baber/WOPTO huggingface dataset:
Patent CZ-20002112-A3 (CZ)
Title: Anti-arrhythmic compounds
Inventor: PAPP GYULA
IPC: A61K31/135
Filed: 1998-12-10
Abstract: The present invention relates to phenoxyalkylamino derivatives of the general formula I, in which Re1 and Re2 represent independently on each another a hydrogen atom, a halogen atom or an alkyl group containing 1 to 4 carbon atoms; Re3, Re4 and Re5 denote independently on each other a hydrogen atom or an alkyl group having 1 to 4 carbon atoms; Re6 represents a hydrogen atom, an alkyl group containing 1 to 4 carbon atoms or a benzyl group; Re7 denotes a nitro group or an amino group, being optionally monosubstituted with alkyl group having 1 to 4 carbon atoms, a benzoyl group, an alkylcarbonyl group containing 1 to 4 carbon atoms, an alkylsulfonyl group containing 1 to 4 carbon atoms, an alkylcarbamoyl group containing 1 to 4 carbon atoms or an alkylthiocarbamoyl group having 1 to 4 carbon atoms; both the n and m are 0 or 1; with the proviso, that Re2 differs from the hydrogen atom provided Re1 is a hydrogen atom, and their stereoisomers or stereoisomer mixtures, acid addition salts and hydrates, precursors and metabolites of all the above-indicated compounds. Disclosed are also pharmaceutical compositions containing the above-described compounds wherein these compounds exhibit a valuable antiarrhythmic activity.
Patent CZ-20004460-A3 (CZ)
Title: Pigment dispersant, process of its preparation, pigment preparation and its use
Inventor: WEBER JOACHIM DR
IPC: C09K23/32
Filed: 2000-11-30
Abstract: Pigment dispersant comprises a 1,4-diketo-3,6-di-(4-biphenyl)-pyrrolo(3,4-c)pyrrole with sulfonamide and optionally sulfonic acid or salt groups. Pigment dispersant comprises a 1,4-diketo-3,6-di-(4-biphenyl)-pyrrolo(3,4-c)pyrrole with sulfonamide and optionally sulfonic acid or salt groups of the formula (I). Q = 1,4-diketo-3,6-di-(4-biphenyl)-pyrrolo(3,4-c)pyrrole group; s = 0.1-4.0; n = 0-2; E<+> = hydrogen (H<+>) cation, the equivalent Mm+/m of a main group 1-5 or sub-group 1, 2 or 4-8 metal cation Mm+ or a (substituted) ammonium cation; Z = Z<1> or Z<4>; Z<1> = -(X-Y)qR<3>; X = (substituted) 2-6 carbon (C) alkylene and/or 5-7 C cycloalkylene;   Y = oxygen, piperazin-1,4-diyl and/or -NR<2>. The full definitions are given in DEFINITIONS. Independent claims are also included for: (a) pigment formulations containing organic basic pigment(s) and dispersant(s) (I); (b) pigment preparations consisting of organic basic pigment(s), dispersant(s) (I) and a high-molecular organic material; (c) the preparation of (I); and (d) the preparation of the pigment formulations.
Patent CZ-20011541-A3 (CZ)
Title: Process for preparing particle suspension
Inventor: BERNINI EVA
IPC: A61K9/72
Filed: 1999-10-28
Abstract: The invention is directed to a process for the preparation of suspensions of drug particles for inhalation delivery, said process providing particles of optimised particle size and distribution homogeneously dispersed in the carrier.  The process, which is also suitable for the preparation of sterile suspensions, includes the step of homogenising and micronising the formulation in a turboemulsifier provided with a high-potency turbine, optionally followed by a treatment in a high-pressure homogeniser.  A further aspect of the invention is directed to a process for preparing micronised sterile beclomethasone dipropionate by gamma-irradiation.
Patent CZ-20012662-A3 (CZ)
Title: Medicament for treating symptoms of weaning away from smoking
Inventor: MENDEL CARL M
IPC: A61P25/34
Filed: 2000-01-19
Abstract: This invention relates to a method to aid smoking cessation by treating a patient who wishes to stop smoking with an effective amount of a compound, in particular a phenylcyclobutylbutylamine, in order to aid the patient in overcoming the craving following smoking cessation. The method relates to preventing weight gain in a patient who ceases to smoke and optionally is using a nicotine patch or other agent or program to aid in ceasing to smoke.
Patent CZ-20012839-A3 (CZ)
Title: Device for measuring surface contamination with particles
Inventor: WOODMANSEE DONALD ERNEST
IPC: G01N1/04
Filed: 2001-08-03
Abstract: An apparatus (10) for measuring surface particulate contamination includes a tool (12,112) for collecting a contamination sample from a target surface, a mask (16) having an opening (28) of known area formed therein for defining the target surface, and a flexible connector (18) connecting the tool (12,112) to the mask (16). The tool (12,112) includes a body portion (13,113) having a large diameter section (20,120) defining a surface (22,122) and a small diameter section (24,124) extending from the large diameter section (20,120). A particulate collector (14) is removably mounted on the surface (22,122) of the large diameter section (20,120) for collecting the contaminants. The tool (12,112) further includes a spindle (30) extending from the small diameter section (24,124) and a spool (32) slidingly mounted on the spindle (30). A spring (34) is disposed between the small diameter section (24,124) and the spool (32) for biasing the spool (32) away from the small diameter section (24,124). An indicator (36) is provided on the spindle (30) so as to be revealed when the spool (32) is pressed downward to compress the spring (34). <IMAGE> <IMAGE>
Patent CZ-20013799-A3 (CZ)
Title: Novel therapeutic preparation
Inventor: BLACKLER PAUL DAVID JAMES
IPC: A61K31/00
Filed: 2000-04-19
Abstract: A polymorphic form of 5-Ä4-Ä2-(N-methyl-N-(2-pyridyl)amino)ethoxyÜbenzylÜthiazolidine-2,4-di one, maleic acid salt (the "Polymorph") characterised in that it:   (i) provides an infra red spectrum containing peaks at 1360, 1326, 1241, 714 and 669 cm<-1>; and/or (ii) provides a Raman spectrum containing peaks at 1581, 768, 670, 271 and 226 cm<-1>; and/or (iii) provides a solid-state nuclear magnetic resonance spectrum containing peaks at chemical shifts substantially as set out in Table I; and/or (iv) provides an X-ray powder diffraction (XRPD) pattern containing peaks substantially as set out in Table II; a process for preparing such a compound, a pharmaceutical composition containing such a compound and the use of such a compund in medicine.
Patent CZ-20021806-A3 (CZ)
Title: Lead, silver, and barium alloy for lead acid battery grids
Inventor: VAZQUEZ DEL MERCADO LUIS FRANC
IPC: H01M4/68
Filed: 2002-05-24
Abstract: A lead alloy for lead acid-battery grids which essentially consists of about 0.05-0.07 wt % calcium; about 0.09-1.3 wt % tin; about 0.006-0.010 %silver; about 0.0100-0.0170 wt% barium and about 0.015-0.025 wt% aluminum with the balance lead. This lead alloy allows the improvement of the age hardening step, by eliminating the high temperature treatment process required for silver alloys in the manufacturing of lead-acid batteries. By using this lead alloy, a longer service life of the lead-acid batteries are also obtained by increasing the corrosion resistance and the mechanical strength of battery grids manufactured by the book molding process. Additionally, the reduced silver level used dramatically mitigates the problem of silver elimination from the stream of recycled lead in the secondary production of this metal. <IMAGE>
Patent CZ-20023496-A3 (CZ)
Title: Receptor modulators for parathyroid glands hormone and protein related to the parathyroid glands hormone
Inventor: KOSTENUIK PAUL
IPC: A61K47/48
Filed: 2001-04-27
Abstract: The present invention concerns therapeutic agents that modulate the activity of PTH and PTHrP. In accordance with the present invention, modulators of PTH and PTHrP comprise: (a) a PTH/PTHrP modulating domain; and (b) a vehicle, such as a polymer (e.g. PEG or dextran) or an Fc domain, which is preferred; wherein the vehicle is covalently attached to the C-terminus of the PTH/PTHrP modulating domain. The vehicle and the PTH/PTHrP modulating domain may be linked through the N- or C-terminus of the PTH/PTHrP modulating domain, as described further below. The preferred vehicle is an Fc domain, and the preferred Fc domain is an IgG Fc domain. Preferred PTH/PTHrP modulating domains comprise the PTH and PTHrP-derived amino acid sequences described hereinafter. Other PTH/PTHrP modulating domains can be generated by phage display, RNA-peptide screening and the other techniques mentioned herein. Such peptides typically will be modulators of both PTH activity and PTHrP activity, although such techniques can be used to generate peptide sequences that serve as selective modulators (e.g., agonists of PTH activity but not PTHrP activity).
Patent CZ-20031815-A3 (CZ)
Title: Sulfamidothienopyrimidine derivative, process of its preparation, use thereof and pharmaceutical preparations in which the derivative is comprised
Inventor: EGGENWEILER HANS-MICHAEL
IPC: A61P19/00
Filed: 2001-12-03
Abstract: The invention relates to compounds of formula (I) wherein R<1>, E<2> and X have the designation cited in the description.
Patent CZ-20033438-A3 (CZ)
Title: Methods for inducing cytotoxic immune reaction and preparations of recombinant monkeyÆs adenovirus, which are usable in these methods
Inventor: ERTL HILDEGUND C J
IPC: C12Q1/70
Filed: 2002-05-13
Abstract: A method of inducing a CD8+ T-cell response against a selected molecule by delivering the molecule via a recombinant simian adenovirus is provided. Also provided are methods of inducing interferon-alpha and interferon-beta by delivering a recombinant simian adenovirus to a subject. The methods of the invention are particularly well suited for prophylaxis and treatment of infections with human immunodeficiency virus and human papilloma virus, among others, and cancer therapy.
Patent CZ-20131033-A3 (CZ)
Inventor: Soukup Viktor
IPC: G08G5/00
Filed: 2013-12-19
Abstract: ﻿Způsob monitorování leteckého hluku s přiřazením identifikované akustické události konkrétnímu letadlu spočívá v tom, že aktuálně snímaná akustická situace daná hladinou akustického tlaku, která je kvantifikovaná některým ze sledovaných akustických deskriptorů (např. LAmax, LAeq, LAE, apod.) v rámci akustického monitorování leteckého provozu v okolí letišť v okamžiku průletu konkrétního letounu v blízkosti měřicího monitorovacího stanoviště automaticky přiradí k přijatému a dekódovanému signálu o aktuální poloze příslušného letounu. Akustická situace se snímá pomocí zvukoměrného zařízení. Přiřazení dat o identifikaci, poloze konkrétního letadla a o naměřené hladině akustického tlaku se provádí přímo v dané měřicí monitorovací stanici, která zaznamenala akustický signál od prolétávajícího letadla. Data a signály jsou přiřazovány pomocí synchronizace času. Tento signál obsahuje časové a identifikační údaje o tomto letadle a je průběžně vytvářen a vysílán palubním navigačním systémem letounu na základě zpracování zaznamenaného signálu ze satelitního navigačního systému. V hlukové monitorovací stanici jsou data o skutečné poloze letounu porovnána s povolenými letovými postupy v daném místě umístění monitorovací stanice, včetně zohlednění povolených odchylek a povolených hodnot hladin akustického tlaku v konkrétním místě monitorováni hluku. Následně po vyhodnocení nastavených kritérií uložených v dané monitorovací stanici a dat o skutečné poloze a hlukovém stavu letounu v daném okamžiku, či předpokládaném dalším letovém postupu letounu, je vyslána informace z daného monitorovacího bodu o případném nedodržení letových postupů, či nedodržení hlukové kvóty s případnou výstrahou zpět určena a na palubu letounu a/nebo výstupní prezentační zařízení letiště. Dále se vynález týká zařízení k provádění tohoto způsobu.
Patent DD-230988-A3 (DD)
Title: Keramischer ferritkopf
Inventor: KODZABASEV PETKO V
IPC: G11B5/133
Filed: 1981-09-21
Abstract: Die Erfindung betrifft einen keramischen Ferritkopf fuer Magnetplattenspeicher, einsetzbar in der Rechentechnik. Aufgabe der Erfindung ist es einen keramischen Ferritkopf zu schaffen, der eine erhoehte Dichte und Zuverlaessigkeit beim Aufzeichnen und beim Lesen von Digitalinformationen aufweist. Diese Aufgabe wird durch einen Ferritkopf geloest, bestehend aus einem kompletten Magnetleiter, der aus einem Aufzeichen- und Lesemagnetleiter, der mit einer Spule versehen ist, und zwei loeschenden Tunnelmagnetleitern, versehen mit einer zweiten Spule sowie aus zwei keramischen Stuetzplatten aufgebaut ist. Der komplette Magnetleiter ist in einer stirnseitigen Oeffnung eines Gehaeuses fest angebracht, wobei an die Rueckseite des Gehaeuses die Spulenenden geleitet sind. Der komplette Magnetleiter ist an Masse angebracht. Die Rueckseite des Gehaeuses ist durch einen Deckel verschlossen, welcher, wie auch das Gehaeuse aus magnetisch weichem Ferrit ausgefuehrt ist, dessen linearer Dehnungskoeffizient dem linearen Dehnungskoeffizienten des kompletten Magnetleiters gleich ist. Der Deckel ist am Gehaeuse mittels eines stromleitenden Harzes angebracht. Der komplette Magnetleiter ist in die stirnseitige Oeffnung des Gehaeuses durch eine Niedertemperatur-Glasverschweissungbefestigt, deren linearer Dehnungskoeffizient dem linearen Dehnungskoeffizienten des kompletten Magnetleiters und des Gehaeuses gleich ist. Die Spulenenden sind auf den Gehaeusedeckel durch eine an demselben starr befestige Anschlussplatte geleitet, wobei der komplette Magnetleiter ebenfalls durch diese Platte geerdet ist. Die Innenflaeche des Gehaeuses ist mit einer stromleitenden, durch Anschlussplatte geerdeten Schicht ueberzogen. Die Vorteile des erfindungsgemaessen keramischen Ferritkopfes sind die erhoehte Dichte und Zuverlaessigkeit beim Aufzeichnen und Lesen von Digitalinformationen.
Patent DD-226733-A3 (DD)
Title: Doppelschalige wand
Inventor: FERNAU ULRICH
IPC: G01N3/12
Filed: 1982-12-16
Abstract: Die Erfindung betrifft eine doppelschalige Wand, vorzugsweise fuer temperatur- und druckbeanspruchte Behaelter, wie Oel- und Gasbehaelter, sowie Sicherheitsbehaelter fuer Kernenergieanlagen. Ziel der Erfindung ist es, die Wand einer doppelschaligen Behaelterwand so auszubilden, dass eine Konzentration der Biege-, Normal- und Zwaengungsspannungen in bestimmten Bereichen ausgeschlossen ist. Erfindungsgemaess wird das dadurch erreicht, dass die aus kraftschluessig miteinander verbundenen Schalen gebildete doppelschalige Wand im mittleren Bereich der temperaturbelasteten inneren Schale horizontale, ringfoermig die Schale umlaufende Dehnungsausgleicher und am Uebergang der Zylinderwand zur Grundplatte oder zum Behaelterdach vertikale Dehnungsausgleicher angeordnet sind. Die horizontalen Dehnungsausgleicher sind vorzugsweise im Stossbereich der aus ringfoermigen Segmenten gefertigten Behaelter angeordnet. Die Laenge der vertikalen Dehnungsausgleicher entspricht maximal dem Abstand benachbarter horizontaler Dehnungsausgleicher. Die Dehnungsausgleicher sind kammerbildend, die Naht der inneren Schale gasdicht umschliessend, angeordnet.
Patent EP-1033824-A3 (EP)
Inventor: SHOJI TAKASHI
IPC: H04J13/00
Filed: 2000-02-29
Abstract: A CDMA receiver which is capable of decreasing the control delay
of the closed-loop power control is provided to be used for a code
division multiple access system. The CDMA receiver comprises a maximum
correlation detector and a de-spreading part for obtaining original
information signals from received signals which have been spread by
a code for transmission. The maximum correlation detector detects a
maximum correlation value among mutual correlations between a received
replica signal and a received signal, calculates a time lag between
the received replica signal and the received signal having the the
maximum correlation value. The de-spreading part performs de-spreading
the received signal by using the reception timing obtained
by the maximum correlation detector and outputting the de-spread .
In addition to these elements, the CDMA receiver is provided with a
reception quality measurement part, which measures a received signal
to interference ratio (SIR) as a reception quality of the received
signal from the received signal and the maximum correlation value
obtained by the maximum correlation detector at the same timing as
the de-spreading part is performing its operation.
Patent EP-1087149-A3 (EP)
Inventor: TAKASHI KATO
IPC: F16B35/04
Filed: 2000-07-26
Abstract: The object of the present invention is to prevent the
encroaching and the seizure between the bolt and the female
screw caused by an oblique screwing of the bolt into the
female screw when the bolt and the female screw are fastened
together. Another object of the present invention is to
manufacture the bolt in a low cost, by using said bolt, the
encroaching and the seizure between the bolt and the female
screw caused by a oblique screwing of the bolt into the
female screw are certainly prevented. Said objects may be
attained by a bolt consisting of a column part and a polygonal
pillar part extending from an end of said column part wherein
a complete thread is formed on said column part and a screw
blade continuing to said complete thread is formed on said
polygonal pillar part.
Patent EP-1069396-A3 (EP)
Inventor: SAEKI AKITOMO
IPC: G01B3/18
Filed: 2000-07-12
Abstract: A micrometer (1) has second vernier numeral (91C) on an outer
circumference of a thimble (61) along circumferential direction and a vernier
scale (91A) on an inner circumference of the thimble (61) along
circumferential direction, the thimble (61) being made of a translucent
material, so that read error during measurement can be reduced.
Patent EP-1075827-A3 (EP)
Inventor: HIMMELSBACH PETER
IPC: A61F13/00
Filed: 2000-07-26
Abstract: Self-adhesive molding comprising adhesive foam high recovery forces, and optional transdermal agent, where adhesion is 1-25 N/cm, expansibility over 10%, thickness greater than 0.5 mm and recovery is more that 50% with tensile stressing of 5N/cm<2>, is new.
Patent EP-1081786-A3 (EP)
Inventor: MITSUI TSUTOMO
IPC: H01Q1/24
Filed: 2000-08-30
Abstract: A 4-line type helical antenna with a simple structure, which can obtain uniform
antenna gain even at a low elevation angle and has a radiation pattern which is not
affected even when the antenna is mounted on the chassis of an automobile. The helical
antenna comprises a circular cone (14), at least a surface of which is made of a metal,
interposed between an antenna body (11), for transmitting and receiving radio waves to/from
a satellite and a satellite terminal for transmitting and receiving the radio waves to/from the
antenna body (11). The circular cone (14), reflects the radio waves of the antenna body
(11). The antenna body (11) has antenna conductors (13), which are spirally formed
thereon, and the circular cone (14), is tapered at a given angle so as to uniformly reflect
the radio waves of the antenna body (11). The circular cone (14), is fixed to one end of
the antenna body (11), such that the tapered angle of the circular cone (14), should be
uniformly allocated with respect to an axis of the antenna body (11).
Patent EP-1093295-A3 (EP)
Inventor: NAKAJIMA MASATO
IPC: H04N1/407
Filed: 2000-10-13
Abstract: In an image processing device (1), when receiving image
data transferred from, for example a digital camera through an
image input section (11), the region division section (13)
divides the image data into a plurality of blocks having optimum
sizes according to a degree of a similarity between density
histograms of the blocks. A contrast enhancement section
(14)obtains an optimum clip value per divided block and then
obtains a density conversion curve based on the density histogram
of the block including a target pixel by using the clip value
in order to perform the density conversion for all of the pixels
optimally. The image data that have been enhanced in contrast
are compensated by a read compensation section (15) according
to a property of a printing device (3) and then printed on a
paper sheet.
Patent EP-1102520-A3 (EP)
Title: Anordnung zur Ansteuerung von LEDs
Inventor: HEITE CHRISTIAN DR-ING
IPC: H05B44/00
Filed: 2000-11-03
Abstract: Die Erfindung bezieht sich auf eine stromsparende Anordnung zur Ansteuerung einer
Anzahl n von lichtemittierenden Dioden LED (L1 bis Ln). Bei dieser Anordnung sind
in abwechselnder Folge jeweils eine LED (L1,L2...Ln) und ein nachgeschalteter
Strombegrenzungswiderstand (R/n) in einer Reihenschaltung angeordnet, und die
jeweils einem Strombegrenzungswiderstand (R/n) folgenden Knotenpunkte (K1 bis
Kn) der Reihenschaltung sind jeweils mit einem Portausgang (P1 bis Pn) einer Ansteuervorrichtung
(A) verbunden. Die Portausgänge (P1 bis Pn) der Ansteuervorrichtung
(A) sind wahlweise in einen der Zustände (Z(P i )): hochohmiger Zustand (H),
getakteter Ausgang (T, T*), Versorgungsspannung (1 = V DD ) oder Masse (0 = GND)
schaltbar.
Patent EP-1103528-A3 (EP)
Inventor: YAMAGATA SHIGERU DR
IPC: H01L21/027
Filed: 2000-11-18
Abstract: An object of the present invention is to provide a silica glass optical material having a
high initial transmittance with respect to vacuum ultraviolet radiation 155 to 195nm
in wavelength, a high precision, a high durability, and an excellent homogeneity, as
well as to a method for producing the same and a projection lens. 
     The silica glass optical material is of ultrahigh purity,
contains from 1 to 10wtppm of OH groups, from 100 to 10,000wtppm of F, and from
1 × 10 17  to 1 × 10 19  molecules/cm 3  of H 2 , and has a distribution in concentration of F
that is axially symmetrical to the central axis.
The silica glass material is produced by flame hydrolysis, fluorine
doping from the gas phase, vitrification, zone melting whilst rotating,
melting and molding in a frame and removing strain by annealing followed
by gas-phase hydrogen doping.
Patent EP-1107037-A3 (EP)
Title: Anordnung zum Scannen einer Objektaufnahmeeinrichtung
Inventor: ENGELHARDT JOHANN DR
IPC: G02B21/26
Filed: 2000-11-21
Abstract: Die Erfindung betrifft eine Anordnung zum Scannen einer Objektaufnahmeeinrichtung
(1) zur Datenaufnahme mit einem Laserscan-Mikroskop, vorzugsweise mit einem
konfokalen Laserscan-Mikroskop (2), mit der die Bildaufnahme großer Objektfelder
mit hinreichender Geschwindigkeit durch das Scannen der Objektaufnahmeeinrichtung
(1) möglich ist, ist dadurch gekennzeichnet, dass die Objektaufnahmeeinrichtung
(1) von einer Dreheinrichtung (3) um eine erste Achse (4) alternierend
drehbar ist.
Patent EP-1108841-A3 (EP)
Inventor: LUEMKEMANN ROLF
IPC: E05D7/04
Filed: 2000-12-14
Abstract: The adjustable band is for the rotatively movable fixture between fixed side parts and panes of complete glass plates (5). A holding piece is securely adhered on the outside with the complete glass plate. In a hollow space (9) of the holding piece, an adjustment device (10) is floatingly located, which through a front-side aperture (11) in the holding piece is connectable with a band flange (2). In the band flange a rear-side recess (12) is formed, which the holding piece overtops with clearance. In the adjustment device threaded bores (15) and in the band flanges bore holes (13) are formed, in which fixture components (14) are formed.
Patent EP-1111898-A3 (EP)
Inventor: FREDLUND JOHN R
IPC: H04N1/107
Filed: 2000-12-08
Abstract: A method and apparatus for capturing an image. The apparatus
includes a support platen for receiving a document having a front image bearing
side and a back side co-extensive with the front side. An image capture element is
disposed below the platen for capturing an image on the front image side. A
reticle forming device is provided for providing a reticle on the platen for assisting
in positioning of the document when a positioning cover is placed over the
document. A second cover is also provided for placement over the positioning
cover. The second cover is substantially opaque and is used for when the image
on the front image side is illuminating for capture of the image.