Patent EP-1992614-A1 (EP)
IPC: C07D207/36
Filed: 2007-05-16
Abstract: The alkoxy-phenyl-substituted compound is new. 4-(2-Alkoxy-phenyl)-substituted tetramate compounds of formula (I), are new. X : 1-6C alkoxy, 1-6C haloalkoxy, 1-4C alkoxy, 2-4C alkyloxy, 1-4C alkoxy-bis-2-4C alkoxy or substituted 3-6C cycloalkyl-1-3C alkanediyl oxy, which is optionally interrupted by heteroatom; W 1>1-6C alkyl; Y 1>Cl, Br or I; G : alkali metal ion, equivalent of an alkaline earth metal ion, equivalent of aluminum ion, equivalent of transition metal ion or ammonium ion in which 1-4 H is replaced by same or different residues from H, 1-5C alkyl, 1-5C isoalkyl or 3-7C cycloalkyl which is optionally substituted by at least 1 F, Cl, CN, OH or one or more O or S or cyclic secondary or tertiary aliphatic or heteroaliphatic ammonium ion like morpholinium, thiomorpholinium, piperidinium, pyrrolidinium or protonated 1,4-diazabicyclo [2.2.2]octane or 1,5-diazabicyclo[4.3.0]undec-7-ene or heterocyclic ammonium cation, protonated pyridine, 2-methyl pyridine, 3-methyl pyridine, 4-methyl pyridine, 2,4-dimethyl pyridine, 2,5-dimethyl pyridine, 2,6-dimethyl pyridine, 5-ethyl-2-methyl pyridine, pyrrole, imidazole, quinoline, quinoxaline, 1,2-dimethylimidazole, 1,3-dimethyl imidazolium methylsulfate, or sulfonium ion or magnesium halogen cation; m : 1-2; n : 1-2; A : H, if necessary substituted by halogen, 1-12C alkyl, 3-8C alkenyl, 1-10C alkoxy-1-8C alkyl, 1-l0C alkylthio-1-6C alkyl or cyclopropyl; B' : H, 1-12 alkyl or 1-8 alkoxy-1-6C alkyl; and D : H or alkyl, alkenyl, alkynyl, alkoxyalkyl, halogen substituted 1-12C alkyl, 3-8C alkenyl, 3-8C alkynyl, 1-10C alkoxy-2-8C alkyl, halogen, 1-4C alkyl, 1-4C alkoxy or 1-4C haloalkyl, saturated or unsaterated cycloalkyl, in which single or multiple ring members are optionally replaced by heteroatom, heteroaryl alkyl, substituted 3-8C cycloalkyl, provided that: (A) A and B' are bonded together with carbon atom, preferably 3-10C or 5-10C unsaturated cycloalkyl or unsubstituted or substituted with heteroatom; and (B) A and D are bonded together with substituted 3-6C alkanediyl or 3-6C-alkenediyl, where methyl group is replaced through a carbonyl, O or S, where substitutents are halogen, hydroxy, mercapto or halogen substituted 1-10C alkyl, 1-6C alkoxy, 1-6C alkylthio, 3-7C cycloalkyl, phenyl or benzyloxy, or 3-6C alkanediyl, 3-6C alkenediyl or butadienyl. Independent claims are included for: (1) a method for producing an agent, which involves utilizing a compound of general formula (I) and a thinner or surface active substance, preferably cultivated plant compatibility improving compound; and (2) a composition, which comprises compound (I), another compound of formula (XIV) and penetration promoters. D : N or P; R 26>-R 29>independently hydrogen or substituted 1-8C alkyl or single or multiple unsaturated, where substituents are halogen, nitro or cyano; n : 1-4; and R 30>an inorganic or organic anion. [Image] [Image] ACTIVITY : Herbicide; Pesticide. 1 part by weight of an active compound was mixed with 78 parts by weight of acetone or 1.5 parts by weight of dimethylformamide and emulsifier 0.5 parts by weight of alkylaryl polyglycol ether. The concentrate was diluted with water to obtain a desired concentration. The brown planthoppers were dipped into prepared active compound having desired concentration. After the desired period of time, the kill in % was determined. The result was evaluated and 80% of planthoppers were killed at a dose of 100 g/hectare. MECHANISM OF ACTION : None given.