baber/WOPTO huggingface dataset:
Patent NZ-595983-A (NZ)
Title: DPP IV inhibitor formulations
Inventor: KOHLRAUSCH ANJA
IPC: A61K38/095
Filed: 2007-04-30
Abstract: Abstract - 595983 Disclosed is a solid pharmaceutical composition comprising as an active ingredient a DPP IV inhibitor compound as represented by the general formula (I) or (II) with a free or primary amino group or a salt thereof, a first diluent, a second diluent, a binder, a disintegrant and a lubricant: wherein the DPP IV inhibitor is selected from 1-[(4-methyl-quinazolin-2-yl)methyl]-3-methyl-7-(2-butyn-1-yl)-8-(3-( R)-aminopiperidin-1-yl)-xanthine, 1-[([1,5]naphthyridin-2-yl)methyl]-3-methyl-7-(2-butyn-1-yl)-8-((R)-3-amino-piperidin-1-yl)-xanthine, 1-[(quinazolin-2-yl)methyl]-3-methyl-7-(2-butyn-1-yl)-8-((R)-3-amino-piperidin-1-yl)-xanthine, 2-((R)-3-amino-piperidin-1-yl)-3-(but-2-yinyl)-5-( 4-methyl-quinazolin-2-ylmethyl)-3,5-dihydro-imidazo[4,5-d]pyridazin-4-one, 1-[(4-methyl-quinazolin-2-yl)methyl]-3-methyl-7-(2-butyn-1-yl)-8-[(2-amino-2-methyl-propyl)-methylamino]-xanthine, 1-[(3-cyano-quinolin-2-yl)methyl]-3-methyl-7-(2-butyn-1-yl)-8-((R)-3-aminopiperidin-1-yl)-xanthine, 1-(2-cyano-benzyl)-3-methyl-7-(2-butyn-1-yl)-8-((R)-3-amino-piperidin-1-yl)-xanthine, 1-[(4-methyl-quinazolin-2-yl)methyl]-3-methyl-7-(2-butyn-1-yl)-8-[(S)-(2-aminopropyl)-methylamino]-xanthine, 1-[(3-cyano-pyridin-2-yl)methyl]-3-methyl-7-(2-butyn-1-yl)-8-((R)-3-aminopiperidin-1-yl)-xanthine, 1-[(4-methyl-pyrimidin-2-yl)methyl]-3-methyl-7-(2-butyn-1-yl)-8-((R)-3-aminopiperidin-1-yl)-xanthine, 1-[(4,6-dimethyl-pyrimidin-2-yl)methyl]-3-methyl-7-(2-butyn-1-yl)-8-((R)-3-amino-piperidin-1-yl)-xanthine, and 1-[(quinoxalin-6-yl)methyl]-3-methyl-7-(2-butyn-1-yl)-8-((R)-3-amino-piperidin-1-yl)-xanthine, or a salt thereof, and the diluents are selected from erythritol, low substituted hydroxypropyl cellulose, mannitol, pregelatinized starch or xylitol, wherein, the binder is selected from copovidone (copolymerisates of vinylpyrrolidon with other vinylderivates), hydroxypropyl methylcellulose (HPMC), hydroxypropylcellulose (HPC), polyvinylpyrrolidon (povidone), pregelatinized starch, or low-substituted hydroxypropylcellulose (L-HPC); the disintegrant is selected from corn starch, crospovidone, low-substituted hydroxypropylcellulose (L-HPC) or pregelatinized starch; and the lubricant is selected from talc, polyethyleneglycol, calcium behenate, calcium stearate, hydrogenated castor oil or magnesium stearate; provided that the solid pharmaceutical composition does not comprise the DPP IV inhibitor together with a first diluent which is mannitol, a second diluent which is pregelatinized starch, a binder which is copovidone, a disintegrant which is corn starch and a lubricant which is magnesium stearate.
Patent NZ-601879-A (NZ)
Title: Analytical and combinatorial fault restoration
Inventor: KANG TAEHYEN
IPC: H02H7/26
Filed: 2012-08-16
Abstract: 601879 Disclosed is a system for fault restoration. The system is comprised of at least one memory that stores computer-executable instructions and at least one processor configured to access the at least one memory and execute the computer-executable instructions. This causes the processor to identify a switch within an area of a power grid that has lost power and compute an alternative source capacity (ASC) value for the identified switch. The processor then identifies and opens at least one second switch. The processor further computes combinations of the switch with each of the at least one second switch that satisfy a rule. The rule includes maximising a number of customers affected and satisfying a power balance equation. The processor then computes a restoration plan based at least in part on the computed combinations.
Patent NZ-602094-A (NZ)
Title: Device for holding and replacing a casting plate in a casting installation, metallic casing of casting plate and casting plate, provided with means interacting with a device detector
Inventor: COLLURA MARIANO
IPC: B22D41/24
Filed: 2011-03-17
Abstract: 602094 The disclosure relates to a device for holding and replacing a casting plate in a continuous casting installation metallurgical vessel. A detector-limit switch assembly automatically moves a casting plate to the casting position or to the sealing position, depending on whether a replacement plate is on standby on the device or not. The disclosure relates to a metallic casing of casting plate and a casting plate, provided with means interacting with the device detector.
Patent NZ-602322-A (NZ)
Title: Vector comprising multiple homologous nucleotide sequences
Inventor: STEIGERWALD ROBIN
Filed: 2009-11-20
Abstract: The invention relates to vectors comprising two or more homologous nucleotide sequences and methods for generating them. The invention concerns substituting bases in the homologous nucleotide sequences with different bases that do not alter the encoded amino acid sequence. The invention allows for the reduction of intramolecular recombination between homologous nucleotide sequences, in particular in mammalian cells. The invention further relates to nucleotide sequences containing substituted bases.
Patent NZ-607554-A (NZ)
Title: Devices for dilating a paranasal sinus opening and for treating sinusitis
Inventor: SCHRECK THOMAS A
IPC: A61M29/00
Filed: 2011-08-26
Abstract: Medical devices (150) for dilating a stenotic opening, such as a stenotic sinus opening, are disclosed. They are adapted to be implanted into a patient for a limited period of time using minimally invasive insertion procedures. The devices and methods can be used for treating sinusitis and other nasal and/or sinus disorders.
Patent NZ-618168-A (NZ)
Title: Tamper-resistant tablet providing immediate drug release
Inventor: BARNSCHEID LUTZ
IPC: A61K31/485
Filed: 2012-07-27
Abstract: Provided is a tamper-resistant tablet comprising: i) a matrix material in an amount of more than one third of the total weight of the tablet ii) a plurality of coated particulates in an amount of less than two thirds of the total weight of the tablet, wherein said particulates comprise a pharmacologically active compound and a physiologically acceptable polymer, preferably a polyalkylene oxide, have a coating comprising a water-soluble polymer, and form a discontinuous phase within the matrix material; wherein under physiological conditions the tablet has released after 30 minutes at least 70% of the pharmacologically active compound originally contained in the tablet.
Patent NZ-624552-A (NZ)
Title: Improved modulators of hec1 activity and methods therefor
Inventor: HUANG YU-LING
IPC: C07D417/14
Filed: 2012-11-29
Abstract: Disclosed are thiozole compounds of formula (I), wherein the substituents are as defined in the specification. The compounds Hec1/Nek2 modulators useful as chemotherapeutic agents for neoplastic diseases. Examples of a compound of formula (I) are: (N-(4-(4-(5-(2-methoxyethoxy)pyrazin-2-ylthio)-2,6-dimethylphenyl)thiazol-2-yl)isonicotinamide N-(4-(2,6-Dimethyl-4-(methylthio)phenyl)thiazol-2-yl)isonicotinamide N-(4-(4-(4-Methoxyphenoxy)-2,6-dimethylphenyl)thiazol-2-yl)-2-nitroisonicotinamide
Patent NZ-624799-A (NZ)
Title: Viral inactivation during purification of antibodies
Inventor: CORREIA IVAN R
IPC: C07K16/24
Filed: 2009-10-20
Abstract: Disclosed is a method for producing a host cell-protein (HCP) reduced antibody preparation from a sample mixture comprising an antibody, an HCP and a viral particle, wherein the preparation comprises a decreased number of viral particles or decreased viral activity in comparison to the sample mixture, the method comprising: (a) subjecting the sample mixture comprising the antibody to a reduction in pH thus forming a primary recovery sample, wherein the reduction in pH is to a pH of 3 to 4 for 0.5 to 2 hours; (b) applying the primary recovery sample to protein A affinity chromatography and eluting the antibody bound to protein A at a pH of 3.5; and (c) applying the eluted antibody to ion exchange chromatography, a hydrophobic interaction chromatography, or a combination thereof.
Patent NZ-710340-A (NZ)
Title: Solar panel and timepiece including solar panel
Inventor: SAITO YUTA
IPC: H01L31/046
Filed: 2014-03-03
Abstract: A solar panel (3) for use in a pointer-type timepiece or measuring instrument formed into a substantially circular shape, above which a pointer (7) mounted on a pointer shaft (6) inserted in a through hole (3a) in a center portion of the solar panel moves. The solar panel (3) includes a plurality of solar cells (11-16) arranged in a substantially circular shape, and these solar cells (11-16) have been divisionally formed into a substantially spiral shape so that the pointer is positioned over two of the plurality of solar cells (11-16). Accordingly, the pointer (7) can always be positioned over two of the plurality of solar cells (11-16), and therefore a decrease of light-receiving area due to the pointer (7) can be distributed between the two solar cells (11-16). As a result, a decrease in the output current of the plurality of solar cells (11-16) over which the pointer (7) is positioned can be suppressed, and the output current of the entire plurality of solar cells (11-16) can be improved.
Patent NZ-714313-A (NZ)
Title: Monoclonal antibodies against tissue factor pathway inhibitor (tfpi)
Inventor: WANG ZHUOZHI
IPC: C12P21/08
Filed: 2009-08-04
Abstract: Disclosed is a monoclonal antibody, or antigen binding fragment thereof which binds to an epitope in human tissue factor pathway inhibitor (TFPI), which epitope is characterised by specific binding by an antibody (2A8) comprising an LCDR1 having an amino acid sequence of SEQ ID NO:176, LCDR2 having an amino acid sequence of SEQ ID NO: 219, LCDR3 having an amino acid sequence of SEQ ID NO: 262, an HCDR1 having an amino acid sequence of SEQ ID NO: 305, an HCDR2 having an amino acid sequence of SEQ ID NO: 348 and an HCDR3 having an amino acid sequence of SEQ ID NO: 391, wherein the antibody or antigen binding fragment shows cross-reactivity to murine TFPI and binds kunitz domain 1 and domain 2.
Patent NZ-730381-A (NZ)
Title: Dynamic bandwidth switching for reducing power consumption in wireless communication devices
Inventor: BHUSHAN NAGA
IPC: H04W52/02
Filed: 2015-09-05
Abstract: Systems, methods, apparatuses, and computer-program products for performing dynamic bandwidth switching between control signals and data signals of differing bandwidths are disclosed. Frame formats are disclosed in which control signals are transmitted at different bandwidths than data signals. Receiver architectures for receiving the signaling formats are disclosed. A receiver can receive a relatively narrowband control signal while consuming a relatively low power and then dynamically adjust characteristics of various components to receive a data signal at a higher bandwidth while consuming a relatively higher power.
Patent NZ-752610-A (NZ)
Title: Pharmaceutical compositions comprising epa and a cardiovascular agent and methods of using the same
Inventor: MANKU MEHAR
IPC: A61K31/202
Filed: 2010-04-29
Abstract: Disclosed is a pharmaceutical composition comprising (a) docosapentaenoic acid in an amount of about 5% to about 10%, by weight, of all fatty acids present in the pharmaceutical composition; (b) eicosapentaenoic acid and (c) is substantially free of docosahexaenoic acid.
Patent NZ-761902-A (NZ)
Title: Use of 3-isoxazolidinones compounds as selective herbicides
Inventor: NICHOLSON PAUL
IPC: A01N43/80
Filed: 2015-02-20
Abstract: Herbicidal compositions are described containing 2-(2,4-dichlorophenyl)methyl- 4,4-dimethyl-3-isoxazolidinone (2,4-DC) and a second herbicide which provide synergistic control of select weed species. Methods of using the same compositions are also described.
Patent PT-104236-A (PT)
Title: Dispositivo para extracção de pó em assentos através de trepidação e aspiração em simultâneo
Inventor: PEREIRA RICARDO NUNO DA SILVA
IPC: A47L5/00
Filed: 2008-10-20
Abstract: O presente invento refere-se a um dispositivo para extracção de pó nos diferentes objectos com material têxtil através de forte trepidação com aspiração em simultâneo, sendo especialmente aplicável a estofos de viaturas, sofás e cadeirões. O dito invento baseia-se em quatro peças em que três delas depois de unidas acabam por formar uma só, estando o dispositivo completo depois de acoplado a um martelo pneumático, bastando acoplar o aspirador para ser utilizado. As quatro peças que formam o dispositivo do presente invento são conjugadas do seguinte modo: as peças n.º 2, 3 e 4 formam uma só peça do conjunto, em que a peça n.º 3 é encastrada na peça n.º 2, no local já referido na descrição geral e por sua vez a peça n.º 4 é encastrada na peça n.º 3 como se pode observar na figura para publicação. Posto isto temos o dispositivo do presente invento pronto a funcionar, a trepidação causada, por exemplo nos estofos do assento de um autocarro, através do conjunto formado pelas peças n.º 2, 3 e 4 faz com que o pó incrustado nos estofos se liberte e venha à superfície do assento, passando através dos orifícios da peça n.º 2, ficando retido no interior da cuba da peça nº 1 e sendo de seguida aspirado pelo aspirador acoplado à peça n.º 1 através da extensão existente na mesma, proporcionando assim ao utilizador um meio rápido e eficaz para o fim a que se destina.
Patent RU-94002473-A (RU)
Inventor: EGOROV D D
IPC: G05D27/00
Filed: 1994-01-20
Abstract: FIELD: apparatus is used in chemical, casting, pharmaceutic industry to control quality of stirring of loose mixtures, consistent lubricants mixtures (gels) between each other and one with another. SUBSTANCE: aim is to increase accuracy of stirring uniformity control. Apparatus uses measuring system, that is laser emission receiver made in the form of sensible two-coordinates detector, in central hole of which laser emission source is mounted so as to be capable to have engagement of laser beam with sensible member mirror reflector. Laser emission receiver has system to transfer electrical signal to electronic unit, that registers and processes reflected from sensible member laser emission. Mixture filled body is placed in tank with liquid and laser beam is directed to its mirror reflector. Any inclination of body caused by nonuniformity of loose materials (gels) stirring makes change of laser beam reflection angle. According to value of laser beam reflection angle they estimate stirring uniformity degree. EFFECT: improved process.
Patent RU-94009801-A (RU)
Inventor: NOVOTRJASOV N I
IPC: A01K1/01
Filed: 1994-03-22
Abstract: FIELD: agriculture, in particular, animal farming. SUBSTANCE: manure removal system has scraper units for moving manure to cross scraper conveyor, feeding funnel, hydraulically driven station with piston pump, manure pipeline, first manure storage and first liquid manure collector with liquid fraction pump. System is further provided with distributing well, second manure storage and second liquid manure collector with liquid fraction pump. Manure storage and liquid manure collector are selectively filled by means of slides with electric drive. Slides are mounted on manure pipeline in distributing well. Control apparatus has control unit with time mode setter, power supply unit, signal receiver for receiving signals indicative of liquid level in liquid manure collectors and signal receiver for receiving signals indicative of manure level in manure storages. Control unit is connected with driving station of scraper conveyor. EFFECT: improved sanitary conditions in animal houses, increased efficiency by automatized processes and improved labor conditions for workers. 3 cl, 5 dwg
Patent RU-94015581-A (RU)
Inventor: GERASIMOVA L G
IPC: C09C1/24
Filed: 1994-04-27
Abstract: FIELD: iron-bearing pigment fillers made of production wastes, thermal power stations ash in particular and used in paint and varnish industry and building. SUBSTANCE: thermal power stations ash is made suspension in water and sulfuric acid or hydrochloric acid are added in suspension till concentration achieves 50 -100 g/l with ratio of solid and liquid phases H : L = 1 : (3 - 5). Mixture is heated up to temperature of 50 - 75 deg C and held for 3 - 10 hours. After the holding suspension is filtered, liquid phase is sent in circulation and sediment is washed with water and calcined to produce iron-bearing pigment filler. To decrease pigment filler covering power index, sediment after acidic treatment is separated from liquid phase, suspended in water, iron compounds (+2) is introduced in suspension in amount of 20 -100 g/l b y FeO and suspension is held under air feeding for 5 - 10 hours under temperature of 70 - 90 C. Method allows to improve labour sanitary conditions and to produce iron-bearing pigment fillers of wide spectrum of action. EFFECT: improved labour conditions and produced universal iron-bearing pigment filler. 2 cl, 1 tbl
Patent RU-94031541-A (RU)
Title: Spring of pneumatic suspension
Inventor: BAKULIN A V
IPC: B60G11/26
Filed: 1994-08-29
Abstract: FIELD: automotive industry; suspensions of buses. SUBSTANCE: pneumatic suspension spring has flexible shell connected by one end to sprung portion of vehicle through flange and ring and coupled through other end with hollow piston connected to unsprung portion of vehicle. Suspension has also shock absorber and support. Surface of piston to which shock absorber, in form of truncated cone, is connected is made in form of end face of truncated cone in center of which one hole is arranged. More than one different diameter holes are located on cone surface. These holes communicate shell and piston spaces. Seating places for shell on ring and piston are provided with chamfer whose angle is equal to angle of chamfer of corresponding seating surfaces of flexible shell, angle of chamfer of shock absorber outer surface being from 44 to 46 degrees, piston cone being from 80 to 85 degrees and chamfer of seats being from 1 to 2 degrees. Piston is made of steel containing vanadium and nitrogen, ratio from 3:1 to 4:1. EFFECT: reduced manufactured and mounting cost of spring suspension, increased load capacity of bus and service life of suspension.
Patent RU-94036127-A (RU)
Inventor: SUCHKOV O V
IPC: H04R3/00
Filed: 1994-09-27
Abstract: FIELD: instrumentation engineering. SUBSTANCE: invention is intended for conversion of electric signals into mechanical translation. Device of electromechanical conversion includes sensor of mechanical translations presenting electromechanical transformer. Device may find use in robotics and other fields where precise linear mechanical translation is required. EFFECT: improved precision and operational reliability of device.
Patent RU-94038117-A (RU)
Inventor: FREJDLIN V B
IPC: C25C3/04
Filed: 1994-10-10
Abstract: FIELD: non-ferrous metallurgy; applicable for production of magnesium by electrolysis of fused chlorides. SUBSTANCE: electrolyzer uses housing 1, lining 2, two working compartments 3 and built-up cell 4 placed between them. The working compartments accommodate cathodes 5 introduced through the longitudinal wall, and anodes 6 introduced through the electrolyzer bottom. The built-up cell is separated from the working compartments by partitions 7 with upper 8 and lower 9 overflow ports. The partition is made of modules 11 with groove 12 and lug 13 in the vertical faces. The upper module has groove 14. EFFECT: enhanced service life of electrolyzer, reduced effluents of chlorine to the servicing zone, improved environment in the shop, enhanced yield of chlorine.
Patent RU-94039038-A (RU)
Inventor: KHOLIN S N
IPC: H01F38/04
Filed: 1994-10-11
Abstract: FIELD: electrical engineering; manufacture of converters and transformers. SUBSTANCE: frequency changer has transformer whose magnetic circuit is built up of N= 2k+1 cores, where k= 1,2,3... made of same magnetic material with rectangular hysteresis loop; each separate core carries different number of primary winding turns Wdifferentially connected in series, where k is core number, according to expression SW=SW, where Sis cross- sectional area of k-th core; Wis number of primary winding turns wound on k-th core. Each separate core also carries secondary winding turns Waccording to expression SW= SW,; each core, except for the last one, carries two isolating windings whose leads are connected through base resistors to emitter-base junctions of isolating transistors to form bidirectional switch which are interconnected so that emitter of each transistor is connected through diode anode-cathode to collector of other transistor and collectors of both transistors are connected to terminal leads of output winding of respective k+1 core. This provides for sequential polarity reversal of same-type cores both in open-circuit and loaded condition with preset sequence and for shaping voltage pulses across output windings equal in amplitude, opposite in polarity, and relatively shifted through angle Φ= K•π/N, where N is total number of cores in magnetic circuit; so, higher-frequency voltage is set up across changer output according to equation f= n•f,, where n = 2k+1, k = 1,2,3,...; fis output voltage frequency; fis input voltage frequency. In order to eliminate disturbance in polarity reversal and to raise loading capacity, as well as to improve output voltage characteristics, during polarity reversal of even-numbered core the next, odd-numbered, core does not reverse its polarity as its output winding is shorted out through conducting transistor of bidirectional switch. Enabling signal arrives at transistor from isolating winding wound on even-numbered core that reverses its polarity. Then odd-numbered core reverses its polarity and output of next, even-numbered, core is shorted out, etc. , until entire magnetic circuit reverses its polarity. This eliminates relative influence of polarity reversal of even- and odd-numbered cores. EFFECT: improved loading capacity of frequency changer and characteristics of its output voltage; simplified design; improved efficiency. 4 dwg
Patent RU-94040417-A (RU)
Inventor: PCHENTLESHEV V T
IPC: F01K27/00
Filed: 1994-11-03
Abstract: FIELD: power mechanical engineering. SUBSTANCE: power plant comprises at least two interconnected power plants that rotate about an axis. Each of the power plants is made up as a tank with a liquid whereto a fluid-operated motor is connected. The outlet of the motor is connected with an evaporator. The outlet of the evaporator is connected with a pipe line. The other end of the pipe line is connected with a condenser. When the power plant is in rotation, the liquid inside the tank is exerted by a centrifugal force. The working member of the motor is exerted by the hydraulic head of the liquid since the motor is at a greater distance from the axis of rotation than the surface of the liquid formed due to the action of the centrifugal force on the liquid. Being passed through the motor, the liquid enters the evaporator where it is fully converted into gas. The pressure of the gas in the evaporator and the pressure of the liquid at the outlet of the motor is less than the hydrostatic pressure of the liquid at the inlet of the motor. The gas from the evaporator is further enters the condenser through the pipe line due to a pressure difference. The condenser is positioned at a less distance from the axis of rotation of the plant than the motor and evaporator. The liquid from the condenser again enters the evaporator and then the cycle is repeated periodically. The heat that gas takes off in condensation in the condenser of the first plant is transferred to an intermediate heat carrier which transfer the heat to the liquid evaporated in the evaporator of the second plant. The boiling temperature of this liquid is lower than the boiling temperature of the liquid evaporated in the evaporator of the first plant. EFFECT: enhanced efficiency.