baber/WOPTO huggingface dataset:
Patent IL-171500-A (IL)
Title: Triaza-and tetraaza-anthracenedione derivatives, their preparation and pharmaceutical compositions comprising them
IPC: C07D471/14
Filed: 2005-10-20
Abstract: A triaza- and tetraaza-anthracenedione derivatives, its stereoisomeric forms or mixture, or salts are new. A triaza- and tetraaza-anthracenedione derivatives of formula (I), its stereoisomeric forms or mixture, or salts are new. [Image] A : CR 6 or N; B : CR 7 or N; R 11-10C alkyl, 3-8C cycloalkyl, 2-10C alkenyl or 2-10C alkynyl (all optionally substituted by halo, CN, 3-8C cycloalkyl, phenyl, biphenylyl, naphthyl, indanyl or heteroaryl); R 2H, 1-4C alkyl, CF 3, -(CH 2) a-3-8C cycloalkyl, -(CH 2) a-phenyl, -(CH 2) a-imidazolyl or -(CH 2) a-pyridinyl; a : 0 - 2; R 3-(CH 2) b-phenyl, -(CH 2) b-imidazolyl, -(CH-2) b-triazolyl, -(CH 2) b-Het or -(CH 2) b-pyridinyl; b : 1 - 4; R 4 - R 7H, 1-4C alkyl, CF 3, 1-4C alkoxy, OCF 3, halo, nitro, CN, -CO-R 1 0, -NR 8R 9, -NH-CO-1-4C alkyl, -SO 2-NR 8R 9, -SO 2-1-4C alkyl or -SO 2-(CH 2) c-phenyl; c : 0 - 2; R 8 and R 9H or 1-4C alkyl; R 1 0OH, 1-4C alkoxy or -NR 8R 9; Het : a residue of a saturated 5- or 6-membered monocyclic heterocycle (contains a ring nitrogen via which it is bonded, and additionally contains a further ring heteroatom selected from N, O and S, and optionally substituted by 1-4C alkyl or -(CH 2) d-phenyl); d : 0 - 2; Heteroaryl : a residue of an aromatic 5 - 10 membered, monocyclic or bicyclic heterocycle (contains 1 - 4 N, O and S). The residues phenyl, biphenylyl, naphthyl, indanyl, heteroaryl, pyridinyl, imidazolyl and triazolyl are optionally substituted by halo, CN, 1-6C alkyl, CF 3, 1-6C alkoxy or OCF 3. A and B are not simultaneously N. An independent claim is included for preparation of (I). ACTIVITY : Cardiovascular-Gen.; Antianginal; Cardiant; Cerebroprotective; Vasotropic; Thrombolytic; Antiarteriosclerotic; Hypotensive; Respiratory-Gen.; Nephrotropic; Antiarrhythmic; Antidiabetic; Ophthalmological; Antiasthmatic; Antiangiogenic; Hepatotropic; Osteopathic. MECHANISM OF ACTION : Endothelial nitric oxide (NO) synthase (eNOS) expression stimulator. (4S)-9-(3-(Imidazo)-1-yl)propyl)-4-isopropyl-6-nitro-2-(4-phenylbutyl)-1,2,9,9a-tetrahydro-2,4a,9-triaza-anthracene- 3,10(4H)-dione trifluoroacetic acid (Ia) was tested for activation of eNOS transcription as described in Li et al., Activation of protein kinase C alpha and/or epsilon enhances transcription of the human endothelial nitric oxide synthase gene, Mol. Pharmacol. 53 (1998) 630. (Ia) Showed an EC 5 0 of 2.2 mM.
Patent IL-187231-A (IL)
Title: Pharmaceutica l compositions of a histone deacetylase (hdac) inhibitor and free arginine or salt thereof' use thereof and products containing the same
IPC: A61K/
Filed: 2007-11-08
Abstract: This invention pertains to pharmaceutical compositions comprising certain carbamic acid compounds (e.g., which inhibit HDAC (histone deacetylase) activity) (e.g., PXD-101, N-hydroxy-3-(3-phenylsulfamoyl-phenyl)-acrylamide)) and one or more additional ingredients selected from cyclodextrin, arginine, and meglumine. The present invention also pertains to the use of such compositions, for example, in the inhibition of HDAC, and in the treatment of conditions mediated by HDAC, cancer, proliferative conditions, psoriasis, etc.
Patent IL-193280-A (IL)
Title: Device for coupling between a plasma antenna and a power signal generator
Filed: 2008-08-06
Abstract: The present invention relates to a device for coupling between a plasma column serving as an antenna and an electric power signal generator, associated with a laser. This device comprises at least two conducting electrodes, each pierced with a hole, these holes being coaxial, the electrodes being connected on the one hand to a high voltage direct current source and on the other hand to power signal alternating current source, the laser(s) being placed do that its (their) beam arrives along the axis of said holes of the electrodes.
Patent IL-198116-A (IL)
Title: Carboxamides of pyrimidine condensed with 5- and 6-membered n-containing rings and pharmaceutical compositions comprising them
IPC: C07D/
Filed: 2009-04-07
Abstract: Provided herein are Heteroaryl Compounds having the following structure: wherein R1, R3, R4, L, X, Y, A and B are as defined herein, compositions comprising an effective amount of a Heteroaryl Compound and methods for treating or preventing cancer, inflammatory conditions, immunological conditions, metabolic conditions and conditions treatable or preventable by inhibition of a kinase pathway comprising administering an effective amount of a Heteroaryl Compound to a patient in need thereof.
Patent IL-201496-A (IL)
Title: Mammalian-type glycosylation in plants by expression of non-mammalian glycosyltransferases
IPC: A01H/
Filed: 2009-10-13
Abstract: The present invention relates to non-mammalian ²-1,4-galactosyltransferases that can be used in their wild-type or in modified forms. The invention further relates to transformed plants and plant cells expressing non-mammalian ²-1,4-galactosyltransferases and methods to produce glycoproteins with altered and preferably mammalian-type glycosylation. The invention additionally provides nucleic acid molecules and expression vectors of non-mammalian ²-1,4-galactosyltransferases.
Patent IL-206570-A (IL)
Title: Trisubstituted 3,4-dihydro-1h-isoquinoline compound, process for its preparation and its use
IPC: C07D/
Filed: 2010-06-23
Abstract: The present invention relates to the compound of formula 7*acetate (see below), a process for its preparation, and its use
Patent JP-S62256166-A (JP)
Title: File correction system
Inventor: YAMAMOTO YOJI
IPC: G06Q50/34
Filed: 1986-04-30
Abstract: PURPOSE:To eliminate a tabulation error generated by the trouble of a terminal controller by transmitting a processing number inquiry instruction for correcting a tabulation file to a terminal side when the trouble is generated and the system in current use is changed over to a spare system and correcting the tabulation file by a tabulation processor based on inquiry data and a processing number. CONSTITUTION:In a totalization processing system in which polling data AD the processing number are transmitted from a terminal, response data RD is returned from the tabulation processor thereby, the totalization of the polling data and the card issuance to the response data are carried out, when the trouble is generated in a terminal controller of a duplex constitution, and the system in current use is changed over to a spare system, the processing number inquiry instruction CD for correcting the tabulation file is transmitted to the terminal side, and the tabulation processor corrects the tabulation file based on the inquiry data AD fed from the terminal to the instruction CD and the processing number. Thereby, the tabulation error generated by the trouble of the terminal controller can be eliminated to improve the reliability of tabulation data.
Patent JP-H06289810-A (JP)
Title: Method and device for image display
Inventor: SUGAWARA MOTOO
IPC: G09G3/28
Filed: 1993-04-02
Abstract: PURPOSE:To suppress a decrease in the luminance of a display image and keep the white balance of the display image by the image display device which displays the image on a PDP. CONSTITUTION:The image display device which displays the image based upon an input digital video signal (R, G, and B signals) on the PDP 1 detects whether or not there is a skin color part as a stored color of said display image by a skin color detection part 2 and detects the luminance of the display image by a luminance detection part 3, and information on the presence or absence of the skin color and the luminance is inputted to an arithmetic part 4 to calculate data for gamma correction corresponding to the information; and a gamma-RAM 5 is rewritten with the data, the gamma correction of the input digital video signal is made with the data in the gamma-RAM 5, and the PDP 1 is driven with the gamma-corrected signal. Then the range of the input digital video signal level for keeping the white balance of the display image is varied according to the luminance of the skin color part (or luminance of the whole display image or means luminance) to keep the white balance below the luminance of the skin color part.
Patent JP-S62257194-A (JP)
Inventor: YANAIDA YOICHI
IPC: G09G3/00
Filed: 1986-04-30
Abstract: (57)【要約】本公報は電子出願前の出願データであるた め要約のデータは記録されません。
Patent JP-H11283913-A (JP)
Title: Filter device
Inventor: OTANI MASAMI
IPC: B01D24/00
Filed: 1998-03-27
Abstract: PROBLEM TO BE SOLVED: To provide a filter device, capable of easily attaching a member provided with a deaeration function and a gas dissolution function, even to an already provided processing liquid supply pipe, minimizing the routing of pipes, keeping compatibility between devices, miniaturizing a processing liquid supplying apparatus and lowering the cost. SOLUTION: For this filter device 24, a planar particle removal member 32 is disposed inside a hermetic container 30 provided with a processing liquid flow-in port 36, a processing liquid flow-out port 38 and a ventilation port 62, a planar gas permeable member 34 for which a ventilation path is formed of a gas permeable film material for transmitting only the gas, and the ventilation path communicating with the ventilation port 62 is disposed inside the hermetic container 30, and the ventilation port 62 communicates with a pressure reduction means or a gas supply means.
Patent JP-H04309038-A (JP)
Title: Congestion control system in packet exchange network
Inventor: TAKAHASHI TOSHIYUKI
IPC: H04L12/811
Filed: 1991-04-05
Abstract: PURPOSE:To implement communication restriction in response to the degree of congestion at the detection of congestion of a packet exchange network. CONSTITUTION:A logic communication line congestion detection section 2 of a packet exchange 1 detects congestion by using control information from other packet exchange inputted through a relay line 3. A restriction inhibiting new call connection is informed to a call control section 4 before a stage that an input restriction is noticed to the call control section 4 to restrict input of a packet to a terminal equipment 5 and sets a stage of rejection when a call connection request comes from the terminal equipment as the congestion detection. Communication is implemented by avoiding a rejected logic communication line. Thus, congestion control is executed in details to the terminal equipment and the service through the communication line with high reliability is offered to the terminal equipment.
Patent JP-H08270062-A (JP)
Title: Device for attaching and removing ditch cover
Inventor: IIJIMA KAZUE
IPC: E02D29/12
Filed: 1995-03-31
Abstract: PURPOSE: To make it possible to safely and speedily attach and remove a road ditch cover by anybody without requiring skill. CONSTITUTION: A device for attaching and removing a ditch cover comprises a pair of parallel levers 11 and 11, an operating handle equipped with a handle lever 12 for connecting and fixing the parallel levers on the upper ends of them and pushing sections 13 provided on the lower ends of the parallel levers, horizontal shafts 21 passing through a pair of parallel levers to provide, and contact sections 25 formed by bending the lower ends of plate bodies 24 vertically hung to the horizontal shafts 25 in a roughly L-shape. Tools 1a and 1b are used in groups of two persons, and a ditch cover is held from both sides by making use of a notched space 102 of the ditch cover 100 with the pushing section 13 and contact sections 25 to attach or remove it.
Patent JP-H01272217-A (JP)
Title: Comb line filter
Inventor: SHINGU YUJI
IPC: H03H9/36
Filed: 1988-04-22
Abstract: PURPOSE:To trim a square chip resistance by a laser after assembling by connecting the square chip resistance across first and second partial patterns and allowing the square chip resistance to face the outside in the assembled state. CONSTITUTION:A storage case 13 is attached which is detained on a printed board 7 so that first - third terminals 11a-11c are projected, and a square chip resistance 14 as the impedance element between the input and the output is connected to first and second partial patterns 9a and 9b. The attached square chip resistance 14 is trimmed from the other surface of the board 7 by the laser to set the resistance value so that the extent of attenuation is maximum, and the filter capacity is considerably improved.
Patent JP-S59226370-A (JP)
Title: Cleaning device
Inventor: SHIODA KEISAKU
IPC: G03G21/00
Filed: 1983-06-06
Abstract: PURPOSE:To prevent the surface of a photosensitive body from being made into a mat to extend the life of the photosensitive body by providing a means which not only runs a web of a cleaning unit in the direction opposite to the rotation direction of the photosensitive body but also moves it back and forth in the axial direction. CONSTITUTION:Simultaneously with the start of rotation of a photosensitive body 1, a web driving motor 11 rotates and drives a pressure roll 4 and a winding roll 7 through a chain 12. Then, a web 6 for polishing and cleaning is carried in the direction opposite to the rotaion direction of the photosensitive body 1 and is wound up by the winding roll 7. Simultaneously, a driving motor 13 is rotated to drive a crank 8. Therefore, a hole 9a in one end of a rod 9 si moved back and forth, and a web cleaning unit 10 is moved back and forth in the axial direction of the photosensitive body 1 to polish and clean the photosensitive body 1 in the axial direction. Thus, the surface of the photosensitive body is prevented from being made into a mat, and the life of the photosensitive body is extended.
Patent JP-H09248979-A (JP)
Title: Method and apparatus for giving folding tendency of saddle stitching folding
Inventor: HORI HACHIRO
IPC: B42C13/00
Filed: 1996-03-14
Abstract: PROBLEM TO BE SOLVED: To provide a method and apparatus for giving the folding tendency of saddle stitching folding capable of sufficiently giving folding tendency by pressing a folding portion of a sheet of paper folded for saddle stitching In a short period of time. SOLUTION: A sheet of paper 3 folded into saddle stitching state is hit against a pair of rollers 82, 83 in a state of its interstice between the front and rear surfaces pressed by a conveyor 80, thereby giving impacts to the rear surface in the proximity of the stitching position, after that, giving a press treatment in turn from the rear of the stitching position by means of the press rollers 82, 83, whereupon the folding tendency of the saddle stitching folding is stiffened.
Patent JP-S5741274-A (JP)
Title: Sheet for bicycle
Inventor: JIYOORU EE BAAKAA
IPC: B62J1/00
Filed: 1981-06-30
Abstract: A bicycle seat according to the invention provides additional comfort for the rider. The seat (9) is made in two portions (10,11) which are mounted on a horizontal mounting member (15) so that they can be moved horizontally and will also have a limited rotational movement round the axis of the member (15). The shape of the top surface of the portions (10,11) is chosen to conform as much as possible to the shape of the human skeleton in the region of the ischium and upper femur. That of the top surface of the portion (11) is shown by graphs in Figures 8-10 of the drawings, and should not deviate by more than 20%. The shape of the portion (10) is a minor image of that of the portion (11).
Patent JP-H01272760-A (JP)
Title: Usage of ceramic heater
Inventor: MATSUDA KOICHI
IPC: C23C14/24
Filed: 1988-04-23
Abstract: PURPOSE:To prevent the overheating of a ceramic heater when Al is vacuum- deposited by a batch process with the heater, by suspending the impression of voltage and calculating voltage to be impressed next time every time the evaporation of Al is finished. CONSTITUTION:When Al is vacuum-deposited by a batch process with a ceramic heater, every time the evaporation of Al is finished, electric current is measured and immediately the impression of voltage is suspended. Voltage to be impressed next time is then calculated on the basis of the measured electric current. This voltage is impressed next time and Al is vacuum-deposited. The shortening of the service life of the heater due to overheating is prevented.
Patent JP-H09288402-A (JP)
Title: Electrophotographic electrifying device
Inventor: ARATAIRA FUMIHIRO
IPC: G03G15/02
Filed: 1996-04-23
Abstract: PROBLEM TO BE SOLVED: To provide an electrophotographic electrifying device in which good electrification characteristics can be maintained for a long time and injection of charges can be performed in a good state. SOLUTION: This electrophotographic electrifying device is equipped with an electrophotographic photoreceptor and an electrifying member disposed in contact with the electrophotographic photoreceptor. By applying voltage on the electrifying member, the electrophotographic photoreceptor is charged. The volume resistance of the photoreceptor is specified to >=1×10<8> Ωcm. The electrifying member has magnetic particles containing 0.05 to 1.2wt.% silicon component. The volume resistance of the magnetic particles is controlled to >=1×10<4> Ωcm and <=1×10<11> Ωcm.
Patent JP-S60244371-A (JP)
Title: Structure of paint outflow part of paint coating brush of painting apparatus with paint coating brush
Inventor: TANADA KATSUNORI
IPC: B05C17/01
Filed: 1984-05-18
Abstract: PURPOSE:To easily and uniformly supply a paint to a brush part, in an apparatus wherein a coating brush is provided to the leading end of the hose connected to the paint feed pump in a paint container, by providing a paint outflow part to the interior or side surface part of the brush. CONSTITUTION:A hose 4 is connected to the pump 2, which is driven by a battery 1 and provided in a paint container 3, and an electric wire 5 is provided to the outer peripheral surface of said hose 4 along the longitudinal direction thereof. One end of an electric wire 5 is connected to a pump driving motor and the other end thereof to the switch 8 provided to a grip pipe 7 mentioned hereinbelow. A chuck pipe 6 is provided to the leading end part of the hose 4 and connected to the pipe 7 while a brush 9 is attached to the leading end of the pipe 7 in a freely detachable manner and a paint outflow part 10 is arranged in the brush 9. Then, the part of the brush 9 connected to the leading end part of the pipe 7 is formed into a flat cylindrical shape from flexible rubber and the leading end part thereof is opened as a paint outflow part and the outlet part of the open end of the pipe 7 is provided so as to be widely opened from the flat base part of the brush 9 toward the intermediate part thereof. This widely opened part is provided so as to be extended toward the leading end of the brush.
Patent JP-S5529254-A (JP)
Title: Sliding contact surface of mechanical seal for submerged motor
Inventor: TSUJIMOTO HARUO
IPC: H02K5/132
Filed: 1978-08-19
Abstract: PURPOSE: To raise the durability of a mechanical seal, by providing a rotary slide ring with a large-diameter part and setting the slide ring in contact with a fixed ring so that intermittent contact surfaces are formed on the contact sides of these rings and communicate with an oil chamber.  
     CONSTITUTION: The fixed ring 6 is provided on an annular support 4 which is fixed in a wall 5 and movably fitted on a motor shaft 1 extending from an oil chamber 3 to a shaft box 2. The rotary slide ring 7 is provided on a rotary annular support 8 mounted on the motor shaft 1. The sides 6a, 7a of both the rings are set in contact with each other by a spring 9. The rotary slide ring 7 is provided with the large-diameter part R2 so that the intermittent contact surfaces 10 are formed on the sides of the rings and communicate with the oil chamber 3. Oil is thus automatically supplied to the sliding sides of the rings 6, 7. This results in maintaining good lubrication and greatly raising the durability of the mechanical seal. 
     COPYRIGHT: (C)1980,JPO&Japio
Patent JP-S5326832-A (JP)
Title: Coating plastic compositions their preparation and applications
Inventor: KOSABE TORAICHI
IPC: C09D5/00
Filed: 1976-08-25
Abstract: PURPOSE: A coating composition capable of forming protective films having improved hardness, wear resistance, etc.  on molded plastic articles, comprising a hydrolyzed tetraalkoxysilane, a hydrolyzed silicon compound and polyvinyl acetate resin. 
     COPYRIGHT: (C)1978,JPO&Japio
Patent JP-H07312649-A (JP)
Title: Data collector
Inventor: ISHIKAWA KEIICHI
IPC: H04B3/54
Filed: 1994-05-16
Abstract: PURPOSE:To provide a data collector capable of easily and efficiently collecting of data or the like without manual aid. CONSTITUTION:Plural terminals 20-1-20-n for sampling and holding the information of measuring instruments every prescribed time are respectively connected to plural measuring instruments 10-1-10-n for measuring information to be changed with time, the sampling data held in the plural terminals are collected through a power line 30 by a power line communication equipment 40, and the collected data are transmitted through a public line to a remote control device 60 by a public line communication equipment 50.
Patent JP-H0841754-A (JP)
Title: Weft inserting method and picking motion in warp opening series arranged loom
Inventor: ROBERUTO BUTSUHAA
IPC: D03D41/00
Filed: 1995-04-25
Abstract: PURPOSE: To surely carry out weft insertion into a weaving rotor of a warp yarn series shed weaving machine. CONSTITUTION: Four weft yarns 7; 71-74 are conveyed from four weft yarn supply units 2a-2d and four metering apparatuses 1a-1d into a weft yarn distribution apparatus 9 which distributes the weft yarns 71-74 delivered thereto to sheds 103a-103d of a weaving rotor 100 and the weft yarns 71-74 are then inserted through stationary fluid nozzles 91-94 into the rotating weaving rotor 100. During normal operation of the warp yarn series shed weaving machine the weft yarns 71-74 are continuously pulled from the weft yarn supply units 2a-2d by the metering apparatuses 1a-1d and conveyed to the weft yarn distribution apparatus 9 which conducts the weft yarns 71-74 into open sheds 103a-103d. The speed of conveyance of the weft yarns 71-74 during the insertion into the sheds 103a-103d is thus determined by the metering apparatuses 1a-1d.
Patent JP-S6069184-A (JP)
Title: Anaerobic microbe-based soil conditioner
Inventor: KOBAYASHI CHIAKI
IPC: A01G1/00
Filed: 1983-06-07
Abstract: PURPOSE:To promote formation of lumps and granules of soil, supply humus of good quality and maintain well-balanced oxidation and reduction in soil, by inoculating an organic substance with a useful anaerobic microbe for selective propagation of the microbe and fixation of decomposition product and microbe in clayey mineral particles. CONSTITUTION:An organic substance consisting of sugar, protein, cellulose, lignin, etc. is inoculated with a useful anaerobic soil microbe which effectively decomposes the above components, to effect propagation of the microbe under anaerobic conditions and decomposition of the organic substance into humus of good quality. The resultant decomposition product and the microbe are mixed with a clayey mineral of good quality so that the microbe may be adsorbed by the mineral for fixation and a soil conditioner consisting mainly of clay, humus and microbe may be formed. Preferred clayey mineral is montmorillonite which has a high base exchange volume and a high swellability.