baber/WOPTO huggingface dataset:
Patent AR-015766-A1 (AR)
Title: Procedimiento para preparar compuestos de 1-h-indol-3-glioxamidas-4-sustituidas, sales farmaceuticamente aceptables de los mismos y derivados prodroga dedichos compuestos.
IPC: C07D209/22
Filed: 1999-04-15
Abstract: Se trata de un procedimiento para preparar compuestos de 1H-indol-3-glioxamidas utiles para inhibir SPLA2 de formula I donde R1 es seleccionado entre el grupo formado por alquilo C7-20, en donde R10 se selecciona entre halo, alquilo C1-10, alcoxi C1-10, -S-alquilo C1-10, y haloalquilo C1-10, y t es un entero de0 a 5 ambos inclusive; R2 se selecciona entre el hidrogeno, halo, alquilo C1-3, cicloalquilo C3-4, cicloalquenilo C3-4, -O(alquilo C1-2), -S(alquilo C1-2),arilo, ariloxi y Het. R4 se selecciona entre -CO2H, -SO2H, y -P(O)(OH)2 o sal o derivados de prodroga de los mismos; R5 se selecciona entre hidrogeno,-alquilo C1-6, alcoxi C1-6, halo (alcoxi C1-6), halo(alquilo C1-6), bromo, cloro, fluoro, yodo y arilo; caracterizado porque comprende las etapas de (a)halogenar un compuesto de formula X donde R8 es alquilo C1-6, arilo o Het, con SO2Cl2 para formar un compuesto de formula IX; b) hidrolizar y descarboxilar uncompuesto de la formula IX para formar compuestos de formula VIII; c)alquilar los compuestos de formula VII con compuestos de formula VIII; para formar loscompuestos de formula VI; d)aminar y deshidratar los compuestos de formula VI con aminas de formula R1NH2 en presencia de solventes que forman azeotropos conel agua para formar compuestos de formula V; e)oxidar los compuestos de formula V por calentamiento con una base y un compuesto de formula RSOX, donde R esalquilo C1-6, arilo, o arilo sustituido y X es alcoxi C1-6, halo o -OCO2 alquilo C1-6 para formar compuestos de formula IV, f) alquilar los compuestos deformula IV con agentes de alquilacion de formula XCH2R4a donde X es un grupo saliente y R4a es -CO2R4a, -SO3R4b, -P(O)(OR4b)2, o -P(O)(OR4b)H, donde R4b es ungrupo ácido protector, para formar compuestos de formula III; g)hacer reaccionar los compuestos de formula III con cloruro de oxalilo y amoníaco para formarlos compuestos de formula II; h) opcionalmente hidrolizar los compuestos de formula II para formar los compuestos de la formula I, e i)opcionalmente salificarde los compuestos de formula I obtenidos. Dichos compuestos son utilizados para inhibir la liberacion mediada por sPLA2 de ácidos grasos en estados tales
Patent AR-021076-A1 (AR)
Title: Base cablecanal con agujeros de fijacion preformados, y su procedimiento de obtencion
IPC: H02G3/10
Filed: 1999-11-04
Abstract: Se trata de una base cablecanal del tipo en el cual fondo (11) presenta al menos dos agujeros de fijacion (17) separados longitudinalmente uno del otro.Cada uno de esos agujeros de fijacion (17) está obturado por un tapon (18) susceptible de serelim inado de este. Aplicacion, en especial, a los cablecanalespara aparatos eléctricos.
Patent AR-024521-A1 (AR)
Title: Derivados de hidrazina, su empleo, un procedimiento para prepararlos, medicamentos que los contienen, un procedimiento para la produccion de unmedicamento, y compuestos intermedios
IPC: A61K31/18
Filed: 1999-11-25
Abstract: Derivados de hidrazina de la formula (1) en donde: R1 representa alquilo inferior, alquenilo inferior, cicloalquilo inferior, cicloalquilo inferior-alquiloinferior, arilo o aril-alquilo inferior; R2 representa heterociclilo o NR5R6; R3 representa hidrogeno, alquilo inferior, halo-alquilo inferior, ciano-alquiloinferior, hidroxi-alquilo inferior, amino-alquilo inferior, alcoxilo inferior-alquilo inferior, alcoxicarbonilo inferior-alquilo inferior, cicloalquiloinferior-alquilo inferior, aril-alquilo inferior, heterociclililo-alquilo inferior, heterociclilcarbonil-alquilo inferior, alquenilo inferior, alquiniloinferior, cicloalquilo inferior, arilo, heteroarilo o aril-alquilo inferior; R4 representa alquilo inferior, alquenilo inferior, cicloalquilo inferior,cicloalquilo inferior-alquilo inferior o una agrupacion de la formula -Z-arilo, -Z-heterociclilo o -(CH2)n-CH=CR7R8; R5 y R6 representan cada uno,independientemente, hidrogeno o alquilo inferior; R7 y R8 representan cada uno, independientemente, hidrogeno o alquilo inferior o R7 y R8 juntos representanalquileno inferior en donde un grupo CH2 está opcionalmente sustituido por un heteroátomo; X y Z representan cada uno un grupo espaciador; y n significa 0, 1 o2; y sus sales farmacéuticamente aceptables, inhiben la liberacion del factor alfa de necrosis tumorales (TNF-alfa) de células. Pueden utilizarse comomedicamentos, especialmente en el tratamiento de enfermedades inflamatorias y autoinmunes, osteoartritis, enfermedades respiratorias, tumores, caquexia,enfermedades cardiovasculares, fiebre, hemorragia y sepsis. Un procedimiento para preparar los derivados de formula (1), un procedimiento para preparar unmedicamento, y compuestos intermediarios.
Patent WO-2007082328-A1 (WO)
Inventor: KARGL HUBERT
IPC: E21C35/24
Filed: 2007-01-18
Abstract: L'invention concerne un procédé de régulation de l'entraînement d'une machine de creusement ou d'extraction destinée à haver un matériau d'abattage, en fonction de grandeurs de réglage telles que la vitesse de déplacement du bras, la position des outils de havage et/ou la puissance consommée par les moteurs d'entraînement ou la pression dans des vérins hydrauliques. Selon ledit procédé, une valeur minimale et une valeur maximale de consigne de la vitesse de déplacement du bras sont déterminées et au moins deux facteurs dont la valeur est comprise entre 0 et 1 sont calculés pour les grandeurs de réglage en fonction de valeurs de mesure. Les valeurs de mesure comprennent au moins des données de position des outils de havage par rapport à des données de consigne qui correspondent à un profil de consigne, des données de mesure de la charge des moteurs et des données de mesure de la vitesse de déplacement du bras, et la vitesse de déplacement du bras est régulée en fonction du produit de la vitesse de consigne et des facteurs respectivement calculés.
Patent WO-2018094437-A1 (WO)
Title: Élément de commande pour une machine à commande électrique
Inventor: FISCHER HARALD
IPC: G06F3/0362
Filed: 2017-11-22
Abstract: L'invention concerne un élément de commande (4) pour une machine à commande électrique (2), lequel élément comprend un corps (7) et une molette (10) pour entrer une instruction dans une commande (3) de la machine (2), cette molette (10) étant disposée sur le corps (7) de l'élément de commande de manière à pouvoir tourner autour d'un axe de rotation (12). La molette (10) est entourée par une surface latérale (11) qui présente une valeur moyenne de diamètre (13) locale prédéterminée dans la direction perpendiculaire à l'axe de rotation (12) et au niveau de laquelle la molette (10) peut être saisie et tournée par un opérateur (5) de la machine. La surface latérale (11) de la molette (10) présente au moins deux parties d'actionnement (14, 15) pourvues de structures de surface différentes, une zone de détection (18, 19) d'un élément de détection (21, 22) étant associée à au moins une des parties d'actionnement (14, 15) et différentes fonctions de machine étant associées à au moins une des parties d'actionnement (14, 15) pour l'entrée d'au moins une instruction dans la commande (3). Les parties d'actionnement (14, 15) sont disposées sur la surface latérale (11) de la molette (10) de telle sorte qu'elles peuvent être saisies par l'opérateur (5) de la machine à l'aide d'une main (6) et/ou des doigts d'une main.
Patent WO-2018102843-A1 (WO)
Title: Procédé de revêtement d'un composant
Inventor: GÄRTNER WALTER
IPC: C23C14/54
Filed: 2017-12-05
Abstract: L'invention concerne un procédé de revêtement d'un composant (2), ledit composant (2) étant disposé sur un support de substrat (1) et étant revêtu sur le support substrat (1) dans une plage de températures prédéfinie. Pour maintenir la température dans cette plage de températures, on utilise un support de substrat (1) qui est pourvu d'un matériau à changement de phase (8) et/ou d'un matériau accumulateur thermochimique. L'invention concerne en outre un support de substrat correspondant.
Patent AU-2002242945-A1 (AU)
Title: Process for the preparation of dimethylcumenes
Inventor: PATRA CHITTA RANJAN
IPC: C07C2/86
Filed: 2002-03-21
Abstract: The present invention relates to a process for the preparation of dimethylcumenes comprising alkylating a substrate comprising of one or more xylene isomers with an alkylating agent in the pesence of a solid acid zeolite catalyst selected from ultrastable zeolite Y (Si/Al=5 to 50) and Beta (Si/Al=10-120), and separating the products formed in vapour phase.
Patent AU-2002253523-A1 (AU)
Title: A vocal connection system between humans and animals
Inventor: PERLO PIETRO GUISEPPE
IPC: G10L15/00
Filed: 2002-03-22
Abstract: A vocal connection system comprises a matrix of sensors ( 2 ) adapted to send signal indicative of a status of the animal, in terms of stimuli, feelings, events, actions or behaviours, of the animal, to a microprocessor ( 3 ). The microprocessor ( 3 ) selects depending upon the signals ( 4 ) which are received, a vocal message recorded in memory means ( 5 ) associated to the microprocessor ( 3 ) and activates a loudspeaker ( 6 ) forming part of the system for emitting the vocal message. The system further comprises vocal recognition means ( 8 ) which activatge stimuli generators ( 11 ) as a function of the contents of a vocal message ( 9 ) emitted by the human user ( 7 ).
Patent AU-2002332897-A1 (AU)
Title: Nucleic acid sequencing by raman monitoring of uptake of precursors during molecular replication
Inventor: NEUBAUER GABI
IPC: C12Q1/68
Filed: 2002-09-05
Abstract: The methods, compositions and apparatus disclosed herein are of use for nucleic acid sequence determination. The methods involve isolation of one or more nucleic acid template molecules and polymerization of a nascent complementary strand of nucleic acid, using a DNA or RNA polymerase or similar synthetic reagent. As the nascent strand is extended one nucleotide at a time, the disappearance of nucleotide precursors from solution is monitored by Raman spectroscopy or FRET. The nucleic acid sequence of the nascent strand, and the complementary sequence of the template strand, may be determined by tracking the order of incorporation of nucleotide precursors during the polymerization reaction. Certain embodiments concern apparatus comprising a reaction chamber and detection unit, of use in practicing the claimed methods. The methods, compositions and apparatus are of use in sequencing very long nucleic acid templates in a single sequencing reaction.
Patent AU-2002346578-A1 (AU)
Title: Purification of onium hydroxides by electrodialysis
Inventor: REITER ROBERT J
IPC: C07C209/68
Filed: 2002-11-27
Abstract: This invention relates to a process for improving the purity of an aqueous onium hydroxide solution. In particular, the invention relates to a process for improving the purity of aqueous onium hydroxide solutions containing undesirable amounts of anions. The invention also relates to the improved high purity onium hydroxide solutions obtained by the above method.
Patent AU-2003207998-A1 (AU)
Title: Catheter with flexible cooled electrode
Inventor: VENTURELLI ANDREA
IPC: A61B17/00
Filed: 2003-01-27
Abstract: A catheter for the treatment of tumors and other affections using hyperthermia induced by radio frequency includes a tubular body with or without an anchoring balloon at its distal end. An active electrode is positioned around the body and connected to a radio frequency generator. At least one thermistor needle measures the temperature around the electrode. The active electrode is flexible and connectable to a supply source of a fluid for cooling the electrode. It includes a helical conduit, which can be metal, conductive ceramic or graphite.
Patent AU-2003212328-A1 (AU)
Title: Ferrocenyl ligands and the use thereof in catalysis
Inventor: ALMENA JUAN
IPC: C07C241/02
Filed: 2003-03-10
Abstract: The invention relates to bidentate organophosphorous ferrocenyl ligands containing ligands of formula (I), to their complex compounds and to their utilization in catalytic processes.
Patent AU-2003241749-A1 (AU)
Title: Polyester composition and packaging material comprising the same
Inventor: NAKAYAMA SEIJI
IPC: C08L67/02
Filed: 2003-06-02
Abstract: The present invention relates to a polyester composition excellent in transparency, thermal stability, and flavor retention or excellent in transparency, thermal stability, flavor retention and gas barrier properties, which is obtained by blending a partially aromatic polyamide to a thermoplastic polyester, and also relates to a packaging material comprising the same. The polyester composition of the invention preferably contains an alkali metal atom in an amount of 0.1 to 300 ppm and phosphorus atom in an amount of 5 to 200 ppm. Further, it is preferable that the Color-L value of the molded article obtained by injection molding of the polyester composition of the invention at a molding temperature of 290 DEG C is 80.0 or more and the haze thereof is 20% or less. As the partially aromatic polyamide, an m-xylylene group-containing polyamide is preferable.
Patent AU-2003255911-A1 (AU)
Title: Method of monitoring a data link
Inventor: WALZ JOCHEN
IPC: H04L69/40
Filed: 2003-08-12
Abstract: In a method of monitoring the reliability of a data link for a data transmission between a server ( 2 ) and a client ( 8 ), a control unit ( 14 ) is triggered by a trigger signal in such a manner that in response to the arrival of the trigger signal the control unit ( 14 ) generates first control data for a predetermined running time which commences anew in response to each trigger signal received. The first control data forms a first control representation ( 23 ) on a client display screen ( 11 ), which first control representation optically indicates the existence of a reliable data link ( 4 ) to a user. The control unit ( 14 ) generates, after expiration of the running time, second control data which generates a second control representation ( 23 ') on the client display screen ( 11 ) which optically indicates the absence of a reliable data link to the user. A control unit ( 15 ) periodically transmits a test message to a test unit ( 18 ). The test unit ( 18 ) returns the incoming test message or another test message to the server ( 2 ). The control unit ( 14 ) is triggered again only if the returned test message is in order. The period with which the control unit ( 15 ) repeats the transmission of the test messages is shorter than the running time during which the control unit ( 14 ) generates the first control data.
Patent AU-2003259748-A1 (AU)
Title: System and method for providing fault tolerant ip services
Inventor: SHAFFER SHMUEL
IPC: H04L69/40
Filed: 2003-08-12
Abstract: A system and method for providing fault tolerant IP services includes establishing a first communication session between an originating telephony device and an application server, through a primary call manager. Failure of the primary call manager may be detected. A second communication session between the application server and a destination telephony device may be established via a back-up call manager. The first communication and the second communication session may be coupled at the application server to establish two-way communication between the originating telephony device and the destination telephony device.
Patent AU-2003268431-A1 (AU)
Title: Preparation of m(co)3-complexes by solid phase techniques via metal assisted cleavage from the solid support
Inventor: ALBERTO ROGER
IPC: C07F15/00
Filed: 2003-09-02
Abstract: The present invention relates to a process for generating a water soluble metal complexed agent, comprising contacting a solid phase bound organic conjugate represented by the formula I with [M(H<SUB>2</SUB>O)<SUB>3</SUB>(CO)<SUB>3</SUB>]<SUP>n+</SUP>, under suitable conditions to cause the formation of a coordinate bond between [M(H<SUB>2</SUB>O)<SUB>3</SUB>(CO)<SUB>3</SUB>]<SUP>n+</SUP> and the tertiary amine nitrogen atom of the solid phase bound organic conjugate and thereby the release of the metal complexed agent thus formed from the support. The invention further relates to the conjugate of formula (I) and to a kit for performing the process.
Patent AU-2003269691-A1 (AU)
Title: Integrated photosensitive structures and passivation method
Inventor: BACH KONRAD
IPC: H01L31/0216
Filed: 2003-08-29
Abstract: The invention relates to an integrated circuit according to CMOS/BiCMOS technology and a method for producing the same. At least one integrated, photosensitive component and one electrical shield are provided, a second layer system (2; 3, 4) being applied to a photosensitive area (1) of the circuit (A) to be protected against an (unwanted) electrical coupling, said second layer system comprising a last layer (3) of a first sealing passivation layer system (5) according to the process, and a subsequent, transparent, electroconductive layer (4). Said layers have adjusted individual thicknesses (d3, d4) in order to obtain an optical thickness of the second layer system (2) having maximum transparency with a reduced thickness tolerance influence.
Patent WO-2005045170-A1 (WO)
Title: An adaptable drive mechanism
Inventor: TONKIN MICHAEL
IPC: E05F15/16
Filed: 2004-11-04
Abstract: A roller curtain drive mechanism (150) for a roller door (10). The roller door (10) including a drum wheel (14) mounted on a shaft (12) and a roller curtain (18) arranged to be rolled onto and off the drum wheel (14) when the roller door (10) is raised or lowered. The drive mechanism (150) includes a drive wheel (152) including means for engagement (152a) with the drum wheel (14) and a slot (170) arranged to fit over the shaft (12) so that the drive wheel (152) can be located thereon. The drive mechanism (150) further includes means for driving the drive wheel (152) about the shaft (12) so as to cause rotation of the drum wheel (14). The driving means is arranged to enable continuous drive of the drive wheel (152).
Patent AU-2004201349-A1 (AU)
Title: Extended articulation orthopaedic implant and associated method
Inventor: COON MICHAEL E
IPC: A61B17/16
Filed: 2004-03-30
Abstract: A prosthesis (20) for use in performing joint arthroplasty is provided. The prosthesis (20) is to be fitted to a long bone (3). The prosthesis includes a first body (22) having a first body articulating surface(24) defining a generally circular outer periphery(26) of the first body articulating surface (24). The first body (22) has a support surface (28) opposed to the articulating surface (24). The support surface (28) is adapted to receive the head of the long bone(3). The prosthesis (20) also includes a second body (30) operably associated with the first body (22). The second body (30) has a second body articulating surface (32) extending from a portion of the circular outer periphery (26) of the first body articulating surface (24).
Patent AU-2004203410-A1 (AU)
Title: Pivoting handle assembly for power tool
Inventor: STONES KEVIN
IPC: A01G3/053
Filed: 2004-07-26
Abstract: There is disclosed a power tool comprising a housing (3), a motor provided in the housing and having a rotary output shaft, a reciprocating output shaft adapted to be caused by the motor to execute reciprocating motion to actuate a blade assembly, and a handle assembly (2, 102) comprising a front handle (6, 106) and a rear handle (7, 107) integral with the front handle. The handle assembly (2, 102) is pivotably mounted to the housing of the power tool and is adapted to be fixed in a plurality of orientations relative to the housing. By providing a handle assembly with integrally formed front and rear handles that is pivotable relative to the body of the power tool, this provides the advantage of avoiding the need for a user to hold the tool upside down when using the blade assembly to perform high-up horizontal cutting, instead of holding the tool above the user's head. The present invention also provides the advantage of reducing the extent to which a user must bend down when using the blade assembly to perform low-down horizontal cutting. The power tool may also comprise fixing means adapted to releasably retain the handle assembly (2, 102) in a plurality of orientations relative to the housing (3). <IMAGE>
Patent AU-2004268542-A1 (AU)
Title: Systems and methods for positioning implants relative to bone anchors in surgical approaches to the spine
Inventor: MELKENT ANTHONY J
IPC: A61B17/86
Filed: 2004-08-13
Abstract: Devices, instruments, systems and techniques for guiding an implant to a location adjacent a bone anchor include a guide member with a connecting portion and a guiding portion. The connecting portion is adjacent the bone anchor, and the guiding portion extends proximally from the connecting portion and is adapted guide an implant therealong toward the bone anchor. The guiding portion is flexible to facilitate manipulation and implant placement in the patient's body.
Patent AU-2004307533-A1 (AU)
Title: Arrangement and method for using a mobile telephone in an aircraft
Inventor: MUIRHEAD ANDREW
IPC: H04B7/185
Filed: 2004-10-25
Abstract: The arrangement has a stationary device for sending/receiving IP data to/from a corresponding device on the vehicle and a device for converting IP data into cell phone data and vice versa. The arrangement also has a device onboard the vehicle for sending/receiving IP data to/from a base station and a device for converting cell phone data into IP data and vice versa. The connection between the sending/receiving device and converting device, located onboard the vehicle, takes place over the intranet.
Patent AU-2004319611-A1 (AU)
Title: Coaxial coupling
Inventor: SCHUTZ CHRISTIAAN ARNOLD
IPC: F16L37/36
Filed: 2004-05-13
Abstract: A coaxial coupling comprising a female part and a male part which are couplable to each other is disclosed. The female part and the male part having an inner passage and a concentric outer passage, wherein the inner passage of the female part is fluidly connected to the inner passage of the male part and the outer passage of the female part is fluidly connected to the outer passage of the male part in the coupled state of the coupling, one of the parts further comprising a by-pass valve that guides the fluid flow internally from the inner passage to the outer passage thereof in a non-coupled state of the coupling, the other part comprising an activator for activating the by-pass valve during coupling of the two parts wherein the by-pass valve is adapted to guide the fluid flow from the inner passage of the one part to the inner passage of the other part during coupling of the two parts.
Patent WO-2005090799-A1 (WO)
Title: Reseau d'attaches pouvant etre activees par un signal
Inventor: RUDDUCK DICKORY
IPC: B64C3/26
Filed: 2005-03-16
Abstract: L'invention concerne un système de fixation (40) comportant une pluralité d'attaches (12). Chaque attache (12) peut être verrouillée ou déverrouillée à l'aide d'un signal adapté, tel qu'un signal électrique, magnétique ou infrarouge. Les attaches (12) sont montées sur un support (38) unique.
Patent WO-2007030854-A1 (WO)
Title: Mécanisme d’avance destiné à maintenir une tension de bande constante dans une imprimante à grand format
Inventor: SILVERBROOK KIA
IPC: B41J33/14
Filed: 2005-09-12
Abstract: La présente invention concerne un mécanisme d’avance pour une imprimante à grand format (1), le mécanisme d’avance comprenant : une bobine débitrice (4) ; une bobine réceptrice (5) ; un moteur récepteur (14) relié de façon opérationnelle à la bobine réceptrice ; un système de contrôle récepteur destiné à contrôler le couple du moteur récepteur (27) ; un système de rouleau d’entraînement (107) positionné entre la bobine débitrice et la bobine réceptrice ; un moteur d’entraînement relié de façon opérationnelle au système de rouleau d’entraînement. Dans ledit mécanisme, durant l’utilisation, une bande (24) fournie à partir du système de rouleau d’entraînement à la bobine réceptrice est maintenue sous une tension sensiblement constante en régulant le couple du moteur récepteur à l’aide du système de contrôle récepteur.