baber/WOPTO huggingface dataset:
Patent IE-840054-L (IE)
Title: Compounds
IPC: C07D295/08
Filed: 1984-01-12
Abstract: This invention relates to compounds of the formula and their pharmaceutically-acceptable salts, wherein A and A min are independently hydroxy, alkoxy, aryloxy, or hydroxyamino; R1, R2, R3, R4, R5 and R6 are defined as in the description; and pharmaceutical preparations made therefrom, having biological utility in the treatment of hypertension in subjects suffering therefrom.
Patent IE-900174-L (IE)
Title: Molecules with antibody combining sites that exhibit¹sterospecific catalysis
IPC: C12N15/02
Filed: 1990-01-16
Abstract: A stereoisomeric analog-ligand having a conformation that substantially corresponds to the conformation of a hydrolytic transition state of an amide or ester reactant ligand and the stereochemistry of the nearby atoms is used to produce receptor molecules of predetermined specificity. The receptor molecules include an antibody combining site that binds stereospecifically to one stereoisomer of the analog-ligand and also to one stereoisomer of the reactant ligand and thereby stabilizes the tetrahedral carbon atom of the amide or ester hydrolysis transition state of that reactant ligand to catalytically hydrolyze the reactant ligand at a predetermined site.
[WO9008185A1]
Patent IE-32712-L (IE)
Title: Audio vision display apparatus
IPC: G09B5/06
Filed: 1967-03-02
Abstract: 1,210,011. Audio-visual apparatus; feeding record tapes. D. J. STAPLETON. 28 Feb., 1968 [2 March, 1967], No. 9596/68. Heading G5R. A magnetic tape transported between spools 12 and 15 has recorded thereon both audio information related to slides 18 carried by a rotatable disc 5 and signals which control the rotation of the disc 5 to bring the relevant slide 18 into operative position in a projector 41. One of these control signals picked up by a head 14c causes brief energization of a solenoid 19 which withdraws a plunger 16 from a hole 17 in the disc 5, closing contacts 27 so that a motor 28, through a pulley 9, a slipping clutch 34, and a drive wheel 8, rotates the disc 5 until the plunger 16, urged by a spring 35, enters the next hole 17 and stops the disc. A manually-operable lever 52, 54 controls the application of a braking ribbon 66 to the spool drive motors and selects the direction of movement of the tape by bring- ing one or other of two pinch-rollers 74, 75 into engagement with its associated capstan 76 or 77.
[GB1210011A]
Patent IE-870245-L (IE)
Title: Platinum complexes
IPC: C07F15/00
Filed: 1987-01-30
Abstract: Organic platinum complexes active as anti-tumor agents in warm-blooded animals, and methods for synthesis of same, are described.
Patent IE-44344-L (IE)
Title: Stress bearing building panel
IPC: B05C9/04
Filed: 1977-02-07
Abstract: 1524734 Coating panels all-round with thermoplastics J LAWRENCE T W AYRE and S RICHARDSON [trading as PRE-SEAL ROOFING CO] 7 Feb 1977 [7 Feb 1976] 04855/76 Headings B2E and B2L [Also in Division B5] A stress bearing building panel comprises a stress-bearing panel with an impervious thermoplastic material completely coating both faces and all the edges; typically it is capable of being walked on, is made of plywood or particle board, and the moisture-impervious thermoplastic material is bitumen; the panel may be 8' x 4'. It may have a layer of roofing felt bonded to one face thereof. Panels 11 are driven by nip rolls 15 to be coated by hot bitumen from hopper 19 and also by bitumen applied from tank 23 by roller 24; this co-acts with roller 21 to spread bitumen on the faces of the panel so as to overflow the edges; the "sides" of the panel are coated by the effect of doctor blades downstream of the rollers; the "ends" are coated by momentarily reversing drive rolls 15 to create a gap between adjacent panels, into which gap bitumen flows. A felt 27 may be immersed in bitumen 28 and fed as shown to be laminated to a panel by roller 21.
[GB1524734A]
Patent IE-810590-L (IE)
Title: Preparing malathion
IPC: C07F9/165
Filed: 1981-03-18
Abstract: Process for the preparation of malathion by reacting O,O-dimethyl-dithiophosphoric acid with ethyl maleate in the presence of a solvent which forms a heterogeneous azeotrope with the O,O-dimethyl-dithiophosphoric acid.
[US4367180A]
Patent IE-830621-L (IE)
Title: Hexahydroindole derivatives.
IPC: C07D209/42
Filed: 1983-03-22
Abstract: The invention relates to compounds of the formula I <IMAGE> (I) in which n denotes 0 or 1, R denotes hydrogen, alkyl or aralkyl, R1 denotes hydrogen or alkyl, which can optionally be substituted by amino, acylamino or benzoylamino, alkenyl, cycloalkyl, cycloalkenyl, cycloalkylalkyl, aryl or partially hydrogenated aryl, which each can be substituted by alkyl, alkoxy or halogen, arylalkyl or aroylalkyl, both of which can be substituted in the aryl radical as defined in the aforegoing, a monocyclic or bicyclic sulfur or oxygen and/or nitrogen heterocyclic radical, or a side chain of a naturally occurring aminoacid, R2 denotes hydrogen, alkyl, alkenyl or arylalkyl, Y denotes hydrogen or hydroxyl, Z denotes hydrogen or Y and Z together denote oxygen and X denotes alkyl, alkenyl, cycloalkyl, aryl, which is monosubstituted, disubstituted or trisubstituted by alkyl, alkoxy, hydroxyl, halogen, nitro, amino, alkylamino, dialkylamino or methylenedioxy or 3-indolyl, and their physiologically acceptable salts, processes for their preparation, agents containing these and their use as medicaments and also bicyclic amino acids as their intermediates and processes for their preparation.
[US4562202A]
Patent IE-900834-L (IE)
Title: Sterile product and method for sterilizing and assembling¹such product
IPC: A61L2/08
Filed: 1990-03-08
Abstract: Methods are disclosed for sterilizing a selected portion of a product and for assembling a sterile product from two or more parts which can not be sterilized with the same form of sterilization. A sterile product produced by these methods is also disclosed. The method for sterilizing may include sterilizing a selected portion of the product by exposing the selected portion to an electron beam, while shielding the remainder of the product from the radiation of the electron beam. The method of assembling a sterile product from two or more component parts may include the steps of sterilizing the first part of the product, isolating a portion of the first part from the remainder of the first part, attaching the second part to the isolated portion of the first part, and exposing the isolated portion to a form of sterilization which is deleterious to the remainder of the first part, while shielding the remainder of the first part from such form of sterilization.
[US5009654A]
Patent IE-37793-L (IE)
Title: 7-(hydroxy-halophenyl)acetamido-3-heterocyclicthiomethyl¹cephalosporins
IPC: C07D501/36
Filed: 1973-06-12
Abstract: 1416503 Cephalosporins SMITHKLINE CORP 12 June 1973 [14 June 1972 15 Sept 1972 11 May 1973] 27794/73 Heading C2C Novel cephalosporins, having antibacterial activity, of formula wherein M is hydrogen, alkali metal or NH 4 , X is F, Cl or Br and Het is a 5- or 6-membered heterocyclic ring containing carbon and up to four N, O or S atoms, the heterocyclic moiety being substituted with up to 2 C 1 -C 4 alkyl, C 1 -C 4 alkenyl, C 1 -C 4 alkoxy, C 1 -C 4 alkoxy, C 1 -C 4 alkyl, CF 3 , OH, halogen, hydroxy- (C 1 -C 4 )alkyl or SR, R being hydrogen or C 1 -C 4 alkyl, are prepared by acylation of the appropriate 7-amino-3-heterocyclicthiomethyl cephalosporin with a 3-halo-4-hydroxyphenylglycine in which the amino group is protected with a removable protecting group such as t-butoxycarbonyl. Following acylation, the protective group may be removed by trifluoroacetic acid, and the resulting salt converted to the Zwitterionic product by means of a basic ion exchange resin. The compounds of Formula I may also be prepared by displacement of the 3-acetoxy group of a 7- acylated - 3 - acetoxymethylcephalosporin with a suitable mercapto-heterocyclic compound under basic conditions. The preparation of 7-[DL-α-amino-α-(3-fluoro-4-hydroxyphenyl) acetamido] - 3 - (5 - methyl - 1,3,4 - thiadiazol- 2 - ylthiomethyl - 3 - cephem - 4 - carboxylic acid, 7 - [DL - α - amino - α - (3 - fluoro - 4- hydroxyphenyl)acetamido] - 3 - (1 - methyl- 1,2,3,4 - tetrazol - 5 - ylthiomethyl) - 3 - cephem- 4 - carboxylic acid, 7 - [DL - α - amino - α- (3 - fluoro - 4 - hydroxyphenyl)acetamido] - 3- (1,2,3 - triazol - 4 - ylthiomethyl) - 3 - cephem- 4 - carboxylic acid and 7 - [DL - α - amino - α- (3 - chloro - 4 - hydroxyphenyl)acetamido] - 3- (1 - methyl - 1,2,3,4 - tetrazol - 5 - ylthiomethyl)- 3 - cephem - 4 - carboxylic acid is described (Examples 6 to 9). N - t - butoxycarbonyl - 3 - fluoro - 4 - hydroxyphenylglycine is prepared by reacting 3-fluoro - 4-hydroxyphenylglyeine with t-butoxycarbonyl azide in the presence of magnesium oxide. The corresponding 3-chloro and 3-bromo cornpounds are prepared in a similar manner.
[GB1416503A]
Patent FI-844738-L (FI)
Inventor: OLSSON MATS
IPC: F23B99/00
Filed: 1984-11-30
Abstract: A reciprocating movement of the combustion air and gas through a glow bed (13) is provided by exposing the bed to a high particle sound velocity. For this, an external low frequency generator (11) of max. frequency of 30 hz is used. The dimensions of the grate in a plane transverse to the reciprocating movement of combustion air and gas are below a quarter of the wave length of the generated sound. The sound generator frequency is determined by a Helmholtz resonator or a reciprocating mechanism. The resonator can be in the form of an electrical loudspeaker.
Patent FI-851356-L (FI)
Inventor: WARD FREDERICK E
IPC: C07D307/58
Filed: 1985-04-03
Abstract: A novel compound useful in detecting leukocytes, esterase and protease in a test sample. The compound has the structurein which: A is an acid residue, R is lower alkyl, aryl, carboxyl, carboxyl ester, amido or cyano, R<sup>*</sup> is H or lower alkyl, and X is 0, S, or NR', in which R' is H, lower alkyl or aryl.
Patent IE-901416-L (IE)
Title: Piperazine derivatives
IPC: C07D295/13
Filed: 1990-04-20
Abstract: Piperazine derivatives of formula <CHEM> and their pharmaceutically acceptable acid addition salts are disclosed. In the formula n is 1 or 2, R is hydrogen or lower alkyl, R<1> is an aryl or nitrogen containing heteroaryl radical, R<2> is hydrogen or lower alkyl, R<3> is aryl, C4-8 alkyl or aryl(lower)alkyl and X is a functionalised group of specified meaning. The compounds exhibit activity as 5-HT1A antagonists and can be used, into alia, for the treatment of CNS disorders, such as anxiety.
Patent IE-35816-L (IE)
Title: Purine sugar derivatives
IPC: C07H19/16
Filed: 1971-11-16
Abstract: 1386585 Purine-sugars WELLCOME FOUNDATION Ltd (Burroughs Wellcome Co) 16 Feb 1972 [16 Nov 1970] 54504/70 Heading C2C [Also in Division A5] Novel threapeutic compounds (I) (including salts thereof) where R<SP>1</SP> is SH or C 1 to C 4 alkylthio and R<SP>2</SP> is NH 2 or H, or R<SP>1</SP> is NH 2 and R<SP>2</SP> is OH, provided that when R<SP>1</SP> is SH or MeS, R<SP>2</SP> is NH 2 , are made by reducing compounds (II) and when desired alkylating a product obtained, or converting a 2,6-diaminoproduct obtained into a 2-hydroxy- 6-aminocompound by diazotization and hydrolysis (Y<SP>1</SP> is protected mercapto or NH 2 and Y<SP>2</SP> is H or NH 2 , provided that when Y<SP>1</SP> is NH 2 , Y<SP>2</SP> is NH 2 , and Z is a blocking group). Compounds (II) where Y<SP>1</SP> is protected mercapto and Y<SP>2</SP> is H or NH 2 , provided that when Y<SP>1</SP> is MeS then Y<SP>2</SP> is NH 2 , are also novel.
[GB1386585A]
Patent IE-38451-L (IE)
Title: Retention of paper on rotary drum
IPC: G03B27/62
Filed: 1973-08-22
Abstract: A rotating drum has a gripper bar mounted for cooperation therewith to convey sheets. The gripper bar is manually moved from a stationary first position spaced from the rotating drum to a second position to grip the sheet against the drum and rotate therewith. After moving through a predetermined angle, the eccentric mounting of the gripper bar causes the bar to move away from the drum and assume the stationary first position.
[US3918707A]
Patent IE-33882-L (IE)
Title: Ultraviolet screening agents
IPC: A61K/
Filed: 1969-12-16
Abstract: 1297126 UV screening compositions F HOFFMANN-LA ROCHE & CO AG 11 Dec 1969 [16 Dec 1968] 60439/69 Heading A5B A UV-screening agent suitable for topical application contains as essential active ingredient cytosine, uracil, guanine and/or chloro-uracil and a solid or liquefied gaseous diluent or a liquid diluent other than a solvent of molecular weight less than 200 except in the presence of a surface active agent. Conventional light-screening substances may also be present.
[GB1297126A]
Patent IE-801729-L (IE)
Title: A morpholine derivative
IPC: A01N43/84
Filed: 1980-08-15
Abstract: Morpholine derivatives of the formula:- <IMAGE> wherein R represents ethyl or phenyl, as well as their salts and N-oxides, possesses fungicidal activity and can be used as antimycotics, especially for combating Candida albicans.
[EP0024334A1]
Patent IE-871958-L (IE)
Title: Methylene chloride-based derivatives
IPC: G03F7/26
Filed: 1987-07-20
Abstract: Composition and its use for removing photoresist films from printed circuits in the electronics industry. Propylene oxide, methanol and methyl tert-butyl ether are added to the methylene chloride.
Patent IE-45938-L (IE)
Title: 1-phenoxy-3-amino-propan-2-ols
IPC: C07C231/00
Filed: 1977-10-06
Abstract: The process is used for preparing the novel amines of the formula (I) <IMAGE> R<1>, R<2> and R<3> are defined in Patent Claim 1. The reactions for preparing the said compounds always take place between primary amines and compounds having a reactive, esterified hydroxyl group or an epoxy group. The novel compounds effectively block beta receptors.
[SE7611125A]
Patent IE-812103-L (IE)
Title: Load carrying trolley.
IPC: B62B3/18
Filed: 1981-09-10
Abstract: Load-handling trolleys of a type in which a load-supporting deck is displaceable into an out-of-use position and opposed load-retaining side walls can be pivoted about rear pivot axes to bring them into mutually inclined positions such that a number of such collapsed trolleys can be nested one into another. The trolley has a wheeled base unit to which the side walls are detachably connectable. The base unit comprises a bridge portion (4) and opposed side beams (2, 3) for supporting the load-retaining side walls. Such side beams are connected to the bridge portion by pivot joints (10, 11) so that the side beams can swing into mutually inclined positions together with the side walls.
[US4456273A]
Patent IE-902249-L (IE)
Title: Improvements in or relating to dispensers
IPC: B65D83/14
Filed: 1990-06-21
Abstract: Dispensing arrangements, comprising a gas-pressurized container for a material to be dispensed with a valve actuable to open a discharge passage through the valve and through a valve and a valve actuator to an actuator discharge outlet, are well known in the art. The invention proposes a non-liquefied gas-pressurized dispensing arrangement capable of being used with relatively low initial gas pressures, and of discharging a relatively high percentage of the dispenser contents with an acceptable spray pattern. The proposed dispensing arrangement attains these advantages by arranging the cross-sectional area of the valve port (17c) to be many times greater than the cross-sectional area of the actuator outlet (22a). In one recited embodiment the actuator outlet has a cross-sectional area in the region of 0.049 mm<2> whilst the total cross-sectional area of the valve ports, the valve having four ports, is some sixteen times greater.
Patent IE-802368-L (IE)
Title: Connector assembly
IPC: A01J7/00
Filed: 1980-11-14
Abstract: A device for closing a fluid flow passage in response to a decrease in vacuum pressure existing in the passage. The device comprises a fluid flow passage with a seating therein. A diaphragm is located so that one face thereof can locate on the seating to close the passage. A chamber is formed partially by the or at least part of the other face of the diaphragm. In use the diaphragm is maintained away from said seating by a higher pressure in the chamber due to a pressure differential existing between chamber and passage. Venting means open the chamber to atmosphere, and means are provided to seal said venting means. Actuating means are provided and engage with said diaphragm when the pressure differential exists. Accordingly when the pressure differential is altered by a decrease in the vacuum in said passage, the resultant movement of the diaphragm causes the actuating means to operate the sealing means such that the venting means vent said chamber and enables the diaphragm to locate on the seat.
[US4347868A]
Patent IE-43329-L (IE)
Title: Drawer assembly
IPC: A47B88/00
Filed: 1976-10-29
Abstract: The invention has as an aim a drawer to assemble kind comprising a basic panel 10, two panels on side it, a panel postpones 12, a panel before 13, and of the means of assembly suitable to solidarize two to two these panels. According To the invention, these means of assembly form a unit with the panels and comprise, for a panel, a male part of enclipsage, for example 15, and for another panel, a part female of enclipsage, for example 38, suitable to receive the aforementioned male part. [FR2355482A1]
Patent IE-45930-L (IE)
Title: Bobbin
IPC: B65H75/12
Filed: 1977-12-05
Abstract: A bobbin on which a package of thread-form or strip-form material can be wound has at one or both ends a reflexive snap ring which is selectively displaceable between first and second positions with an over-center snap action. In the first position of the snap ring the end of the thread or other material to be wound on the bobbin is held fast in a slot at the boundary of a thread-receiving channel which extends circumferentially around the bobbin, while in the second position of the snap ring the channel is opened for access. The snap ring may be integral with the bobbin sleeve and the bobbin made of a synthetic-resin material. The snap ring can be used on bobbins which have a circumferential flange to retain the wound package and on bobbins without such a flange, in which case the snap ring is directly engageable with the end of the package.
[US4165055A]
Patent IE-43895-L (IE)
Title: Inhalation device
IPC: A61M11/02
Filed: 1976-12-10
Abstract: An aerosol inhalation device for dispensing medicine makes use of separate propellant and medicine containers. A valve is provided, which acts in conjunction with a metering chamber, to supply a measured amount of propellant upon each activation of the device.
[SE7514066A]
Patent IE-853322-L (IE)
Title: Micromonospora microorganisms and antibiotic production¹therby
IPC: A61K31/70
Filed: 1985-12-30
Abstract: Novel microorganisms belonging to the genus Micromonospora are capable of producing antibiotics represented by the formula:wherein R represents a hydrogen atom or a formyl group and the dotted line represents a double bond orThe antibiotics are produced by culturing these microorganisms and harvesting the resulting antibiotics.
Patent NO-750581-L (NO)
Inventor: HARSY-VADAS G
IPC: B60G11/30
Filed: 1975-02-20
Abstract: Gassfjær med nødfjær.
Patent NO-821095-L (NO)
Inventor: ERMERT WOLFGANG
IPC: B65D1/28
Filed: 1982-03-31
Abstract: The invention relates to composite packing films shrinkable by deep drawing and consisting of at least one copolyamide layer containing at least 50% by weight of  epsilon -caprolactam units and at least one heat-sealable layer, and optionally, an adhesion-promoting layer.
Patent NO-822455-L (NO)
Inventor: MONDT JOSEF
IPC: C08F220/12
Filed: 1982-07-15
Abstract: 1. A process for the preparation of an aqueous dispersion of copolymers, which can be cross-linked with aminoplasts by the action of heat, by copolymerization of styrene and/or methyl methacrylate, as the hardening component, 2-ethylhexyl acrylate and/or butyl acrylate and/or ethyl acrylate as the plasticizer component, hydroxyethyl (meth) acrylate and/or hydroxypropyl-(meth)acrylate, acrylic acid and/or methacrylic acid and an amide and/or an N-methylolamide and/or an etherified N-methylolamide of an alpha, beta-unsaturated carboxylic acid in the aqueous phase in the presence of an emulsifier and a radical-forming initiator, which comprises copolymerizing a mixture of I. 40-60 % by weight of methyl methacrylate of styrene or a mixture of these monomers, II. 30-50 % by weight of ethyl acrylate, butyl acrylate or 2-ethylhexyl acrylate or a mixture of these monomers, III. 5-15 % weight of hydroxyethyl acrylate, hydroxyethyl methacrylate, hydroxypropyl acrylate or hydroxypropyl methacrylate or a mixture of these monomers, IV. 1-5 % by weight or acrylic acid or methacrylic acid or a mixture of these monomers and VI. 0.5-5 % by weight of an amide or N-methylolamide or an etherified N-methylolamide of an alpha, beta-unsaturated carboxylic acid or a mixture of monomers of this type.
Patent NO-832001-L (NO)
Title: Fremgangsmaate ved fremstilling av 1-sulfo-2-okso-azetidinderivater
Inventor: HOFHEINZ WERNER
IPC: C07F7/08
Filed: 1983-06-02
Abstract: l-sulfo-2-oksoazetidinderivater med den generelle for—. hvor Het er en eventuelt aminosubstituert, 5-eller 6-leddet, aromatisk heterosyklisk ring inneholdende 1. eller 2 nitrogenatomer, evt. også et oksygen- eller svovelatom, R^" betyr hydrogen, lavere-alkyl, fenyl-lavere-alkyl, lavere-alkanoyl, lavere-alkoksykarbonyl, la-,. vere-alkenyl-lavere-alkyl, lavere-alkoksykarbonyl- • lavere-alkyl, fenyl-lavere-alkoksykarbonyl-lavere-alkyl , nitrofenyl-lavere-alkoksykarbonyl-lavere-al-2. kyl eller karboksy-lavere-alkyl, og R betyr hydro-|_j gen, lavere-alkyl, lavere-alkenyl, lavere-alkinyl,. lavere-alkoksykarbonyl, lavere-alkanoyloksy-lavere-alkyl, lavere-alkoksykarbonyl-lavere-alkenyl, hydro-j_I ksyiminometyl, lavere-alkoksyiminometyl, karbamoyl,. karbaraoyl-lavere-alkenyl eller karbamoyloksy-lavere-j ! alkyl, idet gruppen =NORi det minste delvis foreligger i synform,. i. j ji racemisk form eller i form av de 3S-enantiomerer, samt av lett hydrolyserbare estere henh. farmasøytisk fordragelige salter av disse forbindelser. Fremstilling av forbindelsene er beskrevet. Forbindelsene har anti-mikrobiell virkning.
Patent NO-854601-L (NO)
Inventor: VIGNEAU JEAN-LOUIS
IPC: A61M16/00
Filed: 1985-11-18
Abstract: A gas heating process is disclosed in which a gas to be heated and carbonic gas causing an exothermic reaction with soda-lime are caused to pass simultaneously over a charge of soda-lime. The device of the invention includes a cartridge with a first chamber containing the charge of soda-lime and a second chamber containing the amount of carbonic gas required for starting the exothermic reaction, and a means for placing the two chambers in communication. The first chamber is connected to an inlet for the mixture of gas to be heated and carbonic gas for maintaining the reaction, and also is connected to an outlet (3) for the heated gas.
Patent NO-863123-L (NO)
Inventor: KOLL LAUREL A
IPC: A61B10/02
Filed: 1986-08-01
Abstract: The coaxial annular space between a rod and a slidably received outer cylinder is divided into three serial chambers by four seals. Two seals are spaced apart and affixed to the front of the rod. Two seals are spaced apart and affixed to the cylinder rearwardly of the first two. By relative forward rod movement, a specimen capturing zone is exposed at the desired site of a biological specimen. Thereafter, rearward rod movement reseals the capturing zone. Further, rearward rod movement reduces the volume of a media containing chamber and thereby moves the collection zone into contact with the desired medium. The third chamber prevents contamination of the biologically active portions of the structure during operation. Pre-scored break lines formed in the cylinder and rod facilitate severance of unneeded portions after collection of a biological specimen and/or after transportion to a suitable laboratory facility. Color-coded indicia are used on the rod and/or cylinder so as to facilitate proper operation. Reusable extension pieces may be attached to the cylinder and/or rod so as to adapt a standard size module to different desired end uses.