baber/WOPTO huggingface dataset:
Patent WO-03092607-B1 (WO)
Title: Structure cristalline de la proteine aurora-2 et poches de liaison associees
Inventor: CHEETHAM GRAHAM
IPC: C12N9/12
Filed: 2003-05-01
Abstract: La présente invention concerne des molécules cristallines ou complexes moléculaires cristallins contenant des poches de liaison d'Aurora-2 ou de ses homologues. Cette invention concerne également des cristaux contenant Aurora-2 et se rapporte aussi à un ordinateur équipé d'un support de données codé à l'aide des coordonnées structurelles de poches de liaison d'Aurora-2 ainsi que des procédés d'utilisation d'un ordinateur pour évaluer la capacité d'un composé à se lier à ladite molécule ou audit complexe moléculaire. Ladite invention concerne également des procédés d'utilisation desdites coordonnées structurelles pour résoudre la structure de protéines ou complexes protéiques homologues. En outre, cette invention concerne des procédés d'utilisation desdites coordonnées structurelles pour cribler et concevoir des composants, y compris des composants inhibiteurs, se liant à l'Aurora-2 ou à ses homologues.
Patent BG-62764-B1 (BG)
Title: Bicycle transmission
Inventor: ROJDEV STANIMIR V
IPC: B62M1/24
Filed: 1995-10-06
Abstract: The device is designed for stepless changing of the torque of a bicycle transmission by changing the length of the arm depending on the loading of the pedals. The device consists of a driving sprocket (2) on which the arm (4) is mounted, shifted from the center (0) in comparison with it. The device operates by the force which the rider exercises on the pedals by arms (4 & 7). Depending on the size of this force, the appropriate arm is revolving around a point which is the geometrical center of the gear rim transferring the torque to it which torque is dependant on arm R1. Under specific conditions the arms revolve around another center and transmit the torque of the gear rim, dependant on arm R2. The travel of the pedals can be alternated by using small arm R1, and if required to be increased to a maximum, corresponding to arm R2. 2 claims, 4 figures
Patent BG-66218-B1 (BG)
Title: Fungicide compositions
Inventor: HOLAH David
IPC: A01N59/26
Filed: 2003-09-02
Abstract: The invention concerns fungicide compositions, comprising: a) at least a pyridylmethylbenzamide derivative of formula wherein the various radicals are such as defined in the description, and b) at least a compound (II) which is a phosphorous acid derivative, or phosphorous acid itself and their alkaline, alkaline-earth or metal salts. The invention also concerns a preventive or curative method for fighting against phytopathogenic fungi of crops, characterised in that it consists in applying on the aerial parts of plants an efficient and non-phytotoxic amount of said fungicide compositions.
Patent BG-66020-B1 (BG)
Title: Slot machine for sale of ready food or industrial products
Inventor: DIMITROV PARASHKEV
IPC: G07F11/04
Filed: 2008-03-05
Abstract: The invention relates to a slot machine for sale of ready food or industrial products packed in disposable cartons. The machine is technically simple, with a small number of mechanical elements for actuating and control of the feeding-driving mechanisms of the goods. It consists of a mobile parallelepiped piston (12) reciprocally moving over ball bearings (11a) on bearing strips (11) located at the bottom of a module (9) with two rows (A, B) of products (14) arranged one over the other. The piston is driven by a crank mechanism with a short drive arm (19) and a long drive arm (17), which are connected and actuated by a shaft (20) of a motor-reducer (21, 22).
Patent CH-715957-B1 (CH)
Title: Système d'affichage pour mouvement horloger.
Inventor: PIERRE-YVES GRÜRING
IPC: G04B47/06
Filed: 2016-03-30
Abstract: L'invention concerne un système (1) d'affichage pour mouvement horloger (M) comportant : - un mobile d'entrée (11) destiné à être entraîné par ledit mouvement (M) ; - au moins un mobile d'affichage (15a ; 15b ; 15c) destiné à entraîner au moins un organe d'affichage (13a ; 13b ; 13c), ledit mobile d'affichage (15a ; 15b ; 15c) comprenant une came de remise à zéro (43a ; 43b ; 43c) associée à un marteau de remise à zéro (45), - au moins un embrayage (17a, 57a ; 17b, 57b ; 17c, 57c) présentant un état embrayé et un état débrayé, ledit embrayage (17a, 57a ; 17b, 57b ; 17c, 57c) reliant cinématiquement, dans son état embrayé, ledit mobile d'entrée (11) et ledit mobile d'affichage (15a ; 15b ; 15c). Selon l'invention, ledit système d'affichage (1) comprend un système de remise à zéro automatique (9) agencé pour amener automatiquement ledit embrayage (17a, 57a ; 17b, 57b ; 17c, 57c) dans son état débrayé et amener ledit marteau (45) en contact avec ladite came de remise à zéro (43a ; 43b ; 43c) en réponse à un événement prédéfini.
Patent EE-03771-B1 (EE)
Inventor: SENN-BILFINGER JOERG
IPC: C07D471/14
Filed: 1998-03-19
Abstract: Tetrahydropyrido compounds of formula (I)in which the substituents have the meanings mentioned in the description, are suitable for the prevention or treatment of gastrointestinal diseases.
Patent EP-1120632-B1 (EP)
Inventor: MILLER NORBERT DR
IPC: G01C21/34
Filed: 2000-01-24
Granted: 2002-08-21
Abstract: The route guidance method uses a mobile radio system for connecting a user with a central processor (1), supplied with the actual position of the user and the required target location, for calculation of the optimum route based on the local infrastructure. The route is converted into guidance symbols transmitted to the user's mobile radio terminal (2), e.g. mobile telephone, for providing a corresponding route guidance display.
Patent EP-1043145-B1 (EP)
Inventor: SPENCER DUDLEY W C
IPC: B29C65/00
Filed: 2000-04-06
Granted: 2003-09-17
Abstract: A wafer (12) for use in the selective connecting and disconnecting of plastic tubes incorporates a fuse (26) in an aperture. The fuse is made of a three layer laminate (28) having light transmission characteristics which change after the wafer and its laminate have been heated. The three layers comprise two outer transparent layers and an intermediate layer having limited light transmission characteristics. When the wafer (12) is heated the intermediate layer (32) shrinks thereby changing the light transmission characteristics by providing a path for light to pass through the laminate without passing through the intermediate layer. <IMAGE>
Patent EP-1074653-B1 (EP)
Inventor: ERB DAVID F JR
IPC: D04H1/48
Filed: 2000-08-04
Granted: 2006-10-18
Abstract: A durable, low-density, high performance insulating material is suitable for use as a high temperature thermal and acoustic insulation. The insulation includes fiber batting made with non-thermoplastic fibers or blends of fibers such as aramid fibers and ceramic fibers, which are bound within at least some interstices by high temperature non-flammable thermoplastic binder such as polyphenylene sulfide. In addition, a fireblocking layer can be provided on at least one surface of the insulation to further improve fire ablation or flame retardance.  <IMAGE>
Patent EP-1118593-B1 (EP)
Inventor: PEUCHERT ULRICH DR
IPC: C03C3/091
Filed: 2000-11-30
Granted: 2004-08-04
Abstract: Aluminoborosilicate glass contains (in weight %): more than 58-65 SiO2, more than 6-10.5 B2O3, more than 14-25 Al2O3, 0- less than 3 MgO, 0-9 CaO, 0.1-1.5 SrO, more than 5-8.5 BaO, not more than 8.6 SrO + BaO, 8-18 MgO + CaO + SrO + BaO and 0- less than 2 ZnO. The glass has a thermal expansion coefficient alpha 20/300 of 2.8 x 10-6> /K to 3.8 x 10-6> /K.
Patent EP-1056281-B1 (EP)
Inventor: WILF ITZHAK
IPC: H04N9/75
Filed: 1996-09-09
Granted: 2005-12-07
Abstract: Apparatus for automatic electronic replacement of a billboard in a video image including an automatic camera orientation measurement apparatus including motion measurement means operative to measure the Field of View (FOV) of the TV camera relative to a known reference position. <IMAGE>
Patent EP-1033072-B1 (EP)
Inventor: ROYNEBERG ERLING
IPC: A01D87/12
Filed: 2000-02-17
Granted: 2004-07-28
Abstract: A bale wrapper apparatus (10) which can be coupled with a propelling vehicle, and having a wrapping table (14) provided with rollers (15) which are operative, directly or indirectly, to rotate the bale about its axis while stretch film wrapping is applied to the bale, and a bale-handling device (17) mounted forwardly of the table (14) and operative to engage and to grip a bale (16) lying on the ground, and to transfer the bale to the table (14), in which: the bale handling device (17) comprises; first and second lift arms (18, 19) spaced apart laterally from each other to define a receiving space (20) for a bale (16); means (24) permitting relative movement between the first and second lift arms (18, 19) so that the latter can engage opposed end regions (22) of the bale (16) to grip the bale, prior to transfer of the bale (16) rearwardly to the wrapping table (14); and a movable guide surface (21, 21a) which defines part of the receiving space (20) and which is engageable by the bale (16) as the latter enters the receiving space (20), and which can adjust the position of the bale (16) relative to the receiving space (20), when necessary, to locate the bale (16) in a predetermined position axially relative to the centre of the table (14). <IMAGE>
Patent EP-1041525-B1 (EP)
Title: Game system
Inventor: KUSUDA KAZUHIRO
IPC: G06F19/00
Filed: 2000-03-31
Granted: 2006-07-19
Abstract: A game system which is capable of ensuring continuity of a game is provided. A game system for paying for recreation value according to progress of a game, has a magnetic information reading device for reading information in an attachable/detachable recording medium, an SRAM for storing state and history of a suspended game corresponding to each of the recording media, and a medal management device for paying for recreation value according to progress of the game. Specifying information for specifying each of the recording media is recorded in each of the recording media, the state and history of the game are stored in the SRAM corresponding to the specifying information, and the rest of the game is continuously progressed by using the state and history of the game which were stored in the RAM corresponding to the specifying information read by the magnetic information reading device. <IMAGE>   <IMAGE>
Patent EP-1086684-B1 (EP)
Inventor: PLOS GREGORY
IPC: A61K8/66
Filed: 2000-09-14
Granted: 2010-04-14
Abstract: Keratin fibre oxidation staining ready-to-use composition comprises at least one oxidation dye and an enzymatic system. Also claimed is a process utilizing the composition.
Patent EP-1148863-B1 (EP)
Inventor: RESTLE SERGE
IPC: A61Q5/12
Filed: 2000-02-04
Granted: 2002-06-26
Abstract: The invention concerns novel detergent and conditioning compositions comprising, in a cosmetically acceptable medium, at least an anionic surfactant, at least an amphoteric surfactant, at least a selected water-insoluble carboxylic acid ester: the total number of carbon atoms of the ester not exceeding 27 if it contains no unsaturation and 50 if it contains at least one unsaturation, the ester concentration being higher than 1 % and the anionic surfactant/amphoteric surfactant ratio being not more than 3. The invention is useful for hair and skin cleaning and care.
Patent EP-1170989-B1 (EP)
Inventor: TAYLOR WILLIAM
IPC: A01K1/06
Filed: 2000-03-10
Granted: 2003-07-16
Abstract: A confinement device for a four-legged animal is provided. The confinement device comprises a frame to receive the animal and a floor plate for the rear legs of the animal. The floor plate is arranged such that it is stable only when both rear legs of the animal bear down on the floor plate.
Patent EP-1154804-B1 (EP)
Title: Composition cicatrisante antibacterienne bioadhesive
Inventor: LEUNG SAU-HUNG SPENCE
IPC: A61L15/28
Filed: 2000-01-27
Granted: 2008-02-20
Abstract: L'invention se rapporte à une composition cicatrisante bioadhésive comportant du pullulane, du pyruvate, un antioxydant et un mélange d'acides gras saturés et insaturés. Ladite composition peut se présenter sous la forme d'un film qui n'est pas autocollant. Cette composition peut comporter également des agents médicamenteux du type sulfate de polymyxine B, zinc de bacitracine et sulfate de néomycine. L'invention se rapporte également à des procédés de production de cette composition et à des procédés de traitement des plaies à l'aide de ladite composition.
Patent EP-1157069-B1 (EP)
Inventor: YU YUAN
IPC: C09D11/00
Filed: 2000-03-03
Granted: 2003-05-07
Abstract: The present invention relates to a process for preparing surface-modified colored pigments. The process includes the steps of: preparing a reaction batch comprising a treating agent and a diazotizing agent; adding a colored pigment to the batch; and mixing the colored pigment and the batch under high shear conditions to form a reaction product comprising a surface-modified colored pigment. The treating agent has an organic group which comprises at least one diazotizable group. In a preferred embodiment the diazotizable group comprises a) at least one aromatic group or at least one C1-C20 alkyl group, and b) at least one ionic group, ionizable group, nonionic group, or a mixture thereof. The surface-modified colored pigments prepared by the process of the present invention have been found useful in aqueous or solvent based compositions and particularly in ink jet ink compositions.
Patent EP-1165791-B1 (EP)
Inventor: NOVAK JULIE E
IPC: C07K14/52
Filed: 2000-03-09
Granted: 2007-10-31
Abstract: There is provided a method of producing an antibody to an inoculated zalpha11 polypeptide comprising isolating an antibody elicited by the inoculated polypeptide, wherein the polypeptide is selected from the group consisting of: a) a polypeptide consisting of the amino acid sequence of SEQ ID NO: 72; b) a polypeptide consisting of the amino acid sequence of SEQ ID NO: 73.
Patent EP-1173582-B1 (EP)
Inventor: HAWKES TIMOTHY ROBERT
IPC: C12N9/10
Filed: 2000-04-20
Granted: 2006-06-14
Abstract: L'invention concerne, entre autres, un polynucléotide isolé comprenant une région codant un peptide de transit de chloroplaste et une synthase (EPSPS) 3' 5-enolpyruvylshikimate phosphate du peptide résistante au glyphosate, ladite région étant sous contrôle d'expression d'un promoteur de plante fonctionnant, à condition que ledit promoteur n'est pas hétérologue par rapport à ladite région, et le peptide de transit de chloroplaste n'est pas hétérologue par rapport à ladite synthase.
Patent EP-1210947-B1 (EP)
Inventor: KASAMA TOSHIO
IPC: A61K9/06
Filed: 2000-06-28
Granted: 2008-08-20
Abstract: Ophthalmic ointments for treating infective eye diseases which are particularly effective against infective eye diseases caused by methicillin-resistant Staphylococcus aureus (MRSA) or methicillin-resistant Staphylococcus epidermidis (MRSE) and contain as the active ingredient from 0.01 to 5.0% of vancomycin hydrochloride. Compared with intravenous administration, topical administration of these ophthalmic ointments is accompanied with no problem of the occurrence of side effects such as renal toxicity and thus enables the maintenance of a therapeutically effective concentration.
Patent EP-1218063-B1 (EP)
Inventor: STRUMILLO DJACZENKO MARIA
IPC: A61K31/573
Filed: 2000-07-21
Granted: 2004-04-14
Abstract: Pharmaceutical composition for topical use comprising a mixture, in the suitable polymer, of trichloroaceticacid, 2-hydroxybenzoic acid, (1 alpha , 2 beta , 5 alpha )-5-methyl-2-(1-methylethyl)cyclohexanol and, if desired, other pharmaceutically acceptable adjuvants and excipients, uses for the treatment of cutaneous injuries and process for the preparation thereof.
Patent EP-1212288-B1 (EP)
Inventor: JOHNSON BRUCE FLETCHER
IPC: C07C68/00
Filed: 2000-08-08
Granted: 2005-11-16
Abstract: Hydroxyaromatic compounds such as phenol are carbonylated with oxygen and carbon monoxide in the presence of a catalyst system comprising a Group VIII metal having an atomic number of at least 44, preferably palladium; an alkali metal or alkaline earth metal halide, preferably sodium bromide; at least one carboxylic acid amide such as N-methylpyrrolidone or dimethylacetamide; and a cocatalyst which is a compound of one or more metals including copper, titanium, zinc, lead, cerium and manganese.
Patent EP-1204819-B1 (EP)
Inventor: GAGNON FREDERIC
IPC: F02M25/07
Filed: 2000-08-17
Granted: 2007-02-21
Abstract: Système modulaire de recirculation de gaz d'échappement (EGR) comprenant en un seul ensemble, une électrovanne de régulation d'aspiration (EVR) et un capteur de différence de pression (DP). Ce capteur mesure une différence de pression d'échappement au niveau d'emplacements situés en amont et en aval d'un orifice d'un joint obturant le système modulaire EGR par rapport à un collecteur d'admission. L'emplacement de mesure amont est aligné sur l'orifice et en est éloigné.
Patent EP-1198294-B1 (EP)
Inventor: STAEHLER CORD FRIEDRICH
IPC: B01J19/00
Filed: 2000-08-01
Granted: 2005-11-09
Abstract: Microfluid reaction carrier, with a number of reaction zones, has a flow channel structure for fluids to pass through. Feed channels and parallel outflow channels are interlinked by angled connecting channels which also act as part of the feed and outflow channels structure. Microfluid reaction carrier, with a number of reaction zones, has a flow channel structure for fluids to pass through. The flow channel structure (1) is arranged on three flow planes. The feed channels (2) are in parallel on one plane, and the parallel outflow channels (3) are on the third plane. The connecting channels (4), forming the reaction zones, are in the center plane (30), linking the channels together in the outer planes at right angles or virtually at right angles. The projections of the channels in the first and third planes intersect at an angle. Each flow channel has an individual flow control with a valve system for fluid to flow in and for the fluid to be extracted. The fluid taken from each reaction zone is removed without contact with a fluid from other reaction zones. The flow channel structure is covered by a transparent layer on one or both sides (10,20). The transparent cover is of glass or plastics, with an integrated system of micro-lenses to focus light on the reaction zones and concentrate emitted light from reactions. The transparent cover can be composed of a number of parallel and fused glass fibers, forming a transparent honeycomb structure, where incoming and outgoing light is paralleled and scattered light is blocked from spreading into the transparent cover. The walls between the feed and outflow channels are impermeable to light. The connecting channels are formed by a number of fused glass fiber bundles, where the glass fiber cores are etched out to give micro-channels, only at the reaction zones. The connecting plane can be of a silicon layer, with a number of etched channels. A number of flow planes can be assembled together, where their reaction zones do not overlap and can be exposed to light individually which is directed specifically to each reaction zone. A programmable light source matrix is integrated in the reaction carrier for synthesis and analysis. A number of different receptors are fitted to the carrier at specific zones such as nucleic acids such as DNA, RNA, matter similar to nucleic acids such as peptide nucleic acids (PNA), peptides and saccharides. The receptors are of separate synthesis components, synthesized at the carrier. A component is between the receptor and carrier, to split the receptor for a functional group to remain at the carrier for the synthesis of a new receptor.
Patent EP-1244758-B1 (EP)
Inventor: STAVLAND ARNE
IPC: C09K8/502
Filed: 2000-09-15
Granted: 2005-03-16
Abstract: Composition and a process for reducing the water permeability more than the oil permeability using an gelant emulsified in oil. The use of a composition comprising an aqueous gelant emulsified in oil is also included in the present invention.
Patent EP-1220846-B1 (EP)
Inventor: VERMEHREN JAN
IPC: C07D251/42
Filed: 2000-09-28
Granted: 2008-07-09
Abstract: N 1>-Phenylsulfonyl-N 2>-(pyrimidinyl or triazinyl)-urea derivatives are produced from phenylsulfonyl halides by ammonolysis, reaction of the resulting phenylsulfonamides with phosgene and condensation of the phenylsulfonyl isocyanates obtained with an aminopyrimidine or aminotriazole; selected solvent mixtures are used for the ammonolysis and/or condensation. Production of N 1>-phenylsulfonyl-N 2>-(pyrimidinyl or triazinyl)-urea derivatives comprises: (a) ammonolysis of a phenylsulfonyl halide (II) with ammonia, preferably (a1) in a solvent mixture comprising a 20:1 to 1:1, preferably 10:1-1.4:1, by weight mixture of optionally halogenated aromatic hydrocarbon(s) and polar aprotic solvent(s); (b) reaction of the resulting phenylsulfonamide (III) (with or without isolation) with phosgene, preferably (b1) in an organic solvent in the presence of a catalyst comprising isocyanate(s) of the formula R'-NCO (R = optionally substituted hydrocarbyl) and optionally a co-catalyst comprising an amine base; and (c) condensation of the phenylsulfonyl isocyanate (IV) obtained (with or without isolation) with an aminopyrimidine or aminotriazole (V) in an organic solvent; preferably (c1) in a solvent mixture comprising an optionally halogenated hydrocarbon of b.pt. above 110[deg]C and a polar aprotic solvent; provided that steps (a) and/or (c ) are carried out according to (a1) and/or (c1), respectively. [Image] Q : O; S; or N(R 4>); X* : H; halo; CN; NO 2; 1-3C alkyl; or OCH 3; X and Y : CH or N, but are not both CH; R : H; 1-12C alkyl; 2-10C alkenyl; 2-10C alkynyl; 1-6C alkyl substituted with 1-4 halo, 1-4C alkoxy, 1-4C alkylthio, CN, 1-4C alkoxy-CO and/or 2-6C alkenyl; 3-8C cycloalkyl optionally substituted with 1-4C alkyl, 1-4C alkoxy, 1-4C alkylthio and/or halo; 5-8C cycloalkenyl; phenyl-1-4C alkyl optionally ring-substituted with 1 or more halo, 1-4C alkyl, 1-4C alkoxy, 1-4C haloalkyl, 1-4C alkylthio, 1-4C alkoxy-CO, 1-4C alkyl-CO-O, CONH 2, 1-4C alkyl-CO-NH, 1-4C alkyl-NH-CO, (1-4C alkyl) 2N-CO and/or NO 2; 2-oxo-1,3-dioxolan-5-ylmethyl; 2,2-dimethyl-1,3-dioxolan-5-ylmethyl; 1,3-dioxolan-2-ylmethyl; or a group of formula (A-1)-(A-5): X : O; S; SO; or SO 2 and X 1> = CH 2; or X : CH 2 and X 1> = O; S; SO; or SO 2; X 2>O; S; SO; or SO 2; R 1>H or 1-3C alkyl; R 2>H; halo; or 1-3C alkyl or 1-3C alkoxy (both optionally substituted with 1 or more halo or 1-3C alkoxy); R 3>H; halo; 1-3C alkyl, 1-3C alkoxy or 1-3C alkylthio (each optionally substituted with 1 or more halo or optionally substituted with one or two 1-3C alkoxy or 1-3C alkylthio); NR 5>R 6>; 3-6C cycloalkyl; 2-4C alkenyl; 2-4C alkynyl; 3-4C alkenyloxy; or 3-4C alkynyloxy; R 4>H; 1-4C alkyl; or 1-4C alkoxy; R 5> and R 6>H; 1-4C alkyl; 3-4C alkenyl; 1-4C haloalkyl; or 1-4C alkoxy. Independent claims are also included for: (A) step (a) carried out under conditions (a1); (B) step (b) carried out using a phenylsulfonamide (III) with X* = halo and carried out under conditions (b1) (the co-catalyst can be a base other than an amine base); and (C) step (c) carried out under conditions (c1).
Patent EP-1225807-B1 (EP)
Inventor: CHERICI ERNEST
IPC: A22C21/04
Filed: 2000-11-03
Granted: 2006-04-26
Abstract: The invention concerns a method which consists in generating by spraying in the treatment chamber (8) a mist of treating solution, and in causing said mist to pass through the portions to be treated (2). The invention is useful for bactericidal treatment of bird carcasses (2) with a trisodium phosphate solution.
Patent EP-1200867-B1 (EP)
Inventor: LEE JAMES C
IPC: G02B27/00
Filed: 2000-08-11
Granted: 2005-11-16
Abstract: A see through display includes a variably transmissive element positioned between a real world view and an eye of a user, and a generated display optical system for generating a displayed information image superimposed over the real world view in the visual field of the user. The variably transmissive element is controllable to dynamically vary the light intensity passing through the element into the visual field of the user. The variably transmissive element may be spatially addressed to allow selective variable transfer of light intensity through the element into the visual field of the user.