baber/WOPTO huggingface dataset:
Patent NO-170631-B (NO)
Title: Analogifremgangsmaate for fremstilling av terapeutisk aktive 2-pyrimidinaminer
Inventor: TORLEY LAWRENCE WAYNE
IPC: C07D409/04
Filed: 1987-01-14
Abstract: Terapeutisk aktive forbindelser ifølge formelen. hvor Ri er hydrogen, alkyl(Ci-Ca), -COCO2C2 Ho eller N,N-dimetyl-aminoetyl; Rer mono- eller polysubstituert fenyl; Ra er 2-pyridinyl, 3-pyridinyl, 4-pyridinyl, 2-metyl-3-pyridinyl, 4-metyl-3-pyridinyl, 2-furanyl, 5-metyl-2-furanyl, 2,5-dimetyl-3-furanyl, 2-tienyl, 3-tienyl, 5-metyl-2-tienyl, 2-fenotiazinyl, 4-pyrazinyl, 2-benzofuranyl, 2-(pyridin-N-oksyd), 3-(pyridin-N-oksyd), 4-(pyridin-N-oksyd), lH-indol-2-yl, lH-indol-3-yl, 1-metyl-lH-pyrrol-2-yl, 4-kinolinyl, 4-pyridinylmetyljodid, dimetylaminofenyl eller N-acetyl-N-metylaminofenyl; R« er hydrogen eller alkyl (Ci -C3 ) ; og R-i er hydrogen eller alkyl (Ci -C3 ) .Spesielt har forbindelsene anti-astmatisk aktivitet. Fremstilling av forbindelsene er beskrevet.
Patent NO-168243-B (NO)
Inventor: MATSUO MASAAKI
IPC: C07D277/36
Filed: 1988-05-27
Abstract: Alkanesulfonanilide derivatives of the formula : <CHEM>  wherein  Ar is a group of the formula : <CHEM> wherein R<4>, R<5>, R<6> and R<7> are each hydrogen, halogen, halo(lower)alkyl or lower alkoxy,  or heterocyclic group which may have halogen or lower alkyl  X is @@@n , - @@ , -CO-, -NHCO-, -CONH- or - @@-    wherein n is 0, 1 or 2, R<8> is hydrogen or lower alkyl,  R<9> is hydrogen or hydroxy,  R<1> is lower alkyl or halo(lower)alkyl,  R<2> defines certain substituents, R<3> is hydrogen, nitro lower alkyl or halogen, and pharmaceutical acceptable salts thereof, processes for their preparation and pharmaceutical compositions comprising them.
Patent NO-180191-B (NO)
Inventor: DAHL BJARNE HUGO
IPC: A61P25/18
Filed: 1992-03-13
Abstract: A method of treatment with compounds having the formula <CHEM>  wherein  n is 0 or 1; R<1> is hydrogen, C1-6-alkyl which may be branched, C3-7-cycloalkyl, benzyl, phenyl which may be substituted, acyl, hydroxy, C1-6-alkoxy, CH2CO2R' wherein R' is hydrogen or C1-6-alkyl which may be branched, CH2CN, CH2CONR<IV>R<V> wherein R<IV> and R<V> independently are hydrogen or C1-6-alkyl, or CH2C(=NOH)NH2; R<2> is pyridyl or phenyl, both of which may be substituted one or more times preferably in the ortho and para positions with halogen, CF3, NO2, CN, phenyl, SO2NR''R''' wherein R'' and R''' independently are hydrogen, benzyl, or C1-6-alkyl; R<4>, R<5>, R<6>, R<7> independently are hydrogen, C1-6-alkyl which may be branched, phenyl, halogen, C1-6-alkoxy, NO2, CN, CF3, or SO2NR<1><1>R<1><2> wherein R<1><1> and R<1><2> independently are hydrogen, benzyl, or C1-6-alkyl; or R<6> and R<7> together form an additional 4 to 8 membered carbocyclic ring which may be aromatic or partial saturated and which may be substituted with halogen, NO2, CF3, CN, SO2NR<1><3>R<1><4> wherein R<1><3> and R<1><4> independently are hydrogen, benzyl, or C1-6-alkyl, and R<4> and R<5> have the meanings set forth above; or R<4> and R<5> together form an additional 4 to 8 membered carbocyclic ring which may be aromatic or partial saturated and which may be substituted with halogen, NO2, CF3, CN, SO2NR<1><3>R<1><4> wherein R<1><3> and R<1><4> independently are hydrogen, benzyl, or C1-6-alkyl, and R<6> and R<7> have the meanings set forth above. Certain of the compounds are novel. The compounds and pharmaceutical compositions containing the compounds are useful in the treatment of central nervous system disorders and especially conditions sensitive to excitatory amino acids.
Patent NO-180804-B (NO)
Inventor: HORROBIN DAVID FREDERICK
IPC: A61K8/30
Filed: 1992-06-02
Abstract: A natural or synthetic glycerol oil which comprises at least 20% by weight, preferably at least 25 % of di-linoleoyl-mono-gamma-linolenyl-glycerol (DLMG), is used to supplement foods, nutritional compositions and in skin and hair care compositions.
Patent NO-178500-B (NO)
Inventor: OTAKE NOBORU
IPC: C07H19/16
Filed: 1992-07-08
Abstract: Disclosed is a novel spicamycin derivative represented by the formula (I) or a salt thereof: <CHEM> wherein R represents an alkenyl having a given number of carbon atoms, a haloalkyl having a given number of carbon atoms, CH3(CH2)nCH(OH)- or CH3(CH2)n-lCH(OH)-CH2- (wherein n denotes an integer of 9-13), an alkyl with a certain group and a given number of carbon atoms, <CHEM>  (wherein a denotes 2, and b denotes an integer of 10-15),     CH3(CH2)cSO2O(CH2)d- , <CHEM> (wherein c denotes an integer of 0-3 and d denotes an integer of 10-15),     (CH3)3Si(CH2)10- ,     (CH3)3Si-C IDENTICAL C-(CH2)8-, <CHEM>  or <CHEM> (wherein X represents O or S), and R1 and R2 are different from each other and each represents H or OH, which exhibits an excellent antitumor effect and has a high therapeutic index. An antitumor agent containing at least one of the above-described compounds in an effective amount is also disclosed.
Patent NO-180812-B (NO)
Inventor: HAEGGSTROEM THORSTEN
IPC: A21B5/03
Filed: 1993-04-29
Abstract: PCT No. PCT/SE91/00726 Sec. 371 Date Apr. 30, 1993 Sec. 102(e) Date Jun. 30, 1993 PCT Filed Oct. 29, 1991 PCT Pub. No. WO92/07469 PCT Pub. Date May 14, 1992.A method and device for baking dough or batter comprising at least two heatable plates, each of them having a top side, wherein the dough or batter is automatically put on the first and second heated plates for making pastries, pancakes and the like. The method is characterized in that the dough or the batter is baked on its one side on the top side of the first plate whereafter the partly baked dough or batter, is transferred to the second plate and is baked on its other side. The pastry/pancake, completely baked on the second plate is pivotably transferred to a laying off place. Using the device, a plurality of pastries, pancakes, and the like can be automatically and systematically produced.
Patent SE-331303-B (SE)
Inventor: CRANE P
IPC: H02M1/08
Filed: 1966-07-11
Abstract: 1,127,685. Automatic voltage control. MAGNAVOX CO. July 11, 1966 [July 12, 1965], No.30998/66. Heading G3R. A regulated D.C. output at terminals 40, 42 is derived from an A. C. input at terminals 10, 12 by way of a full-wave rectifier 20 and a thyristor 46 which is connected between the rectifier 20 and a smoothing circuit 52, 44 for the D.C. output; firing pulses for the thyristor are derived from the unsmoothed output of rectifier 20 by means of a circuit including resistors 80, 82 and 83, a differentiating capacitor 84, a first transistor 60 and a second transistor 70 which has its collector connected to the control electrode of thyristor 46 over a capacitor 88 having a low resistance to the transient firing pulses but a large resistance to the rectified A. C. which might otherwise have unwanted switching effects on the thyristor. The output voltage at terminals 40, 42 is automatically maintained constant by control of the firing angle of the thyristor 46 in dependence upon output voltage variations as detected by a circuit including a voltage divider 100, 102, 106 and a Zener diode 108 which is connected to the base of transistor 60, and the Specification describes how the required firing pulses are produced with reference to Fig. 2 (not shown).
Patent YU-45956-B (YU)
Inventor: DESPLATS A
IPC: B66D3/02
Filed: 1982-07-12
Abstract: Each half-case of the apparatus comprises a main half-case of pressed steel sheet provided with two chimneys on which is mounted a reinforcement piece, also of pressed steel sheet, having openings corresponding to the chimneys. The main half-case and the reinforcement piece separately each receive an anti-corrosion coating. Two symmetrical half-cases are finally fitted together along a longitudinal plane.
Patent YU-45847-B (YU)
Title: Armirano betonski montažni dvodelni rešetkasti nosač
Inventor: ZLATAN ZLATANOVIC
IPC: E04C3/20
Filed: 1988-11-03
Abstract: ARMIRANO BETONSKI MONTAŽNI DVODELNI REŠETKASTI NOSAČ, naznačen time, što su klasično armirane polurešetke (1,2) medjusobno spojene cevastom, sa navojima maticom (6) navrtnutom na ispuštenu, sa navojnicom (5) primarnu armaturu (4) i što na kraju gornjeg pojasa plurešetke (2) pero (6) zalazi u žljeb (15) na kraju polurešetke (1) pri čemu su polurešetke (1,2) oslonjene i povezane sa stubovima (10) preko čeličnih podvezica (7) vertikalno ubetoniranih jednim krajem u stubove (10) a drugim krajem uvučenim u proreze (8) polurešetke (1,2) i fiksiranih medjusobno poprečnim zavrtnjima (11) a preko uložaka (9) polurešetke (1,2) oslonjene na stubove (10).
Patent YU-47252-B (YU)
Title: Konstrukcija mehaničkog uredjaja za spuštanje kablova
Inventor: NAVEDEN NE ZELI DA BUDE
IPC: E04C5/08
Filed: 1986-12-15
Abstract: KONSTRUKCIJA MEHANIČKOG UREDJAJA ZA SPUŠTANJE KABLOVA, naznačena time, što se sastoji od kuke sa produženim navojem (3), osigurača (4) podložne čelične kutije (6), navrtke (7), i što se kukom (3) obuhvati pravolinijski čelični kabl (5), a osiguračem (4) zaključa položaj kuke (3), i produženi navoj kuke (3) navuče kroz otvor (6a) i navrtku (7) na čeličnoj kutiji (6), koja se sa svojim nožicama odupire na betonske elemente (2), i što se zavrtanjem navrtke (7) pravolinijski čelični kabl (5) postepeno dovede u projektovani položaj (5a), i što se po fiksiranju kabla (5a) uredjaj oslobadja odvrtanjem navrtke (7) i premešta na sledeći pravolinijski kabl.
Patent YU-47602-B (YU)
Title: Mehanizam za naginjanje lestvica na roletni
Inventor: OBREZA I
IPC: E05F5/04
Filed: 1987-12-16
Abstract: MEHANIZAM ZA NAGINJANJE LESTVICA NA ROLETNI, gde je u žljebu (2a) ugradjena pomična letva (5), nataknuta na elastične čepove (4Ab) okova (4A) letvice (3) roletne, naznačen time, što se čep (11), pričvršćen na spojnom članu (9), pruža u otvor (5b) na pomičnoj letvi (5), i što na drugoj strani spojnog člana (9) sa suprotne strane je pričvršćena cilindrična osovinica (10), koja se pruža kroz vodeće proreze (6a) i (6b), iz leve ili desne strane vodjice (6) ručice (7), pri čemu je izmedju bočnih zidova (6e) obrtno-klizno pomično ugradjena ručica (7). Prijava sadrži još 1 zavisan zahtev.
Patent YU-47078-B (YU)
Title: Postupak za konverziju polimorfnog kristalnog oblika
Inventor: BEHME R J
IPC: A61K31/495
Filed: 1989-12-29
Abstract: POSTUPAK ZA KONVERZIJU POLIMORFNOG KRISTALNOG OBLIKA, buspiron hlorhidrata, kako bi se dobio polimorf sa višom tačkom topljenja, P203, naznačen time, što obuhvata razaranje kristalne strukture polaznog polimorfnog kristalnog oblika ili smeše dva polimorfna kristalna oblika buspiron hlorhidrata rastvaranjem u tečnom medijumu i zatim rekristalizacijom na temperaturi višoj od 95В°C, ili mešanjem sa tečnim medijumom, na temperaturi višoj od 95В°C, uz uspostavljanje ravnoteže čvrsta supstanca/tečnost, sve dok se čvrsti buspiron hlorhidrat u potpunosti ne prevede u polimorf P203, nakon čega se dobijeni polimorfni oblik buspiron hlorhidrata odvaja od tečnog medijuma. Prijava sadrži još 3 zavisna zahteva.
Patent ZA-821595-B (ZA)
Title: Process for the preparation of urea
Inventor: BURKS HENK CHRISTIAAN
IPC: C07C239/00
Filed: 1982-03-10
Abstract: A process for the preparation of urea at elevated temperatures and pressures in which ammonium carbamate is decomposed into ammonia and carbon dioxide and separated from the urea product stream in at least two pressure stages. The product urea stream having reduced ammonium carbamate content leaving the first high pressure stage is reduced in pressure to a level intermediate the pressure of the high pressure stage and the next pressure stage in a pressure reducing device in which the energy released by the pressure reduction is converted into kinetic energy by means of which a gaseous mixture of ammonia and carbon dioxide resulting from the carbamate decomposition in a further pressure stage or recovered the process condensate formed in a concentrating stage is compressed to the intermediate pressure. The resulting compressed mixture is thereafter condensed, and the condensate thus formed is pumped to the high pressure stage.
Patent ZA-844322-B (ZA)
Title: Floor-mounted outlet for ventilating and air conditioning systems
Inventor: FEY MICHAEL
IPC: F24F13/06
Filed: 1984-06-07
Abstract: A floor outlet for an air conditioner has a grill which is formed by ring elements whose radial connecting ribs are inclined to impart a vortex flow to the emerging air. A central baffle body is constituted by a disc and a multiplicity of angularly equispaced radially extending blades twisted out of the plane of the disc and projecting therefrom.
Patent ZA-849608-B (ZA)
Title: Method and apparatus for supplying printed products to a continuously operating processing line
Inventor: HONEGGER WERNER
IPC: B65H29/51
Filed: 1984-12-11
Abstract: One stack space is provided for accommodating each stack of a plurality of stacks of printed products to be supplied to the processing line. Each stack space is provided with a powered feed mechanism which urges the associated stack toward a predetermined processing location, such as a product singling or supply device for singly transferring printed products to the processing line. To be able to prepare the supply of printed products at a location remote from or independent of the processing line, a plurality of transportable winding frames are provided. The winding frames are equipped for exchangeably accommodating a wound package of mutually identical printed products. The winding frames are provided with drive and conveying means which drive the wound package in an unwinding direction and convey the printed products unwinding from the printed package to a transfer location. The winding frames are each selectively connectible to any one of the feed mechanisms, while a drive member of the feed mechanism can be simultaneously coupled to a drive member of the drive and conveying means.
Patent ZA-866620-B (ZA)
Title: A method of producing polymers and copolymers of amido-sulfonic acid containing monomers and salts thereof
Inventor: SOPKO THOMAS M
IPC: C08F120/58
Filed: 1986-09-01
Abstract: A fluid loss agent comprising homopolymers or copolymers from amido-sulfonic acid or salt containing monomers obtainable in the presence of high energy mechanical mixing utilizing a final stage polymerisation temperature of from about 93 DEG C (200 DEG F) to below the degradation temperature of the monomer.
Patent ZA-867703-B (ZA)
Title: Oral delivery system
Inventor: RUSSELL-JONES GREGORY JOHN
IPC: A61K38/28
Filed: 1986-10-09
Abstract: The present invention provides a complex of a drug, hormone, bio-active peptide, or immunoger with the carrier molecule vitamin B12 and a method for delivering said complex to the intestine of a host vertebrate in order to deliver the complex to the circulation of the host and thereby elicit a pharmacological response to the drug, hormone, or bio-active molecule or to elicit a systemic immune response to the immunogen. The invention also provides a method for the production of the complex. Further the invention provides medicaments containing the complex.
Patent ZA-876729-B (ZA)
Title: Emanator for volatile liquids
IPC: A01N25/10
Filed: 1987-09-09
Abstract: A device for dispensing a volatile liquid as a vapour includes a porous support of natural or synthetic woven or non-woven fibre, porous glasses, porous plastics (optionally in film form), parchment, leather or rubber provided with an organopolysiloxane material which serves to close the pores of the support to the passage of liquid but permits the passage of vapour from the liquid. The volatile liquid is a perfume, insecticide, insect repellant, insect attractant, higher animal repellant, corrosion inhibitor, a germicidal agent or a medicament. A space treatment vapour emanating device is thus provided the external surface of which device is dry to the touch.
Patent ZA-881739-B (ZA)
Inventor: HOFFMANN RAINER DR
IPC: A61D7/00
Filed: 1988-03-11
Abstract: A plaster containing active ingredients for controlled administration of active ingredients to the skin and possessing a rear side and a skin side, has a rear layer, an active ingredient reservoir containing one or more active ingredients arranged essentially perpendicular to the surface of the plaster in contact with the skin, and an adhesive device on the skin side and possibly a covering layer which is detached before application of the plaster. At least one active ingredient reservoir part (12) can be detached on to the skin while one or more active ingredient reservoir parts remain. For this purpose, the part (13) of the active ingredient reservoir remaining on the skin adheres more strongly to the skin than to the rear side (11).
Patent ZA-905272-B (ZA)
Title: An apparatus for,and a method of,cutting a blank
Inventor: PORUCZNIK PAUL
IPC: B26F1/44
Filed: 1990-07-05
Abstract: When a blank is cut from metal sheet which suffers from crystallographic anisotropy, there is a tendency for ears to be formed during subsequent forming operations, such as drawing or pressing. In order to compensate for this tendency, there may be used a metal blank which is not completely round, but has lobes at positions to cancel at least some of the valleys between the ears. There is described a punch (110) and die (111) which may be used to form such a lobed blank (112). The punch (110) has four circumferentially extending lobe-forming sections (124). Each lobe-forming section is constructed by forming a stepped recess in the cutting edge of the punch (110). In each lobe-forming section, the depth of the recess varies from a maximum at the middle of the section to zero at the ends. The die (111) is conventional.
Patent ZA-911657-B (ZA)
Title: 3-tetrazolylthiomethyl cephalosporin antibiotics
Inventor: JUNG FREDERICK HENRI
IPC: A61K31/546
Filed: 1991-03-06
Abstract: A compound of the formula (II): <CHEM> and pharmaceutically acceptable salts and in vivo hydrolysable esters are described as is their preparation and use as antibacterial agents.
Patent ZA-913992-B (ZA)
Title: A process for preparing a soya food product
Inventor: LEMPKE FREDERICK ERNST VAN
IPC: A23L23/00
Filed: 1991-05-27
Abstract: The invention provides a process for preparing a soya food product including the steps of providing a soya concentrate, and pre-mixing the soya concentrate with a composition including organic flavourants, an amino acid supplementation, an extract of a spice and vitamins. The pre-mixed product is then mixed with water at a temperature below 15 DEG C and then allowed to soak for a period of time sufficient to allow the soya concentrate substantially to absorb the composition. The process may further include a par-cooking step where the product is partially cooked by frying in an oil or fat medium at a temperature above 170 DEG C. The process may also include a cooling step where the product is crust frozen at a temperature below -100 DEG C.
Patent ZA-915437-B (ZA)
Title: Inhaler
Inventor: BRAITHWAITE PHILIP WILSON
IPC: G06M1/24
Filed: 1991-07-12
Abstract: The invention provides an inhaler for delivering a substance in a finely divided form from a storage chamber within the inhaler. The inhaler comprises a metering member operable to transfer a dose of the substance from the storage chamber (10) to an inhalation passage (15), the metering member having a frusto-conical metering surface (7) which is indented to provide at least one dispensing cup (8) and being moveable between a first position in which a dispensing cup (8) is presented to the storage chamber (10) to receive a dose of the substance and a second position in which a dose of the substance is presented to the inhalation passage (15) in an upwardly open dispensing cup (8). The body (4) of the inhaler comprises a seat having an annular, frusto-conical contact surface making sliding contact with the metering surface and defining a socket within which the metering member (6) is journalled for rotation between its first and second positions. The use of a frusto-conical metering member allows a good seal to be obtained between it and the seat and also makes the inhaler relatively compact. <IMAGE>
Patent ZA-928234-B (ZA)
Title: Process for the production of aminoalkanephosphonic acids, salts and/or esters.
Inventor: AXIOTIS GEORGES
IPC: C07F9/40
Filed: 1992-10-23
Abstract: The present invention relates to a new process for obtaining  alpha -aminoalkanephosphonic acids and/or salts or esters of general formula (I): <IMAGE>  with   R1, R2, which are identical or different, chosen from a hydrogen atom, a linear or branched alkyl group with one to six carbon atoms, or an alkali metal or alkaline-earth metal atom. R3 = a hydrogen atom or an alkyl, cycloalkyl, aryl or aralkyl group, it being possible for these groups to be optionally substituted by one or a number of heteroatoms, preferably halogen. R4 = a hydrogen atom or a linear or branched alkyl group with 1 to 4 carbon atoms.
Patent ZA-938611-B (ZA)
Title: Anilines as markers for mineral oils
Inventor: DYLLICK-BRENZINGER RAINER
IPC: C10M171/00
Filed: 1993-11-18
Abstract: PCT No. PCT/EP93/03133 Sec. 371 Date Jun. 22, 1995 Sec. 102(e) Date Jun. 22, 1995 PCT Filed Nov. 9, 1993 PCT Pub. No. WO94/11466 PCT Pub. Date May 26, 1994Anilines of the formula    <IMAGE>  (I)  where R1 and R2 are each hydrogen, unsubstituted or substituted alkyl, alkenyl or unsubstituted or substituted phenyl or R1 and R2, together with the nitrogen atom linking them are a heterocyclic radical or R1 may furthermore be unsubstituted or substituted hydroxyl or unsubstituted or substituted amino, R3 and R7 are each hydrogen, unsubstituted or substituted alkyl, alkenyl, cyano, nitro, acyl, acylamino, unsubstituted or substituted hydroxyl, unsubstituted or substituted carboxymethyl, unsubstituted or substituted amino, unsubstituted or substituted mercapto or unsubstituted or substituted sulfamoyl or, together with R2, are alkylene, alkenylene or phenylalkenylene, R4 is hydrogen, unsubstituted or substituted alkyl, alkenyl, unsubstituted or substituted hydroxyl, unsubstituted or substituted amino, unsubstituted or substituted carboxyl or unsubstituted or substituted sulfamoyl and R5 and R6 are each hydrogen, unsubstituted or substituted alkyl, alkenyl, unsubstituted or substituted phenyl, nitro, acylamino, unsubstituted or substituted hydroxyl, unsubstituted or substituted amino, unsubstituted or substituted sulfamoyl, alkyl-, alkenyl- or arylsulfonyl, acyl or unsubstituted or substituted carboxyl, with the proviso that at least one of the radicals R3, R5 or R7 is hydrogen, are used for marking mineral oils, and the above-mentioned anilines are detected in mineral oils.
Patent ZA-939614-B (ZA)
Title: Dispensing device
Inventor: COFFEE RONALD ALAN
IPC: B05B5/025
Filed: 1993-12-22
Abstract: A dispensing device has liquid supplying means (9, 13) having a liquid outlet and electrical charging means (9) for generating an electrical field to cause liquid issuing from the liquid outlet to be comminuted to provide electrically charged comminuted matter. In an embodiment the electrical charging means are arranged to induce an electrical charge to cause comminution. The device also has electrical discharging means (6;14) for providing ions for at least partially electrically discharging the comminuted matter, and ion attracting means (10,11) for attracting ions generated by the electrical discharging means away from the electrical charging means until a spray cloud of electrically charged comminuted matter has been established by the electrical charging means. <IMAGE>
Patent ZA-957474-B (ZA)
Title: Highly active double metal cyanide catalysts
Inventor: LE-KHAC BI
IPC: C08L71/02
Filed: 1995-09-06
Abstract: A solid double metal cyanide (DMC) catalyst useful for epoxide polymerisation comprises: (a) a double metal cyanide cpd; (b) an organic complexing agent; and (c) about 5-80 wt% based on the amt of catalyst, of a polyether having a number average molecular wt greater than about 500. Also claimed are: Preparing a solid DMC catalyst in the presence of an organic complexing agent and a polyether as above, wherein the solid DMC catalyst contains 5-80 wt% of the polyether. Preparing a soli DMC catalyst useful for epoxide polymerisation.