baber/WOPTO huggingface dataset:
Patent AP-9801322-A0 (AP)
Title: Threshing of harvested grain.
Inventor: VISAGIE ANDRIE DIEDERICH
IPC: A01F11/06
Filed: 1997-02-18
Abstract: Ears, pods, or the like ti be threshed are transported axially into an inclined threshing zone (16). Grain is liberated and falls through a sieve (24)forming a bottom of the threshing zone. Most of the lightweight material or chaff is carried to an exit (32)by means of a fan generated airlow stream. Grain and some chaff falling through the sieve (24)are collected in a trough (34)below the seive. A fan generated auxiliary airfloe stream (37)carries most of the remaining chaff to the exit (32). The larger portion of the grain slides down the trough (34)to exit at (36). The balance of the grain with virtually no entrained chaff exits the trough via an auxiliary grain exit (39). Transverse baffles (29 and 27), in tandem, opposing relationship, caude airflow to be circuitous to promote grain in preference to chaff to enter the exit (39). A final cleaning step may be performed in a cleanining apparatus (112).
Patent IL-80742-A0 (IL)
Title: Method of protecting methionine in a polypeptide chain from irreversible oxidation
IPC: C07K7/00
Filed: 1986-11-24
Abstract: Methionine (I) present in a polypeptide chain is protected from irreversible oxidn. by reacting it with an alkyl halogenide of formula X-CH2-R (II) to obtain the sulphonium salt of formula (III). (III) is subsequently deprotected by reaction with a thiol of formula HS-(M)n-Y (IV). In (II), X = I or Br; R = H, COOH or CONH2; In (IV) M = CH2 or CHOH; Y = OH or SH ; and n = 1-4. Pref. the alkylation is carried out in the presence of excess (II) using e.g. iodo- or bromo- acetamide or methyl iodide or bromide. Deprotection is performed using eg. 2-mercaptoethanol or 1,4-dithiothreitol.
Patent IL-95831-A0 (IL)
Title: Process for making 3-aroyl-2-oxindole-1-carboxamides
IPC: B01J27/053
Filed: 1990-09-27
Abstract: Process for making antiinflammatory 3-aroyl-2-oxindole-1-carboxamides by reductive debromination or deiodination of 3-(bromo- or iodoaroyl)-2-oxindole-1-carboxamides.
Patent IL-96070-A0 (IL)
Title: Liposome micro reservoir composition
IPC: A61K49/00
Filed: 1990-10-21
Abstract: A liposome composition for localizing an anti-tumor compound to a solid tumor via the bloodstream. The liposomes, which contain the agent in entrapped form, are composed of vesicle-forming lipids and between 1-20 mole percent of a vesicle-forming lipid derivatized with hydrophilic biocompatible polymer, and have sizes in a selected size range between 0.07 and 0.12 microns. After intravenous administration, the liposomes are taken up by the tumor within 24-48 hours, for site-specific release of entrapped compound into the tumor. In one composition for use in treating a solid tumor, the compound is an anthracycline antibiotic drug which is entrapped in the liposomes at a concentration of greater than about 50  mu g agent/ mu mole liposome lipid. The method results in regression of solid colon and breast carcinomas which are refractory to anthracycline antibiotic drugs administered in free form or entrapped in conventional liposomes.
Patent AU-PO508497-A0 (AU)
Title: Improvements in poppet valve actuation
IPC: F01L13/00
Filed: 1997-02-13
Abstract: An apparatus for adjusting the motion characteristics of a valve of an engine, comprising an adjustment means to vary the valve opening and closing angle, or the valve lift including a guide element movable from a first position to a second position, and having a path adapted to receive a guide member of a valve actuation means, the guide member received in the guide path having a trajectory, when the adjustment means is in the first position, different of the trajectory of the guide member when the adjustment means is in the second position.
Patent IL-105152-A0 (IL)
Title: Stable conditioning shampoo containing cationic and suspended water-insoluble conditioning agents
IPC: A61K8/891
Filed: 1993-03-24
Abstract: A conditioning shampoo containing water; an anionic surfactant; a water-soluble cationic, preferably polymeric, conditioning compound; a liquid, water-insoluble conditioning compound having a viscosity at 25 DEG C less than about 20 centipoises, a specific gravity less than 1.0, preferably less than about 0.95, and a refractive index of at least about 1.4 at 25 DEG C; and a suspending agent for the water-insoluble conditioning compound; in a suitable carrier, has extended product stability, excellent cleansing properties and provides unexpected overall conditioning to human hair, particularly superior wet and dry combing properties. The composition effectively deposits the water-insoluble conditioning agent onto the hair to substantially improve dry comb and dry lubrication properties that the water-soluble cationic conditioning agent does not substantially improve.
Patent IL-108537-A0 (IL)
Title: Method and machine for producing rolls of web material and tearing the web upon completion of the winding of each roll
IPC: B65H18/16
Filed: 1994-02-03
Abstract: A surface rewinding machine for the formation of logs of web material has a winding roller (1) onto which the web material (N) is fed. The winding roller has a surface portion (1A), extending substantially parallel to the roller axis and having a coefficient of friction lower than that of the adjoining surface. The web is pressed at preset moments by a pusher (3) against that portion of the surface of the winding roller having low coefficient of friction so as to tear the web material. <IMAGE>   <IMAGE>
Patent IL-110099-A0 (IL)
Title: Anti-bacterial, insoluble, metal-chelating polymers
IPC: C08F20/26
Filed: 1994-06-23
Abstract: A soft contact lens which comprises a water-swollen gel of a polymer prepared by polymerizing one or more hydrophilic monomers such as 2-hydroxyethyl methacrylate, one or more cross-linking monomers, and a monomer that contains metal-chelating functionality such as an aminopolycarboxylic acid that contains a polymerizable olefinic group.
Patent IL-116465-A0 (IL)
Title: Pharmaceutical antitumor composition
IPC: A61K31/235
Filed: 1995-12-20
Abstract: Growth or metastasization of malignant tumors can be inhibited by administering to a patient in need thereof sufficient lactose to block crucial lectins on the affected organ so that the tumor cells cannot anchor to other locations in the body. Lactose can be administered alone, or in combination with conjugates of cytotoxic drugs. Preferably, lactose is conjugated to a cytotoxic substance so that the primary tumor is treated concurrently with prevention of metastasis. Additionally, by conjugating a cytotoxic drug to lactose, the cytotoxic drug is maintained in close proximity to the tumor because of the receptors on the tumor which bind the lactose (and therefore the cytotoxic agent bound thereto) to the tumor cells. By using a conjugate of lactose with a cytotoxic agent, one dose is generally sufficient to destroy the receptor sites on the tumor and prevent metastasis of the tumor while treating the tumor.
Patent IL-137248-A0 (IL)
Title: A process for the preparation of 2'-deoxy -2',2' difluoro ribozyl nucleosides and pharmaceutical compositions containing the same
IPC: C07H13/08
Filed: 2000-07-10
Abstract: Anomeric 2,2-difluororibosyl azide and amine intermediates which are useful in the preparation of 2'-deoxynucleosides, and processes thereto.
Patent IL-146778-A0 (IL)
Title: Micropigment mixture
IPC: A61P17/16
Filed: 2000-06-08
Abstract: The use of mixtures of micronised organic UV filters in protecting human and animal skin and hair against the damaging effect of UV readiation and the use thereof in cosmetic and pharmaceutical formulations are described.The micronised mixtures used according to the invention cover a broad UV spectrum and therefore exhibit excellent sunscreen properties.
Patent IL-151997-A0 (IL)
Title: High temperature/high pressure colour change of diamond
IPC: B01J3/06
Filed: 2001-04-02
Abstract: A method is provided for changing the colour of a brown type IIa diamond from brown to pink. The method involves subjecting the diamond to selected conditions of elevated temperature and elevated pressure to produce the colour change.
Patent IL-161226-A0 (IL)
Title: Winding tube
IPC: B65H75/10
Filed: 2002-09-25
Abstract: The coiling sleeve (1) for coiling material sheets comprises an adaptor (4) which is nondestructively detachable from the sleeve body (2).
Patent IL-181076-A0 (IL)
Title: Methods and apparatus for identifying and diagnosing live eggs using heart rate and embryo motion
Filed: 2007-01-30
Abstract: Identifying live eggs includes: a) illuminating eggs with light; b) receiving light passing through each egg at a light detector; c) generating an output signal that corresponds to light received at a light detector for each respective egg; d) analyzing the output signals to identify an indication of an external disturbance; e) analyzing the output signal for each egg to identify the existence of an embryo heart rate and/or embryo movement; and f) designating an egg as a live egg in response to identifying embryo heart rate and/or embryo movement. Steps a) through d) are repeated if output signals from a predetermined number of eggs contain an indication of an external disturbance to the eggs. Steps a) through f) are repeated if the number of eggs designated as live exceeds an expected number, or if embryo movement occurs at about the same time in a predetermined number of eggs.
Patent IL-191069-A0 (IL)
Title: Aminoacid derivatives containing a disulfanyl group in the form of mixed disulfanyl and aminopeptidase n inhibitors
Filed: 2008-04-27
Abstract: Amino acid derivatives (I) are new. Amino acid derivatives of formula H 2NCH(R 1)CH 2SSCH 2CH(R 2)C(O)NHCH(R 3)C(O)OR 4 (I) and their mineral or organic acid addition salts are new. R 1 = 1-6C optionally unsaturated hydrocarbyl (optionally substituted by OR, SR, S(O)R, phenyl or benzyl), phenyl or benzyl (both optionally substituted by OR, SR or S(O)R or 1-5 halo, preferably F) or T; R = H, 1-4C hydrocarbyl, phenyl or benzyl; T = methylene substituted by aromatic or saturated 5-6 membered heterocycle containing heteroatoms such as N or S, preferably as N-oxide or S-oxide; R 2 = phenyl or benzyl (both optionally substituted by OR, SR, S(O)R, amino (optionally mono- or disubsituted by 1-6C aliphatic group), 5-6 membered aromatic ring or 1-5 halogen (preferably F)), 5-6 membered heteroaromatic ring contaning one O, S or N or T; R 3 = H, OH, OR, 1-6C saturated alkyl (optionally substituted by OR or SR), phenyl or benzyl (both optionally substituted by 1-5 halogen (particularly F), OR or SR); and OR 4 = hydrophilic ester where the hydrophilicity of the ester provides an octanol-water division coefficient (log K ow)  1.7 to (I). ACTIVITY : Antidepressant; Antiinflammatory; Analgesic. MECHANISM OF ACTION : Neprilysine inhibitor; N-Amino peptidase inhibitor.
Patent IL-198383-A0 (IL)
Title: An apparatus for percussive harmonic musical synthesis utilizing midi technology (aphams)
Filed: 2009-04-26
Abstract: An Apparatus for Percussive Harmonic Musical Synthesis (APHAMS) which facilitates state-of-the-art musical expression, through generation of melodic sound, bearing well defined tone and note pitch, by the striking of uniquely configured multiple note activitation trigger mechanism surfaces, termed muzi-pads, with an appropriately sized mallet, stick, or other such similar playing implement, for the generation of a desired note, by a given MIDI device and which provides an enhanced emulation of the traditional tenor steelpan, in its interface with the player.
Patent RO-126074-A0 (RO)
Title: Installation for the optimization of power factor in transformer stations of 20/6 kv
Inventor: SIMEREA VASILE
IPC: H02B7/00
Filed: 2010-10-14
Abstract: The invention relates to an installation for the optimization of the power factor in transformer stations of 20/6 kV. According to the invention, the installation comprises three compartments (1, 2 and 3): a low voltage compartment (1) wherein a programmable automaton (a) and the secondary control and signaling circuits for the automatic/local working modes are intended to be mounted; the compartment (2) containing the system of bars of 6 kV, fuses of 100 A/7.2 kV with some sensors (b), some vacuum commutation contactors (c) and some current limiting coils (d); and the compartment (3) wherein some capacitors (e) are mounted, depending on the value and number of stages required, the so obtained energy compensation installation having the role of achieving an accurate control of the power factor in relation to an indexed one, by the commutation of the stages of capacitors (e) depending on the compensation power required as a consequence of the variation of the reactive power.
Patent AP-2003002777-A0 (AP)
Title: Subsea pipeline power transmission
Inventor: HUDSON STEVEN MARTIN
IPC: C23F13/08
Filed: 2001-12-20
Abstract: A subsea pipeline power transmission system comprasing a pipeline (1), an electoral power supply (4) connected to the pipeline at a first location, and connection means provided on the pipeline at a second location for connection of a load (5) to the pipeline. Once connected the load 5 can receive electoral power from the power supply (4) via the pipeline (1). The pipeline has a plurality of cathodic protection anodes (2), each of which is electrically connected via respective impedance means to the pipeline.
Patent LU-87196-A1 (LU)
IPC: A61K8/00
Filed: 1988-04-12
Abstract: Process for the preservation of the dyeing ability of 5,6-dihydroxyindole or its derivatives, corresponding to the formula (I): <IMAGE> in which R1, R2, R3,and R4, which are identical or different, denote hydrogen or C1-C4 lower alkyl, R1, R2 and R3 denoting hydrogen when R4 denotes alkyl, in an aqueous medium, wherein the pH of the aqueous medium is adjusted to a value pHC of between 5 and 10 using a pH regulating agent containing two components (A) and (B), the component (A) being chosen from pH regulating agents having a dissociation constant KCA in aqueous solution at 25 DEG C such that pkCA is:  0 < pkCA-pHC </= 2.5 and the component (B) being chosen from pH regulating agents having a dissociation constant KCB in aqueous solution at 25 DEG C such that pkCB is: 2 < pkCB < pHC.i
Patent LU-87915-A1 (LU)
Title: Drilling machine and associated pinch bars for opening tap-holes in shaft furnaces - includes using machine fitted to carriage pinch bar on carriage to hydraulically advance drilling rod threaded through pinch bar etc.
Inventor: MAILLIET PIERRE
IPC: C21B7/12
Filed: 1991-04-03
Abstract: In the method a drilling rod (22) is introduced into the taphole (24) of a shaft furnace using a drilling machine fitted with a carriage (26) acting against the wall of the furnace (20). A pinch bar (46) mounted on this carriage (26) is able to be displaced longitudinally on the carriage (26) under the action of a hydraulic jack (42) mounted at the front of the carriage (26). After the drilling rod (22) is threaded through the pinch bar (46) the hydrualic jack (42) is operated to advance the drilling rod (22) over a length corresp. to the track of the hydraulic jack (42) whilst it is held by the pinch bar (46). The pinch bar (46) is then opened and is brought back to its start position so that the operation can be repeated until the drilling rod (22) is driven the desired depth into the taphole (24). The drilling rod can then be extd. in a similar manner. The drilling machine is also claimed along with a number of different types of bi-directional pinch bars that can be used to grip the drilling rod.
Patent MA-27502-A1 (MA)
Inventor: ADJE NATHALIE
IPC: A61K31/4164
Filed: 2005-06-22
Abstract: A method and composition for the prevention, amelioration or control of external parasites on animals and humans utilizing a compound of formula I. <CHEM> wherein  R is halogen, OR7, SOmR8, NO2, CN, C1-C6haloalkyl or an optionally substituted C1-C6alkyl group; n is 0 or an integer of 1, 2 or 3; m is 0 or an integer of 1 or 2; R1  is H, halogen, NO2, NR9R10, NR11COR12, NCHNR9R10 or NCHOR13; R2, R3, R4, R5 and R6   are each independently H, halogen or a C1-C4alkyl, aryl or heteroaryl group each optionally substituted; R7  is H or a C1-C6alkyl, C2-C6alkenyl, C2-C6alkynyl, aryl or heteroaryl group each optionally substituted; R8  is a C1-C6alkyl, C2-C6alkenyl, C2-C6alkynyl, aryl or heteroaryl group, each optionally substituted; R9 and R10   are each independently H, C1-C4haloalkyl or a C1-C6alkyl, C2-C6alkenyl, C2-C6alkynyl, aryl or heteroaryl group each optionally substituted or R9 and R10 may be taken together with the atom to which they are attached to form a 5- to 7-membered ring optionally containing 1 or 2 additional heteroatoms selected from O, N or S; R11   is H, COR12 or an optionally substituted C1-C4alkyl group; R12   is a C1-C6alkyl, C2-C6alkenyl, C2-C6alkynyl, aryl or heteroaryl group each optionally substituted; and R13   is H or a C1-C6alkyl, aryl or heteroaryl group each optionally substituted;  or a stereoisomer or tautomer thereof.
Patent MA-38664-A1 (MA)
Title: Portefeuille connecté et procédé de signalement de sa position
Inventor: OUSTOU MUSTAPHA
IPC: A45C13/18
Filed: 2015-12-10
Abstract: Un objet connecté sous forme de portefeuille intelligent. Son objectif consiste à ne jamais perdre les documents ou l'argent qu'il contient. Il dispose également d'une mémoire interne pour le stockage de documents électroniques et d'affichage de photos ou vidéo. Son fonctionnement est simple, il sera connecté à un téléphone portable par connectivité gsm. En cas de perte, une application mobile permettra de savoir son emplacement. Un lecteur d'empreintes digitales renforce la sécurité des documents et biens qui sont à l'intérieur du portefeuille.
Patent MA-54773-A1 (MA)
Title: Nouvelles familles de composés à base de sulfonamides pour le traitement du cancer du sein triple négatif
Inventor: ZYAD ABDELMAJID
IPC: C07C311/46
Filed: 2021-10-29
Abstract: La présente invention concerne de nouveaux dérivés des sulfonamides de formules (i) ou (ii) leurs procédés de synthèse et leur utilisation en thérapeutique pour le traitement de pathologies proliférative notamment les cancers. Plus particulièrement, la présente invention porte sur la synthèse de nouvelles molécules présentant des propriétés biologiques en particulier pour le traitement des cancers et plus spécifiquement le cancer du sien triple négatif. Dans la présente invention de nouveaux composés de formules (i) ou (ii) ont été synthétisés ensuite leurs activités cytotoxiques in vitro et in vivo ont été évaluées sur cancer du sein triple négatif mda-mb-468.
Patent UY-28826-A1 (UY)
Title: Procedimiento de produccion, en forma continua, de un producto en polvo a partir de un producto en estado liquido.
Inventor: JEAN-MARIE BOUVIER
IPC: F26B1/00
Filed: 2005-03-29
Abstract: La invención se refiere a un procedimiento de producción en forma continua de un producto en polvo, especialmente de leche en polvo, a partir del producto en estado líquido, en el cual se efectúa, al menos, una etapa de evaporación al vacío (E1) de la mezcla en estado líquido, para obtener el producto en estado viscoso, y se realiza, al menos, una etapa de secado (E2, E3) del producto en estado viscoso para obtener el producto en forna sólida. De acuerdo con un aspecto de la invención, dicha etapa de secado (E2, E3) comprende, al menos, una primera etapa de tratamiento termomecánico (E2) mediante una máquina de tratamiento termomecánico en la cual se inyecta simultáneamente el producto en estado viscoso que proviene de la etapa de evaporación al vacío y una proporción determinada de producto en polvo de la mima familia del producto en estado líquido.
Patent DZ-3149-A1 (DZ)
Inventor: ZAKARIAN NOEL
IPC: A61K9/00
Filed: 2000-03-30
Granted: 2001-08-16
Abstract: Dispersible tablets containing 20 - 60 % by weight of a macrolid (I) and 1 - 25 % of a disintegration agent (II) together with a sweetening agent. (I) is present as the base and is one or more of the following: pristinamycin, azithromycin, roxithromycin, clarithromycin, and spiramycin. The disintegrating agent (II) is preferably 1 - 16 % polyvinyl pyrrolidone, 1 - 15 % sodium croscarmellose or a 1:1 - 4:1 mixture of these two. The sweetening agent is preferably aspartame, sodium saccharin, potassium acesulfame, ammonium glycerinate, or their mixtures. The tablets may further contain an active nitro-imidazole, especially metronidazole, tinidazole or ornidazole, as well as conventional diluents, surfactants, lubricants, flow agents and flavors. ACTIVITY : Antibiotic. MECHANISM OF ACTION : None given.
Patent ES-166278-A1 (ES)
Title: UN TUBO DE DESCARGA CON ESPEJO ELECTRoNICO Y ELECTRODOS DEFLECTORES
Filed: 1944-05-27
Abstract: Un tubo de descarga en el cual sobre su trayectoria desde el cátodo hacia uno más electrodos colectores una corriente electrónica concentrada es dirigida sobre un espejo electrónico y bajo el efecto del campo de este espejo se desvía de su dirección inicial y sufre una desviación bajo la influencia de uno o más electrodos caracterizado porque los electrodos de desviación están unidos directamente al electrodo espejo pudiendo presentar además este tubo las particularidades siguientes tomadas por separado o según las diversas combinaciones posibles: a)el espejo electrónico ejerce un efecto convergente sobre el haz electrónico b) el electrodo colector está constituido por una pantalla fluorescente c)el electrodo colector está constituido por uno o más ánodos.
Patent ES-172076-A1 (ES)
Title: Un procedimiento de producir una pentosa
IPC: C13K13/00
Filed: 1946-01-08
Abstract: Procedimiento de producir una pentosa caracterizado por calentar una N-pentosida amínica aromática primaria en solución en presencia de agua hasta que la hidrolisis está virtualmente completa separar la amina aromática primaria libertada y aislar la pentosa de al solución acuosa.
Patent ES-187586-A1 (ES)
Title: UN PROCEDIMIENTO ECONoMICO-COMERCIAL CON FINALIDAD DE PROPAGANDA Y COMERCIO
Filed: 1949-03-25
Abstract: Procedimiento económico-comercial con finalidad de propaganda y comercio en el que se reivindica el boleto y hoja encasillada representados en el dibujo adjunto cuyo desarrollo y distribución es objeto del cuerpo de esta memoria que igualmente queda reivindicado por constituir ambos una misma cosa con carácter de imposible separación. Los referidos boletos y hoja encaminada que obrarán en poder de la entidad que adopte el procedimiento y que serán ofrecidos gratuitamente servirán de garantía en los términos expuestos en el cuerpo de la memoria.
Patent ES-189235-A1 (ES)
Title: UN DISPOSITIVO DE PRINCIPIO DE PRODUCCIoN DE CORRIENTES OSCILANTES POLIFáSICAS DE ALTA FRECUENCIA
Filed: 1949-07-27
Abstract: Dispositivo de principio de producción de corrientes oscilantes polifásicas de muy alta frecuencia caracterizado por el hecho de que: prevé el empleo de tubos electrónicos triodos acoplados circularmente comprendiendo el conjunto tantos tubos cuantas son las fases que se desean; un circuito oscilante montado en serie con la placa de cada tubo estando cada placa acoplada a la grilla del circuito siguiente a través de un condensador.
Patent ES-193006-A1 (ES)
Title: Un mecanismo de bloqueo escalonado y conjunto de un sistema de cuatro palancas articuladas a dos
Filed: 1950-05-16
Abstract: Un mecanismo de bloqueo escalonado y conjunto de un sistema de cuatro palancas articuladas dos a dos caracterizado por el hecho de comprender un juego de dos palancas principales articuladas entre sí y cada una de ellas tiene a su vez otra palanca articulada con posibilidad de giro libre en estas articulaciones presentando las dos palancas principales respectivos pestillos oscilantes a lados opuestos cuyos pestillos se relacionan entre sí en el plegado del conjunto por bloqueo de uno sobre el otro llevando cada pestillo medios para acoplar a las palancas secundarias y éstas a su vez medios para relacionarse con dichos pestillos existiendo en una de estas palancas secundarias un fiador excéntrico relacionado con medios de acoplamiento con la palanca secundaria del otro grupo.