baber/WOPTO huggingface dataset:
Patent SK-282467-B6 (SK)
Title: Peptides, pharmaceutical preparation containing them and their use
Inventor: HAUPT ANDREAS
IPC: A61K38/08
Filed: 1996-06-03
Abstract: Peptides of formula R1R2N-CHX-CO-A-B-D-E-(F)t-K (I) and their salts with acids are new. In the formula, R1 = Me, Et or iPr; R2 = H, Me or Et; or NR1R2 = a pyrrolidine ring; A = a valyl, isoleucyl, leucyl, 2-tert-butylglycyl, 2-ethylglycyl, norleucyl or norvalyl residue; B = a N-methyl-valyl, -leucyl, -isoleucyl, -norvalyl, -norleucyl, -2-tert-butylglycyl, -3-tert-butylalanyl or -2-ethylglycyl residue; D = a prolyl, 3,4-dehydroprolyl, 4-fluoroprolyl, 4,4-difluoroprolyl, azetidine-2-carbonyl, homoprolyl, thiazolidine-4-carbonyl or 3-, 4- or 5-methylprolyl residue; E = a 3,4-dehydroprolyl, 4-fluoroprolyl, 3- or 4-methylprolyl, 4,4-difluoroprolyl or azetidine-2-carbonyl residue; F = a valyl, 2-tert-butylglycyl, isoleucyl, leucyl, 2-cyclohexylglycyl, norleucyl, norvalyl, neopentylglycyl, alanyl, ~b-alanyl or aminoisobutyroyl residue; X = alkyl (pref. 2-5C alkyl), cyclopropyl or cyclopentyl; t = 0 or 1; and K = alkoxy (pref. 1-4C alkoxy), benzyloxy or opt. substd. amino.
Patent SK-279050-B6 (SK)
Title: Microbiological process for the preparation of aromatic hydroxylated heterocyclic carboxylic acids, microorganisms pseudomonas acidovorans and alcaligenes faecalis
Inventor: KIENER ANDREAS
IPC: C12R1/38
Filed: 1992-12-04
Abstract: The microbiological process for the preparation of hydroxylated heterocyclic carboxylic acid of the formula (1) is described below. Heterocyclic carboxylic acid is the initial substance. The process is carried out in such a way that aerobic biomass containing Pseudomonas micro-organisms and/or Alcaligenes genus and/or DSM 7202 micro-organisms and absorbing nicotinic acid is cultivated in a molar ratio of nicotinic acid to mineral acid of 1 to 8 ratio. This ratio is kept during the whole process of cultivation followed by hydroxylation of corresponding heterocyclic carboxylic acid of the general formula (II) in this biomass. Under these conditions, microorganisms of the species Pseudomonas acidovorans DSM 7205, of the species Pseudomonas acidovorans DSM 7203, of the species Alcaligenes faecalis DSM 7204 and microorganisms with the identifier DSM 7202 can be isolated in their growth phase.
Patent SK-286079-B6 (SK)
Title: Use of combination of metabolic derivative of loratadine and pseudoefedrine for manufacture of medicament for treatment of cough and other disorders
Inventor: ABERG A K GUNNAR
IPC: A61K31/00
Filed: 1995-12-11
Abstract: The use of a metabolic derivative of loratadine (DCL) or its pharmaceutically acceptable salt and pseudoefedrine or its pharmaceutically acceptable salt for the manufacture of a medicament for treatment of cough, cold, cold-like or flu symptoms and the discomfort, headache, pain, fever and general malaise associated therewith in a human while avoiding the concomitant liability of adverse side-effects associated with the administration of non-sedating antihistamines as are cardiac arrhythmias or tumor promotion.
Patent SK-278458-B6 (SK)
Title: 2-(2-subst.benzoyl)cyclohexane-1,3-diones, herbicidal agents on their base and their use
Inventor: MICHAELY WILLIAM J
IPC: C07C49/76
Filed: 1984-09-17
Abstract: The basic subject of the solution described in this patent are 2-(2-subst.benzoyl)cyclohexane-1,3-diones with a general formula (I), where the symbols R and R1 represent hydrogen, alkyl with 1 up to 4 carbon atoms or the group alkyl-OC(O)- with 1 up to 4 carbon atoms in alkyl, the symbol R2 represents halogen or alkoxyl group with 1 up to 4 carbon atoms and the symbols R3, R4 and R5 represent hydrogen, halogen and another different organic rests, explained in the description in more details. This solution also is dealing with the suppression of an unfavourable vegetation with the use of the above mentioned dions and herbicides made based on these diones.
Patent CZ-304091-B6 (CZ)
Title: Method for producing gas from at least partially gasifiable solid material and apparatus for making the same
Inventor: OCHODEK TADEAS
IPC: B09B3/45
Filed: 2007-11-23
Abstract: The present invention relates to a method of gas production from at least partially gasifiable solid material, using the effect of gasification agent, wherein the method is characterized in that the first portion of particles of at least partially gasifiable solid material is piled inside the reaction zone into a fixed bed of at least partially gasifiable solid material, whereas the other portions of at least partially gasifiable solid material are continually and/or by pulse procedure introduced under the surface of this fixed bed, thereby the particles creating the fixed bed of at least partially gasifiable solid material are transferred from the inside of this fixed bed of at least partially gasifiable solid material towards its periphery, and at the same time, the particles of at least partially gasifiable solid material are exposed to the influence of the gasification agent, which is introduced into the reaction zone, in the process the gasification agent penetrates at least partially under the surface of the fixed bed of at least partially gasifiable solid material and furthermore, the particles of at least partially gasifiable solid material which reached to the surface of this fixed bed pass into the fluidized bed, due to the flow of gases and/or pass into the outlet of the non-gasified residue due to gravity, whereas the particles in the fluidized bed are exposed further to the influence of gases that are present in the reaction zone until the conversion of these particles into the produced gas and the non-gasified residue, which is removed from the reaction zone separately and/or is carried out by the produced gas. The apparatus for making the above-described process comprises a reactor (1), into the reaction zone (2) of which there are introduces the inlet (3) of at least partially gasifiable solid material, at least one inlet (4) of the gasification agent, the outlet (5) of the produced gas and the outlet (6) of the non-gasified residue. A part of the reaction zone (2) is the space (7) for forming the fixed bed (8) of at least partially gasifiable solid material, to which the inlet (3) of at least partially gasifiable solid material is introduced. The reactor (1) involves at least one grate (10) which is located between the reaction zone (2) and the outlet (6) of the non-gasified residue. With advantage, an inlet of gasifiable liquid may be introduced into the reaction zone (2). Equipment for preheating of at least partially gasifiable material may be located at the inlet (3) of at least partially gasifiable solid material. To preheat the gasification agent, the equipment (13) for preheating the gasification agent may be located at the inlet (4) of the gasification agent. The equipment for preheating of gasified liquid may be located in the inlet of gasified liquid. Preferably, the reaction zone (2) is surrounded by thermal insulation (15), which is resistant to the temperature of 1600 degC.
Patent CZ-303477-B6 (CZ)
Title: Process for preparing hard, heat-resistant protective coatings on Al-Si alloys
Inventor: VOJTECH DALIBOR
IPC: C23C18/22
Filed: 2010-08-17
Abstract: The invented process for preparing Ni-P layers on Al-Si alloys containing 5 to 25 percent by weight of silicon, optionally other elements, is carried out in the following three steps: a) surface treatment of the alloy by grinding and degreasing, b) selective dissolution of aluminium in order to increase surface roughness, c) chemical plating in a bath. A method of preparing layers of Ni-P with Ali2Oi3 fiber on Al-Si alloys containing 5 to 25 percent by weight of silicon, optionally other elements, is carried out in the following four steps: a) surface treatment of the alloy by grinding and degreasing, b) selective dissolution of aluminium in order to increase surface roughness, c) activation of aluminium oxide fibers and d) chemical plating in a bath containing aluminum oxide fibers.
Patent CZ-303620-B6 (CZ)
Title: Segment for detection of contact force acting on femoral skeleton for passive safety tests
Inventor: SCHNEJBALOVA ZUZANA
IPC: G01M17/00
Filed: 2010-12-22
Abstract: The present invention relates to a segment for detection of contact force acting on femoral skeleton (1) for passive safety tests, especially a child pedestrian in case of his collision with a vehicle, wherein the segment is formed by the femoral skeleton (1) or a mechanical equivalent of thighbone fitted with two strain gauge semi bridges (2). One strain gauge semi bridge (2) is situated on the side turned towards the impact while the other one on the side turned away from impact. The skeleton (1) is provided with a material in the form of the thigh with properties corresponding to muscle tissue of a child pedestrian.
Patent CZ-305988-B6 (CZ)
Title: Sensor for checking bee colony vitality
Inventor: TEJKL JAROMÍR
IPC: G01K7/00
Filed: 2014-10-14
Abstract: The sensor for checking bee colony vitality according to the present invention is formed by a matrix (2) of eight or more thermistors (2) or the like temperature sensing elements (2), which are distributed regularly all over the surface of the sensor (10) and along with a microprocessor and a battery (6), they are pressed or bonded between two flexible foils. In corners, the sensor can be supplemented by pressure sensing elements (3) and further with a sunlight and external temperature sensing elements (4, 5). Space arrangement of the sensors further comprises two pr four symmetrically arranged openings for free passage of bees when situated between beehive supers (9). The sensors (10), being situated between the beehive supers (9), form a system for measuring the weight of the separate supers (9). The use of the sensor (10) assembly consists in non-invasive method of measuring (without dismounting the beehive) and evaluation of temperature in the beehive 3D space, and measures and evaluates the weight of the separate supers (9) with determination of a hive body size. Based on the change in the hive body size and weight of the separate supers (9), the health state and vitality of the bee colony is also determined relative to the year season.
Patent SK-288195-B6 (SK)
Title: Actuator with artificial muscles - I.
Inventor: PITEL JAN
IPC: B25J13/06
Filed: 2011-05-02
Abstract: Actuator with artificial muscles , which consists of a base plate ( 1 ) with firmly attached two pillars ( 2 ) , which are firmly attached bearing housings ( 3 ) . Through them is pushed onto the shaft ( 4 ) , which is firmly pushed roller ( 7 ) , at the end of what - shaft ( 4 ) is pushed onto the hub ( 6 ) . That is rigidly fixed to the arm (5 ) , at the end of which is screwed onto the load weight (16 ) . Artificial muscles ( 8 ) by means of the rods ( 11 ) coupled to the movable pulley ( 12 ) , through which is threaded through the flexible sheet ( 13 ) , mounted over the roller ( 7 ) . This also passes through the front brackets (14 ) and is secured at spring clip ( 15 ) . Artificial muscles ( 8 ) by means of the rods ( 9 ) connected to the rear support ( 10 ) and are fixed to the pillars ( 2 ) . Resulting from the introduction of the transfer and consequently required less artificial muscle contraction ( which is at - the output power actuator ) is necessary to use artificial muscles with more force ( twice ) .
Patent SK-285366-B6 (SK)
Title: Method of injection (meth)acrylate copolymers with a tertiary ammonium groups
Inventor: PETEREIT HANS-ULRICH
IPC: A61K9/20
Filed: 2000-11-29
Abstract: Method of production moulded parts by injection comprising the steps: a) melting a (meth)acrylate copolymer being present in admixture with 1 to 70 wt. % of a plasticiser and antiadhesive agent in a ratio of 1:1 to 1:20, and 0.05 to 5 wt. % of a mould-release agent , other conventional additives or adjuvants and optionally a pharmaceutical active substance be present in the mixture and before melting the mixture contains more than 0.5 wt. % of low-boiling ingredients with a vapour pressure of at least 190 kPa at 120 °C, b) degassing the mixture in the thermoplastic state at temperatures of at least 120 °C, thereby lowering the content of the low-boiling ingredients with a vapour pressure of at least 190 kPa at 120 °C to not more than 0.5 wt. % and c) injection the molten and degassed mixture containing at most 0.5 wt. % of the low-boiling ingredients with a vapour pressure of at least 190 kPa at 120 °C into the moulding cavity, whereby the moulding cavity being at a temperature which is at least 10 °C below the glass transition temperature of the (meth)acrylate copolymer, cooling the molten mixture and removing obtained moulded body from the mould.
Patent CZ-302748-B6 (CZ)
Title: Interconnect structure
Inventor: EDELSTEIN DANIEL
IPC: H01L21/3205
Filed: 2000-05-15
Abstract: In the present invention, there is disclosed an interconnect structure comprising a layer (1) of copper, a pad-limiting layer (7), a barrier layer (10) and a layer (9) of AlCu, wherein the layer (9) of AlCu and barrier layer (10) are interposed between the layer (1) of copper and pad-limiting layer (7), and wherein the barrier layer (10) being located between the layer (1) of copper and the layer (9) of AlCu ensures a robust interconnection of said layer (1) of copper and said pad-limiting layer (7). In preferred embodiment, the layer (9) of AlCu contains about 96 to about 99.5 atomic percent of aluminium Al, optionally 4 to 0.5 atomic percent of copper Cu and is 0.5 to 1.2 microns thick. The barrier layer (10) can be made of titanium Ti, titanium nitride TiN, tantalum Ta, tantalum nitride TaN, alloys, or combinations thereof. In preferred embodiment, the barrier layer (10) consists of individual layers of the following thicknesses: tantalum nitride TaN layer 50 to 1000 A, titanium layer Ti 200 to 700 A, and a titanium nitride TiN layer 200 to 700 A.
Patent CZ-298618-B6 (CZ)
Title: Method for producing pozzolanic or hydraulic grinding additives from various kinds of basic oxidic slag intended for industrial production of cement
Inventor: EDLINGER ALFRED
IPC: C21B3/06
Filed: 2001-01-18
Abstract: The present invention relates to a method for the production of pozzolanic or hydraulic grinding additives from various kinds of basic oxidic slag for the cement industry from basic oxidic slags, especially steel slags, using a metal bath for reducing metal oxides in the slags. According to said method, the basicity of the liquid slags is adjusted, prior to reduction, to a value that is 0.1 to 0.5 lower than the basicity value (Ca0/Si0i2) of the target slag by adding acid correction materials such as silica sand and/or blast furnace slag and/or correction materials containing SiOi2.
Patent CZ-296902-B6 (CZ)
Title: Process for preparing 6-(4-phenylbutoxy)hexylamine derivative
Inventor: BASSA BELLMUNT JORDI
IPC: C07C213/08
Filed: 1999-09-20
Abstract: In the present invention, there is disclosed a process for preparing 6-(4-phenylbutoxy)hexylamine derivative of the general formula I, in which Ri1 represents the group CHO or the group CHORi3ORi4 wherein Ri3 and Ri4 denote independently on each other alkyl groups containing 1 to 6 carbon atoms, arylalkyl groups having 1 to 6 carbon atoms in the alkyl moiety and 6 to 10 carbon atoms in the monocyclic or bicyclic aryl moiety, or they form 5 or 6-membered cyclic acetals; and Ri2 represents a hydrogen atom, a benzyl group or an alkyloxycarbonyl group, an aryloxycarbonyl group, an arylalkyloxycarbonyl group or an acyl group of the general formula R-CO-, in which R denotes alkyl, being optionally substituted with a halogen, phenyl or phenylalkyl; whereby in the groups represented by Ri2 all the alkyl residues contain 1 to 6 carbon atoms and aryl residues contain 6 to 10 carbon atoms in a monocyclic or bicyclic system, wherein the preparation process is characterized by (i) reacting the compound of the general formula 11 with the compound of the general formula 12 to obtain the compound I, in which Ri1 is the group CHORi3ORi4 wherein Ri3 represents a hydrogen atom or a benzyl group and Ri4 is as defined above; and Ri2 denotes a hydrogen atom or a benzyl group; whereby the compound of the general formula I can be further transformed in order to obtain the full range of the compounds of the general formula I.
Patent SK-288563-B6 (SK)
Title: A process for preparing a composite sorbent for removing contaminants from water
Inventor: NOVAK IVAN
IPC: C02F1/00
Filed: 2014-12-15
Abstract: Method for the preparation of high performance composite sorbents for removing contaminants from nanoporous carbon fiber-based waters coated with nano particles and micro particles of hydrated iron oxides utilizing the synergistic effect of a large surface of nano- and microparticles of hydrated iron oxides and a fibrous structure of the carrier , which reduces resistance to water flow, wherein the effectiveness and capacity of the sorbent in the removal of contaminants in the field of practical use is independent of the pH of the water.
Patent EP-1160204-B8 (EP)
Inventor: HOWSE GEOFFREY
IPC: B01J49/00
Filed: 2001-05-09
Granted: 2007-10-03
Abstract: Water treatment apparatus, such as a water softener, comprises two water treatment components (1, 2) and valve means for causing the two components to be rendered inoperable to treat water at respective different intervals so that at least one component (1, 2) is operable all the time, characterised in that the valve means comprises waterflow controlled valve means and the apparatus includes a water driven flow-meter (16) for controlling said valve means. <IMAGE>
Patent EP-1436208-B8 (EP)
Title: Ebauche de boite a lentille pliable et boite a lentille ophtalmiques formee a partir de cette ebauche
Inventor: MATHIAS GREGORY T
IPC: B65D5/50
Filed: 2002-10-18
Granted: 2012-03-07
Abstract: La présente invention concerne une ébauche (2) de boîte à lentille et une boîte (10) à lentille. L'ébauche de boîte à lentille qui est pliée sous forme d'une boîte à lentille peut, par exemple, comprendre: un alignement (4) d'élément transversal de segments de boîte et un alignement (6) de partie verticale de segments de boîte; les segments d'alignement de partie verticale comprenant au moins un rabat avant (28), un rabat supérieur (24), un rabat inférieur (20) et un rabat arrière (22) séparés par des lignes de pliage; l'alignement de tronçon transversal d'éléments de boîte comprenant de manière symétrique autour du rabat inférieur, au moins deux rabats latéraux (18), au moins deux rabats supérieurs (14) du cadre de support, au moins deux rabats (10) du cadre de support de lentille pourvus d'une ouverture (12) formée dans chaque rabat de support de lentille pour recevoir une lentille et au moins deux rabats (8) de fixation du cadre de support de lentille. L'ébauche de boîte à lentille peut être telle qu'au moins un segment de rabat arrière et le rabat inférieur comporte un prolongement (30) de rabat sur ce dernier. L'ébauche de boîte à lentille peut également comprendre des ouvertures de rabat du cadre de support de boîte à lentille qui sont au moins partiellement courbées. De plus, le rabat supérieur et au moins une partie supérieure du cadre de support peuvent comporter un système (16, 26) de blocage par languettes qui sert à relier le rabat supérieur et le rabat supérieur du cadre de support. Un cadre (402) de boîte en té à ailettes comprend des éléments de blocage additionnels qui permettent de fixer la boîte à lentille en position fermée avec une lentille à l'intérieur.
Patent EP-2004073-B8 (EP)
Inventor: KYPHON SARL
IPC: A61B17/70
Filed: 2007-04-03
Granted: 2010-05-12
Abstract: This device (10) includes an interspinous implant (1) having a flexible structure, capable of being inserted between the spinous processes (100) of two vertebrae, the areas (Z) of these respective spinous processes (100) bearing against the implant (1) defining a longitudinal axis (L) of the implant (1). According to the invention, the device includes at least one cerclage (15) capable of being adjustably engaged around the implant (1), at a centre section (4) of this implant (1), in a plane (P) perpendicular to said longitudinal axis (L); this cerclage (15) is made of a material that is inextensible in the circumferential direction of this cerclage (15), so that it makes it possible to restrain deformation of the implant (1) at the centre section (4), within the entire said plane (P), during exertion on this centre section (4) of opposing compressive forces exerted by the spinous processes of the vertebrae during a posterior movement of the spinal column.
Patent EP-2165774-B8 (EP)
Inventor: RAKSHA VLADIMIR P
IPC: B05D5/12
Filed: 2003-07-01
Granted: 2021-03-17
Abstract: The invention relates to an apparatus (200) for orienting magnetic pigment flakes in a fluid carrier printed on a first side of a substrate (212) in a linear printing process. The apparatus comprises a magnetic structure (202,204,206,208) disposed proximate to a second side of the substrate, the magnetic structure creating a selected magnetic field configuration to orient the magnetic pigment flakes to form an image.
Patent BR-PI0509761-B8 (BR)
Title: compostos de quinolinona-carboxamida como agonistas de receptor de 5-ht4, composição farmacêutica, uso dos referidos compostos e seu processo de preparação
Inventor: ADAM A GOLDBLUM
IPC: A61K31/46
Filed: 2005-04-06
Abstract: compostos de quinolinona-carboxamida como agonistas de receptor de 5-ht~ 4~. a invenção fornece compostos agonistas do receptor de 5-ht~ 4~ de quinolinona-carboxamida inéditos de fórmula (i). a invenção também fornece composições farmacêuticas que compreendem estes compostos, o uso desses compostos para o tratamento de doenças associadas à atividade do receptor de 5-ht~ 4~ e processos e intermediários úteis para preparação desses compostos. onde: r^ 1^ é hidrogênio, halo, hidroxi, c~ 1-4~alquil ou c~ 1-4~alcoxi; r^ 2^ é c~ 3-4~a1quil ou c~ 3-6~cicloalquil; r^ 3^ é hidrogênio ou c~ 1-3~alquil; r^ 4^ é - s (o)~ 2~r^ 6^ ou - c (o) r^ 2^; r^ 5^ é hidrogênio, c~ 1-3~alquil, c~ 2-3~alquil, substituído com -oh ou c~ 1-3~alcoxi ou -ch~ 2~-piridil; r^ 6^ é c~ 1-3~alquil; ou, r^ 5^ e r^ 6^, tomados em conjunto formam c^ 3-4~alquilenil; e r^ 7^ é hidrogênio, c~ 1-3~alquil ou piridil; ou um sal ou solvato ou estereoisômero farmacêuticamente aceitável desses.
Patent BR-PI0511662-B8 (BR)
Title: combinação e usos de um antagonista de receptores muscarínicos m3 e de um agonista beta2 no tratamento de distúrbios respiratórios
Inventor: HAMISH RYDER
IPC: A61K45/00
Filed: 2005-05-31
Abstract: combinação, uso de um agonista beta2 e um antagonista de receptores muscarínicos m3, produto, kit de partes, e, embalagem um combinação que compreende (a) um agonista (beta)2 e (b) um antagonista de receptores muscarínicos m3 que é 3(r)-(2-hidróxi-2,2-ditien-2-il-acetóxi)-1-(3 -fenóxi-propil)-1-azoniabiciclo[2.2.2]octano, na forma de um sal possuindo um ânion x, que é um ânion farmaceuticamente aceitável de um ácido mono ou polivalente.
Patent BR-PI0609634-B8 (BR)
Title: dispositivo de lanceta ativado por dedo
Inventor: ROBERT COLONNA
IPC: A61B5/151
Filed: 2006-04-07
Abstract: dispositivo de lanceta ativado por dedo um dispositivo de lanceta inclui um alojamento com uma mola do tipo cantiléver se estendendo neste e definindo uma lanceta tendo uma extremidade perfurante na mola do tipo cantiléver. um ativador se estende no alojamento através da abertura na extremidade dianteira. o ativador inclui um engate de interferência com a mola do tipo cantiléver. o movimento do ativador no alojamento através da extremidade dianteira articula a mola do tipo cantiléver contra sua condição relaxada e então libera o engate com a mola do tipo cantiléver, desse modo permitindo à mola do tipo cantiléver articular a estrutura de lanceta para uma posição estendida com a extremidade perfurante se estendendo através da abertura dianteira, e retornar para a condição relaxada retraindo a extremidade perfurante de volta no alojamento.