baber/WOPTO huggingface dataset:
Patent PT-719253-E (PT)
Inventor: NAKANE MASAMI
IPC: A61P29/00
Filed: 1994-09-13
Abstract: A compound of the chemical formula (I) and its pharmaceutically acceptable salt, wherein Y is C2-C4 alkylene; Z is a valence bond or C1-C6 alkylene; R<1> is substituted or unsubstituted aryl (e.g., phenyl and naphthyl) or heteroaryl (e.g., thienyl and furyl); R<2> is hydrogen or C1-C6 alkyl; R<3> is hydrogen, hydroxy or the like; R<4> is substituted or unsubstituted benzyl or the like. Typical examples are (2S*,3S*,4S*,5R*)-4-Carboxy-3-[N-(5-Isopropyl-2-methoxy-benzyl)amino]-5-methyl-2-phenylpyrrolidine and (2S*,3S*,5S*)-5-Carboxy-3-[N-(2-methoxy-5-trifluoromethoxybenzyl)amino]-2-phenylpiperidine. The novel substituted azaheterocyclecarboxylic acids in this invention have excellent substance P antagonistic activity and are thus useful for the treatement of gastrointestinal disorders, central nervous system disorders, allergy, inflammatory diseases, asthma, pain, emesis or migraine in mammals, especially humans.
Patent PT-698707-E (PT)
Inventor: HELLWIG VOLKER
IPC: E05B65/462
Filed: 1995-08-16
Abstract: The mechanism comprises two drive elements (7,14), each of which runs along a dimension of the tool trolley. One element (7) is horizontal and the other (14) is vertical. Both drive elements are so joined to each other that they must be moved together. For every object to be secured by a locking action, a locking hook (11,12,19,22) is arranged on one of the two drive elements. The drive elements take the form of displaceable bars (8,9,15) connected by a twin-armed lever (10).
Patent PT-699494-E (PT)
IPC: B23C3/05
Filed: 1995-08-16
Abstract: The milling tool has the tool bit (5) held in a tool holder (3) with axial movement. The servo drive to feed out the tool bit can be powered by a hydraulic cylinder (35) and operates on an axially moving profile section (15) inside the tool holder. The tool head is removable from the mounting by a simple coupling. The coolant flow to the tool head is combined with the hydraulic system. The tool head has a concentric bore and is coupled to the mounting via a simple coupling which can be operated by robotics and which requires no special tools and fittings.
Patent PT-785716-E (PT)
Title: Cytokine designated lerk-6
Inventor: CERRETTI DOUGLAS P
IPC: G01N33/53
Filed: 1995-10-04
Abstract: The invention is directed to LERK-6 as a purified and isolated protein, the DNA encoding the LERK-6, host cells transfected with cDNAs encoding LERK-6.
Patent PT-830797-E (PT)
Inventor: BUYTAERT STEVEN HERWIG CYRIEL
IPC: G01S5/14
Filed: 1996-04-26
Abstract: A method for communicating with an object, for example a vehicle, using a wide area paging network and a cellular mobile communication network that includes the steps of coupling a module with at least a transmitter and a receiver to the object and using the module for communicating with in combination at least three communication networks, the first one being the wide area paging network, the second one being the cellular mobile communication network and the third one being a local network using a spread spectrum modulation method.
Patent PT-974355-E (PT)
Inventor: ASHIDA HIROSHI
IPC: A61K31/19
Filed: 1996-10-23
Abstract: PCT No. PCT/JP96/03079 Sec. 371 Date Mar. 13, 1997 Sec. 102(e) Date Mar. 13, 1997 PCT Filed Oct. 23, 1996 PCT Pub. No. WO98/09624 PCT Pub. Date Mar. 12, 1998There is disclosed a water-soluble vitamin composition which containing about 90 to 99.8% by weight of a water-soluble vitamin, a polymer binder and at least one additive selected from the group consisting of monosaccharides, disaccharides, sugar alcohols, dextrin and organic acids, which can provide a tablet having high mechanical strength (hardness) with less compression problem and easy disintegration, upon compression. A process for producing the composition is also disclosed.
Patent PT-852205-E (PT)
Inventor: WAGNER ARMAND
IPC: B65D41/48
Filed: 1997-12-12
Abstract: The cap (1) has a flat top, an inner ring (10) which fits inside the bottle neck, and an outer skirt (2) with an inner projection (23) which locks the cap in place when it is forced over a collar (C) on the bottle neck. An upper section which forms a security strip (12). One end of the security strip has a tongue (22) which is designed to be gripped to remove the strip, the tongue having an inner surface (22a) which causes it to be pushed outwards when the cap is fitted, making it easier to grip. In a variant of the design the security strip can be made to cover only part of the circumference of the bottle neck, the remainder acting as a hinge for the top of the cap when it is opened and closed.
Patent PT-935684-E (PT)
Inventor: PLEMMONS HAROLD F
IPC: D04B7/34
Filed: 1997-10-20
Abstract: A knitted glove including a thumb and a body, a crotch defined between the thumb and the body, and a thickened knitted portion along at least a portion of the crotch. The present invention is further directed to a method and apparatus for forming such a knitted glove.
Patent PT-901555-E (PT)
Inventor: PERAZZO PIERLUIGI
IPC: E05F11/48
Filed: 1997-05-20
Abstract: A cable transmission connected to a drive unit comprises a pair of flexible sheaths (32, 34) each having a first end anchored to a housing of the drive unit and a second end anchored to a slide (22) which supports a pane and is slidable along a track (20). A flexible cable which extends around a drum of the drive unit comprises two branches (46, 48) slidable in the respective sheaths (32, 34). The slide (22) has a pair of internal ducts (50, 52) for guiding the branches (46, 48) of the cable, the ducts extending between inlet openings, to which the second ends of the sheaths (32, 34) are anchored, and respective opposed outlets facing towards respective opposite ends of the track (20). The two opposite ends of the cable are anchored to the respective ends of the track (20) so that respective portions (46a, 48a) of the cable disposed between the respective outlets and the respective ends of the track (20) extend parallel to the track.
Patent PT-900240-E (PT)
Inventor: MELDER JOHANN-PETER
IPC: C08F8/08
Filed: 1997-05-20
Abstract: PCT No. PCT/EP97/02571 Sec. 371 Date Nov. 5, 1998 Sec. 102(e) Date Nov. 5, 1998 PCT Filed May 20, 1997 PCT Pub. No. WO97/44366 PCT Pub. Date Nov. 27, 1997Polyalkeneamines of the formula (I) where R1, R2, R3, R4, R5 and R6 may have different meanings, are prepared by a process in which a polyalkene epoxide is reacted with an amine and the amino alcohol is dehydrated and reduced to give the compound of the formula (I).
Patent PT-946910-E (PT)
Inventor: MEWES FRANK
IPC: G01F25/00
Filed: 1997-11-13
Abstract: A flow regulation control valve for regulating volume flows in pipelines including valve housing with a flow chamber, a control or shut-off member arranged in the flow chamber for setting a desired flow state through the valve, at least one sensor arranged in the vicinity of the flow chamber of the valve housing for sensing a characteristic value of the flow through the flow chamber, an electronic data store or memory for storing specific characteristic values of the housing of the flow regulation control valve, and an evaluation unit which is connected to the sensor and determines the volume flow from the values measured by the sensor with reference to the characteristic values of the valve stored in the data store.
Patent PT-1032361-E (PT)
Inventor: PLASCHKE KIM
IPC: A61K8/49
Filed: 1998-11-19
Abstract: A flavonoid-containing sunscreen composition having UV absorbency at 282 nm in water contains at least one flavanone and at least one flavone, the flavanone providing 75 to 98% of the UV absorbency at 282 nm and the flavone providing 2 to 25% of the absorbency at 282 nm. The composition is formed of flavonoids extracted from citrus fruit using water, and separating the extracted flavonoids using a sorbent material, and then recovering the flavonoids from the sorbent material using a solvent.
Patent PT-1119448-E (PT)
Inventor: DUFORT JOHN FRANCIS
IPC: B44F1/06
Filed: 1999-06-18
Abstract: A lithophane-like article and a method of forming such an article, for example formed of plastics, confectionery product, soap, wax or liquid, by determining the intensity of different points of an original image (1), and forming the article with a thickness at each point of the article related to the intensity of the corresponding point of the original image (1). <IMAGE>
Patent PT-1141108-E (PT)
Inventor: POUCHELON ALAIN
IPC: C08K9/06
Filed: 1999-12-21
Abstract: The invention concerns a method for preparing a silica suspension in a silicone matrix, said suspension capable of being used for producing organopolysiloxanes crosslinkable by polycondensation. The invention aims at seeking a technical compromise between the rheology of said compositions and the mechanical properties of the resulting crosslinked elastomers. As a solution, the invention discloses a method for preparing a silica suspension treated with organosilazane in a silicone material comprising a linear reactive polyorganosiloxane bearing for example at each chain end a hydroxy group. The invention is characterized in that it consists essentially in introducing the organosilozane in the preparation medium: before and/or substantially simultaneously before bringing together at least part of the silicone material and the particulate filler used, said organosilozane introduction being carried out with a fraction of organosilazane corresponding to a proportion ranging between 8% and 30% by dry weight relatively to the silica filler, and after bringing together the filler and all or part of the silicone material.
Patent PT-1141337-E (PT)
Title: Gram-positive bacteria deprived of htra proteasic activity and their uses
Inventor: POQUET ISABELLE
IPC: C12N15/74
Filed: 1999-12-23
Abstract: The invention concerns bacteria strains, obtained from gram-positive bacteria whereof the genome size is not more than 3.2 Mb, and wherein the HtrA surface protease is inactive. Said strains are useful for expressing exported proteins of interest.
Patent PT-1143937-E (PT)
Inventor: KRISHNAMURTH N THINNAYAM
IPC: A61K9/26
Filed: 1999-12-17
Abstract: The invention is directed to oral modified/controlled release drug formulations which provide a rapid initial onset of effect and a prolonged duration of effect. Preferably, the peak concentration is lower than that provided by the reference standard for immediate release formulations of the drug, and the duration of effect falls rapidly at the end of the dosing interval.
Patent SG-80190-G (SG)
Title: (r)-alpha-ethyl-2-oxo-1-pyrrolidinacetamide
IPC: C07D207/27
Filed: 1990-10-02
Abstract: (R)-alpha-ethyl-2-oxo-1-pyrrolidineacetamide, its preparation and pharmaceutical compositions containing the same. It can be prepared either by reacting (R)-alpha-ethyl-2-oxo-1-pyrrolidineactic acid successively with an alkyl haloformate and with ammonia, or, by cyclizing an (R)-2-amino-butanamide of the formula X-CH2CH2-Y-NHCH (C2H5)CONH2 wherein Y is a -CH2-radical when X represents a ZOOC-radical and Y is a -CO-radical when X represents a HalCH2-radical, Z being a C1-C4 alkyl radical and Hal a halogen atom. This dextrorotatory enantiomer has been found to have significantly higher mnemic activity and lower toxicity than the corresponding racemate.
Patent IE-840011-L (IE)
Title: Thioureidophenyl anthelmintics
IPC: A61K31/325
Filed: 1984-01-05
Abstract: 1-(3,4-bis-(3-lower alkoxycarbonyl)-2-thioureido)-phenyl)-1-phenylethylenes, which have anthelmintic activity, are prepared by reacting various 1-(3,4-diaminophenyl)-1-phenylethylenes with an alkoxycarbonylisothiocyanate which is prepared, in turn, from an alkali metal thiocyanate and a lower alkyl haloformate.
[US4438135A]
Patent IE-820125-L (IE)
Title: Composition
IPC: A01N37/46
Filed: 1982-01-21
Abstract: The use as a fungicide of an N-acyl N-hydroxy amino acetic acid of the general formula RCO - @@ - CH2 - COOH (I) or a salt or an ester thereof, wherein R represents a hydrogen atom, an alkyl group or an aryl group.
[EP0057028A2]
Patent IE-820182-L (IE)
Title: Bandages
IPC: C08G18/22
Filed: 1982-01-27
Abstract: Water hardenable splinting bandages comprising a flexible fabric carrying an isocyanate terminated prepolymer having a reaction functionality of not less than two and a catalyst which bandage is characterised in that the prepo-Iymer is a water absorbing isocyanate terminated prepolymer and the catalyst is water soluble but insoluble in the prepolymer, compositions therefore and processes of manufacture thereof are described.
Patent IE-870382-L (IE)
Title: Locking mechanism for prosthesis components
IPC: F16B21/18
Filed: 1987-02-13
Abstract: A socket insert component (14) of an acetabular cup prosthesis (10) is held securely within its support shell (12) by a locking mechanism comprising a circumferential groove (28) in the shell concavity (18) perpendicular to the longitudinal axis (24) of the concavity, a first circumferential rib (38) on the outer surface (32) of the insert congruent with the groove, and a second circumferential rib (40) on the outer surface (32) of the insert (14) parallel to and proximate the first rib (38), the first rib (38) snapping into the groove (28) and the second rib (40) being deformed and pressed against the concavity (18) when the insert (14) and shell (12) are assembled.
Patent IE-35076-L (IE)
Title: PRODUCTION OF PNPase
IPC: C12P19/34
Filed: 1971-04-29
Abstract: The enzyme (PNPase) is obtd. by (a) suspending a cell mass separated from a Micrococcus lacteus fermentation medium in aqs. saline soln., and homogenising or lysing the suspension to rupture the cells to give a suspension of insol. cell debris in an aqs. PNPase soln.; (b) adding (NH4)2SO4 to a concn. of approx. 24% and centrifuging to remove the cell debris and some protein material; (c) adding to the supernatant of aqs. PNPase sufficient lower alkanol to ppt. almost all of the PNPase, and centrifuging the aqs. alcoholic mixt. to recover the ppted. enzyme. PNPase catalyses the polymerisation of nucleoside diphosphates to polynucleotides. For use as a catalyst, the enzyme is covalently bound to activated cellulose.
[FR2091158A5]
Patent FI-813746-L (FI)
Inventor: PORRMANN HERBERT
IPC: A22C13/00
Filed: 1981-11-24
Abstract: Disclosed is a tubular casing comprising a fiber-reinforced regenerated cellulose wherein the fiber-reinforcement comprises a fiber web comprising first and second edge regions, parallel to the longitudinal axis, which are overlapped and bonded to form a tube; an impregnation layer of a thermoplastic synthetic resin applied on the entire inwardly-facing surface of the fiber-reinforcement and present in a weight per unit area of less than about 50 g/m2, the impregnation layer comprising the bond for the edge regions; and a regenerated cellulose surface on the outer surface of the fiber-reinforcement. Also disclosed is a process for manufacturing the tubular casing.
Patent FI-831849-L (FI)
Inventor: SEGAUD CHRISTIAN
IPC: C08K9/04
Filed: 1983-05-24
Abstract: Molding compositions for the fabrication of shaped articles having enhanced mechanical properties are comprised of (i) a polymeric matrix, (ii) an inorganic reinforcing filler material therefor, and, advantageously, (iii) a polymer/filler coupling agent, said reinforcing filler material consisting essentially of intimate admixture of enstatite and silica advantageously prepared by calcination of a precursor clay at a temperature of at least 800 DEG C.
Patent FI-832348-L (FI)
Inventor: HAAS MAX
IPC: E06B1/62
Filed: 1983-06-28
Abstract: The lift landing door frame arrangement contains horizontally adjustable lateral caulking or sealing elements arranged at uprights of the door frame and a vertically adjustable top caulking or sealing element associated with the topside of the door frame. To avoid retouching due to the caulking elements at the time of placement of the lift landing door frame arrangement and to avoid the formation of gaps in the door frame after placement, each lateral caulking element comprises a rectangular sheet metal panel of a length which exceeds the height of the door frame. Each lateral caulking element engages with and is fixed to the interior of the related upright. Each lateral caulking element is also guided for simultaneous vertical and horizontal adjustment at a guide plate carried by the related upright. The vertically adjustable top caulking element is constituted by a U-shaped sheet metal strap which is disposed astride the front parts of the door frame and is laterally guided thereat. This lift landing door frame arrangement is particularly suitable in cases in which the lift or elevator shaft does not include lateral masonry returns at the landing openings.
Patent FI-844193-L (FI)
Inventor: LUNDBAECK STIG
IPC: A61B5/296
Filed: 1984-10-25
Abstract: The invention relates to an electrode intended, for example, for electrocardiogram examinations, and capable of being held in position by suction. Vacuum conditions are created through a hose or tube (8), through which a measuring conductor (7) is drawn. The electrode comprises an inflexible backpiece (3), an intermediate component (2) made of an elastomeric material, and an electrode plate (1), preferably made of a silver-coated plastics. The intermediate component (2) includes a relatively inflexible sealing ring (9) which, in the operative state of the electrode, supports against the skin of a patient via a sealing lip (13) and against the opposing side of the backpiece (3). The electrode plate (1) is firmly connected to the backpiece, while the sealing ring carried by the intermediate component (2) is movable and can be readily sprung away from the backpiece (via resilient means 17). When no load is exerted on the lip-side of the ring and the ring is thus urged outwardly, a vacuum valve is closed automatically through the intermediate component (2), and is re-opened when the electrode is pressed against the surface of the skin, whereupon the electrode is held firmly by suction.
Patent IE-791014-L (IE)
Title: Method of firing ceramic products
IPC: F27B9/14
Filed: 1979-08-08
Abstract: Clay pipes and the like (3) are fired in a kiln (1) through which they are conveyed by a pusher conveyer (2, 4) as individual articles, instead of being carried on cars or in containers. In the main firing zone of the kiln the pipes (3) roll along a surface (6) to maintain roundness and ensure uniform heating. In the preheating zone of the kiln the pipes are carried by carriers (5) of the conveyer without rotating. The pipes may also be carried without rotating in the final cooling zone of the kiln.
[US4264301A]
Patent IE-36801-L (IE)
Title: Spiral springs
IPC: B21F3/08
Filed: 1972-07-31
Abstract: 1341579 Coiling spirals TENSATOR Ltd 12 May 1972 [25 Aug 1971] 39977/71 Heading B3E [Also in Division F2] A method of making a spiral spring comprises forming a strip of spring material so that one end is set to form a spiral coil while the remainder is straight or is set to coil spirally around the coiled end with a radius of curvature substantially greater than that of the coiled end, and then backwinding at least the coiled end. Fig. 1 shows a configuration before baokwinding, in which one quarter of the total length may be close or open coiled at 1. An attachment part 3 is then secured to an arbor and the spring is reverse wound about the arbor, so as to acquire a permanent set in the reverse sense corresponding to the unstressed configuration of Fig. 3. While still wound on the arbor, the spring is inserted into a casing to which end 4 is attached. The arbor may then be arranged to drive a seat belt reel, providing a rapid rise in torque during initial winding up, followed by a slower rise in torque.
[GB1341579A]
Patent IE-41644-L (IE)
Title: Power supply circuits
IPC: H04M1/31
Filed: 1975-07-29
Abstract: 1472442 Sub-station circuits STANDARD TELEPHONES & CABLES Ltd 30 July 1974 33570/74 Heading H4K A power supply arrangement for maintaining power to the circuitry of a telephone set during loop disconnect signalling comprises a capacitor C charged from the exchange battery via a rectifier bridge 3 and an arrangement of a Zener diode ZD and transistors TR1, TR2. The arrangement of the Zener diode and transistors is such as to ensure that the voltage across capacitor C is mainteined at or below a predetermined limit: To improve the response of the circuit to low line voltages and currents the slope resistance of the Zener diode can be reduced by connecting a parallel arrangement of a resistor and the collector base junction of a transistor in series with the diode, the collector emitter junction of the transistor being connected in the line loop (Fig. 2, not shown). The rectifier bridge 3 may be a diode bridge, or a transistor diode bridge as shown in Fig. 3. The load L may be the circuitry of a pushbutton type dialling apparatus of the type in which the actuation of a push-button causes loop-disconnect impulses to be transmitted.
[GB1472442A]
Patent IE-39686-L (IE)
Title: p-BIPHENYLYL ESTERS OF 15- SUBSTITUTED -16, 17, 18, 19 ,20-¹PENTANORPROSTAGLANDINS
IPC: C07D307/935
Filed: 1973-11-08
Abstract: 1456511 Prostaglandins PFIZER Inc 1 Nov 1973 [8 Nov 1972] 50889/73 Heading C2C The invention comprises prostaglandins of the formula I and the C 15 epimers thereof, wherein A is Ar(CH 2 ) n - or -(CH 2 ) m -OR<SP>2</SP>, W is a single bond or cis double bond, Z is a single bond or trans double bond; m is oxo or n is 0 to 5 when Z is a single bond, or n is 1 to 5 when Z is a trans double bond; m is 2 or 3; R<SP>2</SP> is C 1-4 alkyl; Ar is α- or #-furyl, α- or #-thienyl, α- or #-naphthyl, 3,4-dimethoxyphenyl, 3,4-methylenedioxyphenyl, 3,4,5-trimethoxyphenyl or phenyl optionally monosubstituted by halogen, trifluoromethyl, phenyl, C 1-4 alkyl or C 1-4 alkoxy; R 1 is p-biphenylyl, R is H or C 1-4 alkyl, X and Y together form a single bond or X is H and Y is alpha-hydroxy, with the proviso that when X and Y form a single bond m is oxo; and compounds of the Formulµ II, III and VI or and their C 15 epimers, wherein m is oxo or Compounds of Formula I above are obtained by esterifying the corresponding acids of Formula I in which R<SP>1</SP> and X are hydrogen and Y is alpha-hydroxy with p-phenylphenol, and if desired, dehydrating the resulting compounds in which m is oxo and Y is alpha-hydroxy. The esters of the prostaglandin E and F series may also be obtained by hydrolysing the corresponding 11,15-bis-(tetrahydropyranyl) ethers of Formula VI above which are obtained by reacting compounds of the Formula VII with compounds of the formula and if desired, oxidizing and/or hydrogenating the resulting compounds of formula VI above in which m is Compounds of Formula II and III above are obtained by reacting compounds of formula VII above with compounds of the formula and if desired, oxidizing and/or hydrogenating the resulting compounds of Formula II above. Biphenylyl 9,15 - dioxo - 11α - hydroxy - 17- phenyl - 18,19,20 - trinor - cis - 5, trans - 13- prostadienoate is obtained by oxidizing biphenylyl 9 - oxo - 11α,15# - dihydroxy - 17- phenyl - 18,19,20 - trinor - cis - 5, trans - 13- prostadienoate with manganese dioxide. Pharmaceutical compositions, suitable for oral, intravaginal, intraamniotically, intravenous or intranasal administration, contain the above esters of Formula I together with suitable carriers or diluents. The compound possess similar pharmacological properties to those of the naturally occurring prostaglandins. Reference has been directed by the Comptroller to Specifications 1,386,146, 1,345,934 and 1,324,737.
[GB1456511A]
Patent IE-44472-L (IE)
Title: Producing urethanes
IPC: C07C239/00
Filed: 1976-12-03
Abstract: Aromatic urethans are prepared by reacting aromatic carbonates with aliphatic amines, within an organic solvent or not. It is preferred that a stoichiometric quantity of the amine be employed to prevent the formation of urea by-products which are likely to be formed if an excess of the amine is used. The temperature should not exceed 100 DEG C, the interval between 20 DEG and 40 DEG C being preferred. Nearly quantitative yields are obtained. (From US4097676 A) [FR2333779A1]