baber/WOPTO huggingface dataset:
Patent JP-2011142800-A (JP)
Title: Structure for measuring voltage to be supplied to load circuit of home distribution board
Inventor: FURUMOTO TETSUO
IPC: H02B1/40
Filed: 2010-11-30
Abstract: <P>PROBLEM TO BE SOLVED: To provide a home distribution board equipped with a power-supply voltage measuring structure to check a voltage to be supplied to a load circuit with good workability before an operation handle is turned on in a distribution switch gear having a plug-in terminal structure.  <P>SOLUTION: The power-supply voltage measuring structure is constituted with a bus-bar side voltage measuring unit installed at each of bus bars in first and second voltage poles to be commonly used to a plurality of distribution switch gears, and a switch-gear side voltage measuring unit installed at the side of a plug-in terminal in the distribution switch gear and individually used in each of the distribution switch gears. One of two test leads for the power-supply voltage measuring structure is brought into contact with the first or the second bus-bar side voltage measuring units, while the other is brought into contact individually with each switch-gear side voltage measuring unit at the side of the switch gear. Accordingly, the power-supply voltage applied between the plug-in terminals of the distribution switch gear can be measured.  <P>COPYRIGHT: (C)2011,JPO&INPIT
Patent JP-2012117113-A (JP)
Title: Non-cyanide gold electroplating bath for gold bump formation and method for forming gold bump
Inventor: ISHIZAKI MASASHI
IPC: C25D7/12
Filed: 2010-12-01
Abstract: PROBLEM TO BE SOLVED: To provide a non-cyanide gold electroplating bath for gold bump formation having bump hardness and a bump shape suitable for electrode joining with a substrate electrode, and a method for forming a gold pump using the gold plating bath.SOLUTION: The non-cyanide gold electroplating bath for gold bump formation comprises: an alkali salt of gold sulfite or ammonium gold sulfite; a conducting salt; a crystal stabilizer; a crystal conditioner; a buffer; and a brightening agent. The content of the alkali salt of gold sulfite or ammonium gold sulfite is 1 to 20 g/L as a gold concentration, a conductive salt is sodium sulfite, its content is 5 to 150 g/L, and the content of the brightening agent is 0.5 to 100 mmol/L. As the brightening agent, one or more kinds of compounds selected from a sulfoxide and/or sulfone are preferably used.
Patent JP-2012121079-A (JP)
Title: Dressing device
Inventor: UENO DAISUKE
IPC: B24B53/053
Filed: 2010-12-06
Abstract: PROBLEM TO BE SOLVED: To provide a dressing device which is installed on a grinding machine, reduces the size of a motor, and enhances dressing accuracy.SOLUTION: A rotation drive source 43 is attached to a support member 54 so as to be orthogonal to a rotating shaft 44 and so that a center plane 75 extending through the center of a dressing wheel 45 extends through or near the center 76 of a pivot shaft 53. During dressing operation, the dressing wheel receives a reaction force from a grinding wheel. The direction of the reaction force is aligned with the center plane. The reaction force is directed to the pivot shaft. Therefore, a couple of force (rotating force) hardly acts on the pivot shaft. Consequently, since a motor torque can be reduced, the dressing device having a compact motor and enhanced dressing accuracy can be provided.
Patent JP-2012121258-A (JP)
Title: Drawing machine for sheet-like material
Inventor: NAKAJIMA ICHIRO
IPC: B29C55/16
Filed: 2010-12-09
Abstract: PROBLEM TO BE SOLVED: To provide a drawing machine having a compact structure and enabling highly accurate drawing at high speed.SOLUTION: The drawing machine for a sheet-like material includes an endless link device in which a plurality of clamping devices for gripping ends of the sheet-like material are installed at both side ends of the sheet-like material. The sheet-like material is guided by guide rails arranged from an inlet side sprocket in a parallel state and a folding-fan state and is drawn, and after the drawing, the sheet-like material is detached, is made to pass through an outlet side sprocket and is returned to the inlet side sprocket. Link shaft holders guided by the respective guide rails are provided below link shafts rotatably interconnecting link plates constituting a folding part of the link device. Below the link shaft holder on the sheet-like material side, two pairs of horizontal rollers rolled sandwiching the guide rails are provided and the clamping devices are arranged near the guide rails. Below the link shaft holder on the side opposite to the sheet-like material, a pair of horizontal rollers rolled sandwiching the guide rails are provided.
Patent JP-2012001277-A (JP)
Title: Laminated container and method for manufacturing laminated container
Inventor: TARUNO SHINSUKE
IPC: B65D65/40
Filed: 2010-12-09
Abstract: PROBLEM TO BE SOLVED: To provide a laminated container easily applying vacuum lamination to a body.SOLUTION: A perforated film (21) is laminated on at least one side of a body (5) formed of an air-permeable material.
Patent JP-2012109919-A (JP)
Title: Transmission method, transmitter, reception method and receiver
Inventor: MURAKAMI YUTAKA
IPC: H04B7/04
Filed: 2010-12-09
Abstract: PROBLEM TO BE SOLVED: To improve reception quality for a transmission method which simultaneously transmits from a plurality of antennae a plurality of modulation signals that includes a basic modulation signal consisting of basic stream and an extended modulation signal consisting of extension stream in an environment having dominant direct wave.SOLUTION: A transmission method which simultaneously transmits a first transmission signal and a second transmission signal to the same frequency, selects a precoding matrix while switching one precoding matrix among a plurality of precoding matrices with regularity. The transmission method performs a precoding using the selected precoding matrix, generates an extended modulation signal after the precoding, and generates the first transmission signal and the second transmission signal from a signal based on a basic modulation signal and the extended modulation signal after the precoding.
Patent JP-2012124850-A (JP)
Title: Program and information processor
Inventor: SUZUKI AKIRA
IPC: H04N1/00
Filed: 2010-12-10
Abstract: PROBLEM TO BE SOLVED: To support input work by a user of identification information imparted to each of a plurality of documents.SOLUTION: An ID reception part 100 acquires an ID read by a reader 20 which reads the ID attached to a document from the reader 20. A read mode storage part 102 stores information indicating which of a normal mode and a search mode a present read mode is. An ID registration part 106 registers the ID acquired in the normal mode in a read ID storage part 108. A final ID storage part 110 stores the ID acquired last in the normal mode. An ID type determination part 114 determines which of the ID acquired last in the normal mode, the ID not registered last among the IDs registered in the read ID storage part 108 and the ID not registered in the read ID storage part 108 the ID acquired in the search mode is. An output processing part 116 outputs a determination result of the ID type determination part 114.
Patent JP-2011145287-A (JP)
Title: Visual recognition support apparatus
Inventor: HIKITA KENJIRO
IPC: G01C1/00
Filed: 2010-12-14
Abstract: <P>PROBLEM TO BE SOLVED: To provide a visual recognition support apparatus that allows an optical device, regardless of whether the optical device is held in hand for observation or fixed, to output an azimuth of a target of observation by following a dynamic change and grasp the azimuth without being affected by an error due to accumulation.  <P>SOLUTION: The visual recognition support device includes: an optical device 50 for observing a surrounding environment; a device azimuth detector 52a for detecting a device azimuth of the optical device 50; resetter 51a and 51b for resetting the device azimuth; basic azimuth information acquirer 13a for acquiring basic azimuth information on the optical device 50 when resetting by the resetter 51a and 51b; azimuth calculator 23 for calculating an azimuth of a target of observation by the optical device 50 on the basis of the device azimuth and the basic azimuth information; and output unit 33d for output of at least the azimuth thus calculated, wherein the device azimuth for use in calculation of the azimuth is a device azimuth detected after resetting by the resetter 51b.  <P>COPYRIGHT: (C)2011,JPO&INPIT
Patent JP-2012128613-A (JP)
Title: Travel support system
Inventor: ECHIZEN TAKAMASA
IPC: G08G1/00
Filed: 2010-12-15
Abstract: PROBLEM TO BE SOLVED: To provide a travel support system in which a vehicle group forming a congestion is specified without ITS infrastructure and the congestion of the vehicle group can be resolved.SOLUTION: A travel support system includes: congestion prediction means which makes a congestion prediction by performing the congestion prediction in real time on the basis of an estimated vehicle group distribution; vehicle group congestion information acquisition means which acquires congestion prediction information about a vehicle group obtained by the congestion prediction means; vehicle group end vehicle specification means which specifies a vehicle group end vehicle indicating start or end of a congestion from congestion information about the vehicle group; and travel support information providing means which provides travel support information to the vehicle group end vehicle specified by the vehicle group end vehicle specification means. The travel support information providing means provides travel support information for congestion resolution to at least one vehicle group end vehicle.
Patent JP-2012130441-A (JP)
Title: Bathroom mirror
Inventor: TAKEUCHI SHINICHI
IPC: A47K4/00
Filed: 2010-12-20
Abstract: PROBLEM TO BE SOLVED: To provide a bathroom mirror that has a good appearance because a heat generator disposed on the back of the mirror and a gap provided between the back of the mirror and a bathroom wall are invisible from the lateral sides.SOLUTION: The bathroom mirror includes: a mirror 1; a pair of covers 2; a lower frame 3; and an upper frame 4. The mirror 1 is provided on the back thereof with the heat generator. Each of a pair of the covers 2 is provided with: a fixing piece 21 fixed to the bathroom wall 5; and a covering piece 22 continuously extending forward from a side end of the fixing piece 21 and for covering the side end of the mirror. The lower frame 3 is provided with: a lower fixing piece 31 fixed to the bathroom wall 5; a lower supporting piece 32 continuously extending forward from the lower fixing piece 31 and for supporting the mirror; and a lower holding portion 33 provided at the lower fixing piece 32 and for holding the lower front end of the mirror 1. The upper frame 4 is provided with: an upper fixing piece 41 fixed to the bathroom wall 5; and an upper holding portion 42 provided at the upper fixing piece 41 and for holding the upper front end of the mirror 1.
Patent JP-2012131597-A (JP)
Title: Unnecessary document collection system
Inventor: AOKI HIDEHIRO
IPC: B65F1/00
Filed: 2010-12-21
Abstract: PROBLEM TO BE SOLVED: To improve efficiency of collection of unnecessary documents in terms of timing, in an unnecessary document collection system for collecting, dissolving and recycling unnecessary classified documents by an unnecessary document collection box.SOLUTION: This unnecessary document collection system includes: a fullness notification means 90a to calculate a time the weight of discarded documents reaches a preset caution threshold based on a signal output by a weight sensor 6 of a box 1, and request a notification of the time to a collection side from a communication network N; a warning determination notification means 90b to determine whether the weight of the discarded documents has reached a preset warning threshold based on the signal and request a notification of the determination to the collection side from the communication network when the weight has been determined to reach the warning threshold; and a high gradient determination notification means 90c to calculate the increase of the weight of the discarded documents at every interval of a certain period based on the signal and request, when the increase is determined to be larger than a preset gradient threshold, a notification thereof to the collection side from the communication network.
Patent JP-2012132763-A (JP)
Title: Thermocouple
Inventor: YOSHIKAWA KOJI
IPC: G01K1/08
Filed: 2010-12-21
Abstract: PROBLEM TO BE SOLVED: To provide a thermocouple that allows checking of corrosion and wear of a protection tube without detaching the thermocouple.SOLUTION: A thermocouple 10 has: a long protective tube 2 which has an internal hollow and protects a temperature sensor 1; and a tube fitting 3. The protective tube 2 accommodates the temperature sensor 1 in such a manner that a temperature sensing part 1a is disposed at a tip part. The tube fitting 3 is connected to the protective tube 2 and has a through hole 34 communicating with the inside of the protective tube 2 at its center part. The inside of the protective tube 2 has an internal diameter larger than the external diameter of the temperature sensor 1, and the tube fitting 3 has an inspection hole 3a opened to the outside which communicates with the through hole 34 and allows inspection of the pressure inside the protective tube 2. If a hole penetrates the protective tube 2 due to wear, the internal pressure of the protective tube 2 becomes higher than an atmospheric pressure. Therefore, inspection can be made from the inspection hole 3a communicating with the inside of the protective tube 2 without detaching the thermocouple 10.
Patent JP-2012132074-A (JP)
Title: Method for forming barrier layer
Inventor: KADOKURA YOSHIYUKI
IPC: H01L21/285
Filed: 2010-12-22
Abstract: PROBLEM TO BE SOLVED: To provide a method for forming a barrier layer, by which a barrier layer exhibiting sufficient barrier performance can be formed with satisfactory productivity even when the barrier layer is interposed between conductive layers comprising dissimilar metals.SOLUTION: The method for forming a barrier layer BM includes the steps of: arranging a work piece W with one conductive layer CL1 and a target 2, for example made of Ti, inside a vacuum processing chamber 1a, introducing rare gas in the vacuum processing chamber to form a plasma atmosphere, and sputtering the target to form a first metal layer on a surface of the one conductive layer; introducing gas containing oxygen gas and nitrogen gas in the vacuum processing chamber to form a plasma atmosphere and oxynitriding a surface of the first metal layer while also exposing the target to the plasma atmosphere so that a surface of the target is oxynitrided; and further introducing the rare gas in the vacuum processing chamber to form a plasma atmosphere and sputtering the target to form a second metal layer on the oxynitrided surface.
Patent JP-2012133657-A (JP)
Title: Printing system and function setting method
Inventor: MOTOSUGI TOSHIHISA
IPC: G06F3/0482
Filed: 2010-12-22
Abstract: PROBLEM TO BE SOLVED: To provide a printing system and a function setting method, capable of easily setting even a function requiring transition of a screen for setting, and setting in the same manner for any device connected to a network.SOLUTION: A printing system comprises: a plurality of image forming apparatuses, and a server. The image forming apparatuses each form an image in which options for selecting the image forming device connected to a network and options of functions for transiting a plurality of screens to set are collectively arranged in one page, and print a sheet in which an image area of each option is associated with coordinates. When acquiring the coordinates of the option selected by a user, the server identifies the image forming apparatus and the function associated with the coordinates, and instructs the identified image forming apparatus to set the identified function.
Patent JP-2012136125-A (JP)
Title: Vehicle body frame of motorcycle
Inventor: KAWAI HIDEAKI
IPC: B62K19/40
Filed: 2010-12-24
Abstract: PROBLEM TO BE SOLVED: To provide a vehicle body frame of a motorcycle, which can secure stiffness equal to/higher than that of pipework in a space-saving manner, which can easily secure a space for mounting vehicle accessories, and which has a structure with high mounting workability.SOLUTION: A vehicle body frame 1 includes a frame front section that is extended rearward from a head pipe 2, and a frame rear section that is extended downward or rearward from a back end of the frame front section. The frame front section comprises at least a pair of right and left frame members. A front-side part of the frame rear section enables the vehicle accessories such as a canister 7 and an ABS unit 9 to be easily mounted on the lateral side of a narrow lumber frame 5, while securing the stiffness sufficient for the lumber frame 5 of a closed cross-section structure in which a pair of right and left steel plates 50 and 51 overlap each other.
Patent JP-2012138487-A (JP)
Title: Wall-mountable remote control
Inventor: FUKUSHIMA YOSHIHIKO
IPC: F24H1/00
Filed: 2010-12-27
Abstract: PROBLEM TO BE SOLVED: To provide a wall-mountable remote control that has a preferred thin shape.SOLUTION: In a wall-mountable remote control R having a casing C that stores electric components therein, and packing 5 that, when the casing C is mounted on a mounting wall surface 9, is compressed between the wall surface 9 and a back wall portion 20 of the casing C to seal off a hole portion 15 where electrical wiring is led out, the back wall portion 20 of the casing C has in a position apart from the packing 5 a projecting portion 16 projecting backward of the casing C to a height up to the thickness of the compressed packing 5 and forming a recessed portion 16a inside the casing C, and at least one electric component 39 in the casing C is arranged in front of the projecting portion 16 to enter the recessed portion 16a and avoid interfering with the back wall portion 20.
Patent JP-2012135576-A (JP)
Title: Reel type game machine
Inventor: MANO TOMOKAZU
IPC: A63F5/04
Filed: 2010-12-28
Abstract: PROBLEM TO BE SOLVED: To provide a reel type game machine which promotes the continuation of a reel game by giving a game state where a player's expectation is encouraged in accordance with the game progress situation of a privilege game state, when the special game is given in addition to the privilege game such as an ART game, and then, eliminating the obstructive factor of the expectation, which is induced by the release of the privilege game state in the middle.SOLUTION: When a bonus prize is won during an AT mode, an ART game state is released in the middle to be shifted to a bonus game state, and after the termination of a bonus game, a normal game state is restored. When the release in the middle is performed, the kind of the bonus game related to the prize winning is discriminated, and an advantageous flag is set in a sub RAM 208 when a prize is won in a regular bonus game RB. The additional rate of ART game times in the re-start ART game state after an RB game is increased by setting of the advantageous flag.
Patent JP-2010531257-A (JP)
Title: エネルギー蓄積型空力ブレーキ装置および方法
IPC: B64D41/00
Filed: 2008-03-19
Abstract: 【課題】  空気中を飛行する飛行機などの乗物の速度がいかなるものであっても、効率的な空力ブレーキ力を発生させる。   【解決手段】  本方法は、上記乗物によってエネルギーを生成するステップと、生成されたエネルギーを蓄積するステップと、プロペラを駆動するために、上記乗物の前進運動と対向する力を生成するようなエネルギーを利用するステップとを含む。   エネルギーの生成は、空気に対する乗物の移動を利用してジェネレータを駆動するプロペラを使用することによって、あるいは地面に対する移動を利用してジェネレータを駆動する車輪を使用することによって、あるいは乗物のモータによって駆動されるジェネレータを使用することによって行われる。このエネルギーは、空気式、電気式または動力学的な形で蓄積することができ、その発電／駆動手段は、蓄積手段に使用される技術に応じて選択される。   【選択図】      図５ａ／５ｂ
Patent JP-2010523489-A (JP)
IPC: A61K8/891
Filed: 2008-03-31
Abstract: The present invention relates to a cosmetic composition, for instance an anti deodorant composition, comprising an at least partially dehydrated-aluminium sulphate salt and a carrier liquid. The invention further relates to a method for preparing a composition according to the invention, comprising combining a burnt aluminium salt with the carrier liquid.
Patent JP-2010522307-A (JP)
Title: 軽量複合トラス風力タービンブレード
IPC: F03D1/00
Filed: 2007-09-13
Abstract: 軽量の風力タービンブレードは、複合トラス継手のトラス支持構造アセンブリを有し、複合翼桁および交差部材を含む。複合翼桁および交差部材は、軽量リブパネルの脊椎に、離間状態で取り付けられ、それを支持する。リブパネルは、互いに平行に離間されるよう指向され、個々に周縁部が成形される。周縁部は、完成されたブレードアセンブリのための個々の曲率領域を画成する。トラス支持構造は、軽量のガラス繊維または硬化された織物スキンによって覆われる。ガラス繊維または織物スキンは、翼構造を形成するそれぞれのリブパネル縁部に取り付けられ、適合される。
Patent JP-2010523701-A (JP)
Title: 共蒸留によってジクロロヒドリンを回収する方法および装置
IPC: C07C29/80
Filed: 2008-04-11
Abstract: ジクロロヒドリンと、ジクロロヒドリンのエステル、モノクロロヒドリンおよび／またはそのエステルならびにポリヒドロキシ脂肪族炭化水素化合物および／またはそのエステルから選択される１種以上の化合物と、所望により水、塩素化剤、触媒および／または触媒のエステルを含む１種以上の物質とを含む混合物からジクロロヒドリンを回収する方法および装置を開示する。該混合物は、１工程で該混合物からジクロロヒドリンを含む低沸点留分を分離するために該混合物を蒸留または分留する間にジクロロヒドリンを回収するためにストリッピングされる。利点としては、所与の蒸留塔についてのジクロロヒドリンのより効率的な回収、重質副生成物の形成を助長する条件の回避による廃物の減少、および回収装置における低下された資本投資の低減が挙げられる。 【選択図】なし
Patent JP-2010523291-A (JP)
Title: 遠近の視覚能力を検査および／または訓練するためのシステムおよび方法
IPC: A61H5/00
Filed: 2008-04-14
Abstract: 変化する距離における被検者の視覚能力を自動に検査および／または訓練するためのシステムおよび方法を得る。近位表示装置は、特徴を有する視覚的なマークを表示することができる。表示されたマークが有する視覚的特徴を識別する入力を受信した後に、第２マークを遠位表示装置に表示することができる。遠位表示装置に表示されたマークの特性を識別する入力を受信した後に、さらなる検査を、近位表示装置と遠位表示装置との間で続行することができる。２個以上の表示装置を使用することができ、これら表示装置を被検者に対して互いに異なる距離に配置する。
Patent JP-2010525854-A (JP)
Title: バンドレス聴覚保護具及び聴覚保護方法
IPC: A61F11/08
Filed: 2008-03-27
Abstract: 【課題】人間の耳用の聴覚保護具及び聴覚保護方法を提供する。 【解決手段】聴覚保護具は、プラグ部材が外耳道を塞ぐ又は外耳道に挿入して嵌り込むように形成される。聴覚保護具は、少なくとも一部は加圧パッドによって付勢され、或る程度の力をプラグ部材に加える。プラグ部材を外耳道から一時的に取り外す又はプラグ部材を調節するのを手助けするためにハンドル部が随意的に用いられる。聴覚保護具は、随意的に用いられる弓形部材により耳介の周りにおいてクリップ留めされる。聴覚保護具は、イヤホンとして用いられるように構成することもできる。 【選択図】図１３Ａ
Patent JP-2010526535-A (JP)
Title: 新規な除草剤抵抗性遺伝子
IPC: A01H5/00
Filed: 2008-05-09
Abstract: 本発明は、２，４−Ｄだけではなく、ピリジルオキシ酢酸除草剤に対しても抵抗性である新規な植物を提供する。本発明はまた、１つまたは複数の他の除草剤抵抗性遺伝子と共に「積み重ねられた」本発明の１つまたは複数の酵素を産生する植物を含む。本発明は、除草剤の新規な組合せを新しい形で使用することを可能にする。さらに、本発明は、グリホサートなどの１つまたは複数の除草剤に対して抵抗性である、雑草の系統の発生を予防し、それらを防除するための新規な方法を提供する。本発明による使用に好ましい酵素および遺伝子は、本明細書においてＡＡＤ−１３（アリールオキシアルカノエートジオキシゲナーゼ）と呼ばれる。この非常に新規な発見は、著しい除草剤耐性作物形質および選択可能マーカーの可能性に基づくものである。
Patent JP-2010528213-A (JP)
Title: 燃焼機関のブリーシングシステム用の弁モジュール
IPC: F02D9/06
Filed: 2008-05-20
Abstract: 燃焼機関ブリーシングシステム用の弁モジュール、及びそれを使用する製品及びシステム。
Patent JP-2010529629-A (JP)
Title: 質量分析計の配置
IPC: H01J49/26
Filed: 2008-06-03
Abstract: 【解決手段】本発明は、質量分析計補助真空出口(30)を有する質量分析計補助真空室(20)を囲むハウジング(86)と、少なくとも２つの質量分析計高真空室(21,22,23)と、高真空室(21,22,23)と接続され、補助真空出口(89)を有する一体化されたターボ分子ポンプ(12)とを備えた質量分析計の配置(10)に関する。２つの補助真空出口(30,89) は、ハウジング(86)内の共通の補助真空空間(98)に延びており、補助真空空間はハウジング出口(88)に延びている。
Patent JP-2010530744-A (JP)
Title: アミロイドβに対するヒト化抗体
IPC: A61P35/00
Filed: 2008-06-12
Abstract: 本出願は、キメラ抗体およびヒト化抗体に関し、かつアルツハイマー病などのアミロイドタンパク質と関連する一群の障害および異常であるアミロイドーシスの処置における治療的および診断的使用のための方法および組成物に関する。
Patent JP-2010529577-A (JP)
Title: 画像をエンハンスする方法と装置
IPC: H04N5/20
Filed: 2008-06-05
Abstract: 画像をエンハンスする方法と装置が提供される。短波長赤外線（ＳＷＩＲ）カメラ、センサ、またはあらゆる他の撮像装置のような撮像装置によって生成された入力画像は、処理されて入力画像中のピクセル強度の分布を表す入力ヒストグラムを作成する。ヒストグラムスタートおよびエンドポイントが決定され、所望のエンハンスメントのタイプに依って可変プラトープロファイルが計算される。プラトープロファイルはあらゆる所望の形またはサイズを取ることができ、プロファイル中に2つ以上のプラトー領域を含むことができる。入力ヒストグラムは可変プラトープロファイルに沿ってクリップされる。累積ヒストグラムがクリップされたヒストグラムから作成され、正規化される。入力画像はそれから、正規化累積ヒストグラムをルックアップテーブルとして使ってエンハンス出力画像に変換される。
Patent JP-2010532751-A (JP)
Title: アミノ酸誘導体
IPC: A61P25/16
Filed: 2008-07-04
Abstract: 式(I)または式(II)：     ［式中、R 1 はカルボキシ、カルボキシエステルまたはカルボキシアミド基であり；R 2 は基-C(=O)-NR 3 R 4 または-S(=O) 2 -NR 3 R 4 であり；R 3 およびR 4 は、独立して、水素、任意に置換されていてもよいC 1 -C 6 アルキル、(C 1 -C 5 フルオロアルキル)-CH 2 -、-Qおよび-CH 2 Q（ここで、Qは3〜6の環原子を有し、任意に置換されていてもよい単環式の炭素環または複素環である）から選択されるか；またはR 3 およびR 4 は、それらが結合している窒素と一緒になって、3〜8の環原子を有し、任意に置換されていてもよい単環式のシクロアルキル環もしくは非芳香族複素環を形成し；R 5 は水素、またはペプチド結合を介して結合した天然もしくは非天然のα-アミノ酸の残基であり；R 6 は水素または基R 7 C(=O)-であり；そしてR 7 はC 1 -C 6 アルキル、C 1 -C 6 フルオロアルキルまたはシクロプロピルである］ の化合物は、ドーパミン作用性活性を有する。 【選択図】なし
Patent JP-2010534211-A (JP)
Title: ジヒドロピリジンカルシウムチャンネルアンタゴニストを含む薬学的組成物とその調製方法
IPC: A61K9/48
Filed: 2007-07-23
Abstract: 本発明は、生物学的利用能を向上させ溶解度を改善するためにアエロジル ＴＭ のようなコロイド状二酸化ケイ素と併用して、治療的有効量のレルカニジピン又はその塩のようなジヒドロピリジンカルシウムチャンネルアンタゴニストを含有する固形投薬形態の製剤、及び湿式造粒法によるその調製方法に関する。