baber/WOPTO huggingface dataset:
Patent CY-1124874-T1 (CY)
Title: Διεργασια για την παρασκευη [(5-(3-χλωροφαινυλ)-3-υδροξυπυριδινο-2-καρβονυλ)-αμινο]οξικου οξεος απο 5-((3-χλωροφαινυλ)-3-χλωρο-πυριδιν-2-υλ)-νιτριλιο, και διεργασια για την παρασκευη παραγωγων 5-((αλογονοφαινυλ)-3-αλογονο-πυριδιν-2-υλ)-νιτριλιου
Inventor: LANTHIER CHRISTOPHER M
IPC: C07D213/81
Filed: 2021-12-08
Abstract: Μια διεργασία για την παρασκευή της ένωσης (5):
Patent HR-P20090439-T1 (HR)
Inventor: BRANDT SVEN F A VAN
IPC: C07D403/12
Filed: 2009-08-13
Abstract: Spoj formule (I), N-oksidnog oblika, njegove farmaceutski prihvatljive adicijske soli i njegovi stereokemijski izomerni oblici, naznačen time, dasvaki X je nezavisno N ili CH; R1 je fenil, naftalenil ili heterociklil; gdjesvaki od navedenih fenila ili naftalenila je ponekad supstituiran sa jednim ili dva supstituenta svaki nezavisno izabran među halo, C1-6alkila, C1-6alkiloksi, polihaloC1-6alkila, arila, hidroksi, cijano, amino, C1-6alkilkarbonilamino, C1-6alkilsulfonilamino, hidroksikarbonila, C1-6alkiloksikarbonila, hidroksiC1-6alkila, C1-6alkiloksimetila, aminometila, C1-6alkilaminometila, C1-6alkilkarbonilaminometila, C1-6alkilsulfonilaminometila, aminosulfonila, C1-6alkilaminosulfonila ili heterociklila; R2 je vodik, -CH2-R5, trifulorometil, -C(=O)-R6 ili -CH2-NR7R8; gdje svaki R5 je nezavisno izabran iz vodika, hidroksi, C1-6alkoksi, C1-6alkiloksiC1-6alkiloksi, C1-6alkilkarboniloksi, piperazinila, N-metilpiperazinila, morfolinila, tiomorfolinila, imidazolila ili triazolila; svaki R6 je nezavisno izabran među hidroksi, C1-6alkiloksi, amino ili mono- ili di(C1-6alkil)amino, C1-6cikloalkilamino, hidroksiC1-6alkilamino, piperazinila, mono- ili di(C1-6alkil)aminoC1-6alkilamino N-metilpiperazinila, morfolinila ili tiomorfolinila; svaki R7 i R8 su nezavisno izabrani među vodika, C1-6alkila, C1-6alkilkarbonila, C1-6alkilsulfonila ili mono- ili di(C1-4alkil)aminosulfonila; R3 je vodik, hidroksimetil, aminometil ili mono- ili di(C1-6alkil)aminometil; R4 je vodik ili C1-6alkil; aril u gore navedenom je fenil ili naftalenil; gdjesvaki navedeni fenil ili naftalenil je ponekad supstituiran sa jednim ili dva supstituenta svaki neovisno izabran među halo, C1-6alkila, C1-6alkoksi, trifluorometila, cijano ili hidroksikarbonila; igore navedeni heterociklil je furanil, tienil, pirolil, pirolinil, pirolidinil, dioksolil, oksazolil, tiazolil, imidazolil, imidazolidinil, pirazolil, pirazolinil, pirazolidinil, izoksazolil, izotiazolil, oksadiazolil, triazolil, tiadiazolil, piranil, piridinil, piperidinil, dioksanil, morfolinil, ditianil, tiomorfolinil, piradizinil, pirimidinil, pirazinil, piperazinil, triazinil, tritianil, indolizinil, indolil, indolinil, benzofuranil, benzotifenil, indazolil, benzimidazolil, bentatiazolil, purinil, kinolizinil, kinolinil, cinolinil, ftlazinil, kinazolinil, kinoksalinil ili naftiridinil; gdjesvaki navedeni heterocikal je ponekad supstituiran sa jednim ili više supstituenata, te je svaki nezavisno izabran među halo, C1-6alkila, C1-6alkoksi, C1-6alkiloksi, cijano, amino, mono- ili di(C1-4alkil)amino. Patent sadrži još 11 patentnih zahtjeva.
Patent SI-1400245-T1 (SI)
Title: Boronic acid salts useful in parenteral formulations for selective thrombin inhibition
Inventor: MADGE DAVID JONATHAN
IPC: A61K31/00
Filed: 2003-09-09
Abstract: A pharmaceutical formulation adapted for oral administration, whether directly or after combining with a liquid, and comprising 
a) a first species selected from (a) boronic acids of formula (I), (b) boronate anions thereof, and (c) any equilibrium form of the aforegoing (e.g. an anhydride); and 
(b) a second species selected from the group consisting of pharmaceutically acceptable metal ions.  Formula (I) comprises specified peptidyl boronic acids having anti-thrombotic activity and the formulations are useful for the treatment of thrombosis. An exemplary boronic acid is Cbz-(R)-Phe-(S)-Pro-(R)-Mpg-B(OH) 2 .
Patent SI-1689356-T1 (SI)
Title: Topical compositions associating sodium hyaluronate fragments and retinoid
Inventor: SAURAT JEAN-HILAIRE
IPC: A61K8/00
Filed: 2005-01-27
Abstract: Topical composition (A), contains as active ingredient, one or more fragments (I) of hyaluronate with molecular weight 50-750 kD. ACTIVITY : Dermatological. MECHANISM OF ACTION : (I) increases the number of proliferating cells, particularly fibroblasts, in the epidermis and dermis, so induce epidermal thickening. A standard cosmetic vehicle contained 0.2 % hyaluronate fragments of molecular weight 50-250 kD and was applied twice daily to the skin of SKH1 hairless mice. After an unspecified treatment time, epidermal thickness and the number of proliferating cells were determined. The mean thickness was 0.32 mm (compare 0.07 mm in controls) and the number of cells (per microscope field) was 257 compared with 96 in controls. Also the mean number of proliferating cells (positive for the marker Ki67; per field) was 96 in the epidermis and 5 in the dermis; compare 26 and 0.95 in controls.
Patent SI-1693293-T1 (SI)
Title: Transmission system
Inventor: MARCACCI MAURIZIO
IPC: B62M7/00
Filed: 2006-02-02
Abstract: The present invention relates to a transmission system (100) for a vehicle of the type equipped with an engine group (1), constrained by fixing means to the chassis (5) of the vehicle, a transmission pinion (2) which transfers the movement to the back wheel (27) and a transfer group of the engine torque between the engine group (1) and the pinion (2). The transfer group (3) comprises two articulations (14,15) of which the first is functionally connected to the engine group (1) and the second is functionally connected to the pinion (2) .
Patent SI-1857368-T1 (SI)
Title: Automatic machine and method for the packaging of a series of editorial products in plastic film
Inventor: BALLESTRAZZI ARIS
IPC: B65B61/00
Filed: 2007-05-03
Abstract: An automatic machine for the packaging of a series of editorial products in plastic film comprising feeding means of editorial products (11, 11') and a packaging station (20) equipped with a mechanical conformer (21) for the winding of the film (12) around the products (11, 11') and means for the closing of the same, also comprising two pusher conveyors (14, 16) alongside each other for the feeding of a first product (11) and at least a second product (11') respectively, to the packaging station (20), which comprises at least one longitudinal closing device (23) and a transversal welding station (25) for the formation of a packaging (100), the packaging (100) comprising two closed and separate bags (101) for the first product (11) and the second product (11') respectively.
Patent SI-2003130-T1 (SI)
Title: Novel pyridine derivative having anti-helicobacter pylori activity
Inventor: ITO MASAHARU
IPC: A61K31/00
Filed: 2007-03-07
Abstract: The obj ect is to provide an excellent pharmaceutical having an anti-Helicobacter pylori activity. Disclosed is a novel pyridine derivative represented by the following general formula (I):   
wherein R represents a linear or branched hydroxyalkyl group having 5 to 10 carbon atoms, or a pharmaceutically acceptable salt thereof, which has a potent antibacterial activity against  H. pyroli  ( Helicobacter pyroli ). Examples of the disease which can be prevented/treated by administration of a pharmaceutical agent comprising the compound include gastritis, gastric ulcer, duodenal ulcer, gastric MALT lymphoma, gastric hyperplastic polyp, development of gastric cancer after endoscopic resection of the early stage of gastric cancer and the like.
Patent TR-200100593-T1 (TR)
Title: Bir motorlu araçta bir kampana fren için bir otomatik açıklık dengeleyicisi
Inventor: ANDREIS MARCO DE
IPC: F16D65/56
Filed: 2000-06-27
Abstract: Bir açiklik dengeleyicisinde, bir çubuk (12) fren pabuçlarinin birisine sabitlenir ve diger pabuca bagli olan baska bir çubuga (11) vidalanarak geçen bir ara elemanda (13) kayabilir. Bir isiya karsi hassas metal serit (18), çubugu (12) ara elemandan (13)  uzaga itmek üzere çalisan bir yaprak yaydan (14) çikinti yapar. Çift metal serit (18) ara elemana (13) sabitlenen bir mandal çarkina (17) büyük ölçüde teget sekilde yönlendirilir; serbest ucunda , çift metal serit (18) mandal çarkina (17) geçen bir durak elemanina (18a) sahiptir. Önceden belirlenmis bir degerin üzerindeki sicakliklarda, serit (18) durak elemaninin (18a) çarktan (17) çiktigi bir isidan kaynaklanan bükülme konumuna gelir.
Patent DE-3687551-T2 (DE)
Inventor: JANSKI ALVIN M
IPC: A61K9/22
Filed: 1986-07-15
Granted: 1993-05-13
Abstract: The present invention provides improved controlled release implants for subcutaneous administration to an animal of a growth promoting amount of a recombinant protein having growth hormone activity, characterised in that said protein is present in a form having a salt content of less than 5% by weight based on the weight of said protein.
Patent DE-3783185-T2 (DE)
Inventor: BOUJU MARIE-CHRISTINE
IPC: C11D1/90
Filed: 1987-09-07
Granted: 1993-07-01
Abstract: A thickened acidic aqueous composition, containing a betaine of formula: <IMAGE> in which R is a C9-C17 alkyl or alkenyl radical, x and y are independent of each other and are integers between 0 and 5 inclusive,  as well as:  at least one weak acid,  at least one salt,  optionally perfume,  optionally a bactericide,  optionally a colorant,  water. Application to the cleaning of sanitaryware.
Patent DE-3850672-T2 (DE)
Inventor: BUCKNELL JOHN WENTWORTH
IPC: B25B29/02
Filed: 1988-09-29
Granted: 1995-03-02
Abstract: PCT No. PCT/AU88/00381 Sec. 371 Date May 7, 1990 Sec. 102(e) Date May 7, 1990 PCT Filed Sep. 29, 1988 PCT Pub. No. WO89/02807 PCT Pub. Date Apr. 6, 1989.A hydraulic nut (20) for tensioning a bolt (232) is disclosed having a stepped annular piston (22) slidable within a housing (21) for reducing the complexity of manufacture. The locking collar (27) is threaded to the housing (21) on a buttress thread (28) to minimize distortion due to thread loads and locks against the piston (22) instead of the clamped article for minimizing tensile relaxation during transfer of load from the hydraulic tensioner to the locking collar (27).
Patent DE-3876336-T2 (DE)
Inventor: DENIS ASCOT
IPC: C10N10/04
Filed: 1988-02-19
Granted: 1993-06-17
Abstract: Oil based compositions are disclosed which are comprised of oil having a multi-functional additive component therein. The additive component is present in sufficient amounts so as to provide improved performance characteristics to the composition such as water tolerance and antiwear characteristics. The additive is a compound represented by the general structural formula (I):   <IMAGE> (I) wherein R is a hydrocarbyl, preferably iso-stearyl, R1, R2, and R3 are independently hydrogen or alkyl, preferably hydrogen, n is 1 to 20, preferably 5, and X is a cation, preferably Ca. Overbased and mixed salts of the additive compound are also disclosed. The additive is an effective EP agent, water tolerance fix in a variety of functional fluids and lubricating compositions.
Patent DE-3878571-T2 (DE)
Inventor: WACHI SHIGEAKI C O PATENTS DIV
IPC: G11B33/10
Filed: 1988-03-28
Granted: 1993-08-05
Abstract: An optical disc recording and reproducing apparatus includes a servo circuit (1 to 7) incorporating an element (3) which has high response characteristics to run out frequency. An output of the element (3) is monitored by a defective disc detecting circuit (8).
Patent DE-3886762-T2 (DE)
Inventor: SUMNER CHARLES
IPC: C07C59/64
Filed: 1988-10-05
Granted: 1994-07-28
Abstract: Alkylene or dialkyl ketal of an alpha-acetyl cinnamic acid or ester therof are obtained by reacting alpha-acetyl cinnamic acid or an ester thereof with a ketalizing agent selected from the group consisting of alkyl glycols, dialkyl detals and trialkyl orthoesters in the presence of the transition metal catalyst and an acid catalyst. Also, alkyl alpha-enol ethers of alpha-acetyl cinnamic acid are obtained by heating the alkylene or dialkyl ketals.
Patent DE-3889463-T2 (DE)
Inventor: BARMAN ROLF
IPC: A46D3/00
Filed: 1988-12-13
Granted: 1994-08-18
Abstract: PCT No. PCT/NO88/00091 Sec. 371 Date Aug. 21, 1990 Sec. 102(e) Date Aug. 21, 1990 PCT Filed Dec. 13, 1988 PCT Pub. No. WO90/06701 PCT Pub. Date Jun. 28, 1990.A process for producing a toothbrush produced thereby have the cavities (11, 12) arranged on the back side of the tooth brush head. The longitudinal axes (14a, 15a) for angling the head portions (13, 14, 15) relative to each other are arranged on or at the bristle-carrying side of the head portion directly opposite the associated cavity (11, 12). A blank for carrying out the process and a toothbrush produced thereby have the cavities (11, 12) arranged on the back side of the toothbrush head. The longitudinal axes (14a, 15a) for angling the head portions (13, 14, 15) relative to each other are arranged on or at the bristle-carrying side of the head portion directly opposite the associated cavity (11, 12).
Patent TR-199801874-T2 (TR)
Inventor: DICKENS R ROBERT
IPC: C03B35/26
Filed: 1997-03-05
Abstract: Kenarli cam esya üzerinde dekoratif model olusturma aparati (10) ayakli (64) bir kaide (60), mil monte edici ayak (68),sekil verici alet (150), harekete geçirici ve kontrol edici araç içerir. Harekete geçirici ve kontrol edici araç ayak baglama levhasi (72) üzerine monte edilmis el topuzuna (76) sahip dikey bir saft kanali (74) içerir. Buda (74) dikey saft (78) içerir. Mengene blok (80), bir mil düzenegiyle (82) dikey saft (78) üzerine monte edilir. Yatay saft (88) birinci uç (90) ile ikinci  uç (92) içerir. Yatay el çarki (96), yatay saftla (88) baglantilidir. Saft (88) ile mengene blogun (80) ilgili hareketi ölçme aletinde (100) belirtilir. Hava akimi karsilik gelen hava girisinde (138) hava ile çalisan kontrol valfiyle (120) düzenlenir; egzos hava girisiyle baglantilidir. Dekoratif model olusturma aleti (104) geri silindirle (200) harekete ettirilebilen bir izleme aksami (174) içerir.
Patent TR-199901510-T2 (TR)
Inventor: KARPPANEN HEIKKI OLAVI
IPC: A23L13/40
Filed: 1997-12-17
Abstract: Bitki sterolleri ve/veya stanolleri veya bunlarin türevleri ile magnezyum, kalsiyum ve potasyum minerallerinden bir veya birden fazlasinin seviyesinin yükseltilmesini içeren gida lezzetlendiricileri, gida malzemeleri ve gida ürünleri hazirlama metodu gösterilmektedir. Bahsi geçen bilesim içeren verilen gidanin alimi sonucu kolestrol ve tansiyonda önemli bir azalma görülmektedir. Bu azalma bitki sterollerinin ve minerallerin beklenilen toplam etkisinden daha fazladir. Ayni zamanda, gidalarin hazirlanmasinda kullanilan, bahsi geçen özellikler tasiyan gida lezzetlendiricileri tarif edilmektedir.
Patent TR-199901645-T2 (TR)
Inventor: LYNDA KAYE JOHNS N
IPC: C07C251/08
Filed: 1998-01-13
Abstract: Selected olefins such as ethylene and  alpha -olefins are polymerized by nickel [II] complexes of certain monoanionic ligands. The polyolefins are useful in many applications such as molding resins, film, fibers and others. Also described are many novel nickel compounds and their precursors, as well as novel ligands.
Patent DE-60002343-T2 (DE)
Inventor: EMCH J
IPC: B05D3/02
Filed: 2000-05-15
Granted: 2004-03-04
Abstract: Processes for coating metal or polymeric substrates are provided which include the steps of: (a) applying a liquid basecoating composition to a surface of the substrate; (b) exposing the basecoating composition to air having a temperature ranging from about 10° C. to about 50° C. for a period of at least about 5 minutes to volatilize at least a portion of volatile material from the liquid basecoating composition, the velocity of the air at a surface of the basecoating composition being less than about 0.5 meters per second; (c) applying infrared radiation and hot air simultaneously to the basecoating composition for a period of at least about 2 minutes, the velocity of the air at the surface of the basecoating composition being less than about 4 meters per second, the temperature of the metal substrate being increased at a rate ranging from about 0.4° C. per second to about 1.2° C. per second to achieve a peak substrate temperature ranging from about 120° C. to about 165° C., such that a dried basecoat is formed upon the surface of the substrate; and (d) applying a powder topcoating composition over the dried basecoat.
Patent DE-60002448-T2 (DE)
Inventor: GURNY ROBERT
IPC: A61K9/00
Filed: 2000-05-26
Granted: 2004-03-25
Abstract: The aqueous ophthalmic formulation for the treatment and prevention of infections contains ofloxacin as active ingredient and a chitosan having a weight average molecular weight of 500,000 - 5,000,000 Daltons and a deacetylation degree of 30 - 90 % as solubilizing agent of ofloxacin. Chitosan having a deacetylation degree of 30 - 90 % may be also used for solubilizing ofloxacin suspended in an aqueous media having a substantially neutral pH in any other applications.
Patent DE-60009774-T2 (DE)
Inventor: BARBEY JEAN-PIERRE
IPC: H04L29/12
Filed: 2000-02-10
Granted: 2004-09-23
Abstract: The supplementary machine network connection technique has a machine (M4) in a network of addressable machines (M1,M2,M3) and having input ports connected to the addressable machines. Each supplementary machine port has an address (A1,A2,A3) which represents an address designating the machine but not the machine to which the port is connected.
Patent DE-60014525-T2 (DE)
Inventor: KAKEHI T
IPC: B60R13/02
Filed: 2000-07-27
Granted: 2006-02-02
Abstract: To provide a method for bonding a plastic clip onto a natural fiber based porous member and a plastic clip for use in the bonding method that the clip can be bonded with a low energy without any of heat affection and any dent on a rear side of the clip, and the excessive molten portions will be handled well.  A plastic clip 1 comprises a base 5 having a bonding side including a welding region 6 and a non-welding region 7. The welding region 6 includes a plurality of fusible projections 9 extending to the natural fiber based porous member and a plurality of recesses 10 adjacent the projections for receiving the excessive molten portions of the projections. The non-welding region 7 is formed with a reference level portion 11 to set the welding height of the plastic clip.  <IMAGE>
Patent DE-60015283-T2 (DE)
Inventor: PATIL MANOJ
IPC: H04W4/14
Filed: 2000-11-27
Granted: 2005-10-27
Abstract: A wireless station user 10 is provided with a unified messaging protocol that enhances the currently available messaging capabilities of SMS. The user is provided with the capability to compose at least one distribution list for SMS messages. The list can be stored in a memory 24, 29 of the station, or in a message server 40. The user is also provided with the capability to send messages to at least one distribution list on a user determined, periodic basis. The user is further provided with the capability to obtaining content from an external source 60, to composing an SMS incorporating the content, and send the SMS to recipients 70 defined in the distribution list. <IMAGE>
Patent DE-60026743-T2 (DE)
Inventor: KNOPP MICHAEL V
IPC: A61K49/00
Filed: 2000-12-21
Granted: 2006-08-17
Abstract: This invention relates to the use of particular contrast agents to prepare diagostic compounds suitable for non-invasive visualisation under physiological conditions of the intestinal tract, and the colon in particular.
Patent DE-60026838-T2 (DE)
Inventor: BELLWOOD ALEXANDER
IPC: H04L29/08
Filed: 2000-06-28
Granted: 2006-09-07
Abstract: A method of enabling a proxy to participate in a secure communication between a client and a set of servers. The method begins by establishing a first secure session between the client and the proxy. Upon verifying the first secure session, the method continues by establishing a second secure session between the client and the proxy. In the second secure session, the client requests the proxy to act as a conduit to a first server. Thereafter, the client and the first server negotiate a first session master secret. Using the first secure session, this first session master secret is then provided by the client to the proxy to enable the proxy to participate in secure communications between the client and the first server. After receiving the first session master secret, the proxy generates cryptographic information that enables it to provide a given service (e.g., transcoding) on the client's behalf and without the first server's knowledge or participation. If data from a second server is required during the processing of a given client request to the first server, the proxy issues a request to the client to tunnel back through the proxy to the second server using the same protocol.
Patent DE-60029138-T2 (DE)
Inventor: LIPSON KEN
IPC: A61P11/00
Filed: 2000-12-22
Granted: 2007-06-06
Abstract: The present invention concerns compounds and their use to inhibit the activity of a receptor tyrosine kinase. The invention is preferably used to treat cell proliferative disorders such as cancers characterized by over-activity or inappropriate activity c-kit kinase.
Patent DE-60029606-T2 (DE)
Inventor: UPTON M
IPC: C12M3/00
Filed: 2000-09-22
Granted: 2007-07-12
Abstract: The present invention relates to culturing devices that are compact, utilize small amounts of cell culture media to establish and maintain cell cultures, and produce a large number of cells in a short period of time when compared to other cell culturing devices and techniques. Such devices are useful in the culture of all cell types, but are particularly useful in the culture of cells that are known in the art to be difficult to culture, including cells that lose one or more of their particular attributes/characteristics (e.g., pluripotentiality), or cells that are difficult to establish cultures of (e.g. primary cells), during culturing in traditional cell culture devices.
Patent DE-60031304-T2 (DE)
Inventor: ROSE G
IPC: G06F21/33
Filed: 2000-12-21
Granted: 2007-05-24
Abstract: A method of authenticating anonymous users while reducing potential for "middleman" fraud includes the step of constructing a puzzle in response to information received from a software user. The puzzle includes the received information. The puzzle is sent to the user by a software provider. The user solves the puzzle and returns the solution to the provider. The puzzle includes a portion of a value derived from an encrypted "cookie" and an exponentiation of the derived value. The cookie includes information about the user.
Patent DE-60034466-T2 (DE)
Inventor: WILLIAMS PETER C
IPC: F16L19/06
Filed: 2000-09-12
Granted: 2008-01-03
Abstract: An intrinsic gauging device for a ferrule type tube fitting (10) of the type having a coupling nut (14), a coupling body (12) and at least one ferrule (32), includes a precisely formed marking on the coupling body that is visually perceptible when the coupling is in a finger tight position, and that is covered or visually imperceptible or otherwise has a predetermined relationship with the coupling nut when the fitting has been initially pulled-up. In a preferred form, the marking is realized as a precision groove (50) or recess machined into a surface of the coupling body. The groove can be made more easily visually perceptible such as by roughening or knurling the surface, or coloring the surface, for example. The groove defines an edge (50b) at a precise position that corresponds to a predetermined axial displacement of the nut relative to the body for initial pull-up. The marking may also be formed with a precise dimension such as an axial length to provide a second edge that corresponds to a predetermined axial displacement of the nut relative to the body beyond initial pull-up for fitting assemblies that are remade.
Patent DE-60102694-T2 (DE)
Inventor: MARTY EMMANUEL
IPC: G06F9/44
Filed: 2001-06-14
Granted: 2005-03-31
Abstract: The method identifies required functionalities in an initial phase and then creates components which fulfill the associated functionality using computer means. Each component is declared in relation to a system loading component and loading is assisted. The architecture is dynamic and a component (31) may be replaced (32) by a component giving the same functionality without changing any other component in the system.