baber/WOPTO huggingface dataset:
Patent PT-1113014-E (PT)
Inventor: PEGLION JEAN-LOUIS
IPC: A61P9/00
Filed: 2000-12-26
Abstract: Piperidinyl- or piperazinyl-substituted linear or cyclic urea derivatives (or analogs) (I) are new. Piperidine or piperazine derivatives of formula (I) and their isomers, hydrates, solvates and acid addition salts are new. [Image] V, M : direct bond or linear or branched 1-6C alkylene; A, E : N or CH, provided that at least one is N; W : diaza-cyclic group of formula (a) or bicyclic group of formula (b), or may also be a bicyclic group of formula (c) if V = direct bond and A = N; [Image] * : attachment point; X : CO, SO or SO 2; G 12-4C n-alkylene (optionally containing a double bond and/or substituted by OH); G 2direct bond; and G 32-3C n-alkylene (optionally containing a double bond); or G 2CH 2; and G 31-2C n-alkylene (optionally containing a double bond); T : fused benzene or pyridine ring; R 1H, alkyl, Ar or Ar-alkyl; R 2 a, R 2 bH, halo, alkyl, OH, alkoxy, SH, alkylthio, trihaloalkyl, CN, NO 2, NH 2, mono- or dialkylamino, trihaloalkoxy, Ar-alkoxy, alkylsulfonate, trihaloalkylsulfonate or alkylsulfonyl; or R 2 a + R 2 bOCH 2O, O(CH 2) 2O, O(CH 2) 3O or CH 2CH 2 (optionally substituted by CN, CH 2OH, alkoxycarbonyl, ArOCO, or Ar-alkoxycarbonyl); R 3Ar or Het 1 (both optionally substituted by one or more R 2 a); Y : OAr, OHet 1 or Het 2 (all optionally substituted by one or more R 2 a); Ar : phenyl, biphenyl, naphthyl, dihydronaphthyl, tetrahydronaphthyl, indanyl, indenyl or benzocyclobutyl; Het 15-12 membered mono- or bicyclic aromatic system containing 1 or 2 of O, S and N as heteroatom(s), where in the case of bicyclic systems one of the rings may be partially hydrogenated; and Het 25-12 membered mono- or bicyclic aromatic system containing 1-3 of O, S and N as heteroatom(s). alkyl moieties have 1-6C unless specified otherwise; provided that: (i) if V = direct bond, W = (a) and R 3 = Ph, then Y cannot be 3-indolyl; (ii) if M = direct bond, W = (a) and Y = bicyclic Het 2 in which one ring is a benzene ring, then Y cannot be bonded to M via this benzene ring; and (iii) if M = direct bond, V = CH 2CH 2, W = (a) and R 3 = Ph, then Y cannot be 1,2-benzisoxazol-3-yl. An independent claim is included for the preparation of (I). ACTIVITY : Vasotropic; antiarteriosclerotic; cardiant; hypotensive. MECHANISM OF ACTION : Endothelial nitrogen monoxide (NO) synthase inhibitor antagonist; superoxide antagonist; antioxidant. (I) reduce endothelial dysfunction and reduction in vascular NO availability induced by inhibition of endothelial NO synthase or by oxidative stress associated with production of superoxide anion. In tests in rat aortic rings, N-(2-(4-(phenoxymethyl)-1-piperidinyl)-ethyl)-1-indoline-carboxamide (Ia) at a concentration of 30 nM gave 26 % inhibition of endothelial dysfunction induced by the NO synthase inhibitor N(G)-nitro-L-arginine.
Patent PT-1173393-E (PT)
Inventor: KOCH ERNST-CHRISTIAN
IPC: F41H9/00
Filed: 2000-01-07
Abstract: The invention relates to a method of producing a screening smoke which is one-way transparent in the infrared spectrum (780 nm-14.0 mum) and opaque in the visible spectrum. According to the invention a known pyrotechnic screening smoke which is highly absorbent in the visible spectrum (380 nm-780 nm) is generated in the form of an aerosol, pyrotechnic scattered particles between 10 and 100 mum in size are simultaneously produced in said aerosol, and the resulting two-component smoke is irradiated by an infrared radiation source (spectrum: 780 nm-14.0 mum) from the smoke producer side.
Patent PT-1148897-E (PT)
Inventor: ZHANG RENWEN
IPC: A61K38/22
Filed: 2000-01-31
Abstract: Methods and compositions are provided for the treatment of articular cartilage defects and disease involving the combination of the tissue, such as osteochondral grafts, with active growth factor. The active growth factor is preferably a composition containing at least one bone morphogenetic protein and a suitable carrier. The method results in the regeneration of functional repair of articular cartilage tissue.
Patent PT-1276646-E (PT)
Inventor: CASTAGNER BERNARD
IPC: B60R21/26
Filed: 2001-04-25
Abstract: The invention concerns a protective device comprising an airbag worn by a person, a pyrotechnic gas generator for inflating the airbag, and an actuator for the gas generator. The invention is such that the gas generator has a dual state combustion. Preferably, the generator is single-piece with single ignition. The invention device enables to provide a first inflating phase lasting about 60 ms at most, preferably between 30 and 50 ms; then a second phase maintaining inflation lasting at least a few seconds, preferably at least 4 s, more preferably still between 5 and 8 s.
Patent PT-1261980-E (PT)
Title: Emergency shutdown key
Inventor: BURS MARC
IPC: H01H3/02
Filed: 2001-03-02
Abstract: The device has an actuating knob, a button guide (4) and a locking arrangement. The guide has a first guide path (21) parallel to the longitudinal axis, a locking arrangement protruding into the path under spring force and a first protrusion in the path so that only unlocking by pulling is possible. A second guide path (26) and protrusion allow only unlocking by turning. The locking arrangement can be inserted into one of the two guide paths
Patent PT-1302926-E (PT)
Inventor: PARK JONG-BOO
IPC: G02F1/133
Filed: 2002-09-18
Abstract: An apparatus and method for preventing lock-up of an LCD is provided, in which a voltage on a pin of the LCD is monitored, and determined whether an electrostatic discharge (ESD) has been applied to the LCD based on the monitored voltage, and the LCD is reset if an ESD has been applied to the LCD. In a preferred embodiment, the LCD pin which voltage is monitored exhibits a voltage level change, in response to an ESD, that is greater than a voltage level change exhibited by all other individual pins of the LCD. Because the LCD is reset only when an ESD condition has been detected, periodic blinking of the LCD is prevented. <IMAGE>
Patent PT-1397313-E (PT)
Title: Press bending station and method for bending heated glass sheets
Inventor: BENNETT TERRY A
IPC: C03B23/025
Filed: 2002-06-17
Abstract: A press bending station (12) for heated glass sheets includes a lower wheel bed (36) having a lower support (38) and wheel assemblies (40) with detachable connections (46) to a drive mechanism (48) of the lower support to provide rotational driving of a wheel (44) of each wheel assembly. An actuator (62) provides relative vertical movement that lifts a heated glass sheet received by the wheel bed (36) to provide press bending thereof between a lower press ring (52) and an upper press mold (58). The wheel bed (36) can have a curved shape or a flat shape. Connection and detachment of the wheel assemblies (40) facilitates switching from one production job to the next.
Patent PT-1364717-E (PT)
Title: Decanter centrifuge for extracting fruit- or vegetable juices having a worm-conveyor for discontinous transport
Inventor: HAIDER GUENTER
IPC: A23N1/00
Filed: 2003-05-23
Abstract: Decanting centrifuge comprising a conveyor screw (10) rotating in a rotor, devices for introducing material, and outlet openings for the liquid phase and the solids, is new. The screw has spirals (24) part of which are formed as paddles (26) arranged on gaps for the discontinuous conveying of the material (20).  Preferred Features: The paddles are adjusted on their inlet edges at an angle to the radial surfaces. The paddles are planar. The inlet edges of the paddles lie vertical to the shaft body of the screw.
Patent PT-1484970-E (PT)
Title: Benzamides and compositions comprising benzamides for use as fungicides
Inventor: FOOR STEPHEN RAY
IPC: A01N57/18
Filed: 2003-03-18
Abstract: Compositions for controlling plant diseases caused by fungal plant pathogens are described, comprising:   
(a) a fungicidally effective amount of a compound of Formula I (including all geometric and stereoisomers,  N -oxides, and agriculturally suitable salts thereof) wherein A, B, W, R 1 , R 2 , and R 3  are as defined in the disclosure; and 
(b) at least one compound selected from the group consisting of (b9) fosetyl-aluminum.  Also disclosed are methods for controlling plant diseases caused by fungal plant pathogens that involves applying an effective amount of the combinations described.
Patent PT-1573208-E (PT)
Title: Intake duct
Inventor: BROSS STEPHAN
IPC: F04D29/40
Filed: 2003-10-23
Abstract: A centrifugal pump with a housing having one or more impellers having an axial or semiaxial, open or closed design disposed therein and an intake channel mounted upstream of the first impeller. A plurality of grooves that are distributed around the circumference and extend in the direction of flow are arranged within the wall area of the intake channel. In the housing wall of the intake channel there is a closed annular wall area constructed between a point of entry of the first impeller and the proximate ends of the grooves, whereby the grooves are operatively connected exclusively with the space in the intake channel.
Patent PT-1654241-E (PT)
Title: Macrocyclic compounds having aspartic protease inhibiting activity and pharmaceutical uses thereof
Inventor: BETSCHART CLAUDIA
IPC: C07D273/02
Filed: 2004-07-02
Abstract: The present invention relates to macro-cyclic compounds of formula (I), wherein R<SUB>1</SUB>, is (C<SUB>1-8</SUB>)alkyl, (C<SUB>1-4</SUB>)alkoxy(C<SUB>1-4</SUB>)alkyl, hydroxy(C<SUB>1-6</SUB>)alkyl, (C<SUB>1-4</SUB>)alkylthio(C<SUB>1-4</SUB>)alkyl, (C<SUB>1-6</SUB>)alkenyl, (C<SUB>3-7</SUB>)cycloalkyl, (C<SUB>3-7</SUB>)cycloalkyl(C<SUB>1-4</SUB>)alkyl, piperidinyl or pyrrolidinyl, R<SUB>2 </SUB>and R<SUB>4</SUB>, independently, are hydrogen or optionally substituted (C<SUB>1-8</SUB>)alkyl, (C<SUB>3-7</SUB>)cycloalkyl, (C<SUB>3-7</SUB>)cycloalkyl(C<SUB>1-4</SUB>)alkyl, aryl, aryl(C<SUB>1-4</SUB>)alkyl, heteroaryl or heteroaryl(C<SUB>1-4</SUB>)alkyl, or R<SUB>2 </SUB>and R<SUB>4</SUB>, together with the nitrogen to which they are attached, form an optionally substituted piperidino, pyrrolidinyl, morpholino or piperazinyl group, R<SUB>3 </SUB>is hydrogen or (C<SUB>1-4</SUB>)alkyl, X<SUB>1 </SUB>is CH<SUB>2</SUB>, X<SUB>2 </SUB>is CH<SUB>2</SUB>, O, S, CO, COO, OCO, NHCO, CONH, or NR, R being hydrogen or (C<SUB>1-4</SUB>)alkyl, Y is (C<SUB>1-8</SUB>)alkylen or (C<SUB>1-8</SUB>)alkylenoxy(C<SUB>1-6</SUB>)alkylen, (C<SUB>1-8</SUB>)alkenylen or (C<SUB>1-8</SUB>)alkenylenoxy(C<SUB>1-6</SUB>)alkylen, Ar is a phenyl ring optionally mono- di or trisubstituted by, independently, hydroxy or halogen, whereby X<SUB>1</SUB>, and X<SUB>2 </SUB>are in meta or para position to each other, and either Z is CO, AA is a natural or unnatural alpha-amino-acid, and n is 0 or 1, or Z is S0<SUB>2</SUB>, AA is an optionally substituted ethylencarbonyl group (derived from a natural or unnatural alpha-amino acid by replacement of the nitrogen by a methylen group), and n is 1; processes for the preparation of these compounds; pharmaceutical compositions and combinations comprising the same; and their use in the treatment of neurological and vascular disorders related to beta-amyloid generation and/or aggregation.
Patent PT-1641862-E (PT)
Title: Silyl ester copolymer compositions
Inventor: FINNIE ALISTAIR ANDREW
IPC: C08G77/04
Filed: 2004-06-29
Abstract: The invention relates to a silyl ester copolymer solution having a solids content of at least 55 weight percent and a viscosity of less than 20 poise at 25° C., comprising a silyl ester copolymer having a weight-average molecular weight of less than 20,000. The invention further relates to coating compositions comprising a silyl ester copolymer and to substrates and structures having a cured coating prepared from such a coating composition.
Patent PT-1636593-E (PT)
Title: Modulating the interaction between hgf beta chain and c-met
Inventor: LAZARUS ROBERT A
IPC: G01N33/574
Filed: 2004-06-04
Abstract: The invention provides methods and compositions for modulating the HGF/c-met signalling pathway, in particular by regulating binding of HGF ² chain to c-met.
Patent PT-1759373-E (PT)
Title: Equipment for displaying information carriers especially for advertising purposes
Inventor: SERDUELT GYULA
IPC: A47F11/06
Filed: 2004-10-11
Abstract: Equipment for displaying information carriers, especially objects, mainly goods and products and/or devices introducing human, mainly service-providing activities, favourably for advertising purposes, which equipment has a cabinet 1 suitable for accommodating the information carrying device to be displayed, constructed in a way that it is possible to look inside its internal space, which cabinet contains light sources, especially lighting units. The equipment is characterised by that the cabinet's 1 side-walls (1,2), bottom-wall (5) and upper-wall 6, made of non-transparent material, contain a strip running around situated at a distance e from the back-wall (4), and the edges of a transparent plate 7 are in contact with this strip; -the information carrier, especially object (8) to be displayed is situated on the front of the transparent plate 7 with respect to the viewing direction a of the inside of the cabinet 1; - the side-walls (1,2), the bottom-wall (5) and the upper-wall (6) contain at least one strip running around of the same construction as the strip touching the transparent plate (7), situated at a distance from the transparent plate (7), in front of it, favourably parallel to the contact strip; and - looking at it from the viewing direction a there are lighting units 10 behind the transparent plate (7).
Patent PT-1624105-E (PT)
Title: Alkanol-ammonia containing triazinylflavonat brightener
Inventor: HEINZ GIESECKE DR
IPC: D21H21/30
Filed: 2005-07-23
Abstract: Method for whitening paper in the size press comprises a size press fleet containing an alkanolammonium containing triazinyl flavone compound (I) as the optical whitener. Method for whitening paper in the size press comprises a size press fleet containing an alkanolammonium containing triazinyl flavone compound of formula (I) as the optical whitener. X : alkyl compounds of formula (a) or (b); either R 1>, R-1a : 1-6C alkyl; and R 2>, R-2a : H; or R 3>, R-3a : H, CH 3, CH 2CH 3, CH 2CH 2OH or CH 2CH 2OCH 3; R 4>H or 1-4C alkyl; M : an equivalent inorganic cation (preferably Li, Na, K, Ca, Mg or ammonium) or a substituted ammonium of formula (II) (where at least 10 mol.% of all cation corresponds to formula (II)); R 5>-R 7>H, 1-4C alkyl or optionally substituted 2-4C hydroxyalkyl; and R 8>optionally further substituted 2-4C hydroxy alkyl. Independent claims are also included for: (1) an optical whitener preparation comprising more than 50 (preferably more than 95) wt.% of (I); and (2) a size press fleet comprising (I) or an optical whitener preparation and at least a surface sizing agent (preferably starch). [Image] [Image] [Image].
Patent PT-1753566-E (PT)
Title: Method for the production of niobium and tantalum powder
Inventor: HAAS HELMUT
IPC: C22B34/24
Filed: 2005-04-09
Abstract: In the production of metal valve powders, especially niobium and tantalum, the metal oxide powders are reduced by reduction metal vapors and/or their hydrides in an inert carrier gas. The reduction is at a partial vapor pressure of the reduction metal/hydride of 5-110 hPa and at a total pressure of = 1000 hPa. The preferred metal oxides are of titanium, zirconium, hafnium, vanadium, niobium, tantalum, molybdenum and/or tungsten, and especially tantalum pentoxide. The reduction metal is a magnesium vapor.
Patent PT-1776323-E (PT)
Title: Batch for producing a fireproof ceramic moulded body, method for the production of the same and use thereof as a diesel particulate filter
Inventor: KRIEGESMANN JOCHEN
IPC: C04B35/565
Filed: 2005-06-30
Abstract: The invention relates to a batch for producing a fireproof ceramic moulded body comprising a porous matrix, containing a non-oxidic, ceramic component with at least one grain size and an organic binding agent. The invention also relates to a method for producing the moulded body and to the use of said body as a diesel particulate filter.
Patent PT-1749700-E (PT)
Title: Large sized vehicle for passenger transportation, especially railway or omnibus
Inventor: SCHILLINGS DIRK
IPC: B64C1/12
Filed: 2006-06-14
Abstract: Large capacity vehicle has lining element (1) for door pillar and one of the fitting components grip bar (2), wind screen (3), light barrier (4), stop request button (5) forms a complete premounted and pretested assembly unit. The premounted and pretested assembly unit is wired incase of electric fitting components (4,5).
Patent PT-1962926-E (PT)
Title: Injection device
Inventor: MEJLHEDE SIGNE THORNING
IPC: A61M5/142
Filed: 2006-12-22
Abstract: A device for delivering fluid, comprising an injection part (1), a fluid delivery part (3,4), and a base plate (10), wherein the fluid delivery part and the base plate can be separated and rejoined, the fluid delivery part comprising a reservoir (4) having an outlet, transfer means, and a housing (3), the injection part comprising a cannula part comprising a body with a through going opening provided with a cannula (9) configured to extend past the proximal side of the base plate, the base plate comprising means for fixation of the base plate to the skin of the user, wherein the injection part comprises a first part (1a) which is fastened unreleasably to the base plate and a second part (1b) comprising the cannula part, the second part being configured to lock to the first part upon insertion of the second part.
Patent PT-2042509-E (PT)
Title: Modulators of the function of fas receptors and other proteins
Inventor: WALLACH DAVID
IPC: A61K48/00
Filed: 1996-06-14
Abstract: The present invention provides proteins capable of modulating or mediating the FAS receptor ligand or TNF effect on cells carrying FAS receptor or p55 receptor by binding or interacting with MORT-1 protein, which in turn binds to the intracellular domain of the FAS receptor or to another protein TRADD which binds to the p55 receptor. In addition, peptide inhibitors which interfere with the proteolytic activity of MORT-1-binding proteins having proteolytic activity are provided as well as a method of designing them.
Patent PT-2200841-E (PT)
Title: Multilayer body and method for producing a multilayer body
Inventor: TOMPKIN WAYNE ROBERT
IPC: B29D11/00
Filed: 2008-10-15
Abstract: The invention concerns a multilayer body and a process for producing a multilayer body. The multilayer body has a transparent first layer in which a multiplicity of cylindrical lenses of a length of more than 2 mm and a width of less than 400 mum are shaped, which are arranged in accordance with a microlens grid spanning a first co-ordinate system having a co-ordinate axis X1 which is determined by the focal point lines of the cylindrical lenses, and a co-ordinate axis Y2 perpendicular thereto.
Patent PT-679156-E (PT)
Inventor: HOLTON ROBERT A
IPC: C07C233/46
Filed: 1994-01-14
Abstract: A process for abstracting a C10 hydroxy, acyloxy or sulfonyloxy substituent from a taxane in which the C10 hydroxy, acyloxy or sulfonyloxy substituted taxane is reacted with samarium diiodide.
Patent PT-676635-E (PT)
Inventor: RINGLIEN JAMES A
IPC: G01N21/90
Filed: 1995-04-05
Abstract: Apparatus for inspecting the bottom (12) of a container (14) that includes a light sensor (26) positioned to view the container bottom through the open container mouth (28), a light source (24 or 46) positioned externally of the container on the opposite side of the container bottom, and electronics (34) for detecting commercial variations in the container bottom as a function of light energy incident on the sensor. The light source, as viewed by the sensor through the container bottom, is characterized by being elongated radially of the container bottom and narrow transversely of the container bottom. In this way, any variations (38) in the container bottom that refract the line of sight of the sensor in the radial direction, such as mold code rings and baffle scars, are essentially transparent as viewed by the sensor. On the other hand, variations (40) that refract the sensor line of sight laterally of the container bottom, such as glass particles, knots and lumps, produce a dark image at the sensor since the sensor cannot see the light source through the variation. <IMAGE>
Patent PT-811058-E (PT)
Inventor: HOFFER LUTZ
IPC: C12N9/64
Filed: 1996-02-14
Abstract: PCT No. PCT/EP96/00636 Sec. 371 Date Nov. 26, 1997 Sec. 102(e) Date Nov. 26, 1997 PCT Filed Feb. 14, 1996 PCT Pub. No. WO96/27003 PCT Pub. Date Sep. 6, 1996A process for the preparation of factor IX from a biological source by chromatography involves prior treatment with ammonium sulfate as a protein precipitant at a concentration of from 1.5-2.3 mol/l.
Patent PT-857231-E (PT)
Inventor: NORDEN SOLVEIG
IPC: D21C9/10
Filed: 1996-09-18
Abstract: Methods for oxygen delignification of a pulp are disclosed, including initially delignifying the pulp at a delignification temperature of less than 90° C., adding oxygen to the pulp so that the oxygen is present during the initial delignification step, and further delignifying the pulp at a delignification temperature of greater than 90° C., the difference between the two delignification temperatures being less than about 20° C., and the pressure being greater in the initial delignification step. The method also includes adding alkali solely to the initial delignification step in order to obtain high alkalinity therein.
Patent PT-880484-E (PT)
Inventor: BLOMKIST OVE
IPC: C02F11/143
Filed: 1997-02-12
Abstract: PCT No. PCT/NO97/00041 Sec. 371 Date Aug. 10, 1998 Sec. 102(e) Date Aug. 10, 1998 PCT Filed Feb. 12, 1997 PCT Pub. No. WO97/30008 PCT Pub. Date Aug. 21, 1997Liquid containing organic waste material and chemicals are continually introduced into the upper part of a vertical, cylindical treatment chamber. While sinking through the chamber, the material is beaten by fast rotating treating elements which also mix the material. The treating elements also move in axial direction to free vapors and gases from the material. Vapors and gases are removed from the top of the chamber.
Patent PT-927027-E (PT)
Inventor: LEFEVRE HERVE
IPC: A61K31/00
Filed: 1997-08-29
Abstract: The invention concerns a novel use of antagonists of the 5-HT4 receptor in pathological conditions where the aldosterone and cortisol blood levels are abnormally high.
Patent PT-940401-E (PT)
Inventor: NAKAZATO ATSURO
IPC: A61K31/425
Filed: 1997-09-19
Abstract: This invention provides a 2-carbonylthiazole derivative represented by formula (I): <CHEM> Äwherein each of Ar<1> and Ar<2> represents a phenyl group, a phenyl group having one or two substituents selected from "a halogen atom, an alkyl group having 1 to 5 carbon atoms, a trifluoromethyl group, an alkoxy group having 1 to 5 carbon atoms and a hydroxyl group" or a thienyl group; R<1> represents an alkoxy group having 1 to 5 carbon atoms, a hydroxyl group or an amino group represented by formula N(R<3>)R<4> (wherein each of R<3> and R<4> represents a hydrogen atom or an alkyl group having 1 to 5 carbon atoms, or R<3> and R<4>, together with the nitrogen atom to which they are bound, form a pyrrolidino, piperidino, morpholino or piperazino group, or a pyrrolidino, piperidino, morpholino or piperazino group having one to four substituents selected from "an alkyl group having 1 to 5 carbon atoms, an alkoxy group having 1 to 5 carbon atoms and a hydroxyl group"); Y<1>-Y<2> represents CH-CO or C=C(R<2>) (wherein R<2> represents a hydrogen atom or an alkyl group having 1 to 5 carbon atoms); and n is an integer of from 1 to 4Ü or a pharmaceutically acceptable salt thereof. It also provides a medicament which comprises the 2-carbonylthiazole derivative of formula (I) or a pharmaceutically acceptable salt thereof and a dopamine D4 receptor antagonist which contains the same as the active ingredient, which are useful as drugs for preventing and treating dopamine D4 receptor-related morbid states such as schizophrenia and problematic behavior caused by cerebrovascular accidents and senile dementia, and also as the drugs which do not induce extrapyramidal disorders as side effects.