baber/WOPTO huggingface dataset:
Patent EA-002547-B1 (EA)
Title: Selective epoxidation process for preparing pharmaceutical compounds
Inventor: HOARD DAVID W
IPC: C07D303/40
Filed: 1998-02-25
Abstract: 1. A process for preparing a compound of the formula   wherein G is phenyl, optionally subsitituted with substituent, selected form the group, comprising halo and C1-C6 alkyl; R<3> is C1-C6-alkyl; R<4> and R<5>, taken together form a second bond between C-13 and C-14; R<83> is hydrogen, C1-C6-alkyl, trichloroethyl, or -CH2SR<81>; R<30>' is hydrogen, protecting group for alcohol or the group of formula   R<7> and R<8> are each independently hydrogen or C1-C6 alkyl; or R<7> and R<8> taken together form a cyclopropyl or cyclobutyl ring; R<10> is C1-C6 alkyl; R<50> is (=O); R<6> is halogenC1-C6 alkoxyphenyl; R<81> is C1-C6 -alkyl, and R<82> is a base labile protecting group; or a pharmaceutically acceptable salt thereof; with proviso that when R<83> is -CH2SR<81>, R<30> is not a hydrogen or a protecting group for alcohol, comprising epoxidation of the compound of formula   wherein G, R<3>, R<4>, R<5>, R<6>, R<30>, and R<83> are as defined above; oxidant and chiral ketone with forming the compound of formula (II); and optionally forming a pharmaceutically acceptable salt thereof. 2. A process according to Claim 1 wherein G is phenyl, para-fluorophenyl, R<30>' is hydrogen. 3. A process according to Claim 1 wherein said oxidant is oxone and the compound of formula   is a chiral ketone. 4. A process according to Claim 2 wherein G is phenyl and R<83> is trichloroethyl. 5. A process according to Claim 1 wherein said compound of formula (II) is represented by the formula   6. A compound of the formula   wherein G is phenyl, optionally substituted halo and C1-C6 alkyl; R<3> is C1-C6 alkyl; R<4> and R<5> taken together form a second bond between C-13 and C-14; R<6> is halogenC1-C6 alkoxyphenyl; or a pharmaceutically acceptable salt thereof. 7. A compound according to Claim 6 wherein G is phenyl, para-fluorophenyl. 8. A compound according to Claim 6, which is represented by formula   9. A compound of formula   wherein G is phenyl, optionally subsitituted with substituent, selected form the group, comprising halo and C1-C6 alkyl; R<3> is C1-C6-alkyl; R<4> and R<5>, taken together form a second bond between C-13 and C-14; R<7> and R<8> are each independently hydrogen or C1-C6 alkyl; or R<7> and R<8> taken together form a cyclopropyl or cyclobutyl ring; R<10> is C1-C6 alkyl; R<50> is (=O); R<6> is halogenC1-C6 alkoxyphenyl; R<82> is a base labile protecting group; or a pharmaceutically acceptable salt thereof; 10. A compound according to Claim 9 wherein G is phenyl, parafluorophenyl. 11. A compound according to Claim 9, which is represented by formula   12. A compound according to Claim 9, which is represented by formula
Patent EA-005787-B1 (EA)
Title: Ceramic filtering element and method for production thereof
Inventor: KRASNY BORIS LAZAREVICH
IPC: B01D33/23
Filed: 2002-11-26
Abstract: The invention relates to filtering devices, in particular to the structural design of the filtering elements of disc ceramic filters and to methods for the production thereof. In order to increase the performance and the strength of a device, the inventive ceramic filtering element comprises a hollow block made of porous ceramic material whose inside elements are arranged in rows and offset along the arcs of a concentric circle and form with walls (4) a hollow volume (3). The ratio of the radius of the transition line between walls inside the hollow block (1) in the bottom part (6) of a sector element with respect to the radius of said interface line in the top part thereof rages from 0.5 to 0.75. An outlet fitting (7) is connected to the hollow block (1) with the aid of a screw joint provided with a seal (8). The inventive method for producing a ceramic filtering element consists in producing the replication thereof of a mixture of paraffin hydrocarbons, forming a porous blank by compaction and using vibration load, and, in order to protect environment, in removing the material of said replication at a temperature below the inflammability point of paraffin hydrocarbons.
Patent EA-009605-B1 (EA)
Title: Method for characterising polynucleotides
Inventor: LEXOW PREBEN
IPC: C12Q1/6874
Filed: 2004-04-16
Abstract: The method of the invention is used to identify specific characteristics of a target polynucleotide in a sample, and comprises the steps of: i) attaching to one end of each target polynucleotide in the sample a polynucleotide signal sequence that is specific for the characteristic under study; ii) contacting the target polynucleotides with a molecule that interacts with the target polynucleotide if the characteristic is present; iii) attaching a polynucleotide adapter sequence to those targets polynucleotides that interact with the molecule of step (ii), the adapter being attached at the end of the target polynucleotide opposite that at which the signal sequence is attached; iv) carrying out a polynucleotide amplification reaction on those target polynucleotides that comprise both the adapter and signal sequence, optionally repeating steps (i) to (iv) for other characteristics; and (v) identifying which signal sequences are present on the amplified products, and in which order, to thereby determine the characteristics of each target polynucleotide.
Patent EA-011230-B1 (EA)
Title: Optically active carboxamides and use thereof to combat undesirable microorganisms
Inventor: DUNKEL RALF
IPC: C07D207/34
Filed: 2004-12-06
Abstract: Novel optically active carboxamides of formula (1)wherein R, M and A have the meanings cited in the description.There described several methods for the production of said substances and the use thereof to combat undesirable microorganisms, in addition to novel intermediate products and the production thereof.
Patent EA-013447-B1 (EA)
Title: Apparatus for adjusting an electrode for a metallurgical furnace
Inventor: KUMMER KARL-HEINZ
IPC: H05B7/10
Filed: 2006-12-07
Abstract: In an apparatus (1) for adjusting an electrode (5) of a metallurgical furnace, in particular a furnace for resistance operation having a furnace lid (15), comprising a clamping ring (3) and a holder ring (4, 14), the holder ring (4, 14) is designed to be arranged in the furnace lid (15).
Patent EA-017321-B1 (EA)
Title: N,n-dibemzyl-2-aminopyrimidine derivatives and medicine comprising them
Inventor: OHGIYA TADAAKI
IPC: A61K31/505
Filed: 2008-04-10
Abstract: This invention provides a compound represented by general formula (I) having a high level of inhibitory activity against a cholesterol ester transfer protein (CETP)wherein R, R, R, Rand Rrepresent a hydrogen atom, and represent hydrogen atom, a halo(C-Calkyl) group, or cyano group, Rrepresents a C-Calkyl group, R, R, Rand Rare the same or different, and represent hydrogen atom, a halogen atom, a C-Calkyl group, a halo(C-Calkyl) group, or a C-Calkoxy group, Rand Rare the same or different, and represent a C-Calkyl group, or a (C-Ccycloalkyl)(C-Calkyl) group (this (C-Ccycloalkyl)(C-Calkyl) group may have one hydroxycarbonyl(C-Calkyl) group or (C-Calkoxy)carbonyl(C-Calkyl) group as a substituent on the cycloalkyl group), or Rand Rcombine to form morpholino group or piperidino group together with the adjacent nitrogen atom (the morpholino group or the piperidino group may have 1 or 2 of C-Calkyl groups as a substituent), and Rrepresents a (C-Calkyl)thio(C-Calkoxy) group, a (C-Calkyl)sulfinyl(C-Calkoxy) group, or a (C-Calkyl)sulfonyl(C-Calkoxy) group.
Patent EA-022472-B1 (EA)
Title: Telomerase activating compounds and methods of use thereof
Inventor: GAZIT AVIV
IPC: A01N43/04
Filed: 2008-06-04
Abstract: The present invention is directed to the use of compounds of formula I wherein R-R, Z are disclosed in the claims and compositions comprising the same for stimulating or increasing telomerase expression, activity or a combination thereof in a cell or tissue in a subject having a disease mediated by telomerase expression/activation or a combination thereof.
Patent EA-016067-B1 (EA)
Title: Fungicidal mixtures of triticonazole and difenoconazole
Inventor: LINDHOLM DON CRAIG
IPC: A01N43/653
Filed: 2008-09-10
Abstract: Fungicidal mixtures comprising, as active components: 1) triticonazole of Formula (I)and 2) difenoconazole of Formula (II)in a synergistically effective amount, and also compositions comprising these mixtures.
Patent EA-018288-B1 (EA)
Title: Base station device, mobile station device, wireless communication system and wireless communication method
Inventor: HAMAGUCHI YASUHIRO
IPC: H04J1/00
Filed: 2008-11-26
Abstract: A wireless transmission device converts signals having been subjected to a first modulation into frequency domain signals, and allocates the frequency domain signals converted to subcarriers for transmission. The wireless transmission device includes: a controller that selects, based on channel qualities of the subcarriers to which the frequency domain signals are allocated, a value satisfying a predetermined communication quality as control information indicative of the number of frequency domain signals included in each of segments into which the frequency domain signals are segmentalized; and an allocating unit that segmentalizes the frequency domain signals into segments, each of the segments including the same number of frequency domain signals as the value selected as the control information by the controller, and allocates the frequency domain signals included in each of the segments to sequential subcarriers.
Patent EA-019534-B1 (EA)
Title: 3-(3-PYRIMIDIN-2-YLBENZYL)-1,2,4-TRIAZOLO[4,3-b]PYRIDAZINE DERIVATIVES AS Met KINASE INHIBITORS
Inventor: DORSCH DIETER
IPC: A61K31/5025
Filed: 2009-05-25
Abstract: The invention relates to compounds of the formula (I) in which R, R, R, R', Rare each as defined herein which are inhibitors of tyrosine kinases, especially of Met kinase, and can be used for treatment of neoplasms.
Patent EA-029354-B1 (EA)
Title: Preparation of caprolactam from 6-amino caproic acid obtained in a fermentation process
Inventor: GUIT RUDOLF PHILIPPUS MARIA
IPC: C07D223/10
Filed: 2010-12-22
Abstract: The present invention relates to a method for preparing caprolactam comprising recovering a mixture containing 6-aminocaproic acid, from a culture medium comprising biomass, and thereafter cyclising the 6-aminocaproic acid in the presence of superheated steam, thereby forming caprolactam, wherein the weight to weight ratio carbohydrate to 6-aminocaproic acid in said mixture is 0.03 or less.
Patent EA-021127-B1 (EA)
Title: Method of cutting fragile nonmetallic materials
Inventor: KONDRATENKO VLADIMIR STEPANOVICH
IPC: B23K26/402
Filed: 2012-10-08
Abstract: The invention relates to the methods of cutting fragile nonmetallic materials, in particular quartz glass and other fragile heat-resistance materials. The technical result provides expanded possibilities of a method of cutting fragile nonmetallic materials due to application of LUT cutting method for cutting quartz glass and other fragile heat-resistance materials. The assigned task is solved by that the known method of cutting fragile nonmetallic materials comprising making a local notch at workpiece edge in cutting line, heating the latter by laser beam and subsequent cooling it by coolant at relative displacement of material and laser beam with coolant, for cutting quartz glass and other heat-resistance materials workpiece is heated by laser beam before making a local notch and the local notch is made in laser beam zone or immediately behind it, wherein the notch is made at relative displacement of workpiece at the rate v with time delay with respect to beginning of heating t by laser beam defined by equation t=Ak/v, where A is half of the elliptic beam in direction of displacement or round beam radius, k varies from 1 to 2.5.
Patent EA-023810-B1 (EA)
Title: Wearing article
Inventor: TAKINO SHUNSUKE
IPC: A61F13/49
Filed: 2008-09-03
Abstract: The aim of the present invention is to provide an improved wearing article which is not easily torn and makes it possible to see the skin of an article wearer through. The wearing article includes a belt member 4 constituting front and back waist areas and a liquid absorbing structure 5 constituting a crotch area, wherein the belt member 4 is provided with a waist side opening edge 19 comprising two segments of the front and back waist areas separately facing the anteroposterior direction Y. The front and back belt parts 6 and 7 of the belt member 4 include see-through possible areas where all light beam transmissivity is 55% or more in the front and back waist areas 1 and 2 and the skin of the article wearer is seen through, the see-through possible areas occupy 40% or more of the front and back waist areas 1 and 2. A reinforcing elastic member 35 to the front and back belt members 6 and 7 is attached in the width direction X along the waist side opening edge 19.
Patent EA-028180-B1 (EA)
Title: Multi filter lubricant purification system
Inventor: JACOBS WILLIAM A
IPC: F01M11/03
Filed: 2011-03-22
Abstract: A lubricant reclamation configuration includes a series of fluid inlets that distribute the fluid to a series of parallel arrangement of individual filter assemblies. A filter control valve assembly is assembled between the distribution manifold and each respective filter assembly individually controlling fluid flow between the distribution manifold and each respective filter assembly. The filter assembly processes the fluid, after which the processed fluid is collected and retuned to the system via a series of collection channels. The distribution manifold is preferably fabricated of a series of plates.
Patent EA-026196-B1 (EA)
Title: Biomass torrefaction system and method
Inventor: TEAL WILLIAM B
IPC: F27B7/16
Filed: 2011-10-06
Abstract: A biomass torrefaction system is provided which enables a continuous torrefaction process that involves the introduction of biomass particles into a rotating reactor drum having a low oxygen environment. The particles are conveyed through the drum by a heated gas stream and simultaneously torrefied thereby. Gas exiting the drum is recirculated back to a heat source for reheating the gas prior to reentering the drum. A method of biomass torrefaction is also provided.
Patent EA-034462-B1 (EA)
Title: Anti-clusterin antibodies and antigen binding fragments and their use to reduce tumor volume
Inventor: TREMBLAY GILLES BERNARD
IPC: C07K14/775
Filed: 2010-11-24
Abstract: Novel antibodies and antigen binding fragments that specifically bind to clusterin are described. In some embodiments, the antibodies block the biological activity of clusterin and are useful in composition in certain cancers, more particularly in cancers, such as endometrial carcinoma, breast carcinoma, hepatocellular carcinoma, prostate carcinoma, a renal cell carcinoma, ovarian carcinoma, pancreatic carcinoma, and colorectal carcinoma. The invention also relates to cells expressing the humanized or hybrid antibodies. Additionally, methods of detecting and treating cancer using the antibodies and fragments thereof are also disclosed.
Patent EA-027223-B1 (EA)
Title: Process and apparatus for winning oil from a vapor gas mixture
Inventor: SIEGER HERMANN
IPC: B03C3/00
Filed: 2012-10-10
Abstract: In a process for winning oil from a vapor gas mixture (VGM) obtained by the pyrolysis of a hydrocarbon containing material, such as oil shale, the VGM containing several oil fractions is dedusted and the oil fractions are separated based on their condensation temperature. To separate the desired oil fractions contained in the vapor gas mixture the dedusted VGM is cooled and subsequently fractionated in at least two electrostatic precipitator stages at a temperature adapted to the boiling point of the respective oil fraction to be separated.
Patent EA-029526-B1 (EA)
Title: Process for producing crustless sandwich bread
Inventor: MAUCOTEL THIERRY
IPC: A21D13/00
Filed: 2014-07-03
Abstract: The invention provides a process for producing crustless sandwich bread, which comprises the following steps: depositing semifinished products of a sandwich bread dough in moulds, oven-baking these semifinished products, obtaining corresponding loaves of sandwich bread, cooling the loaves of sandwich bread and removing the crust from all the sides thereof, the oven-baking step being performed in an oven at a temperature of 145-175°C for a time period comprised between 50 and 70 minutes.
Patent EA-029641-B1 (EA)
Title: Integrated circuit metallization
Inventor: NALIVAJKO OLEG YURIEVICH
IPC: H01L23/48
Filed: 2015-02-04
Abstract: The invention is related to the field of microelectronics, in particular, to submicron integrated circuit manufacture technology. The invention is based on solution of the problem of improving the passivation coating quality and increasing the yield of metallization structures in ICs of submicron design standards. The essence of the invention is in provision of metallization of an integrated circuit comprising active and passive components formed on the surface of a semiconductor plate, a pattern of current-conductive material with contact pads for connection of external terminals, a silicon oxide layer, and a passivating silicon nitride layer, wherein the silicon oxide layer is made in the form of near-wall spacers on side surfaces of the current-conductive material, and the passivating silicon nitride layer has a thickness of 0.8-1.2 μm.
Patent EA-032974-B1 (EA)
Title: Massage portable mat
Inventor: GALLAGHER ALI
IPC: A61H7/00
Filed: 2013-11-15
Abstract: A device or system useful for temporarily reducing the appearance of cellulite and increasing local circulation, including a base with an array of protrusions having a size, shape, durometer and spacing selected to indent a user's skin under pressure. A user may position the device such that the protrusions are in contact with skin or separated from the skin by thin fabric, and then apply pressure to cause the protrusions to indent but not penetrate the skin.
Patent EA-030768-B1 (EA)
Title: System for dispensing active agents to agricultural or forestry products
Inventor: EUBELER JAN
IPC: B26F1/26
Filed: 2014-09-13
Abstract: Claimed is a system for dispensing active agents to agricultural or forestry products, said system comprising an adhesive layer (11) that contains at least one active agent (12), adheres to a surface (23) and connects a covering layer (13) to this surface (23), wherein the covering layer (13) has a plurality of openings (14) for dispensing the active agent (12), is perforated with vacuum and has bulges (15) protruding by a height (17) from a plane (16) of the covering layer (13) and forming said openings (14).
Patent EA-038112-B1 (EA)
Title: Novel compounds and therapeutic uses thereof
Inventor: GLOSSOP MELANIE
IPC: A61K47/64
Filed: 2017-09-13
Abstract: The invention relates to novel compounds with the ability to link an immune response to a pathogen, to the use of said compounds in a disease or disorder mediated and/or caused by an infective agent, to compositions containing said compounds, processes for their preparation and to novel intermediates used in said process.
Patent EA-039159-B1 (EA)
Title: Flotation machine apparatus and method of using the same
Inventor: WALKER MATHEW
Filed: 2019-03-22
Abstract: Described herein is a flotation machine including a wash water system that is connectable adjacent a tank to direct sprays of water into froth within a froth zone. Wash water panel assemblies of the system can be positioned adjacent the tank so that each of the wash water panel assemblies are moveable between an open position and a closed position. Each wash water panel assembly can include an outer panel body that at least partially defines a reservoir in which wash water is passable and a spray membrane positionable adjacent the outer panel body. The spray membrane can have a plurality of spray holes in fluid communication with the reservoir such that water is passable from the reservoir and through the spray membrane via the spray holes for spraying water into the froth in the froth zone.
Patent ES-2193833-B1 (ES)
Title: Anilla embellecedora para cortinas.
Inventor: TERRADAS RIULAS ISIDOR
IPC: A47H13/02
Filed: 2001-04-10
Granted: 2005-02-16
Abstract: Anilla embellecedora para cortinas. La anilla está prevista para su aplicación sobre cada uno de los orificios que se realizan en una cortina (7) para el colgado de ésta respecto de una barra, constituyendo no solamente el medio de suspensión sino un medio embellecedor que además facilita el deslizamiento de la cortina a través de la barra. Dicha anilla la forman dos cuerpos anulares (1 y 2) que se acoplan entre sí, contando el cuerpo (1) con un cuello (3) que en su superficie externa cuenta con nervios (4), mientras que el cuerpo (2) presenta una sección en "U" cuya rama interna (2'') está afectada de rebajes (5) complementarios de resaltes (4) para determinar entre ambos el medio de retención entre sí, cuando se acopla por deslizamiento un cuerpo sobre el otro, quedando entre ambos retenida la cortina (7), ya que dichos cuerpos quedan a uno y otro lado de la propia cortina.
Patent ES-2196951-B1 (ES)
Title: Encofrado recuperable.
Inventor: UBINANA FELIX JOSE LUIS
IPC: E04G11/38
Filed: 2001-04-18
Granted: 2004-10-16
Abstract: Encofrado recuperable. El encofrado presenta paneles de encofrado dotados de rebordes laterales, susceptibles de quedar retenidos en rebordes de retención de las vigas de soporte de los paneles, las cuales quedan apoyadas en cabezales desplazables verticalmente sobre los extremos de pies derechos ajustables, entre una posición alta de encofrado y una posición más baja de desmontaje de los paneles, en la que se posibilita el levantamiento de los mismos por un lado, previo a su traslación lateral, liberando una de las vigas de soporte y permitiendo la basculación del panel para su retención en suspensión o para su desmontaje.
Patent ES-2216651-B1 (ES)
Title: Compacto de tono metalico y metodo de formacion del mismo.
Inventor: OHTSUKA YOSHIAKI
IPC: C08K3/40
Filed: 2001-05-23
Granted: 2005-12-16
Abstract: Compacto de tono metálico y método de formación del mismo. Cuando se forma un compacto de tono metálico de resina, que está coloreado en un tono metálico mezclando una matriz de resina con un material que proporciona aspecto metálico (1), se utiliza un polvo de vidrio de alta luminosidad (2), alrededor del cual se forma una capa de revestimiento de resina (3) con una temperatura de fusión más alta que la matriz de resina, como material que proporciona aspecto metálico.
Patent ES-2204274-B1 (ES)
Title: Method for modification of trajectory of fluid eliminates mixed or dissolves substances and generates energy
Inventor: DORADO GONZALEZ MANUEL
IPC: B01D17/06
Filed: 2002-02-21
Granted: 2005-03-01
Abstract: The method for modification of the trajectory of a fluid eliminates mixed or dissolves substances and generates energy. A unit is formed by a deposit containing fluid which has an electric or magnetic dipolar moment and causes the deviation of the fluid. It has collector deposits of the outgoing fluid and the rest of the components. - The fluid is canalized towards the entry to the unit. Whilst it crosses the unit, the flow of fluid is deviated in its trajectory. In this deviation, the various substances accompanying the fluid are separated as the result of following different trajectories.