baber/WOPTO huggingface dataset:
Patent CZ-76597-A3 (CZ)
Title: 2-amino-1,2,3,4-tetrahydronaphthalene derivatives, process of their preparation and pharmaceutical composition containing thereof
Inventor: MONTANARI STEFANIA
IPC: C07C323/25
Filed: 1995-09-11
Abstract: Compounds of formula    <IMAGE>  (I)  wherein R, R', R'', R1, R2, R3, R4, R5, R6, X, Y, m, n and p have the meanings reported in the description; and their pharmaceutically acceptable salts are described. The compounds of formula I are useful in the treatment of arterial hypertension and congestive heart failure, of renal failure, of peripheral arteriopathies, of cerebrovascular insufficiencies and of ischemic cardiopathy.
Patent CZ-76995-A3 (CZ)
Title: Derivatives of 1-(oxoacetyl)pipridine-2-carboxylic acid, process of their preparation pharmaceutical composition containing thereof and their use
Inventor: ARMISTEAD DAVID M
IPC: C07D235/00
Filed: 1993-09-27
Abstract: The present invention relates to novel compounds of formula (I) which maintain, increase, or restore sensitivity of cells to therapeutic or prophylactic agents. This invention also relates to pharmaceutical compositions comprising these compounds. The compounds and pharmaceutical compositions of this invention are particularly well-suited for treatment of multi-drug resistant cells, for prevention of the development of multi-drug resistance and for use in multi-drug resistant cancer therapy.
Patent CZ-83698-A3 (CZ)
Title: Process and apparatus for determining thickness of film and covering of pattern of cells being plated on induction payment cards
Inventor: DE OLIVEIRA LOPES PAULO HENRIQ
IPC: G01B7/06
Filed: 1996-09-17
Abstract: A device for determining the thickness of conductive metal patterns plated on insulating surfaces, such as credit cells in prepaid telephone debit cards, comprising a plurality of sensing modules equal in number to the credit cells in said cards, each module consisting of an oscillator (30) wherein the inductance is provided by a pair of collinear sensing coils (24a, 24b), aligned with the true position of its relative credit cell (25), the output (26) of said sensing assembly being connected to the input of an A/D converter (40) whose output is connected to computing means (11, 21) provided with memory means. Said oscillators are enabled by turns, the output voltage being converted to a numeric value. The converter parameters are adjusted for each sensing module according to coefficients stored in said memory, to compensate for component variations, sensing coil position and so on. The resultant numeric value is processed by the computing means according to a transfer curve (53) which is specific for each sensing module, so as to furnish the film thickness. Said coefficients and transfer curves are previously determined for each one of the positions in the cell array by means of individual calibration, using standard cards of known metal film thickness.
Patent SK-48097-A3 (SK)
Title: Process for producing liquid raw iron or steel basic products and iron sponge and plant for implementing it
Inventor: DIEHL JOERG
IPC: C21B13/00
Filed: 1995-10-12
Abstract: In a process for producing liquid raw iron or steel basic products and iron sponge from charges consisting of iron ore and possible additives, the charges are directly reduced to iron sponge in a fixed-bed reducing region (12), the iron sponge is melted in a melt gasification region (8) with the addition of carbon vehicles and oxygen-containing gas and a reduction gas containing CO and H2 is produced which is taken into the reducing region (12), reacted there and drawn off as the export gas, CO2 is extracted from the export gas drawn off and taken as an at least largely CO2-free reducing gas together with some of the reducing gas formed in the melt gasification region (8) to a further reducing region (21) for the direct reduction of iron ore. In order to reduce the investment costs of a plant for implementing this process and improve productivity, part of the reducing gas generated in the melt gasification region (8) is diverted and taken to the further reduction region (21), by-passing the CO2 elimination stage.
Patent SK-54194-A3 (SK)
Title: Preparation with controlled releasing of medicine and method of its manufacture
Inventor: MILLER RONALD B
IPC: A61K47/44
Filed: 1994-05-10
Abstract: A controlled release preparation for oral administration contains tramadol, or a pharmaceutically acceptable salt thereof, as active ingredient.
Patent SK-62799-A3 (SK)
Title: Glass fibres for reinforcing organic and/or inorganic materials
Inventor: GALLO MARCELO HERNAN
IPC: C03C13/00
Filed: 1998-09-10
Abstract: The invention concerns reinforcing glass fibres whereof the composition comprises the following constituents, within the limits defined as follows expressed in weight percentages: 58 to 62 % SiO2, 10 to 16 % Al2O3, more than 18 % CaO, more than 1.5 % MgO, less than 28 % CaO + MgO, less than 2 % Na2O + K2O + Li2O, less than 1.5 % TiO2, less than 0.5 % Fe2O3, less than 2 % B2O3, less than 2 % F2; said composition further comprising 1 % of other constituent(s) and comprising more than 0.5 % of at least three F2, B2O3, Li2O constituents. Said glass fibres have a composition providing excellent compromise between its cost and its fibre drawing capability.
Patent SK-62993-A3 (SK)
Title: Novel methylenebisphosphonic acid derivatives
Inventor: NIKANDER HANNU
IPC: A61P19/08
Filed: 1991-12-18
Abstract: Compositions having formula (I) wherein R1, R2, R3 and R4 independently are straight or branched, optionally unsaturated C1-C10 alkyl group or hydrogen, whereby in formula (I) at least one of the groups R1, is hydrogen and at least one of the groups R1, R2, R3 and R4 is different from hydrogen, Q1 is hydrogen or hydroxyl group, Q2 is straight or branched C1-C10-alkyl C3-C10-cycloalkyl, C2-C10 hydroxyalkyl or C2-C10-aminoalkyl, where amino is optionally substituted by one or two C1-4-alkyls and stereoisomers of these compositions, such as the geometrical isomers and the optically active isomers, as well as the pharmacologically acceptable salts of these compounds. Disclosed is also the method for preparation of the said derivatives and pharmaceutical means containing them.
Patent SK-65797-A3 (SK)
Title: Food on the milk product base enriched with ground eggshell
Inventor: SCHAAFSMA ANNE
IPC: A23L1/304
Filed: 1995-11-21
Abstract: The invention relates to the use of aseptic or sterile fine ground eggshell in foods based on milk products. As a result, products of good taste are obtained, which are enriched with calcium and which give improved calcium absorption and retention of the total calcium fraction compared with milk product-based food products enriched with calcium from other calcium sources.
Patent CS-271891-A3 (CS)
Title: Diphenyl compounds inhibiting substitution of arachidonic acid and their use in pharmaceuticals
Inventor: SCHEFE TANKRED PROF DR
IPC: A61K31/055
Filed: 1991-09-04
Abstract: Pharmaceutical compositions, which comprise a compound of the general formula I  <IMAGE>  in which X is oxygen, sulfur or -CH2-, Y is chlorine or bromine, Z is an SO2H, NO2 or C1-C4alkyl radical, r is a number from 0 to 3, o is a number from 0 to 3, p is the number 0 or 1, m is the number 1 or 2 and n is the number 0 or 1, have having a lipoxygenase- and prostaglandin H synthase-inhibiting action. The compositions are useful in particular for the local (topical) or inhalative treatment of inflammatory, allergic and spasmolytic diseases, as well as psoriasis, bronchial asthma and diseases with disturbances in cell proliferation.
Patent CZ-117998-A3 (CZ)
Title: Stabilization process of biological materials and preparations for making the same
Inventor: MATTERN MARKUS
IPC: A61K38/44
Filed: 1996-10-24
Abstract: The present invention concerns processes for the production of dry, partially amorphous products containing biologically active and in particular therapeutically active material which are macroscopically homogeneous substance mixtures, the substance mixtures being selected from at least one substance of each of the groups (i) carbohydrate or zwitterion with a polar residue and derivatives thereof, and (ii) zwitterion with an apolar residue and derivatives thereof, wherein a solution is prepared of the biologically or therapeutically active material and of substances (i) and (ii) and the solution is dried at a product temperature above the freezing point of the solution. In addition the invention concerns new substance mixtures which are obtained by the said process as well as the use thereof in diagnostic or therapeutic methods.
Patent CZ-9301304-A3 (CZ)
Title: Single-crystal nickel-based high alloy
Inventor: ERICKSON GARY L ING
IPC: C30B29/52
Filed: 1993-06-29
Abstract: A nickel-based superalloy comprises the following elements in percent by weight: from about 5.0 to about 7.0 percent rhenium, from about 1.8 to about 4.0 percent chromium, from about 1.5 to about 9.0 percent cobalt, from about 7.0 to about 10.0 percent tantalum, from about 3.5 to about 7.5 percent tungsten, from about 5.0 to about 7.0 percent aluminium, from about 0.1 to about 1.2 percent titanium, from about 0 to about 0.5 percent columbium, from about 0.25 to about 2.0 percent molybdenum, from about 0 to about 0.15 percent hafnium, and the balance nickel + incidental impurities, the superalloy having a phasial stability number NV3B less than about 2.10. <IMAGE>
Patent CZ-156796-A3 (CZ)
Title: Benzimidazoles derivatives, their preparation and their therapeutical application
Inventor: FUJITA TAKASHI
IPC: A61K31/4245
Filed: 1996-05-30
Abstract: Compounds of formula (I): <CHEM> Äin which: X represents an optionally substituted benzimidazole group; Y represents an oxygen or sulphur atom; Z represents a 2,4-dioxothiazolidin-5-ylidenylmethyl, 2,4-dioxothiazolidin-5-ylmethyl, 2,4-dioxo-oxazolidin-5-ylmethyl, 3,5-dioxooxadiazolidin-2-ylmethyl or N-hydroxyureidomethyl group; R represents hydrogen, alkyl, alkoxy, halogen, hydroxy, nitro, amino or aralkyl; and m is an integer from 1 to 5Ü; have valuable activity for the treatment and/or prophylaxis of a variety of disorders, including one or more of: hyperlipemia, hyperglycemia, obesity, impaired glucose tolerance (IGT), insulin resistance and diabetic complications.
Patent CZ-164999-A3 (CZ)
Title: Process of strengthening flat glass by coating edges, brittle oxide object and window assembly
Inventor: PAPANU VICTOR DENNIS
IPC: C03C17/32
Filed: 1998-09-01
Abstract: A method is described for strengthening or restoring strength to a flat brittle oxide substrate (12) which includes the steps of coating the edges of the brittle oxide substrate (12) with a strengthening composition without coating a significant portion of the major flat surfaces of the substrate (12). The strengthened brittle oxide substrate (12), such as glass, and a window containing as a window pane the edge strengthened glass (12) are also provided.
Patent CZ-189097-A3 (CZ)
Title: Amorphous silicates of alkali metals
Inventor: GONZALES ARTIGA
IPC: C11D3/08
Filed: 1995-12-14
Abstract: Water-soluble builder substances partially or totally replace zeolite in washing or cleaning agents. They should above all be suitable for production and use with extruded and granulated washing or cleaning agents. For that purpose, amorphous alkaline silicates are used with a secondary detergent power and a molar ratio between M2O and SiO2 (M being an alkaline metal) from 1:1.5 and 1:3.3. These amorphous alkaline silicates have at least 300 g/l apparent density and are impregnated with active ingredients of washing or cleaning agents, in particular non-ionic surfactants.
Patent CZ-200442-A3 (CZ)
Title: Novel heterocyclic compounds functioning as bacterial DHFR selective inhibitors and their use
Inventor: MOE SCOTT T
IPC: C07D471/04
Filed: 2002-06-28
Abstract: The invention is based on the discovery of a new class of heterocyclic compounds having, for example, antibacterial properties. The D-Ala-D-Ala ligase enzyme is a critical pathway enzyme in the bacterial cell-wall synthesis. The compounds can bind to and inhibit the enzyme D-Ala-D-Ala ligase. The new compounds' activity combined with their ability to cross bacterial cell membranes makes them suitable for use as antibacterial drugs or other antibacterial applications.
Patent CZ-201232-A3 (CZ)
Inventor: KATOLICKY ZDENEK
IPC: F02C9/52
Filed: 2012-01-19
Abstract: Regulátor palivových trysek s obtokem sestává z hlavního odtlacného prvku, telesa (2) vstupního tlaku a telesa (3) výstupního tlaku, pricemž obe telesa (2 a 3) jsou spolu pevne spojeny šrouby (16). Teleso (2) vstupního tlaku je opatreno stredovým výklenkem (18) s vyrovnávacím prostorem (13) a teleso (3) výstupního tlaku je uzavreno krycím telesem (19), s kterým je spojeno šrouby (20). Do krycího telesa (19) je zašroubováno vedení (6) jehly (5) pístu (4) a pružiny (7), pricemž pružina (7) se opírá o dosedací výstupek (21) a o hlavu (22) pístu (4). Teleso (2) vstupního tlaku je opatreno prívodní tryskou (8), pro prívod paliva do vyrovnávacího prostoru (13) ve stredovém výklenku (18) z vnejší strany membrány (1). Jehla (5) je opatrena vybráním (25), které má drážku (23) a nábehovou cást (9), orientovanou k hlave (22) pístu (4) pro zajištení plynulého prechodu z plne otevreného obtoku do plne uzavreného obtoku.
Patent CZ-201755-A3 (CZ)
Inventor: Mašek Bohuslav
IPC: E04C3/292
Filed: 2017-01-31
Abstract: Způsob výroby dřevěných nosníků zahrnuje kroky: nahřátí ocelové výztuže (2) na teplotu austenitu materiálu, ze kterého je vyrobena; nahřátí dřevěné voštiny (3) na teplotu ležící mezi Ms a Mf materiálu, ze kterého je vyrobena výztuž (2); nanesení teplotně odolného lepidla na povrch nejméně jedné výztuže (2) a/nebo dřevěné voštiny (3); zalisování výztuže (2) do povrchu dřevěné voštiny (3) v lisovacím přípravku definujícím budoucí tvar dřevěného nosníku (1); udržení dřevěného nosníku (1) v lisovacím přípravku alespoň po dobu vyrovnání teplot výztuže (2) a voštiny (3) a jejich společného ochlazení, zahrnujícího proces stabilizace zbytkového austenitu a popuštění martenzitu v oceli výztuže (2) a vytvrzení lepidla. Nosník může obsahovat více střídajících se vrstev výztuží (2), lepidla a dřevěných voštin (3). Výztuž (2) může být opatřena vystupujícím tvarovým zámkem (4), který je při lisování zalisován do dřevěné voštiny (3). Voština (3) může být na povrchu opatřena sníženou oblastí (6), do které je nejméně jedna výztuž (2) uložena.
Patent CZ-206195-A3 (CZ)
Title: Controlled transcription of target genes and other biological materials
Inventor: CRABTREE GERALD R
IPC: C10G7/06
Filed: 1994-02-14
Abstract: Dimerization and oligomerization of proteins are general biological control mechanisms that contribute to the activation of cell membrane receptors, transcription factors, vesicle fusion proteins, and other classes of intra- and extracellular proteins. We have developed a general procedure for the regulated (inducible) dimerization or oligomerization of intracellular proteins. In principle, any two target proteins can be induced to associate by treating the cells or organisms that harbor them with cell permeable, synthetic ligands. To illustrate the practice of this invention, we have induced: (1) the intracellular aggregation of the cytoplasmic tail of the ¶ chain of the T cell receptor (TCR)-CD3 complex thereby leading to signaling and transcription of a reporter gene, (2) the homodimerization of the cytoplasmic tail of the Fas receptor thereby leading to cell-specific apoptosis (programmed cell death) and (3) the heterodimerization of a DNA-binding domain (Gal4) and a transcription-activation domain (VP16) thereby leading to direct transcription of a reporter gene.  Regulated intracellular protein association with our cell permeable, synthetic ligands offers new capabilities in biological research and medicine, in particular, in gene therapy. Using gene transfer techniques to introduce our artificial receptors, one can turn on or off the signaling pathways that lead to the overexpression of therapeutic proteins by administering orally active "dimerizers" or "de-dimerizers", respectively. Since cells from different recipients can be configured to have the pathway overexpress different therapeutic proteins for use in a variety of disorders, the dimerizers have the potential to serve as "universal drugs". They can also be viewed as cell permeable, organic replacements for therapeutic antisense agents or for proteins that would otherwise require intravenous injection or intracellular expression (e.g., the LDL receptor or the CFTR protein).
Patent CZ-209895-A3 (CZ)
Title: Sound evaluation method
Inventor: KEIPER WINFRIED
IPC: G01H3/08
Filed: 1994-12-05
Abstract: In a sound evaluation process, a digital signal that corresponds to the sound is subjected to a Fourier time transformation (FTT 14). Partial tones are derived from the result for predetermined frequencies within an equally predetermined evaluation interval. Thanks to the frequency-dependent definition of the evaluation interval for determining a partial tone, sound, in particular a technical sound, are reproduced in a manner that corresponds to the perception of the human ear. The determination of partial tone lines reduces the data to be processed and makes the representation of the result clearer. A criterion that allows the perception of knocks to be recognised is derived from the progression in time of a selected partial tone line. This process is particularly suitable for evaluating technical, industrial sounds and is therefore particularly applicable to acoustic quality control.
Patent CZ-252699-A3 (CZ)
Title: Distillation process with reduced clogging
Inventor: KRESNYAK STEVE
IPC: C02F1/04
Filed: 1998-01-14
Abstract: A method for removing a contaminant from a fluid feed stream containing the contaminant. The method includes the steps of providing a feed stream and heating it in a first step to at least partially remove some of the contaminants and recover energy from a concentrate and distillate generated. Further heating the feed stream in a second heating step in a heated separator generates a saturated vapor fraction and a concentrated liquid contaminant fraction. The vapor fraction may be compressed to generate a temperature differential in the reboiler exchanger with the vapor fraction being passed into contact with a reboiler exchanger to provide a stream of condensed vapor from the reboiler. The stream may be circulated through the reboiler exchanger and the heated separator to maintain from about 1% to about 50% by mass vapor in the stream. The apparatus includes a unique configuration of a vapor compressor, heated separator in combination with a forced circulation circuit to generate the decontamination result.
Patent CZ-9702552-A3 (CZ)
Inventor: WHITAKER RICHARD JEFFREY
IPC: F16M13/02
Filed: 1996-02-22
Abstract: Podpěrný držák TV-přijímače obsahuje plošinu (9) pro
uchycení a podepření televizního přístroje. Plošina (9) je
podepřena podpěrnými prostředky. Výztužný článek (5) vede
od prostředků, podpírajících plošinu (9), ke stěnové desce (3),
přizpůsobené k namontování podpěrného držáku. Stěny pláště
určují prostor pro přijímání kabelu. TV-přijímač je montován
na podpěrný držák. Držákje uspořádaný tak, že kabely TVpřijímače
jsou vedeny nejmenší částí podpěrného držáku pro
připojení na síť.
Patent CZ-258695-A3 (CZ)
Inventor: HAJEK JAROMIR
IPC: F17D1/00
Filed: 1995-10-05
Abstract: Podtlakový zásobník {1) je potrubím (4) s uzávěrem
(8) spojen s nádobou (2) opatřenou odváděcím
potrubím (5) s uzávěrem (9), do nádoby
(2) ústí potrubí (6) pro zdroj podlaku a
potrubí (7) pro zdroj tlakového vzduchu.
Alternativně je odváděči potrubí (5) napojeno
na čerpadlo (13).
Patent CZ-264098-A3 (CZ)
Title: Syringe with electronic presentation of parameters
Inventor: JENSEN JENS MOLLER
IPC: A61M5/31
Filed: 1997-02-20
Abstract: A syringe having a dose setting mechanism, a button which can be operated to inject a set dose, a switch operated at a time between the start and the completion of the injection and an electronic representation of parameters such as magnitudes of the set dose and the latest injected dose, which syringe further has a stop watch which is reset and started when the switch is operated. The status of the watch function is electronically represented and is together with the electronic represented parameters reproduced in a display showing the number of hours passed since the operation of the switch by switching on a corresponding number of 30 DEG  segments of a circle. Dose sizes are shown by common Arabic numerals.
Patent CZ-9903927-A3 (CZ)
Title: Casing, preferably for ventilation, heating and/or air conditioning devices
Inventor: SCHUBASCHITZ KLAUS
IPC: F16M1/08
Filed: 1999-11-05
Abstract: A sheet metal housing (1) for an air conditioning, heating or ventilation unit consists essentially of top and bottom panels, and sidewalls. The sheet metal edges have especially a U-shaped profile which forms the link between adjacent panels, secured by rivets, screws, spot welding or welded seams. The panel inner faces bear insulation material.
Patent CZ-410497-A3 (CZ)
Title: Axial mounting of open-end spinning machine
Inventor: WINZEN LOTHAR
IPC: F16C39/06
Filed: 1997-12-18
Abstract: A thrust bearing for an open-end spinning rotor (1) supported by its rotor shaft (2) in the bearing slot of a support-disk bearing arrangement (4). The thrust bearing has a magnetic bearing system (10) or (25) comprising magnetic support elements (12), (13) stationarily arranged on a thrust bearing housing (11) and a rotating magnetic bearing device (14) fastened to rotor shaft (2). Bearing element (15) of magnetic bearing device (14) is releasably connected to rotor shaft (2) via an elastic connection (20), (21) positively supported in corresponding receiving grooves (22), (23) of either the rotor shaft or the magnetic bearing device (14).
Patent ES-181395-A3 (ES)
Title: MEJORAS EN LA CONSTRUCCIoN DE VEHiCULOS MOTORES PARA FERROCARRILES DE JUGUETE
IPC: A63H19/22
Filed: 1947-12-31
Abstract: Mejoras en la construcción de vehículos motores para ferrocarriles de juguete, caracterizadas porque en cada uno de sus carros giratorios y solidario del eje de las ruedas motrices va dispuesto un cilindro estriado, de forma y dimensiones adecuadas para que, en todas las posiciones que en las curvas tome el referido carro, engrane con la rueda dentada de accionamiento, situada en la caja del vehículo y movida por el motor dispuesto en él.
Patent ES-194756-A3 (ES)
Title: Un perfeccionamiento en el cierre hermético de envases.
Filed: 1950-09-23
Abstract: Perfeccionamiento en el cierre hermético de envases que consiste esencialmente en la aplicación sobre la junta del cierre recubriéndolo suficientemente una cinta de una materia plástica tal como una resina sintética fenólica polivinílica o acrílica o de otra materia similar que aplicada superficialmente reblandecida por la acción de un mordiente o agente levemente disolvente de dichas materias pueda adherirse fácilmente en parte al envase y en parte a su tapa o tapón o medio obturador fabricados de materiales absolutamente impenetrables quedando al secarse el mordiente o disolvente empleado fijada uno y otra recubriendo sobradamente la junta sin dejar el menor resquicio para el paso del aire o de la humedad incluso por sus extremidades que al quedar superpuestas quedan en iguales condiciones de hermeticidad sin perjuicio de que pueda retirarse fácilmente el recubrimiento cuando sea necesario abrir el envase bastando para ello sujetar una de tales extremidades y tirar violentamente de la misma para producir el desprendimiento total de la cinta que se realiza generalmente dada la consistencia y continuidad del material de que está formada sin peligro de roturas dificultadoras.
Patent ES-8802472-A3 (ES)
Title: Tubular components for gymnastic equipment
IPC: A63G31/00
Filed: 1986-02-18
Abstract: A structure is assembled from components which can be spatially arranged in a number of different ways. The components have at least one circular end face with a screw thread connector. Each component has an internal thread (10) at one end and an external thread (11) at the other end. - The screw threads are multiple start so that two components can be screwed together in several different relative angular positions.