baber/WOPTO huggingface dataset:
Patent JP-2788118-B2 (JP)
IPC: C07C303/30
Filed: 1990-09-05
Granted: 1998-08-20
Abstract: PCT No. PCT/GB90/01371 Sec. 371 Date Apr. 10, 1992 Sec. 102(e) Date Apr. 10, 1992 PCT Filed Sep. 5, 1990 PCT Pub. No. WO91/03460 PCT Pub. Date Mar. 21, 1991.4-[(2-chloroethyl)-(2-hydroxyethyl)-amino]benzoyl amino acids of formula (IV), wherein X represents a group (a), where Pro represents hydrogen or a straight or branched chain C1-6 alkyl group, and salts thereof, and processes for their production. The compounds are useful for the production of nitrogen mustard prodrugs    <IMAGE>  (IV)   <IMAGE>  (a)
Patent JP-3365634-B2 (JP)
IPC: A61K9/20
Filed: 1993-11-17
Granted: 2003-01-14
Abstract: Prepn. of a tablet contg. a bisphosphonic acid deriv. (BP), comprises (a) forming a mixt. contg. the BP, anhydrous or fast flow lactose, dry binder and disintegrant; (b) opt. adding compression aids, flavours, flavour enhancers, sweeteners, and preservatives; (c) lubricating with a lubricant; and (d) compressing to the desired tablet form. The (BP) are chosen from 4-amino-1-hydroxybutylidene-1,1-bisphosphonic acid; and its N-methyl and N,N-dimethyl analogues, 3-amino-1-hydroxypropylidene-1,1-bisphosphonic acid and its N,N-dimethyl and N-methyl-N-pentyl analogues; 1-hydroxy-2-(3-pyridyl)ethylidene-1,1-bisphosphonic acid and 4-hydroxymethylene-1,1-bisphosphonic acid piperidine; or their salts. More pref. is 4-amino-1-hydroxybutylidene -1,1-bisphosphonic acid (BP-1) partic. as monosodium salt trihydrate (BP-2). The dry binder is microcrystalline cellulose (MC). The disintegrant is modified starch or cellulose polymer, croscarmellose sodium (CC-Na) or a mixt. esp. CC. The lubricant is Mg stearate. Compsn. range is basic BP 0.5-25, lactose 30-70, MC 30-50, CC-Na 0.5-5 and mg stearate 0.1-2, all %. Closer limits, for BP-2 are BP-2 1-25, lactose 40-60, MC 35-45, CC-Na 0.5-2, and Mg stearate 0.1-1 all %.
Patent JP-3441458-B2 (JP)
IPC: C07D409/12
Filed: 1993-12-13
Granted: 2003-09-02
Abstract: This invention provides 7-deoxy-taxol analogs of Formula I: The compounds of Formula I (including II and III) are useful for the same cancers for which taxol has been shown active, including human ovarian cancer, breast cancer, and malignant melanoma as well as lung cancer, gastric cancer, colon cancer, head and neck cancer, and leukemia.
Patent JP-3679806-B2 (JP)
IPC: D21D5/26
Filed: 1994-12-21
Granted: 2005-08-03
Abstract: PCT No. PCT/FI94/00578 Sec. 371 Date Jun. 19, 1996 Sec. 102(e) Date Jun. 19, 1996 PCT Filed Dec. 21, 1994 PCT Pub. No. WO95/17235 PCT Pub. Date Jun. 29, 1995A process and apparatus for pumping a fluid mixture of a gas and a liquid and for separating said gas and liquid from each other, said apparatus having a fluid inlet (14) at one end (18) and at the opposite end (22) a pump housing (16) with a liquid outlet (28) and, between said inlet (14) and said pump housing (16), a hollow elongated gas separation part (30) of an essentially circular cross section with a generally central outlet (26) for separated gas. Said gas separation part (30) is provided by a hollow rotor (12) between said inlet (14) and said pump housing (16), the inner wall of said rotor (12) providing a large rotatable gas separation surface (32). The diameter of said rotor (12) increases at said opposite end (22) of the apparatus to form a larger diameter pumping zone (17) extending into said pump housing (16). Said rotor (12) is provided with a blade wheel (24) extending into said pump housing (16). The apparatus is especially well suited for the gas-free re-cycling of backwater drained through a forming fabric in a papermaking process. The invention is also applicable to the removal of air from fluid materials separated by flotation.
Patent JP-3468515-B2 (JP)
IPC: A61P43/00
Filed: 1991-10-30
Granted: 2003-11-17
Abstract: A combined preparation for simultaneous combined, simultaneous separate, or sequential use in the therapy or prophylaxis of disorders associated with undesirably high levels of TNF, e.g. septic or endotoxic shock and immunoregulatory and inflammatory disorders, which comprises an antibody to TNF or a TNF binding fragment thereof and a xanthine derivative. Particular preferred xanthine derivatives are 3,7-dimethyl-1-(5-oxo-hexyl)xanthine (known as Pentoxifylline or Trental) and 1-(5-hydroxy-5-methylhexyl)-3-methylxanthine and similar compounds. The anti-TNF antibody or fragment is preferably monospecific especially a humanised recombinant antibody or fragment. The ratio of xanthine derivative to anti-TNF antibody component used may be in the range between 450:1 and 1:10 and doses of anti-TNF component in the range 0.001-30mg/kg/day and doses of xanthine derivative in the range 0.5 to 100mg/kg/day may be administered during treatment of human or animal subjects. It has been found that when an anti-TNF antibody and a xanthine derivative are used together in some experimental models of septic shock, a surprising combination effect is observed.
Patent JP-3502637-B2 (JP)
IPC: F21V21/03
Filed: 1994-12-29
Granted: 2004-03-02
Abstract: A fitting (70) for covering the fixation point of a cord (80) to a ceiling surface has a hollow body (71) which defines an outer curved plane and an inner cord passage cavity (72). To facilitate a fitting or fixation of the fitting (70) after the suspension and connection of an electrical appliance such as a swinging lamp, and to facilitate a subsequent dismantling of the fitting (70) for the purpose of cleaning and/or replacement, the hollow body (71) has two parts (82, 84) which are interconnected through a hinge (86) and thus rotatable with respect to each other between a first position, in which the body (71) is opened so that the cord (80) can be introduced freely into the inner cord passage cavity (72), and a second position, in which the body (71) is closed and encircles the cord (80), the cord being received in the inner cord passage cavity. The fitting (70) preferably has locks (90, 92, 94 and 96) for locking the two parts (82 and 84) in said second position, i.e. in the position in which they encircle the cord.
Patent JP-3157165-B2 (JP)
IPC: C07F7/18
Filed: 1994-03-24
Granted: 2001-04-16
Abstract: The present invention is directed to novel taxanes useful as chemotherapeutic agents or their precursors. Processes for preparing the novel taxanes include coupling reactions, in the presence of a base, of baccatin of formula (III) or (IV)    <IMAGE>rmula (V).    <IMAGE>  (V)  The invention also provides pharmaceutical compositions including the novel taxanes and method for treatment of certain cancers with these new compounds.
Patent JP-3420238-B2 (JP)
IPC: B41M1/40
Filed: 1994-05-05
Granted: 2003-06-23
Abstract: A molded closure for a liquid container comprising a thermoplastic elastomer and a blowing agent. The molded closure is particularly suitable for use as a synthetic wine cork in a wine bottle. The molded closure does not permit passage of oxygen into the container, does not absorb oxygen from the contents of the container, can be removed from the container using a corkscrew without significant expansion, crumbling or disintegration, does not significantly taint a liquid in the container, permits the container to be placed horizonzally immediately after insertion of the molded closure, and can permanently retain printed matter on its surface. <IMAGE>
Patent JP-3197277-B2 (JP)
IPC: C12Q1/68
Filed: 1994-04-28
Granted: 2001-08-13
Abstract: An assay reagent and a kit whereby nonspecific capture of a labeled substance by a solid phase can be suppressed and more than one antibody or more than one antigen can be detected via a simple assay by using one reagent. An immunological ligand assay reagent comprising components selected from the following groups (A) and (B) at the same time is reacted with immunogical ligands to thereby form complexes, which are captured by separate solid phases (C) and analyzed based on the labeling substance contained in each complex: group (A): more than one type of immunological antiligand-nucleotide conjugates wherein antibodies having specific avidities respectively for immunological ligands of different types are bonded to nucleotides which are specific respectively for said immunological ligands and each has an arbitrarily selected base sequence; group (B): labeled substances having specific avidities respectively for the immunological antiligands of different types which are to be assayed; and group (C): solid phase-nucleotide conjugates wherein nucleotides having base sequences capable of complementarily binding respectively to the nucleotides of the group (A) are bonded to a water-insoluble carrier. Either antigens or antibodies are applicable to said immunological ligands and immunological antiligands. <MATH>
Patent JP-3983303-B2 (JP)
IPC: F24C7/04
Filed: 1998-01-15
Granted: 2007-09-26
Abstract: Electric toaster with a first heating element arranged at one side of a toasting compartment and a second heating element arranged at an opposed side of the toasting compartment. The first heating element is divided into two sub-elements. Two diodes and a switch provide the possibility to switch over from a normal two-sided toasting mode to an asymmetric single-sided toasting mode. In the normal mode the switch is closed and the sub-elements receive power only during different half-waves of the mains supply voltage, so that the effective radiant power of the sub-divided first element is equal to the radiant power of the second heating element. In the asymmetric mode the switch is opened and the resistance of the first heating element is greater than the resistance of the second element, as a consequence of which relatively more radiant power is emitted by the first heating element than by the second heating element.
Patent JP-4263243-B2 (JP)
IPC: B29C45/26
Filed: 1997-05-20
Granted: 2009-05-13
Abstract: A process for the manufacturing of a pressure vessel made from a thermoplastic material or a thermosetting resin. The vessel comprises a first and a second vessel end part, and possibly an intermediate tube part. The vessel end parts include a circumfering shell (4) and each one dome (3). A number of partition and load distributing walls (5) stretch from the domes (3) towards the open part of each vessel end part. The possible intermediate tube part includes similar walls (5). The edges of the walls (5) will meet when the different parts are joined. A number of cells (6) are formed between the walls (5). A number of crossing areas are formed between intersecting walls (5). At least one crossing area is provided with a determination by achieving a hole (14) from the outside of the dome. The hole (14) is bigger than the crossing area and has a depth greater than thickness of the dome part (3).
Patent JP-4057069-B2 (JP)
IPC: B23B13/12
Filed: 1999-03-05
Granted: 2008-03-05
Abstract: The devices guides a bar that is advanced by the retractable collet of a bar feeder magazine to the mandrel of a lathe by employing an insert which is slidable with slight clearance within a duct that is connected to the mandrel. The insert has therethrough an axial passage registering at one end with an inlet end of the duct, which is disposed to receive the bar and collet, and the opposite end of the passage designed to be traversed by the bar with slight clearance. The insert is disposed to be engaged and impelled by the advancing collet along the duct a predetermined distance towards the mandrel, after which means is provided to engage and effect return of the insert to a starting position close to the inlet end of the duct upon re-extraction of the collet from the duct.
Patent ES-2293845-B2 (ES)
Title: Sistema de monitorizacion y control de procesos de tratamiento termico superficial de materiales con laser mediante un control neuronal adaptativo mediante modelo de referencia.
Inventor: PEREZ RODRIGUEZ JOSE ANTONIO
IPC: B23K26/352
Filed: 2006-09-25
Granted: 2008-12-16
Abstract: Sistema de monitorización y control de procesos de tratamiento térmico superficial de materiales con láser mediante un control neuronal adaptativo mediante modelo de referencia. Consiste en un sistema de monitorización y control en tiempo real de procesos de tratamiento térmico superficial de materiales con láser mediante control neuronal mediante modelo de referencia, que emplea como variable de entrada la máxima temperatura en la superficie del material y como variable de actuación la potencia de salida de la fuente láser. El sistema calcula cíclicamente la señal de actuación sobre la potencia de la fuente láser (8), en base al error de seguimiento (4). La señal de control sobre la potencia de la fuente láser (8) es calculada en dos etapas: en primer lugar, el controlador lineal tipo Proporcional, Integral y Derivativo, PID (5) genera, en base al error de seguimiento (4), la correspondiente actuación (6), y posteriormente, a partir de dicha señal y el estado del proceso (2), el controlador neuronal mediante modelo de referencia (7) calcula la señal de actuación sobre la fuente láser (8).
Patent ES-2346025-B2 (ES)
Title: Sistema para la simulacion de practicas quirurgicas.
Inventor: BAYONA BERISO SOFIA
IPC: A61B17/00
Filed: 2008-06-02
Granted: 2011-11-16
Abstract: Sistema que comprende un equipo informático (1) con una base de datos (11) de una parte anatómica y unos medios de visualización (2) de recreación visual de un modelo virtual, estando asociado un simulador (4) de la parte anatómica, palpable, posicionable y orientable en el entorno virtual generado por el equipo informático (1), mediante unos medios que proporcionan al usuario una información táctil específica de las diferentes zonas de la parte anatómica reproducida, con el fin de permitir un número indefinido de prácticas de localización táctil en dicho simulador -sin deteriorar el modelo anatómico- (4) de posibles portales de entrada para la zona subsidiaria a ser intervenida quirúrgicamente, mediante técnicas de cirugía de mínimo abordaje. El sistema comprende un simulador (5) de la herramienta posicionable sobre el simulador (4) de la parte anatómica para la interactuación de ambos en el entorno virtual mediante unos medios (3) de seguimiento y posicionamiento del simulador (4) y del simulador (5).
Patent ES-2337012-B2 (ES)
Title: Sistema y metodo de ajuste de retardo audio/video.
Inventor: MARTINEZ BARBERO JESUS
IPC: H04N5/04
Filed: 2009-12-17
Granted: 2010-09-17
Abstract: Sistema y método de ajuste de retardo
audio/vídeo que comprende las siguientes  etapas: extraer parámetros
característicos de una fuente de audio (3);  introducir los
parámetros extraídos de la fuente de audio (3) en el vídeo 
procedente de una fuente de vídeo (1); extraer de la señal de audio,
tras  el procesado del vídeo, los mismos parámetros extraídos en la
primera etapa;  obtener de la señal de vídeo, tras el procesado del
vídeo, los parámetros  de audio introducidos en la segunda etapa;
comparar los parámetros de audio  extraídos en la tercera etapa y
obtenidos en la cuarta; calcular el retardo  existente entre los
parámetros de audio comparados; almacenar el retardo  calculado; y
finalmente retardar la señal de audio un valor de retardo 
configurable en función del retardo calculado y del retardo
almacenado  procedente de una ejecución anterior del método.
Patent ES-2598902-B2 (ES)
Title: Mortero estructural aligerado y de baja porosidad fabricado con residuos de poliuretano
Inventor: CALDERON CARPINTERO VERÓNICA
IPC: C04B18/20
Filed: 2015-07-30
Granted: 2017-09-14
Abstract: La invención trata de un nuevo producto que incluye una base de mortero donde parte del árido o la totalidad del árido se ha sustituido por residuo de poliuretano espumado triturado. También se refiere a un método para preparar morteros aligerados pero con propiedades estructurales que comprende las etapas de amasado y dosificación de los diferentes componentes y la adición de una solución acuosa que comprende un 0.5% de al menos un agente tensioactivo que se introduce en la mezcla del conglomerado fresco en el momento del amasado.
Patent ES-2636713-B2 (ES)
Title: Dispositivo fotónico sensor, método de análisis de muestras que hace uso del mismo y usos de dicho dispositivo
Inventor: MUÑOZ MUÑOZ PASCUAL
IPC: G02B6/12
Filed: 2016-12-02
Granted: 2018-05-18
Abstract: Dispositivo fotónico sensor, método de análisis de muestras que hace uso del mismo y usos de dicho dispositivo.#Se describen en este documento un dispositivo sensor y un método de análisis de muestras que hace uso dicho dispositivo, basándose ambos en el uso de una sub-agrupación de guías que se usa como referencia junto con otra sub-agrupación de guías que presenta una serie de ventanas definidas en las guías de onda de tal manera que se dan variaciones en el campo de evanescencia de cada porción de las guías de onda de la ventana, o de las ventanas en el caso de formaciones de ventanas, que está en contacto óptico mediante la ventana con una porción de la muestra a analizar. Las mediciones de dichas variaciones con respecto a una medida de referencia que se toma de la sub-agrupación de referencia permiten determinar y cuantificar el analito de la muestra.
Patent AU-2001233744-B2 (AU)
Title: Exhaust system for watercrafts
Inventor: HELLMANN HANS KURT
IPC: B63H21/32
Filed: 2001-02-08
Granted: 2005-06-30
Abstract: Prior to leaving the exhaust pipe (1), the exhaust gases are made to flow through a section used to help reduce the heat of the sea water around the pipe exit. In this section at least one sump is provided, with a drainage tube (25) extending from the deepest point of the sump to a point around the boat.
Patent AU-2001239029-B2 (AU)
Title: Method for treating solid waste with an organic fraction
Inventor: VANDEVIVERE PHILIPPE
IPC: B03B9/06
Filed: 2001-03-06
Granted: 2004-10-14
Abstract: The present invention concerns a method for treating solid waste with an organic fraction. A slurry (4) of the waste (1) diluted with water (3) is sieved, at least by means of a sieving device (5) which lets pieces through whose dimension in at least one direction, and preferably in at least two standing directions, is situated between 2 and 20 mm, after which, from the slurry (7) which has passed through, a part of the ferrous metals (8) which are present in the waste (1) is removed from said waste by means of magnets, and the slurry (7) is finally dewatered.
Patent AU-2001286939-B2 (AU)
Title: Oximeter sensor with digital memory encoding patient data
Inventor: MANNHEIMER PAUL D
IPC: G01D18/00
Filed: 2001-08-31
Granted: 2005-03-24
Abstract: Embodiments of the present invention include systems and methods that relate to pulse oximetry. Specifically, one embodiment includes an oximeter sensor comprising a light emitting element configured to emit light, a light detector configured to detect the light, and a memory chip having a built-in trimmed resistor, the trimmed resistor having a resistance value that is detectable by a monitor.
Patent AU-2001294437-B2 (AU)
Title: Flame retardant for polymeric materials
Inventor: BUTYLKINA NATALIYA GRIGORIEVNA
IPC: B27K3/36
Filed: 2001-07-16
Granted: 2007-11-29
Abstract: A flame retardant predominantly of polymeric materials, appearing as a novel chemical compound, viz, ammonium salt of nitrolotris(methylene)phosphonic acid amide.
Patent AU-2002326898-B2 (AU)
Title: Load transfer plate for in situ concrete slabs
Inventor: PARKES NIGEL K
IPC: E01C11/14
Filed: 2002-09-13
Granted: 2008-01-17
Abstract: A tapered load plate transfers loads across a joint between adjacent concrete floor slabs. The top and bottom surfaces may taper from approximately 4 inches wide to a narrow substantially pointed end over a length of approximately 12 inches. The tapered load plate accommodates differential shrinkage of cast-in-place concrete slabs. When adjacent slabs move away from each other, the narrow end of the tapered load plate moves out of the void that it created in the slab thus allowing the slabs to move relative to one another in a direction parallel to the joint. Tapered load plates may be assembled into a load-plate basket with the direction of the taper alternating from one tapered load plate to the next to account for off-center saw cuts. A tapered load plate and an end cap may be used to provide load transfer across an expansion joint.
Patent AU-2002343969-B2 (AU)
Title: Floor laying material, piece mat, and arranging structure thereof
Inventor: NAKAMURA TOSHIYUKI
IPC: B32B7/02
Filed: 2002-10-10
Granted: 2008-01-03
Abstract: A floor laying material, a piece mat, and an arranging structure thereof whose sound absorbing property and sound insulating property are optimized. Floor laying material (10) comprises carpet layer (11) having joining strips (11a) of thermoplastic resin discontinuously arranged on the back surface thereof, and buffer material layer (12) layered to the back surface of carpet layer (11) through joining strips (11a). Carpet layer (11) has its front-to-back flow resistance value adjusted between 100 Nsm<-3> and 1000 Nsm<-3.> Further, buffer material layer (12) is made of a material having an air wrapping property and has its front-to-back flow resistance value adjusted between 40 Nsm<-3> and 800 Nsm<-3>. <IMAGE>
Patent AU-2003222830-B2 (AU)
Title: Core material
Inventor: SCHREY ALEXANDER
IPC: B22C9/12
Filed: 2003-04-19
Granted: 2008-10-09
Abstract: A method for the production of cores and molds for casting molds, based on a base molding material and an organic or inorganic binding agent and an additive. According to the method, pre-forming substances are used in order to dispense with the use of sizing substances and to prevent the formation of ribs.
Patent AU-2003236729-B2 (AU)
Title: Method and device for reducing the NOx and N2O of gases
Inventor: SCHWEFER MEINHARD
IPC: B01D53/86
Filed: 2003-06-10
Granted: 2009-05-07
Abstract: To reduce the content of NO 2 and NOx in process and exhaust gases, they are passed over two catalyst beds (4,5) in succession, containing one or more zeolites charged with iron, between the gas inflow (1) and outflow (2). An agent for the reduction of NOx is fed (3) into a mixer (6) between the catalyst beds, and the bed temperatures are set at = 500 [deg] C. The gas pressure is adjusted to at least 2 bar in both beds. The spatial speed is selected through the ring channel gaps (7-10) at the beds, so that the NO 2 content is degraded in the first bed at the most by 90 % of its content on the entry of the gas into the bed and is degraded in the second bed by at least 30 % of the content on entering the second bed.
Patent AU-2003263071-B2 (AU)
Title: Pyrazolopyrimidines as cyclin-dependent kinase inhibitors
Inventor: RIVERA JOCELYN
IPC: C07D487/04
Filed: 2003-09-03
Granted: 2007-03-15
Abstract: In its many embodiments, the present invention provides a novel class of pyrazolo[1,5-a]pyrimidine compounds as inhibitors of cyclin dependent kinases, methods of preparing such compounds, pharmaceutical compositions containing one or more such compounds, methods of preparing pharmaceutical formulations comprising one or more such compounds, and methods of treatment, prevention, inhibition, or amelioration of one or more diseases associated with the CDKs using such compounds or pharmaceutical compositions.
Patent AU-2005215906-B2 (AU)
Title: Process for the preparation of enantiomerically pure 1-substituted-3-aminoalcohols
Inventor: JOHN MCGARRITY
IPC: C07D333/22
Filed: 2005-02-21
Granted: 2011-08-18
Abstract: Provided is a process for the preparation of enantiomerically pure 1-substituted-3-aminoalcohols, particularly of (S)-(-)- and (R)-(+)-3--methylamino-l-(2-thienyl)-1-propanol, by asymmetrically hydrogenating salts of a carboxylic acids with an aminoketone of formula (II), wherein R is selected from the group consisting of 2-thienyl, 2-furanyl and phenyl, each optionally substituted with one or more halogen atoms and/or one or more C-alkoxy groups, and wherein R is C-alkyl or phenyl, each optionally substituted with one or more halogen atoms and/or one or more C-alkyl or C-alkoxy groups, and wherein the corresponding aminoalcohols are obtained by subsequent hydrolysis of their salts. Furthermore provided are salts of a carboxylic acid with said aminoketones and the aminoalcohols obtained by asymmetriacally hydrogenating said aminoketones, respectively.