baber/WOPTO huggingface dataset:
Patent FI-883218-A0 (FI)
Inventor: BOWMAN ROBERT M
IPC: C07D471/04
Filed: 1988-07-06
Abstract: Disclosed are 1,2-benzisoxazole and 1,2-benzisothiazole derivatives represented by formula I    <IMAGE>  (I)  wherein X represents oxygen or sulfur; Z rep;esents carbon (CH) so as to complete the imidazol-1-yl ring radical or Z represents nitrogen (N) so as to complete the 1,2,4-triazol-1-yl ring radical; R1 represents hydrogen, lower alkenyl, lower alkynyl, aryl-lower alkyl or lower alkyl; R2 represents hydrogen, lower alkenyl, lower alkynyl, aryl-lower alkyl or lower alkyl; or R1 and R2 combined represent lower alkylene; or R1 combined with R5 located on the Z-carbon atom of the imidazolyl radical represents C2-C4-alkylene; R3 and R4 independently represent hydrogen, lower alkyl, cycloalkyl, halogen, trifluoromethyl, cyano, nitro, amino, hydroxy, lower alkanoyloxy, carbocyclic aroyloxy, lower alkoxy, or carbocyclic aryl; or R3 and R4, together when located on adjacent carbon atoms, represent lower alkylenedioxy; or R3 and R4, together when located on the carbon atoms to which attached a benzo-fused or C5-C7-cycloalka-fused ring, respectively; R5 located on carbon represents hydrogen, lower alkyl or hydroxy-lower alkyl; R6 located on carbon represents hydrogen or lower alkyl; or when Z represents carbon, R5 located on the Z-carbon atom combined with R6 located on the adjacent carbon atom represents C3-C5-alkylene; and pharmaceutically acceptable salts thereof; which are active in mammals as anticonvulsant agents.
Patent FI-885451-A0 (FI)
Inventor: BOLL WERNER
IPC: B65D75/36
Filed: 1988-11-24
Abstract: The package for the sale and transport of a small article consists of a carrying part (1) and a transparent receiving part, which is held on the carrying part, for the small article which projects into a pouch (4) of the carrying part, which pouch is open upwards and is connected on three sides to the carrying part. Based on the above, a package is to be provided which allows, in addition to the possibility of effective viewing of the small article, a repeated removal of the receiving part from the carrying part and repeated removal of the small article from the package, it being possible for the small article firstly to remain and be viewed in the receiving part until its ultimate removal. This is achieved in that the receiving part (12) is formed from a front wall (16) and a rear wall (15), a curvature (23) for receiving the small article is provided only in the front wall (16), and the lower portion of the receiving part (12) has a removal opening (Ö) between the two walls (15, 16) and projects into the receiving pouch (4) of the carrying part (1), the upper portion of the receiving part (12) and of the carrying part (1) being connected by a repeatably detachable connection in a manner secure against longitudinal displacement relative to each other. 
<IMAGE>
Patent FI-893818-A0 (FI)
Inventor: VAN HARTINGSVELDT WIM
IPC: C12R1/66
Filed: 1989-08-14
Abstract: Transformation of Aspergillus, particularly A. niger is demonstrated. Integration at the glucoamylase locus is exemplified. A chymosin expression construct is inserted at a locus, where the chymosin may be joined to a signal sequence for efficient secretion.
Patent FI-896075-A0 (FI)
Inventor: OHTA MITSUAKI
IPC: C07D235/08
Filed: 1989-12-19
Abstract: 4,5,6,7-Tetrahydrobenzimidazole derivatives (I) and salts thereof show 5-HT3 antagonizing activity <CHEM>  wherein R<1>, R<2>, R<3> independently represent hydrogen atom, hydroxy group, a halogen atom, a lower alkyl group which may optionally be substituted with a halogen atom, a lower alkoxy group, a lower alkylthio group, an aralkyloxy group, an aryloxy group, a lower alkanoyl group, carboxy group, a lower alkoxycarbonyl group or nitro group; R<4>,R<5> and R<6> can each be a hydrogen atom or a lower alkyl group; and X is an oxygen atom or sulfur atom. d
Patent FI-900512-A0 (FI)
Inventor: RUNGGALDIER DIETHARD
IPC: H02P27/02
Filed: 1990-02-01
Abstract: When using phase control of semiconductor valves (4) for controlling AC voltage converters, in order to regulate the power factor it is necessary to determine the phase angle between the current I and the voltage U by measuring the time difference between the points at which the current and voltage pass through zero. However, disturbances superimposed on the mains voltage cause considerable random fluctuations, particularly in the measurement of the times of the voltage zero-passages, which are transferred to the phase angle and can result in an unstable regulation characteristic. It is therefore proposed according to the invention to make use of a reference time for the voltage zero-passage when determining the time difference, which reference time is derived from the measured values for the true times of the preceding voltage zero-passages. 
<IMAGE>
Patent FI-911556-A0 (FI)
Inventor: JAEPOELAE JARI ILMARI
IPC: F16K31/60
Filed: 1991-03-28
Abstract: The invention concerns a valve stem adjustment device suitable for setting the valve handle to a predetermined height from the wall surface irrespective of the valve recessing depth in the wall. The device is comprised of an extension shaft (4) fitted between the stem (2) of the valve (1) and the valve handle (3) and of a protective bushing (5) enclosing the extension shaft. The extension shaft (4) can be trimmed steplessly according to installation instructions so that the handle (3) of the valve (1) remains at a predetermined height from the wall surface when mounted to the end of the extension shaft. <IMAGE>
Patent FI-911801-A0 (FI)
Inventor: SEEL TIMOTHY P
IPC: F23N5/02
Filed: 1991-04-12
Abstract: A control assembly in combination with a thermostatically responsive apparatus. In a preferred mode the principles of the present invention are applied to an infra-red heating system of the type including burner assemblies (12, 12 min ) connected in series by a heating pipe (14), the assemblies being further connected by heating pipes (14) to a vacuum pump (40). The pump (40) is driven by a variable-speed electric motor (42) which is responsive to a thermostat (16) which may initiate, through control panel (15), operation of the burner assemblies. The burning rate of the burner assemblies is controlled by varying the speed of the electric motor and this is accomplished by the control assembly (44) which is responsive to indoor and outdoor temperature sensing devices (48, 50). The control assembly is initially programmed with climatic data which is correlated with operational speeds of the pump to give desired thermal operational characteristics of the burners at differing temperature ranges. <IMAGE>
Patent FI-913957-A0 (FI)
Inventor: WETTLAUFER DAVID GORDON
IPC: C07D413/06
Filed: 1991-08-21
Abstract: This invention relates to 6,7-dihydro-3-phenyl-1,2-benzisoxazol-4(5H)-ones and -ols of the formula <CHEM>  wherein X is <CHEM> or loweralkyl; Y is hydrogen, halogen, loweralkyl, loweralkoxy, trifluoromethyl, nitro or amino; R is H when the bond between the oxygen atom and the carbon atom in question is a single bond; otherwise the dotted line signifies part of a double bond to the oxygen atom; R1 is hydrogen, loweralkyl or arylloweralkyl; R2 and R3 are independently hydrogen, loweralkyl or arylloweralkyl, or R2 and R3 taken together with the nitrogen atom form an optionally substituted heterocycle selected from the group consisting of piperidinyl, pyrrolidinyl, morpholinyl, imidazol-1-yl, 1-piperazinyl, said substituents being hydrogen or loweralkyl; 4-substituted-1-piperazinyl of the formula <CHEM>  where R6 is loweralkyl, aryl, arylloweralkyl, <CHEM>  2-pyrimidyl, <CHEM>  2-pyridinyl of the formula <CHEM>  or 4-pyridinyl of the formula <CHEM>  4-substituted-1-piperidinyl of the formula <CHEM> wherein R7 is hydrogen, loweralkyl, aryl, arylloweralkyl, 2-pyridinyl of the formula <CHEM>  4-pyridinyl of the formula <CHEM>  2-pyrimidinyl of the formula <CHEM>  arylcarbonyl, <CHEM> R8 is hydrogen or -OH; R4 is hydrogen, loweralkoxycarbonyl or aryloxycarbonyl; Z is chlorine, bromine or fluorine; m is an integer of 1 to 4; n is an integer of 1 to 4 or a pharmaceutically acceptable acid addition salt thereof and where applicable the geometric and optical isomers and racemic mixtures thereof. The compounds of this invention display utility as antipsychotic agents and analgesic agents.
Patent FI-922418-A0 (FI)
Inventor: SCHLIENGER ALBERT
IPC: B61D45/00
Filed: 1992-05-26
Abstract: The cargo carrier (1), for example an interchangeable container, is secured on the turntable (2) of a railway wagon by means of swivellable holding claws (11, 11') which are articulated below the turntable. The holding claws are permanently acted on by an energy store, preferably in the form of a spring 14, and are pressed into the engagement position. This engagement position is reached as soon as the two parallel support rails (4, 4') of the turntable (2) are in the travel position parallel to the longitudinal sides of the railway wagon. <IMAGE>
Patent FI-923348-A0 (FI)
Inventor: HANSEN JOHN-ERIK STIG
IPC: A61P31/18
Filed: 1992-07-23
Abstract: A monoclonal or other antibody to the carbohydrate antigen Tn can be used to inhibit or slow the progression of AIDS or ARC. The atigen can be used in a vaccine, for immunisation.
Patent FI-930644-A0 (FI)
Inventor: RUDELLA MICHAEL D
IPC: A61K9/70
Filed: 1993-02-12
Abstract: The invention relates to a process of sealing transdermal drug delivery system components together which comprises contacting the surfaces of the components to be sealed together with each other and exposing the contacted surfaces to ultrasonic radiation while said surfaces are still in contact to produce a seal of said surfaces in a predetermined manner.
Patent FI-932158-A0 (FI)
Inventor: KJELLMAN HELENA
IPC: A47C7/00
Filed: 1993-05-12
Abstract: PCT No. PCT/FI94/00176 Sec. 371 Date Nov. 9, 1995 Sec. 102(e) Date Nov. 9, 1995 PCT Filed May 6, 1994 PCT Pub. No. WO94/26149 PCT Pub. Date Nov. 24, 1994The present invention is related to a hub for a rotatable chair, said hub comprising an essentially pyramidal body having its side faces (1) suited for the mounting of the chair's leg element (2) thereon and further including a centrally aligned cylindrical cavity (3) suited for accommodating the center rod (4) of the chair seat cushion. The hub is characterized in that the lower part of each side face (1) is flared outwardly forming a slanting flank (5) with at least one hole (6) suited to accommodate a fixing screw (7) adapted to be screwed from underneath the hub into each leg element (2), and that each side face (1) further includes an essentially radially projecting support element (8) adapted for insertion into a mating groove (9) provided to each leg element (2).
Patent FI-943121-A0 (FI)
Inventor: ERKOBONI DAVID FRANK
IPC: C08J3/00
Filed: 1994-06-29
Abstract: A particulate co-processed unattrited microcrystalline cellulose:hydrocolloid composition wherein the respective components are present in a weight ratio of from about 99:1 to 70:30. The composition is useful as a spheronizing agent for producing spheroids of uniform size and sphericity and having high drug loadings. The composition is produced by drying a slurry of the microcrystalline cellulose in an aqueous solution of the hydrocolloid. The preferred hydrocolloid is methylcellulose.
Patent FI-943285-A0 (FI)
Inventor: KIISKI ERKKI
IPC: D21F3/08
Filed: 1994-07-11
Abstract: The invention relates to the manufacture of paper machine roll shells of stainless steel. According to the invention, powder is made of molten steel by gas-atomizing, a roll shell preform is made of the powder, and the roll shell preform is machined to form a roll shell. The main advantage of the rolls shells according to the invention is their good corrosion fatigue resistance. <MATH>
Patent FI-953838-A0 (FI)
Inventor: SENN-BILFINGER JOERG
IPC: A61K31/407
Filed: 1995-08-14
Abstract: PCT No. PCT/EP94/00335 Sec. 371 Date Aug. 15, 1995 Sec. 102(e) Date Aug. 15, 1995 PCT Filed Feb. 7, 1994 PCT Pub. No. WO94/18199 PCT Pub. Date Aug. 18, 1994The invention relates to novel compounds of the formula I    <IMAGE>  (I)  and the therapeutic use thereof.
Patent FI-954447-A0 (FI)
Inventor: PATTERSON ALAN
IPC: A61K9/06
Filed: 1995-09-20
Abstract: A sustained release veterinary composition, for intra-muscular and subcutaneous administration comprises Tylosin and an oily vehicle containing a gelling agent, wherein the gelling agent may be an aluminium salt of a fatty acid such as stearic acid and the oily vehicle may be a low viscosity polyol diester of a short chain naturally derived fatty acid such as propylene glycol dicaprylate/dicaprate.
Patent FI-954580-A0 (FI)
Inventor: VACCA JOSEPH P
IPC: C07D241/04
Filed: 1995-09-27
Abstract: Compounds of formula <CHEM> where R1 and R2 are independently hydrogen or optionally-substituted C1-4alkyl or aryl, or R1 and R2 are joined together to form a monocyclic or bicyclic ring system, are HIV protease inhibitors. These compounds are useful in the prevention or treatment of infection by HIV and in the treatment of AIDS, either as compounds, pharmaceutically acceptable salts, pharmaceutical composition ingredients, whether or not in combination with other antivirals, immunomodulators, antibiotics or vaccines. Methods of treating AIDS and methods of preventing or treating infection by HIV are also described.
Patent FI-955436-A0 (FI)
Inventor: JOHANSSON LARS
IPC: B62B5/04
Filed: 1995-11-10
Abstract: A parking device for parking a handtruck on the floor of a truck or like vehicle so as to prevent accidental movement of the handtruck on the floor during movement of the truck. The device includes a frame structure (4) which is comprised of four mutually joined frame parts, of which one part (2) is longer and thicker than the remaining sides of the frame. This longer and thicker side extends at both ends beyond the remainder of the frame, i.e. the frame parts that extend generally at right angles to the longer and thicker part (2) are joined thereto slightly inwards from the ends of the part. The cavity (5) defined by the frame is intended to receive the wheels of the handtruck, whereas the upper surface (3a) of the longer and thicker frame part (2) is intended to receive the remainder of the handtruck and thus support the general weight thereof.
Patent FI-960856-A0 (FI)
Inventor: KLAUS MICHAEL
IPC: C07C59/64
Filed: 1996-02-23
Abstract: Novel nonatetraenoic acid derivatives of the formula <CHEM> wherein the dotted bond is optional and R1 and R2 are as defined in the specific ation selectively bind to retinoic acid X-receptors (RXR) have anti-acne acitvity and potentiate the activity of retinoids having RAR alpha  activity.
Patent FI-971489-A0 (FI)
Inventor: CHASIN MARK
IPC: C07D417/06
Filed: 1997-04-10
Abstract: Novel compounds which are effective PDE IV inhibitors are disclosed. The compounds possess improved PDE IV inhibition as compared to theophylline or rolipram, with improved selectivity with regards to, e.g., PDE III inhibition.
Patent FI-973806-A0 (FI)
Inventor: HAUMONT SERGE
IPC: H04L12/56
Filed: 1997-09-26
Abstract: Method and arrangement for intercepting a target mobile station in a GPRS network. A legal interception node is installed into the land-based portion of the radio network. An "intercepted" status is defined for mobile stations that are to be intercepted. In response to an order from a law-enforcement authority to intercept one of said mobile stations the status of such mobile station is changed to "intercepted" and at least some of the packets originating from such a mobile station or terminated thereto are routed and/or copied from at least one of the support nodes via the legal interception node to the law-enforcement authority.
Patent FI-974185-A0 (FI)
Inventor: LENTO KYOESTI
IPC: B29D11/00
Filed: 1997-11-10
Abstract: The invention relates to a method and an arrangement in connection with a secondary coating line, in which method a fiber, fibers or fiber bundles are unwound from payoff reels (1) and guided to a press (4) by which a secondary sheath is formed around the fiber(s) or the fiber bundles and grease is fed into the secondary sheath, and in which method the assembly formed by the secondary sheath and the fiber(s) or the fiber bundles is pulled at a constant rate and low tension to a winding device (15) through cooling means (5, 6). In order to control the difference in length between the fibers and the secondary sheath, the difference in length between the fibers and the secondary sheath is arranged to be adjusted by adjusting fiber tension by moving the fixing point between the fibers and the secondary sheath along a straight part formed in the relaxation part by using wheel structures (8, 10).
Patent IL-76502-A0 (IL)
Title: Multiprocessor shared pipeline cache memory
IPC: G06F12/084
Filed: 1985-09-26
Abstract: A cache memory unit is constructed to have a two-stage pipeline shareable by a plurality of sources which include two independently operated central processing units (CPUs). Apparatus included within the cache memory unit operates to allocate alternate time slots to the two CPUs which offset their operations by a pipeline stage. This permits one pipeline stage of the cache memory unit to perform a directory search for one CPU while the other pipeline stage performs a data buffer read for the other CPU. Each CPU is programmed to use less than all of the time slots allocated to it. Thus, the processing units operate conflict-free while pipeline stages are freed up for processing requests from other sources, such as replacement data from main memory or cache updates.
Patent IL-88657-A0 (IL)
Title: Preparation of certain cyclopropane derivatives
IPC: C07C33/50
Filed: 1988-12-12
Abstract: The invention provides a process for the preparation of a compound of the general formula (I): <CHEM> wherein X, Y and R<1> to R<7> are as defined. In the process, the olefinic analog of the compound of general formula (I) is treated with a halogen-bearing compound in the presence of metallic zinc.
Patent IL-93246-A0 (IL)
Title: Flame-retardant thermostable homopolyimides and method of producing these
IPC: D01F6/74
Filed: 1990-02-01
Abstract: In order to prepare novel flame-retardant, thermostable homopolyimides containing structural units of the formula 
<IMAGE>
 by reacting 3,3',4,4'-benzophenonetetracarboxylic dianhydride with an, in total, equimolar amount of 2,4- and/or 2,6-tolylene diisocyanate, the reaction is carried out in the presence of a polymerisation accelerator. 
<??>The novel homopolyimides have a glass transition temperature of at least 320 DEG C and can be converted into mouldings having a similar structural strength to that observed hitherto only for copolyimides. In addition, the novel homopolyimides can be spun to form fibres.
Patent IL-94335-A0 (IL)
Title: Method and circuit for controlling oscillation current in an oscillator
IPC: H03L5/00
Filed: 1990-05-09
Abstract: An automatic voltage-controlled oscillator (VCO) current control circuit, that senses a voltage in the VCO representative of the current of the VCO, compares that voltage to a reference voltage, and applies the voltage resulting from that comparison back to the VCO at a point therein that changes its bias state in such a manner as to maintain the noise level in the VCO at a minimum and also maintains the power output of the oscillator substantially constant.
Patent IL-94587-A0 (IL)
Title: Polymer base blend compositions containing destructurized starch
IPC: C08L69/00
Filed: 1990-06-01
Abstract: A thermoplastic polymer composition comprising     a) a destructurized starch, and b) an effective amount of at least one polymer which contains at least two different types of functional groups, one of said types of these groups being hydroxyl groups.   The composition may contain further conventional additives as well as hydrophobic, substantially water-insoluble polymers.
Patent IL-108704-A0 (IL)
Title: Preparation of a cetrorelix lyophilisate
IPC: A61K38/00
Filed: 1994-02-18
Abstract: Sterile freeze-dried cetrorelix acetate (a peptide described in EP299402) is used in the treatment of female infertility. Independent claims are also included for the following: (1) use of sterile freeze-dried cetrorelix acetate for protecting gonads against noxious agents that damage germ cells, e.g. radiation treatment and chemotherapy; (2) a composition comprising sterile freeze-dried cetrorelix acetate and optionally excipients for use in the treatment of female infertility; (3) a composition comprising sterile freeze-dried cetrorelix acetate and optionally excipients for protecting gonads against noxious agents that damage germ cells, e.g. radiation treatment and chemotherapy with cytostatic agents.
Patent IL-110403-A0 (IL)
Title: Terminal block for high transmission rates in the telecommunication and data technique
IPC: H01R9/22
Filed: 1994-07-21
Abstract: The invention relates to a connection block for high transmission rates in telecommunications and data technology. The connection block 1 consists of a plastic housing 2 and of metallic insulation piercing terminal contact elements 10 which are inserted in pairs, in at least two parallel rows, into the housing 2 and have connected contact fingers 15 forming spring contacts 16. In order to reduce the capacitances between adjacent insulation piercing terminal contact elements 10 and between adjacent pairs of insulation piercing terminal contact elements 10, and thus to improve the crosstalk levels, the flat insulation piercing terminal contact elements 10 are formed only out of the base web 13 and the very narrow side webs 12 which enclose the contact slots 11 between them. The width of the contact fingers 15 is as small as possible. <IMAGE>
Patent IL-115753-A0 (IL)
Title: System for supplying consumers with heat energy and apparatus therefor
IPC: F28F27/02
Filed: 1995-10-24
Abstract: The output pipe from the at least one heat source (A,B,8) is connected to the input of at least one associated distributor device (1,2). This is formed with several outlets to which are attached the header pipes (71-79') for the consumers of heat energy at different temperature levels. One of the consumers is chosen by the distributor device so that the heated carrier medium can be supplied to it. The consumers of heat energy at different temperature level are connected in series so that the carrier medium flows through same in succession. At least one heat source is formed by a sun collector (A,B). The return lines of consumers at low temperature level are connected to the inputs of a collector device (6) formed with a single outlet pipe which can be attached to the input of a heat pump (8).
Patent IL-118217-A0 (IL)
Title: Sensor platform for the parallel detection of a plurality of analytes and method for its production
IPC: G01N21/27
Filed: 1996-05-10
Abstract: The invention relates to a sensor platform based on at least two planar, separate, inorganic dielectric waveguiding regions on a common substrate and to an apparatus for the parallel evanescent excitation and detection of the luminescence of identical or different analytes. The invention relates also to a sensor platform having the planar, separate, inorganic dielectric waveguiding regions and one or more organic phases immobilised thereon. A further subject of the invention is the use of the sensor platform in a luminescence detection method for quantitative affinity sensing and for the selective quantitative determination of luminescent constituents of optically opaque solutions.
Patent IL-120151-A0 (IL)
Title: Improved stability of azadirachtin-containing solid
IPC: A61K36/58
Filed: 1996-06-05
Abstract: The stability of an azadirachtin-containing solid preparation is increased if the preparation contains about 5% or less volatile polar solvents and 1% or less water. Reduction of the percentage of volatile polar solvents present in preparations of azadirachtin-containing solids to such levels improves the storage-stability of the solids without significantly degrading the azadirachtin in the solid. Solvents are preferably removed by drying the preparation at a suitable temperature for a time sufficient to reduce the level of water and volatile polar solvents to acceptable levels.