baber/WOPTO huggingface dataset:
Patent MC-2144-A1 (MC)
Inventor: COY DAVID H
IPC: A61P9/10
Filed: 1989-10-13
Abstract: In general, the invention features a linear (i.e., non-cyclic) bombesin analog of biologically active mammalian gastrin-releasing peptide (GRP) and amphibian bombesin, having an active site and a binding site responsable for the binding of the peptide to a receptor on a target cell; cleavage of a peptide bond in the active site of naturally occuring bombesin or GRP is unnecessary for in vivo bilogical activity. The analog has one of the following modifications: (a) a deletion of a residue within the active site and a modification of a residue outside of the active site, or (b) a remplacement of one or two residues within the active site with a synthetic amino acid. The analog is capable of binding to the receptor and acting as a competitive inhibitor of the naturally occurring peptide by binding to the receptor and, by virtue of one of the modifications, failing to exhibit the in vivo biological activity of the naturally occurring peptide.
Patent IE-910749-A1 (IE)
Title: Aromatic copolyamides, preparation thereof and structures formed therefrom
Inventor: KEIL GUENTER
IPC: C08G69/36
Filed: 1991-03-06
Abstract: Aromatic copolyamides, preparation thereof and structures formed therefrom There are described aromatic copolyamides which are soluble in organic solvents for polyamides and which comprise at least 95 mol % of recurring structural units of formulae   OCArCO A  NHAr'NH B <IMAGE> C  <IMAGE> D  and up to 5 mol % of meta-bonded structural units E and/or F derived from aromatic dicarboxylic acids (E') and/or from aromatic diamines (F'), the sum total of the mole fractions of structural units A+E and the sum total of the mole fractions of structural units B+C+D+F being essentially of equal magnitude. The copolyamides of the present invention can be processed into fibers having high strengths and high breaking extensions.
Patent LU-88851-A1 (LU)
Inventor: WAGNER ARMAND
IPC: B65D41/48
Filed: 1996-12-13
Abstract: The cap (1) has a flat top, an inner ring (10) which fits inside the bottle neck, and an outer skirt (2) with an inner projection (23) which locks the cap in place when it is forced over a collar (C) on the bottle neck. An upper section which forms a security strip (12). One end of the security strip has a tongue (22) which is designed to be gripped to remove the strip, the tongue having an inner surface (22a) which causes it to be pushed outwards when the cap is fitted, making it easier to grip. In a variant of the design the security strip can be made to cover only part of the circumference of the bottle neck, the remainder acting as a hinge for the top of the cap when it is opened and closed.
Patent MA-25024-A1 (MA)
Inventor: WOBBEN ALOYS
IPC: F03D7/04
Filed: 1999-11-09
Abstract: Wind power installations generally have an active drive for wind direction tracking. The active drive rotates the machine housing of the wind power installation in such a way that the rotor blades of the rotor are oriented in the direction of the wind. Multiple azimuthal drives are typically used for larger wind power installations. The present invention includes a wind power installation comprising a machine housing, a rotor with at least one rotor blade, and a displacement device for orientating the rotor in the direction of the wind. The displacement device has a three-phase asynchronous motor drive that is supplied with three-phase current and is at times or completely acted upon with direct current during the stoppage time of the machine housing. Thus improved displacement devices, such as azimuthal drives, are provided ensuring uniform load distribution for each drive and preventing unwanted torque fluctuations in the individual drives.
Patent MA-27596-A1 (MA)
Title: Derives d'heteroarylamides benzocondenses de thienopyridines utiles comme agents therapeutiques, compositions pharmaceutiques les contenant et methodes pour leur utilisation
Inventor: ROMINES WILLIAM HENRY III
IPC: C07D495/04
Filed: 2004-12-08
Abstract: Société dite : PFIZER INC. REVENDICATION DE PRIORITES US 14 Juin 2002	60/389,110 Voir en annexe le titre de l'invention et le texte de l'abrégé Dérivés d'hétéroarylamides benzocondensés de thiénopyridines utiles comme agents thérapeutiques, compositions pharmaceutiques les contenant et méthodes pour leur utilisation L'invention concerne des composés représentés par la formule I ainsi que leurs précurseurs médicamenteux ou métabolites, ou les sels ou produits de solvatation pharmaceutiquement acceptables desdits composés, desdits précurseurs médicamenteux et desdits métabolites, formule dans laquelle Z, Y, R11 et R14, R15, R16 et R17 répondent aux définitions figurant dans le présent mémoire. L'invention concerne également des compositions pharmaceutiques contenant les composés de formule I et des méthodes pour le traitement de troubles hyperprolifératifs chez un mammifère par administration des composés de formule I.
Patent MA-38834-A1 (MA)
Title: Composition de ciment faite de materiaux isolants ou de materiaux ayant une bonne conductivite thermique de differents types, particulierement applicable dans le domaine du batiment et procede de sa fabrication
Inventor: PELUSI CLAUDIO
IPC: C04B28/02
Filed: 2016-02-08
Abstract: L'invention concerne une composition de ciment de matériaux isolants de divers types, qui est applicable en particulier dans le domaine de la construction avec la fonction d'isolation thermique et acoustique, en utilisant des matériaux d'usage courant et économiquement avantageux, pour obtenir des niveaux élevés d'isolation thermique et acoustique, et concerne également un procédé pour la fabrication de cette composition de ciment. L'invention se rapporte également en alternative à une composition de ciment de bons matériaux conducteurs thermiques, pour l'obtention de hautes performances de conductivité thermique. Sont décrit en détail tous les matériaux utilisés, qui sont mélangés les uns aux autres, et les quantités maximales et minimales de l'ensemble des mêmes matériaux.
Patent MA-51948-A1 (MA)
Title: Composition pharmaceutique ou diététique contenant l’extrait aqueux de la lavande et utilisable comme antidiabétique
Inventor: BOUTAHIRI SALIMA
IPC: A61K36/53
Filed: 2020-12-18
Abstract: Composition pharmaceutique ou diététique à base d'extraits aqueux de lavande pour son utilisation pour soigner le syndrome métabolique et le diabète. Selon l'invention, cette composition peut en outre comprendre un extrait aqueux d'au moins une deuxième plante issue de la liste 1.
Patent MA-53572-A1 (MA)
Title: Procédés de production et formes cristallines d'un inhibiteur mdm2
Inventor: BIO MATTHEW
IPC: C07D498/04
Filed: 2014-06-09
Abstract: La présente invention concerne des procédés de production d'acide 2-((3r,5r,6s)-5-(3- chlorophényl)-6-(4-chlorophényl)-l-((s)-l-(isopropylsulfonyl)-3-méthylbutan-2-yl)-3- méthyl-2-oxopipéridin-3-yl)acétique ainsi que des intermédiaires et des procédés de production des intermédiaires. L'invention concerne également des formes cristallines du composé et les intermédiaires
Patent UY-24362-A1 (UY)
Title: D-tartrato de (-)-cis-6(s)-fenil-5(r)-(4-(2-pirrolidin-1-il etoxi)fenil)-5,6,7,8-tetrahidronaftalen-2-ol
Inventor: CHARLES K CHIU
IPC: A61K31/40
Filed: 1996-11-04
Abstract: Un procedimiento ventajoso de preparación de D-tartrato de (-)-cis-6(S)-fenil-5(R)-[4-(2-pirrolidin-1-iletoxi)fenil]-5, 6, 7, 8-tetrahidronaftalen-2-ol, que es útil como agonista de estrógenos. También aporta procedimientos para tratar o prevenir enfermedades o estados que son susceptibles de ser tratados o prevenidos por agonistas de estrógenos, los cuales comprenden administrar a un mamífero que necesite tal tratamiento o prevención, una cantidad eficaz del compuesto. Dicho procedimiento comprende: a- disolver cis-6-fenil-5-[4-(2-pirrolidin-1-iletoxi)fenil]-5, 6, 7, 8-tetrahidronaftalen-2-ol racémico, o enriquecido ópticamente de forma parcial, en etanol acuoso en ebullición para formar una disolución, b- añadir a dicha disolución una cantidad molar igual de ácido D-tartárico disuelto en etanol acuoso para formar una segunda disolución; c- enfriar dicha segunda disolución; y d- recoger el producto formado en el paso c. Este procedimiento es útil para tratar osteoporosis, enfermedades cardiovascular o hiperlipidemia, para disminuir los niveles séricos de colesterol, obesidad cáncer de mama, endometriosis.
Patent UY-26386-A1 (UY)
Title: Empleo del aceite de oliva en la elaboración de un producto para la higiene oral para la eliminación o reducción de la placa bacteriana y/o bacterias presentes en la cavidad bucal
Inventor: FERNANDEZ MARIA ALVAREZ
Filed: 2000-10-10
Abstract: Se describe el empleo del aceite de oliva en la elaboración de un producto destinado a la higiene oral, por ejemplo, una pasta dentífrica, un colutorio bucal, un spray o inhalador bucal o un chicle, para eliminar o reducir la placa bacteriana y/o bacterias presentes en la cavidad bucal, consiguiéndose de esta manera una reducción en la aparición de enfermedades dentales (caries, enfermedad periodontal) y halitosis.
Patent UY-28880-A1 (UY)
Title: Atomizador para la distribución de líquidos para fines médicos
Inventor: SPALLEK MICHAEL
IPC: A61M11/00
Filed: 2005-04-29
Abstract: Atomizador medicinal distribuidor de líquidos desde al menos un cartucho insertable en el atomizador así como un cartucho y un sistema constituido por atomizador y cartucho insertable en el mismo. Útiles para aplicación de formulaciones medicinales líquidas activas por inhalación comprendiendo como módulos esenciales, porta-cartuchos dispuesto en la carcasa, boquilla configurada en la carcasa, donde se dispone dispositivo de atomización y sistema de tubo de unión conectando el atomizador y el porta-cartuchos donde el atomizador presenta al menor un cuerpo de toberas y el tubo de unión presenta al menos un canal con pistón hueco alojado de forma desplazable en el mismo, donde el pistón hueco comprende un cuerpo de válvula.
Patent UY-29468-A1 (UY)
Title: Nuevos derivados de isoindoles, composiciones que los contienen, su preparación y sus utilizaciones farmacéuticas, especialmente como inhibidores de las actividades de la proteína chaperona hsp90.
Inventor: PATRICK MAILLIET
IPC: C07D487/04
Filed: 2006-04-07
Abstract: La invención se refiere a productos nuevos isoindoles de fórmula (I) en la que los sustituyentes y parámetros son tales como se definieron el Memoria Descriptiva y en las reivindicaciones, estando estos productos en todas las formas isómeras y las sales, como medicamentos.
Patent UY-29988-A1 (UY)
Title: Compuestos de oxazolidinona y su uso como potenciadores del receptor metabotrópico de glutamato
Inventor: SWIERCZEK KRZYSZTOF
IPC: C07D263/24
Filed: 2006-12-05
Abstract: La presente invención se relaciona con compuestos de fórmula I: donde R1, R2, Y, m y n son como se los define con mayor detalle en la descripción, La invención también se relaciona con procesos para la preparación de los compuestos, y con nuevos intermdediarios empleados en la preparación, con composiciones farmacéuticas que contienen los compuestos, y con el uso de los compuestos en terapia.
Patent AT-523795-A1 (AT)
Title: Prothesenkomponente für eine Endoprothese
IPC: A61F2/40
Filed: 2020-04-21
Abstract: Bei einer Prothesenkomponente für eine Endoprothese zum Ersatz eines anatomischen Gelenks, zumindest mit einem Gleitflächenelement (6, 12) und einem zur Festlegung an einem Knochen eines Patienten ausgebildeten Festlegungsteil (1, 11), wobei das Gleitflächenelement (6, 12) an dem Festlegungsteil (1, 11) starr festlegbar ist und weist das Gleitflächenelement (6, 12) an einer einer Gleitfläche (8) des Gleitflächenelements (6, 12) abgewandten Seite (9) zumindest eine Ausnehmung (10) auf, in welcher ein Magnetelement (20) zumindest teilweise aufgenommen ist. Weiters eine Prothesengegenkomponente mit einem Gleitflächengegenelement, (13) aufweisend ein ferromagnetisches Material sowie ein Gleitflächenelement und eine Endoprothese.
Patent ES-180736-A1 (ES)
Title: UN MOTOR DE EXPLOSIoN ROTATIVO
Filed: 1947-11-21
Abstract: Motor rotativo de explosión caracterizado por estar constituído por una envolvente externa que forma una cámara interior, cerrada por dos superficies planas y paralelas y por una superficie curvada entre las mismas, presentando esta cámara una sección aproximadamente ovalada o aplanada, en cuyo interior se mueve un cuerpo cilíndrico o rotor solidario de un eje que atraviesa las superficies planas o culatas y puede girar sobre cojinetes apropiados de las misma, estando este rotor provisto de varias ranuras según planos radiales, en las cuales se alojan una o más paletas, desplazables radialmente y provistas en su borde o extremo interno de unos rodillos que sobresalen ligeramente de la paleta y se apoyan contra sendos nervios o resaltos excéntricos formados en la pared interior de las culatas, estando además, provistas estas paletas en su borde exterior de unas tiras o nervios sujetados elásticamente que están en contacto y rozan continuamente con la superficie curvada interna de la envolvente y con los bordes de las culatas planas extremas, estableciéndose entre cada dos paletas consecutivas, pequeñas cámaras parciales cuyo volumen varia, aumentado y disminuyendo durante la rotación del rotor.
Patent ES-182995-A1 (ES)
Title: Un revestimiento interior para hornos industriales con ladrillos o bloques de material crudo
Filed: 1948-03-11
Abstract: Un revestimiento interior para hornos industriales, caracterizado por el hecho de que los ladrillos o bloques refractarios, a base de cuarcita con alto contenido de sílice, se emplean crudos, realizándose directamente la cocción en el sitio de empleo, es decir en el horno mismo del cual constituyen el revestimiento, y durante las operaciones corrientes de encendido del horno.
Patent ES-185560-A1 (ES)
Title: PERFECCIONAMIENTOS INTRODUCIDOS EN LOS PROCEDIMIENTOS DE DEPURACIoN DE GASES INDUSTRIALES
IPC: C10K1/32
Filed: 1948-10-13
Abstract: Perfeccionamientos introducidos en los procedimientos de depuración de gases industriales caracterizados por eliminarse el hidrógeno sulfurado de dichos gases industriales tratando éstos con anhídrido sulfuroso en presencia de un absorbente sólido que favorece la reacción entre el hidrógeno sulfuroso y el anhídrido sulfuroso.
Patent ES-197084-A1 (ES)
Title: UN MECANISMO DE CAMBIO DE PESADA PARA LAS BALANZAS AUTOMáTICAS.
Filed: 1951-03-15
Abstract: Mecanismo de cambio de pesada para balanzas automáticas que comprende un pilón que puede ocupar sobre el balancín varias posiciones correspondientes a otras tantas capacidades de pesada de la balanza caracterizado porque las diferentes posiciones del pilón se determinan mediante un juego de palancas que accionado desde el exterior de la balanza desplaza longitudinalmente al balancín un par de horquillas que abrazan los muñones del pilón.
Patent ES-279253-A1 (ES)
Title: Derivatives of ajmaline
Filed: 1962-07-14
Abstract: The invention comprises mono- and di-esters of the alkaloid ajmaline with saturated or unsaturated aliphatic mono- or poly-carboxylic acids having more than 2 carbon atoms in the molecule, or with partial esters of the polycarboxylic acids, or with halogenated saturated aliphatic carboxylic acids, or with halo-, nitro- or alkoxy-benzoic acids, and the acid addition and quaternary ammonium salts thereof, and the preparation of the esters by esterifying ajmaline with the appropriate acid halides or anhydrides. Pharmaceutical preparations, useful for regulating cardiac rhythm, comprise the foregoing compounds, with or without other medicaments, and an inert pharmaceutical carrier. They may be in forms suitable for enteral or parenteral administration, e.g. tablets or ampoules. Salts specified include ascorbates, salicylates and p-aminosalicylates. The Provisional Specification comprises also esters with acyloxybenzoic acids.
Patent ES-320310-A1 (ES)
Title: Method of making thyristors having electrically interchangeable anodes and cathodes
IPC: H01L29/73
Filed: 1965-12-02
Abstract: A device of the type described in Specification 1,030,669 has a fifth region 4 of the same conductivity type as the central (base) region of the wafer diffused into the anode region 1, a first metallic contact 8 applied to the cathode (3) and gate regions, and a second metallic contact 5 applied to the anode and fifth regions. Control electrodes 6 and 7 are provided, and the contacts 5 and 8 serve interchangeably as anode and cathode. In a modification, Fig. 2 (not shown), a further region (10) is diffused into the gate region and the control electrodes 6 and 7 are replaced by a single electrode (11) making contact with this further region (10) and with the gate region.
Patent ES-332556-A1 (ES)
Title: Mechanism for effecting the positional adjustment of nuclear reactor control rods
IPC: G21C7/14
Filed: 1966-10-21
Abstract: A mechanism for effecting the positional adjustment of nuclear reactor control rods comprises first and second vertical operating members 10, 14 pivotally coupled to an intermediate member 12 which forms a lever arm, the first member 10 terminating in a grab 9 for the control rod 8 and the second member 14 extending outside the biological shield wall 2 of the reactor, the intermediate member 12 being provided with a transverse fulcrum pin 15 which is pivotally mounted in a bearing secured to a vertical support rod 16 which also extends outside the shield wall 2. The leak-tightness of the shield wall 2 where it is traversed by the second member 14 is ensured by means of a bellows seal (not shown). The intermediate member 12 terminates at one end in a fork 19 in which is engaged a pivot pin 13 for the second member 14, the fork being intended to permit any lateral movements of these members when they perform either simultaneous or separate movements. The shield wall 2 consists of a shield slab 3 through which are formed openings which provide access to the reactor tank 1 and which are normally closed by means of plugs 4, 5. The drive mechanism also comprises a graboperating device (not shown) consisting of a first vertical rod which causes the grab to open as a result of the displacement of the rod, which rod is pivotally connected to one end of a relay rod pivoted about a pin carried by the intermediate member 12, the other end of the relay rod being pivotally connected to a second vertical or drive rod. The position of the control rod 8 is controlled externally of the reactor, from a control station located above the shield slab 3, by vertical displacement of the member 14. This displacement is considerably less than that of the member 10, thus facilitating the sealing of the member 14 in its passage through the shield wall 2. When the control rod 8 is to function as a safety rod for controlled shutdown of the reactor, the rod is propelled towards the reactor core 7 by rapid movement of the member 14 which is produced for example by the expansion of a spring. The removal of the drive mechanism, after shut down of the reactor, so as to completely clear the space above the core 7 in order that various fuel element handling operations may be effected is described.
Patent ES-351349-A1 (ES)
Title: Apparatus for production of printed web materials
IPC: B42D15/00
Filed: 1968-03-07
Abstract: Apparatus for printing monetary transfer documents such as cheques comprises a plurality of stations 12-15, Fig. 3, for printing on a web supplied by a roll 10, each station including an impression roller 18 and a plate cylinder 16 having a retractable section 19 carrying a printing surface, and a pair of further printing stations 23, 24, Fig. 4, at which the printed web 61 is printed with personalized information by computer-controlled printers. The fully printed web is cut by a pair of disc-type rotary cutters 26 which slit it longitudinally and remove waste 8 and by a shear cutter 28 which cuts it transversely. Cutters 26 may be re-sited to produce left-hand cheque books. The cut sheets 30 are removed by a conveyer 29. The web may be serrated at 22 and re-reeled before overprinting. Rotary printing apparatus.-Cylinder 16 at station 12 prints a background tint on five cheques and a line outline of a credit slip, the credit slip plate is mounted on section 19 and may be tripped as required. At station 13 a second colour is overprinted on the web. At station 14 the reverse side of the web is printed and the plate on the respective section 19 prints the reverse side of the credit slip if required. At 15 the original side of the web is printed by a plate carrying " re-order " information on the respective section 19. In operation cylinders at stations 12- 14 make five complete revolutions with their sections 19 operative and a sixth with the sections retracted the section 19 at station 15 is only operative during the said sixth revolution. Selective computer-controlled printing.-At 23, branch variables and cheque numbers are printed and at 24 the account number, the branch code and the cheque numbers are printed in magnetic or magnetizable ink. Information is fed into the printers at 23, 24 from a computer control centre supplied with coded information derived from a punched card or analogous information store system relating to a particular account. Both computer controlled printers at 23 and 24 print different personalized information on adjacent cheques.
Patent ES-356277-A1 (ES)
Title: Method for depositing on a support a thin layer of a solid ceramic electrolyte for a fuel cell
IPC: H01M8/12
Filed: 1968-07-19
Abstract: A process has been provided for preparing thin solid electrolyte layer suitable for use in fuel cells. This process comprises the following steps: making electrically conductive at least one substance intended to form the electrolyte layer maintaining said substance placed on at least one conductor in an enclosure under a vacuum, said support being connected to at least one anode of at least one electron beam accelerating anode and being at the same potential thereof bombarding said substance by at least one focused electron beam increasing the energy of said beam to bring gradually the substance being bombarded to a temperature close to the melting point of the substance and maintaining this temperature, for a sufficient time to obtain by progressive evaporation, a layer of electrolyte of a desired thickness deposited on a support placed within the enclosure.