baber/WOPTO huggingface dataset:
Patent FI-942598-A0 (FI)
Inventor: LANG HANS-JOCHEN
IPC: C07C279/22
Filed: 1994-06-02
Abstract: There are described benzoylguanidines of the formula I <IMAGE>  where   R(1) is H, Hal, -NO2, -C IDENTICAL N, Xo-(CH2)p-(CF2)q-CF3, R(5)- SOm, R(6)-CO- or R(6)R(7)NO-SO2-, where X is O, S, NR(14), m is 0-2, o is 0, 1, p is 0-2, q is 0-6, R(5) and R(6) are alk(en)yl, -CnH2n-R(8), CF3, n is 0-4, R(8) is cycloalkyl, phenyl, R(6) also being H,   R(2) is <IMAGE> where Y is O, -S- or -NR(12)-; R(11), R(12) = H, alkyl, and h is zero or 1, and i, j and k are 0-4,  but where h, i and k are not simultaneously zero, R(3) is defined as R(1), or is alkyl, -X-R(13) where X is O, S, NR(14), R(14) is H, alkyl, R(13) is H, (cyclo)alkyl, -CbH2b-R(15) where b is 0-4,  R(15) is phenyl,   R(4) is H, -OR(16) or -NR(16)R(17) where R(16), R(17) are H, alkyl  and their pharmaceutically tolerable salts. They are obtained from a compound II <IMAGE> by reaction with guanidine, in which R(1) to R(4) have the meaning indicated and L is a leaving group which can be easily nucleophilically substituted. The compounds are outstandingly suitable as antiarrhythmic medicaments having a cardioprotective component for infarct prophylaxis and infarct treatment and also for the treatment of angina pectoris, where they also preventively inhibit or severely decrease the pathophysiological processes in the formation of ischaemically induced damage, in particular in the elicitation of ischaemically induced cardiac arrhythmias.
Patent FI-946053-A0 (FI)
Inventor: ILM MYOEH
IPC: A22C13/00
Filed: 1994-12-23
Abstract: The invention is concerned with a method of destruction of sausage skins and other mainly cellulosic substances by means of dissolution with an enzyme solution. In the method enzymes are added to a reactor that contains a water solution, after or before which the substances to be dissolved are added to the reactor. The substances to be dissolved are dissolved partly or completely, after which a new amount of substances to be dissolved are added to the reactor. When the enzymes have been adsorbed into the new substances to be dissolved, the solution containing the substances dissolved are recovered by separating the solution and the substances to be dissolved from each other, whereby water is added to the substances to be dissolved and if desired, the four foregoing steps are repeated a wished amount of times.
Patent FI-951556-A0 (FI)
Inventor: EVAIN ERIC J
IPC: D06M101/00
Filed: 1995-03-31
Abstract: A process for preparing thermal bondable fibers including exposing molten fiber grade polymer to electromagnetic radiation at the one or more orifices of the spinneret and the upper portion of the spin line, and the fibers prepared therefrom.
Patent FI-954798-A0 (FI)
Inventor: HOFMANN KARL-HEINZ
IPC: E04D13/17
Filed: 1995-10-09
Abstract: The invention relates to a ventilation strip (10; 110) for ventilating the eaves, a ridge or an edge of a roof, with at least one section (12; 114, 116) extendable along the ventilation strip (10; 110) which can be fitted to the shape of contoured roofing panels, and a section (14; 112) which is substantially rigid along the ventilation strip (10; 110) and parallel to the first section. The extendable section (12; 114, 116) has elongated holes and/or slots (30) in mutually staggered rows transversely to the ventilation strip (10; 110) and the elongated holes and/or slots (30) in one row are separated by at least one longitudinal web (34) running along the ventilation strip (10; 110). A ventilation strip (10) for the eaves may have apertures (20) for guttering brackets (70) and in a strip (110) for ridges or edges there may be an extendable section (114, 116) on either side of the rigid section (112). The extendable section (114, 116) may be folded in a zigzag with longitudinal fold lines (122, 124, 126, 128). There may ben an air-permeable and/or waterproof material covering (134) extendable longitudinally and transversally at least in the extendable section (12).
Patent IL-63038-A0 (IL)
Title: Vinblastine derivatives
IPC: A61K31/395
Filed: 1981-06-04
Abstract: Amino acid derivatives of vinblastine, including peptide derivatives, methods of their preparation and pharmaceutical compositions containing such vinblastine derivatives for use as antitumor agents are described.
Patent IL-74842-A0 (IL)
Title: Method of modifying taste
IPC: A23G9/52
Filed: 1985-04-09
Abstract: The sweetness of an ingestible product or oral composition containing a sweetening sugar or sugar alcohol in relatively large quantities can be reduced and/or the flavour enhanced by incorporation of at least one compound of the general formula (I)in which m represents 0 or 1, A represents a homocyclic or heterocyclic aromatic group with one or more rings; and B represents a hydrogen atom, a lower aliphatic group with 1-3 carbon atoms or a phenyl group; or, when m represents 0, A and B together represent a bivalent homocyclic or heterocyclic aromatic group with two or more rings, or a methylidene group carrying as a substituent a homocyclic or heterocyclic aromatic group with one or more rings; an aromatic ring of A, or of A and B together, optionally carrying one to three substituents selected from lower alkoxy groups, lower alkyl alkenyl groups, formyl or acetyl groups, hydroxy groups or acyloxy groups, and halogen atoms;C represents a hydrogen atom or an alkyl group or, when m represents 0, a hydroxy or alkoxy group;D represents an oxygen or sulphur atom;X<sup>+</sup> represents a hydrogen ion or another physiologically compatible cation;with the proviso that m represents 1 when S represents a substituted or unsubstituted phenyl group and Band C both represent hydrogen atoms; or when A represents an unsubstituted phenyl group, B represents an alkyl group and C represents a hydrogen atom.
Patent IL-80510-A0 (IL)
Title: Improved yeast strains
IPC: A21D8/04
Filed: 1986-11-05
Abstract: Process for increasing the rate of production of carbon dioxide, ethanol and other fermentation products such as citric acid, produced by yeast such as Saccaromyces cerevisiae during fermentation and decreasing biomass production by regulating the rate of glycolysis indirectly through changing the energy balance of the cell, i.e. by reducing intracellular ATP levels. Modifications for so altering the glycolysis rate involve the use of either a regulated ATP hydrolysis within the cell or a regulated leakage of ATP from the cell. This invention encompasses several ways for altering the yeast ATP level including (a) engaging futile metabolic cycles to increase ATP consumption; (b) using an altered exocellular acid phosphatase so that it becomes intracellular to increase intracellular ATP hydrolysis; (c) using a drug which uncouples the plasma membrane ATPase thereby consuming an abnormally high level of ATP; and (d) using a drug which allows the release of ATP from the cell to lower the intracellular ATP level. This invention further encompasses regulating the genetic modifications described in greater detail herein. By these means, such modifications may be turned off during growth of the yeast on a commercial scale, and then turned on before or during, and preferably before or at a very early stage of, the dough-rising phase.
Patent IL-90428-A0 (IL)
Title: Precipitated calcium carbonate-cationic starch binder as retention aid system for papermaking
IPC: D21H17/29
Filed: 1989-05-26
Abstract: A two component binder system comprising a highly dispersible, high specific surface area precipitated calcium carbonate (colloidal PCC) and a cationic starch, especially a cationic potato starch, for improving filler retention, opacity and strength during papermaking.
Patent IL-92222-A0 (IL)
Title: New insulin derivatives,the use thereof,and pharmaceutical compositions containing them
IPC: C07K14/62
Filed: 1989-11-06
Abstract: Insulin derivatives of the formula II with an isoelectric point between 5 and 8.5, with improved stability in weakly acid aqueous medium and with specific action profile and the physiologically tolerated salts of these insulin derivatives for the treatment of diabetes mellitus; formula II is: <IMAGE> in which R<1> is H or H-Phe, R<2> is a genetically encodable L-amino acid which contains no amide group, R<3><0> is the residue of a neutral, genetically encodable L-amino acid, R<3><1> is a physiological acceptable organic group which is basic in nature and has up to 50 C atoms, in whose structure 0 to 3  alpha -amino acids are involved and whose terminal carboxyl group which is present where appropriate can be free, in the form of an ester, in the form of an amide, in the form of a lactone or reduced to CH2OH, and X is a genetically encodable L-amino acid.
Patent IL-94049-A0 (IL)
Title: Benzimidazole derivatives,their preparation and pharmaceutical compositions containing them
IPC: C07D487/04
Filed: 1990-04-08
Abstract: The invention relates to benzimidazoles of the formula <IMAGE>  in which R1 to R6 are defined as in claim 1, their 1- and 3-isomer mixtures and their acid addition salts, which have useful properties. The novel compounds are in particular angiotensin II antagonists.
Patent FI-20040537-A0 (FI)
Inventor: LINDBERG HARRI
IPC: B65B25/14
Filed: 2004-04-14
Abstract: An assembly for moving paper, board and cellulosic web rolls in a roll packaging system includes a plurality of roll handling stations incorporating at least one receiving station for the entry of rolls into the system, one wrapping station for winding at least one wrapper course on the periphery of the rolls, and at least one other station, and an indexing conveyor having a car for moving the rolls which is adapted to move synchronously into positions coinciding with each one of said roll handling stations. The car of the indexing conveyor is adapted to move on at least three different elevation levels named as a base elevation level 0, a first elevation level and a second elevation level. Additionally, at least a portion of the car coinciding with one station is on an elevated level in regard to the other parts of the car coinciding with the other stations.
Patent FI-20090317-A0 (FI)
Inventor: RAHARDJO ANDHIKAPUTRA
IPC: E06B/
Filed: 2009-09-03
Abstract: Door arrangement, more particularly a sliding door arrangement of an automatic door of an elevator or of a building, which comprises a door panel, and a guide arrangement for controlling the path of movement of the door panel, which guide arrangement comprises at least one guide connected to the aforementioned door panel, and a guide rail, closely along which the aforementioned guide is arranged to move, and from which guide rail the guide takes lateral support force with respect to the longitudinal direction of the guide rail. The guide comprises a first guide roll for taking the support force from the guide surface of the guide rail on the side of a first side of the guide, and a second guide roll for taking support force from the guide surface of the guide rail on the side of a second side of the guide.
Patent IL-111293-A0 (IL)
Title: Pharmaceutical compositions comprising 5 alpha-reductase type 2 inhibitor for treating androgenic alopecia
IPC: A61P29/00
Filed: 1994-10-13
Abstract: The instant invention involves a method of treating and/or reversing androgenic alopecia and promoting hair growth, and methods of treating acne vulgaris, seborrhea, and female hirsutism, by administering to a patient in need of such treatment a 5 alpha -reductase 2 inhibitor such as finasteride, in a dosage amount under 5 mgs/day.
Patent IL-118417-A0 (IL)
Title: Impact absorbing macadam
IPC: E01C7/26
Filed: 1996-05-26
Abstract: PCT No. PCT/GB96/01240 Sec. 371 Date Mar. 23, 1998 Sec. 102(e) Date Mar. 23, 1998 PCT Filed May 23, 1996 PCT Pub. No. WO96/37658 PCT Pub. Date Nov. 28, 1996An impact absorbing macadam comprises 10 to 75% (preferably 25 to 45%) of a particulate rubber having a particle size of up to 40 mm, 25 to 90% (preferably 45 to 65%) of an aggregate having a particle of up to 40 mm and from 5 to 9% of a polymer modified bituminous binder. Typically such a macadam has a void volume, interconnected or unconnected, of from 5 to 25%. The polymer which modifies the bituminous binder is preferably an unbranched styrene butadiene styrene block copolymer forming about 7% of the modified binder. The macadam is suitable as a base for sports pitches and athletic tracks without a rubber shock pad overlay.
Patent IL-124357-A0 (IL)
Title: Device for image projection
Inventor: KRAENERT JUERGEN DR
IPC: H04N5/74
Filed: 1997-09-06
Abstract: PCT No. PCT/EP97/04834 Sec. 371 Date May 28, 1998 Sec. 102(e) Date May 28, 1998 PCT Filed Sep. 6, 1997 PCT Pub. No. WO98/15127 PCT Pub. Date Apr. 9, 1998In an arrangement for displaying images on a projection screen, which arrangement includes a laser, which emits a laser beam, and a deflecting device, which is provided for deflecting the laser beam, and an image-generating device which is connected to a controlling device for controlling the laser and the deflecting means. The image-generating device is switchable in two operating modes, the first operating mode being the standard operating mode for projecting, and the second being an operating mode in which the laser radiation is harmless to a person disposed in the region to which the laser has access. In this regard, a safety circuit is provided and comprises at least one sensor, by which a monitored region, which is larger than the region accessible to the laser, between the image-generating means and the projection screen is monitored as to the presence of objects, wherein the image-generating means is switchable into the second operating mode by means of the safety circuit, in the event of an object being present.
Patent IL-132068-A0 (IL)
Title: A stab-resisting material a coated carrier to be used therewith and clothing made of said material
IPC: A41D31/00
Filed: 1998-04-03
Abstract: A stab-resisting material includes a carrier coated with solid particles, which is provided on a packet of fabrics, in which the coating on the carrier includes abrasive particles having a diameter of 0.1-3 mm, and in which the packet of fabrics is thicker than 1.5 mm. The abrasive particles may be provided on the carrier by an adhesive, which forms an elastic film after curing. In particular, a fabric made of Aramid or Nylon fibres may be used as the carrier material. The preferred adhesive is a bituminous adhesive or an adhesive with a base of polyurethane. This material is used in particular in protective clothing.
Patent IL-132077-A0 (IL)
Title: Process for producing 1-chlorocarbonyl-4- piperidinopiperidine or hydrochloride thereof
IPC: C07D211/60
Filed: 1998-03-31
Abstract: The present invention provides a highly safe and easily operable process for producing 1-chlorocarbonyl-4-piperidinopiperidine or hydrochloride thereof in a high yield. Described specifically, the present invention relates to a process for producing 1-clorocarbonyl-4-piperidinopiperidine or hydrochloride thereof, which comprises reacting 4-piperidinopiperidine with a trialkylsilyl halide to obtain a 4-piperidinopiperidinyl trialkylsilyl, reacting it with a carbon dioxide gas to obtain a 4-piperidinopiperidinyl trialkylsilyl carbamate derivative, reacting the derivative with thionyl chloride or the like to obtain 1-chlorocarbonyl-4-piperidinopiperidine hydrochloride and optionally treating it with a strong base.
Patent IL-136409-A0 (IL)
Title: Morpholino end-capped, hindered amine substituted aminotriazine and their use as light stabilizers
IPC: C07D401/14
Filed: 1998-11-03
Abstract: Novel morpholino end-capped polyamino-1,3,5-triazines, methods for their use as light stabilizers for materials which are subject to degradation (for example, by actinic radiation), stabilizer compositions based on these morpholino end-capped polyamino-1,3,5-triazines and methods for their synthesis are herein described.
Patent IL-139163-A0 (IL)
Title: A method of predicting the ability of compounds to modulate the biological activity of receptors
IPC: C07K1/04
Filed: 1999-03-26
Abstract: The ability of a query compound to modulate the biological activity of a receptor in a multicellular organism is predicted on the basis of its interaction with that receptor in the presence of various member of a panel of BioKeys. The BioKeys are ligands, especially peptides or nucleic acids, known to modify the conformation of the receptor. This interaction data, known as a "fingerprint", is compared to the fingerprints for reference compounds with known biological activities mediated by that receptor. In the "molecular braille" (MB) embodiment of the present invention, the reference and test fingerprints are based on in vitro (cell-free) assays. In the "cellular-braille" (CB) embodiment of the present invention, the reference and test fingerprints are based on cellular assays (but not on assays of whole multicellular organisms, or their organs or tissues).
Patent IL-146631-A0 (IL)
Title: Diagnostics and therapeutics for cardiovascular disorders
IPC: C12N15/09
Filed: 2000-05-26
Abstract: The kits and methods of the present invention relate to the diagnosis of cardiovascular disorders.
Patent IL-154198-A0 (IL)
Title: Unidirectional, adjustable flap valves
IPC: F24F11/00
Filed: 2003-01-30
Abstract: The invention provides a flap valve (2) for controlling the air pressure within a protected space defined by walls, the flap valve including a valve frame (6) attachable to an opening made in the walls, a valve flap (8), articulated at least indirectly to the frame and being subjectable to both a sealing force which forces the valve flap against the valve frame and to an opening force which lifts a portion of the flap off the valve frames. The flap valve (2) has a first position in which the protected space is sealed off from a contaminated environment, and a second position in which air from the protected space is allowed to escape into the environment via the opening, wherein the sealing force is constituted by at least one spring (22) at least indirectly attached to the valve flap (8) and the valve frame (6). <IMAGE>
Patent IL-154265-A0 (IL)
Title: System for enhanced chemical debridement
IPC: A61M1/00
Filed: 2001-07-30
Abstract: A device, system and method for enhancing the functionality and efficiency of a chemical and/or enzymatic debriding agent with a physical debriding mechanism. The debriding agent alone and the physical mechanism alone are each capable of at least some debriding activity separately, without being used in the combination. In combination, however, they are more effective, such that the debriding efficacy is increased for the combination. Preferably, the physical debriding mechanism comprises an ultrasound source.
Patent IL-172731-A0 (IL)
Title: Barrier formulation comprising a silicone based emulsion
IPC: A61K8/06
Filed: 2005-12-21
Abstract: The present invention provides an improved barrier formulation that is useful in a number of applications, and a method for its manufacture. The formulation comprises an emulsion having at least an oil phase and an aqueous phase wherein the oil phase comprises a silicone compound wherein the viscosity of the formulation is 20000 cps or less.
Patent IL-187879-A0 (IL)
Title: A method of treating fruit or vegetables, and a corresponding plant
Filed: 2007-12-04
Abstract: The process for treating fruits or vegetables, comprises collecting a conditioning means (33) containing the fruits or vegetables in a block (35) significantly compact in a housing (8) bounded by a belt on the side walls (9, 11) inside an enclosure (3), bringing each deformable side wall in its thread configuration of the block, and longitudinally passing the housing by a treating composition having a temperature of 48-52[deg] C with a flow of 50-100m 3>/m 2>/h and a duration of 2-3 minutes. The sidewalls extend according to a longitudinal direction. The process for treating fruits or vegetables, comprises collecting a conditioning means (33) containing the fruits or vegetables in a block (35) significantly compact in a housing (8) bounded by a belt on the side walls (9, 11) inside an enclosure (3), bringing each deformable side wall in its thread configuration of the block, and longitudinally passing the housing by a treating composition having a temperature of 48-52[deg] C with a flow of 50-100m 3>/m 2>/h and a duration of 2-3 minutes. The sidewalls extend according to a longitudinal direction, where one of the side wall is deformable between a thread configuration and release configuration of the block. The treating composition contains phosphorous acid, which has a concentration of 2000-4000 ppm. The treating composition is applied at a rate of 3000-10000 liters for 100-300 ton of fruits or vegetables to be treated. An independent claim is included for an installation for treating fruits or vegetables.
Patent IL-197385-A0 (IL)
Title: Methods for determining a cursor position from a finger contact with a touch screen display
Filed: 2009-03-03
Abstract: A portable device with a touch screen display detects a contact area of a finger with the touch screen display and then determines a first position associated with the contact area. The cursor position of the finger contact is determined, at least in part, based on: the first position, one or more distances between the first position and one or more of the user interface objects; and one or more activation susceptibility numbers, each associated with a respective user interface object in the plurality of user interface objects. If the cursor position falls into the hidden hit region of a virtual push button on the touch screen display, the portable device is activated to perform operations associated with the virtual push button.
Patent RO-131090-A0 (RO)
Title: Ecological toothpaste with multiple implications
Inventor: EARAR KAMEL
IPC: A61K8/97
Filed: 2015-10-16
Abstract: The invention relates to an ecological toothpaste. According to the invention, the paste comprises, in gravimetric parts, 35...40 parts of egg shell crumb, 12...15 parts of decorticated rice crumb, 12...15 parts of aromatic plants crumb: mint and rosemary and cardamom seeds, 6...8 parts of sodium bicarbonate, 2...3 parts of sea salt, and the remainder up to 100 parts, emulgel consisting of 55...60% deionized or distilled water, 5...6% mint essential oil, 8...10% pineapple juice and pomegranate juice, respectively, in which 20...25% colloidal cream of sesame and hemp seeds is dispersed in a mass ratio of 3 : 2, the product having a good paste stability, without phase segregation, and a consistency similar to commercial toothpastes.
Patent RO-135389-A0 (RO)
Title: Anti-friction alloys improved by micro-alloying
Inventor: AVRAM VASILE
IPC: F16C33/00
Filed: 2021-08-23
Abstract: The invention relates to anti-friction alloys micro-alloyed with Ca and Mg, of YSn83Ca and YSn83Mg type,  which confer the alloys properties directly related to the lubrication process or contribute to the improvement of their workability. According to the invention, the alloys have the following chemical composition: a. the YSn83Ca alloy comprises 0.2...0.5% Ca, 82...84% Sn, 10...12% Sb, 5.5...6.5% Cu and impurities of maximum 0.25% and b. the YSn83Mg alloy comprises 0.2...0.5% Mg, 82...84% Sn,  10...12% Sb, 5.5...6.5% Cu and impurities of maximum 0.25%, for which values of the friction coefficient ranging between 0.0663...0.1286 were obtained, values which are improved by 59% as compared to those of the commercial alloy YSn83.
Patent AP-2001002319-A0 (AP)
Title: Pyrimidine-2,4,6-trione metalloproteinase inhibitors.
Inventor: NOE MARK CARL
IPC: A61P1/16
Filed: 2001-10-17
Abstract: The present inventin relates to pyrimidine-2,4,6-trione metalloproteinase inhibitors of the formula wherein x, y, a, b and r1 are as defined in the specification, and to pharmaceutical compositions and methods of treating infalammation, cancer and other disorders.