baber/WOPTO huggingface dataset:
Patent IE-42971-L (IE)
Title: 2-arylpropionic acids and intermediates
IPC: C07C51/00
Filed: 1976-03-31
Abstract: 1514812 2-Arylpropionic acids; 2-arylacrylic acids BOOTS CO Ltd 31 March 1976 [4 April 1975] 13817/75 Heading C2C Compounds III (including novel 2-(fluorobiphenylyl)-2-hydroxypropionic acids) in which Ar is aryl and Y is OH or NR 1 R 2 , where R 1 and R 2 are alkyl, alkenyl or aryl or together with the adjacent N atom form a 5- to 7-membered ring, are prepared by reacting a compound Ar 1 MgBr, where Ar 1 is Ar or a group convertible to Ar on acidification, with a compound CH 3 CO.COZ, where Z is OM or NR 1 R 2 , M being an alkali metal, and acidifying the resulting mixture to give a compound III. Compounds III can be converted to antiinflammatory compounds Ar-CH(CH 3 )COOH by known methods, e.g. by dehydration to the corresponding acrylic acid followed by hydrogenation and when Y is NR 1 R 2 , by hydrolysis to a carboxylic acid before or after dehydration or hydrogenation.
[GB1514812A]
Patent IE-780812-L (IE)
Title: Denitrosation of organic nitrosamines.
IPC: C07B/
Filed: 1978-04-24
Abstract: The invention relates to a method for the denitrosation of organic nitrosamines with aliphatic and cycloaliphatic ketones or aliphatic aldehyes in the presence of a strong acid, and optionally an inert organic solvent.
[US4134917A]
Patent IE-820862-L (IE)
Title: Aminophosphinylalkanoyl compounds
IPC: A61K31/675
Filed: 1982-04-14
Abstract: Compounds of the formula  <IMAGE>  wherein X is an imino acid or ester and R1 is hydrogen,  <IMAGE>  are useful hypotensive agents due to their angiotensin converting enzyme inhibition activity.
Patent IE-810919-L (IE)
Title: Composition
IPC: A61K31/495
Filed: 1981-04-24
Abstract: 1. Anti-inflammatory compositions for local topical administration containing an effective amount of a compound of the general formula see diagramm : EP0039059,P10,F2 wherein X signifies a sulphur or oxygen atom, Y signifies the group -CH=, -CH2 - or -N=, R signifies lower alkyl or hydroxy-lower alkyl, R' signifies lower alkyl, halogen, cyano, lower alkylthio, carboxy or lower alkylcarboxy and Z signifies the number 0 or 1, with the proviso that R' signifies bromine and X signifies a sulphur atom when Y signifies the group -CH2 -, and X signifies an oxygen atom when Y signifies the group -N=, or a pharmaceutically acceptable salt thereof and a pharmaceutically acceptable carrier material which is designed for local topical application.
[EP0039059A2]
Patent IE-44837-L (IE)
Title: Tertiary imidazolyl alcohols
IPC: E04G21/20
Filed: 1977-05-10
Abstract: The bricklaying or plaster finishing trowel has holding handle on its upper face. The tool is designed for reliable carrying of mortar without loss of dropping from the trowel. The trowel tip end has vertically raised side walls, with sloping edges which taper downwards towards the trowel tip. The side walls can be fixed and their edges can also taper downwards towards the handle end of trowel. These side walls can be held on a carrier bracket with springs and with a hinge with pivoting axis for adjusting the position of the side walls and placing it over trowel as an attachment.
[DE2623159A1]
Patent FI-810509-L (FI)
Inventor: BECK GERHARD
IPC: C07D209/52
Filed: 1981-02-19
Abstract: What are disclosed are prostacylin PGI2 analogs of the formula <IMAGE>   having a more specific or longer lasting pharmacological action than PGI2, methods of making these analogs; and methods and pharmaceutical preparations for inhibiting blood platelet aggregation, for treating hypertension, for the treatment or prophylaxis of gastrointestinal ulcers, and for the treatment of asthma.
Patent FI-812194-L (FI)
Inventor: LANGE WOLFGANG
IPC: B01J20/26
Filed: 1981-07-10
Abstract: The invention relates to a process producing porous powdery polymer particles. A homogeneous mixture having two components minimum, one a meltable polymer, the other fluid inert to the polymer, both forming a system having a range of complete miscibility and a miscibility gap are introduced to a bed of solid-substance particles, then cooling the mixture to below solidification of the polymer and comminuting the obtained cake-like mass. The polymer is separated then from the inert fluid and solid-like substance particles.
Patent FI-812309-L (FI)
Inventor: FISCHER KARL
IPC: H01H37/34
Filed: 1981-07-22
Abstract: An electric hot plate has an overheating safety switch having a steatite housing which is inserted into the lower sheet cover plate of the hot plate and is supported with two feet on the lower side of the heating elements of the hot plate. A bimetallic member is positioned parallel between these feet which acts on a snap switch positioned in the steatite housing via a transmission rod. The transmission rod is continuously pressed against the snap switch by a plate spring and a guide on the snap switch. As a result of this, it is fixed precisely in its position. The overheating safety switch simultaneously forms the lead-through passages for the electric hot plate connections.
Patent IE-33927-L (IE)
Title: Separating carboxylic acids from solvent extracts of¹micro-organisms grown on hydrocarbons
IPC: C07C51/48
Filed: 1969-08-01
Abstract: 1,271,516. Separation of carboxylic acid-esters from growth media. BRITISH PETROLEUM CO. Ltd. 30 July, 1969 [30 Aug., 1968], No. 41539/68. Heading C2C. Carboxylic acids and esters obtained by microbiological treatment of hydrocarbons are separated from a lipid extract (defined as meaning that portion of a micro-organism culture grown on a hydrocarbon substrate separated from the micro-organisms by solvent extraction) by converting the acids and esters into alkali metal salts by saponification, extracting the hydrocarbons in a solvent in which the alkali metal salts are insoluble, and then converting the salts back into acids or esters.
[GB1271516A]
Patent IE-37198-L (IE)
Title: Making containers
IPC: B31B50/44
Filed: 1972-12-01
Abstract: 1376454 Making boxes AIRFIX INDUSTRIES Ltd 11 Dec 1972 [14 Dec 1971] 58080/71 Heading B5D To enable blanks used to form boxes to be positioned close together on the blank stackwhich may be flexible board, paper, plastics or metal foil-without wastage each box is formed of two or more blanks the abutting edges of which are connected, preferably by injection moulding. The blanks may be frusto-conical as shown in Fig. 2 or rectangular if the box is to be rectangular. A base may be formed of overlapping flaps secured together by injection moulding or the base may be formed by injection moulding. Apparatus for assembling the blanks comprises stacks of blanks 14, 15, and arms 22, 23 having suction pads 24 and swingable by the action of a jack 27 to remove blanks from the stacks and present them to the cavity of a tool 21. Actuation of a further jack 20 moves the blanks and arms 22, 23 into the cavity with the blank edges abutting. Vacuum ports may be provided in the walls of the cavity. The cavity tool is then closed by a core tool that injects material to form the seams, and if required the base. There may be two cavity tools mounted on rails so that they can be moved into and out of the moulding machine, one tool being loaded with blanks whilst the seams are being moulded in the other tool. When the blanks include base forming flaps an additional member (30, Fig. 7) having a suction cap is provided on the arms 22, 23.
[GB1376454A]
Patent IE-33999-L (IE)
Title: (3-benzoylphenyl) alkanoic acids
IPC: C07C59/64
Filed: 1969-12-18
Abstract: 1,241,880. Benzoylphenylalkanoic acids. RHONE POULENC S.A. 18 Dec., 1969-[20 Dec., 1968], No. 161844/69. Heading. C2C. Novel compounds (I) in which R<SP>1</SP> is 1-4C alkyl are prepared by demethylation of compounds (II) by methods known per se Intermediates isolated are (III) 2-(3-benzoyl- 2-methoxyphenyl) propionic acid, prepared by reaction of (IV) 2-(3-benzyl-2-methoxyphenyl) propionic acid with alkaline KMnO 4 ; compound (IV), prepared by simultaneous hydrolysis and methylation of (V) 2-oxo-3-methyl-7-benzyl- 2,3-dihydro-benzofuran; compound (V), prepared by reaction of (VI) 2-ethoxycarbonylamino - 3 - methyl 7 benzyl - benzofuran with 12N HCl; compound (VI) prepared by reaction of ethanol with (VII) 2-azidocarbonyl- 3 - methyl - 7 - benzyl - benzofuran; compound (VII), prepared by reaction of sodium azide with (VIII) 2-chlorocarbonyl-3-methyl-7-benzyl-benzofuran; compound (VIII), prepared by reaction of SOCl 2 with (IX) 2-carboxy-3-methyl- 7-benzyl-benzofuran; compound (IX), prepared by hydrolysis of (X) 2-ethoxycarbonyl-3- methyl-7-benzyl-benzofuran; compound (X), prepared by cyclization of (XI) ethyl α-(2- benzylphenoxy)-acetyl-acetate; and compound (XI), prepared by reaction of 2-hydroxydiphenylmethane - with NaH and ethyl α- chloroacetylacetate. Pharmaceutical compositions comprise a compound (I) together with a suitable carrier and/or diluent, are administered orally, rectally, parenterally or topically and have anti-inflammatory activity.
[GB1241880A]
Patent IE-821689-L (IE)
Title: Bicyclic pyrimidin-5-one derivatives
IPC: A61K31/519
Filed: 1982-07-14
Abstract: Novel 5_H-thiazolo- and 5_H-1,3,4-thiadiazolo[3,2-a]pyrimidin-5-one and 3,4-dihydro-2_H,6_H-pyrimido[2,1-b] [1,3]-thiazin-6-one derivatives, which compounds are useful psychotropic agents.
[US4443451A]
Patent IE-861894-L (IE)
Title: Chemical compounds
IPC: A61P35/00
Filed: 1986-07-15
Abstract: Vitamin D analogues represented by general formula (I), in which formula X stands for hydrogen, lower alkyl, halogen or hydroxy; Y stands for hydrogen or hydroxy; R<1> and R<2>, which may be the same or different, stand for lower alkyl, optionally substitutedwith halogen or hydroxy with the proviso that R<1> and R<2> cannot both be methyl when X is other than lower alkyl, or, taken together with the carbon atom numbered 25, R<1> and R<2> can form a saturated or unsaturated C3-C9 carbocyclic ring which may optionally be substituted at any possible position(s) with lower alkyl, halogen or hydroxy; R<3> stands for hydrogen or lower alkyl; R<4> and R<5> represent either each hydrogen, or when taken together constitute a bond, with the result that a double bond connects carbon atoms numbered 22 and 23; and bioreversible derivatives thereof. The compounds of the invention have a favourable therapeutic index and are particularly useful in the treatment of human and veterinary disorders which are characterized by abnormal cell proliferation and/or cell differentiation.
[WO8700834A1]
Patent IE-902362-L (IE)
Title: Packing pressure sensitive adhesive substrate sections
IPC: B05D5/10
Filed: 1990-06-29
Abstract: The device for increasing the storage stability of flat substrate portions which are packaged in bags, are equipped to be self-adhesive, whose self-adhesive surface is protected by a carrier layer which projects at least partially over said self-adhesive layer, and in which bonding of the carrier layer to the packaging occurs due to migration of the adhesive as a result of cold flow, is characterised in that elevations, which are fixed on the carrier layer in the part of the carrier layer projecting over the self-adhesive surface or are shaped from the carrier layer itself, are mounted as spacers between the carrier layer and the packaging. 
<IMAGE>
Patent IE-822801-L (IE)
Title: Compositions for topical application
IPC: A01N25/02
Filed: 1982-11-24
Abstract: A composition for topical application to animals to control ectoparasites comprising a mixture of a synthetic pyrethroid in a carrier comprising particular combinations of an alcohol solvent with an ester co-solvent.
[GB2110092A]
Patent IE-823087-L (IE)
Title: Azetidinones.
IPC: C07D205/08
Filed: 1982-12-23
Abstract: Antibacterial activity is exhibited by compounds having the formula <CHEM> and salts thereof, wherein R1, R2, R3, R4, R5 and R6 represent various organic groups.
[EP0085291A1]
Patent IE-873467-L (IE)
Title: Aryloxy and arylacyloxymethyl aminomethylketones
IPC: C07C239/00
Filed: 1987-12-21
Abstract: Thiol protease inhibitors are disclosed having the formula: <CHEM> or an optical isomer thereof, or a pharmaceutically acceptable salt thereof, wherein: n is 0 or 1; m is 0, 1 or 2; X is H or an N-protecting group; each Y is independently an optionally protected alpha -amino acid residue; R is an optionally protected alpha -amino acid side chain that is H or CH3 or that is bonded to the alpha -carbon atom to which it is attached by a methylene, methine or phenyl radical; and R' is optionally substituted aryl.
[EP0272671A2]
Patent NO-781951-L (NO)
Title: Flytende plattformkonstruksjon
Inventor: EINSTABLAND TOMAS BERGE
IPC: B63B/
Filed: 1978-06-05
Abstract: Flytende plattformkonstruksjon
Patent NO-832252-L (NO)
Inventor: HAWKES GRAHAM S
IPC: B25J3/04
Filed: 1983-06-21
Abstract: A powered, electromechanical manipulator assembly is disclosed which includes an electrically powered input device (21) coupled by a hydraulic circuit (29) to a mechanical manipulator. The hydraulic circuit (29) is a fixed-volume, closed circuit in which a master piston-cylinder assembly (32) is driven by a D.C. motor (26) and a hydraulically coupled for direct and proportional displacement of a slave piston-cylinder assembly (33) to enable smooth, accurate and easily controlled displacement of a manipulator arm (61). The manipulator arm (61) is formed of a plurality of modules (62a, 62b, 62c, 62d) each having a fixed- volume, closed, hydraulic circuit (29) and a slave cylinder (33). Both the slave and master cylinders include ambient pressure surfaces (53,54) which are exposed to the water pressure at the operating depth of the assembly so that variation in depth does not materially affect the response or dexterity of the remote manipulator apparatus. An improved terminal module or jaw assembly (68) is also disclosed.
Patent NO-862532-L (NO)
Inventor: GRELL WOLFGANG
IPC: A61K31/395
Filed: 1986-06-24
Abstract: 1. Two new solid forms of 2-ethoxy-4-[N-(1-(2-piperidino- phenyl)-3-methyl-1-butyl)-aminocarbonylmethyl]-benzoic acid, the form designated (B) being characterised by the melting point of 140-142 degrees C and by the IR(KBr) spectrum according to Figure B' and the form designated (C) being characterised by a melting point of 75-85 degrees C and by the IR(KBr) spectrum according to Figure C'.
Patent NO-864561-L (NO)
Inventor: MOHN FRANK
IPC: F04D17/02
Filed: 1986-11-17
Abstract: PCT No. PCT/GB86/00156 Sec. 371 Date Jan. 20, 1987 Sec. 102(e) Date Jan. 20, 1987 PCT Filed Mar. 18, 1986 PCT Pub. No. WO86/05557 PCT Pub. Date Sep. 25, 1986.A pump or compressor unit (1) suited particularly for mixed phase fluids, e.g. mixed gas and oil, has a multistage axial flow compressor device with contra-rotating vanes. An upstream mixer device (10) and a downstream centrifugal impeller device (32) can each be driven by the compressor device (21, 26, 27, 29), which may be shaped to provide a flow passage of decreasing cross-section in the flow direction. The compressor drives may be supplied by axially adjacent electric motors (24, 25) which may surround rotating sleeves (21) carrying the compressor vanes. A fluid can be circulated through the unit, e.g. for electrical insulation, and may be leaked into the pump fluid through seals, when it may contain a corrosion inhibiting agent. The unit may be arranged to be movable along a pipeline under fluid pressure to engage power supply contacts at a predetermined location.
Patent NO-872779-L (NO)
Inventor: FABRE JEAN-LOUIS
IPC: C07D519/00
Filed: 1987-07-02
Abstract: A compound of the general formula I;    <IMAGE>  (I)  in which R is hydrogen or a halogen or an alkyl, alkyloxy, alkylthio, trifluoromethyl, amino, alkylamino, dialkylamino, hydroxy, cyano, carboxy, alkylsulphinyl, alkylsulphonyl, sulphamido, alkylsulphamido, dialkylsulphamido, carbamoyl, alkylcarbamoyl, dialkylcarbamoyl, phenylcarbamoyl, diphenylcarbamoyl, pyridylcarbamoyl, dipyridylcarbamoyl, benzyl, alkylcarbonyl, benzoyl, alkyloxycarbonyl, phenoxycarbonyl, alkylcarbonyloxy, benzoyloxy, alkylcarbonylamino, benzamido, phenyl, phenoxy or phenylthio group, X is oxygen or sulphur or an imino, alkylimino, phenylimino, benzylimino, sulphinyl, sulphonyl, carbonyl, carbonylmethylene, methylenecarbonyl, carbonylvinylene or vinylenecarbonyl group, or X represents a valency bond or a straight-chain alkylene group containing 1 to 4 carbon atoms and Ar is a phenyl, naphthyl, pyridyl, quinolinyl, isoquinolinyl, thienyl, benzothienyl, thieno[3,2-b]thien-2-yl or thieno[2,3-b]thien-2-yl group, it being possible for the group Ar to be unsubstituted or substituted with one or more halogen or alkyl, alkyloxy, alkylthio, trifluoromethyl, amino, alkylamino, dialkylamino, hydroxy, cyano, carboxy, alkylsulphinyl, alkylsulphonyl, sulphamido, alkylsulphamido, dialkylsulphamido, carbamoyl, alkylcarbamoyl, dialkylcarbamoyl, phenylcarbamoyl, diphenylcarbamoyl, pyridylcarbamoyl, dipyridylcarbamoyl, benzyl, alkylcarbonyl, benzoyl, alkyloxycarbonyl, phenoxycarbonyl, alkylcarbonyloxy, benzoyloxy, alkylcarbonylamino or benzamido group; each alkyl moiety containing 1 to 4 straight- or branched-chain carbon atoms; the compound being in separate enantiomeric form or mixtures thereof or a pharmaceutically acceptable salt thereof is useful in the treatment of all the pathological conditions in which PAF-acether may be directly or indirectly implicated.
Patent NO-883478-L (NO)
Inventor: DREVET MICHEL
IPC: F01B3/02
Filed: 1988-08-04
Abstract: Rotating machine with pistons (7) and barrel (2) comprising a thrust plate (15) inclined in relation to its geometric axis of rotation which coincides with the geometric axis of the barrel, the central part of the inclined plate (15) comprising a spherical bearing (17) which turns freely about a fixed central trunnion (16) anchored to the central section of the barrel (2) whilst the latter is connected to a rigid peripheral housing (1), the central trunnion being firmly attached to a rigid half-shaft (33) linked to the rear section of the housing (1), characterised by at least one rod (38) rigidly connected to the trunnion (16) and to a piston (46) arranged in a bore (47) in the barrel (2) and subjected to the action of a pressurised liquid in such a way that at least some of the axial stresses applied to the trunnion (16) are transmitted to the barrel (2) without being applied to the housing (1). 
<IMAGE>
Patent NO-890285-L (NO)
Inventor: DOHRER KATHRYN K
IPC: B29D7/00
Filed: 1989-01-23
Abstract: Draw resonance problems previously encountered when extrusion casting or extrusion coating linear low density polyethylene, LLDPE, are substantially alleviated by use of a polymer designed to have an I2 melt index of from 0.1 to 25 gm/10 minutes, and an I10/I2 ratio from 4.0 to 8.3. Line speeds approaching and even surpassing those attained with LDPE are made possible. This invention can even be used in conjunction with known prior methods for alleviating draw resonance problems with LLDPE and obtain the benefits of the combination.
Patent NO-893970-L (NO)
Inventor: CLARK JOSEPH DEGANT JR
IPC: A61K31/195
Filed: 1989-10-05
Abstract: There are described compositions of 2-(2,6-dichloro-3-methylphenylamino)benzoic acid and its physiologically acceptable salts which are effective in inhibiting the conversion of gingivitis to periodontitis and thus useful in treating destructive periodontal disease. The therapeutic agent can be applied directly to the gingival tissue in a topically administerable pharmaceutical composition or can be introduced and released in the buccal cavity for contact with the gingival tissue through the fluid motion present in the mouth.
Patent NO-903367-L (NO)
Inventor: ROESSLER KARL-HEINZ
IPC: H02B11/133
Filed: 1990-07-30
Abstract: A draw (2) for an electrical cabinet has two switches (4, 5) arranged next to one another and each with a drive shaft (6, 7). A locking device ensures that only one of the switches (4, 5) can ever be actuated, and that this is possible only when the draw (2) is in a position in the electrical cabinet provided for this purpose. The locking device comprises a two-armed lever (13) having detent noses (12) and a projecting detent lever (15) with a recess (16), and a respective detent disc (8) with a recess (10) for each of the drive shafts (6, 7) of the switches (4, 5). A tension spring (22) exerts a symmetrical return force on the two-armed lever (13). The device described is intended for switch installations with draws, for example motor control cabinets. <IMAGE>
Patent NO-910983-L (NO)
Inventor: MODY RUSTOM K
IPC: E21B33/127
Filed: 1991-03-12
Abstract: An inflatable packing element (10) for an inflatable packer or bridge plug utilized in subterranean wells comprises a tubular elastomeric sleeve (30) which is surrounded by a plurality of circumferentially overlapping flexible metal ribs (12). The opposite ends of the ribs (12) are respectively welded to an external surface provided on a force transmitting sleeve (14). The sleeve (14) is provided with a shoulder (14a) having an abutting relationship with an internally projecting shoulder (20a) provided on the tubular mounting structure (20) for the inflatable element (10). <IMAGE>
Patent NO-911525-L (NO)
Inventor: KENNIS LUDO EDMOND JOSEPHINE
IPC: A61K31/4523
Filed: 1991-04-18
Abstract: Compounds of formula <CHEM> pharmaceutically acceptable acid addition salts thereof, and stereochemically isomeric forms thereof, wherein  Alk is C1-4alkanediyl, and D is <CHEM>  wherein R<1> represents C1-4alkyl, hydroxyC1-4alkyl, carboxaldehyde, carboxyl, C1-10alkylcarbonyloxyC1-4alkyl;  each R<2> represents hydrogen or C1-4alkyl; R<3> represents C1-4alkyl, hydroxyC1-4alkyl or methyl substituted with phenyl, 5-methyl-2-furanyl or 3-pyridinyl; and R<4> represents C1-3alkyl, phenyl, 5-methyl-2-furanyl or 3-pyridinyl,   which compounds are potent antagonists of dopamine and are therapeutically useful in treating patients suffering from acute psychoses. Compositions containing these compounds as active ingredient and processes of preparing said compounds and compositions.
Patent NO-912868-L (NO)
Inventor: PAULMICHL DIETER
IPC: E04H6/22
Filed: 1991-07-23
Abstract: A mechanical automobile parking facility with auto parking pallets, in which a vehicle is driven onto an auto parking pallet which is moved with the vehicle thereon to a predetermined space inside the facility. In order to guarantee reliable and abrasion free parking, a driving unit on rails is included whereby the driving unit with the auto parking pallet lying thereon, proceeds along a parking aisle and the auto parking pallet is pushed sideways from the driving unit by telescopic cylinders over glide rails into a free parking space, or conversely the auto parking pallet is taken from there onto the driving unit.
Patent NO-914797-L (NO)
Inventor: TOMKA IVAN
IPC: C08L3/00
Filed: 1991-12-05
Abstract: A single or multiple layer foil with an essentially reduced gas permeability has at least one layer composed at least in part of an essentially thermoplastic starch. In order to obtain a single or multiple layer foil which is at least almost completely insensitive to humidity, the one layer has at least one additional hydrophobic polymer, such as a polyolefine, which is mixed with the starch during the production of the one layer, and/or the starch is at least partially cross-linked at the surface of the one layer and/or the one layer is covered with at least one other layer which is at least almost completely insensitive to humidity.
Patent NO-924088-L (NO)
Inventor: ADAIR JOHN ROBERT
IPC: C12P21/08
Filed: 1992-10-22
Abstract: The present invention discloses humanized chimeric antibodies which are capable of binding to the intercellular adhesion molecule ICAM-1. Specifically, disclosed are humanized anti-ICAM-1 antibodies of the IgG1, IgG2, and IgG4 subtype. These antibodies are useful in treating specific and non-specific inflammation, rhinoviral infection, HIV infection, the dissemination of HIV infected cells, and asthma. In addition, the humanized antibodies disclosed can be useful in methods of diagnosing and localizing sites of inflammation and infection and tumors expressing ICAM-1.