baber/WOPTO huggingface dataset:
Patent IL-70519-A0 (IL)
Title: Cephalosporin derivatives and a process for their preparation
IPC: A01N/
Filed: 1983-12-21
Abstract: For the Contracting States : BE, CH, DE, FR, GB, IT, LI, LU, NL, SE 1. Cephem derivatives of the general formula  see diagramm : EP0111935,P10,F1  and physiologically acceptable acid addition salts thereof in which R**1 denotes hydrogen, R**2 denotes hydrogen, R**3 denotes C1 -C4 -alkyl optionally substituted by fluorine, A denotes a quinolinium or an isoquinolinium radical, each of which can also be substituted once or twice by C1 -C4 -alkyl and in which the R**3O group is in the syn position. For the Contracting State : AT A process for the preparation of cephem derivatives of the general formula I  see diagramm : EP0111935,P11,F1  and physiologically acceptable acid addition salts thereof in which R**1 denotes hydrogen, R**2 denotes hydrogen, R**3 denotes C1 -C4 -alkyl optionally substituted by fluorine, A denotes a quinolinium or an isoquinolinium radical, each of which can also be substituted once or twice by C1 -C4 -alkyl and in which the R**3O group is in the syn position, which comprises a) reacting a compound of the general formula II  see diagramm : EP0111935,P11,F2  or salts thereof or a reactive derivative of the compound II in which R**1, R**2 and R**3 have the abovementioned meaning and R**8 denotes an amino group or a protected amino group and R**9 denotes a group which can be replaced by quinoline, isoquinoline or substituted quinolines or isoquinolines corresponding to the radicals A of the formula I, with quinoline, isoquinoline or one of their derivatives, and alpha) splitting off a protective group which is present where appropriate and beta) if necessary, converting the resulting product into a physiologically acceptable acid addition salt, or b) reacting a 7-aminocephen compound of the general formula III  see diagramm : EP0111935,P12,F3 or acid addition salts thereof in which R**2 and A have the abovementioned meaning, it also being possible for the amino group to be present in the form of a reactive derivative, with a 2-(2-aminothiazol-4-yl)-2-syn-oximinoacetic acid of the general formula IV  see diagramm : EP0111935,P12,F4 in which R**1, R**3 and R**8 have the above meaning, or with an activated derivative of this compound, and alpha) splitting off a protective group which is present where appropriate and beta) if necessary, converting the resulting product into a physiologically acceptable acid addition salt
Patent IL-73459-A0 (IL)
Title: Fiber optic directional coupler
IPC: G02F1/01
Filed: 1984-11-08
Abstract: A modal coupler, for coupling between modes of an optical fiber, such as between first and second order modes or between orthogonal polarization modes, comprises a single continuous strand of optical fiber (24), and a device (14) including a plurality of coupling surfaces (18) for applying stress to the optical fiber at spaced intervals along the fiber. The stress deforms the fiber and abruptly changes the fiber geometry at the beginning and end of each stressed region. The change in fiber geometry causes coupling of light from the fundamental mode to the second order mode or between polarization modes. Under certain conditions with nonbirefringent fiber the coupler exhibits polarization dependence, and thus, may be utilized as a fiber optic polarizer. In addition, the device couples coherently, and may be used in interferometric systems.
Patent IL-82550-A0 (IL)
Title: Spring coil and spring assembly
IPC: A47C27/06
Filed: 1987-05-17
Abstract: A spring coil (11) has an open-ended terminal convolution (11b, 11c) which is connected to the body (11a) of the coil through a gradient arm (20) which can be varied in length in manufacture to alter the spring compression and firmness. Offset portions (12, 13, 14) are formed on each terminal convolution with a major straight part (13a) which is outwardly spaced from minor straight parts (13c) for a three point engagement for the offset portion to a border wire (18). The offset portions (12, 14) have inside (25a) and outside (25b) shoulders adjacent their ends, with the pitch of joing cross-helicals (17) chosen so that a cross-helical simultaneously engages the outside shoulders of a pair of overlapped offset portions (12, 14). The spring rows are further arranged across the width of the mattress, with the columns extending along the length. Cross-helicals (28) can then be used across portions of the width for extra firmness for the entire mattress, or for selected areas, such as the middle third.
Patent IL-94592-A0 (IL)
Title: Heterocyclic compounds,their preparation and pharmaceutical compositions containing them
IPC: C07D498/04
Filed: 1990-06-01
Abstract: A heterocyclic compound represented by formula (I): <CHEM> and salts thereof, and intermediates therefor are disclosed. The compound of formula (I) and salts thereof exhibit selective serotonin 2-receptor antagonistic activity and are useful for the prevention or treatment of circulatory diseases, e.g., ischemic heart diseases, cerebral vessel disturbances, and peripheral circulation disturbances.
Patent IL-98109-A0 (IL)
Title: Oxalylamino acid derivatives,processes for their preparation and their use as medicaments for inhibiting proline hydroxylase
IPC: A61K31/395
Filed: 1991-05-10
Abstract: The invention relates to oxalylamino acid derivatives of the formula I  <IMAGE>  in which R and R' are identical or different and are C1-C6 -alkyl or hydrogen, R1 is hydrogen or C1-C4-alkyl, R2 is hydrogen, C1-C6-alkyl, C1-C3-alkoxy, carboxyl, C1-C6-alkoxycarbonyl, aryl, SH, NH2 or halogen, where the alkyl radicals are unsubstituted or substituted by aryl, OH, SH or NH2  or R1 and R2 together are a C2-C4-alkylene chain and the compounds in their predominantly pure D- and L-form and the physiologically tolerable salts. The compounds are distinguished as excellent inhibitors of prolyl hydroxylase and lysine hydroxylase.
Patent IL-99683-A0 (IL)
Title: Hydroxy alkylquinoline ether acids and pharmaceutical compositions containing them
IPC: A61P9/00
Filed: 1991-10-09
Abstract: Compounds having the formula I: <CHEM> are leukotriene antagonists and inhibitors of leukotriene biosynthesis. These compounds are useful as anti-asthmatic, anti-allergic, anti-inflammatory, and cytoprotective agents. They are also useful in treating angina, cerebral spasm, glomerular nephritis, hepatitis, endotoxemia, uveitis, and allograft rejection.
Patent IL-125475-A0 (IL)
Title: Process and device for determining an analyte contained in a scattering matrix
IPC: A61B5/00
Filed: 1997-01-23
Abstract: PCT No. PCT/DE97/00168 Sec. 371 Date Jul. 28, 1997 Sec. 102(e) Date Jul. 28, 1997 PCT Filed Jan. 23, 1997 PCT Pub. No. WO97/27469 PCT Pub. Date Jul. 31, 1997Method for determining an analyte in a scattering matrix. In a detection step detection measurements are made in which light is irradiated into the matrix as primary light and light leaving the scattering matrix is detected as secondary light, in order to determine as a measurement quantity a measurable physical property of the light which is variable due to the interaction of the light with the matrix. Information on the presence of the analyte in the matrix is determined in an evaluation step. The determination of optically weakly absorbing analytes against a strongly absorbing interference background is improved by the use of two selection methods for the depth selective detection of the secondary light in combination with one another. Primary light is focused by means of a primary light optically focussing element onto a region of focus lying in the matrix at a predetermined measuring depth and the region of focus is imaged by means of a secondary light optically focusing element onto a light entry aperture arranged in the light path of the secondary light to the detector. In addition to this first depth selection by a confocal arrangement, a second depth selection device is used to detect light reflected from a defined measuring depth as secondary light, with the measuring depth coinciding with the depth of focus.
Patent IL-125982-A0 (IL)
Title: 2-(arylphenyl) amino-imidazoline derivatives
IPC: C07D401/12
Filed: 1998-08-28
Abstract: The invention relates to IP receptor antagonists selected from the group of compounds represented by formula <CHEM>  wherein     R<1> is a group represented by formula (A), (B) or (C): <CHEM> and other substituents as defined in the specification, and their pharmaceutically acceptable salts, crystal forms therof and pharmaceutical compositions containing them.
Patent IL-129332-A0 (IL)
Title: suPAR STIMULATING ACTIVITY OF tcuPA-MEDIATED FIBRINOLYSIS AND DIFFERENT USES THEREOF
IPC: A61P9/10
Filed: 1999-04-05
Abstract: The present invention relates to a complex (tcuPA/suPAR) of the two chain urokinase plasminogen activator (tcuPA) with the soluble urokinase plasminogen activator (suPAR), to pharmaceutical compositions comprising this complex and to different uses of the compositions in the treatment and/or prevention of thrombotic events, particularly those associated with the formation of fibrin clots. In the complex (tcuPA/suPAR), the suPAR stimulates firbrinolytic activity mediated by tcuPA under physiological conditions. The complex acts preferably on freshly-formed clots and is specific to such clots.
Patent IL-134641-A0 (IL)
Title: No-spill drinking cup apparatus
IPC: B65D51/16
Filed: 1998-08-21
Abstract: An improved no-spill cup construction and valve assembly which provides an extremely secure seal against accidental liquid flow from the cup spout. The act of sucking at the cup spout creates negative pressure or a partial vacuum against a valve near the spout, causing the valve to invert which unblocks an opening in the valve. When the opening is unblocked, liquid can flow freely through the valve and spout. When not in use, the valve sits in a resting, closed position, with the valve pressed against a center seal-off, sealing off the opening in the valve assembly. The closed position provides an extremely secure seal against fluid leakage, such that inadvertent spills or even deliberate attempts to force liquid outside of the cup, such as by turning the cup upside down, or shaking the cup, are ineffective. The cup assembly further allows liquid flow to be regulated between regular or maximum flow and minimal flow levels or rates by rotating the position of the valve assembly in the cover of the cup.
Patent IL-138170-A0 (IL)
Title: Counter top paper towel holder
IPC: A47G/
Filed: 2000-08-30
Abstract: A counter-top paper towel holder (10) having a base (18), a mounting rod (20) extending upward from the base, and a stabilizing extension (26) extending upward from the base at a position radially spaced from the mounting rod. The stabilizing extension (26) includes a handle portion (28) and a presser arm (32) spaced radially outward from the handle potion. The presser arm (32) is resilient, and includes a free end for abutting the roll of paper towels mounted on the mounting rod. Grasping the handle with one hand provides support for the paper towel holder against gross movement as the free towels are pulled from the roll using the other hand. The thumb of the grasping hand may press against the presser arm to force the free end against the roll. The free end thus prevent further rotation of the roll, and assists in breaking the lines of perforation to dispense the towels. <IMAGE>
Patent IL-141161-A0 (IL)
Title: Synthesis of acyclic nucleoside derivatives
IPC: C07D473/18
Filed: 1999-08-05
Abstract: A process for preparing a compound of the formula: <CHEM> wherein R10 is a C3-C21 saturated or monounsaturated, optionally substituted alkyl residue, the process comprising the steps of:  a) reacting a compound of the formula: <CHEM> wherein R6 and R7 are lower alkyl or benzyl residues, or R6 and R7 taken together are -CH2CH2-, -CH2CH2CH2- or -CH2CH2CH2CH2- with R10COOH or an activated derivative thereof, wherein R10 is a C3-C21 saturated or monounsaturated, optionally substituted alkyl residue, to provide a compound of the formula: <CHEM> wherein R6, R7 and R10 are defined as above, b) de-protecting the acetal of the product of step a), and c) reducing the aldehyde substituent of the product of step b),  characterized in that the products of steps a) and b) are not isolated.
Patent IL-146082-A0 (IL)
Title: Treatment of fibrosis by antagonism of il-13 and il-13 receptor chains
IPC: A61P1/16
Filed: 2000-04-28
Abstract: Methods are provided for treating or inhibiting the formation of tissue fibrosis using IL-13 antagonists, including without limitation soluble forms of the IL-13 receptor.
Patent IL-158210-A0 (IL)
Title: Propellant and a method and device for producing the same
IPC: C06B45/00
Filed: 2002-03-28
Abstract: The present invention relates to a method and a device for producing perforated propellant in the geometric form of block, stick, slab, cylindrical or tubular propellant (2) with high charge density and high progressivity. The propellant as claimed in the present invention is characterised by a large number of perforations, densely and evenly distributed over the entire propellant segments, made by perforation members (6) that are pressed down into the propellant. The perforations are thereby made in a plurality of steps with a predetermined step feed between each perforation operation. The device as claimed in the present invention also comprises a mobile pin die (5) away from but facing the feed path (1) for the propellant (2), and containing at least one row of pins for perforation of the propellant whereby each such row of pins comprises the number of pins (6) required to cover the complete width of the propellant segment across its direction of advance. Between each perforation operation the propellant is step fed by a step feed device (15) a distance equivalent to the distance between two desired perforations multiplied by the number of rows of pins arranged across the direction of advance of the propellant. Additionally, in the propellant as claimed in the present invention the distance between two burning surfaces of the propellant shall be equal to double the desired burning length (2b).
Patent IL-220131-A0 (IL)
Title: Cloning and expression of biologically active alpha- galactosidase a
IPC: C12N15/54
Filed: 1993-11-30
Abstract: The present invention discloses a method for producing a secreted biologically active mature ±-galactosidase A that contains ±2,6-sialic acid residues, comprising culturing an engineered mammalian cell that expresses ±-galactoside ±2,6-sialyltransferase such that the cell is capable of peptide sialylation, wherein the cell further comprises a nucleotide sequence that regulates gene expression operatively associated with an ±-galactosidase A gene sequence under conditions in which the ±-galactosidase A is sufficiently overexpressed by the engineered mammalian cell so as to be selectively secreted into the mammalian cell culture as a biologically active mature ±-galactosidase A that contains ±2,6-sialic acid residues; and isolating biologically active mature ±-galactosidase A that contains ±2,6-sialic acid residues from the mammalian cell culture.
Patent BE-1015434-A0 (BE)
Title: Anti-theft device for motor vehicle, has capacitive sensor for reading and recognizing internal finger prints of skin i.e. between skin and flesh, of driver to verify whether driver is authorized to use vehicle
Inventor: SAGNIER JOSEPH
IPC: B60R25/00
Filed: 2003-02-27
Abstract: The device has an AFS 8500 type capacitive sensor (2) for reading and recognizing internal finger prints of skin i.e. between skin and flesh, of a driver to verify whether the driver is authorized to use a vehicle. An acceptance signal is sent towards a central processing unit (8) of a computer, if the driver is authorized, to activate an engine or to open the door of the vehicle.
Patent RO-128165-A0 (RO)
Title: Process for making telephone subway ducts in highways
Inventor: NICULICEA SANDU
IPC: G02B6/50
Filed: 2012-08-17
Abstract: The invention relates to a process for making telephone subway ducts servicing highways. According to the invention, the process comprises a telephone duct site embedded in the highway body (), at the border of the emergency lane, in the vicinity of a protection fence (), which is physically made by machining a vertical channel into the body of the practicable road (), at the border of the emergency lane, said vertical mini trench () of a certain width () and depth (), being meant for some single tubes () to be laid as a support wherein the fiber optics and electric cables will be installed, after which the rest of the space existing in the mini trench () is filled with concrete or asphalt, depending on the composition of the practicable road ().
Patent MC-2207-A1 (MC)
Inventor: TAKATOSHI TAKEMOTO
IPC: A63F7/02
Filed: 1991-10-04
Abstract: The apparatus of the invention includes folded transmission lines (22) for sending a current for generating a magnetic field, and folded reception lines (26) disposed at a position at which they can electromagnetically couple with the transmission lines (22), for detecting the change of the magnetic flux due to the approach of a metal. The transmission lines (22) are disposed on a first plane, and the reception lines (26) are disposed on a second plane in parallel with the first plane in such a manner that the transmission lines are perpendicular to the reception lines in order to constitute a detection matrix (20).The detection matrix (20) is disposed on a panel surface, along which a metallic member to be detected moves, in such a manner as to oppose each other while keeping at least a space through which the metallic member can pass. Transmission means (50) and reception means (40) are connected to the detection matrices (20) so as to detect the existing position of the metallic member. <IMAGE>
Patent LU-82671-A1 (LU)
Inventor: HURST R
IPC: C09C1/50
Filed: 1980-07-30
Abstract: This disclosure relates to an improved furnace process for producing carbon blacks by the incomplete combustion of hydrocarbonaceous feedstock wherein the resultant blacks have higher surface areas than the carbon blacks normally prepared from the feedstocks, as a result of which the blacks are particularly suitable for use in imparting conductivity properites to plastic materials and the like. This disclosure also relates to the production of a novel class of furnace blacks having excellent conductivity properites and which are characterized by high surface areas and low pH values.
Patent MA-52331-A1 (MA)
Title: Macrocycles à groupes hétérocycliques p2' servant d'inhibiteurs du facteur xia
Inventor: ORWAT MICHAEL J
IPC: C07D471/08
Filed: 2015-01-30
Abstract: La présente invention concerne des composés de formule (i) ou des stéréo-isomères, des tautomères ou des sels de qualité pharmaceutique de ceux-ci. Dans ladite formule, toutes les variables ont la signification indiquée dans la description. Ces composés sont des inhibiteurs sélectifs du facteur xia ou des inhibiteurs doubles de fxia et de la kallicréine du plasma. Cette invention concerne également des compositions pharmaceutiques comportant ces composés et des méthodes pour traiter des troubles thrombo-emboliques et/ou inflammatoires à l'aide de celles-ci.
Patent UY-23219-A1 (UY)
Title: Recipiente para almacenar y distribuir articulos
Inventor: K J PIETER DECOSTER
IPC: B65D81/26
Filed: 1991-05-07
Abstract: Receptáculo con nervaduras de guía internas (28) que se extienden verticalmente, las cuales terminan en resaltos de soportes superiores (30) en una relación espaciada hacia abajo al extremo superior abierto del receptáculo. Un inserto (16) se monta para el deslizamiento vertical dentro del receptáculo e incluye una charola de fondo (32) que tiene rebajos (34) en puntos espaciados periféricamente, que corresponden a la posición de las nervaduras de guía. Los rebajos complementan las nervaduras para la guía vertical no rotacional del inserto. La charola, arriba de los resaltos, gira para el asentamiento sobre los resaltos. La figura 1 ilustra la presente invención.
Patent UY-23957-A1 (UY)
Title: Sistema inteligente de modulos electro-computarizados para identificacion de infractores a la ordenanza de transito
IPC: G08G1/07
Filed: 1995-05-02
Abstract: Se describe un sistema inteligente de módulos electro-computarizados para identificación de infractores a la ordenanza de tránsito que permite registrar interrumpidamente el flujo de tránsito, censar sistematicamente la velocidad de todos los vehículos infractores y registrar los vehículos infractores, con la posibilidad de anunciar a los conductores el estado de legalidad o ilegalidad de sus maniobras o conducción, caracterizado por consistir de elementos en los puntos de fiscalización, que son aparatos incorporados en columnas, dispositivos colgantes o en carteles indicadores, que están vinculados a una red con un programa central que dirige y colecta las informaciones. Los puntos de fiscalización están constituidos por un núcleo o comando central, constituido por un sistema computarizado autónomo, un sistema sensor para identificar al infractor, una cámara para registración del infractor, una interfase para comunicación de datos al programa central, un sistema de abastecimiento y almacenamiento energético, una interfase para conexión de periféricos para ingreso y egreso de datos y, opcionalmente, sistemas de advertencia in-situ al conductor infractor. El programa central consiste en un nodo de red que está constituido por un sistema central de administración y procesamiento, unidades interfases para comunicación con los puntos de fiscalización y periféricos de salida de resultados para el control e impresión de reportes, fotografías, etc.
Patent UY-30429-A1 (UY)
Title: Vida util y estabilizacion en la semilla mejoradas de inoculantes bacterianos liquidos
Inventor: YANG GUOPING
IPC: A01N63/27
Filed: 2007-06-21
Abstract: La presente invencion incluye un método para producir un inoculante líquido que contiene un desecante. El método puede mejorar la supervivencia y estabilidad de bacterias en inoculantes líquidos en envase o en semillas. El método incluye proporcionar un inoculante líquido de una bacteria cultivada a una fase sustancialmente estacionaria. Se anade un tratamiento desecante que contiene un desecante al inoculante líquido para formar un producto inoculante parcialmente desecado. El producto inoculante parcialmente desecado puede envasarse y almacenarse. El producto inoculante parcialmente desecado también puede aplicarse a las semillas.
Patent UY-31592-A1 (UY)
Title: Compuestos de n-fenil-imidazo[1,2-a]piridin-2-carboxamidas, su preparacion y su aplicacion en terapéutica
Inventor: JEAN-FRANCOIS PEYRONEL
IPC: A61K31/165
Filed: 2008-12-30
Abstract: COMPUESTOS DE N-FENIL-IMIDAZO[1,2-a]PIRIDIN-2-CARBOXAMIDAS de formula (I) en el estado de vase o de sal de adision a un ácido, en la que los sustituyentes y los índices son segun están especificados en la Memoria descriptiva y en las reveindicaciones. Se divulga los métodos de preparacion, la de los intermediarios y su aplicacion en el tratamiento o prevencion de enfermedades que implican los receptorea nucleares Nurr-1 denominados NR4A2, NOT, TINUR, RNR-1 y HZF3.
Patent ES-178456-A1 (ES)
Title: Sistema de radio-ruta de planeo para sistemas de radioaterrizaje a ciegas
IPC: G01S1/02
Filed: 1947-06-14
Abstract: Un sistema de radio-ruta de planeo para aeronaves de la clase en que la ruta de planeo es una línea de intensidades de campo de relación constante producida por las partes solapadas de dos campos radiados contenidos en un plano vertical caracterizado en que uno o ambos de los orígenes de dichos campos está o están desplazados en el plano horizontal de la línea de intersección de dicho plano vertical con el plano horizontal y las características de radiación tienen tal forma una con respecto a la otra que dicha línea de intensidades de campo de relación constante se acerca al terreno en un punto alejado de los orígenes de los dos campos o características de campo.