along the roll length, wherein the measurements obtained by the sensors are transmitted to a computer and a display, to provide tabular, numerical and graphical representations of the pressure at one or more locations on the roll. Optionally a control system may be incorporated in the system for determining the pressure distribution along the roll and initiating corrective measures. The system of the instant invention can further measure temperature variations, if desired, as thermal sensors can be used on the sensing roll, or a computerized correlation scheme can relate sensor readings to temperature as well as pressure.
Patent JP-3771276-B2 (JP)
IPC: A61F13/53
Filed: 1997-03-27
Granted: 2006-04-26
Abstract: Absorbent article comprises an absorbent core comprising a crotch region and one or more waist regions. The crotch region has a lower ultimate fluid storage capability than the waste regions together. The article has a crotch region Post Acquisition Collagen Rewet Method value of less than 180 mg.
Patent JP-4118962-B2 (JP)
IPC: C08L23/04
Filed: 1998-04-21
Granted: 2008-07-16
Abstract: Halogen-free thermoplastic blends of a polar rubber, ethylene vinyl acetate and a polyolefin. are provided which are flexible and are particularly useful in replacing polyvinyl chloride for production of various products.
Patent PL-119823-B2 (PL)
Title: Fungicide
IPC: C07D233/60
Filed: 1979-10-16
Abstract: New compounds of the formula   <IMAGE>   which have a good fungicidal action, their manufacture, fungicides containing these compounds as active ingredients, and processes for combating fungi with these compounds.
Patent PL-160694-B2 (PL)
Title: Method of purifying crude sulfite wood turpentine
IPC: C09F3/00
Filed: 1989-07-04
Abstract: 1. A method of refining raw sulphate turpentine oil with the use of a water solution of alkali metal hypochlorite, characterised in that the solution of the hypochlorite is entered into the continuously flowing stream of turpentine oil in counter stream, where the amount of the hypochlorite per one part of turpentine is divided into at least two separate streams introduced in various places into the stream of turpentine, and the final product is discharged behind the last hypochlorite feeding point.
Patent ES-2498490-B2 (ES)
Title: Método para la generación de modelos realistas en tres dimensiones de células neuronales
Inventor: MATA FERNANDEZ SUSANA
IPC: G06T17/20
Filed: 2013-02-20
Granted: 2015-02-23
Abstract: Esta invención presenta un método para la generación de modelos tridimensionales de células neuronales partiendo de la información morfológica incompleta extraída mediante métodos de muestreo estándar. Los modelos generados incluyen un soma realista, árboles dendríticos y axonales, y espinas dendríticas, pudiendo ser generados a diferentes niveles de resolución. La invención propone una técnica innovadora que permite obtener una forma realista del soma partiendo de una definición simple del mismo (tal como centro y radio) que resulta incompleta para reconstruir la forma 3D original. El método propuesto se basa en la deformación de una forma inicial, guiada por restricciones establecidas de acuerdo a las propiedades morfológicas de los árboles dendríticos y axonales (por ejemplo: posición y grosor de las dendritas de primer orden). La distribución de un conjunto de espinas a lo largo de las dendritas completa el modelo, generando un modelo tridimensional adecuado para su visualización en una amplia gama de entornos 3D.
Patent ES-2472140-B2 (ES)
Title: Método de proyección de sólidos sobre una superficie
Inventor: TOMAS CLARAMONTE JOSÉ VICENTE
IPC: B28B19/00
Filed: 2014-02-07
Granted: 2015-01-29
Abstract: Método para la deposición de sólidos sobre una superficie, mediante la asociación de al menos una boquilla o inyector, que contiene al menos un orificio de eyección, asociado con al menos un transductor, de forma que la activación de dicho transductor, en contacto con alguna de las superficies del inyector, produzca sobre éste, movimientos oscilantes o vibratorios de la superficie que contiene el orificio de eyección y de tal forma que un material sólido, pulverulento o granulado, situado en su interior sea proyectado por la parte inferior de dicha boquilla o inyector a través del orificio del inyector y en una dirección (z) perpendicular al plano en que se sitúa dicho orificio, de forma que dicho material se deposita sobre una superficie situada bajo el inyector.
Patent AU-2001216117-B2 (AU)
Title: Method for converting oxygenates to olefins
Inventor: LATTNER JAMES R
IPC: C07B61/00
Filed: 2000-11-16
Granted: 2005-02-17
Abstract: The present invention provides a method for converting a feed containing oxygenates to olefins and comprises the following steps: providing a feed including an oxygenate; contacting the feed in a reactor apparatus with a catalyst including a molecular sieve, the contacting taking place under conditions effective to convert the oxygenate to a product including a light olefin, the conditions including a gas superficial velocity of at least two meters per second at least one point in the reaction zone; and recirculating a first portion of the catalyst to recontact the feed.
Patent AU-2001277935-B2 (AU)
Title: Alpha v integrin receptor antagonists
Inventor: WANG JIABING
IPC: A61K31/4745
Filed: 2001-07-20
Granted: 2005-08-04
Abstract: The present invention relates to novel chain-fluorinated alkanoic acid derivatives thereof, their synthesis, and their use as alphav integrin receptor antagonists. More particularly, the compounds of the present invention are antagonists of the integrin receptors alphavbeta3 and/or alphavbeta5 and are useful for inhibiting bone resorption, treating and preventing osteoporosis, and inhibiting vascular restenosis, diabetic retinopathy, macular degeneration, angiogenesis, atherosclerosis, inflammation, inflammatory arthritis, viral disease, cancer, and metastatic tumor growth.
Patent AU-2002310250-B2 (AU)
Title: Compositions of alkanolamine salts of alkyl phosphate esters
Inventor: SOMAN SUBHASH
IPC: C09K23/00
Filed: 2002-06-03
Granted: 2007-08-16
Abstract: Disclosed are pumpable surfactant compositions of alkanolamine salts of alkyl phosphate esters. The compositions have a solids content of about 60% by weight or more. Alkanolamines useful in preparation of the alkyl phosphate ester salts of the compositions of the present invention have the following formula III:wherein R4 to R6 are, individually, hydrogen or C1-8, linear or branched alkyl, alkenyl, alkaryl or aralkyl hydrocarbon moieties, which optionally may contain carbocyclic rings. At least one of the amine substituents is different from the other two. For at least one of the three substituents on the amine nitrogen, the sum of s and t (s+t) or v and w (v+w) or x and y (x+y) is equal to or greater than 1 and the corresponding R (R4, R5 or R6) is hydrogen. The subscripts p and q, individually, may be the same or different and are integers from 2 to 4. The subscripts s, t, v, w, x, and y, individually, may be the same or different and are integers of from 0 to 10, with the proviso that the sum of all six of the subscripts is less than or equal to 12.
Patent AU-2002342135-B2 (AU)
Title: High speed embossing and adhesive printing process and apparatus
Inventor: TOUSSANT JOHN WILLIAM
IPC: C09J7/20
Filed: 2002-10-25
Granted: 2006-05-25
Abstract: A high speed embossing and adhesive printing process using a first and second embossing rolls having complementary embossing pattern disposed thereon. A web of sheet material is placed in contact with an adhesive applied to the first embossing roll. The adhesive forms an adhesive pattern on the web of sheet material in register with the first embossing pattern of the first embossing roll. The web of sheet material is then passed between the first and second embossing rolls which emboss the web with the complementary embossing pattern.
Patent AU-2002345075-B2 (AU)
Title: Panel with sound insulation layer and production method
Inventor: RUHDORFER HERBERT
IPC: E04B5/43
Filed: 2002-06-28
Granted: 2007-09-20
Abstract: The invention relates to a method for applying to a flooring panel a layer designed to reduce the footfall sound on the floor, and a panel of this kind. With the prior art, it is disadvantageous that the sound-insulation layer is glued onto the laminate panel in a subsequent manufacturing stage. Accordingly, the panel is initially manufactured by pressing with the associated gluing of layers and/or papers. The sound-insulation layer is glued in place in a subsequent operational stage. PVA-glues, thermoplastics or wood glues may be used, for example, to attach the sound-insulation layer. In the manufacture of a panel with a carrier board, decorative paper, counteracting paper and/or a wood veneer, an additional layer, preferably in the form of a sheet or a roll, is provided. The material of this roll or sheet product is designed to provide the desired sound-insulation properties as described above and/or provides these properties when a panel is being walked over. The roll or sheet product is placed in a press and pressed together with the other components at a temperature of at least 100° C.
Patent AU-2003243089-B2 (AU)
Title: Novel compounds, their use and preparation
Inventor: SJOBERG BIRGER
IPC: A61P1/14
Filed: 2003-06-18
Granted: 2010-01-07
Abstract: The invention relates to compounds of the general Formula (I). The compounds may be prepared by per se conventional methods and can be used for treating a human or animal subject suffering from a serotonin-related disorder. The invention also relates to such use as well as to pharmaceutical compositions comprising a compound of Formula (I).
Patent AU-2003275209-B2 (AU)
Title: UV led based water purification module for intermittantly operable flow-through hydration systems
Inventor: MAIDEN MILES
IPC: C02F1/32
Filed: 2003-09-24
Granted: 2009-11-26
Abstract: A wearable or portable intermittently operable hydration system (10) includes a purification module (22, 50) that contains one or more solid state UV devices that are positioned in the path of hydrating fluid, or water, flow through the hydration system to a mouthpiece (18). The UV LEDs are instant on devices with essentially no ramp-up required, and a sensor (20) or the opening of a push-pull valve (53) controls the turning on of the UV LEDs. The fluid flow path may run from a bladder (12) in a backpack (19) worn by the user, a sports bottle (54) worn by or carried by the user or may be through a water filtration system that a user operates via a pump. The power for the purification module may come from batteries, solar cells, fuel cells, power converted from pumping or winding action or any combination thereof.
Patent AU-2003296596-B2 (AU)
Title: Halothenoyl-cyclopropane-1-carboxylic acid derivatives
Inventor: CACCIA CARLA
IPC: A61P25/00
Filed: 2003-11-25
Granted: 2010-03-04
Abstract: Compounds of formula (I) <CHEM> wherein R is hydroxy, linear or branched C1-C6 alkoxy, phenoxy, benzyloxy, a group -N(R<1>R<2>) wherein R<1> is hydrogen, linear or branched C1-C4 alkyl, benzyl, phenyl and R<2> is hydrogen or linear or branched C1-C4 alkyl, or R is a glycoside residue or a primary alkoxy residue from ascorbic acid, optionally having one or more hydroxy groups alkylated or acylated by linear or branched C1-C4 alkyl or acyl groups; X is a halogen atom and n 1 or 2 are long lasting inhibitors of kynurenine 3-monooxygenase (KMO) and potent glutamate (GLU) release inhibitors.
Patent AU-2004200454-B2 (AU)
Title: Enrolling/sub-enrolling a digital rights management (DRM) server into a DRM architecture
Inventor: KOSTAL GREGORY
IPC: G06Q20/36
Filed: 2004-02-10
Granted: 2009-10-29
Abstract: A Digital Rights Management (DRM) system has a plurality of DRM servers performing DRM functionality and an entering DRM-E server is enrolled into the system by an enrolling DRM-R server such that the entering DRM-E server is to be trusted within the system. The DRM-E server sends an enrollment request to the DRM-R server including a proffering identification and a public key (PU-E). The DRM-R server validates the proffering identification, and, if the request is to be honored, generates a digital enrollment certificate with (PU-E) for the DRM-E server to enroll such DRM-E server into the DRM system. The now-enrolled DRM-E server with the generated enrollment certificate is able to employ same to issue DRM documents within the DRM system. <IMAGE>
Patent AU-2004209426-B2 (AU)
Title: Method for preparing single-stranded DNA libraries
Inventor: WEINER MICHAEL P
IPC: G01N21/25
Filed: 2004-01-28
Granted: 2008-04-17
Abstract: An apparatus and method for performing rapid DNA sequencing, such as genomic sequencing, is provided herein. The method includes the steps of preparing a sample DNA for genomic sequencing, amplifying the prepared DNA in a representative manner, and performing multiple sequencing reaction on the amplified DNA with only one primer hybridization step.
Patent AU-2004220183-B2 (AU)
Title: Photochromic multilayer body and method for producing same
Inventor: IZUMI SHINOBU
IPC: C09D7/62
Filed: 2004-03-09
Granted: 2009-09-03
Abstract: A photochromic laminate comprising a base material of a thermoplastic resin having light-transmitting property, a crosslinked resin layer formed on the surfaces of the base material and containing inorganic colloidal particles in an amount of 20 to 40% by mass, and a photochromic coating formed on the surfaces of the crosslinked resin layer. Though the laminate has the layer exhibiting photochromic property formed thereon by the coating method, the surfaces of the base material of a thermoplastic resin are suppressed from being whitened or swollen. Therefore, the base material exhibits excellent optical properties, a high adhesiveness to the photochromic coating, and superior durability.
Patent AU-2004261045-B2 (AU)
Title: Disinfection of a contaminated environment
Inventor: CAUNT PHILIP
IPC: A61Q17/00
Filed: 2004-07-29
Granted: 2007-12-13
Abstract: A formulation to reduce the numbers of bacteria, particularly Gram positive bacteria, in a space such as a waste disposal bin, via the vapour phase, and active over a long period, typically several weeks. The product comprises one or more essential oil components plus a mixture of volatile and non-volatile solvents, on a carrier such as a non-woven sintered plastic or cardboard.
Patent AU-2004281226-B2 (AU)
Title: Water-soluble glass composition
Inventor: HAHN KARLHEINZ ULRICH GERHARD
IPC: C11D3/02
Filed: 2004-10-18
Granted: 2009-10-29
Abstract: A zinc and bismuth containing, water-soluble glass composition comprising from 10 to 75 mole % P<SUB>2</SUB>0<SUB>5</SUB>, 5-50 mole % alkali metal oxide, up to 40 mole % ZnO and up to 40 mole % Bi<SUB>2</SUB>0<SUB>3</SUB>.
Patent AU-2004308632-B2 (AU)
Title: Probiotic tablet formulations
Inventor: HENRIKSEN KRISTIAN LUND
IPC: A23L33/15
Filed: 2004-12-21
Granted: 2010-07-01
Abstract: A probiotic tablet comprising a probiotic micro-organism and other nutritionally active ingredients in two zones, a first zone comprising said probiotic micro-organism and precisely selenium, and a second zone comprising at least one said other active ingredient such as iron, other minerals and vitamin B6 kept separated from the probiotic micro-organism of said first zone, the water activity in said probiotic micro-organism containing first zone being no greater than 0.2 and the water content of said tablet being as much as 3% by weight. Good viability of the micro-organisms is obtained despite the relatively high overall moisture content.
Patent AU-2005289753-B2 (AU)
Title: CRC counter normalization
Inventor: TZANNES MARCOS C
IPC: H04L1/24
Filed: 2005-09-23
Granted: 2008-12-04
Abstract: The ability to accurately and efficiently calculate and report communication errors is becoming more important than ever in today's communications environment. More specifically calculating and reporting CRC anomalies in a consistent manner across a plurality of communications connections in a network is crucial to accurate error reporting. Through a normalization technique applied to a CRC computation period (e.g., the PERp value), accurate error identification and reporting for each individual connection can be achieved. In particular, severly errored seconds are detected and reported.
Patent AU-2005308881-B2 (AU)
Title: Process for preparing halogenoalkylnitrates
Inventor: RIVOLTA ROMANO
IPC: C07C205/08
Filed: 2005-11-09
Granted: 2010-10-28
Abstract: A process for preparing a compound of formula (I) X-(CH2)n-ONO2  (I) wherein: X is a halogen atom selected from Cl, Br, I; n is an integer from 3 to 6; said process comprising the slow addition of a compound of formula (II) X-(CH2)n-OH  (II) wherein X and n are as defined above to a nitrating agent selected from the group consisting of concentrated nitric acid/concentrated sulfuric acid (sulfonitric mixture), nitric acid alone, NaNO2 in trifluoroacetic acid, nitronium salts such as NO2BF4 and an organic solvent selected from the group consisting of CH2Cl2, CHCl3, CCl4, perfluorohexane, perfluoroheptane. The invention refers also to solutions containing: a compound of general formula (I) and a solvent selected from the group consisting of CH2Cl2, CHCl3, CCl4, perfluorohexane, perfluoroheptane, characterized in that the compound of formula (I) is present in a concentration not higher than 20% by weight.
Patent AU-2006247447-B2 (AU)
Title: Method and apparatus for conducting a game of chance
Inventor: YANOWITZ JASON
IPC: A63F13/00
Filed: 2006-05-16
Granted: 2012-07-05
Abstract: A system and method are provided for playing a game of chance. The game of chance may include, for example, a lottery-type game. A result of the game of chance is revealed to a player in another medium. In one example, the result is revealed during multiple game instances of one or more online games. In one example, the online game includes a slot machine type game.
Patent AU-2006256530-B2 (AU)
Title: Scaffold
Inventor: KO FERRIGNO PAUL
IPC: A61P31/10
Filed: 2006-06-08
Granted: 2012-12-20
Abstract: The present invention relates to the use of Stefin A as a scaffold protein for the display of inserted peptides, particularly wherein the Stefin A is a human Stefin A. Several mutations are advantageously made in the wild type stefin A sequence to improve it as a scaffold; preferably the Stefin A comprises a heterologous peptide insertion at the Leu 73 site. Furthermore, preferably the scaffold protein comprises a V48D mutation; preferably the scaffold protein comprises a G4W mutation. Preferably the scaffold comprises Leu73, V48D and G4W mutations. The invention also relates to the scaffold proteins themselves, in particular a stefin A polypeptide having the Leu73, V48D and G4W mutations, such as shown as SEQ ID NO: 1. The invention also relates to a method for identifying binding proteins and to peptide A (RLNKPLPSLPV) and its use in treating yeast infections.