baber/WOPTO huggingface dataset:
Patent EA-002023-B1 (EA)
Title: Pharmaceutical topically applicable preparation for introducing a peptidaceous pharmacon in a living organism
IPC: A61K31/165
Filed: 1997-09-08
Abstract: 1. A pharmaceutical topically applicable preparation for introducing a peptidaceous pharmacon in a living organism, which comprises: (i) a peptidaceous pharmacon, (ii) capsaicine, histamine and/or cantharis extract, and (iii) an epithelizing agent in admixture with carriers and/or diluents conventionally applicable in topical pharmaceutical preparations, optionally applied onto a support capable of adhering to skin. 2. A preparation as claimed in claim 1, which comprises as peptidaceous pharmacon a natural hormone or a synthetic analogue or derivative thereof. 3. A preparation as claimed in claim 2, which comprises insuline as peptidaceous pharmacon. 4. A preparation as claimed in claim 3, which comprises 0.001-0.3 g of component (ii) for 10 IU of insuline. 5. A preparation as claimed in claim 4, which comprises 0.003-0.1 g of component (ii) for 10 IU of insuline. 6. A preparation as claimed in claim 5, which comprises 0.005-0.05 g of component (ii) for 10 IU of insuline. 7. A preparation as claimed in any of the preceding claims, which comprises components (ii) and (iii) in a weight ratio of 1:(0.01-10). 8. A preparation as claimed in claim 7, which comprises components (ii) and (iii) in a weight ratio of 1:(0.03-3). 9. A preparation as claimed in claim 8, which comprises components (ii) and (iii) in a weight ratio of 1:(0.05-2). 10. A preparation as claimed in any of the preceding claims, which comprises salicylic acid, sodium chloride, resorcinol or urea as component (iii). 11. A preparation as claimed in any of the preceding claims, which also comprises an indicator which reacts to the presence or absence of the peptidaceous pharmacon by a visually observable change. 12. A preparation as claimed in claim 11, which comprises ninhydrine as indicator.
Patent EA-001830-B1 (EA)
Title: Refrigerator container
Inventor: GUBAREV OLEG ALEXEEVICH
IPC: B60P3/20
Filed: 2000-01-10
Abstract: A refrigerator container, comprising a heat-insulated body with a cargo compartment with a door and floor, a refrigerating unit in the form of compressor-refrigerating apparatus with an air cooler (air heater), mounted in of the container's body corners, characterized in that the container body is provided with an additional door, the refrigerating unit is equipped with an additional air cooler (air heater) mounted in a free corner of the container body, and the cargo compartment is provided with control sensors of temperature monitoring, floor gratings hingedly mounted on its side walls enabling them to be raised vertically and an additional loading shelves mounted at a predetermined distance from the floor enabling to be raised vertically in posts fixed in the floor, the doors are arranged on both sides of the container body and shifted relative to each other.
Patent EA-007886-B1 (EA)
Title: Electrical connectors
Inventor: NICHOLSON ALLAN
IPC: H01R43/00
Filed: 2001-12-20
Abstract: An electrical connector and method of making the electrical connection are disclosed for use in particularly arduous conditions, such as down hole oil production applications. The invention provides high electrical integrity with an ability to accommodate steady and/or fluctuating mechanical forces placed via the cable into the connector. Synergy between the mechanical and electrical aspects of the design is taught in which an insulating member, fitted with annular upstands, co-operates with a mechanically soft, essentially incompressible, insulating substance (gel) to cause vibrations in the cable to be dissipated over a length of the insulated cores inside the connector rather that at a single point where it would cause the core to fracture. In addition, annular collars of the gel are provided between the insulating member and the crimped pin-core connections and between the annular upstands and insulated cores to give further cushioning. Because the core insulation sits deep inside the annular upstand of the insulating member and gel collars, this creates a good electrical interface with a long creepage distance. The method covers the creation of the gel collars, alignment of contact pins and insulated cores and assembly of the connector.
Patent EA-005985-B1 (EA)
Title: Cellular communication method
IPC: H04B7/185
Filed: 2004-02-26
Abstract: The aim of said invention is to increase the efficiency of a cellular communication network. The inventive method consists in pre-entering an electronic file, which contains fragments of a digital local geographic map with the co-ordinates and characteristics of base stations arranged in cells and the geographic co-ordinates of said cell boundaries, into a cellular communication network control centre, in determining location data of a corresponding mobile station during a radio communication with the aid of a satellite positioning system receiver which is incorporated into said mobile station and in transmitting said data to the cellular communication network control centre through the base station. The file containing the fragments of the digital local geographic map with the co-ordinates and characteristics of the base station of a cell wherein said mobile station is located and of the adjacent cells with the boundary co-ordinates thereof is transmitted from the cellular communication network control centre through a corresponding base station to the mobile station wherein the comparison of the current data of the location of said station with the cell boundary co-ordinates is carried out.
Patent EA-006349-B1 (EA)
Title: Vehicle mounted concrete mixing drum and method of manufacturing thereof
Inventor: KHOURI ANTHONY
IPC: B28C5/18
Filed: 2003-05-31
Abstract: A method of manufacture of a vehicle mounted rotary concrete mixing drum of the type having an opening at one end for receiving and/or discharge of concrete therefrom and at the other end, means for engaging a drive assembly so as to rotate the drum for mixing or discharging concrete. The drum is manufactured from at least one mould using at least plastics material and further includes integrally attached vanes stand out from the internal surface of the drum forming an archimedian spiral disposed such that when the drum is rotated in a first direction, the concrete contents are mixed and when the drum is rotated in a second direction the contents are discharged from the drum; wherein, the method comprises the steps of: a) preparing a first generally helical inner mold part containing a surface extending between first and second helical edges; b) mounting the first helical inner mould part on a support; c) enclosing the inner helical mold assembly within an outer mould formed by at least one outer mold part; d) fitting a second mating inner helical mold part to the first inner mould part to form an inner mold assembly; e) injecting a polyurethane elastomer into a cavity defined by said inner mold assembly and the outer mould assembly to form an inner wall element comprising one half of an interior wall of the mixer and one helical blade; f) allowing said polyurethane to cure; g) removing said at least one outer mold parts to expose said inner wall element; h) removing said inner wall element one said inner molds.
Patent EA-007016-B1 (EA)
Title: Jacking frame for coiled tubing operations
Inventor: POLSKY YAROM
IPC: E21B19/22
Filed: 2003-06-23
Abstract: A modular system for performing work on a rig or platform comprises a jacking frame for movement perpendicular to the wellbore and for supporting coiled tubing loads.
Patent EA-018066-B1 (EA)
Title: Nuclear receptor binding agents
Inventor: DALTON JAMES T
IPC: A61K31/165
Filed: 2006-11-28
Abstract: The present invention relates to a novel class of selective estrogen receptor modulators (SERMs) of formulanamely 3-fluoro-N-(fluorophenyl)-4-hydroxy-N-(4-hydroxyphenyl)benzamide. The SERM compounds are applicable for use in the prevention and/or treatment of a variety of diseases and conditions including prevention and treatment of cancers such as prostate and breast cancer, osteoporosis, hormone-related diseases, hot flashes or vasomotor symptoms, neurological disorders, cardiovascular disease and obesity.
Patent EA-017145-B1 (EA)
Title: Process for the conversion of hydrocarbons into ethanol
Inventor: DANIEL BERIAN JOHN
IPC: C07C29/151
Filed: 2008-12-12
Abstract: The present invention relates to a process for the production of ethanol, and optionally methanol, from synthesis gas. In particular the present invention relates to a process for the production of ethanol from a carbonaceous feedstock; wherein the carbonaceous feedstock is first converted to synthesis gas which is then converted to methanol, which is then converted to ethanoic acid, which is then esterified and which is then hydrogenated to produce ethanol in the same alcohol synthesis unit in which the said synthesis gas is converted to methanol.
Patent EA-026302-B1 (EA)
Title: Motor controller system and method for maximizing energy savings
Inventor: KELLEY PAUL H
IPC: H02P5/00
Filed: 2008-09-15
Abstract: Provided are a motor controller (4) and method for maximizing the energy savings in an AC induction motor (3) at every load wherein the motor is calibrated at two or more load points to establish a control line (6), which is then programmed into a non-volatile memory (30) of the motor controller. A DSP-based closed-loop motor controller observes the motor parameters of the motor such as firing angle/duty cycles (23), voltage (37), current (9) and phase angles to arrive at a minimum voltage necessary to operate the motor at any load along the control line. The motor controller performs closed-loop control to keep the motor running at a computed target control point, such that maximum energy savings are realized by reducing voltage through pulse width modulation.
Patent EA-023017-B1 (EA)
Title: Fuel assembly
Inventor: BASHKIRTSEV SERGEY MIKHAILOVICH
IPC: G21C21/10
Filed: 2011-05-11
Abstract: Nuclear fuel assemblies include fuel elements that are sintered or cast into billets and co-extruded into a spiral, multi-lobed shape. The fuel kernel may be a metal alloy of a metal fuel material and a metal-non-fuel material, or ceramic fuel in a metal non-fuel matrix. The fuel elements may use more highly enriched fissile material while maintaining safe operating temperatures. Such fuel elements according to one or more embodiments may provide more power at a safer, lower temperature than possible with conventional uranium oxide fuel rods. The fuel assembly may also include a plurality of conventional UOfuel rods, which may help the fuel assembly to conform to the space requirements of conventional nuclear reactors.
Patent EA-020486-B1 (EA)
Title: N-((1R,2S,5R)-5-(TERT-BUTYLAMINO)-2-((S)-3-(7-TERT-BUTYLPYRAZOLO[1,5-a][1,3,5]TRIAZIN-4-YLAMINO)-2-OXOPYRROLIDIN-1-YL)CYCLOHEXYL)ACETAMIDE AS A DUAL MODULATOR OF CHEMOKINE RECEPTOR ACTIVITY, CRYSTALLINE FORMS AND PROCESSES
Inventor: CARTER PERCY H
IPC: C07D487/04
Filed: 2010-10-12
Abstract: The present invention provides N-((1R,2S,5R)-5-(tert-butylamino)-2-((S)-3-(7-tert-butylpyrazolo[1,5-a][1,3,5]triazin-4-ylamino)-2-oxopyrrolidin-1-yl)cyclohexyl)acetamideand a crystalline form N1 thereof, having dual CCR-2 and CCR-5 receptor inhibitory activity. Compositions based on said compounds and use of the compounds and compositions for modulating CCR-2 and CCR-5 receptor activity and for the treatment of inflammatory, allergic, autoimmune, metabolic, cancer and/or cardiovascular diseases are disclosed. The present disclosure also provides a process for preparing N-((1R,2S,5R)-5-(tert-butylamino)-2-((S)-3-(7-tert-butylpyrazolo[1,5-a][1,3,5]triazin-4-ylamino)-2-oxopyrrolidin-1-yl)cyclohexyl)acetamide.
Patent EA-022254-B1 (EA)
Title: Pipe connecting structure of water heater with tap water pipe and hot water pipe
Inventor: MIN TAE-SIK
IPC: F24H9/00
Filed: 2010-11-11
Abstract: The present invention relates to a pipe connecting structure of a water heater, wherein individual parts in the water heater are integrally coupled with a pipe body, which is injection-molded, so as to form paths of direct water and hot water, thereby reducing the number of pipes connecting the individual parts and simplifying the connection structure of the pipes. In order to realize this, according to the present invention, the pipe connecting structure of a water heater comprising a direct water inlet pipe connected from a direct water inlet to a heat exchanger; a hot water supply pipe connected from the heat exchanger to a hot water outlet; a flow sensor for measuring the flow rate of the direct water introduced via the direct water inlet; a flow control valve for controlling the flow rate of the hot water discharged via the hot water outlet; is characterized in that the pipe body which connects the direct water inlet, the direct water inlet pipe, the hot water supply pipe and the hot water outlet is formed integrally therewith.
Patent EA-023900-B1 (EA)
Title: Method for material testing for friction and wear and device for implementation thereof
Inventor: BASINYUK VLADIMIR LEONIDOVICH
IPC: G01N19/02
Filed: 2013-06-24
Abstract: The invention is related to the field of mechanical engineering, in particular, to methods and means for tribotechnical tests. The problem addressed by the invention is higher reliability of determining antiwear and/or antifriction properties of sliding friction pairs. The problem is solved by provision of a method for material testing for friction and wear, wherein the counter specimen is connected rigidly to a permanent magnet and fixed in the space by indenter specimens that are pressed to the counter specimen with a force corresponding to the static component of the load, and a resilient element coupled with the indenter specimens is connected to a software controlled module for provision of a variable component of the pressing force, the permanent magnet being arranged, with a radial gap, in the hole of a magneto-electric module that creates reciprocating motion of the counter specimen under action of the magnetic field. The absence of any guides or rolling supports makes it possible to eliminate associated errors in friction force control and to improve reliability of determining antiwear and/or antifriction properties of sliding friction pairs in conditions of non-stationary loads and sliding speeds.
Patent EA-027889-B1 (EA)
Title: Biaryl diphosphine ligands, intermediates of the same and their use in asymmetric catalysis
Inventor: ABDUR-RASHID KAMALUDDIN
IPC: C07F9/53
Filed: 2011-09-09
Abstract: The present disclosure relates to biaryl diphosphine ligands of the formula (B), processes for the production of the ligands and the use of the ligands in metal catalysts for asymmetric synthesis. The disclosure also relates to intermediates used for the production of the biaryl diphosphine ligand.
Patent EA-025315-B1 (EA)
Title: Swing adsorption processes utilizing controlled adsorption fronts
Inventor: DECKMAN HARRY W
IPC: C01B32/50
Filed: 2012-02-27
Abstract: A process for reducing the loss of valuable products by improving the overall recovery of a contaminant gas component in swing adsorption processes. The present invention utilizes at least two adsorption beds, in series, with separately controlled cycles to control the adsorption front and optionally to maximize the overall capacity of a swing adsorption process and to improve overall recovery a contaminant gas component from a feed gas mixture.
Patent EA-034610-B1 (EA)
Title: Isolated il-18 binding antibodies and uses thereof
Inventor: BARDROFF MICHAEL OTTO
IPC: A61K39/395
Filed: 2013-09-05
Abstract: The present invention relates to an isolated fully human, humanized or chimeric antibody or a fragment thereof that specifically binds IL-18, but does not bind the IL-18/IL-18 binding protein complex. Also provided are an isolated polynucleotide encoding said antibody or a fragment thereof, a cloning or expression vector comprising said one or more polynucleotides, a host cell comprising said one or more vectors, a stably transformed or transfected host cell comprising said one or more polynucleotides, a method of producing said isolated antibody or a fragment thereof. Furthermore, provided are a pharmaceutical composition comprising said isolated antibody or a fragment thereof and the uses of the antibody or a fragment thereof and the uses of said pharmaceutical composition.
Patent EA-028526-B1 (EA)
Title: ALKYL-AMIDE-SUBSTITUTED PYRIDYL COMPOUNDS USEFUL AS MODULATORS OF IL-12, IL-23 AND/OR IFNα RESPONSES
Inventor: MOSLIN RYAN M
IPC: C07D471/04
Filed: 2013-11-07
Abstract: Compounds having the following formula I:or a stereoisomer or pharmaceutically acceptable salt thereof, where the meanings of R, R, R, R, and Rare defined herein, are useful in treating inflammatory and autoimmune diseases.
Patent EA-035110-B1 (EA)
Title: Macrocyclic deaza-purinones as tlr7 modulators
Inventor: BONFANTI JEAN-FRANCOIS
IPC: C07D473/00
Filed: 2014-03-28
Abstract: The invention relates to macrocyclic deaza-purinones derivatives of formula (I), processes for their preparation, pharmaceutical compositions and the use thereof as TLR7 modulators in treating viral infections.
Patent EA-033439-B1 (EA)
Title: Fuel assembly
Inventor: BASHKIRTSEV SERGEY MIKHAILOVICH
IPC: G21C21/10
Filed: 2014-05-01
Abstract: Fuel assemblies (710) include non-symmetrical fuel elements (730) with reduced lateral dimensions on their outer lateral sides that facilitate fitting the fuel assembly (710) into the predefined envelope size and guide tube position and pattern of a conventional nuclear reactor. Fuel assemblies (910) alternatively comprise a mixed grid pattern that positions generally similar fuel elements (920) in a compact arrangement that facilitates fitting of the assembly (910) into the conventional nuclear reactor.
Patent EA-034927-B1 (EA)
Title: Aromatic heterocyclic compounds as antiinflammatory compounds
Inventor: LONGSHAW ALISTAIR IAN
IPC: C07D401/14
Filed: 2015-02-13
Abstract: The invention relates to a compound of formula (I) as defined in the specification which is a p38 MAP kinase inhibitor for use as medicament for the treatment inter alia of inflammatory diseases.
Patent EA-033294-B1 (EA)
Title: Pyridazinone herbicides
Inventor: SELBY THOMAS PAUL
IPC: A01N43/58
Filed: 2015-04-27
Abstract: Disclosed are compounds of Formula 1, including N-oxides and salts:wherein X is O, S or NR; or X is C(R)=C(R), wherein the carbon atom bonded to Ris also bonded to the carbon atom bonded to R, and the carbon atom bonded to R7 is also bonded to the phenyl ring moiety in Formula 1; and R, R, R, R, R, R, R, G and W are as defined in the disclosure. Also disclosed are compositions containing the compounds of Formula 1 and methods for controlling undesired vegetation comprising contacting the undesired vegetation or its environment with an effective amount of a compound or a composition of the invention.
Patent EA-036029-B1 (EA)
Title: Railroad traffic control and safety system
Inventor: PRONKIN ALEXANDER VASILIEVICH
IPC: B61L27/04
Filed: 2018-06-29
Abstract: The invention relates to the railroad transport. The technical result of the invention is: enhancement of functionality, improvement of information content and security, reduction of the number of operating personnel for railroad traffic control and reduced human factor influence. The system contains automated traffic control, microprocessor control, train safety, technical diagnostics and monitoring subsystems, as well as a digital radio communication system, the central switchboard of which is included in the operational digital data network with base stations installed along the rail track. The automated traffic control subsystem is provided in the rail traffic control center, microprocessor control systems are installed at stations and combined in a local transmission network of the united microprocessor control. Safety subsystems are installed in trains with each of them providing receipt and processing of data from the microprocessor control subsystems via two channels from track circuits and a radio interlocking unit, and train handling by the systems in accordance with the traffic safety requirements and "obstacle" stop requirement.
Patent EA-036203-B1 (EA)
Title: Composite material
Inventor: LESIV ALEKSEY VALERYEVICH
IPC: G08B17/00
Filed: 2016-08-10
Abstract: The invention relates to the means for controlling pre-fire situations resulting from local overheating of electrical equipment and is intended to prevent fires arising as a result of such malfunctions, in particular faults in wall outlets. Essence of the invention: a polymer composite material which polymeric matrix consists of a thermosetting polymer, is filled with an odorant that is sulfur dioxide, low-molecular-weight mercaptans, dialkyl sulfides, dialkyl disulfides or mixtures thereof and has an explosive destruction temperature in the range of 80-200°C, can be used to generate a signal for local overheating of electrical equipment. In some embodiments of the invention, the odorants, in pure form or as a solution, can be contained inside the microcapsules with a shell of polymeric material distributed in the polymer matrix. In other embodiments of the invention, the polymeric composite material is a polymer gel formed by crosslinked polymer particles swollen in an odorant solution placed in the polymeric matrix. In other embodiments of the invention, the polymeric composite material is a sorbent particles with an odorant occluded thereon, placed in the polymeric matrix. In other embodiments of the invention, the polymeric composite material is porous polymer particles with closed-type pores or channels filled with an odorant or odorant solution placed in the polymeric matrix.
Patent EA-036361-B1 (EA)
Title: Low pressure separator having an internal divider and uses thereof
Inventor: SCHULTZ MICHAEL ANTHONY
IPC: C12P7/06
Filed: 2017-02-03
Abstract: Improvements in biological conversion processes and associated apparatuses are disclosed for the generation of useful end products such as ethanol, through metabolic pathways of C1-fixing bacteria that utilize, as a nutrient, a C1-carbon source from a C1-containing substrate such as an industrial waste gas. Particular aspects of the disclosure relate to the downstream recovery of ethanol and/or isopropanol from bleed and permeate streams and more particularly to performing such recovery with improved efficiency that can advantageously reduce capital (e.g., equipment) and/or operating (e.g., utility) costs. Particular aspects related to the downstream recovery of ethanol and/or isopropanol using a low pressure separator having an internal divider.
Patent EA-038498-B1 (EA)
Title: Disposable diaper
Inventor: YOSHIOKA TOSHIYASU
Filed: 2017-02-03
Abstract: A disposable diaper (1) comprises a waist section (40) and an absorbent main body (10). Elastic member (43) extending and contracting in the horizontal direction are provided at the upper end of the waist section (40) in the vertical direction, and a cutout (45) is formed on the front side of the waist section (40) in the front-back direction at the upper end thereof in the vertical direction. The waist section (40) has a plurality of folding sections (170) folded in the horizontal direction. The folding sections (170) include two inner folding sections (172) formed on the innermost side in the side direction, and two outer folding sections (171) formed on the outermost side in the side direction. The absorbent main body (10) has a belly-side section located at the front side from the center in the front-back direction, and a back-side portion located at the back side from the center in the front-back direction. Two inner folding sections (172) are located at the back side in the front-back direction relative to the belly-side section of the absorbent main body (10), and two outer folding sections (171) are located outside the cutout (45) in the side direction.