baber/WOPTO huggingface dataset:
Patent BR-112022018534-A2 (BR)
Title: Agonistas de receptores de glp oral
Inventor: GILES ALBERT BROWN
IPC: A61K38/26
Filed: 2021-03-16
Abstract: AGONISTAS DE RECEPTORES DE GLP ORAL. A presente invenção refere-se a novos compostos de fórmula (1a) ou fórmula (1b):  e seus sais, em que S, T, W, Z, AA1, AA2, AA3, AA4, AA5, AA6, AA7, AA8, AA9, AA10, AA11, AA12, AA13, AA14, AA15, A16, AA17, AA18, AA19, AA20, AA21, AA22, Sa, Ta, Wa, Xa, Ya, Za, AA1a, AA2a, AA3a, AA4a, AA5a, AA6a, AA7a, AA8a, AA9a, AA10a, AA11a, AA12a, AA13a, AA14a, AA15a, A16a, R, R1 e R2 são definidos neste documento, e seu uso no tratamento, prevenção, melhoria, controle ou redução do risco de distúrbios associados a receptores de peptídeo semelhante a glucagon (GLP).
Patent BR-112022021469-A2 (BR)
Title: Moléculas bifuncionais e métodos de uso das mesmas
Inventor: Nathan Wilson STEBBINS
IPC: A61K31/7105
Filed: 2021-04-21
Abstract: MOLÉCULAS BIFUNCIONAIS E MÉTODOS DE SUA UTILIZAÇÃO. A presente revelação se relaciona geralmente às composições de moléculas bifuncionais sintéticas que compreendem um primeiro domínio que se liga especificamente a um ácido ribonucleico-alvo e um segundo domínio que se liga especificamente a uma proteína-alvo, e usos destas.
Patent BR-112022024856-A2 (BR)
Title: Processo para preparação de fluoxastrobina e seus intermediários
Inventor: DIGISHKUMAR MANUBHAI PANCHAL
IPC: C07D413/12
Filed: 2021-06-08
Abstract: PROCESSO PARA PREPARAÇÃO DE FLUOXASTROBINA E SEUS INTERMEDIÁRIOS. A invenção fornece um processo melhorado para a preparação de fluoxastrobina e seus intermediários. A presente invenção fornece um processo para a preparação de fluoaxastrobina, 4,6-dicloro-5-fluoropirimidina e 2-cloromalonato de dietila que são substancialmente isentos de impurezas indesejadas.
Patent BR-112022026012-A2 (BR)
Title: Unidade de transmissão, trem de força de veículo e veículo
Inventor: STEFAN KARLSSON
IPC: B60K17/08
Filed: 2021-07-27
Abstract: UNIDADE DE TRANSMISSÃO, TREM DE FORÇA DE VEÍCULO E VEÍCULO. A presente invenção refere-se a uma unidade de transmissão (4), um trem de força de veículo (2) e um veículo. A unidade de transmissão (4) compreende um primeiro eixo de transmissão (10) formando um eixo de entrada da unidade de transmissão (4), e um segundo eixo de transmissão (20) compreendendo uma primeira parte de eixo (20a) e uma segunda parte de eixo (20b). A primeira parte de eixo (20a) é conectada de forma rotativa ao primeiro eixo de transmissão (10) através de um primeiro par de engrenagens (11). A unidade de transmissão compreende ainda um terceiro eixo de transmissão (30) conectável de forma rotativa à primeira parte de eixo (20a) por meio de um segundo par de engrenagens (21) e conectável de forma rotativa à segunda parte de eixo (20b) por meio de um terceiro par de engrenagens (31). O segundo e o terceiro par de engrenagens estão dispostos a uma distância um do outro em uma direção paralela ao eixo longitudinal do segundo eixo de transmissão (20) de modo que, quando a unidade de transmissão (4) estiver disposta no trem de força do veículo (2), uma máquina elétrica (3) pode ser disposta entre eles.
Patent BR-112023001112-A2 (BR)
Title: Sistema de travamento para uma tampa de veículo
Inventor: MARCO CIARMATORI
IPC: E05B83/34
Filed: 2021-07-08
Abstract: SISTEMA DE TRAVAMENTO PARA UMA TAMPA DE VEÍCULO. Sistema de travamento (100) para travar uma tampa de veículo compreendendo: uma tampa (103), um atuador de movimento (105) para mover a tampa (103), uma trava (106) compreendendo um pino de rototranslação (2) com uma cabeça (20) adequada para ser engatada em uma base (130) da tampa, um atuador (1) da trava que movimenta o pino de rototranslação (2); o atuador (1) compreende: um motor elétrico (7), e meios de redução de movimento (R); o motor elétrico (7) é configurado adequadamente de forma a girar em uma primeira direção de rotação para mover o pino de rototranslação de uma posição retraída para uma posição extraída, e em uma segunda direção de rotação para mover o pino de rototranslação da posição extraída para a posição retraída.
Patent BR-112023019592-A2 (BR)
Title: Condimento emulsificado
Inventor: BREANNE J MCDAVID
IPC: A23L13/40
Filed: 2022-03-22
Abstract: condimento emulsificado. um condimento emulsificado incluindo sementes de mostarda trituradas, quebradas ou moídas, um componente ácido tal como vinagre, água e uma quantidade em peso significante de um óleo comestível, provê um condimento com uma textura espessa, espalhável, uma sensação cremosa na boca e estabilidade de separação sem a inclusão de gomas ou aditivos que formem emulsão. o processo para fabricar o condimento inclui quebrar grosseiramente sementes de mostarda, misturar as sementes de mostarda com água, um óleo, um componente ácido e água para se obter uma mistura, embeber a mistura com agitação moderada, moer a mistura de pedra e desaerar a mistura.
Patent BR-122016030831-A2 (BR)
Title: sistemas, dispositivos e métodos para interoperação entre evolução a longo prazo e área local sem fio
Inventor: ALEXANDER SIROTKIN
IPC: H04W88/06
Filed: 2015-04-22
Abstract: ?sistemas, dispositivos e métodos para interoperação entre evolução a longo prazo e área local sem fio? as modalidades da presente revelação descrevem sistemas, dispositivos e métodos para a interoperação entre evolução a longo prazo e área local sem fio. várias modalidades podem incluir utilizar as regras de seleção de rede de acesso e direcionamento de tráfego com base nos parâmetros de assistência de rede de acesso de rádio. outras modalidades podem ser descritas ou reivindicadas.
Patent BR-122020014015-A2 (BR)
Title: Aparelho para decodificar um vídeo
Inventor: IL-KOO KIM
Filed: 2011-07-07
Abstract: o método para codificar inclui: determinar um modo de codificação, indicando uma unidade atual de dados para codificação de um quadro e um método de codificação incluindo codificação de predição realizada para a unidade atual de dados; determinar uma ocorrência de mesclagem com pelo menos uma unidade vizinha de dados, baseado em pelo menos um dentre o modo de codificação e o modo de predição; e determinar informações do modo de predição, informações relacionadas à mesclagem, e informações relacionadas à predição, e determinar informações de codificação da unidade de dados, incluindo as informações do modo de predição, as informações relacionadas à mesclagem, e as informações relacionadas à predição.
Patent SK-4996-A3 (SK)
Title: Sugar covering agent and compressed tablet containing its
Inventor: BARCOMB REGINALD J
IPC: A61K47/38
Filed: 1996-01-11
Abstract: A sugar coating composition for application to a compressed medicinal tablet comprising a sugar, a dose of a hormonal steroid and a steroid release rate controlling amount of microcrystalline cellulose.
Patent CZ-20497-A3 (CZ)
Title: Collapsible support plate
Inventor: OHMAN GERTH
IPC: A61G1/01
Filed: 1994-07-26
Abstract: A lying underlay comprises on the one hand a thin first layer (2) of an all-round flexible material of large wear and tear strength, having a substantially elongate basic form and being intended for forming a strong carrier, and on the other hand a considerably thicker second layer (3) which is permanently joined or integrated with the carrier layer (2) and which consists of a porous or fluffy soft material being intended for forming a mattress part. The mattress part (3) is divided into several elongate sections (5, 6, 7) by longitudinal slits (4, 4'), which sections are jointly held together by the carrier layer (2), more precisely in portions (8, 8') forming longitudinal folding lines which permit a folding of the lying underlay into a package in which two mattress sections (6, 7) are folded inwards towards another one (5), the carrier layers (2) of the respective sections being turned towards each other.
Patent CZ-30099-A3 (CZ)
Title: Process and apparatus for bending glass sheets
Inventor: TAKEDA TAKASHI
IPC: C03B35/16
Filed: 1998-06-02
Abstract: In a bending apparatus for glass sheets, at least some of distances between conveyor rolls are set so as to be unequal, forming glass sheets having good quality and free from optical distortion. For the purpose, the distances between conveyor rolls 12A-12G which are provided from an outlet 17 of a heating furnace 16 are set so as to be unequal and to gradually expand toward a downstream direction. <IMAGE>
Patent CZ-31094-A3 (CZ)
Inventor: KUBICEK JAN ING
IPC: C02F1/74
Filed: 1994-02-14
Abstract: Aerační element pro nádrže na úpravu a čištění vody. Obsahuje
rozvodné potrubí (1) a propustnou membránu (2) s
jemným děrováním. Plášť rozvodného potrubí (1) je opatřen
otvory, které jsou membránou (2) překryté, přičemž
membrána (2) je vzduchotěsně pomocí přítlačných pásů (3)
a přítlačných lišt (4) k potrubí připevněna
Patent CZ-9900373-A3 (CZ)
Title: Process for producing waste paper board, waste paper board produced in such a manner and use thereof
Inventor: MACHACEK JAN
IPC: D21B1/32
Filed: 1999-02-04
Abstract: To produce a board material from waste paper, the paper is mixed with water into a paste, and poured into a mold as a pulp. The water is extracted rapidly and the mold contents are compressed in a vertical press. Remaining water is extracted and the resulting material is dried out.  To produce boards from waste paper, additional additives are mixed with the paper mass, and especially colorants, impregnation or waterproof agents which are preferably soluble in water. When the mold is partially filled, strengthening materials are added, and the mold is then topped up and filled. The strengthening materials are of plastics, metal or textiles with their weight reduced by holes or profiles. The dry board material is given a surface treatment as required, and especially a wood veneer, an outer film, paint, plaster, staining, wallpaper or a resin coating. Surplus pulp and water from the mold is returned to the pulp preparation stage. The finished board is composed of 70-80% of bonded paper fibers and 20-30% residual moisture.
Patent SK-89395-A3 (SK)
Title: Container base
Inventor: MOGENSEN ERLING K
IPC: B62B3/02
Filed: 1994-01-14
Abstract: A container base (5) is adapted to receive various types of side-boards owing to a new corner structure. The corner structure is characterized in that coupling means can be inserted in two mutually perpendicular horizontal directions and in a vertical direction. This is achieved in that a pair of pipe profiles (10, 11) has open ends to receive coupling means, and by the provision of a further pipe profile (12) which extends perpendicularly to the pipe profiles (10, 11). The further pipe section is terminated at the same level as or below the lower side wall of the substantially horizontal pipe parts and is secured to the lower wall edges of these. All pipe profiles are located in such a way that they do not prevent introduction of a coupling means into any of the pipe profiles of the corner.
Patent SK-91799-A3 (SK)
Title: Material intended to remineralise organomineral tissues
Inventor: VALIENTE MALMAGRO M
IPC: A61K6/884
Filed: 1997-12-30
Abstract: Together with other accessory products, includes a mixture of ion-exchange resins, cationic and anionic, charged with Ca<2+>, F<-> and PO4<3-> ions, in an approximate molar ratio of 2:1:1, respectively. Particularly preferred is a material in which the resins also have a charge of Zn<2+> ions representing a proportion of less than 1%, preferably close to 0.2% of the dry weight of the resin. The preferred resins are those whose base is cross-linked polystyrene with 2-14% divinylbenzene. The material is useful as first filler in the treatment of caries, especially deep caries, leading to remineralization of the dentin with a composition very close to the original composition, together with high microhardness. It is also useful as a component of dentifrice products such as pastes, elixirs and dental floss.
Patent SK-91997-A3 (SK)
Inventor: LAURO JAN
IPC: F42B33/00
Filed: 1997-07-04
Abstract: Spôsob delaborácie striel plnených bielym fosforom
spočíva v tom, že vo vylievacej nádrži (1) sa pod hladinou
vody (11) s teplotou 60 až 70 °C postupne vyskrutkujú
a vyberú trhacie puzdrá (3) z delaborovaných
striel (2), následne sa strely otočia o 180 °, biely fosfor
v dutine strely (4) sa vplyvom vody (11) s teplotou 60
až 70 °C zohreje, premení sa na tekuté skupenstvo, vytečie
z delaborovanej strely (2) a hromadí sa v spodnej
časti vylievacej nádrže (1) pod hladinou vody (11) bez
styku so vzdušným kyslíkom
Patent AT-522362-A3 (AT)
Title: Halterung für die lösbare Befestigung eines Schilds
Inventor: Roger Gogniat
IPC: G09F7/16
Filed: 2020-03-27
Abstract: Die Halterung sieht ein Halteelement (4,40,60) zur Befestigung der Halterung (1,50,70) am Objekt und ein Verbindungselement (5,41,61) zur Befestigung am Schild (2) vor, wobei das Halteelement (4,40,60) und das Verbindungselement (5,41,61) miteinander lösbar verbindbar sind, dadurch gekennzeichnet, dass das Halteelement (4,40,60) zwei seitlich voneinander und im Abstand zueinander angeordnete, je federelastisch deformierbare fixierende Enden (11,11',44,44', 64,64') aufweist, die sich gegen das betriebsfähig positionierte Verbindungselement (5,41,61) erstrecken und dazu bogenförmig gegen dieses hin gekrümmt sind und das Verbindungselement (5,41,61) zwei gegengleich zu den fixierenden Enden (11,11',44,44',64,64') des Halteelements (4,40,60) angeordnete, je federelastisch deformierbare sich fixierende Enden (14,14', 51,51', 71,71') aufweist, die sich gegen das Halteelement (4,40,60) erstrecken und dazu bogenförmig und gegengleich zu den fixierenden Enden (11,11',44,44',64,64') gekrümmt sind, derart, dass sie mit diesen je eine lösbare Rastverbindung bilden, und dass weiter das Halteelement (4,40,60) im Abstand über eine Höhe zu den fixierenden Enden wenigstens eine Einschubrinne (12,12',46,66,66') für eine am Verbindungselement (5,41,61) vorgesehene, im gleichen Abstand zu den sich fixierenden Enden (14,14'51,51',71,71') angeordneten Einschubführung (15,15', 53,73,73') aufweist, derart, dass das Verbindungselement (5,41,61) mit der Einschubführung (15,15',53,73,73') voran in die Einschubrinne (15,15',53,73,73') hinein steckbar ist und durch eine Verschwenkbewegung mit in der Einschubrinne (15,15',53, 73,73') positionierten Einschubführung (15,15',53,73, 73') mit dem Halteelement (4,40,60) in die Rastverbindung gebracht und aus dieser wieder gelöst werden kann.
Patent CZ-109393-A3 (CZ)
Title: Bonded proteins
Inventor: KUBIAK TERESA M
IPC: A61K38/26
Filed: 1991-12-12
Abstract: A non-naturally-occurring fusion protein comprising an extension peptide portion covalently linked at its C-terminus to the N-terminus of a biologically active portion is disclosed. The extension peptide portion can be removed by DPP IV cleavage. A use of fusion proteins with DPP IV cleavable extension peptide portions in medecinal preparations is disclosed. A method of purifying desired proteins from a mixture containing a fusion protein is disclosed.
Patent CZ-106798-A3 (CZ)
Title: Holder for elongation of brush handle
Inventor: LEH NORBERT
IPC: A46B3/12
Filed: 1998-04-08
Abstract: The holder (5) comprises a handle (4), two plastics clamping arms (1), and a plastics clamping ring (2). The clamping arms form a mounting (7) for the paint brush shaft end. The clamping ring is slidable along the clamping arms, such that by sliding the ring in the direction of the free ends (8) of the clamping arm, the inserted shaft end is gripped between the arms. The clamping arms have knubs (3) at the inner surfaces of the free arms. The handle has a mounting opening (9) in which a rod-end of a telescopic rod may be inserted.
Patent CZ-117797-A3 (CZ)
Title: Heterocyclic compounds and pharmaceutical compositions based thereon
Inventor: STEVENS RODNEY W
IPC: A61P43/00
Filed: 1995-05-29
Abstract: Novel compounds having the ability to inhibit 5-lipoxygenase enzyme and having formula (I) and the pharmaceutically acceptable salts thereof, wherein Ar<1> is a heterocyclic moiety which is selected from imidazolyl, pyrrolyl, pyrazolyl, 1,2,3-triazolyl, 1,2,4-triazolyl, indolyl, indazolyl and benzimidazolyl, which is bonded to X<1> through a ring nitrogen atom, and which may be optionally substituted with one or two substituents selected from halo, hydroxy, cyano, amino, C1-4 alkyl and the like; X<1> is a direct bond or C1-4 alkylene; Ar<2> is phenylene optionally substituted with halo, hydroxy, cyano, amino and the like;  X<2> is -A-X- or -X-A- wherein A is a direct bond or C1-4 alkylene and X is oxy, thio, sulfinyl or sulfonyl; Ar<3> is phenylene, pyridylene, thienylene, furylene, oxazolylene or thiazolylene optionally substituted with one or two substituents selected from halo, hydroxy, cyano, amino, C1-4 alkyl and the like; R<1> and R<2> are each C1-4 alkyl, or together they form a group of formula -D<1>-Z-D<2>- which together with the carbon atom to which it is attached defines a ring having 3 to 8 atoms, wherein D<1> and D<2> are C1-4 alkylene and Z is a direct bond or oxy, thio, sulfinyl, sulfonyl, or vinylene, and D<1> and D<2> may be substituted by C1-3 alkyl; and Y is CONR<3>R<4>, CN, C(R<3>)=N-OR<4>, COOR<3>, COR<3> or CSNR<3>R<4>, wherein R<3> and R<4> are each H or C1-4 alkyl. These compounds are useful in the treatment or alleviation of inflammatory diseases, allergy and cardiovascular diseases in mammals and as the active ingredient in pharmaceutical compositions for treating such conditions.
Patent CZ-128096-A3 (CZ)
Title: Charged liposome preparation
Inventor: KRAUSE WERNER
IPC: A61K9/127
Filed: 1994-11-04
Abstract: The invention relates to a method of administering a liposome preparation having an effective amount of an electrically charged component which is effective in reducing adverse effects of a liposome preparation, e.g., in reducing hemodynamic effects, and improving host tolerance.
Patent CZ-145693-A3 (CZ)
Title: Novel herbicides
Inventor: CRAMP SUSAN MARY
IPC: C07C49/84
Filed: 1993-07-20
Abstract: 4-Benzoylisoxazole derivatives of formula (I): <CHEM>     wherein:     R represents hydrogen or -CO2R<4>; R<1> represents alkyl, haloalkyl or optionally substituted cycloalkyl; R<2> represents halogen, alkyl, haloalkyl or alkyl substituted by -OR<5>, or a group selected from nitro, cyano, -CO2R<4>, -S(O)pR<6>, -O(CH2)rOR<5> and -OR<5>;     R<3> represents optionally substituted phenyl;     X represents oxygen or -S(O)q-;     n represents zero or an integer from one to four;     R<4> and R<5> independently represent alkyl or haloalkyl; R<6> represents alkyl, haloalkyl or optionally substituted phenyl;  R<7> represents halogen, alkyl or haloalkyl or a group selected from nitro, cyano, -OR<5> and -S(O)pR<6>;     p represents 0, 1 or 2; q represents 0, 1 or 2;     r represents 1, 2 or 3; the herbicidal properties of these derivatives and their application to crop protection is described.
Patent CZ-149697-A3 (CZ)
Inventor: KOULISIANIS ANASTASIOS ING
IPC: F41B11/62
Filed: 1997-05-15
Abstract: Vynález se týká expanzní pistole, zejména plynovky
nebo akustické pistole, obsahující vratně
přestavitelný zápalník /7/ uložený ve vratně
přestavitelném závěru /6/ proti nábojové
komoře /3/, přičemž zápalník /7/ je spřažen
se západkou pojistky /9/. Minimální vzdálenost
dna nábojové komory /3/ od čelní plochy
/62/ je rovna délce vkládané nábojky /4/,
přičemž zápalník / 7 / je spřažen s prostředky,
které zabraňují jeho pohybu při vložení delšího
ostrého náboje /41/ do nábojové komory
/3/.
Patent CZ-174999-A3 (CZ)
Title: Novel utilization of 2-amino-1,3-propanediole derivatives
Inventor: COTTENS SYLVAIN
IPC: A61K31/137
Filed: 1997-11-17
Abstract: Combined use of a compound of formula I  wherein     R1   is an optionally substituted straight- or branched carbon chain having 12 to 22 carbon atoms which may be optionally interrupted by an optionally substituted phenylene, and    each of R 2 , R 3 , R 4  and R 5 , independently, is H or lower alkyl,  in free form or in pharmaceutically acceptable salt form, with 40-O-(2-hydroxyethyl)-rapamycin or with an immuno-suppressive monoclonal antibody.
Patent CZ-9502000-A3 (CZ)
Title: Process of separating by flotation and apparatus for making the same
Inventor: CHUDACEK MICHAEL WENZEL
IPC: B03D1/14
Filed: 1994-01-20
Abstract: A suitably conditioned slurry feed is introduced to a trough (1) from which it is distributed into a slurry layer-flow forming chamber (2). Chamber (2) is provided with a discharge weir (3) which discharges an evenly spread layer of slurry (4) onto an inclined plate (5) feeding into a mixing passage (6). Recirculated slurry from vessel (7) is also fed into mixing passage (6) via a recycle gate (8) which forms it into a layer of slurry (9). An array of clean liquid jets (12) accelerates thin gas envelopes and impinges between layers of slurry (4) and (9) causing intensive mixing of all streams in mixing passage (6). The high shear rate produces high intensity turbulence and shears gas into very small bubbles. A multiphase mixture flow is discharged from mixing passage (6) into vessel (7), where it flows past one or more longitudinal stabilizing baffles (13). Gas bubbles loaded with hydrophobic particles disengage from the stream, rise towards the liquid surface and are diverted by bubble diverting guides (14) towards the froth discharge end of the vessel. A layer of froth travels towards froth weir (15) where it is discharged. The residual slurry leaves discharge launder (19) via a weir (20) to the next flotation cell or process stage.
Patent CZ-201038-A3 (CZ)
Inventor: STACH JAN
IPC: A61K31/40
Filed: 2010-01-19
Abstract: Rešení se týká nového, pro prumyslovou výrobu vetších množství vhodného zpusobu výroby amorfní formy hemivápenaté soli (3R,5R) 7-[3-fenyl-4-fenylkarbamoyl-2-(4-fluorfenyl)-5-isopropylpyrrol-1-yl]-3,5-dihydroxyheptanové kyseliny (atorvastatinu vzorce I) s nízkým specifickým povrchem založeného na rízeném srážení a jeho použití v lékové forme.
Patent CZ-220599-A3 (CZ)
Title: Camptothecine analogs, their use as medicaments and pharmaceutical compositions containing thereof
Inventor: BIGG DENNIS
IPC: A61K31/4709
Filed: 1997-12-05
Abstract: The invention concerns novel counterparts of camptothecin and particularly the products complying with the following formulae: -5-ethyl-9,10-difluoro-4,5-dihydro-5-hydroxy-12- (4-methyl piperidinomethyl) -1H-oxepino[3', 4':6,7]indolizino[1,2-b] quinolein-3,15(4H,13H)-dione; -5-ethyl-12-diethylaminomethyl-9-fluoro-4,5-dihydro-5-hydroxy-10-methyl-1H-oxepino [3',4':6,7] indolizino[1,2-b]quinolein-3,15(4H,13H)-dione; -5-ethyl-9-fluoro-4,5-dihydro-5-hydroxy-10-methyl-12- (4-methyl piperidinomethyl) -1H-oxepino[3',4':6,7]indolizino[1,2-b]quinolein-3,15(4H,13H)-dione. The invention also concerns their application as medicines, the pharmaceutical compositions containing them and their use in producing tumoricidal, antiviral or parasiticide medicines.
Patent CZ-250098-A3 (CZ)
Inventor: KALINDJIAN SARKIS BARRET
IPC: C07D401/12
Filed: 1997-02-10
Abstract: Sloučeniny obecného vzorce I a II, ve kterémR1 představuje G^o
hydrokarbylovou skupinu, R2 znamená atomvodíku nebo Q_3
alkylovou skupinu, mje 1 až 15, nje 2 až 6, každá ze skupinX
znamená navzájemna sobě nezávisle skupinu a nebojedna ze
skupin Xznamená skupinu -NR4/-, -O- nebo -S- azbývající
skupinyXznamenají nezávisle na sobě skupiny/a/, ve kterých: R3
znamená atomvodíku, C,.6 alkylovou skupinu, skupinu -CQ2R5, -
COjNR5, -CR5 2QR6 nebo -OR5 /ve kterýchR5 aR6 znamenají
vodík nebo Ci_3 alkylovou skupinu/, aR4 je vodík nebo Cw
alkylová skupina, každá ze skupin Yznamenánavzájemna sobě
nezávisle skupinu -CZR3/R4- nebo až dvě tyto skupiny Y
představují nezávisle skupinu -NU4/-, -O- nebo -S- azbývající
skupinyYpředstavují na sobě nezávisle skupinu -C/R3/R4-, aZ
znamená skupinuX7R7/NR2- nebo >N-, kde R7 znamená
libovolnou skupinou uvedenou výše v případě R3, a farmaceuticky
přijatelné soli těchto sloučenin, které představují ligandy na