baber/WOPTO huggingface dataset:
Patent AU-4600393-A (AU)
Title: Excitatory amino acid receptor antagonists
Inventor: ARNOLD MACKLIN BRIAN
IPC: C07D417/06
Filed: 1993-08-31
Abstract: This invention provides novel decahydroisoquinoline compounds which are useful as excitatory amino acid receptor antagonists and in the treatment of neurological disorders. This invention also provides synthetic methods for preparing decahydroisoquinolines, as well as, novel intermediates in the synthesis thereof. The novel pharmaceutical compounds have the formula <CHEM>  wherein: R<1> is hydrogen, C1-C10 alkyl, arylalkyl, alkoxycarbonyl or acyl;  R<2> is hydrogen, C1-C6 alkyl, substituted alkyl, cycloalkyl, or arylalkyl;     R<3> is CO2H, SO3H, CONHSO2R<8>, or a group of formula <CHEM>   <CHEM>   <CHEM>     W is (CH2)n, S, SO, SO2;     Y is CHR<7>, NR<4>, O, S, SO, or SO2;     Z is NR<6>, CHR<7>, or CH; or W and Y together are HC=CH or C IDENTICAL C, or Y and Z together are HC=CH or C IDENTICAL C;     R<4> is hydrogen, C1-C4 alkyl, phenyl, or acyl; R<5> is hydrogen, C1-C4 alkyl, CF3, phenyl, hydroxy, amino, bromo, iodo, or chloro;     R<6> is acyl; R<7> is independently hydrogen, C1-C4 alkyl, phenyl, or substituted phenyl;     R<8> is C1-C4 alkyl or tetrazole-5-yl; and     n is 0, 1, or 2; provided that when Y is NR<4>, O, S, SO, or SO2, W is (CH2)n and Z is CHR<7> or CH; further provided that when W is S, SO, or SO2, Y is CHR<7>, Z is CHR<7> or CH, or Y and Z together are HC=CH or C IDENTICAL C;     further provided that when W and Z are CH2, Y is not S; further provided that when W and Y together are HC=CH or C IDENTICAL C, Z is CHR<7>; or a pharmaceutically acceptable salt thereof. 1,
Patent AU-4641293-A (AU)
Title: Glycine receptor antagonists and the use thereof
Inventor: WEBER ECKARD
IPC: C07D241/44
Filed: 1993-06-17
Abstract: Methods of treating or preventing neuronal loss associated with stroke, ischemia, CNS trauma, hypoglycemia and surgery, as well as treating neurodegenerative diseases including Alzheimer's disease, amyotrophic lateral sclerosis, Huntington's disease and Down's syndrome, treating or preventing the adverse consequences of the hyperactivity of the excitatory amino acids, as well as treating anxiety, chronic pain, convulsions, inducing anesthesia and treating psychosis are disclosed by administering to an animal in need of such treatment a compound having high affinity for the glycine binding site, lacking PCP side effects and which crosses the blood brain barrier of the animal. Also disclosed are novel 1,4-dihydroquinoxaline-2,3-diones, and pharmaceutical compositions thereof. Also disclosed are highly soluble ammonium salts of 1,4-dihydroquinoxaline-2,3-diones.
Patent AU-4769101-A (AU)
Title: Improved easy-open end and method of making
Inventor: ZYSSET EDGAR
IPC: B21D51/38
Filed: 2001-03-23
Abstract: A method of making an easy-open end for a container includes steps of forming first and second grooves in a panel of a can end blank, the grooves extending below the level of the panel to form inner and outer beads and forming a central bead in the panel between the first and second grooves so that the central bead extends above the panel. A score is then formed along the central bead by simultaneously forming the score and compressing the central bead, so that the depth of the score and the thickness of the central bead are both positively controlled. The inner and outer beads are then forced toward each other and then toward the panel, and the central bead is forced toward the panel. A pull-tab is then fixed to the end. This process permits the score residual to be controlled to a greater tolerance than the conventional processes, and is also more material efficient.
Patent AU-4969100-A (AU)
Title: New composition
Inventor: BERGGREN ANNA
IPC: A23L33/00
Filed: 2000-05-22
Abstract: The invention describes a sports drink, which in addition to conventional additives contains viable lactobacilli having a positive effect on human intestinal mucosa. The sports drink preferably also contains micronutrients and proteins. The invention also refers to a tablet for the preparation of such a sports drink, containing viable freeze-dried lactobacilli in combination with micronutrients. In addition to providing liquid and nutrients replacement, the sports drink also relieves the stress symptoms, which are associated with long physical exercise.
Patent AU-5057599-A (AU)
Title: Disc brake system
Inventor: BUNKER KENNETH JAMES
IPC: F16D65/12
Filed: 1999-07-26
Abstract: A disc brake comprises discs 12, 14, a hub 16, and a plurality of rollers 34 by which the discs are mounted on the hub for rotation therewith and for axial sliding movement thereon. Each roller is received in a recess in the hub and in recesses 24,26 in the discs so that the rollers transmit rotational drive between the hub and the discs and also provide bearing surfaces for said sliding movement. Disc 12 projects into a groove 36 provided in each roller so that the roller slides with that disc on the hub and that disc acts to retain each roller in its pocket. Disc 14 slides on the rollers, and leaf springs 40 are provided between each circumferentially adjacent pair of rollers.
Patent AU-5119485-A (AU)
Title: Process for the manufacture of aminothiazole acetic acid derivatives
Inventor: HEBEISEN PAUL
IPC: C07D277/20
Filed: 1985-12-13
Abstract: There is described a process for the manufacture of a compound of the formula    <IMAGE>  IV  wherein R1 is lower alkyl, lower alkanoyl, lower alkenyl or the group -CH2COOR2 or -C(CH3)2COOR2 and R2 is a readily cleavable group, by reacting a compound of the formula <IMAGE> II  wherein R is lower alkyl, with an alkali metal allylate and reacting the resulting compound of the formula    <IMAGE> I wherein M is an alkali metal atom, with a compound of the formula R1-X, wherein X is a leaving group. This process can be used to manufacture antimicrobially active mono- beta -lactam, cephalosporin and penicillin derivatives.
Patent AU-5129690-A (AU)
Title: Anti-human sperm antibody, and its production
Inventor: OKABE MASARU
IPC: C07K16/18
Filed: 1990-03-15
Abstract: A monoclonal or polyclonal antibody having a specific binding property to an antigenic site on the human sperm acrosome is disclosed, which is produced by a hybridoma obtained by fusing a mammalian cell producing an antibody to the antigenic site on the human sperm acrosome with a cell having permanent proliferation potency. Furthermore, methods and kits for the evaluation of the fertilizability of human sperms are disclosed.
Patent AU-5148785-A (AU)
Title: New imidazo ``1,2-a``-pyrimidines and salts thereof, processes for their preparation and uses thereof
Inventor: GILLESPIE ROGER JOHN
IPC: C07D487/04
Filed: 1985-12-19
Abstract: Novel compounds selected from the group consisting of the formula <IMAGE>  I  wherein R1 is selected from the group consisting of 1,2,4-oxadiazol-5-yl and 1,3,4-thiadiazol-2-yl, both optionally substituted with alkyl of 1 to 3 carbon atoms or alkenyl of 2 to 5 carbon atoms and 1,2,4-oxadiazol-3-yl and 1,3,4-oxadiazol-2-yl, both optionally substituted with alkenyl of 2 to 5 carbon atoms, alkyl of 1 to 3 carbon atoms or alkyl of 1 to 3 carbon atoms substituted with at least one fluorine, R2 and R3 are individually selected from the group consisting of hydrogen, alkyl of 1 to 3 carbon atoms and alkenyl of 2 to 5 carbon atoms or together form alkylene of 3 to 5 carbon atoms, X is selected from the group consisting of -O- and -S-, R4 is alkyl of 1 to 3 carbon atoms and their non-toxic, pharmaceutically acceptable acid addition salts having anxiolytic sedative and hypnotic activity and a novel process and novel intermediates therefor.
Patent AU-5157190-A (AU)
Title: Etoposide analogues
Inventor: LEE KUO-HSIUNG
IPC: C07D493/04
Filed: 1990-02-23
Abstract: Compounds that are analogs of etoposide and exhibit antitumor activity are disclosed. The compounds of the present invention have formula (I), where R1 is  beta -OCH2CH2NH2,  beta -NHCH(CH3)CH2OH, beta -NHCH2CH(CH3)OH,  beta -Cl,  beta -Br,  beta -OH,  alpha -OH, beta -NH2,  alpha -NH2,  beta -NHCH2CH2OH,  alpha -NHCH2CH2OH,  beta -NHCH2CH2CH3,  beta -NHCH2CH2OCH3,  beta -NHCH2CH=CH2,  beta -NHCH2CH(OH)CH3,  beta -NHCH2CH2CH2OH,  beta -OCH2CH2OH, (a), (b), (c), (d), (e), (f), (g), (h), (i), (j), (k), (l), (m), (n), (o), (p), (q), (r), (s), (t), (u), (v) or (w). R2 is H, or Br; R3 is H, or Br; R4 is H, or Br; R5 is H, or Br; and R6 is H, or -CH3.
Patent AU-5164996-A (AU)
Title: Support leg
Inventor: NILSSON HANS
IPC: B60S9/12
Filed: 1996-02-15
Abstract: A support leg (1) comprises a pivotable upper part (2) and a lower part (3) that is protrudable relative to the former, said lower part having a support foot (4). On the upper leg part (2) is arranged a rod (14) being displaceable movable which at one end is connected with a flexible tractive means (11), e.g. a chain, and at the opposite end is actuatable by the support foot (4). The tractive means (11) is laid over a pulley means (20) that separates inner and outer parts (11', 11'') of the tractive means. When pushing in the lower leg part (3), the rod is carried with the same, while lengthening the inner chain part (11') at the same time as the outer part (11'') is shortened, as the support leg pivots in the direction of a raised position. When pushing out the lower leg part, the rod (14) is allowed to move in the opposite direction, while shortening the inner chain part (11') and simultaneously lengthening the outer part (11''). In this way, a pivoting of the support leg in the direction of a lowered position is made possible.
Patent AU-5193693-A (AU)
Title: Process for recharging a part by means of a plasma transferred arc
Inventor: PRONER ALAIN
IPC: B23K9/04
Filed: 1993-11-26
Abstract: The invention relates to a method for the build-up of a workpiece by means of a transferred-arc plasma device. According to this method, there is deposited onto the workpiece (1) to be built up at least one weld bead (7a, 7b, 7c) of the said material solely by means of the transferred-arc plasma device (5), by moving the plasma device with respect to the workpiece at a speed of 1.5 to 50 m/min and by using a power of the plasma device such that the surface of the workpiece is melted to a depth at least equal to 0.5 mm and such that the coarsening of the grains in the molten zone does not exceed 10 %, without cooling the workpiece during the build-up. <IMAGE>
Patent AU-5205996-A (AU)
Title: Means of handling multiple sensors in a glucose monitoring instrument system
Inventor: BONNER LYDIA M
IPC: B01L99/00
Filed: 1996-05-03
Abstract: Fluid sensor dispenser comprises a magazine (26) with slots holding sensors (38) and located in a housing (22) opening, and an actuator (58) to advance through a slot to place the sensor in position of use. After use the actuator can be moved further to eject the used sensor and in returning to standby position activates an indexing drive (56) to turn the magazine and place the next sensor in ready position. The magazine is pref. a right cylinder with detent along its outer periphery each corresponding to one slot and with detents and slots equally spaced. The magazine pref. also has cavities holding desiccant and each communicating with one slot.
Patent AU-5255696-A (AU)
Title: Method and apparatus for frequency agility in a communication system
Inventor: BALACHANDRAN KUMAR
IPC: H04W48/08
Filed: 1996-03-18
Abstract: A method and apparatus used in the context of a first and a second communications network, wherein the second communications network is overlaid upon the first communications network. The invention generates and utilizes a number of flags and indicators to determine which channel, from among a plurality of shared channels assignable to a first communications network (e.g., an AMPS network) and a second communications network (e.g., a CDPD network), will be used next for communicating information by the second network (e.g., a CDPD information). The invention provides a means for generating an ordered Idle-Channel list. The Idle-Channel list includes each assignable channel that is not currently used by the first or second communications network. In one embodiment of the present invention, the order of the channels in the Idle-Channel list at any given time determines the order of the channels to be selected for transmission of a signal by the second communications network. In alternative embodiments of the present invention, the idle channels are ordered based upon the likelihood that they will be assigned for use by the first communications network when an additional channel is required by the first communications network.
Patent AU-5325998-A (AU)
Title: Method for simultaneously controlling and programming a plurality of transponders and device for implementing this method
Inventor: PAGNOL FREDERIC
IPC: G06K7/00
Filed: 1997-12-04
Abstract: The method involves using an external transmitter to transmit energy (1) to a group of read and write transponders. After a time delay (TRR) the transponders emit identification signals (2-3,4-5) through allocated time windows. An external receiver receives the signals during the first window and determines if there is dispersion. If there is dispersion the supply of transmitted energy is interrupted quickly enough to deactivate all the transponders. Energy transmission is resumed and if no transponder signal dispersion is now detected, a window of reception is used to send groups of data to the transponders which are simultaneously programmed into their memories.
Patent AU-5328100-A (AU)
Title: Urea substituted imidazoquinolines
Inventor: CROOKS STEPHEN L
IPC: A61P1/02
Filed: 2000-06-08
Abstract: Imidazoquinoline and tetrahydroimidazoquinoline compounds that contain urea, thiourea, acylurea, or sulfonylurea functionality at the 1-position are useful as immune response modifiers. The compounds and compositions of the invention can induce the biosynthesis of various cytokines and are useful in the treatment of a variety of conditions including viral diseases and neoplastic diseases.
Patent AU-5478096-A (AU)
Title: Improved barb and expandable transluminal graft prosthesis for repair of an aneurysm
Inventor: CHUTER TIMOTHY A
IPC: A61B17/115
Filed: 1996-06-06
Abstract: An improved prosthesis assembly (422) for placement at an aneurysm in the bifurcated lumen of the aorta and the common iliac arteries extending therefrom. The prosthesis assembly includes a single lumen graft (1) or a bifurcated lumen graft having a main body and ipsilateral and contralateral limbs extending therefrom. The main body and ipsilateral and contralateral limbs each have a spring assembly (12,31) about their orifices for conforming that portion of the graft to the wall of the vessel lumen. The main body spring assembly has an improved barb (10) with first (401) and second (414) attachment arms for securely anchoring the spring assembly to the vessel wall. The improved barb includes two forms of mechanical attachment such as, for example, a helical coil body (405) positioned around a spring assembly arm (15) and, secondly, a bonding material such as, for example, solder for fixedly attaching the coil and spring assembly arm. The attachment arms of the barb are positioned longitudinally along the spring assembly arm for engagement with the vessel wall without engaging each other when the spring assembly is in a collapsed condition. The ipsilateral and contralateral spring assemblies (31) also include the improved barb with only a single attachment arm for anchoring the spring assembly to the vessel wall. <IMAGE>
Patent AU-5571496-A (AU)
Title: Air bed with fluidized bead surface and related methods
Inventor: VRZALIK JOHN H
IPC: A47C27/10
Filed: 1996-04-24
Abstract: A therapeutic patient treatment bed (20) with features to enhance the care and comfort of burn patients and others subject to extensive recuperative periods. Among the features are patient engaging fluidized bead surfaces (22) integral with the upper surfaces (27) of air cushions (21) provided by an air bed (20). Detachable conformation of the fluidized bead surfaces (22) is also provided.
Patent AU-5603190-A (AU)
Title: Hiv p24 quantitation panel
IPC: C07K14/16
Filed: 1990-05-28
Abstract: The present invention is directed to improved immunoassay methods, and compositions and kits for carrying out the methods, for quantitating HIV p24 antigen in a biological sample. The method involves contacting a sample with an antibody specific for HIV p24 antigen, whereby a detectable antigen-antibody complex is formed, and quantitating the amount of the complex formed by employing a quantitation panel as a standard with which the amount of the complex formed can be compared. The method involves utilizing purified HIV p24 antigen in the quantitation panel. Preferably, the quantitation panel comprises lyophilized standards containing immunoaffinity-purified viral p24 antigen. The composition includes purified viral HIV p24 and a buffer. The kit includes a panel of purified viral HIV p24 compositions.
Patent AU-5662800-A (AU)
Title: Method and system for user registration on terminal
Inventor: LAPSTUN PAUL
IPC: H04L12/16
Filed: 2000-06-30
Abstract: A binding printer is provided which has a media transport assembly configured to transport individual sheets of media along a media path, a printhead assembly configured to print on the sheets transported along the media path, and a binding assembly configured to bind together the printed sheets transported along the media path. The binding assembly has a binding platen configured to press each printed sheet transported onto a support platen to preceding sheets supported on the support platen to bind the printed sheets together, and a chassis defining an inlet for receiving the transported printed sheets and an exit hatch from which the bound printed sheets are removable.
Patent AU-5745196-A (AU)
Title: Catalyzed packing material for regenerative catalytic oxidation
Inventor: NGUYEN PASCALINE H
IPC: B01J23/42
Filed: 1996-05-13
Abstract: Homogeneous catalytic regenerative heat transfer packing material is made by impregnating ceramic packing material with a solution of a catalyst precursor and then fixing the precursor into catalyst form. The catalyzed packing material is suitable for use in a process for the regenerative catalytic oxidation of waste gases, in particular, gases that include volatile organic compounds, carbon monoxide or combinations thereof.
Patent AU-5911490-A (AU)
Title: Catalyst for the selective oxidation of sulphur compounds
Inventor: BRINK PETER JOHN VAN DEN
IPC: B01J35/10
Filed: 1990-07-19
Abstract: Catalyst (I) has a specific surface area above 20 sq.m/g, average pore radius of 25 Angstroms at least with no activity w.r.t. the Claus reaction. (I) may be supported e.g. on SiO2. Active component in (I) is pref. an iron and/or chromium cpd. plus a phosphorus cpd. promotor. H2S contg. gas and O2 contg. gas are passed over (I) in a fixed or fluid bed at below 300 deg.C to obtain elemental sulphur.
Patent AU-6091180-A (AU)
Title: Series switch-mode converter
Inventor: BRAKUS B
IPC: H02M3/335
Filed: 1980-07-30
Abstract: 1. A single-ended forward converter with a pulse-width controlled semiconductor switch (41) in the converter main circuit, and with a power transformer (31) having a plurality of secondary windings (311, 312) for the generation of electrically isolated d.c. output voltages, where at least one output circuit of the single-ended forward converter contains a transistor switch (42) which is pulse-width controlled in dependence upon the output voltage (U22) of this output circuit and which possesses its own auxiliary control circuit whose output pulses occur within the output pulses of the semiconductor switch (41) in the main circuit and which is rendered conductive at the same time as the control transistor located in the converter main circuit, the transistor (42) being arranged in an output circuit that is rendered inoperative by short-circuiting a winding (71) of a pulse-control transformer (7) in dependence upon the output voltage (U22) of the corresponding output circuit, the pulse transformer (7) being preceded by a switch-on device and a switch-off device and the emitter-collector path of a transistor (43) of the switch-off device arranged parallel to a winding (71) of the pulse transformer (7), characterised in that the switch-on device is formed by a series arrangement of a resistor (12) and a diode (57), and that a winding (74) of the pulse transformer is connected via the series arrangement (12, 57) to a separate switch-on winding (311) of the power transformer (31), and that the switch-off device contains a threshold-value switch (81) having an open collector output, whose first input (+) is supplied with a control value which is dependent upon the output voltage and whose other input (-) is supplied with a comparison value (URef ) and which has its output connected via a timer circuit in the form of a mono-stable flip-flop stage which contains a capacitor (21) and a charge resistor (13 ... 15), to that transistor (43) of the switch-off device whose emitter-collector path is arranged parallel to a separate switch-off winding (71) of the pulse transformer (7).
Patent AU-6224090-A (AU)
Title: Nonwoven fabric laminates
IPC: B32B5/26
Filed: 1990-09-06
Abstract: There is disclosed a nonwoven fabric laminate formed from an olefin copolymer, olefin terpolymer, or a blend of olefin polymers. Particularly, the improved fabric laminate is formed from a polymer having a crystallinity of less than 45% and preferably between 31-35% and most preferably about 32%. The fabric laminates formed from layers that are spun-bonded (28,36) or melt-blown (32) have improved characteristics including higher tear strength, greater tensile energy, greater abrasion resistance, better fabric drape and softness, and less particulate emission. There is also disclosed a low particle emission, sterilizable garment for use in clean rooms, paint rooms, and operating rooms.
Patent AU-6323496-A (AU)
Title: Distributor comprised by a one-pipe-system for a heating or cooling apparatus
Inventor: ENGELBREKTSSON ANDERS
IPC: F24H9/12
Filed: 1996-06-25
Abstract: A distributor (7) in a single-pipe system (1, 2) in a heating or cooling apparatus has a feed pipe (3), a return and bypass pipe (4), radiators or cooling elements (5), valves (6) for the latter, and a housing (8) with an axially through-going conduit (9), one end of which forms a return inlet (10), and to which are laterally connected a return outlet (11), a feed inlet (12) and a feed outlet (13). Through the other end of said conduit (9) is inserted a control spindle (17, 21) having a cone (18) for throttling or shutting off said return inlet (10) against a seat (19) in said housing (8). According to the invention, said spindle (17, 21) is provided with a throttling cone (22) acting on a surrounding seat (23) being a circular-cylindrical restriction of said housing (8), which restriction constitutes a bypass of said system jointly with said feed inlet, said return outlet and portions of said conduit interconnecting same.
Patent AU-6469796-A (AU)
Title: 4,5-diaryl oxazole derivatives
Inventor: TANIGUCHI KIYOSHI
IPC: A61P1/16
Filed: 1996-07-18
Abstract: Heterocyclic compounds of the formula: <CHEM>     wherein     R<1> is carboxy or esterified carboxy,   R<2> and R<3> are phenyl or (C1-C6)alkylphenyl,   A<1> is (C1-C6)alkylene, and   n is 0 or 1, for the treatment or prevention of arterial obstruction, hepatitis, hepatic insufficiency, restenosis after percutaneous transluminal coronary angioplasty, arteriosclerosis, cerebrovascular disease or ischemic heart disease.