baber/WOPTO huggingface dataset:
Patent BR-112023015219-A2 (BR)
Title: Derivados de 3h,4h,5h,6h,7h-pirimido [4,5-b][1,4]oxazina-4,6-diona como inibidores de trpa1
Inventor: FLORIAN PAUL CHRISTIAN BINDER
IPC: C07D498/04
Filed: 2022-04-13
Abstract: derivados de 3h,4h,5h,6h,7h-pirimido [4,5-b][1,4]oxazina-4,6-diona como inibidores de trpa1. a presente invenção fornece determinados derivados de 3h,4h,5h,6h,7h-pirimido[4,5-b][1,4]oxazina-4,6-diona que são inibidores do receptor do potencial de anquirina 1 transitório (trpa1) e são, portanto, úteis para o tratamento de doenças tratáveis por inibição de trpa1. também são fornecidas composições farmacêuticas que contêm os mesmos e processos para preparar os ditos compostos.
Patent BR-112023019781-A2 (BR)
Title: Fosfolipídeos como agentes quelantes de ânions em formulações farmacêuticas
Inventor: GIANG HOANG THUY AU
IPC: A61K9/00
Filed: 2022-03-31
Abstract: fosfolipídeos como agentes quelantes de ânions em formulações farmacêuticas. são descritas aqui formas de dosagem incluindo um material de preenchimento que incorpora um agente quelante aniônico, tal como lecitina, e uma forma de sal de um ingrediente farmacêutico ativo básico ou ácido e um íon livre. a relação molar do agente quelante aniônico, tal como a lecitina, para o íon livre varia de cerca de 0,5 a cerca de 3. da mesma forma descritos aqui são métodos de estabilização de formas de dosagem que incluem uma forma de sal de um ingrediente farmacêutico ativo básico ou ácido, métodos de preparação de tais formas de dosagem e métodos de utilização de tais formas de dosagem.
Patent BR-112023020345-A2 (BR)
Title: Transmissão multi-slot para pontos de recepção multi-transmissão
Inventor: SRIDHARAN GOKUL
IPC: H04L5/00
Filed: 2022-04-12
Abstract: transmissão multi-slot para pontos de recepção multitransmissão. certos aspectos da presente revelação fornecem técnicas para transmissão de bloco de transporte multi-slot com salto de frequência. um método que pode ser executado por um equipamento de usuário (ue) inclui a programação de recebimento de pelo menos um bloco de transporte a ser transmitido, através de múltiplos slots e a transmissão do bloco de transporte em múltiplas ocasiões de transmissão, através de múltiplos slots, de acordo com o salto de frequência aplicado para variar os recursos de frequência usados em ocasiões de transmissão.
Patent BR-122020025357-A2 (BR)
Title: sistemas para uso no fraturamento de formações subterrâneas e para uso na entrega de fluido pressurizado a um furo de poço a ser fraturado e método de entrega de fluido pressurizado a furo de poço para ser fraturado
Inventor: ELDON SCHELSKE
IPC: E21B43/12
Filed: 2012-04-06
Abstract: A presente invenção provê um método e sistema para fornecer energia elétrica no local para uma operação de fraturamento, e um sistema de fraturamento alimentado eletricamnente. Gás natural pode ser utilizado para acionar um gerador de turbina na produção de energia elétrica. Uma frota de fraturamento alimentada eletricamente, escalonável é fornecida para bombear fluidos para a operação de fraturamento, evitando a necessidade de um fornecimento constante de combustível diesel para o local e reduzindo a pegada do local e infraestrutura exigida para a operação de fraturamento, quando comparado com sistemas convencionais.
Patent CZ-73589-A3 (CZ)
Inventor: BAUDYS BOHUSLAV
IPC: H02B5/02
Filed: 1989-02-03
Abstract: Transformační stanice sestává z transformátorů'(3), na než
je připojeno primární vedení (13) a sekundární vedení (12).
Transformační stanice je umístěna na dvojici základů (1) a
hlavním základu (2), případně monobloku (18), kde v hlavním
základu (2) nebo monobloku (18) jsou uloženy dva
sloupy (9), k nimž jsou přivedeny přívody (10). Na konci
přívodů (10) jsou umístěny kotevní izolátory (8) a za nimi
jsou na konzoli (17) na konci sloupu (9) umístěny závěsné
izolátory (14), pod nimiž jsou na sloupech (9) a mezi nimi v
primárním vedení (13) umístěny tři bleskojistky (7) a pod
nimi ještě podpěrné izolátory (6). Bleskojistky (7) jsou spojeny
s na primárním vedení (13) umístěnými pojistkami (5),
za nimiž jsou na primárním vedení (13) umístěny izolátory
(4) a primární vedení (13) je za nimi napojeno na
transformátory (3), uložené na základech (1) a hlavním základu
(2), případně monobloku (18). Kolem transformátorů
(3) je provedeno oplocení (11) a mezi základy (1), hlavním
základem (2), případně monoblokem (18) a oplocením (11)
je uložen makadam (15) pro zachycení oleje při havárii a
vně kolem oplocení (11) je vytvořena izolační vrstva (16).
Mezi pojistky (5) a podpěrné izolátory (6) mohou být do primárního
vedení (13) umístěny měřicí transformátory (19)
proudu a napětí.
Patent CZ-24796-A3 (CZ)
Title: Cable chain
Inventor: BLASE GUNTER
IPC: H02G11/00
Filed: 1994-07-26
Abstract: PCT No. PCT/DE94/00868 Sec. 371 Date Jan. 25, 1996 Sec. 102(e) Date Jan. 25, 1996 PCT Filed Jul. 26, 1994 PCT Pub. No. WO95/04231 PCT Pub. Date Feb. 9, 1995It is envisaged in the case of a power transmission chain (1) for guiding cables, hoses and the like in a cavity surrounded by the chain links, with several chain straps (2, 3) which can be connected in detachable fashion by upper and lower cross-members, which are assembled to form two parallel strands, overlap each other and can be angled in relation to each other, and which interlock positively in the area of the mutual overlap, that each of the parallel chain strands includes inner straps (2) and outer straps (3). Each outer strap (3) overlaps two inner straps (2). The areas of the chain straps (2, 3) which are intended to overlap the adjacent chain straps (2, 3) are arranged in a common plane which roughly forms the mid-length plane of the chain straps (2, 3). (FIG.
Patent CZ-31693-A3 (CZ)
Inventor: PESL ALES ING CSC
IPC: F41G3/00
Filed: 1993-03-03
Abstract: Bezkontaktní ovládání laserového zaměřovače (2) je založeno
na jeho aktivací přirozeným pohybem, provádéným
při ovládání spouště ruční zbraně (1). Bezkontaktní laserový
zaměřovač (2) má za tím účelem ve své sestavě zabudován
pyrodetektor (3) pro snímání dynamických změn
gradientu teplotního pole ve svém okolí.
Patent CZ-33199-A3 (CZ)
Title: 1,4-disubstituted piperidine derivatives containing fluorine
Inventor: TSUCHIYA YOSHIMI
IPC: C07D211/58
Filed: 1997-07-28
Abstract: This invention relates to novel fluorine-containing 1,4-disubstituted piperidine derivatives represented by a general formula ÄIÜ <CHEM>  and pharmaceutically acceptable salts thereof,  Äwherein:   Ar represents an aryl group or a hetero-aryl group having 1 to 2 hetero atoms selected from a group consisting of nitrogen, oxygen and sulfur (any 1 to 3 hydrogen atoms on the ring of said aryl or heteroaryl group may be substituted with lower alkyl, etc.); R<1> represents C3-C6 cycloalkyl whose any 1-4 hydrogen atmos may be substituted with fluorine atoms(s); R<2> represents C5-C15 saturated or unsaturated aliphatic hydrocarbon groups whose any 1 to 6 hydrogen atoms may be substituted with fluorine atom(s), aralkyl, arylalkenyl, heteroarylalkyl or heteroarylalkenyl group having 1 to 2 hetero atoms selected from a group consisting of nitrogen, oxygen and sulfur (optionally any 1 to 3 hydrogen atoms on the ring in said aralkyl, arylalkenyl, hetero-arylalkyl or heteroarylalkenyl group may be substituted with lower alkyl, trifluoromethyl, cyano, hydroxyl, nitro, lower alkoxycarbonyl, halogen, lower alkoxy or amino, etc. ; and   X stands for O or NH, provided that at least either one of R<1> and R<2> contains one or more fluorine atomsÜ.   The compounds of the present invention have selective antagonistic activity for muscarinic M3 receptors, and exhibit excellent oral activity, duration of action and pharmacokinetics, so that they have little side effects and are safe and effective. Therefore they are useful for treatment or prophylaxis of respiratory diseases, urinary diseases and digestive diseases.
Patent CZ-45298-A3 (CZ)
Inventor: STARZEWSKI JIRI
IPC: A62B35/00
Filed: 1998-02-16
Abstract: Zařízení k humánnímu systému dopravy raněných,
zejména při přepravě pacientů na nosítkách
je tvořeno popruhy /1, 3, 4/, jakož i
úchyty /7/ s otvory /8/ a vybráním /9/ k připevnění
karabin /11/ na oka nosítek /12/ i
přezkami /6/ pro úchýt karabinek /10/ na
přední části. Hlavní popruh /1 / je vředu spojen
sponou /2/, přičemž popruhy /1, 3, 4/
jsou spojeny ve spojeních /5/.
Patent CZ-54397-A3 (CZ)
Title: Composite materials from silicon dioxide and zeolite in spherical form, process of their preparation and their use
Inventor: BALDUCCI LUIGI
IPC: C01B39/02
Filed: 1997-02-21
Abstract: The present invention relates to silica/zeolite composite materials in spherical form and the process for their preparation which occurs by the dispersion of submicronic particles of titanium silicalite, beta zeolite, or mixtures of beta zeolite with titanium silicalite, in a silica sol synthesized by acid hydrolysis of silicon alkoxides; the hybrid sol thus obtained, subjected to emulsification and gelation techniques in organic mediums, produces these materials in a spherical form with an average diameter of between 20 and 150  mu m and containing up to 70% by weight of titanium silicalite, beta zeolite or mixtures of titanium silicalite/beta zeolite. The materials of the invention, having a high mechanical resistance and characterized by a surface area of between 300 and 800 m<2>/g, are applied as catalysts; in particular, those consisting of titanium silicalite or mixtures of titanium silicalite/beta zeolite are advantageously used in oxidation reactions of organic compounds with hydrogen peroxide.
Patent CZ-54798-A3 (CZ)
Title: Toothbrush and process for producing thereof
Inventor: HALM HANS
IPC: A46B7/06
Filed: 1996-08-22
Abstract: A toothbrush in which the head comprises a base region adjoining the handle, and a tip region, the tip region being flexibly and resiliently linked at the link region to the base region in a manner which enables the tip region to pivot resiliently relative to the base region during toothbrushing. The base region or tip region are in the form of two limbs which partly surround a part of the tip or base region respectively, which extends in the respective base or tip direction between these two limbs.
Patent CZ-71896-A3 (CZ)
Title: Apparatus for detecting identifiers of elements within a telecommunications system
Inventor: IJKELENSTAM EVERT PIETER
IPC: H04M3/28
Filed: 1994-09-08
Abstract: System for detecting the identifier of a component of a telecommunication system such as a terminal component, transmission component or switching component. The system comprises a detector (2) which is connected to the component (3), furthermore a remitter (4) which is connected to a second component (5). The detector dials the second component, and the telecommunication system transmits the identifier of the first component to the remitter ("calling number display" service). The remitter sends the identifier of the first component back to the detector, where the requested identifier can be read out on a display. To summarize, relatively large savings are obtained by only one operator instead of two necessary for testing; time gained in the event of malfunctions; direct and undistorted data exchange; recording of the data on a printer possible; fits into a system for guaranteeing quality; increases the performance of the telecommunication system; avoids unnecessary investment in cable/bundle/channel capacity.
Patent CZ-82698-A3 (CZ)
Title: Use of 5-ht3 receptor antagonists for preparing a pharmaceutical preparation for treating dikinesis
Inventor: RICE GEORGE PETER ARTHUR
IPC: A61K31/40
Filed: 1996-09-16
Abstract: The invention provides the use of a 5-HT3 receptor antagonist or a pharmaceutically acceptable derivative thereof for use in the treatment of dyskinesia.
Patent SK-16195-A3 (SK)
Title: Benzoxazinone derivatives, pharmaceutical agents containing thereof and method of production of these derivatives
Inventor: YOUNG STEVEN D
IPC: A61K31/54
Filed: 1993-08-06
Abstract: Benzoxazinone derivatives of general formula (I), which can be used for inhibition of reverse transcriptase HIV including their resistant variants, for prevention or treatment of HIV infection and for treatment of AIDS; their pharmaceutically acceptable salts; pharmaceutical preparations containing them in combination with other antiviral substances, immunomodulators, antibiotics or vaccines and their use.
Patent SK-33198-A3 (SK)
Title: Integrated reactor for biological treatment of waste waters
Inventor: SALAT MIROSLAV
IPC: C02F3/12
Filed: 1998-03-12
Abstract: An integrated reactor for biological cleaning of all sorts of wastewater with biologically removable pollution is compactly designed in one tank. A V - shaped settling chamber (2) is located between a denitrification zone (1) and a nitrification zone (3), which separates the mentioned zones and is used to separate biological sludge from cleaned water by countercurrent sedimentation. The wastewater is fed into the denitrification zone (1), in which a stirrer (10) is installed, designated for thorough mixing of the activated reverse sludge with the wastewater. From there, the mixture of the denitrificated sludge and water flows through a pipe (8) to the opposite wall of the reactor, into the nitrification zone (3). The required amount of oxygen is supplied by an aeration system (9) to the nitrification. The nitrification zone (3) is linked with the settling chamber (2) through a stabilising zone (4), whose lower part at the same time serves as a place for cumulating of the settled sludge. In this part, there is a device (7) installed for draining of the sludge, to which a pump (16) of the reverse sludge is connected, whose delivery ends directly above the level of the denitrification zone (1). The cleaned water mixed with the activated sludge, free of oxygen, flows into the settling area, where the sludge settles and at the same time a lifted layer of sludge is formed, throughout which the cleaned water is strained. The cleaned water flows out through a discharge channel. Where appropriate, it is possible to use the broken scumboards to intensify the whole process.
Patent SK-36196-A3 (SK)
Title: Two-step masonry impregnation water repelling method
Inventor: WEBER HELMUT
IPC: C04B41/49
Filed: 1996-03-15
Abstract: Making new or old masonry water repellent Impregnation of masonry to make it water repellant is effected in 2 steps by: (1) treating with a highly dispersed aqueous emulsion of (A1) an organoalkoxysilane and/or (A2), alkoxy group containing organosiloxane and (B) salts of water-soluble (in)organic acids and organopolysiloxanes, there being siloxane units monovalently attached to SiC groups containing basic N such that there is at least 0.5 wt. % basic N based on the organopolysiloxane wt.; and (2) treating with an aqueous solution of (C1) alkali silicate and/or alkali siliconate (C2) or mixture of alkali silicate and alkali siliconate in water.
Patent SK-43897-A3 (SK)
Title: Treatment of multiple sclerosis (ms) and other demyelinating conditions using lofepramine in combination with l-phenylalanine, tyrosine or tryptophan and possibly a vitamin b12 compound
Inventor: LODER CARI
IPC: A61K31/66
Filed: 1995-10-05
Abstract: The use of a combination of a tricyclic antidepressant or a monoamine oxidase inhibitor with a amino acid compound neurotransmitter-inducing for the preparation of medication for the treatment or prevention of multiple sclerosis or other demyelinating conditions. Indicating compound it that is L-phenylalanine, tyrosine or tryptophan, lofepramine is an antidepressant with addition of vitamin B12.
Patent SK-78096-A3 (SK)
Title: Method of reducing a steam consumption at the tyre production and device for carrying out this method
Inventor: BAFRNEC MILAN
IPC: B29C48/92
Filed: 1996-06-14
Abstract: At the moment when the liquid is displaced from the membrane (1) the gas starts to flow through effluent pipe (2). Sensor (6) placed in this pipe measures the size of medium parameter, which changes by hop-off, when the liquid stops to flow aroung the sensor (6) and the gas starts to flow. Signal sent by sensor (6) is evaluated by control computer (7) or automatic controller (7) and/or alarm unit (7), which sends commands to close actuating device (4) of inflow of extruding gas to the membrane and to close actuating device (5), through which the liquid is displaced from the membrane (1). At the same time the concerned period of the production run is finished. Device for realization for this method consists of membrane (1), pipe for displaced liquid abstraction (2), pipe for inlet of the extruding gas (3), actuating devices (4) and (5), sensor (6), control computer (7) or automatic controller (7) and/or alarm unit (7), liquid accumulating pipe (8).
Patent SK-93999-A3 (SK)
Title: Expandable gastro-retentive therapeutic system with controlled active substance release in the gastro-intestinal tract
Inventor: ASMUSSEN BODO
IPC: A61M31/00
Filed: 1998-01-09
Abstract: The invention concerns a device for the controlled release of active substances in the gastro-intestinal tract with a retarded passage through the pylorus, the device comprising a component which can expand on contact with gastric juice and is surrounded by a polymer casing which is permeable to gastric juice and active substances. The device comprises at least one active substance in the form of a multi-particle preparation which releases the active substance into the gastric juice in retarded manner. The release of active substance from a device according to the invention can be controlled better than conventional medicaments with a retarded passage through the pylorus. Similarly, the device can easily be rolled or folded and inserted in capsules without difficulty.
Patent CZ-184693-A3 (CZ)
Title: Concentrated textile plasticizing mixtures
Inventor: HUBESCH BRUNO ALBERT JEAN
IPC: C11D1/835
Filed: 1992-01-30
Abstract: Concentrated fabric softening compositions are described which retain viscosity upon dilution in water. The compositions comprise cationic fabric softening actives, as well as a specific combination of emulsifiers and polymers. The present invention also encompasses a method for the softening of fabrics.
Patent CZ-223793-A3 (CZ)
Title: Method of detecting and measuring activity of neurotrophins, method of cloning a gene for tyrosinkinase and a recombinant molecule of nucleic acid, cell, micro-organisms and protein thereof
Inventor: SQUINTO STEPHEN P
IPC: G01N/
Filed: 1992-04-23
Abstract: The present invention provides for assay systems that may be used to detect and/or measure neurotrophin activity or to identify agents that exhibit neurotrophin-like activity. It is based, at least in part, on the discovery that the trkB proto-oncogene encodes a tyrosine kinase receptor that may serve as a functional binding protein for BDNF and NT-3. The present invention also provides for diagnostic and therapeutic methods based on the interaction between BDNF and/or NT-3 and trkB, and for a number of orphan receptor molecules. <IMAGE> <IMAGE> <IMAGE> <IMAGE> <IMAGE> <IMAGE> <IMAGE> <IMAGE> <IMAGE>
Patent CZ-601989-A3 (CZ)
Inventor: PRACHAR OLDRICH ING
IPC: E02B7/20
Filed: 1989-10-25
Abstract: V průtočném otvoru klapkového uzávěru mezi jednotlivými
uzavíracími klapkami (1) umístěna pevná svislá žebra (2),
jejichž čela jsou zkosena a opatřena těsněním (3). Tato
žebra (2) tvoří opěry uzavíracích klapek (1) v zavřené poloze
uzávěru.
Patent CZ-119095-A3 (CZ)
Title: Process for preparing n-methylmorpholinoxide with a low content of nitrosomorpholine
Inventor: PASEK JOSEF PROF ING DRSC
IPC: C07D295/24
Filed: 1995-05-09
Abstract: A method of preparation of a 50 to 60 % mass of NMMO solution with a content of 100 to 300 ppb NOMOR by oxidation of a mix of NMM and an aqueous solution of hydrogen peroxide at a temperature of 55 to 70 degrees C. The working molar ratio of H2O2/NMM=0.4 to 0.7, preferably 0.5 to 0.65, whereas the peroxide solution is added to an amine solution for 2 to 5 hours and the mixture is left to react at reaction temperature for 3 to 5 hours. Unprecipitated NMM is removed from the reaction mix by vacuum rectification.
Patent CZ-120998-A3 (CZ)
Inventor: DYNTAR MILOS
IPC: G05D16/20
Filed: 1998-04-21
Abstract: Zevní stínící zařízení pro otočné střešní okno
zahrnuje pás /54/ ze stínícího materiálu,
který je navinut na pružně předpjatěm válci
/11/ a je spojen se spodní tyčí /7/ vedenou v
bočních vodících kolejničkách /9, 10/, která
je spojena přes lankový pohon /14, 15/ s odvinovací
hnací jednotkou /12, 13/. Boční vodící
kolejničky /9, 10/ pro spodní tyč /7/ probíhají
podél částí /3/ bočních částí rámu, situovaných
nad osou /2/ otáčeni, a podél částí
/4/ bočních částí rámu, situovaných pod
osou /2/ otáčení. K stínícímu pásu /5/ je
upevněno nosné zařízení /8/ v podstatě ve
tvaru tyče, které prochází přes tento pás /5/ a
je vedeno v bočních vodících kolejničkách /9,
10/ tak, že v poloze použití pro stínící zařízení
je umístěno v ose /2/ otáčení nebo v blízkosti
osy /2/ otáčení a paralelně s ní. Zařízení
může být opatřeno prostředky pro opětovné
napnutí a vyhlazení pásu /5/ v plně vytažené
poloze a v průběhu převíjení.
Patent CZ-200253-A3 (CZ)
Title: Resin for a binding agent, product, manufacturing process and use
Inventor: HANSEN RRLING
IPC: C04B14/46
Filed: 2000-07-07
Abstract: Resin for a binder suitable for mineral fibers such as glass or stone wool, said resin comprising the reaction product of a polymer free mixture of an amine with a first anhydride and a second anhydride, characterized in that the first and second anhydrides are different anhydrides.
Patent CZ-200785-A3 (CZ)
Inventor: KAZEHARE HIROYUKI
IPC: D05B47/04
Filed: 2007-02-01
Abstract: Zarízení pro napínání nite obsahuje dvojici napínacích kotoucu (31, 32), které mezi sebou pridržujínit, hnací mechanismus (4), ovladatelný pro zajištování pohybu jednoho napínacího kotouce smerem k nebo smerem od druhého napínacího kotouce, a hnacízdroj (5) ovladatelný pro pohánení pohánecího mechanismu. Hnací zdroj obsahuje pohybové ústrojí (6), obsahující hrídel (51) pohybového ústrojí, kterýse pohybuje v osovém smeru, a permanentní magnety(52,53,54,55), pripevnené ke hrídeli (51) pohybového ústrojí (6), stator (7), obsahující cívky (57,58,59,60), které jsou navinuty kolem permanentníchmagnetu s predem stanoveným intervalem vzhledem kpermanentním magnetum, a ložiska (40,8), která nesou príslušné konce hrídele pohybového ústrojí. Ložisko (40,8), které nese konec hrídele (51) pohybového ústrojí (6) na vzdálené strane od dvojice napínacích kotoucu (31,32) je deskové pružinové ložisko (8), vytvorené z deskové pružiny.
Patent CZ-202893-A3 (CZ)
Inventor: UTIKAL JAROSLAV
IPC: E03F5/10
Filed: 1993-09-29
Abstract: Zařízení pro čištění odpadní vody a výrobu bioplynu, sestávající
z vyhnívací nádrže (1) opatřené vtokem (11) odpadu
WC a venkovním vhozovým skluzem (13) domovního biologického
odpadu z hydrotermické jímky (2). Hydrotermická
jímka (2) je opatřena přítokem (21) domácí odpadní vody,
obklopující alespoň jednu boční stěnu vyhnívací nádrže (1).
Vyhnívací nádrž (1) je opatřena jímacím zvonem (5) a s
hydrotermíckou jímkou (2) je spojena s prvním přepadem
(14).
Patent CZ-207696-A3 (CZ)
Title: Attachment of nose support to a spectacles rim
Inventor: WINKLER ROLF
IPC: G02C5/22
Filed: 1995-01-11
Abstract: A retainer for securing a nose pad on an eyeglasses frame, the retainer being composed of a flat, one-piece pad arm having a receiving opening in the form of an elongated hole, and a retaining element of plastic secured to the nose pad, the retaining element having a constriction and being receivable in the receiving opening of the pad arm to be locked in the receiving opening by engagement of the constriction in the opening. The pad arm is a bilaterally symmetrical structure having a first end in which the opening is formed, is made of material which extends continuously around the opening and is substantially inelastic around the opening. The opening cross section of the elongated hole is selected and the retaining element is formed such that when the constriction engages in the receiving opening, a transition surface of the retaining element is engageable with the pad arm for allowing the retaining element and the nose pad to be pivotable and tiltable relative to the pad arm.