baber/WOPTO huggingface dataset:
Patent ES-8800225-A1 (ES)
Title: 6-substituted mitomycin analogs
IPC: C07D487/14
Filed: 1985-09-03
Abstract: Novel methods for treatment of neoplastic disease states in animals, which methods comprise administering a therapeutically effective amount of a compound of the formula IV, < IMAGE > IV wherein: Y is hydrogen or lower alkyl and Z is a radical of the formula -O-R, wherein R is: a substituted lower alkyl radical selected from the group consisting of mono- and di-hydroxy lower alkyl, cyano lower alkyl, halo lower alkyl, lower alkyl amino lower alkyl, hydroxy lower alkylthio lower alkyl, hydroxy lower alkyldithio lower alkyl, di-lower alkoxy lower alkyl, hydroxy or lower alkoxy substituted lower alkoxy lower alkyl, and cyclo lower alkyl substituted lower alkyl or a lower alkenyl radical or a lower alkynyl radical or a substituted or unsubstituted oxygen-containing heterocyclic radical selected from the group consisting of tetrahydro furanyl or lower alkyl substituted derivatives thereof, lower alkyl substituted oxiranyl, lower alkyl substituted dioxolanyl, lower alkyl substituted pyranyl, or lower alkyl substituted furanyl.
Patent ES-8705442-A1 (ES)
Title: Novel beta-lactams and their production.
IPC: C07F7/18
Filed: 1985-12-27
Abstract: A beta-lactam compound of the formula: <CHEM contiene="yes"> wherein R1 and R2 are, the same or different, each a hydrogen atom or a lower alkyl group, R3 is a lower alkyl group, R4 is a hydrogen atom, a carboxyl-protecting group or a thiolcarboxyl-protecting group, X is a hydrogen atom, a hydroxyl group or a protected hydroxyl group, Y is an oxygen atom or a sulfur atom and COZ is a carboxyl group, an activated or protected carboxyl group, a thiolcarboxyl group or an activated or protected thiolcarboxyl group, which is useful as a valuable intermediate in the stereospecific production of 1-alkylcarbapenem compounds.
Patent ES-8900008-A1 (ES)
Title: Antigens and monoclonal antibodies reactive against sporozoites of eimeria spp.
IPC: A61K39/012
Filed: 1986-01-31
Abstract: Monoclonal antibodies against sporozoites of the Eimeria spp. are obtained by use of hybridoma technology. Specific sporozoite antigens for use as vaccines in the prevention and treatment of coccidiosis and hybridoma cultures producing monoclonal antibodies are described.
Patent ES-8801284-A1 (ES)
Title: Benzothiophenes and benzofurans having antiallergic activity.
IPC: C07D307/92
Filed: 1987-01-16
Abstract: There is disclosed a compound having the following general formula (I) <CHEM contiene="yes"> or a pharmaceutically acceptable salt thereof, wherein: R<1>, R<4>, and R<5> are each, independently, H, an alkyl having from one to twelve carbon atoms, an alkoxy having from one to twelve carbon atoms, a hydroxy, an aryl, a nitro group, an amino group, a substituted amino group, a mercapto radical, an alkylthio radical having from one to four carbon atoms, an alkylsulphinyl radical having from one to four carbon atoms, an alkylsulphonyl radical having from one to four carbon atoms, an arylthio radical, an arylsulphinyl radical, an arylsulphony radical or a halogen, R<1> being further chosen from a methylenedioxy radical attached to adjacent carbon atoms of the benzene ring R<2> is an alkoxy having from one to twelve carbon atoms, an arylmethoxy, an amino group, a substituted amino group., a mercapto group, an alkylthio having from one to four carbon atoms, an alkylsulphinyl having from one to four carbon atoms, an alkylsulphonyl having from one to four carbon atoms, an arylthio, an arylsulphinyl, or an arylsulphonyl and R<3> is A or B <CHEM contiene="yes"> X is oxygen or S(O)q wherein q is zero, one, or two. Also disclosed is a process for preparing the compounds, compositions comprising the compounds and pharmaceutical uses of the compounds. The novel benzothiophene and benzofuran derivatives have antiallergic activity. The disclosure describes the use of derivatives for prevention of the release of mediators including histamine and leukotrienes from basophils and mast cells, and prevent respiratory burst in neutrophils providing activity useful in cardiovascular disorders as well as in antiinflammatory, psoriasis, and antimigraine treatment.
Patent IE-901793-A1 (IE)
Title: Pyranyl cyanoguanidine derivatives
IPC: C07D311/70
Filed: 1990-05-18
Abstract: Novel compounds having the formula <CHEM>  wherein <CHEM> are disclosed. These compounds have potassium channel activating activity and are useful, for example, as cardiovascular agents, especially as antiischemic agents.
Patent IE-912032-A1 (IE)
Title: New cephalosporins containing, in position 3, a propenyl¹radical substituted by a quaternary ammonium, their¹preparation process, their use as medicaments, the¹compositions containing them and the new intermediates¹obtained
IPC: C07D501/24
Filed: 1991-06-14
Abstract: The invention relates to the products of formula: in which: R1 =, in particular, or Rb and Rc = H or acyl A and A' =, in particular H, alkali metal equivalent, aminated organic base, readily cleavable ester group, or CO2A represents CO2<(-)> to a process for their preparation, to their use as medicaments, to compositions containing them and to the new intermediates obtained.
Patent IE-913129-A1 (IE)
Title: Synergistic composition and method of selective weed control
Inventor: MAURER WILLY
IPC: A01N43/90
Filed: 1991-09-05
Abstract: The present invention relates to a synergistic agent containing a herbicidally active sulphonylurea of the formula I <IMAGE>  in which   Z represents a substituted phenyl, thiophenyl, benzyl, pyridinyl, pyrazinyl, hetero-fused phenyl, or alkylsulphonylamino radical;   M represents hydrogen; or C1-C4-alkyl; and Het represents a substituted five- or six-membered heterocycle having 2 or three nitrogen atoms, and a synergistically active amount of a 5,6,7,8-tetrahydro-1H,3H- (1,3,4)thiadiazolo-[3,4-a]-pyridazine or 7,8-dihydro-1H,3H- (1,3,4)-thiadiazolo-[3,4-a]-pyridazine of the formula II <IMAGE> in which     X represents oxygen; or sulphur;   A-B represents -CH2-CH2-; or -CH=CH-; and   Phe represents a substituted phenyl radical.   The agent according to the invention is suitable for selective control of weeds in crops of useful plants, in particular in cereals, maize, rice or soybeans. The invention also relates to a method of controlling weeds in crops of useful plants, preferably in cereals, maize, rice or soybeans, and to the use of this novel agent.
Patent IE-904382-A1 (IE)
Title: Substituted cyclohexanols as central nervous system agents
Inventor: CAPRATHE BRADLEY WILLIAM
IPC: A61K31/535
Filed: 1990-12-05
Abstract: Substituted cyclohexanols and cyclohexylamines and derivatives thereof of the formula I as well as methods for the preparation and pharmaceutical composition of same, which are useful as central nervous system agents and are particularly useful as dopaminergic, antipsychotic, and antihypertensive agents as well as for treating hyperprolactinaemia-related conditions and central nervous system disorders.
Patent IE-922463-A1 (IE)
Title: Apparatus for the handling of electrophoretic transfer¹membranes and for the chemiluminescent detection of blots¹contained thereon, and processes using the apparatus
Inventor: ANDERSON LYNNE ELIZABETH
IPC: G01N27/447
Filed: 1992-07-29
Abstract: Improved apparatus for the handling and detecting of an electrophorectic transfer membrane is disclosed herein, the improvement comprising guide apparatus designed to accomodate the transfert membrane, a pressure head positioned relative to the guide apparatus to releasably engage the membrane, and light shielding apparatus positioned relative to the guide apparatus to selectively enclose about the transfer membrane. The apparatus is operated so that the pressure head engages a flexible portion of the transfer membrane containing an electrophoretic blot while it is in a position appropriate for detection. There is also disclosed herein a process for utilizing the apparatus of the invention. In the process drying and optionally heating of the membrane where the blot has been contacted with enzyme-triggered 1,2-dioxetanes, to enhance the resulting chemiluminescent signal, is disclosed.
Patent IE-922537-A1 (IE)
Title: Improved method of applying metal coatings on cubic boron nitride and articles made therefrom
Inventor: IACOVANGELO CHARLES DOMINIC
IPC: C09K3/14
Filed: 1992-07-31
Abstract: Cubic boron nitride particles are electrolessly nickel plated with a nickel alloy formed with a metalloid, such as boron. Electrolessly plated particles are then gradually heated at a steady rate from room temperature to a desired heat treatment temperature in a non-oxidizing atmosphere formed by argon containing 10% hydrogen. Exemplary articles made by the aforementioned process include a grinding wheel having uniformly dispersed abrasive cubic boron nitride particles having the Ni/B alloy coat thereon.
Patent IE-922554-A1 (IE)
Title: Device for emptying containers
Inventor: RECK HERBERT
IPC: B65F3/04
Filed: 1992-07-31
Abstract: In order to make it possible to empty in particular, large containers with a crew of just one person, an emptying device with a tilting/lifting device 1 and a control unit 4 is described to which a trigger switch 2 is connected which is actuated by the container to be emptied as it approaches the lifting/tilting device and which triggers the raising phase of the lifting/tilting process automatically. When a preset raised level of the lifting/tilting device is reached the control unit interrupts the raising phase. In addition, a first manual actuator 8 to trigger the automatic emptying process, which actuator has an effect upon the control unit 4 only after the interruption of the lifting process, is connected to the control unit. The control unit 4 contains a programmable device 5 into which the preset raised level can be inputted. The programmable device 5 also assumes the function of monitoring the preset time spans, such as the time span between the actuation of the trigger switch 2 and the actuation of the acknowledgement signal switch 3. After the container is emptied, putting the container back down completely is accomplished by means of a second manual actuator 9.
Patent LU-101323-A1 (LU)
Title: Dynamic testing device for mechanical properties of pile and soil
Inventor: TAN JUNKUN
Filed: 2019-07-22
Abstract: The present disclosure relates to the technical field of civil engineering, in particular to a dynamic testing device for mechanical properties of piles and soils, including a top plate, a support plate and a bottom plate fixedly connected in series through a set of support columns from top to bottom. A film box is embodied and installed between the support plate and the bottom plate. The film box includes a circular rubber film cylinder, a bottom supporting board and a cover plate; the bottom supporting board is coaxially embedded in the middle of the bottom plate, the bottom supporting board is arranged at the lower end of the rubber film cylinder, and the cover plate is used for sealing the upper port of the rubber film cylinder. The cover plate passes through the support plate and is fixedly connected to the top plate through a set of mounting columns; a vertical loading device is arranged in the middle of the top plate, and at least one horizontal loading device is arranged on the outer ring of the rubber film cylinder. The present disclosure controls the displacement stroke of each telescopic rod. When the strokes of the telescopic rods are the same, the corresponding horizontal pressures are applied to the piles in the respective directions, and different states of different side pressures are realized when the strokes are different, which is more flexible and suitable for to different experimental requirements.
Patent LU-502619-A1 (LU)
Title: Method for control of grab bucket in pit cleaning
Inventor: LAN JIANGSONG
IPC: B25J9/16
Filed: 2022-01-13
Abstract: The invention relates to a method for control of a grab bucket in pit cleaning, including the steps of: performing spatial vectorization on the pit structure to construct a spatial coordinate system and calibrating the position coordinates of the pit edge; determining the position of the grab bucket in the pit and calibrating the position coordinates in dynamic state of the grab bucket based on the size of the grab bucket; driving, by a sliding assembly and a lifting assembly, the grab bucket to move in the pit, and in cooperation with the action of the grab bucket, driving the grab bucket for dynamic adjustment, so that the position coordinates in dynamic state of the grab bucket are controlled never to exceed coordinates of the edge; and setting a laser scan device to move along with the grab bucket to detect the material distribution state in the pit. With the method for control of a grab bucket in pit cleaning in the present invention, the position of the grab bucket relative to the pit is defined by coordinatograph processing and the position of the grab bucket is dynamically adjusted, thereby accomplishing grabbing of the material at the pit edge.
Patent LU-56947-A1 (LU)
IPC: C08J5/22
Filed: 1968-09-24
Abstract: 1,199,668. Ion - exchange membranes. RHONE-POULENC S.A. 24 Sept., 1968 [25 Sept., 1967], No. 45369/68. Headings C3G and C3P. [Also in Divisions D1-D2] An ion-exchange membrane is formed of a vinyl chloride polymer or copolymer grafted with an aromatic vinyl monomer comprising an intranuclear or juxtanuclear tertiary nitrogen atom, or of a mixture of a vinyl chloride polymer or copolymer and a polymer of an aromatic vinyl monomer comprising an intranuclear or juxtanuclear tertiary nitrogen atom, all or part of the said tertiary nitrogen atoms having been quaternized by an alkylene or alkenylene dihalide or bis-(haloalkyl)-benzene. Specified aromatic vinyl monomers are vinyl pyridines and N,N-dialkylaminostyrenes. The polymer may be partially quaternized with the dihalide and the quaternization completed using a monofunctional quaternizing agent, e.g. an alkyl, cycloalkyl or aralkyl halide or sulphate. In the examples, (1) polyvinyl chloride is grafted with 4-vinylpyridine, the resulting graft polymer being quaternized with p-dodecylbenzyl chloride and bis - 1,4 - (chloromethyl) - benzene then treated with methyl iodide, (2) a membrane is formed as in Example 1, except that no dodecylbenzyl chloride is used, (3) a polyethylene glycol terephthalate fabric is soaked in a solution of the graft copolymer obtained in Example 1 and the supported film obtained is quaternized as in Example 1, (4) a solution of polyvinyl chloride and p-dimethylamino-styrene in cyclohexanone is poured on to glass, dried and then quaternized as in Example 2, (5) and (7) polyvinyl chloride and poly-p-dimethylaminostyrene are dissolved in cyclohexanone and a film formed from the solution is quaternized as in Example 2 and (6) a membrane reinforced with fabric is formed as in Example 3, using the solution of polymers prepared in Example 5.
Patent SU-237073-A1 (SU)
Title: Способ бурения электрическими импульсными разрядами
IPC: E21C37/18
Filed: 1959-04-14
Granted: 2004-04-10
Abstract: Способ бурения электрическими импульсными разрядами, отличающийся тем, что для разрушения породы разряд осуществляют в буримом твердом теле под слоем жидкости, например воды, трансформаторного масла и др., со временем нарастания напряжения импульса до пробоя менее 5•10c.
Patent AT-500084-A1 (AT)
IPC: B65G1/137
Filed: 2004-03-18
Abstract: Device for supplying stackable goods (2) comprises a detecting unit (30) having a positioning carriage (32) arranged above a supply hopper (13). The carriage is provided with a measuring device (33) for measuring the distance between the uppermost goods and a maximum filling level of a supply hopper to determine the level of the goods in one hopper. Preferred Features: The positioning carriage has a guiding arrangement (35) by which it is guided on a guiding strip running in the longitudinal direction of a storage unit (4).
Patent AT-514771-A1 (AT)
Title: Siloxanbasierter Adhäsionsgreifer
Inventor: CAKMAK UMUT DIPL ING
IPC: B65G47/90
Filed: 2013-08-27
Abstract: Haltevorrichtung (1), insbesondere Adhäsionsgreifer, mit einer Halterung (2) und einem in oder an der Halterung (2) befestigten Greifstempel (3), wobei der Greifstempel (3) eine elastomereKontaktfläche (4) aufweist, wobei die Kontaktfläche (4) aus einem vernetzten Siloxan besteht.
Patent WO-9318902-A1 (WO)
Title: Device for processing synthetic thermoplastic material
Inventor: BACHER HELMUT
IPC: B29B17/00
Filed: 1993-03-16
Abstract: A device for pre-processing a synthetic thermoplastic material, such as polyester waste, comprises at least two containers (1, 13) connected in series, in each of which a comminuting and mixing tool (5) rotates at the base of the containers (1, 13) about a vertical axis. At least the downstream container has an evacuation duct (18) which can also be used to introduce an inert gas if required. The containers (1, 13) are connected by a sleeve (12) in which there is a stop valve (20) to facilitate trouble free maintenance of the vacuum in the downstream container (13) until the valve (20) is opened, thus allowing the vacuum in the container (13) to draw in the material in the upstream container (1). In the upstream container (1) (as seen in the flow-direction of the material), the material is pre-comminuted, pre-heated, pre-dried and pre-compacted and that process is enhanced by the turbulence in the material as it is sucked into the downstream container (13). Completely homogenous material is thus transported for further processing by a worm (16) which is connected to the last container (13).
Patent WO-9600830-A1 (WO)
Inventor: NEUMAYER HARALD
IPC: E05B27/00
Filed: 1995-06-30
Abstract: L'invention concerne un dispositif de blocage électromagnétique du barillet de fermeture (2) d'une serrure (1), qui comporte un réducteur de rotation comprenant une bobine (12) et un rotor (7). Selon la position dans laquelle la gâchette (4) mobile est tournée, elle peut être sortie de la cavité (3) du barillet de fermeture dans laquelle elle est engagée. En position de fermeture, une butée située sur la face avant (11) du rotor empêche la gâchette de se déporter.
Patent WO-9903474-A1 (WO)
Inventor: BURGHART WALTER
IPC: A61K9/00
Filed: 1998-07-15
Abstract: The invention relates to a method for producing stable acetylsalicylic acid solutions with non-aqueous pharmaceutically acceptable organic solvents such as dimethylisosorbide, propylene glycol or diethylene glycol monoethyl ether, wherein 0.005 - 2 wt. % of a cyclic acidic imide and/or 0.005 - 2 wt. % of a sulphamic acid and preferably 1 - 40 wt. %, in relation to the weight of the solution, of a compound of general formula (I) is added to the solution. In said general formula, R1 stands for H, CH3 or C2H5, n = 0 or 1 and R2 is H or one or more low alkyl, low alkyloxy or low alkenyl radicals with 1 to 5 C atoms.
Patent WO-0061919-A1 (WO)
Title: Reglage de jeux de soupape sur des moteurs a combustion interne a arbre a cames en tete
Inventor: HADAWAY ROBERT JOHN
IPC: F01L1/20
Filed: 2000-04-10
Abstract: La présente invention concerne un procédé et un dispositif pour régler des jeux de soupape sur des moteurs à combustion interne à arbre à cames en tête. Un élément cale (82) allongé, amovible et de section rectangulaire, présente une rainure (94) s'étendant longitudinalement sur cet élément. Cet élément cale (82) se loge par coulissement dans un évidement (88) ménagé dans une paroi latérale d'un corps (84) de galet de came. Le remplacement de l'élément cale (82) permet de régler le jeu de soupape entre une surface de compression (86) du corps (84) de galet de came et un lobe d'arbre à cames. L'élément cale (82) peut être remplacé avec des articles en stock de différentes épaisseurs, de façon à faciliter le réglage rapide et efficace du jeu de soupape. Une grande partie du travail et du temps passés au réglage du jeu de soupape avec les procédés classiques est ainsi éliminée et il n'est pas nécessaire d'enlever le(s) arbre(s) à cames et l'engrenage d'entraînement.
Patent WO-0183363-A1 (WO)
Title: Actionneur a flexion thermique ameliore
Inventor: SILVERBROOK KIA
IPC: B41J2/14
Filed: 2001-05-02
Abstract: L'invention concerne un actionneur à flexion thermique (6) présentant des bras supérieurs (23, 25, 26) et des bras inférieurs (27, 28) non plans, de manière à accroître la rigidité des bras. Les bras (23, 25, 26, 27, 28) peuvent être espacés transversalement les uns des autres et sans recouvrir l'autre, en vue en plan, permettant ainsi que tous les bras soient formés en déposant une seule couche de matériau formant le bras.
Patent WO-0220598-A1 (WO)
Title: Mucine
Inventor: MCGUCKIN MICHAEL ANDREW
IPC: A61K38/17
Filed: 2001-07-27
Abstract: L'invention se rapporte, de façon générale, à une mucine épithéliale. Plus particulièrement, l'invention se rapporte à une nouvelle mucine trans-membrane, à des séquences génétiques codant pour celle-ci, à des anticorps ayant pour cible la mucine et des compositions renfermant la mucine, à ses anticorps ou séquences génétiques codant pour celle-ci. L'invention concerne en outre des méthodes de détection d'états maladifs ou de tendance au développement d'états maladifs, par dépistage d'aberrations dans la mucine ou dans sa séquence génétique de codage.
Patent WO-02084511-A1 (WO)
Title: Reseau dependant virtuel pour clients et utilisateurs de fournisseurs de services et procede associe
Inventor: YOGESAN KANAGASINGAM
IPC: G16H30/20
Filed: 2002-04-10
Abstract: La présente invention concerne un système de soins de santé électronique. Ledit système comprend un certain nombre de stations (12) connectées par l'intermédiaire d'un réseau local d'entreprise ou par l'intermédiaire de l'Internet. Des stations de service clients (13) sont utilisées pour capturer et traiter des images numériques qui sont ensuite téléchargées sur une station de service centrale (21). Des stations de service primaires (14) et des stations de service spécialisées (15) permettent à des spécialistes des soins de santé et à des fournisseurs de soins de santé primaires d'accéder aux informations multimédia téléchargées pour proposer un diagnostic et un traitement ainsi que d'autres services. Une station gestionnaire (16) et une ou plusieurs stations d'analyse (18) permettent de gérer le système ainsi que d'effectuer l'analyse des données. L'accès aux données est accordé sur permission. Le système peut être appliqué à de nombreux scénarios de soins de santé, mais peut être notamment appliqué pour le dépistage, le diagnostic et le traitement ophtalmique et dentaire.
Patent WO-2004016588-A1 (WO)
Title: Derives de furanone et leurs procedes de production
Inventor: KUMAR NARESH
IPC: A01N43/36
Filed: 2003-08-19
Abstract: L'invention concerne de nouveaux procédés de synthèse, des produits obtenus par lesdits procédés et les utilisations de ces produits. En particulier, l'invention concerne des procédés permettant de mettre en réaction des furanones, notamment des fimbrolides, avec des amines. L'invention présente une application particulière dans la synthèse de 1,5-dihydro-pyrrol-2-one halogéné, de 1,5-dihydropyrrol-2-ones substitués par 5-halométhylène (analogues de lactame de fimbrolides), de furanones substitués par 5-amino et de 5-aminométhylène-2(5H)-furanones et de leurs analogues synthétiques. L'invention concerne également de nouveaux composés et leurs utilisations.
Patent WO-2004024342-A1 (WO)
Title: Buse pour cartouches de materiau d'etancheite
Inventor: WILLERS ANDREW
IPC: B05C17/005
Filed: 2003-09-10
Abstract: L'invention concerne une buse (1) pour cartouches de matériau d'étanchéité que l'on utilise généralement pour les pistolets de calfeutrage. La buse (1) comprend une extrémité d'admission (2) qui permet sa fixation à une cartouche. La buse (1) comprend en outre un corps conique (9) qui se termine en sortie (4). Le corps conique (9) comporte une cavité à profil en triangle, courbe ou en forme de croissant. Ledit profil produit un bourrelet de forme correspondante qui permet de travailler ce bourrelet selon un savoir-faire moins élaboré, donnant au matériau d'étanchéité le chanfrein ou le biseau approprié.