baber/WOPTO huggingface dataset:
Patent HU-T73141-A (HU)
Title: Process for preparing benzoic acid derivative intermediates and benzothiophene pharmaceutical agents
Inventor: KJELL DOUGLAS PATTON
IPC: C07C213/00
Filed: 1995-08-30
Abstract: The present invention provides a novel process for preparing novel compounds of formula I <CHEM>  wherein R<1> and R<2> each are independently C1-C4 alkyl, or combine to form piperidinyl, pyrrolidinyl, methylpyrrolidinyl, dimethylpyrrolidinyl, morpholino, dimethylamino, diethylamino, or 1-hexamethyleneimino; and     n is 2 or 3;  or a pharmaceutically acceptable salt thereof, comprising     a) reacting a haloalkyl amine of formula III <CHEM>  wherein     X is a halogen; and R<1>, R<2>, and n are as defined above, with a compound of formula IV   <CHEM> wherein R is C1-C6 alkyl, in the presence of an alkyl acetate solvent and a base; b) extracting the reaction product of step a) with an aqueous acid; and c) cleaving the ester of the reaction product from step b) to form an acid.   The present invention further provides a novel process for preparing compounds of formula V <CHEM>  wherein R<1> and R<2> each are independently C1-C4 alkyl, or combine to form piperidinyl, pyrrolidino, methylpyrrolidino, dimethylpyrrolidinyl, morpholino, dimethylamino, diethylamino, or 1-hexamethyleneimino;     R<3> and R<4> each are H or a hydroxy protecting group; and     n is 2 or 3;  or a pharmaceutically acceptable salt thereof, comprising     a) reacting a haloalkyl amine of formula III <CHEM>  wherein     X is a halogen; and R<1>, R<2>, and n are as defined above, with a compound of formula IV   <CHEM> wherein R is C1-C6 alkyl, in the presence of an alkyl acetate solvent and a base; b) extracting the reaction product from step a) with an aqueous acid;   c) cleaving the ester of the reaction product from step b) to form an acid; d) reacting the extracted product from step c) with a compound of formula V <CHEM> wherein R<3> and R<4> are as defined above, or a pharmaceutically acceptable salt thereof; e) optionally removing the R<3> and R<4> hydroxy protecting groups of the reaction product form step d); and f) optionally forming a salt of the reaction product from either steps d) or step e).
Patent HU-T74293-A (HU)
Title: Process for the production of aminoalkylguanidines and products of the method
Inventor: NYSTROEM JAN-ERIK
IPC: C07D231/12
Filed: 1994-06-01
Abstract: PCT No. PCT/SE94/00517 Sec. 371 Date Jun. 28, 1994 Sec. 102(e) Date Jun. 28, 1994 PCT Filed Jun. 1, 1994 PCT Pub. No. WO94/29269 PCT Pub. Date Dec. 22, 1994A process for the production of guanidino protected  omega -aminoalkyl guanidines comprising reacting a diamine selectively at one amino group with an alkoxycarbonyl or aralkoxycarbonyl protected electrophilic guanylation reagent. The process of the invention is general and may be performed efficiently in one step yielding a product with high purity and in useful yields. The invention further refers to some compounds that are novel per se and to some novel compounds useful in the process of the invention.
Patent HU-T77693-A (HU)
Title: A pant diaper or sanitary panty having a detachably connected front part
Inventor: ROMARE ANETTE
IPC: A61F13/62
Filed: 1995-04-11
Abstract: PCT No. PCT/SE95/00389 Sec. 371 Date Sep. 30, 1996 Sec. 102(e) Date Sep. 30, 1996 PCT Filed Apr. 11, 1995 PCT Pub. No. WO95/27460 PCT Pub. Date Oct. 19, 1995A pant diaper or a sanitary panty which includes a front part, a rear part, and an intermediate crotch part, which includes an absorbent body enclosed between an inner and an outer casing sheet. The front part is detachably joined to the rear part by means of a first fastening. A piece of flexible material extends over the front part and is joined thereto over a larger part of its surface by means of a first releasable fastening, which extends on both sides of a centrally located region of the piece of material, from the edges of the central region to the respective side edges of the front part. The piece of material is also joined to the rear part.
Patent HU-T76171-A (HU)
Title: Roof window
Inventor: GEIB JOERG
IPC: E04D13/035
Filed: 1995-06-14
Abstract: The invention relates to an opening roof window (10) for a pitched roof, with a base frame (12) and a glazed wing (14) which may be secured as desired to one of at least two equal-length sides of the base frame (12), in which the glazed wing (14) is articulated on the base frame (12) by at least one hinge (16) having a movable section (18) fastened to the glazed wing (14) and a fixed section (20) and a catch (26) spaced away from the hinge (16) for securing the glazed wing (14) to at least one engaging component (28) securable to the base frame (12). To provide a roof window through which access can safely be gained to the roof and which is economical to produce, it is proposed that the hinge sections (18, 20) be pivotably combined into a unit, the fixed hinge section (20) have a retainer (22) which can be fitted to the selected side of the base frame (12) and there be bearing surfaces (34) on the base frame (12) for the fitting as desired of the retainer (22) or the engaging component (28).
Patent IL-43528-A (IL)
Title: Tone detector
IPC: H04L27/26
Filed: 1973-10-31
Abstract: 1412897 Selective signalling MOTOROLA Inc 7 Nov 1973 [7 Nov 1972] 51635/73 Heading G4H [Also in Division H3] The invention relates to a switchable frequency filter which is capable of responding to a plurality of predetermined tones in rapid succession. The filter has a predetermed energy build up and decay rate in response to the tones, and speed of operation is ensured by temporarily increasing the bandwidth of the filter after detection of a tone frequency to increase the decay rate before selecting the next frequency to which the filter is to respond. The filter 19 comprises operational amplifiers 38, 43, 50 with a resistor 48 and a capacitor 49 which respectively determine the pass frequency and the bandwidth of the filter. Connection of a capacitor 60 in parallel with capacitor 49 increases the bandwidth, and connection of one or more resistances 67 ... 90 in parallel with resistor 48 alters the frequency to be passed. A signal containing an audio part and a sequence of tones constituting an address is received at 10, 11 and passed to amplifier 12 which is held inoperative until a circuit 15 containing filter 19 has detected the required tone sequence. Detection of a frequency causes a counter 21 to be incremented and a timing circuit 22 to switch capacitor 60 into filter 19 so as to increase the bandwidth for a predetermined time. The output from 21 causes a diode matrix 23 to output a signal 24 to the filter to switch in a new combination of resistors 67 ... 90 so as to select the next frequency. When all the tones have been detected, counter 21 actuates an "audio alert" device 30 and enables amplifier 12.
[GB1412897A]
Patent IL-88473-A (IL)
Title: Substituted alkylamine derivatives, their preparation and pharmaceutical compositions containing them
IPC: C07C255/36
Filed: 1988-11-24
Abstract: A substituted alkylamine derivative represented by the general formula <CHEM> wherein A represents a methine group, a nitrogen atom, an oxygen atom or a sulfur atom; Q represents a group which may contain one or two hetero atoms selected from the group consisting of nitrogen, oxygen and sulfur atoms and forms a 5- or 6-membered aromatic ring together with the adjacent carbon atoms and A (the aromatic ring may contain one substituent, or two identical or different substituents, selected from the class consisting of halogen atoms, hydroxyl groups, lower alkyl groups and lower alkoxy groups); X and Y may be identical or different and each represents an oxygen atom, a sulfur atom, a carbonyl group, a group of the formula -CHR<a>- in which R<a> represents a hydrogen atom or a lower alkyl group, or a group of the formula -NR<b>- in which R<b> represents a hydrogen atom or a lower alkyl group, or when taken together, X and Y represent a vinylene or ethynylene group; R<1> represents a lower alkenyl group which may be substituted, a cycloalkenyl group which may be substituted, a lower alkynyl group which may be substituted, an aryl group which may be substituted, or a heterocyclic group which may be substituted; R<2> represents a hydrogen atom or a lower alkyl group; R<3> represents a hydrogen atom, a lower alkyl group, a lower alkenyl group, a lower alkynyl group or a cycloalkyl group; R<4> and R<5> may be identical or different and each represents a hydrogen atom or a halogen atom; and R<6> represents an acyclic hydrocarbon group which may be substituted (which may contain 1 or 2 unsaturated bonds selected from double and triple bonds); a cycloalkyl group which may be substituted, or a phenyl group which may be substituted; provided that when either one of X and Y represents an oxygen or sulfur atom, or the group -NR<b>- in which R<b> is as defined above, the other represents a carbonyl group or the group -CHR<a>- in which R<a> is as defined above, and a nontoxic salt thereof. The said compound is useful as pharmaceuticals, particularly for the treatment and prevention of hypercholesterolemia, hyperlipemia and arteriosclerosis.
Patent IL-89335-A (IL)
Title: 6-oxo-pyridazine derivatives, a process for their preparation and pharmaceutical compositions containing these compounds
IPC: C07D401/14
Filed: 1989-02-17
Abstract: Novel 6-oxopyridazine derivatives of the general formula I 
<IMAGE>
 which are novel positively inotropic compounds which have a higher, more selective, inotropism-enhancing activity. 
<??>A preparation process and the pharmaceutical use of these substances or of a medicament containing these substances are also described.
Patent IL-91518-A (IL)
Title: Antibiotic ge 2270, its preparation and pharmaceutical compositions containing it
Inventor: SELVA ENRICO
IPC: A61K35/66
Filed: 1989-09-04
Abstract: The present invention is directed to a new antibiotic substance denominated antibiotic GE 2270, by cultivating Planobispora rosea ATCC 53773 or a GE 2270 producing variant or mutant the addition salts thereof, the pharmaceutical compositions thereof and their use as medicaments, particularly in the treatment of infectious diseases involving microorganisms susceptible to them.
[EP0359062A2]
Patent IL-93485-A (IL)
Title: Tetrahydropyridines process for their preparation intermediates therefor compositions containing them and process for use of such compositions
IPC: A61K8/00
Filed: 1990-02-21
Abstract: The invention provides UV-absorbing compounds of formula (I), processes for preparing compounds of formula (I) and compositions, including sunscreens, containing compounds of formula (I), wherein A and B are alkyl, haloalkyl or together form a carbocyclic ring; R<1> is alkyl, haloalkyl, substituted alkyl where the substituent is selected from hydroxy, amino, alkoxy, alkanoyl, alkoxycarbonyl, phenyl and the radical of formula (I(a)), wherein A, B, R<2> and R<3> are as herein defined; alkenyl, cycloalkyl; phenyl; the groups phenyl and benzyl; said groups being substituted in the benzene ring by alkyl, alkenyl and alkoxy; and wherein R<1> and R<2> may form a carbocyclic ring; R<2> is hydrogen or alkyl; R<3> is alkyl, substituted alkyl, alkenyl, cycloalkyl and substituted benzyl; and the invention also provides for compounds of formula (VII); wherein A and B are methyl; R<2> is hydrogen; and R<3> is alkyl.
[WO9009995A1]
Patent IL-95452-A (IL)
Title: Bimetallic coin blank, particularly for coins and the like
IPC: A44C3/00
Filed: 1990-08-21
Abstract: A coin blank, particularly for minting of coins and the like, is formed by an external element (1) of metal or metal alloy having a central aperture, on the edge surface (4) of which are cut perimetrally a series of spaced grooves (5), and by an internal element (6), of metal or metal alloy different from the former, on the edge surface of which is formed a perimetral ridge (8,9), said external and internal elements being coupled inseparably during the minting operation through the plastic flow of the material from said perimetral ridge (8,9) into said grooves (5) in said external element (1) and through the firm fitting of the material from said ridge into the portions of the edge surface of said central aperture in said external element (6), provided between adjacent grooves (5).
Patent IL-97753-A (IL)
Title: 4-Quinolyl and 4-isoquinolyl-dihydropyridines, their preparation and pharmaceutical compositions containing them
IPC: A61P9/06
Filed: 1991-04-03
Abstract: Compounds of the general formula I 
<IMAGE>
 in which 
 
  R<1> and R<5> are identical or different and represent straight-chain or branched alkyl having up to 8 carbon atoms, 
  R<2> represents nitro or cyano, 
 or 
 
  R<1> and R<2> together form a lactone ring of the formula 
<IMAGE>
 
  R<3> represents a radical of the formula 
<IMAGE>
 in which 
 
  R<6> denotes hydrogen, halogen or straight-chain or branched alkyl or alkoxy each having up to 8 carbon atoms, 
  R<7> denotes optionally substituted aryl having 6 to 10 carbon atoms, or
 denotes thienyl or pyridyl, each of which is optionally substituted by halogen, 
  R<4> represents hydrogen, or straight-chain or branched alkyl, alkenyl, alkadienyl or alkynyl each having up to 10 carbon atoms, each of which is optionally monosubstituted or disubstituted by identical or different substituents from the series comprising halogen, hydroxyl, carboxyl, cyano, nitro and phenoxy or by straight-chain or branched alkylthio, alkoxy, alkoxycarbonyl, acyl or acyloxy each having up to 8 carbon atoms or by phenoxy or phenyl, where the latter can in turn be monosubstituted or disubstituted by identical or different halogen or by straight-chain or branched alkyl or alkoxy each having up to 6 carbon atoms 
 
 A process for their preparation and their use in medicaments, in particular in compositions having a positively inotropic action.
Patent IL-99195-A (IL)
Title: Process for enhancing the surface area of adsorbent aromatic copolymers
IPC: C08F2/18
Filed: 1991-08-15
Abstract: Highly crosslinked adsorbent copolymers are treated to enhance their surface area by reacting the copolymers in the presence of non-swelling liquid and Lewis-acid catalyst.
Patent JP-H11213342-A (JP)
Title: Magneto-resistance effect type magnetic head and its production
Inventor: KOMURO MATAHIRO
IPC: G11B5/39
Filed: 1998-01-22
Abstract: PROBLEM TO BE SOLVED: To provide a magneto-resistance effect magnetic head which has a high-precision track width by using a thin gap film of high film thickness precision, and its production. SOLUTION: In this magneto-resistance effect type magnetic head, upper and lower gap films 2 and 7 are provided between two shield films 8 and 10, and a magneto-resistance effect film 1 is provided between upper and lower gap films 2 and 7, and an electrode film 4 which causes a current to flow to this magneto-resistance effect film 1 is provided in electric contact with the magneto-resistance effect film 1. The electrode film 4 is provided so as to come into contact with both ends through the upper gap film 2 formed on the magneto-resistance effect film 1.
Patent JP-S61169099-A (JP)
Title: Ultrasonic transmitter-receiver
Inventor: TONE MASAYUKI
IPC: G10K11/02
Filed: 1985-01-22
Abstract: PURPOSE:To reduce the attenuation of ultrasonic waves by utilizing a high polymer film including air foams for the acoustic matching film and thereby making the density of the tone adjusting layer small. CONSTITUTION:On the main surface 11 of a piezoelectric vibrator 10 that transmits/receives ultrasonic waves, an acoustic matching layer made of the high polymer porous film 12 which incorporates holes 3 for matching acoustic impedance between the air that functions as an acoustic load and the surface. As the result of this constitution with the film 12 which does not utilize small hollow globes of compound materials, the density of the film can be made small, and also, scattering due to the said globes is prevented. Therefore, the attenuation of the ultrasonic waves are reduced.
Patent JP-S57124744-A (JP)
Title: Standard copy mode setter for copying machine
Inventor: UCHIDA HIROYASU
IPC: G03B27/00
Filed: 1981-01-28
Abstract: PURPOSE:To optimize an automatic return time in accordance with the situation of users, by providing a standard copy mode return time setting switch to a copying machine having a standard copy mode automatic return function. CONSTITUTION:A CPU1, an ROM2, an RAM3, an input board 4 and an output board 5 are mutually connected via a common bus 19, and they form a control section for a copying machine main body 15. On the other hand, the body 15 is provided with a standard copy mode setting switch 6 and a standard copy mode return time setting switch 7, which are connected to an input board 4. After the end of copying, when a time set to the switch 7 elapses, the mode returns to the standard copy mode automatically. Since the automatic return time can freely be selected like this, the automatic return time can be optimized according to the situation of users.
Patent JP-S61167618-A (JP)
Inventor: ASHIYOKU BUI KATODEERE
IPC: A61K9/20
Filed: 1986-01-22
Abstract: (57)【要約】本公報は電子出願前の出願データであるた め要約のデータは記録されません。
Patent JP-H07215571-A (JP)
Title: Sheet storing device
Inventor: SHINNO TATSUYA
IPC: B65H5/06
Filed: 1994-02-01
Abstract: PURPOSE:To form punch holes at accurate positions without affecting on the treatment speed of a copying machine main body and without applying excessive load onto a sheet transporting system in a sorter. CONSTITUTION:Pair of rollers 51, 52, 53, and 54 to transport the sheets delivered from a copying machine main body are provided inside a sorter 4, and a punch mechanism 60 to form punch holes in the sheets is provided immediately after the pair of rollers 52. Also an electromagnetic clutch is installed on a mechanism to transmit driving power to the pair of rollers 53 and 54 so as to turn on and off the transmission of the driving force. The electromagnetic clutch is turned on immediately before the rear end part of the sheets passes the pair of rollers 52 so as to stop the rotation of the pair of rollers 53 and 54. For the sheet S, its rear end part is transported by the pair of rollers 52, curved part S1 is formed, and the rear end is resisted by the pair of rollers 52. This time, the punch mechanism 60 is operated, and punch holes are formed in the sheets.
Patent JP-S60153535-A (JP)
Title: Computer
Inventor: ASAI NORIHIRO
IPC: G06F15/00
Filed: 1984-01-24
Abstract: PURPOSE:To operate a computer in accordance with a request without using a manual by arranging a liquid crystal display and function keys correspondingly on a keyboard. CONSTITUTION:If ''END'' is inputted from normal keys 2 except the function keys on the keyboard 1, the message of ''END'' is displayed on the liquid crystal display LCD3 and the messages of functions in the lower layers are displayed on respective peripheral edge display parts 31-3n. In addition, the message of ''END'' can be displayed on the LCD3 also by depressing function keys F1-F6 adjacent to the ''END'' of the commands displayed on the peripheral edge display parts of the LCD3. A ''HELP'' message is formed in a memory to provide the message with a retrieving function, so that a correct command name can be optionally retrieved is spite of uncertain storage by depressing a HELP key F6 in the function key.
Patent JP-H11212639-A (JP)
Title: Method and device for detecting malfunction in traveling controller for automatic traveling machine
Inventor: HATSUMOTO SHINTAROU
IPC: G05D1/02
Filed: 1998-01-22
Abstract: PROBLEM TO BE SOLVED: To detect a car body gets out of an operating route when an internal sensor is normal. SOLUTION: When traveling an automatic traveling machine 1, GAS position data are provided from a GAS satellite 100 by a controller 6, and correction data are provided from a fixed satellite 110 so that a current position under control is found as position finding data but when these position finding data are transmitted to a state monitoring device part 202, based on the transmitted information, this state monitoring device part 202 confirms and checks the position of the automatic traveling machine 1 in the specified area. Thus, since it is discriminated whether the automatic traveling machine 1 malfunctions or not, the malfunction of the automatic traveling machine 1 can exactly be detected even while the internal sensor of the automatic traveling machine 1 is normally operated. Further, since the automatic traveling machine 1 is stopped in the case of malfunction, the automatic traveling machine 1 can be prevent from working in the specified area while malfunctioning and not only erroneous work is eliminated but also no danger occurs as a result.
Patent JP-S60154911-A (JP)
Title: Fuel tank structure for automobile
Inventor: SATOU YOSHITAKA
IPC: B60K15/077
Filed: 1984-01-24
Abstract: PURPOSE:To aim at an increase in the measure of capacity, by separating a subtank to the opposite side from a gas-liquid separator, while fitly installing a pair of pipes into solidification in a higher position than a fulltank's full lever in time of a car body's maximum tilt as well as installing the subtank in the point midway in a connecting tube interposingly between a main tank and the gas-liquid separator. CONSTITUTION:When a car body M is tilted in a counterclockwise direction, a gas-liquid separator 16 is situated in a higher position than a full tank's full lever 24 as far as a position for H2 so that there is no fear of any outflow of fuel. Likewise, when it is tilted in a clockwise direction, a subtank 25 is installed in the point midway in a tube 21 and in a higher position than the said fuel level 24 as far as a portion for H2 interposingly, therefore even if there is any inflow of the fuel, its amount is as little as negligible whereby it is in no case reached to the subtank 25 further away, and what is more, no fear of its outflow. And, with fittedness between an inlet side 21A and an outlet side 21B of the tube 21, a tank is constituted into solidification, thus both detachment and assembling operations for the gas-liquid separator can be made so easily.
Patent JP-S5294128-A (JP)
Title: Exposure control systemfor flash shooting
Inventor: NAKAMURA ZENZOU
IPC: G03B7/16
Filed: 1976-02-04
Abstract: PURPOSE: To reduce the fluctuation of reference voltage and form a precise diaphragn control signal by energizing the reference voltage from the electric source to the flash means. 
     COPYRIGHT: (C)1977,JPO&Japio
Patent JP-S61171178-A (JP)
Title: Cryogenic coolant carrier
Inventor: KIMURA SHINICHI
IPC: F25B9/00
Filed: 1985-01-25
Abstract: PURPOSE:To obtain the titled apparatus which can largely reduce the time of e-cooling a liquid helium container or a superconductive device, by a method wherein a connecting pipe 17 moving up and down by the operation of an outer peripheral supporter is provided at the tip of a liquid-feeding pipe projecting inward the liquid-storing bath. CONSTITUTION:In order to pre-cool a liquid helium container inner bath 13, low-temperature gas helium evolved in a helium liquifier 1 is fed to the container inner bath 13 through the liquid-feeding pipe 3 of a helium carrier pipe 22. During this pre-cooling, the connecting pipe 17 is moved downward by loosing two caulking members 15; then, the carrier pipe 22 and an outer peripheral support pipe 18 are fixed by tightening said members 15. Such an operation enables low-temperature gas helium to be released through the connecting pipe 17 to the bottom of the inner bath 13 and to be returned after pre-cooling the whole inner bath 13, through a vent hole provide at a proper position of the pipe from a return pipe 4 18 to the helium liquifier 1. During liquid storing, the connecting pipe 17 is moved upward by the same operation, and the liquid should not be stirred even in a state of liquid accumulation; therefore, the liquid can be fed without boiling.