baber/WOPTO huggingface dataset:
Patent BR-112023001351-A2 (BR)
Title: Escetamina-suspensão-tts
Inventor: FLORIAN HAMMES
IPC: A61P29/02
Filed: 2021-07-22
Abstract: ESCETAMINA-SUSPENSÃO-TTS. A presente invenção refere-se a um sistema terapêutico transdérmico, compreendendo uma camada de suporte, que não é permeável ao ingrediente ativo, e pelo menos uma camada matriz em um lado da camada de suporte, em que a camada matriz contém pelo menos um adesivo sensível à pressão e cetamina ou um sal ou solvato farmaceuticamente aceitável da mesma, em que o pelo menos um adesivo sensível à pressão compreende um adesivo de silicone sensível à pressão, bem como seu uso como fármaco, em particular para o tratamento de depressão e dor.
Patent BR-112023016026-A2 (BR)
Title: Variante de enzima maltotriose amilase, enzima maltotriose e método de produção de xarope de glicose com teor reduzido de açúcar
Inventor: GARNER ASHLEY
IPC: C12N9/24
Filed: 2022-02-07
Abstract: variante de enzima maltotriose amilase, enzima maltotriose e método de produção de xarope de glicose com teor reduzido de açúcar. essa revelação provê enzimas maltotriose amilase úteis para a produção em escala comercial de xaropes de glicose com teor reduzido de açúcar (rsgs) a partir de um amido. as enzimas úteis (variantes de amilase ou variantes de enzima) podem ser variantes de uma amilase de bacillus subtilis ou enzimas com pelo menos 90% de identidade de sequência projetada com mutações que melhoram a tolerância térmica e a atividade a uma temperatura acima de 50°c em comparação às enzimas matrizes.
Patent BR-112023016582-A2 (BR)
Title: Sistema e processo de registro global unificado e identificação universal de doadores
Inventor: Fernando Latorre Lopez
IPC: G06Q30/02
Filed: 2022-02-18
Abstract: sistema e processo de registro global unificado e identificação universal de doadores. trata-se de um sistema, processo e produto de computador para o registro global unificado e identificação universal de doadores. o método inclui a criação de um ou mais perfis de doadores, perfis de dados médicos relevantes e um identificador de doador público comum a partir de um registro inicial. o procedimento inclui ainda a identificação do doador por uma central de doação por meio de um código pessoal e intransferível para acesso aos dados, ao identificador público comum de doador e aos perfis armazenados. o procedimento atualiza automaticamente os dados, perfis e histórico de doações dos doadores em um banco de dados acessível por diferentes centros de doação.
Patent BR-112023018133-A2 (BR)
Title: Composição de revestimento, poliéster insaturado, substrato, métodos para produzir um substrato de metal revestido e para produzir corpos de latas revestidos e extremidades de lata, e, uso da composição de revestimento
Inventor: LUNZER FLORIAN
IPC: B65D1/12
Filed: 2022-03-10
Abstract: composição de revestimento, poliéster insaturado, substrato, métodos para produzir um substrato de metal revestido e para produzir corpos de latas revestidos e extremidades de lata, e, uso da composição de revestimento. a presente invenção refere-se a uma composição de revestimento compreendendo uma mistura de poliésteres, a dita mistura compreendendo: - de 0,1 a 99,9% em peso de um ou mais poliésteres saturados (a) e - de 99,9 a 0,1% em peso de um ou mais poliésteres insaturados (b), com base no peso total de poliésteres (a) e (b); os ditos um ou mais (a) e um ou mais (b) tendo um peso molecular médio ponderal (mw) de pelo menos 15.000 g/mol, conforme medido por cromatografia de permeação em gel usando tetra-hidrofurano como solvente e uma temperatura de transição vítrea, conforme medida por calorimetria exploratória diferencial, segundo din en 61006, método a, de pelo menos 60°c. a presente invenção também se refere a um poliéster de alto peso molecular propriamente dito, ao método para produzir um substrato revestido, ao substrato revestido propriamente dito e ao uso da composição de revestimento.
Patent BR-112023018525-A2 (BR)
Title: Técnicas para operação full-duplex em sidelink e downlink em sistemas de comunicações sem fio
Inventor: BALASUBRAMANIAN ANANTHARAMAN
IPC: H04W72/04
Filed: 2021-03-23
Abstract: técnicas para operação full-duplex em sidelink e downlink em sistemas de comunicações sem fio. métodos, sistemas e dispositivos para comunicações sem fio são descritos. geralmente, as técnicas descritas proporcionam um primeiro equipamento do usuário (ue) para estabelecer um link de comunicação com uma estação base e um link de comunicação de sidelink com um segundo ue utilizando diferentes pontos de recepção e de transmissão associados ao primeiro ue. o primeiro ue pode realizar uma medição de interferência entre as comunicações de downlink recebidas no link de comunicação e as comunicações de sidelink transmitidas no link de comunicação de sidelink. o primeiro ue pode determinar se é capaz de executar operações full-duplex no link de comunicação e no link de comunicação de sidelink baseado na medição de interferência e pode transmitir uma indicação da capacidade do primeiro ue para a estação base. em alguns exemplos, o segundo ue pode realizar medições de interferência de sinais de downlink no link de comunicação de sidelink, onde as medições podem informar a determinação de utilizar comunicações full-duplex no primeiro ue.
Patent BR-112023019948-A2 (BR)
Title: Dispositivo médico implantável para a entrega de partículas encapsuladas com ácido nucleico
Inventor: Brian d wilson
IPC: A61K9/48
Filed: 2022-03-29
Abstract: dispositivo médico implantável para a entrega de partículas encapsuladas com ácido nucleico. é fornecido um dispositivo médico implantável. o dispositivo compreende uma camada de liberação de fármaco, em que a camada de liberação de fármaco contém partículas dispersas dentro de uma matriz polimérica. as partículas de lipídio incluem um componente carreador que contém um carreador (por exemplo, peptídeo, proteína, carboidrato, lipídio, polímero, etc.) e encapsula um ácido nucleico, em que a matriz polimérica inclui um copolímero de acetato de vinila de etileno. a razão da temperatura de fusão do copolímero de acetato de vinila de etileno à temperatura de fusão do carreador é cerca de 2 °c/°c ou menos.
Patent BR-112023021251-A2 (BR)
Title: Método para inibir florescimento de cana de açúcar
Inventor: CAIO VITAGLIANO SANTI ROSSI
IPC: A01P21/00
Filed: 2022-04-13
Abstract: método para inibir florescimento de cana de açúcar. trata-se de novo método que compreende tratar cana de açúcar com florpirauxifeno-benzila durante o período de indução de florescimento da cana de açúcar e que aumenta a produção de açúcar e eficiência de extração.
Patent CZ-17893-A3 (CZ)
Title: Process and apparatus for saving electric power of a hydraulic elevator drive
Inventor: NAGEL HEINZ-DIETER
IPC: B66B9/04
Filed: 1993-02-11
Abstract: With this method and arrangement for conserving electric power for driving a hydraulic elevator, it is possible to drive the elevator car in the ascending direction with virtually constant power output at any load. The maximum rated speed in the ascending direction is selected for a load which from experience occurs most frequently. The requisite drive variable is set in accordance with this selection. The lifting speed is correspondingly reduced in the case of higher loads and correspondingly increased in the case of smaller loads. The variable lifting speed is obtained either by an adjusting pump (8) with a variable displacement volume, controlled by a pressure regulator (14), or by a displacement pump (28) with a constant displacement volume which is driven by a frequency-controlled electric motor (31) with continuously variable adaptation of the speed of the electric motor (31) as a function of the effective load present. <IMAGE>
Patent CZ-17994-A3 (CZ)
Title: Flaky tantalum powder and method of using thereof
Inventor: FIFE JAMES A
IPC: B22F9/04
Filed: 1992-07-28
Abstract: An improved flaked tantalum powder and process for making the flaked powder are disclosed. The powder is characterized by having a mean particle size in the range of about 2 to about 55 micrometers and a BET surface area in the range of about 0.5 to about 5.0 m<2>/g. Preferably, the mean particle size and BET surface area are selected so that the flakes have an aspect ratio (D/T) in the range of about 2 to about 50. Agglomerates of the flaked tantalum powder, provide improved flowability, green strength and pressing charactistics compared to conventional flaked tantalum powders. The improved flaked tantalum powder can be made by preparing a flaked tantalum and then reducing the flake size until such mean particle size and BET surface areas are achieved such that the flakes have an aspect ratio (D/T) in the range of about 2 to about 50.
Patent CZ-23094-A3 (CZ)
Title: Process and apparatus for treating packages containing residual materials
Inventor: PAULS MATHIAS
IPC: C08J11/08
Filed: 1994-02-03
Abstract: A method is disclosed for processing residue-containing packages so as to recover valuable materials, in particular pressure containers for dispensing polyurethane foams with propellant gases. For that purpose, extraction with a solvent is carried out essentially in atmosphere of propellant gas and/or solvent vapours.
Patent CZ-70097-A3 (CZ)
Title: Composite water-swelling elastomers and process for preparing thereof
Inventor: SULC JIRI ING
IPC: C08L7/00
Filed: 1997-03-07
Abstract: The present invention relates to composite water swellable elastomers consisting of a hydrophobic elastomeric component and hydrophilic polymeric component in which the hydrophobic as well as the hydrophilic component are forming a continuous or communicating matrix. The hydrophobic elastomeric component is selected from the group consisting of a filled or unfilled, vulcanized or non-vulcanized silicone, natural rubber, synthetic butadiene-styrene rubber, butadiene rubber, isoprene rubber, isobutylene-isoprene rubber, ethylene-propylene rubber, ethylenepropylenediene rubber, chlorobutyl rubber, bromobutyl rubber, chloroprene rubber, butadiene-acrylonitrile rubber, acrylate rubber, urethane rubber, fluorocarbon rubber, chlorosulfonated rubber, polyethylene rubber, chlorinated polyethylene rubber, ethylene vinyl acetate rubber, polysulfide rubber, hydrine rubber. The hydrophilic polymeric component is being formed by a polymer based on the hydrophilic monomers being selected from the group consisting of glycolmonomethacrylates and acrylates, dihydroxyestermonomethacrylates, acrylamide, methacrylamide, N-substituted acrylamide and methacrylamide, N,N-substituted acrylamide and methacrylamide, methacrylic and acrylic acids, N-vinylpyrrolidon and their combinations. The method of preparation of the water swellable elastomers according to the invention consists in that in the inside of the hydrophobic elastomeric component matrix and/or the filler the precipitation or solution polymerization of a hydrophilic monomer or monomer mixture in the presence of one or more solvents, a cross-linking agent and initiator of radical polymerization is performed. The process of precipitation or solution polymerization according to the invention can be repeated one or more times using the same or different monomers, solvents, cross-linking agents and initiators. According to the invention the precipitation or solution polymerization can be performed either only in the swollen surface layer or only in the hydrophobic matrix or only in the hydrophilic filler or in the hydrophobic matrix and the hydrophilic filler.
Patent CZ-90598-A3 (CZ)
Title: Mould for injection moulding of a plurality of press button corpuscles or the like individual shaped parts
Inventor: WANDINGER FRANZ
IPC: H01H13/705
Filed: 1996-09-26
Abstract: The invention concerns a method and device for the final assembly of a computer keyboard in which all the key bodies (5) of the keyboard are injection-moulded in the predetermined keyboard arrangement in a common injection-moulding process. A removal device (2) comprising a plurality of suction heads (7) then sucks up and removes the key bodies, which project out of the ejector part (6) when the injection-moulding die is opened, at the upper side of the key caps. The connection channels, which remain between the individual key bodies in the region of the lower edge of the caps for material flow purposes, are separated. Finally, the key bodies held by the removal device (2) are lowered onto a prepared keyboard housing (4) where they are inserted in the correct positions in the respective associated key guides (11).
Patent SK-17698-A3 (SK)
Title: Sulfonamide substituted compounds, a medicament containing same and their use
Inventor: GERLACH UWE
IPC: A61K31/382
Filed: 1998-02-09
Abstract: Sulphonamide-substituted compounds of formula (I) and their salts are new. X = S, SO, SO2, or CO etc.; R1, R2 = H, CF3, C2F5, C3F7, 1-6C alkyl or phenyl (optionally substituted); or R1+R2 = 2-10C alkylene; R3 = R12-CaH2aÄNR13Üm; R12 = H, 3-8C cycloalkyl, CF3, C2F5, or C3F7; a = 0-10; m = 0 or 1; R13 = H or 1-6C alkyl; or R12+R13 = 4-8C alkylene, where one of the CH2 groups may be replaced by O, S, SO, SO2, CO etc.; R4 = R14-CrH2r, where one of the CH2 groups may be replaced by O, CH=CH, C  IDENTICAL  C, CO, CO-O etc.; r = 1-20; R14 = H, 3-8C cycloalkyl, piperidyl, 1-pyrrolidinyl, N-morpholino, or phenyl (optionally substituted) etc.; or R3+R4 = 3-8C alkylene, one of whose CH2 groups may be replaced by O, CO, S, SO, SO2 etc.; R5+R6 = CR15=CR16-CR17=CR18, CR15=CR16-CR17=N, CR15=CR16-N=CR18, CR15=N-CR17=N, CR15=N-N=CR18, N=CR16-CR17=N or S-CR15=CR16; R15-R18 = H, F, Cl, Br, I, 1-4C alkyl, 3-8C cycloalkyl, CN, CF3 etc.; R7 = H, OH, 1-4C alkoxy, 1-4C acyloxy, Cl, Br, F or 1-4C alkyl; R8 = H or 1-6C alkyl.
Patent SK-22296-A3 (SK)
Title: Substituted benzenesulfonylureas and benzenesulfonylthioureas, method of their manufacture, their use for production of pharmaceutical compositions, and medicaments containing them
Inventor: ENGLERT HEINRICH
IPC: C07C335/42
Filed: 1996-02-19
Abstract: Substituted benzene sulphonylurea and benzenesulphonyl-(thio)urea derivatives of general formula (I), wherein R1, R2, R3, R4, R5, R6, E, X and Y have the meaning stated in the claims. These compounds are effective in cardiovascular system.
Patent SK-26594-A3 (SK)
Title: Safety cannula
Inventor: ATTERMEIER KURT
IPC: A61M5/24
Filed: 1993-06-25
Abstract: A coupling system (10) for transferring fluids from a medicament-containing cartridge to an injection site comprises a fluid flow channel, a blunt cannula (16), defining the distal end of the fluid flow channel (14), a needle cannula (18) defining the proximal end of the fluid flow channel (12), and means for fixedly connecting the needle cannula (18) to the blunt cannula (16).
Patent SK-29198-A3 (SK)
Title: Terminal or jointing clamp for a coated overhead cable and moment screw used therein
Inventor: TURUNEN HARRI
IPC: H01R4/24
Filed: 1998-03-04
Abstract: The invention relates to a terminal or jointing clamp for a coated overhead cable and to a moment screw, the latter serving as a terminal clamping element. The moment screw includes a moment transmission nut (11), provided with a fracture point (12) and engaged with a head (7) of a clamping screw (5) through the intermediary of an insulation layer (9). Such a terminal or jointing clamp is capable of voltage work, while enabling an accurate calibration for the operation of the moment screw. <IMAGE>
Patent CS-243591-A3 (CS)
Title: Substituted pyrroles, process of their preparation, medicaments prepared therefrom and process for preparing thereof
Inventor: DAVIS PETER DAVID CHEM
IPC: C07D487/02
Filed: 1991-08-06
Abstract: Compounds of the formula <CHEM> wherein R<1> and R<3> together form a bond and R<2> represents hydrogen or R<1> and R<2> together form a bond and R<3> represents hydrogen; R<4>, R<5>, R<6> and R<7> each independently represent hydrogen, halogen, alkyl, haloalkyl, alkoxy, nitro, amino, alkanoylamino, aroylamino, alkylthio or alkylsulphonyl; R<8> represents hydrogen, alkyl or aralkyl; X represents -N(R<9>)- or -CHN(R<1><0>,R<1><1>)- in which R<9>, R<1><0> and R<1><1> each represent hydrogen, alkyl, aralkyl or alkanoyl; m stands for 0-2 and n stands for 1-3, with the proviso that the sum of m and n is 1-3; p stands fo 0-4 and q stands for 0-4, with the proviso that the sum of p and q is 2-4 when X represents -N(R<9>)-, that the sum of p and q is 1-5 when X represents -CHN(R<1><0>,R<1><1>)- and R<1> and R<2> together form a bond, that the sum of p and q is 0-4 when X represents -CHN(R<1><0>,R<1><1>)- and R<1> and R<3> together form a bond and that p stands for 1-4 when X represents -N(R<9>)-, R<1> and R<3> together represent a bond and m stands for 0, as well as pharmaceutically acceptable salts of acidic compounds of formula I with bases and of basic compounds of formula I with acids, are useful in the control or prevention of inflammatory, immunological, oncological, bronchopulmonary, dermatological or cardiovascular disorders or for the treatment of asthma, AIDS or diabetic complications or for the stimulation of hair growth. They can be prepared from correspondingly substituted furandiones.
Patent CS-261791-A3 (CS)
Title: Process for preparing preparations in the form of tablets or coated tablets containing light, heat and moisture sensitive active component having a monoclinic crystal structure
Inventor: KOVACS ISTVAN
IPC: A61K47/38
Filed: 1991-08-23
Abstract: PCT No. PCT/HU91/00039 Sec. 371 Date Jun. 5, 1992 Sec. 102(e) Date Jun. 5, 1992 PCT Filed Aug. 23, 1991 PCT Pub. No. WO92/03126 PCT Pub. Date Mar. 5, 1992.The invention relates to a process for the preparation of a tablet or dragée composition containing a moisture-, heat- and light-sensitive compounds having monoclinic crystalline structure as active ingredients, which comprises homogenizing the active ingredient with 0.2 to 1.5 parts by weight of an anhydrous alkaline earth metal salt and 0.5 to 2.5 parts by weight of microcrystalline cellulose calculated for the active ingredient and optionally with one or more pharmaceutically acceptable carrier(s) and/or additive(s) and compressing the homogeneous mixture obtained to tablets in a manner known per se and, if desired, coating the tablet thus obtained in a manner known per se.
Patent CZ-100895-A3 (CZ)
Title: Enantiomeric cis-3-(4,6-dihydroxychroman-3-ylmethyl)benzoic acids
Inventor: MURTIASHAW CHARLES W
IPC: C07D311/22
Filed: 1993-06-30
Abstract: This invention relates to enantiomerically pure cis-3-(4,6-dihydroxychroman-3-ylmethyl)benzoic acids and processes for the preparation of such compounds. The compounds are intermediates useful in the preparation of optically pure enantiomers of cis-3-(6-arylmethyloxy-4-hydroxy-chroman-3-ylmethyl)aniline sulfonamides which are useful in the treatment of asthma, arthritis, psoriasis, ulcers, myocardial infarction and related diseases. More particularly it relates to (3R-cis)-3-(4,6-dihydroxychroman-3-ylmethyl)benzoic acid. It also relates to an improved process for the preparation of racemic cis-3-(4,6-dihydroxychroman-3-ylmethyl)benzoic acid.
Patent CZ-188397-A3 (CZ)
Title: Oral preparations containing dimethicone co-polyols
Inventor: HUGHES IAIN ALLAN
IPC: A61K8/38
Filed: 1995-11-21
Abstract: An oral composition in the form of a toothpaste, powder, liquid dentifrice, mouthwash, denture cleanser, chewing gum or candy comprising a lipophilic compound selected from flavorants, physiological cooling agents and antimicrobial compounds and a dimethicone copolyol selected from alkyl- and alkoxy-dimethicone copolyols having formula (I) wherein X is selected from hydrogen, alkyl, alkoxy and acyl groups having from about 1 to about 16 carbon atoms, Y is selected from alkyl and alkoxy groups having from about 8 to about 22 carbon atoms, n is from about 0 to about 200, m is from about 1 to about 40, q is from about 1 to about 100, the molecular weight of the residue (C2H4O-)x(C3H6O-)yX is from about 50 to about 2000, and x and y are such that the weight ratio of oxyethylene:oxypropylene is from about 100:0 to about 0:100. The composition provides improved antiplaque and anti-bacterial activity together with enhanced substantivity, impact and/or efficacy of the lipophilic components on teeth or dentures.
Patent CZ-189997-A3 (CZ)
Title: Bicyclic compounds, process of their preparation and pharmaceutical composition based thereon
Inventor: DIMAIO JOHN
IPC: A61K31/435
Filed: 1995-12-21
Abstract: This invention relates to the discovery of heterocyclic competitive inhibitors of the enzyme thrombin having formula (I), their preparation, and pharmaceutical compositions thereof. As well, this invention relates to the use of such compounds and compositions in vitro as anticoagulants and in vivo as agents for the treatment and prophylaxis of thrombotic disorders such as venous thrombosis, pulmonary embolism and arterial thrombosis resulting in acute ischemic events such as myocardial infarction or cerebral infarction. Moreover, these compounds and compositions have therapeutic utility for the prevention and treatment of coagulopathies associated with coronary bypass operations as well as restenotic events following transluminal angioplasty.
Patent CZ-192998-A3 (CZ)
Title: 2,7-SUBSTITUTED OCTAHYDROPYRROLO[1,2-a]-PYRAZINE DERIVATIVES, INTERMEDIATES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS BASED THEREON
Inventor: SANNER MARK A
IPC: C07D487/04
Filed: 1996-11-06
Abstract: This invention relates to compounds of formula (I), wherein R1 is phenyl, naphthyl, benzoxazolonyl, indolyl, indolonyl, benzimidazolyl, quinolyl, furyl, benzofuryl, thienyl, benzothienyl, oxazolyl, benzoxazolyl; R2 is H or (C1-C6)alkyl; R3 is phenyl, pyridinyl, pyrimidinyl, pyrazinyl, or pyridazinyl; X is O, S, SO, SO2, NR4, C=O, CH(OH), CHR4, (a), (b), (c), or (d); m is 0, 1 or 2; n is 0, 1 or 2. The compounds of this invention are ligands for dopamine receptor subtypes, especially the dopamine D4 receptor, and are therefore useful in the treatment of disorders of the dopamine system.
Patent CZ-201853-A3 (CZ)
Inventor: MATĚJŮ TOMÁŠ
IPC: F21S41/36
Filed: 2018-01-31
Abstract: Řešení se týká optického systému obsahujícího dvě řady zdrojů (1a, 1b) světla tvořených LED. Každá řada zdrojů (1a, 1b) světla je celá uspořádána na jedné straně oboustranné desky (2) plošných spojů a každému zdroji (1a, 1b) v každé řadě je přiřazen vlastní reflektor (3a, 3b), přičemž před oběma řadami reflektorů (3a, 3b) je uspořádán jeden optický filtr (4), který je společný pro obě řady reflektorů (3a, 3b) a na jehož výstupní ploše jsou vytvořeny polštářky (5), které jsou rozděleny do dvou skupin (51, 52), z nichž každá skupina (51, 52) je uzpůsobena k lomu paprsků (6a, 6b) světla z příslušné řady zdrojů (1a, 1b) světla, po odrazu těchto paprsků (6a, 6b) od příslušné řady reflektorů (3a, 3b) přiřazené příslušné řadě zdrojů (1a, 1b) světla a po průchodu těchto odražených paprsků (6a, 6b) filtrem (4), do směru (x) svícení.
Patent CZ-284395-A3 (CZ)
Title: Process for preparing substances suitable for synthesis of fungicidal agents
Inventor: SAKSENA ANIL K
IPC: C12P7/04
Filed: 1994-04-28
Abstract: Disclosed is a process for preparing chiral compounds of the formula (I)    <IMAGE>  (I)  wherein: X1 and X2 are independently F or Cl; and E is -SO2R2, wherein R2 is C1-C6 alkyl, -C6H4CH3 or -CF3; its enantiomer and racemates thereof, useful in the synthesis of tetrahydrofuran azole antifungals. Novel compounds of the formula   <IMAGE>   or   <IMAGE>   wherein: X1 and X2 are independently F or Cl; B represents -C(O)Q* or -CH2OR''; Q* represents a chiral auxiliary group; R'' represents a hydroxy protecting group selected from -CH2C6H5, or -C(O)R1, wherein R1 is C1-C6 alkyl; and A represents Cl, Br, I or triazolyl; are also disclosed.