baber/WOPTO huggingface dataset:
Patent FI-954750-A0 (FI)
Inventor: GARCIA HERVE
IPC: C07D471/04
Filed: 1995-10-05
Abstract: PCT No. PCT/US94/11832 Sec. 371 Date Jun. 7, 1995 Sec. 102(e) Date Jun. 7, 1995 PCT Filed Oct. 20, 1994 PCT Pub. No. WO94/24113 PCT Pub. Date Oct. 27, 1994Method of preparation of 6-fluoro-2-halogen quinoline of general formula (I) wherein R is a hydrogen atom or an alkyl radical and Hal and Hal' are identical or different halogen atoms. The invention is characterized in that a halogenating agent is made to act on hydroxy-1 quinoline of general formula (II) wherein Hal is defined as above and R1 is defined as R excepting a hydrogen atom, the acid function being optionally released if a 6-fluoro-2-halogen quinoline is to be obtained for which R is a hydrogen atom.
Patent FI-964002-A0 (FI)
Inventor: BASTART JEAN-PIERRE
IPC: C07F7/18
Filed: 1996-10-04
Abstract: PCT No. PCT/FR95/00420 Sec. 371 Date Oct. 3, 1996 Sec. 102(e) Date Oct. 3, 1996 PCT Filed Apr. 3, 1995 PCT Pub. No. WO95/26961 PCT Pub. Date Oct. 12, 1995This invention relates to a process for the preparation of 7-hydroxy taxanes of general formula (I) from 7-trialkylsilyl taxanes of general formula (II), wherein R1 is hydrogen, alkoxy, acyloxy, or alkoxyacetoxy, and Z is a hydrogen atom or a radical of general formula (III), wherein R2 is an optionally substituted benzyl radical or an R'2-O-CO- radical wherein R'2 is an alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, bicycloalkyl, optionally substituted phenyl or heterocyclyl radical, R3 is an aromatic alkyl, alkenyl, alkynyl, cycloalyl, phenyl, naphthyl or heterocyclyl radical and either R4 is a hydrogen atom and R5 is a hydroxyl function protecting group, or R4 and R5 together form a saturated 5- or 6-membered heterocylic ring. In general formula (II), each R, which are the same or different, is an alkyl radical optionally substituted by a phenyl radical.    <IMAGE>  (I)   <IMAGE>  (II)   <IMAGE>  (III)
Patent FI-971583-A0 (FI)
Inventor: MALCOLM PETER BRYAN
IPC: G06F21/12
Filed: 1997-04-15
Abstract: In an improved method for accessing files in a computer system, file open requests are intercepted at the level of the operating system. The identity of the file to be opened is extracted from the request and a determination is made as to whether the identity of the requested file should be replaced with the identity of a substitute file to be opened instead of the requested file. If it is determined that the identity should be so replaced, the file open request is amended by substituting the identity of the substitute file for the identity of the requested file, and the request is passed on to its original destination for execution. This technique can be used to cause execution of a substitute program without the knowledge of the user. As an example, software metering can be implemented in a network system by substituting a different program from that requested when the number of copies of the requested program in use on the network has reached the maximum licensed number, so as to provide a user-friendly rejection of the program execution request.
Patent FI-973879-A0 (FI)
Inventor: CHAN MING FAI
IPC: A61K31/381
Filed: 1997-10-03
Abstract: Biphenylsufonamides of the following formula and methods for modulating or altering the activity of the endothelin family of peptides are provided. The sulfonamides may be used for inhibiting the binding of an endothelin peptide to an endothelin receptor by contacting the receptor with the sulfonamide <CHEM> or a pharmaceutically acceptable salt, acid or ester thereof, wherein Ar<2> is <CHEM> and wherein Ar<1>, R<13> and R<26> are as defined herein.m
Patent IL-83618-A0 (IL)
Title: Procedure for incorporating timing parameters in the synthesis of logic circuit design
IPC: G06F17/50
Filed: 1987-08-23
Abstract: During the synthesis of a logic circuit in which a plurality circuit components are examined and, in the presence of certain criteria, are changed in accordance with preestablished rules, timing parameters are estimated for selected circuit locations. Forward timing delays are determined by adding the timing delays associated with the intervening circuit components and media paths between an input terminal or latch component output terminals and a successive locations on the signal path. Similarly, a derived budget timing delay constant is calculated by designating a budget or design delay at any location in the circuit and by subtracting timing delays asssociated with the intervening components between that location and the previous location along the signal path in the reverse direction. The derived budget timing delay constant is substracted from the forward timing delay at each selected location to derive a timing debt for each selected location. The timing debt can be used as a criterion to determine when the implementation of circuit component should be changed. The timing information is stored in data structures associated with terminals of components and can include data with respect to a multiplicity of designated paths for complex circuits for which examination of all signal paths requires a prohibitive amount of time, the technique can be used between groups of latches that are activated by timing signals having known signal delays. The resulting timing data can be derived and stored for all latch (input signal and output signal) paths affecting each selected location.
Patent IL-85488-A0 (IL)
Title: Thermodynamic printing method and means
IPC: G03G15/32
Filed: 1988-02-22
Abstract: In a method of printing on a printing medium (S) a variable thickness ink dot pattern representing an original image in response to an incoming digital data stream, a printing member, e.g. a cylinder (72), is formed which defines a multiplicity of discrete, independently electrically chargable capacitor microcells (94) adjacent to a printing surface of that member. Selected ones of the microcells (94) are activated in accordance with the incoming data stream so that the activated microcells are geometrically related to the dots in the pattern to be printed. Then, electrical charges are deposited on the microcells (94) selected for activation at controlled variable coulombic charge levels to create at the printing surface localized electrical fields of various strengths that are proportional to the print densities desired for the related dots in the pattern to be printed. Following this, the printing surface is contacted by a two-component, voltage sensitive, thermoplastic whereby the ink, under the influence of the fields, is deposited on the printing surface only at the locations of the microcells selected for activation, with the thickness of each ink deposit being proportional to the strength of the field at that microcell, thereby to form a variable-thickness ink pattern on the printing surface. That ink pattern is then transferred completely to the printing medium to provide a faithful hardcopy reproduction of the original image. Apparatus for practicing the method are also disclosed.
Patent IL-86169-A0 (IL)
Title: Substituted quinoxalyl-imidazolidine-2,4-diones,processes for their preparation and pharmaceutical compositions containing them
IPC: C07D403/04
Filed: 1988-04-25
Abstract: 5-Quinoxalylimidazolidine-2,4-diones of the formula I 
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 in which R<1>, R<2>, R<3>, R<4> and R<5> have the meanings indicated, their physiologically tolerable salts and a process for their preparation are described. The compounds inhibit aldose reductase and can be used as medicaments.
Patent FI-20001874-A0 (FI)
Inventor: LAHDENSIVU KIMMO
IPC: H04L29/12
Filed: 2000-08-24
Abstract: The present invention relates to a method for centralized configuration of a telecommunication network, which telecommunication network comprises one or more IP networks with their addresses. From a set of IP addresses, an IP alias is generated. In the method, a predetermined change is made at least in one service parameter of the IP alias or of the devices belonging to the IP alias; those IP additional services are defined whose parameters are affected by the change in question, and the necessary configuration changes are made in the devices generating the IP additional services in question. According to the invention, a device configuration database is created that comprises the configuration information of the additional service devices; the aforementioned change is focused on the IP alias in question, and the aforementioned configuration changes of the additional service devices are made automatically and in parallel utilizing the aforementioned device configuration database.
Patent FI-20041010-A0 (FI)
Inventor: DE GODZINSKY CHRISTIAN
IPC: G03B42/02
Filed: 2004-07-22
Abstract: This invention relates to mutual positioning of an x-ray beam and an intra-oral x-ray sensor in connection with an imaging process by utilizing at least one measurement signal, which is achieved by arranging means for producing a magnetic field resp. for measuring the magnetic field in connection with a radiation source resp. the sensor.
Patent FI-20105279-A0 (FI)
Inventor: HARTIKKA YRJOE
IPC: H05B45/50
Filed: 2010-03-19
Abstract: A LED tube (41) comprises one or more LED components (34) and a current control unit (33) installed therein. Both ends of the LED tube (41) are provided with a contact pin pair (37, 38, 39, 40) for connecting the LED tube mechanically and electrically to tube holders of a fluorescent tube lighting fixture. The LED tube includes a safety unit (42, 43, S1) arranged to prevent a voltage from passing through the LED tube (41) from its one end to the other end thereof until at both ends of the LED tube, a voltage (U1, U2) fed from the corresponding tube holder of the lighting fixture to the contact pin pair (37, 38, 39, 40) has been detected separately.
Patent FI-20115771-A0 (FI)
Inventor: KALLIONIEMI ANTTI
Filed: 2011-07-28
Abstract: The invention relates to an elevator system and also to an electricity supply device (1, 2, 3) for supplying electric power in the elevator system. The electricity supply device (1, 2, 3) comprises a controllable power output stage (4, 5), comprising a connection to the load (6, 7, 8) of the elevator system to be supplied. The power output stage (4, 5) comprises one or more controllable solid-state switches (9) in the form of silicon carbide (SiC) solid-state switches.
Patent IL-103089-A0 (IL)
Title: Process for manufacture of insecticidal,nematicidal and acaricidal 2-aryl-3-substituted-5-(trifluoromethyl)pyrrole compounds from n-(substituted benzyl)-2,2,2-trifluoroacetimidoyl chloride compounds
IPC: C07D207/34
Filed: 1992-09-07
Abstract: There is provided a process for the manufacture of insecticidal, nematicidal and acaricidal 2-aryl-3-substituted-5-(trifluoromethyl)pyrrole compounds via the condensation of an N-(substituted benzyl)-2,2-2-trifluoroacetimidoyl chloride compound with an  alpha -halo- alpha , beta -unsaturated nitrile, ester or nitro compound.
Patent IL-105772-A0 (IL)
Title: Methods and materials for combating pests
IPC: A01M1/02
Filed: 1993-05-21
Abstract: The subject invention pertains to materials and methods useful for management of certain pests. The invention is particularly well suited for the control of social insect pests and, particularly, termites. The invention concerns unique toxicant-containing matrices as well as apparatuses for monitoring pest activity and presenting a toxicant. The invention is useful as part of an Integrated Pest Management Program and can greatly reduce the introduction of harmful chemicals into the environment.
Patent IL-109581-A0 (IL)
Title: Tetrazole derivatives of bile acids, processes for their preparation and the use of these compounds as medicaments
IPC: A61P9/10
Filed: 1994-05-06
Abstract: Tetrazole bile acid derivatives of the formula I  G1 - X - G2      I in which G1, G2 and X have the stated meanings, and processes for their preparation are described. The compounds have valuable pharmacological properties and can therefore be used as medicines.
Patent IL-111745-A0 (IL)
Title: Feed comb arrangement
Inventor: EGERER JOSEF
IPC: D01G19/08
Filed: 1994-11-23
Abstract: In a feed-comb arrangement for a combing machine, comprising an intermittently driven pair of feed rollers, preceding the feed-chamber arrangement in the direction of transport of the fibre web to be combed, and a draw-off arrangement, especially in the form of draw-off rollers, following the feed-chamber arrangement, in order to increase the quiet running, avoid accumulations of impurities and achieve efficient transport there is provision for the feed-comb arrangement to be formed by a plurality of needle bars (13) which are intermittently driven synchronously with the comb cycle and are equipped with needles or sawtooth-shaped stampings (14) and which run at their two outer ends in guide tracks (12) in such a way that, over part of the rotational travel, the needles or sawtooth tips (14) engage into the fibre web (2), and, on the other hand, the needles or sawtooth tips (14), after executing a transport movement, emerge upwards out of the fibre web (2). <IMAGE>
Patent IL-113918-A0 (IL)
Title: Process for preparing delta 9,11 and 21-chloro corticosteroids
IPC: C07J5/00
Filed: 1995-05-30
Abstract: Described is a process for the regioselective dehydration of 11-hydroxy steroids using PCl5, PCl3, POCl3 or either SO2Cl2 and imidazole, or PPh3 and CCl4. The disclosed process selectively forms  DELTA <9,11> steroids from either 11- alpha - or 11- beta -hydroxy steroids, and can also be used for the one-step conversion of 11,21-dihydroxy steroids to 21-chloro- DELTA <9,11> steroids. Also disclosed are processes for the regioselective conversion of 11- beta -chloro steroids to  DELTA <9,11> steroids, and for regioselectively converting an 11,17,21-trihydroxy steroid to a 21-chloro-11,17-dihydroxy steroid.
Patent IL-114724-A0 (IL)
Title: Dihalopropene compounds insecticidal/acaricidal agents containing same and intermediates for their production
IPC: C07C69/712
Filed: 1995-07-25
Abstract: The dihalopropene compounds of the general formula [I] have excellent insecticidal/acaricidal activity, so that they are satisfactorily effective for the control of noxious insects, mites and ticks.
Patent IL-121218-A0 (IL)
Title: Polypropylene fibers
IPC: D01F6/06
Filed: 1997-02-11
Abstract: The present invention relates to polypropylene fibers and nonwoven fabrics produced from spunlaid or staple fibers having improved natural bulk. Said polypropylene fibers are made of a blend of sPP and iPP.
Patent IL-124883-A0 (IL)
Title: Amidino protease inhibitors and pharmaceutical compositions containing the same
IPC: A61P1/00
Filed: 1996-12-20
Abstract: Amidino and benzamidino compounds, including compounds of the formula: wherein R1-R4, R6-R9, Y, Z, n and m are set forth in the specification, as well as hydrates, solvates or pharmaceutically acceptable salts thereof, that inhibit a number of proteolytic enzymes are described. Also described are methods for preparing the compounds of Formula I.
Patent IL-143613-A0 (IL)
Title: A process for the preparation of antihistaminic piperidine derivatives
IPC: A61P11/08
Filed: 2001-06-06
Abstract: The present invention is related to novel intermediates and processes which are useful in the preparation of certain antihistaminic piperidine derivatives of formula (I) wherein W represents -C(=O)- or -CH(OH)-; R 1  represents hydrogen or hydroxy; R 2  represents hydrogen; R 1  and R 2  taken together form a second bond between the carbon atoms bearing R 1  and R 2 ; n is an integer of from 1 to 5; m is an integer 0 or 1; R 3  is -COOH or -COOalkyl wherein the alkyl moiety has from 1 to 6 carbon atoms and is straight or branched; each of A is hydrogen or hydroxy; and pharmaceutically acceptable salts and individual optical isomers thereof, with the proviso that where R 1  and R 2  are taken together to form a second bond between the carbon atoms bearing R 1  and R 2  or where R 1  represented hydroxy, m is an integer 0.
Patent IL-148360-A0 (IL)
Title: A herpes viral mutant and pharmaceutical compositions containing the same
IPC: C07K14/035
Filed: 2000-02-02
Abstract: The present invention relates to herpes viral mutants and methods of using these viral mutants for selectively targeting tumor cells or other populations of target cells. The viral mutants of the invention are capable of selective targeting due to the use of tumor-specific and/or cell-specific promoters to drive expression of the herpes  gamma 34.5 gene.
Patent IL-151638-A0 (IL)
Title: Method and system for controlling data traffic in a network
IPC: G01R31/08
Filed: 2001-03-15
Abstract: A method and a system for optimizing the routing of data to be communicated in a network. In one embodiment, the system achieves an improved control for routing of data traffic in a network by minimizing link costs between nodes of the network.
Patent IL-156808-A0 (IL)
Title: Method and system for gemstone color prediction
IPC: G01N21/87
Filed: 2003-07-07
Abstract: Predicting a first color of a gemstone to be cut to have a first geometry, from an uncut gemstone having a second color and a second geometry, is performed by means of a system comprising gemstone-mapping device for measuring the second geometry of the uncut gemstone, a spectral measurement device for measuring the second color of the uncut gemstone; and a processor adapted to determine an absorption coefficient of the uncut gemstone's material based on data from the gemstone-mapping and the spectral measurement devices, and on calculations relating to behavior of light in the uncut gemstone. The processor is adapted to deduce the first color based on the first geometry, the deduced coefficient and calculations relating to behavior of light in the cut gemstone.
Patent IL-157540-A0 (IL)
Title: N-(aryl)-2-arylethenesulphonamides and therapeutic uses thereof
IPC: A61K31/18
Filed: 2002-02-28
Abstract: N-(Aryl)-2-arylethenesulfonamides and pharmaceutically acceptable salts and compositions thereof are useful as antiproliferative agents, including, for example, anticancer agents. They are also useful as radioprotective agents.
Patent IL-159665-A0 (IL)
Title: Locking device for connecting housing sections of an administration appliance
IPC: A61M5/28
Filed: 2002-07-22
Abstract: An administering apparatus for delivering a dosage of product including a casing with a reservoir for the product, a piston within the reservoir to deliver the product, a piston rod for engaging the piston, a drive device for driving the piston rod, and a dosage setting member mechanically engaging the piston rod and a stopper for the dosage setting member. The casing includes a front casing section containing a reservoir for the product and a rear casing section detachably connected to the front casing section. The front casing section is connected to or forms a first latching element, and the rear casing section is connected to or forms a second latching element. The latching elements are in latching engagement when the casing sections are connected. The casing sections may be axially fixed to one another by the latching engagement. The casing sections may alternately be fixed to one another, secured against rotating, with respect to a rotational movement about a longitudinal axis of the casing sections parallel to the advancing direction, by the latching engagement. The administering apparatus further includes a latching block coupled to the drive element such that the latching engagement can only be released in a releasing position of the drive element.
Patent IL-189204-A0 (IL)
Title: Heteroaryl-substituted diazatricycloalkanes, methods for its preparation and use thereof
Filed: 2008-02-03
Abstract: The present invention relates to amide and urea derivatives of heteroaryl-substituted diazatricycloalkanes, pharmaceutical compositions including the compounds, methods of preparing the compounds, and methods of treatment using the compounds. More specifically, the methods of treatment involve modulating the activity of the α7 nAChR subtype by administering one or more of the compounds to treat or prevent disorders mediated by the α7 nAChR subtype. The diazatricycloalkanes typically consist of a 1-azabicyclooctane fused to pyrrolidine ring. The substituent heteroaryl groups are 5- or 6-membered ring heteroaromatics, such as 3-pyridinyl and 5-pyrimidinyl moieties, which are attached directly to the diazatricycloalkane. The secondary nitrogen of the pyrrolidine moiety is substituted with an arylcarbonyl (amide type derivative) or an arylaminocarbonyl (N-arylcarbamoyl) (urea type derivative) group. The compounds are beneficial in therapeutic applications requiring a selective interaction at certain nAChR subtypes. That is, the compounds modulate the activity of certain nAChR subtypes, particularly the α7 nAChR subtype, and do not have appreciable activity toward muscarinic receptors. Radiolabeled versions of the compounds can be used in diagnostic methods.
Patent IL-195126-A0 (IL)
Title: Substituted 5-phenylamino-1,3,4-oxadiazole-2-
Filed: 2008-11-05
Abstract: Compounds of formula (I), or salts thereof, which inhibit acetyl CoA (acetyl coenzyme A):diacylglycerol acyltransferase (DGAT1) activity are provided, wherein R1, R2 and R3 are each independently selected from hydrogen, fluoro, chloro, cyano, trifluoromethyl, trifluoromethoxy and difluoromethoxy; together with processes for their preparation, pharmaceutical compositions containing them and their use as medicaments.
Patent IL-209749-A0 (IL)
Title: A method of producing fatty acids for biofuel, biodiesel, and other valuable chemicals
Filed: 2010-12-02
Abstract: The present invention relates to a method of producing fatty acids, by (i) inoculating a mixture of at least one of cellulose, hemicellulose, and lignin with at least one microorganism strain that produces one or more cellulases, hemicellulases and laccase, that hydrolyze at least one of cellulose, hemicellulose and lignin, under conditions to produce at least one of glucose, cellobiose, xylose, mannose, galactose, rhamnose, arabinose or other hemicellulose sugars; (ii) inhibiting growth of the at least one microorganism strain; (iii) inoculating the mixture of step (ii) with at least one algae strain that metabolizes the at least one of glucose, cellobiose, xylose, mannose, galactose, rhamnose, arabinose or other hemicellulose sugars, under conditions so that the at least one algae strain produces one or more fatty acids; and optionally (iv) recovering the one or more fatty acids from the at least one algae strain.
Patent RO-131453-A0 (RO)
Title: Self-heating reducer-vaporizer for supplying lpg to internal combustion engines
Inventor: CIOBANU MIHAI-MĂRŢIŞOR
IPC: F02M21/06
Filed: 2016-06-27
Abstract: The invention relates to a self-heating apparatus for supplying liquefied petroleum gas to internal combustion engines. According to the invention, the apparatus has a sealed enclosure for heating the liquid fuel gas, wherein electric insulating oil, needed to heat the enclosure, is introduced, while on the external wall, inside the heating enclosure, there are two glow plugs immersed in the oil, which are controlled by a temperature relay, set according to the temperature of the fuel gas within the enclosure, so that the temperature of the gas introduced into the intake manifold of an engine may be kept constant, at 20...25°C, in stabilized operating conditions.
Patent AP-2001002217-A0 (AP)
Title: Oxygenated esters of 4-iodo phenylamino benzhydroxamic acids.
Inventor: BARRETT STEPHEN DOUGLAS
IPC: C07C259/00
Filed: 2001-07-12
Abstract: The present invention relates to oxygenated esters of 4-iodophenylamino benzhydroxamic acid derivatives, pharmaceutical compositions and methods of use thereof. The present invention also relates to crystalline forms of oxygenated esters of 4-iodophenylamino benzhydroxamic acid derivatives, pharmaceutical compositions and methods of use thereof.