baber/WOPTO huggingface dataset:
Patent CZ-285028-B6 (CZ)
Title: 3-substituted 1-arylindole compounds and pharmaceutical compositions containing thereof
Inventor: ANDERSEN KIM
IPC: A61K31/445
Filed: 1994-12-15
Abstract: 3-substituted 1-arylindole compound having general Formula I <CHEM>       wherein Ar is an optionally substituted aryl group; X represents a bond, a divalent hydrocarbon group or methyleneoxy or -thioxo; R<1>_R<4> are hydrogen or substituents; R<5> is hydrogen, hydroxy, alkoxy, halogen, trifluoromethyl, alkyl or alkenyl; R<6> and R<7> are hydrogen, alkyl or alkenyl;   R<8> is alkyl or alkenyl a group of Formula 1a or 1b : <CHEM>   wherein; W is O or S; U is N or CH ; Z is (CH2)m, 1,2-phenylene, CH=CH, COCH2 or CSCH2-; V is O, S, CH2, or NR<10>, wherein R<10> is hydrogen or alkyl; U<1> is O, S, CH2 or NR<11>, wherein R<11> is as R<10>; and V<1> is NR<12>R<13>, OR<14>, SR<15> or CR<16>R<17>R<18>, where each of R<12>-R<18> are as the R<10>-substituents; R<9> is hydrogen or alkyl; or R<9> is linked to R<7> to form a ring; or R<8> and R<9> together form a morpholinyl or piperidinyl ring, the latter optionally substituted by alkyl or a group of Formula 1a or 1b, or a carbamoyl group, show central antiserotonergic activity and possibly also antidopaminergic activity and are, accordingly, useful in the treatment of central nervous system (CNS) disorders. The compounds are prepared by methodt known pr. se.
Patent CZ-290398-B6 (CZ)
Title: Method and device for measuring permanent linear deformations of materials
Inventor: ZEMAN JINDRICH ING
IPC: G01N3/06
Filed: 1999-05-28
Abstract: The proposed method for measuring permanent linear deformations of materials by determining change in initial distance between two points on the material surface is characterized by making on a removable impression body (9) impressions (15) of measuring points created on the material surface and measuring precise distance of the identifiable spots of both the measuring points on the measuring point impressions. A device for making the method includes two measuring marks, fastened at a certain distance from each other onto a material to be measured, whereby it contains a fixed part (1) arranged on a material measured section (2) and a portable part (3), from which parts (2, 3) the fixed part (1) is provided with two measuring elements (7) with identifiable measuring points placed apart from each other and the portable part (3) is formed by an impression body (9) having an impression surface (10) for making impressions (15) of the measuring points.
Patent CZ-287485-B6 (CZ)
Title: Pharmaceutical preparation stabilization process
Inventor: AGHARKAR SHREERHAM NARAHARI
IPC: A61K47/44
Filed: 1998-06-23
Abstract: In the present invention there is disclosed a stabilization process of a pharmaceutical preparation containing at least one pharmaceutical agent being selected from a group comprising paclitaxel, camptothecin and derivatives thereof and a solvent system comprising ethanol and a solubilizing agent being represented by polyoxyethylated castor oil, preferably condensation product of the castor oil and 20 to 40 moles of ethylene oxide per one mole of the castor oil, preferably volume ration of ethanol : polyoxyethylated castor oil 50 : 50, at which the carboxylate anion content in this pharmaceutical preparation is reduced to a value being less than or equal to 0.6 x 10e-6 of the carboxylate anion gramequivalent per ml of the pharmaceutical preparation by addition of an acid to the solvent system or by contacting of at least one component of the solvent system with aluminium oxide.
Patent CZ-298763-B6 (CZ)
Title: Open-end spinning apparatus
Inventor: WASSENHOVEN HEINZ-GEORG
IPC: D01H4/30
Filed: 1999-08-03
Abstract: In the present invention, there is disclosed an open-end spinning apparatus (1) having a spinning rotor (3) and a spinning rotor (3) spinning cup being capable of revolving with a high number of revolution in a rotor casing 2 capable of being closed by a fiber passage-plate and attracting. The open-end spinning apparatus (1) is installed with a fiber-guiding passage (14) arranged between an opening device (26) and the spinning cup and the fiber-guiding passage (14) has a wall partition having an enhanced coefficient of friction. The fiber-guiding passage (14) has two passage sections (29 and 30) and each of their walls having a different roughness. The wall of the entrance side passage section (29) has much greater roughness (Rt) than that of the exit side passage section (30). At the same time, the roughness depth in the region of both the sections (29 and 30) of the fiber-guiding passage (14) is less than average diameter of the individual fibers (22) amounting to about 10 microns.
Patent CZ-291508-B6 (CZ)
Title: Method for removing gaseous contaminants from air
Inventor: MATZKE VLADIMIR
IPC: B01D53/66
Filed: 1998-09-29
Abstract: The invented method for removing gaseous contaminants from air, particularly sulfur oxides, nitrogen oxides, carbon monoxide and ozone is characterized in that air to be purified is heated to a temperature in the range of 15 to 85 degC, whereupon it is forcibly passed over a surface of reactor plates the active portion of which is formed by solidified mixture of urea, cyanuric acid and allophanic acid amide, whereby during forcible passage of air to be purified over the surface of the reactor plates gaseous contaminants are bound to or react with urea and/or allophanic acid amide and/or cyanuric acid to thereby achieving removal or reduction of gaseous contaminant amount in the purified air.
Patent CZ-290490-B6 (CZ)
Title: Method for the reduction of NOx in a flue gas and a system for making the same
Inventor: HINKE THOMAS V
IPC: B01D53/56
Filed: 1996-05-29
Abstract: In the present invention there is disclosed a method for reducing the NOx content of a flue gas, comprising the steps of preparing a Pi4 in water liquid/liquid emulsion (39); injecting a selected amount of the emulsion (39) as a mist into the flue gas at a preselected location; and removing NOi2 from the flue gas at a distance downstream from the predetermined location, the distance being selected such that the phosphorus-accelerated oxidation of nitrous oxide  NO in the flue gas induced by injecting the emulsion and being carried out at a temperature ranging from ranging from 180 degC to 280 degC is substantially complete prior to the removal of NOi2 Further disclosed is a system for reducing the NOx content of a flue gas stream in an intake manifold (51), comprising means for preparing a Pi4 in water liquid/liquid emulsion (39); means for injecting a metered amount of the emulsion (39) as a mist into the flue gas stream inside the intake manifold (51) at a preselected location, means for regulating temperature of the flue gas in the countercurrent section of the intake manifold (51) immediately above the injection location and for initiation of phosphorus Pi4 and nitrous oxide NO in the flue gas gaseous phase at a temperature ranging from 180 degC to 280 degC and means for wet purification being connected to said flue gas intake manifold (51) and intended for removing nitrogen dioxide NOi2 from the flue gas.
Patent SK-283927-B6 (SK)
Title: Farnesyl transferase inhibiting 1,8-annelated quinolinone derivatives substituted with N- or C-linked imidazoles
Inventor: VENET MARC GASTON
IPC: C07D498/06
Filed: 1998-03-03
Abstract: This invention concerns compounds of formula (I), the pharmaceutically acceptable acid additions salts and the stereochemically isomeric forms thereof, wherein the dotted line represents an optional bond; X is oxygen or sulphur; -A- is a bivalent radical of formula; R1 and R2 each independently are hydrogen, hydroxy, halo, cyano, C1-6alkyl, trihalomethyl, trihalomethoxy, C2-6alkenyl, C1-6alkyloxy, hydroxyC1-6alkyloxy, C1-6alkyloxyC1-6alkyloxy, C1-6alkyloxycarbonyl, aminoC1-6alkyloxy, mono- or di(C1-6alkyl)aminoC1-6alkyloxy, Ar, Ar-C1-6alkyl, Ar-oxy, Ar-C1-6alkyloxy; or when on adjacent positions R1 and R2 taken together may form a bivalent radical; R3 and R4 each independently are hydrogen, halo, cyano, C1-6alkyl, C1-6alkyloxy, Ar-oxy, C1-6alkylthio, di(C1-6alkyl)amino, trihalomethyl, trihalomethoxy; or when on adjacent positions R3 and R4 taken together may form a bivalent radical; R5 is an imidazolyl substituted with hydrogen or C1-6alkyl; R6 hydrogen, hydroxy, halo, cyano, optionally substituted C1-6alkyl, C1-6alkyloxycarbonyl or Ar; or a radical of formula -O-R7, -S-R8, -N-R8R9; and Ar is optionally substituted phenyl; having farnesyl transferase inhibiting activity; their preparation, compositions containing them and their use as a medicine.
Patent SK-281807-B6 (SK)
Inventor: THURALRAJAH PADMANATHAN
IPC: A61K31/505
Filed: 1996-11-29
Abstract: Je opísaný spôsob výroby N-[3-(3-kyanopyrazolo[1,5- a]pyrimidin-7-yl)fenyl]-N-etylacetamidu reakciou 3-dimetylamino- 1-(3-N-etyl-N-acetylaminofenyl)-2-propén-1-ónu s 3-aminopyrazol- 4-karbonitrilom v prostredí vodnej kysliny octovej.ŕ
Patent SK-278269-B6 (SK)
Title: Compressor or gas pump
Inventor: GAJDOS LUBOMIR
IPC: F04B43/04
Filed: 1991-11-13
Abstract: A driving shaft carries co-axial, one another separated and eccentrically mounted antifriction bearings (4, 41) in such a manner, that at least one first bearing (4) is with its outer ring mounted with prestressing on at least one first area (5) of the first holder (6) and at the same time at least one second bearing (41) is with its outer ring mounted with prestressing on at least one second area (51) of the second holder (61). The first and the second holders (6, 61) are each other permanently joined and every first and second bearing (4, 41) is mounted on one corresponding first or second area (5, 51), parallel each other. Individual holders (6, 61) are joined with pistons (20) which are moving in cylinders (22); said cylinders (22) form one unit together with a crankcase, so called compressor body (23). Coupling elements (7) bear, with their side areas, on the outer rings of the guiding antifriction bearings (4, 41), gripping in the compressor body (23) or in its front cover.
Patent SK-288496-B6 (SK)
Title: Dendritic constructal object with foam structure
Inventor: RYBAR RADIM
IPC: F28F7/02
Filed: 2014-09-16
Abstract: The dendritic constructal object with a foam structure formed by the folders comprising the pillars is symmetrical and hierarchically divided into several levels of the branches (1), consisting of the tandems (2) comprising two each other by a cross wall (3) separated the flow channels (4). The branches (1) of the next level of the branches (1) in the previous level are separated in the board (5) of the tandem (2) and in the last - the finest level are the branches (1) sequentially rotated about its longitudinal axis by 180 ø.
Patent CZ-298527-B6 (CZ)
Title: Medicament for treating or preventing diabetes, insulin resistance or diabetes complications and use thereof
Inventor: HORROBIN DAVID FREDERICK
IPC: A23L33/00
Filed: 1998-07-22
Abstract: In the present invention, there is described the use of an essential fatty acid, particularly one beyond the 6-desaturation step in the n-6 and n-3 metabolic pathways, and a biocompatible disulphide, particularly alpha-lipoic acid for the preparation of a medicament intended for treating or preventing diabetes, insulin resistance or diabetes complications.
Patent CZ-297920-B6 (CZ)
Title: Safety system of key protection against unauthorized handling therewith
Inventor: KALOUS JAN
IPC: G07C11/00
Filed: 2001-03-14
Abstract: The invented safety system of key protection against unauthorized handling therewith is characterized in that when manufacturing or purchase of an original cylinder-type safety lock, a customer evidence record is established. In this customer evidence record there are made the following entries: safety card and/or system card serial number, and serial numbers of all the keys supplied to the cylinder-type safety lock. Customer specimen signature is issued on both the safety card and evidence record. The specimen signature is then entered into a database. When manufacturing another replacement key, checks of the cylinder-type safety lock card and/or the system card, specimen signature entered in the database and present on the customer evidence record where serial number of the key and date of its manufacture is specified. When producing a replacement key reject, an evidence card of the reject is established, serial number of the key is recorded in the evidence card and the key is put in a safe. Serial number of the key is marked on the bill of sale or invoice.
Patent CZ-302875-B6 (CZ)
Title: Textile machine drafting mechanism
Inventor: EAFAR VACLAV
IPC: D01H5/00
Filed: 2010-06-21
Abstract: In the present invention, there is disclosed a textile machine drafting mechanism comprising drafting rollers /1, 2, 3, 4, 5, 6/ arranged in pairs with mutual thrust for controlling fibers and with gradually growing velocity. A contact insert /13, 30, 40, 50, 60/ bearing against a fiber strand /22/ magnetically presses during drafting the fiber strand /22/ to a lower belt /8/. A permanent magnet /10, 61/ can be used for applying thrust to the contact insert /13, 30, 40, 50, 60/.
Patent CZ-304151-B6 (CZ)
Title: Circuit arrangement for integrated control and management in service networks of smart buildings
Inventor: JANECEK JAN
IPC: G05B6/02
Filed: 2012-10-09
Abstract: The present invention covers a device for efficient solution and project of service network of smart buildings, which is based on sharing a harness that is primary used for making local computer networks of Ethernet, i.e. four-pair cables UTP Cat.5, optionally Cat.6. The device comprises a central processor (1), which supports any program needful for the device function. Interface (2) 802.3 for communication by IEEE 802.3c protocol interconnects the device with two pairs (1-2 a 3-6) of the UTP cable normally used by the Ethernet technology. Interface (3) of the RS-485 bus uses in common Ethernet local networks and devices used therein such as routers, switches, servers, memory centers, printers, and other unused pairs (5-4) of the UTP cables as a bus complying with the standard RS-485 in the synchronous communication (peer-to-peer) operational mode. The described device can also be provided with a suitable input/output module (4), making it possible to operate with optional own sensors or own control elements, and/or it can locally provide for the user information about the state and to ensure control of the device itself, as well as through the mediation of the central processor (1) and the IEEE 802.3 interface (2) for the communication through the protocol IEEE 802.3c and the interface (3) of the RS-485 bud of arbitrary other device of the service network, and/or it can serve for processing optical information of a camera sensor, i.e. to provide storage of data, its evaluation, for example detection of movement and its preparation for transmission to the central processor of the service network computer or to a remote indicator. A power supply unit (5) for other parts of the device uses the free pairs (7-8) of the UTP cables and makes it possible to feed sensors and control elements of the busses RS-485 as well as mutual backup of other devices. The connection of contacts between the interface (3) of the RS-485 bus and the two pairs (1-2) and (3-6) makes it possible to use the cables connected to connectors (B, C) of the RJ-45 type and unused for Ethernet transmission for additional bus according to RS-485 in the asynchronous communication mode of operation.
Patent CZ-306895-B6 (CZ)
Title: A biotelemetric system for the support of monitoring the psychophysiological state of a human being
Inventor: KAŠPAR JAN
IPC: A61B5/16
Filed: 2014-12-31
Abstract: The invention relates to a multifunctional biotelemetric system for the support of monitoring the psychophysiological state of a human being in real time, in which the physiological quantities are detected, which are further evaluated. The system comprises at least one compact wireless scanning unit (1) provided with at least one wifi access point translation unit (2) and one control/collection unit (3), wherein each scanning unit (1) comprises the ECG sensor (4), the sensor (5) for measuring skin resistance, the sensor (6) for measuring the pulse and respiration curve, the sensor (7) of body temperature, the ambient temperature sensor (8), the 3D actigram activity sensor (9), the sensor (10) for measuring and evaluating HRV variability of the heart rhythm and, further, the signal LED (11) and the event button (12).
Patent CZ-308880-B6 (CZ)
Title: Safety barrier
Inventor: DUFKA DUŠAN
IPC: F16G11/14
Filed: 2020-09-25
Abstract: The safety barrier, in particular to prevent vehicles from entering confined spaces, is formed by a system of anchored posts, which are connected by a system of horizontally arranged ropes. The columns are hollow column profiles (1), in the walls of which there are through-holes (2) for passing at least one steel rope (3) into their interior spaces. In these spaces of the hollow column profiles (1), the steel rope (3) has at least one divided rope clamp (4). If a vehicle hits it, it abuts the inner wall of the hollow steel section (1) and allows, depending on the assumed maximum impact size of the vehicle and the degree of tightening of the clamping bolts (5) connecting the two parts of the rope clamps (4), it to slide on the surface of the steel rope (3).
Patent CZ-309257-B6 (CZ)
Title: Modification of geopolymer material to increase water wettability
Inventor: LOUDA PETR
IPC: C04B28/26
Filed: 2021-10-08
Abstract: The treatment of the geopolymer material to increase the wettability by water consists of subjecting the surface of the geopolymer composite to the action of a low-temperature plasma for at least one second and this is repeated one or more times for at least one second, using atmospheric plasma with a temperature of up to 80 ° C. By applying atmospheric plasma, the surface layer of the geopolymer composite is modified by applying reactive ones and hydrophilic hydroxyl particles and the surface of the geopolymer composite is simultaneously nitrided.
Patent SK-284577-B6 (SK)
Title: Oxazolidinone derivatives, pharmaceutical compositions containing them and their use
Inventor: HESTER JACKSON B
IPC: A61K31/551
Filed: 1998-10-30
Abstract: Oxazolidinone derivative of formula (I) or a pharmaceutically acceptable salt thereof, which is antimicrobial agent, effective against various human and veterinary pathogens, including gram positive aerobic organisms, gram negative organisms, and anaerobic organisms.
Patent CZ-296086-B6 (CZ)
Title: Isolated polypeptide and polynucleotide, process of their preparation, cell and vaccine
Inventor: VINALS Y DE BASSOLS CARLOTA
IPC: A61P31/04
Filed: 1999-05-31
Abstract: In the present invention, there are disclosed polypeptides BASB027 and polynucleotides encoding for the polypeptides BASB027, processes for preparing such polypeptides using recombinant techniques and method for expression of the polynucleotides. There are also provided immunogenic fragments and fusion proteins containing the above-indicated polypeptides, expression vectors, microorganisms and cells in which these polynucleotides are comprised, vaccines, antibodies and pharmaceutical compositions, as well as their use in diagnostics, prophylaxis and therapy.
Patent CZ-293717-B6 (CZ)
Title: Recycling process of waste gas mixture to a thermoplastic tenacious material
Inventor: KRULIS ZDENEK ING CSC
IPC: C08L23/02
Filed: 2002-10-30
Abstract: The present invention relates to a recycling process of a waste gas mixture of plastics containing at least 30 percent by weight of  polyolefins to thermoplastic tenacious material wherein the process is based on the fact that polymeric components of the plastic waste mixture are made compatible by addition of 2 to 15 percent by weight of ethylene-propylene copolymer, or block styrene-butadiene copolymer, or combination of ethylene-propylene copolymer and styrene-butadiene copolymer in arbitrary weight ratio and 0.1 to 2,5 percent by weight of a secondary aromatic amine, followed with subsequent treatment of the mixture in melt.
Patent CZ-297446-B6 (CZ)
Title: Process for preparing oral solid medicamentous form and oral medicamentous form prepared thereby
Inventor: FRANC ALES
IPC: A61K31/138
Filed: 2004-09-30
Abstract: In the present invention, there is disclosed a process for preparing a solid oral medicamentous form capable of instantaneous release of the active substance which antiestrogen, particularly tamoxifen citrate, characterized in that the antiestrogen is pre-mixed with a water-insoluble and/or alcohol-insoluble filling agent and optionally with at least one further pharmaceutically acceptable excipient whereby 80 percent of particles of the filling agent or a mixture thereof with at least one further pharmaceutically acceptable excipient are smaller than 355 micrometers and at the most 10 percent of these particles are smaller than 40 micrometers, whereupon the triturate obtained is mixed with a water-insoluble and/or alcohol-insoluble filling agent and with a water-soluble and/or alcohol-soluble binding agent whereby 80 percent of particles of the mixture of the filling agent and the binding agent are smaller than 355 micrometers and at the most 10 percent of these particles are smaller than 40 micrometers. So obtained mixture is then granulated in the presence of water and/or alcohol being used in an amount smaller than or equal to 8 percent by weight, based on the total weight of the wet granulated mixture, whereupon the granulate obtained is dried. The invention also relates to the solid oral medicamentous form obtained in the above-described manner.
Patent BR-PI9913097-B8 (BR)
Inventor: HIROYUKI EGAWA
IPC: A61K31/495
Filed: 1999-08-18
Abstract: Nitrogen-containing heterocyclic carboxamide derivatives represented by the following general formula: <CHEM> wherein ring A is a substituted or unsubstituted pyrazine, pyrimidine, pyridazine or triazine ring; R<1> is O or OH; R<2> is a hydrogen atom, an acyl group or a substituted or unsubstituted carbamoylalkyl or carboxyalkyl group; and the broken line represents a single bond or a double bond; or salts thereof are useful for preventing and treating virus infections and especially influenza virus infections.
Patent GB-2271451-B8 (GB)
Title: Data recovery after error correction failure
Inventor: WENG LIH-JYH
IPC: G11C29/00
Filed: 1993-03-12
Granted: 1996-03-11
Abstract: A method of data recovery in systems employing error-correction coding techniques is described. The technique may be used, for example, in conjunction with a data storage device or a data communications network. Several trials of accessing or transmitting the ECC-protected data are performed. The data from each trial is decoded, and is also saved. If none of the trials results in the successful decoding of the data, then a reconstruction function is employed to create a reconstructed version of the data from the sequence of data created by the trials. One method of reconstruction involves majority voting on a symbol-by-symbol basis. The reconstructed data created that way is then decoded in the same fashion as for each trial. A more powerful reconstruction function employs a threshold to determine whether each voted-on symbol is sufficiently "reliable". If not, it is marked as an erasure. The reconstructed data created by this reconstruction function is decoded according to an error-and-erasure algorithm, which increases the error-correcting power of the ECC.
Patent EP-1294498-B8 (EP)
Inventor: DAVENPORT CHRISTOPHER JOHN
IPC: B21B1/40
Filed: 2001-06-22
Granted: 2006-02-01
Abstract: A method of reducing the thickness of metal sheet by cold rolling the metal sheet at least once using work rolls, whereby at least one of the work rolls has an effective Young's Modulus less than that of steel. A work roll for use in this method having an effective Young's Modulus less than that of steel. <IMAGE>
Patent EP-1598366-B8 (EP)
Inventor: GIUNTINI MAURO
IPC: A61P35/00
Filed: 2005-03-10
Granted: 2009-03-18
Abstract: Compounds of formula (I) <CHEM> useful as agonists of Somatostatin are described, processes for their preparation and pharmaceutical preparations containing them are also described.