baber/WOPTO huggingface dataset:
Patent BR-PI1100858-B1 (BR)
Title: Transmissão manual automática
Inventor: ANDREA PALAZZETTI
IPC: F16H61/22
Filed: 2011-03-21
Abstract: transmissão manual automática equipada com dispositivo de trava de estacionamento. transmissão manual automática (1) que possui: pelo menos um eixo primário (5); pelo menos um eixo secundário (7); uma série de pares de embreagens (8, 9), cada um dos quais acopla mecanicamente o eixo primário (5) ao eixo secundário (7); uma série de sincronizadores (10), cada um dos quais montado coaxialmente a um eixo (7), é acoplada a uma engrenagem (9) de pelo menos um par de engrenagens e é adaptada para acionamento para engate da marcha (9) ao eixo (7); uma série de forquilhas (11), que acionam os sincronizadores (10) e são móveis; um dispositivo de trava de estacionamento (20) que pode ser acionado para evitar a rotação do eixo secundário (7); e um dispositivo de conexão (21), que é conectado mecanicamente sobre um lado a uma primeira forquilha (11d) e, do outro lado, ao dispositivo de trava de estacionamento (20) para transmitir o movimento da primeira forquilha (11d) ao dispositivo de trava de estacionamento (20), de forma a controlar a ativação e a desativação do próprio dispositivo de trava de estacionamento (20) por meio de exploração do movimento-da primeira forquilha (11d).
Patent EA-000846-B1 (EA)
Title: Medical powder
Inventor: NAKATSUKA KATSUTO
IPC: A61K9/50
Filed: 1997-06-06
Abstract: 1. A medical powder comprising a base particle of a ferromagnetic metal with a coating layer provided on the surface thereof, characterized in that at least the outside of the coating layer comprises a bioinactive material. 2. The medical powder according to claim 1, characterized in that the coating layer comprising the bioinactive material comprises a layer of a hydrolyzate of an alkoxide compound.
Patent EA-005749-B1 (EA)
Title: Coke drum discharge system
Inventor: MALSBURY ALLEN S
IPC: C10B57/04
Filed: 2002-11-06
Abstract: An apparatus including a coke drum for coking hydrocarbon substances, a valve disposed near the bottom of the coke drum, and a discharge conduit for removing coke from the coke drum, wherein the discharge conduit is connected to the valve such that when the valve is open, the coke may be removed via the discharge conduit.
Patent EA-006835-B1 (EA)
Title: A process for the production of hydrocarbon fluids
Inventor: GUYOMAR PIERRE-YVES
IPC: C09K3/00
Filed: 2003-02-28
Abstract: Hydrocarbon fluids are produced by hydrocracking a vacuum gas oil stream, fractionating and/or hydrogenating the hydrocracked vacuum gas oil. The fluids typically have ASTM D86 boiling point ranges within the range 100°C-400°C the range being no more than 75°C, they also have a naphthenic content greater than 60%, the naphthenics containing polycyclic materials, an aromatic content below 2% and an aniline point below 100°C. The fluids are particularly useful as solvents, for printing inks, drilling fluids, metal working fluids and as silicone extenders.
Patent EA-007289-B1 (EA)
Title: Phosphonates and derivatives thereof as enhancers of the activity of insecticides
Inventor: STOCK DAVID
IPC: A01N43/40
Filed: 2003-05-22
Abstract: An insecticidal composition having as an adjuvant a phosphonate or an alkoxylated derivative or dimer thereof. Preferred phosphonates are bis-(2-ethylhexyl)-2ethylhexylphosphonate, bis-(2-ethylhexyl)-octylphosphonate and bis-(butyl)butylphosphonate.
Patent EA-008968-B1 (EA)
Title: Selective hydrogenation process and catalyst therefor
Inventor: BAILEY STEPHEN
IPC: B01J23/63
Filed: 2004-05-26
Abstract: A catalyst suitable for use in hydrogenation, especially the selective hydrogenation of acetylenic compounds to olefinic compounds, which comprises palladium supported upon an alumina support material characterised in that said catalyst further comprises a compound of a lanthanide, wherein the atomic ratio of Pd to lanthanide metal is in the range 1: 0.5-1 : 3.5.
Patent EA-010719-B1 (EA)
Title: Process for forming light olefins integrated with air separation unit
Inventor: VAN EGMOND COR F
IPC: B01J38/12
Filed: 2005-03-25
Abstract: A process for regenerating catalyst in a reaction system, integrated with a system for air separation from oxygenates, and optionally from natural gas. The integrated system includes an air separation unit, which separates air components into an oxygen stream and a nitrogen stream, and which also forms a compressed air stream. The oxygen stream, the nitrogen stream and/or the compressed air stream from the air separation unit may serve as a reactant in syngas generation, as a regeneration medium in the methanol-to-olefins reaction system, as a fluidizing stream, as a blanketing medium, as a stripping medium, as instrument air, and/or as a reactant in a sulfur removal unit. In particular, according to the present invention the process comprises the steps of: (a) separating air components in an air separation unit to form an oxygen stream and a nitrogen stream, wherein the air separation unit also forms a compressed air stream; b) separating from the natural gas-containing stream and HS a majority of the HS to form a separated HS-containing stream; c) contacting the separated HS-containing stream with a portion of the oxygen stream and/or with a portion of the compressed air stream under conditions effective to convert a portion of the HS in the separated HS-containing stream to SO; d) contacting the SOwith residual SOin the presence of a catalyst composition under conditions effective to form elemental sulfur and water; e) contacting the natural gas separated from sulfur compounds in the natural gas-containing stream with at least o portion of the oxygen stream in a syngas generator under conditions effective to convert the natural gas to syngas; g) contacting the syngas with a catalyst composition in a methanol synthesis unit under conditions effective to convert at least a portion of the syngas to methanol; h) contacting the methanol with a molecular sieve catalyst composition in a reactor under conditions effective to convert the methanol to light olefins; and j) regeneration, at least partially coked molecular sieve catalyst composition at step h) using oxygen-containing regeneration medium formed in the air separation unit.
Patent EA-018014-B1 (EA)
Title: Kinesin inhibitors as cancer therapeutics
Inventor: ABRAMS TINYA
IPC: A61K31/4164
Filed: 2008-12-12
Abstract: The invention provides novel imidazole compounds of the formulathat inhibit the activity of kinesin spindle protein (KSP, also called Eg5). Inhibitors of KSP can reduce undesired cellular proliferation and provide other therapeutic effects. The invention also provides pharmaceutical compositions containing these novel compounds, and methods of using the novel KSP inhibitors and their pharmaceutical compositions to treat various types of cancers. The compounds, compositions and methods of the invention are especially useful for treating certain classes of cancers that are resistant to conventional drug treatments, because such cancers are shown to remain sensitive to the compounds of the invention.
Patent EA-019206-B1 (EA)
Title: Pyrazine compounds as phosphodiesterase 10 inhibitors
Inventor: ALLEN JENNIFER R
IPC: A61K31/497
Filed: 2009-11-16
Abstract: Pyrazine compounds of formula Iare provided, and compositions containing them, and a process for preparing such compounds. Provided herein also are methods of treating disorders or diseases treatable by inhibition of PDE10, such as obesity, non-insulin dependent diabetes, schizophrenia, bipolar disorder, obsessive-compulsive disorder, and the like.
Patent EA-021708-B1 (EA)
Title: Hydroconversion multi-metallic catalyst and method for making same
Inventor: KUPERMAN ALEXANDER E
IPC: C07F19/00
Filed: 2010-04-08
Abstract: A catalyst with low volumetric shrinkage and a process for making the stable catalyst with low volumetric shrinkage is disclosed. The catalyst is made by sulfiding a catalyst precursor containing at least a Group VIB metal compound; at least a promoter metal compound selected from Group VIII, Group IIB, Group IIA, Group IVA and combinations thereof, having an oxidation state of either +2 or +4; optionally at least a ligating agent; optionally at least a diluent. In one embodiment, the catalyst precursor is first shaped then heat treated at a temperature of 50 to 200°C for 15 minutes to 12 hours, wherein the catalyst precursor has a low (less than 12%) volumetric shrinkage after exposure to at least 100°C for at least 30 minutes, e.g., in sulfidation or in a hydrotreating reactor. In one embodiment, the catalyst precursor has an essentially monomodal pore volume distribution with at least 90% of the pores being macropores, and a total pore volume of at least 0.08 g/cm. In another embodiment, the catalyst is suitable for hydrotreating heavy oil feeds having a boiling point in the range of 343 to 454°C, an average molecular weight Mn ranging from 300 to 400, and an average molecular diameter ranging from 0.9 to 1.7 nm.
Patent EA-022218-B1 (EA)
Title: Composite reinforcement
Inventor: ZUBKOV VJACHESLAV DMITRIEVICH
IPC: E04C5/07
Filed: 2012-12-29
Abstract: The invention relates to reinforcements, particularly, to alternate-profile reinforcements for production of articles from concrete and aerated concrete by hot moulding at simultaneous effects of aggressive media. A composite reinforcement comprises bar with winding composed by fibrous filler impregnated with epoxy resin-based polymer binder and hardener. The reinforcement contains 60-80% of fibrous hardener and 20-40% of binder comprising, wt.%: epoxy-novolak resin - 50-60, amine hardener - 40-50. Said resin comprises the following components, wt.%: diane epoxy resin - 47-80, modifier based on polyesters including glycidyl groups - 10-25, component produced by epoxidation of hydroxyphenylene oligomer from alkyl resorcinol - 10-28. The effect is higher resistance of the reinforcement to continuous exposure to high temperatures, high strength and elasticity rates, resistance against aggressive media and high binder hardening rate.
Patent EA-024241-B1 (EA)
Title: Optically active dibenzylamine derivative, and method for preparing the same
Inventor: OHGIYA TADAAKI
IPC: C07D239/47
Filed: 2011-06-03
Abstract: The present invention relates to a substantially optically pure (S)-trans-{4-[({2-[({1-[3,5-bis(trifluoromethyl)phenyl]ethyl}{5-[2-(methylsulfonyl)ethoxy]pyrimidine-2-yl}amino)methyl]-4-(trifluoromethyl)phenyl}(ethyl)amino)methyl]cyclohexyl}aceitic acid or a pharmaceutically acceptable salt thereof, having the effect of reducing the amount of PCSK9 proteins and increasing the amount of LDL receptors. Disclosed is a medicament for prophylactic and/or treatment of a disease selected from hyper-LDL cholesterolemia, dyslipidemia, arteriosclerosis, atherosclerosis, peripheral vascular diseases, hypercholesterolemia, familial hypercholesterolemia, cardiovascular functional disorders, angina pectoris, ischemia, cardiac ischemia, thrombosis, myocardial infarction, reperfusion disorders, angioplasty restenosis, and hypertension, comprising the above-stated compound or a pharmaceutically acceptable salt thereof as an active ingredient. The invention also relates to a method for preparing (S)-trans-{4-[({2-[({1-[3,5-bis(trifluoromethyl)phenyl]ethyl}{5-[2-(methylsulfonyl)ethoxy]pyrimidine-2-yl}amino)methyl]-4-(trifluoromethyl)phenyl}(ethyl)amino)methyl]cyclohexyl}aceitic acid or a pharmaceutically acceptable salt thereof.
Patent EA-026677-B1 (EA)
Title: Method and system for thermal energy storage
Inventor: DUCHEYNE WOUTER
IPC: F28D20/00
Filed: 2012-01-24
Abstract: The present invention relates to a method of thermal energy storage in a reaction mixture by means of an endothermic condensation reaction, said reaction mixture comprising a polyphosphoric acid compound and/or its salt and water, said reaction being enabled by the heat input from a heat source distinct from said reaction mixture, the energy in the heat source being stored by means of the endothermic condensation reaction removing water from the reaction mixture and forming the polyphosphoric acid and/or salts thereof. The present invention further provides a system for storing energy to carry out said method, the system comprising at least one reaction vessel at least partially filled with a reaction mixture comprising a polyphosphoric acid compound and/or its salt and water, suitable for having an endothermic condensation reaction performed on said reaction mixture, and comprising a heating element in thermal communication with said vessel.
Patent EA-026181-B1 (EA)
Title: Device for optical identification of measurement channels of a built-in non-destructive control system based on fiber-optic bragg gratings
Inventor: KARASIK VALERIY EFIMOVICH
IPC: G02B6/34
Filed: 2012-12-21
Abstract: The invention relates to devices for registering signals from a set of fiber-optic Bragg gratings in a built-in non-destructive object control system. The device for optical identification of measurement channels in a built-in non-destructive control system comprises a source of optical radiation, a tripolar optical splitter, a reference Bragg grating having a known reflected radiation wavelength, several measurement channels with fiber Bragg gratings located on the object being tested, a system for insulating the reference Bragg grating from external disturbing effects, a photodetector device and a unit for registering and converting signals, said unit being connected to a computer. One addressable reference Bragg gratings having non-repeating reflected radiation wavelengths is built into each measurement channel. All reference gratings are placed in a body insulated for protection against external disturbing effects. A superluminescent diode (SLD) is used as a continuous broad-band source of optical radiation. The device further includes an optical insulator and an optical switch, the optical insulator being installed between the output of the source and the input pole of the tripolar optical splitter, one output pole of which is connected to the common input of the optical switch. Each connectable output of the optical switch is connected to its own measurement channel. The other output pole of the splitter is connected to an input of the photodetector device and of the signal registering and converting unit. The technical result is simultaneous significant simplification of the device circuit with warranted assurance of reliability of identification (addressing) of measurement channels connected to the computer, and an increase in dynamic range of optical signals being measured.
Patent EA-038489-B1 (EA)
Title: Anticholinergic neuroprotective composition and methods
Inventor: CLARENCE-SMITH KATHLEEN E
IPC: A61K31/00
Filed: 2013-09-05
Abstract: The invention relates to a pharmaceutical composition for inducing neuroprotection in a patient suffering from Alzheimer type dementia, the composition being in the form of immediate release preparation. The provided composition comprises from 10 to 80 mg of solifenacin succinate and from 25 to 70 mg of donepezil hydrochloride in admixture with a pharmaceutical carrier. The invention also relates to the use of a combination of an acetyl choline esterase inhibitor (AChEI) consisting of donepezil hydrochloride at a daily dose of 25 to 151 mg and a non-selective peripheral anticholinergic agent (nsPAChA) consisting of solifenacin succinate at a daily dose of 10 to 80 mg for inducing neuroprotection in a patient suffering from Alzheimer type dementia.
Patent EA-030155-B1 (EA)
Title: 1,2,4-oxadiazole derivatives as immunomodulators
Inventor: SASIKUMAR POTTAYIL GOVINDAN NAIR
IPC: C07D285/08
Filed: 2014-09-05
Abstract: The present invention relates to 1,2,4-oxadiazole compounds as therapeutic agents capable of inhibiting the programmed cell death 1 (PD1) signaling pathway. The invention also refers to derivatives of these therapeutic agents. The invention also encompasses the use of the said therapeutic agents and derivatives thereof for treatment of impairments and disorders via immunopotentiation comprising inhibition of immunosuppressive signal induced due to PD-1, PD-L1, or PD-L2 and therapies or treatment using them.
Patent EA-033452-B1 (EA)
Title: Tap-hole refurbishing
Inventor: CLESEN ROMAIN
IPC: F27D3/15
Filed: 2014-12-09
Abstract: The present invention relates to a method for refurbishing a tap-hole, comprising making a tap-hole channel trough a tap-hole block in a lower section of an arc, blast or smelter furnace; restoring the tap-hole channel; detachably connecting a sealing rod to a clay gun; inserting the sealing rod into a prefabricated, hollow, refractory tap-hole insert so that there is a space between the tap-hole insert and the sealing rod; detachably connecting to said clay gun the tap-hole insert comprising a shell and having a first end with an opening, a second blocked end, a hollow passage in axial direction, said hollow passage being accessible through the opening, and a plurality of lateral through holes aligned in a longitudinal direction with a constant interval in-between and covering between 10 and 25% of the shell of the tap-hole insert; inserting the tap-hole insert into the tap-hole channel, wherein the clay gun is fluidly coupled with the tap-hole insert and the tap-hole channel; injecting a clay material in the space between the tap-hole insert and the sealing rod; holding the sealing rod in place until the clay material has at least partially cured; injecting a grouting material from the clay gun into the tap-hole insert and into the tap-hole channel; disconnecting the sealing rod from the clay gun such that the sealing rod remains in the tap-hole; and disconnecting the tap-hole insert from the clay gun.
Patent EA-033476-B1 (EA)
Title: Synthesis of anionic surfactants and their use as collectors in froth flotation of non-sulphidic ores
Inventor: SMOLKO-SCHVARZMAYR NATALIJA
IPC: B03D1/016
Filed: 2014-07-02
Abstract: The invention relates to a compound obtainable by reacting an N-acyl neutral amino acid or a salt thereof, or an N-acyl neutral amino acid oligopeptide or a salt thereof with a monohydroxy monocarboxylic acid or a salt thereof. The compound has structural formulaThis compound is useful as a collector in a process for froth flotation of non-sulfidic ores, especially phosphate ores. The invention also relates to a method which comprises the steps of a) conditioning a pulped phoshate ore, wherein the ore comprises a calcium phosphate mineral or a mixture of such minerals, and gangue minerals, with an effective amount of a calcium phosphate mineral collector reagent, which is the above-mentioned compound, and optionally other flotation aids, and b) performing a froth flotation process to recover the calcium phosphate mineral(s).
Patent EA-035338-B1 (EA)
Title: Composition of hematopoietic stem cells with reduced inflammatory activity, production and use thereof
Inventor: De Munter Johannes Petrus Jozef Maria
IPC: C12N5/0775
Filed: 2014-10-24
Abstract: The invention relates to the field of cell therapy, more particularly to stem cell transplantation therapy. Provided are methods and compositions for improving the efficacy of stem cell transplantation therapy by reducing the inflammatory activity of a stem cell transplant. In particular, provided is a method for preparing a stem cell transplant with reduced inflammatory activity comprising a step of suspending a composition comprising stem cells in a fibrinogen depleted plasma and/or in a fibrinogen and C-reactive protein depleted plasma.
Patent EA-034662-B1 (EA)
Title: Combine header reel apparatus for sunflowers
Inventor: DIETRICH DAVE
IPC: A01D45/00
Filed: 2016-09-08
Abstract: A plant pushing apparatus for mounting on a reel of a combine where the reel comprises a center shaft rotatably mounted at each end thereof to the combine header, a plurality of contact members mounted to the center shaft in a horizontal orientation radially spaced from the center shaft, and a drive operative to rotate the center shaft such that the contact members below the center shaft move in a rearward direction toward the combine header. For each contact member, a projecting shield member is adapted at an inner portion thereof for attachment to the contact member such that an outer edge of the projecting shield member is substantially horizontal and rearward of the contact member, and such that the outer edge of the projecting shield member contacts plant stalks, particularly sunflower plant stalks, and pushes the plant stalks toward the combine header ahead of the following attached contact member.
Patent EA-037498-B1 (EA)
Title: Pharmaceutical composition containing 8-[(3r)-3-amino-1-piperidinyl]-7-(2-butyn-1-yl)-3,7-dihydro-3-methyl-1-[4-methyl-2-quinazolinyl)methyl]-1h-purine-2,6-dione or a pharmaceutically acceptable salt thereof
Inventor: KREKELER ANDREAS
IPC: A61K9/20
Filed: 2016-10-07
Abstract: The invention relates to a pharmaceutical composition comprising linagliptin or a pharmaceutically acceptable salt thereof as active ingredient, wherein the pharmaceutical composition does not comprise a binder and wherein the pharmaceutical composition is obtained by direct compression.
Patent EA-038774-B1 (EA)
Title: Smoking article with liquid-filled capsule
Inventor: ONO HIROYOSHI
Filed: 2017-10-30
Abstract: A smoking article is disclosed which includes a rod element comprising smokeable material and a filter element having a first end for connection to an end of the rod element and an opposite, second end for insertion into a mouth of a user. A liquid-filled capsule is arranged between the first and second ends of the filter element and the liquid-filled capsule is configured to break upon application of an external force to release the liquid. A tipping wrapper connects the filter element and rod element. The tipping wrapper has a wet tensile strength of at least about 0.15 kN/m. The smoking article is resistant to breakage even after the liquid is released.
Patent EA-039853-B1 (EA)
Title: Tetracyclic heterocycle compounds useful as hiv integrase inhibitors
Inventor: GRAHAM THOMAS H
Filed: 2017-11-30
Abstract: The invention relates to tetracyclic heterocycle compounds of formula (I) and pharmaceutically acceptable salts or prodrug thereof, wherein A, X, R1, R2, R3 and R7 are as defined herein. The invention also relates to compositions comprising at least one tetracyclic heterocycle compound, and methods of using the tetracyclic heterocycle compounds for treating or preventing HIV infection in a subject.
Patent ES-2190703-B1 (ES)
Title: Composicion de lana mineral.
Inventor: VIGNESOULT SERGE
IPC: A01G31/00
Filed: 2000-07-28
Granted: 2004-07-01
Abstract: Composición de lana mineral. Lana mineral susceptible de disolverse en un medio fisiológico, y que comprende los componentes mostrados a continuación con los porcentajes expresados seguidamente: **FIGURA** y que representan el criterio basado en el ratio R{sub,1} de forma que R{sub,1} = (SiO{sub,2}+Al{sub,2}O{sub,3})/P{sub,2}O{sub,5} donde R{sub,1} está comprendido entre 12 y 20.
Patent ES-2169009-B1 (ES)
Title: Algoritmo auto-organizativo de datos de expresion genica
Inventor: DOPAZO BLAZQUEZ JOAQUIN
IPC: G16B40/30
Filed: 2000-12-14
Granted: 2003-11-01
Abstract: Algoritmo auto-organizativo para el análisis masivo de datos de expresión génica provenientes de experimentos de arrays de ADN, que comienza partiendo de una estructura compuesta por dos neuronas "hijas" conectadas a una neurona "madre", las cuales se componen por una lista de valores o perfil, inicialmente de datos aleatorios. El algoritmo, en una serie sucesiva de ciclos, va dividiendo el conjunto de datos en subconjuntos. Cada uno de los ciclos consta de una serie de épocas en las que se presentan los datos a las neuronas terminales y éstas se van actualizando. Cuando entre dos épocas consecutivas la actualización producida está por debajo de un cierto nivel mínimo preestablecido, se considera que la red ha convergido en ese ciclo y se decide si la red debe seguir creciendo o si ya ha acabado de crecer, en cuyo caso se da por finalizado el proceso o algoritmo.