baber/WOPTO huggingface dataset:
Patent IL-101506-A0 (IL)
Title: Use of 2-iminothiazolidin-4-one derivatives as novel pharmaceutical active ingredients
IPC: C07D277/38
Filed: 1992-04-06
Abstract: Compounds of the formula I   <IMAGE> (I)  in which R1 is lower alk-2-en-1-yl, lower alk-3-en-2-yl, lower alk-2-yn-1-yl or lower alkyl substituted in the 2,3-position by radicals which can be eliminated to give a double bond, R2 is hydrogen and R3 is methyl which is unsubstituted or substituted by radicals which can be eliminated together with hydrogen R2 to give a double bond or R2 and R3 are both hydrogen or lower alkyl or are together methylene and R4 is a group of the formula Ia, Ib or Ic   <IMAGE> (Ia)  <IMAGE> (Ib) <IMAGE> (Ic)  in which R5 is hydrogen, lower alkyl, lower alk-2-en-1-yl or lower alk-2-yn-1-yl and R6 is a group of the formula Id or Ie   <IMAGE> (Id)  <IMAGE> (Ie)  in which R1, R2, R3 and R5 are as defined, and their pharmaceutically acceptable salts can be used in a novel manner for the treatment of diseases of the rheumatoid type.
Patent IL-109988-A0 (IL)
Title: Acid derivatives
IPC: A61K31/445
Filed: 1994-06-12
Abstract: The invention concerns acid derivatives of formula I R<1>-CON(R<2>)-N(R<3>)CO-X<1>-Q-X<2>-G   I and pharmaceutically acceptable metabolically labile esters or amides thereof, and pharmaceutically acceptable salts thereof, wherein R<1> represents a group of formula II or III <CHEM> in which A is attached meta or para to the position where the group CONR<2>NR<3>CO is attached and is selected from aminomethyl, guanidino and R<a>N=C(NH2)-  T is N or CH, and  X<3> is a bond, (1-4C)alkylene or, when T is CH, oxy(1-3C)alkylene; R<2> and R<3>, which may be the same or different, represent hydrogen, (1-4C)alkyl or ar(1-4C)alkyl;  X<1> is a bond or (1-4C)alkylene;  Q is a group of formula IV or V <CHEM> X<2> is a bond, (1-4C)alkylene, oxy(1-3C)alkylene or a group of formula CH2CH(NHXR<4>) in which X is SO2, CO or CO2 and R<4> is (1-6C)alkyl, (6-12C)aryl or (6-12C)aryl(1-4C)alkyl in which the aryl group may optionally be substituted by (1-4C)alkyl; and  G is a carboxy group. The invention also concerns processes for the preparation of the acid derivatives of formula I, pharmaceutical compositions containing them and their use as inhibitors of the binding of fibrinogen to glycoprotein IIb/IIIa.
Patent IL-112515-A0 (IL)
Title: N,n-dimethyl-1-Ú1-(4-chlorophenyl) cyclobutyl¾-3-methylbutylamine in the treatment of non-insulin dependent diabetes mellitus
IPC: A61K31/137
Filed: 1995-02-01
Abstract: A compound of formula I    <IMAGE>  I  or a pharmaceutically acceptable salt thereof in which R1 and R2 are independently H or methyl (for example N,N-dimethyl-1-[1-(4-chlorophenyl)cyclobutyl]-3-methylbutylamine hydrochloride optionally in the form of its monohydrate) is used for improving the glucose tolerance of humans having non-insulin dependent diabetes mellitus.
Patent IL-113474-A0 (IL)
Title: Biaromatic acetylene compounds containing an adamantyl group pharmaceutical and cosmetic compositions containing them and uses
IPC: C07C43/225
Filed: 1995-04-24
Abstract: Bi-aromatic acetylenic cpds. with an adamantyl gp. of formula (I), their chiral analogues and their salts, are new. X = H or halo, R1 = H, -CH3, -CH2-O-R4, -CH2-O-CO-R5, -OR6, -O-(CH2)m-(CO)n-R7, -(CH2)p-CO-R8, -(CH2)p-CO-O-R9 or -S(O)p-R10, Ar = a gp. of formula (a)-(f), R2 = H, halo, 1-20C alkyl, -O-CH2-O-CH2-CH2-O-CH3 or -O-R13, R3 = -O-CH2-O-CH2-CH2-O-CH3, -(Y)n-(CH2)q-R14 or -CH=CH-(CH2)t-R14, m = 1-3, n = 0 or 1, p = 0, 1-3, q = 0, 1-12, t = 0, 1-10, R4, R6, R10 = H or lower alkyl, R5, R12 = lower alkyl, R7 = lower alkyl or a heterocyclic gp., R8 = H, lower alkyl or -N(R')R", R', R" = H, lower alkyl, mono- or poly-hydroxyalkyl, aryl (opt. substd.) or an aminoacid, sugar or peptide residue, or R'+R"= heterocyclic gp., R9 = H, 1-20C alkyl, alkenyl, mono- or poly-hydroxyalkyl, aryl or aralkyl (opt. substd) or a sugar, aminoacid or peptide residue; R11 = H, halo, lower alkyl, hydroxy, -O-R12 or -O-OR12, R13 = H or 1-20C alkyl, R14 = H, lower alkyl, 3-6C cycloaliphatic gp., mono- or poly-hydroxyalkyl, aryl, aralkyl, -CO-R8, -S(O)p-R10, -N(R')R" or, when n = 0, hydroxy, -O-R12 or -O-COR12, Y = O, S or -S(O)p.
Patent IL-115145-A0 (IL)
Title: A method of adaptive digital filtering and an adaptive digital filter
IPC: H03H21/00
Filed: 1995-09-01
Abstract: PCT No. PCT/GB95/02122 Sec. 371 Date May 28, 1997 Sec. 102(e) Date May 28, 1997 PCT Filed Sep. 8, 1995 PCT Pub. No. WO96/08867 PCT Pub. Date Mar. 21, 1996In adaptive digital filtering, first steps of adapting a filter coefficient dependent on a received data sample, and second steps of filtering by applying an adapted filter coefficient to a received data sample, are alternated so that adapted filter coefficients and modulated data samples are alternatively determined. In consequence, each adapted filter coefficient can be provided for immediate use in filtering.
Patent IL-126408-A0 (IL)
Title: Glass article carrying a transparent protective layer
IPC: C09D7/12
Filed: 1997-06-04
Abstract: The glassware, in particular hollow ware, bears a coating resulting from the deposit, in one or two steps, on the glass surface, of at least one monoaminosilane and at least one lubricating substance such as an optionally oxidised or partly oxidised polyolefin.
Patent IL-134234-A0 (IL)
Title: Coating compositions with a base consisting of silanes containing epoxide groups
IPC: C09D183/06
Filed: 1998-08-17
Abstract: The present invention provides a coating composition which comprises at least one silicon compound (A) which has at least one radical which is bonded directly to Si, is not able to be separated hydrolytically and contains an epoxy group, a particulate material (B) which is selected from among oxides, oxide hydrates, nitrides and carbides of Si, Al and B and of transition metals and has a particle size within the range 1 to 100 nm, a Si, Ti, Zr, B, Sn or V compound (C) and at least one hydrolysable Ti, Zr or Al compound (D), which comprises the following ratio1 mol of the silicon compound (A),0.42 to 0.68 mol of the particulate material (B),0.28 to 1.0 mol of the compound (C)and 0.23 to 0.68 mol of the compound (D).
Patent IL-134903-A0 (IL)
Title: Drop-on demand multi-tone printing
IPC: B41J2/01
Filed: 1998-09-07
Abstract: A drop-on-demand multi-tone printing apparatus has a series of channels arranged to receive ink from a source. Each channel has a respective ink outlet. Each adjacent pair of the channels is separated by a respective dividing wall, and each dividing wall is movable in response to a respective pulsed electrical signal to apply pressure pulses to the respective pair of the channels, whereby ink can be ejected from the outlets and deposited onto a recording medium. A respective pulsed electrical signal is developed for each channel in dependence upon whether ink is to be ejected from that channel, the signals for adjacent pairs of the channels temporally overlapping each other and not being in phase with each other.
Patent IL-145877-A0 (IL)
Title: System for accessing a synchronous network comprising a transmitter equipment and a receiver equipment
IPC: H04Q11/04
Filed: 2000-04-13
Abstract: A synchronous frame is formed by inserting data in virtual containers that are inserted in the fame. The containers are concatenated with each other. Each concatenated container indicates the total number of containers, and the order number of the particular container. A receiver responsive to the frame delivers to its output only the containers with the indications in the order of the order numbers.
Patent IL-155977-A0 (IL)
Title: Transgenic transchromosomal rodents for making human antibodies
IPC: A01K67/027
Filed: 2001-11-30
Abstract: The present invention provides novel transgenic nonhuman mammals capable of producing human sequence anti-bodies, as well as methods for producing and using these antibodies.
Patent IL-174034-A0 (IL)
Title: Security holster with locking lever
IPC: F41A/
Filed: 2006-03-01
Abstract: Holster (10) is provided having shroud (20) with top (28), sides (34, 34′), slide bearing stop (22) with hole (24) facing slide guard. Cam slot (44) is provided through shroud (20). Protuberance slots (36, 36)′ are provided in shroud (20) for receiving pistol protuberance (99). Screw (84) pivotally secures lever (70) to shroud (20). Lever (70) includes lever arm (72) having actuator (74) with bearing (76) and cam arm (78) having guide cam (80) positioned in cam slot (44) into side of shroud (20). A method for using holster is provided.
Patent IL-181373-A0 (IL)
Title: Procedure for the recognition of interfering transmitter a communication terminal and an evaluation unit
Filed: 2007-02-15
Abstract: The invention relates to a method for recognizing a jamming transmitter (STOR), a communication terminal (KEG), and an evaluation unit (AE). The inventive method is used for recognizing a jamming transmitter (STOR) affecting a communication terminal (KEG) that operates in cellular radio networks (FN), particularly the GSM mobile radio network, and taking a countermeasure to reduce the action of the jamming transmitter (STOR). The communication terminal (KEG) and a base station (B) are part of a cellular radio network (FN) while the base station (B) has its own service range (ZB) and services at least one radio channel (FB). The communication terminal (KEG) evaluates radio channel signal levels (FSP) that are received at periodic intervals on the radio channel (FB) determined by the base station (B) while receiving and evaluating another message (M) which originates from the base station (B) and concerns the message content when the communication terminal (KEG) is registered in the radio network. In case the communication terminal (KEG) discovers a radio channel signal level (FSP) exceeding a given threshold value on the specified radio channel (FB) without being able to decode the additional message (M), the communication terminal (KEG) interprets said state as an interfering state and outputs an alarm signal (AS). Also disclosed are an adequately configured communication terminal (KEG) and an adequately configured evaluation unit (AE).
Patent IL-183064-A0 (IL)
Title: Phenylpiperazine derivatives with a combination of partial dopamine-d2 receptor agonism and serotonin reuptake inhibition
Filed: 2007-05-08
Abstract: The invention relates to a group of novel phenylpiperazine derivatives with a dual mode of action: serotonin reuptake inhibition and partial agonism on dopamine -D2 receptors. The invention also relates to the use of a compound disclosed herein for the manufacture of a medicament giving a beneficial effect. The compounds have the general formula (1) wherein the symbols have the meanings given in the specification.
Patent IL-184286-A0 (IL)
Title: Shortened wound healing processes by means of novel fiber non-wovens
Filed: 2007-06-28
Abstract: Multilayered wound dressing (A) comprises a fleece (1), in contact with the wound; a watertight membrane (3) made of at least one water-insoluble polymer (P1), and, between (1) and (3), a loose, easily removed adhesive compound (I), or no adhesive at all. Multilayered wound dressing (A) comprises a fleece (1), in contact with the wound; a watertight membrane (3) made of at least one water-insoluble polymer (P1), and, between (1) and (3), a loose, easily removed adhesive compound (I), or no adhesive at all. (3) is (a) an adherent plaster, with a part able to adhere to the skin surrounding the wound or (b) it has no adhesive part, and the part surrounding the wound will adhere only when an adhesive has been applied to the skin.
Patent IL-195907-A0 (IL)
Title: Protein-binding methotrexate derivatives, and medicaments containing the same
Filed: 2008-12-11
Abstract: The invention relates to methotrexate derivatives which contain a protein-binding group and can be enzymatically cleaved in the body such that the active substance or a low-molecular active substance derivative is released. Also disclosed is a method for producing methotrexate derivatives, the use thereof, and medicaments comprising methotrexate derivative.
Patent IL-196985-A0 (IL)
Title: Security peripheral integrated with a contactless object of secure document type with radiofrequency device
Filed: 2009-02-09
Abstract: The invention concerns a contactless portable object (10, 30, 60) featuring a main radiofrequency device made up of a main chip (18, 38, 68) and a main antenna (16, 36, 66) connected together so that, when the portable object enters the magnetic field of a suitable reader, the main radiofrequency device provides power to the chip and ensures communication between the chip and the reader. According to the main characteristic of the invention, the portable object includes a secondary contactless device featuring a secondary antenna (12, 32, 62) and an electric circuit set up in such a way that, when the two antennas enter the magnetic field of a suitable reader at the same time, the amount of energy required to power the electric circuit and have it operational being less than the amount of energy required to power the main chip (18, 38, 68) and have it operational, the electric circuit is powered and makes the reading of data of the main chip impossible.
Patent IL-210668-A0 (IL)
Title: Glucagon - like - peptide - 2 (glp-2) analogues and pharmaceutical composiitons containing them
Filed: 2011-01-16
Abstract: GLP-2 analogues are disclosed which comprise one of more substitutions as compared to [hGly2]GLP-2 and which improved biological activity  in vivo  and/or improved chemical stability, e.g. as assessed in  in vitro  stability assays. More particularly, preferred GLP-2 analogues disclosed herein comprise substitutions at one or more of positions 8, 16, 24 and/or 28 of the wild-type GLP-2 sequence, optionally in combination with further substitutions at position 2 (as mentioned in the introduction) and one or more of positions 3, 5, 7, 10 and 11, and/or a deletion of one or more of amino acids 31 to 33 and/or the addition of a N-terminal or C-terminal stabilizing peptide sequence. The analogues are particularly useful for the prophylaxis or treatment of stomach and bowel-related disorders and for ameliorating side effects of chemotherapy.
Patent RO-127678-A0 (RO)
Title: System and method for orienting a flat thermal solar collector depending on the thermal need
Inventor: VIŞA ION
IPC: F03G6/00
Filed: 2012-02-20
Abstract: The invention relates to a system and method for orienting a flat thermal solar collector depending on the thermal need. According to the invention, the system consists of a fixed frame (0) and a movable platform (2) , with a fixed rotation axis (A-A) therebetween, said axis being situated in the middle plane of the location and inclined to an optimum angle (( γ *) depending on the geo-meteorological peculiarities of the considered location, a linear actuator (1), articulated at the base of the fixed frame (0) and to the platform (2), which ensures the orientation step-by-step of the platform (2), on a stroke ( Δ β *) of up to 130°, by means of a deformable triangle type mechanism, some flexible connections (4) between the pipes mounted on the platform (2) and the fixed pipes in the network, two shadowing screens (5) provided with mirrors on the inner faces, adjacent to the collector, arranged on the eastern and western sides of the platform (2), means for measurement and control, such as temperature and position transducers of the orientation system and for establishing the level of the solar radiation incident in horizontal plane. The method claimed by the invention, ensures the collected solar energy to be adapted to the specificity of the null or non-null thermal load, according to a composed algorithm, in a first step there being entered as input data the required null or non-null thermal load, the temperature (T) of the water in the boiler and the instantaneous solar radiation in the horizontal plane, the global radiation (G) and the diffuse radiation (D), in the second step if the thermal load is null there is applied a reverse phase orientation program, thereafter if the thermal load is not null, the temperature (T) is lower than the maximum allowable temperature (Tadm) and the direct radiation is preponderant (clear sky or relatively clear sky, G>kxD) - program of step-by-step orientation, in the forth stage, in the same thermal conditions (with clouded sky, G<=kxD) - fixed orientation southwards, and in the last stage, if the load is not null and the temperature (T) is close to the temperature (Tadm) - reverse phase orientation.
Patent RO-130391-A0 (RO)
Title: Shoe with golden sole
Inventor: STAVAR IORDAN
IPC: A43B3/35
Filed: 2015-03-26
Abstract: The invention relates to a medical shoe which ensures a uniform foot sole blood supply by using reflexogenic zones located on the sole of the foot. According to the invention, the shoe comprises a sole (1) of leather which is mounted over a golden plate (2) mounted on a support (3) and coupled, by means of a conductor (4), to a wear element (5).
Patent RO-130890-A0 (RO)
Title: Seasonal method and apicultural kit (skep) for obtaining honey in natural honeycombs
Inventor: COŢOP NICOLAE
IPC: A01K47/00
Filed: 2015-10-26
Abstract: The invention relates to a seasonal method intended for a period of time between one month and four months and to an apicultural kit named skep, meant to be employed to obtain honey in natural honeycombs, even by unspecialized persons, the method aiming at producing honey in natural honeycombs and giving incentive to current apiculture by creating apicultural services. According to the invention, the method consists in creating a network of apicultural accredited units from which interested persons can purchase the swarm of bees along with the apicultural kit suitably packaged by the specialists in the field, in order for it to be transported to the selected meliferous area, at the harvesting time the purchaser being intended to come back with the closed beehive, for exploiting the bees family and harvesting the honeycombs, where the apicultural units which are part of the network are able to lend specialized advice for cost optimization in the honey production activity, as well as for calibrating the swarms of bees in connection with the potential of the meliferous areas of interest. The apicultural kit, as claimed by the invention, is an enclosure made of food-compatible material, such as stainless steel, plastics or other materials, heat- and rain-insulated, which has a stand and a bee entrance/bee-family closing system, a suitable venting system and to which a pollen collector may be attached, a handle for transportation purposes and a landing board, the apicultural kit mainly consisting of a stand and two vertical parts which can be assembled/disassembled so that, by detaching the two halves of the skep, it allows the honeycombs to be harvested.
Patent IE-910411-A1 (IE)
Title: Expandable base shelf assembly for display gondolas
IPC: A47F5/00
Filed: 1991-02-07
Abstract: Shelving for supporting merchandise includes a sloping base shelf (12) that extends outwardly from a gondola wall and slightly upwardly toward a shopping aisle. The base shelf is supported by a framework (16) that rests upon the floor. An extension shelf (14) is mounted on a framework that is slidably mounted to the base shelf (12). The extension shelf and base shelf are substantially parallel and spaced apart. A pin (70) on the frame of the extension shelf is selectably positioned in any of a plurality of stop positions (50) provided on the base shelf framework. In a first position the base shelf (12) overlies the extension shelf (14) and in a second position the extension shelf extends beyond the base shelf into the aisle. Where a large inventory is desired on the selling floor, the base shelf surface is supplemented by pulling out the extension shelf from beneath the base shelf. A grid (78) of spaced rods extends perpendicularly from the base shelf (18) until it contacts the back wall of the gondola, providing a sloping surface against which the product leans while standing on the slopes base shelf. <IMAGE>
Patent IE-910539-A1 (IE)
Title: Surgical gripping instrument
Inventor: BENCINI ROBERT F
IPC: A61B17/221
Filed: 1991-02-15
Abstract: A surgical gripping instrument, e.g. for gripping and removing intestinal polyps, includes a sheath (60), gripping means (59) at the distal end of the sheath movable with respect to the sheath by a predetermined distance for actuating the gripping means, a support assembly (10) and a slide (30) movable with respect to the support assembly. The slide (30) is connected to at least one of the sheath and the gripping means for movement thereof. In accordance with the invention, means are provided responsive to movement of the slide relative to the support assembly by a distance less than the predetermined distance to cause the gripping means to be moved relative to the sheath by the predetermined distance in order to actuate the gripping means. This enables the throw of the instrument, i.e. the distance the surgeon needs to move his or her fingers, to be reduced to a comfortable level while retaining the desired travel of the gripping means relative to the sheath.
Patent MA-19541-A1 (MA)
IPC: C22B1/00
Filed: 1982-07-19
Abstract: The invention relates to a method for converting metal-containing waste material having substantial quantities of organic constituents, such as plastics, rubber, paper and greases, to a product from which metal can readily be recovered. The waste material is introduced into a reactor vessel arranged for rotation about its longitudinal axis, the vessel being provided with a bottom and a common charge and discharge opening, whereafter the reactor vessel is rotated with its axis inclined to the horizontal plane at an angle of less than 90 DEG . The reactor vessel is maintained during this rotation at a temperature which is sufficiently high to expel organic constituents in the form of a combustible gas for as long as such a gas continues to be generated. The combustible gas is combusted continuously at a location external of the reactor vessel, and the residual content of the reactor vessel is taken out in a molten and/or non-molten state. During at least a part of the expulsion process, air or gas containing free oxygen can be supplied to the reactor vessel through a lance in sub-stoichiometric amount.
Patent MA-21756-A1 (MA)
Inventor: WAYNE DANIEL MICHEL
IPC: B01J13/02
Filed: 1990-02-26
Abstract: Microcapsules which are prepared using coacervation processes and/or which have a complex structures in which there is a large central core of encapsulated material, preferably perfume, and the walls contain small wall inclusion particles of either the core material or some other material that can be activated to disrupt the wall are disclosed. The microcapsules that are prepared by coacervation and contain perfume are especially desirable for inclusion in fabric softener compositions that have a pH of about 7 or less and which contain cationic fabric softener. The encapsulated perfume preferably does not contain large amounts of relatively water-soluble ingredients. Such ingredients are added separately to the fabric softener compositions. Ingredients that have high and low volatilities as compared to, e.g., the desired perfume, can either be added to, or removed from, the perfume to achieve the desired volatility.
Patent MA-27974-A1 (MA)
Inventor: NORON MARK RICHARD THOMAS
IPC: A23L27/00
Filed: 2006-01-06
Abstract: A coffee product and process are provided which produce a coffee product having elevated levels of 3,7-dimethylocta-1,6-dien-3-ol. In various forms, the coffee product is dry roast and ground coffee or a dry soluble coffee product such as a powder or granule form. The process includes adding 3,7-dimethylocta-1,6-dien-3-ol to roast and ground coffee or a soluble coffee to produce an enhanced coffee flavor beverage, or to an extract or solution thereof.