baber/WOPTO huggingface dataset:
Patent MA-38986-A3 (MA)
Title: Inhibiteurs marqués de l'antigène membranaire spécifique de la prostate (psma), leur utilisation comme agents d'imagerie et agents pharmaceutiques pour le traitement du cancer de la prostate
Inventor: EDER MATTHIAS
IPC: C07D295/145
Filed: 2014-10-17
Abstract: La présente invention concerne de façon générale le domaine des produits radio-pharmaceutiques et leur utilisation en médecine nucléaire comme marqueurs, agents d'imagerie et pour le traitement de divers stades du cancer de la prostate. Ainsi, la présente invention concerne des composés qui sont représentés par la formule générale (ia) ou (ib).
Patent SK-49897-A3 (SK)
Inventor: HLADKY TEODOR SR
IPC: A23L27/14
Filed: 1997-04-21
Abstract: Zmes kôprového korenia pozostáva z vysušených Častí
rastliny kôpru voňavého, ktorého podstatu tvori obsah
listových Častí, byle a nedozretých plodov, ktoré po sušení
a mletí vytvoria prísadovú zmes.
Patent SK-50099-A3 (SK)
Title: Polyolefins having greater than 5 percent 2-hydroxyethyl methacrylate grafted thereto
Inventor: WANG JAMES HONGXUE
IPC: C08F255/00
Filed: 1997-09-30
Abstract: A polyolefin, such as polyethylene or polypropylene, is modified by grafting onto the polyolefin backbone from 5 weight percent to about 30 weight percent of 2-hydroxyethyl methacrylate. Suitable polyethylene compositions for grafting include ultra high molecular weight polyethylene, high density polyethylene, ultra low density polyethylene, low density polyethylene, linear low density polyethylene and polypropylene.
Patent SK-55595-A3 (SK)
Title: Herbicidal compositions containing triazolines and method of regulation of growth of plants
Inventor: POSS KATHLEEN M
IPC: C07D249/12
Filed: 1993-10-20
Abstract: This invention relates to compositions comprising 1-aryl-4,5-dihydro-1,2,4-triazol-5(1H)-ones (triazolinones) in combination with the herbicide (2,4-dichlorophenoxy)acetic acid (2,4-D), or like substituted phenoxyalkanoic acids, or esters, or alkali metal or ammonium salts thereof; or with certain herbicidal sulfonylureas, or mixtures of these classes of compounds, to provide herbicidal compositions which are highly effective against a broad array of crop weeds, particularly broadleaf weeds, in crops such as wheat.
Patent SK-69895-A3 (SK)
Title: Shunting mechanics for perforated sheat
Inventor: BENE CARL M
IPC: B42F13/24
Filed: 1994-01-28
Abstract: A loose leaf binder mechanism has a bottom plate (2), a guide (3, 4) for turning punched sheets consisting of fixed rods and of rods movable by means of a spring-actuated pivot arm (5), and an actuating lever (10) whose actuating head (11) engages, via a guiding device, a bearing plate which projects upwards from the bottom plate (2). The actuating lever (10) further engages the pivot arm (5) by means of an actuating element (22). In order to control the movements of the actuating lever (10), at least two control cams (19, 20) for engaging at least one control cam (21) of the actuating head (11) are spaced apart on the bearing plate (9). An additional control cam (23) for determining when the actuating lever (10) is in its open position is provided on the bearing plate (9) or on the actuating head (11). The additional control cam may be integrated in the front end of the actuating head (11), in the guiding device or in the actuating element (22).
Patent SK-73398-A3 (SK)
Title: Water desalination
Inventor: GRAHAM WILLIAM
IPC: B01D65/08
Filed: 1996-12-13
Abstract: A desalination plant (10) is disclosed which includes a pump for pumping water at a pressure of between 50 and 65 Bar to a generally cylindrical filter element (30) which includes a plurality of reverse osmosis membranes defining salt passages. Immediately upstream of the filter element (30) there is a disc (40) with a plurality of holes (44) in it. The disc (40) forms an obstruction which causes a pressure drop between the upstream side thereof and the downstream side. It also divides the water flow into a series of separate streams which impinge on the end of the filter element and flow into the salt passages. The water downstream of the obstruction is not only at a lower pressure than the water upstream of the obstruction but also is flowing turbulently. The disc (40) and filter element (30) are in a cylindrical casing (12). The brine which emerges from the filter element, and which is still at a substantial pressure, can be fed through a device such as a Pelton wheel to recover some of the residual energy therefrom.
Patent SK-95499-A3 (SK)
Title: Distillation process with reduced fouling
Inventor: KRESNYAK STEVE
IPC: B01D3/32
Filed: 1998-01-14
Abstract: A method for removing a contaminant from a fluid feed stream containing the contaminant. The method includes the steps of providing a feed stream and heating it in a first step to at least partially remove some of the contaminants and recover energy from a concentrate and distillate generated. Further heating the feed stream in a second heating step in a heated separator generates a saturated vapor fraction and a concentrated liquid contaminant fraction. The vapor fraction may be compressed to generate a temperature differential in the reboiler exchanger with the vapor fraction being passed into contact with a reboiler exchanger to provide a stream of condensed vapor from the reboiler. The stream may be circulated through the reboiler exchanger and the heated separator to maintain from about 1% to about 50% by mass vapor in the stream. The apparatus includes a unique configuration of a vapor compressor, heated separator in combination with a forced circulation circuit to generate the decontamination result.
Patent CZ-364192-A3 (CZ)
Inventor: STOJAN LUBOMIR ING
IPC: C02F1/20
Filed: 1992-12-11
Abstract: Způsob úpravy pitné vody míšením, to je pitné vody, případně alespoň částečně demineralizované vody, s přírodní minerální vodou z jednoho nebo více zdrojů, zejména pro výrobu balené pitné vody stolní a kojenecké , nealkoholických nápojů a piva. Nejprve se s chemickou analýzou určí složení přírodních minerálních vod a ostatních vod míšených, vzniklá směs vody o proměnné celkové koncentraci rozpuštěných látek v rozmezí 200 až 2 000 mg/1 se provzdušňuje, filtruje, dezinfikuje, stáčí do láhví a termizu- je.
Patent CZ-106399-A3 (CZ)
Inventor: KOSAR KAREL RNDR CSC
IPC: C12C11/09
Filed: 1999-03-24
Abstract: Způsob spočívá v tom, že v bioreaktoru se na
nosič biomasy z polyesteru a/nebo polyamidu
a/nebo skleněných vláken a/nebo regenerované
celulosy a/nebo po vysterilizování horkou
vodou nebo parou sorbují mikroorganismy
a/nebo bezbuněčné preparáty a/nebo
enzymy ve formě suspenze o sušině 1 až 20 %
/hmotn./obj./ při teplotě 0É až 30° C a po
dobu 10 až 48 h, načež se k navázaným buňkám
přidá fermentovatelný substrát tvořený
mladinou a/nebo roztoky cukrů a/nebo jiných
fermentovatelných látek a vlastní
fermantace probíhá po dobu 1 až 72 h při
teplotě 0° až 40°C.
Patent CZ-142794-A3 (CZ)
Inventor: DOHANYOS MICHAL DOC ING CSC
IPC: C12S3/18
Filed: 1994-06-09
Abstract: Způsob zneškodňování organických materiálů, obsahujících
polychlorované bifenyly spočívá v tom, že na materiál,
obsahující polychlorované bifenyly se působí anaerobními
mikroorganismy, přičemž biologicky rozložitelné organické
látky se rozkládají na methan, oxid uhličitý a vodu, nerozložené
polychlorované bifenyly, přítomné ve
zpracovávaném materiálu se zachytí do anaerobně stabilizovaného
kalu, kde na ně působí anaerobní mikroorganismy
obsažené ve stabilizovaném kalu. Organické materiály, obsahující
polychlorované bifenyly jsou s výhodou přidávány
do zapracovaného systému anaerobní fermentace substrátů
jako jsou čistírenské kaly, nebo prasečí kejda. Na nerozložené
polychlorované bifenyly, zachycené a anaerobně stabilizovaném
kalu, působí anaerobními mikroorganismy
stabilizovaného kalu v dalším samostatném anaerobním reaktoru
nebo na anaerobní skládce, kde je kal deponován.
Patent CZ-150196-A3 (CZ)
Title: Detection method of yarn supply in a yarn storage and supply facility and the yarn storage and supply facility
Inventor: HUSS ROLF
IPC: B65H63/06
Filed: 1994-11-03
Abstract: In the detection of the movement of a yarn storage limit on the storage surface of a storage body of a yarn storage and feed device, different sensing properties of at least two storage-surface circumference portions offset in the circumferential direction are sensed simultaneously and are converted into non-identical storage-surface signals which are discriminated by the same sensors in relation to identical yarn signals which are formed from the sensing property of the yarn turns when the yarn store is present in the sensing zone. On a yarn storage and feed device (F) suitable for carrying out the method, there are provided first and second storage-surface circumference portions (8, 9) with sensing properties (A, B) different from one another and a plurality of sensors (SA, SB, S) which are spaced from one another approximately in the circumferential direction of the storage body (1), in such a way that at least one first storage-surface circumference portion (8) can be sensed by one sensor and simultaneously a second storage-surface circumference portion (9) can be sensed by at least one further sensor. <IMAGE>
Patent CZ-152994-A3 (CZ)
Title: Railway vehicle travel
Inventor: HANNEFORTH WOLFGANG
IPC: B61F5/30
Filed: 1994-06-21
Abstract: Running gear for railway vehicles, which, by virtue of the particular arrangement of the damping components, improves damping, permits high travel speeds and ensures that bends can be travelled through safely. This object is achieved by means of the arrangement of the vertical and horizontal shock absorbers in such a way that as a result of the horizontal shock absorber force a rotational deflection of the axle bearing housing is produced, which rotational deflection is in turn additionally damped by the vertical shock absorber, the longitudinal movements of the wheel sets being simultaneously damped by the horizontal shock absorber and the vertical shock absorber and this also applying to a lesser degree to the transverse movements of the wheel sets. The vertical shock absorber is included in the damping characteristic of the horizontal shock absorber. By changing the attachment point of the horizontal shock absorber and thus by changing the points of intersection of the median lines of the shock absorbers and the median line of the axle bearing housing in the vertical and horizontal planes by means of an attachment bracket arranged in a defined manner it is possible to vary the damping ratio of the shock absorbers. The invention is suitable in particular for sets of running gear which are to be used for high speed transport. <IMAGE>
Patent CZ-153399-A3 (CZ)
Title: Polyolefins and their functionalized derivatives
Inventor: RATH HANS P
IPC: C10L1/2387
Filed: 1997-11-03
Abstract: PCT No. PCT/EP97/06068 Sec. 371 Date Jul. 27, 1999 Sec. 102(e) Date Jul. 27, 1999 PCT Filed Nov. 3, 1997 PCT Pub. No. WO98/20053 PCT Pub. Date May 14, 1998The present invention relates to at least simply unsaturated polyolefins with a number mean molecular weight in the range of 400 to 1,500 dalton and a dispersibility of MW/MN<1.2, obtained through catalytic dimerization from at least simply unsaturated olefin-oligomers, as well as to the method for their production. The present invention further relates to derivatives of these polyolefins which can be obtained by functionalizing at least a double link of the polyolefin. The invention also relates to the use of polyolefins and/or functionalization products as additives for fuels or lubricants.
Patent CZ-159796-A3 (CZ)
Title: Process of fermentation industrial production of enzyme preparation phytase
Inventor: VOLFOVA OLGA RNDR DRSC
IPC: C12N1/14
Filed: 1996-05-31
Abstract: This method of producing a phytase enzyme preparation by industrial fermentation through the submerged cultivation of an Aspergillus strain on a medium containing starch with a growth limitation with phosphorus, consisting of the submerged cultivation of the strain of the Aspergillius niger 921 CCF 2951 at a temperature of 25-27 degrees C, at a pH of 2.0 to 6.0, particularly 2.5 to 3.5, with aeration and agitation providing an oxygen concentration of 10-99% of the coefficient of the dissolubility of the gases, mainly of 20-60%, with the subsequent separation of the fungal mycelium, dialysis and ultrafiltration of the supernatant and lyophilisation of the concentrated solution of enzymes.
Patent CZ-181993-A3 (CZ)
Title: Contact adhesive responsive to pressure and hand-tearable adhesive tapes produced by means of such contact adhesive for embroidery and textile industries
Inventor: GRABEMANN JUERGEN
IPC: B32B7/12
Filed: 1993-09-02
Abstract: Pressure-sensitive contact adhesive which is characterised in that it contains a mixture of   A) from 0 to 90% by weight of acrylate-vinyl acetate-acrylic acid copolymer having 2 to 8 carbon atoms in the alcohol component of the acrylate and, based on the copolymer, from 10 to 60% by weight of vinyl acetate and from 1 to 10% by weight of acrylic acid (Fikentscher K value in the range from 50 to 110, measured in accordance with DIN 51562 in tetrahydrofuran), B) from 10 to 80% by weight of acrylate-acrylic acid-N-methylolmethacrylamide copolymer having 4 to 8 carbon atoms in the alcohol component of the acrylate and, based on the copolymer, from 1 to 10% by weight of acrylic acid and from 1 to 10% by weight of self-crosslinking N-methylolmethacrylamide (Fikentscher K value in the range from 70 to 130, measured in accordance with DIN 51562 in tetrahydrofuran), C) from 0 to 90% by weight of acrylate-ethyl acrylate-N-methylolmethacrylamide-acrylic acid copolymer having 4 to 8 carbon atoms in the alcohol component of the acrylate and, based on the copolymer, from 1 to 10% by weight of acrylic acid and from 1 to 10% by weight of self-crosslinking N-methylolmethacrylamide and from 20 to 80% by weight of ethyl acrylate (Fikentscher K value in the range from 80 to 130, measured in accordance with DIN 51562 in tetrahydrofuran), D) from 0 to 25% by weight of phthalic esters (phthalates) having 2 to 12 carbon atoms in the alcohol component of the ester, where at least one of components A) and C) is present in addition to component B). It is suitable for the production of manually tearable contact adhesive tapes for the embroidery and textile industries.
Patent CZ-200058-A3 (CZ)
Title: Epothilone derivatives
Inventor: VITE GREGORY D
IPC: C07D277/26
Filed: 1998-06-16
Abstract: The present invention relates to compounds of the formula
         Q is selected from the group consisting of
         G is selected from the group consisting of alkyl, substituted alkvl, substituted or unsubstituted aryl, heterocyclo,
         W is O or NR 15 ; 
   X is O or H,H; 
   Y is selected from the group consisting of O; H,OR 16 ; OR 17 ,OR 17 ; NOR 18 ; H,NOR 19 ; H,NR 20 R 21 ; H,H; or CHR 22 ; OR 17  OR 17  can be a cyclic ketal; 
   Z 1 , and Z 2  are selected from the group consisting of CH 2 , O, NR 23 , S, or SO 2 , wherein only one of Z and Z 2  is a heteroatom; 
   B 1  and B 2  are selected from the group consisting of OR 24 , or OCOR 25 , or O 2 CNR 26 R 27 ; when B 1  is H and Y is OH, H they can form a six-membered ring ketal or acetal; 
   D is selected from the group consisting of NR 28 R 29 , NR 30 COR 31  or saturated heterocycle    R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , R 7 , R 13 , R 14 , R 18 , R 19 , R 20 , R 21 , R 22 , R 26 , and R 27  are selected from the group H, alkyl, substituted alkyl, or aryl and when R 1  and R 2  are alkyl can be joined to form a cycloalkyl; R 3  and R 4  are alkyl can be joined to form a cycloalkyl; 
   R 9 , R 10 , R 16 , R 17 , R 24 , R 25 , and R 31  are selected from the group H, alkyl, or substituted alkyl; 
   R 8 , R 11 , R 12 , R 28 , R 30 , R 32 , R 33 , and R 30  are selected from the group consisting of H, alkyl, substituted alkyl, aryl, substituted aryl, cycloalkyl, or heterocyclo; 
   R 15 , R 23  and R 29  are selected from the group consisting of H, alkyl, substituted alkyl, aryl, substituted aryl, cycloalkyl, heterocyclo, R 32 C=O, R 33 SO 2 , hydroxy, O-alkyl or O-substituted alkyl, the pharmaceutically acceptable salts thereof and any hydrates, solvates or geometric, optical and stereoisomers thereof, with the proviso that compounds wherein 
   W and X are both O; and 
   R 1 , R 2 , R 7 , are H; and 
   R 3 , R 4 , R 6 , are methyl; and 
   R 8 , is H or methyl; and 
   Z 1 , and Z 2 , are CH 2 ; and 
   G is 1-methyl-2-(substituted-4-thiazolyl)ethenyl; and 
   Q is as defined above 
are excluded.
Patent CZ-200441-A3 (CZ)
Title: Structure-based medicament design methods for identifying D-Ala-D-Ala ligase inhibitors as antibacterial medicaments
Inventor: NAVIA MANUEL
IPC: C12N9/00
Filed: 2002-06-28
Abstract: The invention is based on the discovery that certain small molecules can bind to the ATP binding site of D-Ala-D-Ala ligase, even in the absence of the enzyme's substrate, and can cause a conformational change in the enzyme structure similar to that which occurs upon binding of ATP and substrate to the enzyme. Without wishing to be bound by any theory, it is believed that such a conformational change is required for either activation or inhibition of the enzyme. The information obtained from this discovery has enabled identification of key interactions in the active site of the enzyme, as well as the design and opimization of inhibitors.
Patent CZ-211399-A3 (CZ)
Title: 1-Phenylalkyl-1,2,3,6-tetrahydropyridines for treating Alzheimer's disease
Inventor: BARONI MARCO
IPC: A61K31/444
Filed: 1997-12-12
Abstract: PCT No. PCT/FR97/02286 Sec. 371 Date Jul. 27, 1999 Sec. 102(e) Date Jul. 27, 1999 PCT Filed Dec. 12, 1997 PCT Pub. No. WO98/25903 PCT Pub. Date Jun. 18, 1998The invention relates to compounds of the formula in which: Y is -CH- or -N-; R1 is hydrogen, a halogen or a CF3, (C1-C4)alkyl or (C1-C4)alkoxy group; R2 is a methyl or ethyl group; R3 and R4 are each hydrogen or a (C1-C3)alkyl; and X is: (a) a (C1-C6)alkyl, a (C1-C6)alkoxy, a (C3-C7)carboxyalkyl, a (C1-C4)alkoxy-carbonyl(C1-C6)alkyl, a (C3-C7)carboxyalkoxy or a (C1-C4)alkoxycarbonyl-(C1-C6)alkoxy; (b) a radical selected from (C3-C7)cycloalkyl, (C3-C7)cycloalkoxy, (C3-C7)-cycloalkylmethyl, (C3-C7)cycloalkylamino and cyclohexenyl, it being possible for said radical to be substituted by a halogen, hydroxyl, (C1-C4)-alkoxy, carboxyl, (C1-C4)alkoxycarbonyl, amino or mono- or di-(C1-C4)-alkylamino; or (c) a group selected from a phenyl, phenoxy, phenylamino, N-(C1-C3)alkyl-phenylamino, phenylmethyl, phenylethyl, phenylcarbonyl, phenylthio, phenylsulfonyl, phenylsulfinyl and styryl, it being possible for said group to be monosubstituted or polysubstituted on the phenyl group by a halogen, CF3, (C1-C4)alkyl, (C1-C4)alkoxy, cyano, amino, mono- or di-(C1-C4)alkyl-amino, (C1-C4)acylamino, carboxyl, (C1-C4)alkoxycarbonyl, aminocarbonyl, mono- or di-(C1-C4)alkylaminocarbonyl, amino(C1-C4)alkyl, hydroxy(C1-C4)alkyl or halogeno(C1-C4)alkyl; to a method of preparing them and to the pharmaceutical compositions containing them. These compounds have neurotrophic and neuroprotective activity.
Patent CZ-245294-A3 (CZ)
Title: Process of treating railway bed and apparatus for making the same
Inventor: NEMEC BRONISLAV ING
IPC: E01B27/06
Filed: 1994-10-05
Abstract: At first, the original ballast is excavated in the excavating section from the track bed, whereby it is transported out of the excavating section or the excavated original ballast of the track bed is led into the cleaning section, where it is cleaned and after it has been cleaned the cleaned original ballast is transported back into the excavating section, into which reinforcing material is introduced for inserting the reinforcing layer. The power supply section and the excavating section are connected with the cleaning section to create a machine for cleaning of the whole cross-section of the original ballast from the track bed and a machine for increasing the load capacity of the sleeper subsoil using cleaned original ballast.
Patent CZ-255497-A3 (CZ)
Title: Process for preparing genome of recombinant adenoviruses
Inventor: CROUZET JOEL
IPC: C12N15/09
Filed: 1996-02-09
Abstract: A novel method for preparing recombinant adenoviruses and the use of such adenoviruses in gene therapy are disclosed. Plasmids used in the construction of said adenoviruses are also disclosed.
Patent CZ-259398-A3 (CZ)
Title: Safety circuit arrangement
Inventor: BRITZ WOLFGANG
IPC: F01D21/18
Filed: 1997-01-17
Abstract: The invention relates to a safety circuit for controlling a hydraulic drive (10) with a drive part (12) movable in at least two different directions of movement and controllable for any movement  by a control switching circuit. A safety circuit which ensures the required safety function in an absolutely safe manner, even in the event of a power failure, is obtained in that at least one safety switching circuit is hydraulically combined with the control switching circuit in such a manner that when the latter is switched off the drive part (12) can only be controlled by the respective safety switching circuit. Consequently, the highest-priority operation provided in an emergency, for example in the form of the defined closing or opening of a vapour control valve, is safely executed and the otherwise usual control process is interrupted by the control switching circuit.
Patent CZ-296798-A3 (CZ)
Title: Sealing device and steam turbine
Inventor: REMBERG AXEL
IPC: F01D11/02
Filed: 1997-05-12
Abstract: The invention relates to a seal arrangement (18) to seal off a first area (19) from a second area (20). Fluid (17) can flow through each area (19, 20) the pressure of which can be maintained on a different level. The seal arrangement comprises a rotary component (12, 10) rotating about a main axis (14) and a stationary component (11, 13). One of the components (12, 13) comprises a recess (16a, 16b) running in the direction of the periphery and the other component (11, 10) an end piece (5). Adjoining to the end piece (5) follows a sealing web (6) with a crosswise arranged area (8) running essentially parallel to the main axis (14) at a distance from the end piece (5), which protrudes radially into the recess (16a, 16b) with the recess (16a, 16b) being geometrically similar to the sealing web (6).
Patent CZ-312399-A3 (CZ)
Title: Apparatus for testing urine
Inventor: DAVARZAN HAMID
IPC: C12Q1/04
Filed: 1997-03-05
Abstract: The present invention concerns a device for testing resistance in microorganisms present in e.g. urine. The device comprises a cylindric container (1) fitted with a spout (3) of a considerably lesser diameter and a plunger (2) making a tight seal against the wall of the container (1), having a radially extending gasket (6) and being partly coated with nutrients for growing microorganisms, the coated part being arranged at the front part of the plunger (2) and comprising at least three angularly arranged test laminate (4A, 4B, 4C), at least one of which is coated with nutrients and antibiotics of different kinds and concentrations. The lower end surface (Ä) of the container (1) is conically shaped with a peak turning into the spout (3) preventing urine from remaining on the surface (Ä) when the container (1) is emptied after the laminae (4A, 4B, 4C) have been wetted with urine and before the device is incubated.
Patent CZ-325194-A3 (CZ)
Title: Switch with rotary control contacts
Inventor: SINTHOMEZ DANIEL
IPC: H01H71/04
Filed: 1993-04-20
Abstract: The on (14) and off (13) buttons are mounted pivotably in the casing of the circuit breaker and exhibit, in the front projection, a difference in height (h) of their lower ends (20b, 20b'). Their upper ends (20a, 20a') alternately uncover and cover display elements (32, 32') provided on the anterior face (17) of the casing. <IMAGE>