baber/WOPTO huggingface dataset:
Patent TW-I411645-B (TW)
Title: Adhesive composition of low molecular weight polyaminopolyamide-epichlorohydrin (pae) resin and protein
Inventor: SPRAUL BRYAN K
IPC: B27N3/00
Filed: 2007-08-24
Granted: 2013-10-11
Abstract: The invention is directed to compositions containing polyamidoamine-epihalohydrin resins (PAE resins) of low molecular weight and a soy protein or lignin in which the weight ratio of protein or lignin to PAE is 100:0.1 to 0.1:100. The invention is also directed to the use of the compositions as adhesives for binding wood materials. The lower adhesive viscosity provides better handling properties, as well as allowing for less water in the adhesive formulation. The lower viscosity provides for both ease of handling of the adhesive material and the pot life if the adhesive formulation
Patent TW-I406455-B (TW)
Inventor: UKITA YOSHIO
IPC: H01R13/46
Filed: 2008-01-18
Granted: 2013-08-21
Abstract: An outlet device, which is to be arranged on a wall surface, includes an outlet box in which electric wiring and optical interconnection are to be accommodated, and a cover plate which covers the outlet box. The cover plate includes a plate surface formed with an opening section through which an electric connection port of at least one of a telephone jack and an electric power supply outlet is to be exposed, and a bulged portion formed, on left or right side of the plate surface, to bulge frontward from the plate surface. The bulged portion is operable to accommodate a connection adaptor to which an optical connector attached directly to an end portion of an optical fiber is fitted, and includes a bottom face formed with an opening through which an optical connection port of the connection adaptor is to be exposed so as to be oriented downward.
Patent TW-I409899-B (TW)
IPC: H01L21/67
Filed: 2008-08-28
Granted: 2013-09-21
Abstract: This invention is an automatic tray-changing device. A feeding tray and a collecting tray with different specification are individually placed on a feeding platform and a collecting platform. The memory of a controller is preset with the location information of each storage tank of the aforementioned feeding tray, and the location information of each groove of the collecting tray. Therefore, the controller can control a picking and placing device to pick the chip out one at a time from the feeding tray and place it one at a time into the collecting tray. It is beneficial in performing the automatic IC tray exchanging operation between the feeding tray and the collecting tray, which are different in specification. It can improve the work efficiency in picking and placing chips and reduce the defective rate of chip. In addition, both the feeding tray and the collecting tray can individually recede to the empty tray position in the back along its sliding rail. Finally, empty trays or full trays can be automatically collected by a tray-collecting device to further improve the work efficiency.
Patent TW-I411983-B (TW)
IPC: G09F19/12
Filed: 2009-07-14
Granted: 2013-10-11
Abstract: The invention relates to an image-text picture exhibition structure, in which one independent image-text picture is generated respectively at two opposite observation directions. The technological means for the invention is: a picture device is a prismatic body with bottom faces upward and isosceles triangle shape, two vertex angles of the prismatic body are calculated by a formula; the fixing base corresponding to each picture device is equipped with a positioning slot respectively; a first and a second holding surfaces are disposed on the positioning slot wherein its surface sides are equipped with image-text portions. The image-text portion of the first and/or the second holding portion of each positioning slot is fully reflected through the picture device so that the image-text picture of the image-text portions of the second and/or the first holding surfaces can be observed from each of two opposite observation directions within the scopes of first and second vision line; furthermore, the picture device is disposed on the slot by a non-adhesion method, where a gap filled with air is formed between the picture device and the fixing base.
Patent TW-I411829-B (TW)
IPC: G02B7/04
Filed: 2009-09-02
Granted: 2013-10-11
Abstract: The present invention discloses an assembling and adhesive drying method for optical lens, which comprises: a lens components assembling step, a cushion assembling step, an adhesion disposing step, a pre-drying step, an encapsulation step and an after-drying step. The UV drying lamp is used to half-drying the adhesion disposed on the optical lens in which a filter has not been assembled for preventing the mist caused by re-drying of the adhesion from adhering to the lens of the optical lens, hence the optical quality of the lens could be improved.
Patent TW-I413898-B (TW)
Title: Method and system for data protection, storage device, and storage device controller
Inventor: YU HSIANG HSIUNG
IPC: G06F21/62
Filed: 2009-09-15
Granted: 2013-11-01
Abstract: A method and a system for protecting data, a storage device, and a storage device controller are provided. In the present method, when a host accesses data in the storage device, whether the host performs a play operation or a copy operation on the data is first determined. If the host performs the play operation on the data, the storage device continues to execute the play operation so as to allow the host to access the data. On the other hand, if the host performs the copy operation on the data, the storage device executes an interference procedure so as to prevent or retard the data from being copied into the host.
Patent TW-I400012-B (TW)
Title: Conformal reference planes in substrates
Inventor: VELAYUDHAM KARIKALAN SAMPATH KOMARAPALAYAM
IPC: H05K9/00
Filed: 2009-10-28
Granted: 2013-06-21
Abstract: Methods, systems, and apparatuses for circuit boards are provided herein. An electrically insulating material is formed over one or more traces on a circuit board. One or more further electrically conductive features are present on the circuit board. A layer of an electrically conductive material is formed over the one or more traces that is electrically isolated from the one or more traces by the electrically insulating material, and is in electrical contact with the one or more further electrically conductive features. The electrically conductive material confines magnetic and electric fields produced when the one or more traces conduct an alternating current. By confining the magnetic and electric field distributions in this manner, problems of interference and/or crosstalk with adjacent signal traces are reduced or eliminated.
Patent TW-I408617-B (TW)
Title: Method for testing and classifying performance of graphic processing unit under overclock operation
Inventor: HUANG SHUN CHIH
IPC: G06F1/08
Filed: 2010-05-05
Granted: 2013-09-11
Abstract: A method is applied to test and classify the performance of a graphic processing unit (GPU) under overclock operation. The GPU has a testing overclock band, and the testing overclock band includes a plurality of testing overclock frequencies. In the method, it is necessary to input an operating voltage to the GPU to make the GPU operate under the testing overclock frequencies, so as to obtain a frequency-standard power consumption curve. Following up, it is necessary to increase the operating voltage for the GPU to make the GPU also operate under the testing overclock frequencies, so as to obtain a frequency-increase power consumption curve. Finally, it is necessary to compare the slope of the frequency-standard power consumption curve and the slope of the frequency-increase power consumption curve to accordingly classify the GPU.
Patent TW-I394598-B (TW)
Title: Particle beam irradiation apparatus and particle beam therapy apparatus
Inventor: IWATA TAKAAKI
IPC: G21K1/093
Filed: 2010-08-09
Granted: 2013-05-01
Abstract: The objective is to eliminate the effect of the hysteresis of a scanning electromagnet so that there is obtained a particle beam irradiation system that realizes high-accuracy beam irradiation.  There are provided a magnetic-field sensor (20) that measures the magnetic field of a scanning electromagnet (3) and an irradiation control apparatus (5) that controls the scanning electromagnet (3) based on a measurement magnetic field Bs measured by the magnetic-field sensor (20) and target irradiation position coordinates Pi of a charged particle beam (1b). The irradiation control apparatus (5) is provided with an inverse map means (22) that calculates a target magnetic field Bi, based on the target irradiation position coordinates Pi of the charged particle beam (1b); and a compensator (23) that outputs a control input Io, to the scanning electromagnet (3), for controlling the magnetic-field error Be between the target magnetic field Bi and the measurement magnetic field Bs to be the same as or smaller than a predetermined threshold value.
Patent TW-I403509-B (TW)
Title: A pharmaceutical composition for treating cancer
Inventor: CHANG LI CHIEN
IPC: C07D413/06
Filed: 2010-12-27
Granted: 2013-08-01
Abstract: Disclosed herein is a new use of a pyrrolidone derivative, particularly, the use of the pyrrolidone derivative for treating a subject suffering from a cancer. A pharmaceutical composition for treating cancer is provided accordingly. The pharmaceutical composition includes a pyrrolidone derivative, a salt or a solvate thereof; and a pharmaceutically acceptable carrier. The pharmaceutical composition may further include a chemo therapeutic agent.
Patent TW-I404553-B (TW)
Title: Lower limb strength enhancement device
Inventor: CHEN DAR ZEN
IPC: A63B23/04
Filed: 2010-12-28
Granted: 2013-08-11
Abstract: A lower limb strength enhancement device for training or rehabilitation is disclosed. The lower limb strength enhancement device comprises a first fixing element, a first linkage set, a second linkage set, a first elastic element and a second elastic element. The first linkage set comprises a first end and a second end, the first end of the first linkage set is connected to the first fixing element. The second linkage set comprises a first end and a second end, the first end of the second linkage set is connected to the first fixing element. Two ends of the first elastic element are pivoted individually to a first pivoting point and a second pivoting point of the first linkage set. Two ends of the second elastic element are pivoted individually to a third pivoting point and a fourth pivoting point of the second linkage set.
Patent GB-2488972-B (GB)
Title: A locking pin
Inventor: SARGEANT MICHAEL JOHN
IPC: B65F1/16
Filed: 2011-02-23
Granted: 2013-04-24
Abstract: A locking pin is formed of two sheet like components, the edge of one 34 being secured perpendicularly against the planar face of the other 28 to reinforce it. The reinforcing component 34 includes a hook formation extending around the end of the planar component into its plane. Both sheets have generally constant width. The ends of both sheets preferably include a rounded tapered so that the pins entire tip is has a rounded taper but a flat end. The components ideally engage by tabs on the reinforcing sheet extending into slots on the planar sheet and secure to the far side of the planar sheet. The planar component and/or the reinforcing component may be made of two layers, in this case the tabs of each layer could be staggered.
Patent GR-7535-B (GR)
Title: Βελτιωσεις εν σχεσει με την ιδια βροχοποιησιν υφαντουργικων ινων, ελασματων και παρομοιων.
Inventor: HIGGINS ERIC BERKELEY
Filed: 1938-05-27
Abstract: εφεύρεσης αυτή αναφέρεται εις την κατεργασία υφαντουργιών ινών δια να καθιστά ταύτας αδιάβροχα καιβασίζεται επί της παρατηρήσεως ότι συνδυασμοί, οιτινες συμβαίνουν μεταξύ ενίων αμφοτερικών μετάλλων, ιδίως ψευδαργύρου, αλουμινίου ή άλλων συνθέτων οωιδίων και αμφοτερικών πρωτεϊνών, ιδίως καζείνης, υπό όρων ελέγχου οξέων, κατέχουν εν ψιλό βαθμό ιδιότητος δι' αδιαβροχοποίησιν όταν αποσυντεθούν και μεταδίδουν την ιδιότητα ταύτη επί υφαντουργικών ινών εντός των οποίων απεροφήθησαν ή εντός ή εφ' ωνπαρήχθησαν, εν ω υπό συνθήκες αλκακίνης ουδεμία ένωσης λαμβάνει χώρα μεταξύ τούτων των αμφοτερικών σωμάτων .
Patent GR-16443-B (GR)
Title: Τελειοποιησεις εις η εν σχεσει προς χημικας συνθεσεις και παρασκευασματα αυτων.
Filed: 1954-06-09
Abstract: ία μέθοδος δια την παρασκευήν της 2-υποκατεστημένης ενώσεως της ιμιδαζολίνης, ήτις περιλαμβάνει τηνσυμπύκνωσιν μιάς ενώσεως επιλεγείσης εκ μιάς ομάδος αποτελουμένης εξ ενός καρβοξυλικού οξέος έχοντος τον τύπον (Ι) ένθα το n είναι 2 ή 3, και των εστέρων και του νιτριλίου τούτου, μετά αιθυλενοδιαμίνης.
Patent GR-16494-B (GR)
Title: Συγκροτημα αποχωριζομενης διαταξις συνδεσεως.
Filed: 1955-03-09
Abstract: μέθοδος κατασκευής ενός συγκροτήματος αποχωριζομένον συνδέτου του τύπου όστις έχει ένα στοίχον εκ στοιχείων εμπλοκής, στερεωμένων, εν σχέσει αποστάσεως από αλλήλων, κατά μήκος ενός δρομέως και τα οποία είναι κατάλληλα να εμπλέκονται κατά τρόπον θετικής αλληλεμπλοκκής, με ένα στοίχον εξ ομίων στοιχείων εμπλοκής στερεωμένων κατά την διεύθυνσιν του μήκους επί ενός άλλου δρομέως και όστις τύπος έχειεν ολισθαίνον μέλος διά την κατά αποχωριζομενον τρόπον σύνδεσιν και δια τον αποχωρισμόν των ρηθέντων στοιχείων εμπλοκής, ιδιά ταστάδια άτι να περιλαμβάνουν την κατασκευήν, επί τινος κορδονιοειδούς σώματος  επί μιάς συμβατικής ταινίας, και η ρηθείσα βάσις έχει τοιαύτην κατά εγκαρσίαν τομήν επιφάνειαν ώστε ο ηνωμένος εγκάρσιον όγκος ενός ζεύγους τοιούτων αλληλοσυνδεσμένων συγκροτημάτων συνδετών περιβάλλεται τελείως υπό του ολισθαίνοντος μέλους πρός οδήγησιν τούτου κατά μήκος των κορδονιοειδών σωμάτων.
Patent GR-17132-B (GR)
Title: Φορητη διαμορφωσεως γωνιας.
Filed: 1955-09-30
Abstract: ύκλωμα φωρατού γωνιακής διαμορφώσεως προς απόληψιν από γωνιακώς διαμορφωμένου σήματος τάσεως εξόδουεχούσης μέγεθος εξαρτώμενον από την διαμόρφωσιν του ρηθέντος σήματος, του ρηθέντος κυκλώματος φωρατού έχοντος μέσα προς σχηματισμόν του ρηθέντος σήματος εις κύματα των οποίων η αμοιβαία φασική σχέσιςμεταβάλλεται με την ρηθείσαν διαμόρφωσιν και προςδιανυσματικήν πρόσθεσιν των ρηθέντων κυμάτων ούτως ώστε να σχηματίζωνται δύο ταλαντώσεις μεταβλητώνευρών, ένθα μία των ρηθεισών ταλατώσεων εφαρμόζεται εις πρώτην ημιαγώγιμον ενισχυτικήν συσκευήν καιη άλλη των ρηθεισών ταλαντώσεων εφαρμόζεται εις δευτέραν ημιαγώγιμον ενισχυτικήν συσκευήν προς ανόρθωσιν και ενίσχυσιν αυτής, των ρηθεισών υμιαγωγίμων ενισχυτικών συσκευών ουσών αντιθέτου τύπου αγωγιμότητος, προβλέπονται δε μέσα προς συνδυασμόν των ρηθεισών ανορθωθεισών και ενισχυθεισών ταλαντώσεωνπρος παραγωγήν της ρηθείσης τάσεως εξόδου.
Patent GR-18166-B (GR)
Title: Μεθοδος και μεσα δια την παραγωγην υψηλων θερμοκρασιων.
Filed: 1956-05-12
Abstract: υσκευή διά την παραγωγήν υψηλών θερμοκρασιών, περιλαμβάνουσα μέσα διά την δημιουργίαν ενο συμπεπυκνωμένου μαγνητικού πεδίου περιβάλλοντος κατά ουσίανένα χώρον αντιδράσεως ,χαρακτηριζομένη εν μέσων διά την παραγωγήν ενός νέφους ή πλάσματος (plasma)ιόντων είς τον ρηθέντα χώρον αντιδράσεων παρουσία του ρηθέντος μαγνητικού πεδίου, ένθα ο χώρος αντιδράσεων είναι κατά ουσίαν ελεύθερος μαγνητικού πεδίου.
Patent GR-21717-B (GR)
Title: Μεθοδος παρασκευης νεων παραγωγων του αδαμαντανιου.
Filed: 1961-01-21
Abstract: αράγωγα του αδαμαντανίου του γενικού τύπου:
[*]
εις τον οποίον το Α παριστά δισθενή ρίζαν αλιφατικού υδρογονάνθρακος, κεκορεσμένην ή μη, μετ' αλύσεωςευθείας ή διακεκλαδισμένης, περιέχουσαν το πολύ 4άτομα άνθρακος ή δισθενή μονοπυρηνικής αρωματικήνρίζαν, καθώς και τα άλατα των παραγώγων του τύπου(1).
Patent GR-21873-B (GR)
Title: Συμπλοκον λιπασμα επι τη βασει του τριπολυφωσφορικου καλιου.
Filed: 1961-04-17
Abstract: προκειμένη εφεύρεσις έχει ως αντικείμενον:
1. Μίαν μέθοδον παρασκευής ενός συμπλόκου λειπάσματος επί τη βάσει του τριπολυφωσφορικού καλίου, ήτις μέθοδος συνίσταται εις την διαδροήν του τριπολυφωσοφικού καλίου δι' υδατικού διαλύματος φωσφορικού οξέος, και εις την υπό μορφήν κόκκων διαμόρφωσιν του μίγματος, εντός ατμοσφαίρας αμμωνίας.
2. Την χρησιμοποίησιν της κατά την αξίωσιν 1 μεθόδου, ήτις χαρακτηρίζεται εκ των ακολούθως σημείων λαμβανομένων μεμονωμένως ως κατά συνδυασμούς:
α. Το τριπολυφωσφορικόν συνδέεται με μίαν λιπαντική αζωτούχον ουσίαν.
β. Η λιπαντική αζωτούχος ουσία κατά την παράγραφον α είναι ουρία ή διαμμωνιακόν φωσφορικόν.
γ. Η αμμωνίωσις κατά την διάρκειαν της διαμορφώσεως εις κόκκους συνεχίζεται μέχρι του σχηματισμού διαμμωνιακού φωσφορικού.
Patent GR-22521-B (GR)
Title: Τελειοποιησεις εν σχεσει προς μηχανας στεγνωματοσδια περιδινησεως.
Filed: 1961-01-10
Abstract: ηχανή φυγοκεντρικού ξηραντηρίου περιλαμβάνουσα φυγοκεντρικόν θάλαμον συναρμολογημένον ώστε να περιστρέφεται πέριξ άξονος κεκλιμένου περί την κατακόρυφον κατά ουσιαστικήν γωνίαν εντός ακινήτου δοχείουτο οποίον αναρτάται ελαστικώς από υποστήριγμα χαρακτηριζομένη υπό μέσων παρεμποδισμού κινήσεων του σώματος του δοχείου κατά μίαν ή αμφοτέρας τας διευθύνσεις κατά μήκος του άξονος, περιλαμβνομένων συν_δεσμων συνδεδεμένων προς το δοχείον εις αντιθέτους πλευράς και εκτεινομένων εντεύθεν ουσιαστικώς παραλλήλως προς τον άξονα με τα άκρα των τα επιμεμακρυσμένα εκ του δοχείου συνδεδεμένα υπό διαφορικής διατάξεως επιτρεπούσης εις τον ένα σύνδεσμον να κινηθή κατά την μίαν διεύθυνσιν ενώ ο άλλος κινείταικατά την αντίθετον διεύθυνσιν ουσιαστικώς παραλλήλως προς τον άξονα.
Patent GR-34579-B (GR)
Title: Μεθοδος και διαταξις δια την απομακρυνσιν ακαθαρσιων εξ ορυκτων.
Filed: 1967-12-28
Abstract: έθοδος πρός απομάκρυνισν θειούχων ακαθαρσιών ώς π.χ. θειούχου αρσενικύ, έξ ορυκτών περιεχόντων τάς ακαθαρσίας ταύτας προ  της φρύξεως τούτων, χαρακτηριζομένη έκ του ότι τηρουεν τα ορυκτά ταύτα καθ' ομορροήν μετά ή κατ' αντιρροήν πρός α απαέρια της φρύξεως και άν χρειάζεται προσθέτων θερμών αερίων-φορέων έν αιωρήσει και εξαχνούμεν τάς ακαθαρσίας είς θεμοκρασίας καωθεν του σημείου μαλακύνσεως των ορυκτών, είς μίαν περιοχήν θερμοκρασιών από 650 βαθμους έως 1100 βαθμούς Κελσίου ενώ πρέπει να ληφθείπρός τούτο μέριμνα όωπς τα άερια δέν παρουσιάζουνή (παρουσιάζουν) μιάν κατα το δυνατόν μικράν περιεκτικότητα θείου.
Patent GR-77442-B (GR)
Inventor: GLICKMAN MICHAEL NEIL
IPC: E01C5/00
Filed: 1983-08-16
Abstract: A block for use in construction, particularly though not exclusively paving, has top and bottom surfaces one of which is a rectangle and the other of which is a square or a rectangle. In the case where the other surface is a rectangle the block has the major axes of the rectangles mutually perpendicular and has a shape at mid-height in horizontal cross-section which is substantially a square and the length of the side of said square is within the range 66% to 300% of the height of the block. In the case where the other surface is a square, the major axis of the rectangle is greater in length than the side of the square and the said square has a side of length within the range 66% to 300% of the height of the block.
Patent GR-850301-B (GR)
Inventor: CURRO JOHN JOSEPH
IPC: B29C67/00
Filed: 1985-02-04
Abstract: The present invention provides for a process for transforming a substantially continuous web of substantially planar, deformable material having an indefinite length, a first surface, and a second surface into a formed material. The material has a transofrmation temperature range. The process comprises the following steps:(a) The web of material is provided on a forming structure with the first surface of the web of material proximate a forming surface of the forming structure. The forming surface moves in a direction of the length of the web of material and carries the web of material in that direction.(b) A liquid stream is applied to the second surface of the web of material. The liquid stream has sufficient force and mass flux to cause the web of material to be deformed toward the forming surface, such that the material acquires a substantial three-dimensional conformation.(c) The temperature of the web of material is controlled such that it remains below the transformation temperature range of the material throughout the process.
Patent GR-851089-B (GR)
Inventor: GEORGIEV VESSELIN JORDANOV
IPC: A01G25/16
Filed: 1985-05-06
Abstract: A hydro-automatic valve with a cylindrical housing mounted vertically and having rigid upper and bottom ring shaped rests between which, within the cylindrical housing, interconnected upper and bottom face closure members are freely disposed. The upper face closure member is shaped as a disc with a hole in the central axis and has small legs arranged around its periphery extending vertically downwards with small teeth turned inwards towards the central axis. The small teeth are disposed freely in a shallow ring shaped groove in the surrounding surface of the bottom face closure member, which is shaped with a conical peak in the axis. At the bottom end of the bottom face closure member there is a deep ring shaped groove. This deep ring shaped groove is connected via parallel channels with the space between the upper and bottom face closure member. The cylindrical housing is connected to a centrally disposed lateral inlet hole and an outlet elbow above the upper ring shaped rest, to the basic distribution piping of the sprinkling irrigation system, and via a chamber with a lateral outlet hole, disposed underneath the bottom ring shaped rest, to the branch piping. In the bottom of the chamber, coaxial to the cylindrical housing, there is mounted a cylinder with a piston pin. The space of this cylinder underneath the piston is connected via a hole to additional control piping of the irrigation system.
Patent GR-860679-B (GR)
Title: Novel 3-pyridylmethylnaphthyl derivatives method for their preparation and their use as medicine
Inventor: HERMANN-HANS LAU
IPC: C07D213/26
Filed: 1986-03-12
Abstract: Compounds of the formula I    <IMAGE>  I  in which R1, R2, R3 and Y have the indicated meanings, their physiologically tolerated acid addition salts, and a process for the preparation of these compounds, are described. The compounds inhibit thromboxane synthetase and can thus be used as medicaments.
Patent IN-176618-B (IN)
Inventor: BEISSWENGER THOMAS
IPC: C07D339/04
Filed: 1993-09-01
Abstract: RS-Thioctic acid with a new morphology which is obtainable by a recrystallisation process is described.
Patent RS-52809-B (RS)
Inventor: SO SUNG-SAU
IPC: A61K31/185
Filed: 2009-11-09
Abstract: Jedinjenje koje ima formulu 1:ili njegove farmaceutski prihvatljive soli ili estri, gde:W je C(H)2, C(H)2-C(H)2, C(H)(CH3), CH2-C(H)(CH3), ili C(H)(CH3)-CH2;X je odabrano iz grupe, koja se sastoji od:(1) O,(2) N(H),(3) N(CH3),(4) S,(5) S(O) i(6) S(O)2;Y je ugljenik ili azot;R1 je odabrano iz grupe, koja se sastoji od:(1) vodonika,(2) halogena,(3) metila opciono supstituisanog sa fluoro,(4) C1-7 alkoksi opciono supstituisanog sa fluoro,(5) cijano i(6) nižeg alkilsulfonila;R2 je vodonik, fluoro, hloro, C1-7 alkil, ili niži alkoksi;R3 is vodonik, fluoro, hloro, bromo, ili metil; R4 je odabrano iz grupe, koja se sastoji od:(1) vodonika,(2) halogena,(3) C1-7 alkila opciono supstituisanog sa fluoro,(4) C3-7 cikloalkila i(5) etenila;R5 i R6, nezavisno jedan od drugog, odabrani su iz grupe koja se sastoji od:(1) vodonika,(2) halogena,(3) C1-7 alkila,(4) cijano i(5) C3-7 cikloalkila;R7 je cijano ili S(O)2-R8, pri čemu je R8 odabrano iz grupe, koja se sastoji od:(1) C1-7 alkila,(2) C3-7 cikloalkila,(4) C1-7 alkilamino,(5) C1-7 dialkilamino,(6) nižeg heterocikloalkila opciono supstituisanog sa halogenom, C1-7 alkilom, ili C1-7alkoksikarbonilom i(7) 2-oksa-6-aza-spiro[3.3]hept-6-ila.pri čemu"niži heterocikloalkil" se odnosi na zasićeni ili delimično nezasićeni ne-aromatični deo prstena koji ima 3 do 7 atoma u prstenu povezana zajedno kako formiraju prstenastu strukturu, gde su jedan, dva ili tri atoma prstena heteroatomi, dok su ostali atomi ugljenikovi atomi; ifarmaceutski prihvatljivi estri su metil i etil estri kiselina koje imaju formulu I, koji su za korišćenje kao prolekovi.Prijava sadrži još 17 patentnih zahteva.