baber/WOPTO huggingface dataset:
Patent BR-112021003652-B1 (BR)
Title: Composto derivado de amina heterocíclica, composição farmacêutica compreendendo o mesmo e uso do dito composto para prevenir ou tratar doenças autoimunes ou cânceres
Inventor: DEOK KI EOM
IPC: A61K31/496
Filed: 2019-08-27
Abstract: A presente divulgação refere-se a um novo derivado de amina heterocíclica representado pela seguinte Fórmula Química 1 e a uma composição farmacêutica compreendendo o mesmo, e o composto, de acordo com a presente divulgação, pode ser usado de maneira útil para a prevenção ou tratamento de doenças autoimunes ou cânceres. Fórmula Química 1 em que, na Fórmula Química 1, R1, R2, X1, X2, L, Y, A e B são iguais aos definidos no relatório descritivo.
Patent BR-122017006111-B1 (BR)
Title: métodos para controlar ervas daninhas
Inventor: ANTHONY J KINNEY
IPC: C12N15/82
Filed: 2007-10-30
Abstract: a presente invenção fornece métodos e composições relacionados com plantas de soja transgênicas de alto teor de ácido oleico / tolerantes a inibidores de als. especificamente, a presente invenção fornece plantas de soja com um evento dp-305423-1 que transmite um fenótipo de alto teor de ácido oleico e tolerância a, pelo menos, um herbicida inibidor de als. as plantas de soja que carregam o evento pd-305423-1 compreende a junção genômicas/transgene tendo pelo menos a sequência polinucleotídica de seq id no: 8, 9, 14, 15, 20, 21, 83 ou 84. a caracterização do sítio de inserção genômica do evento dp-305423-1 fornece uma eficiencia de produção melhorada e permite a utilização de marcadores moleculares para rastrear o transgene inserido nas populações reprodutoras e descendentes destas. são fornecidas vários métodos e composições para a identificação, detecção e utilização da soja evento pd-305423-1.
Patent BR-122017010425-B1 (BR)
Title: Method of producing an analytical measurement using a test strip
Inventor: HENNING GROLL
IPC: G01N27/416
Filed: 2005-06-20
Abstract: a presente invenção refere-se a método de produzir uma medição de um analito usando uma tira de teste (800) que compreende uma célula de medição, um eletrodo contador (216a), e um eletrodo de trabalho (814a). o método compreendendo as etapas de receber a tira de teste (800) no dispositivo biossensor; aplicar estímulo ao eletrodo contador (216a) para produzir o potencial através da célula de medição; medir a diferença de potencial desenvolvido através da célula de medição pela aplicação do estímulo; e adaptar o estímulo aplicado ao eletrodo contador com base na diferença de potencial medido desenvolvido através da célula de medição.
Patent BR-122017023426-B1 (BR)
Title: Sistema de circulação para uma extensão de água em um tanque
Inventor: COREY M SIMNIONIW
IPC: C02F1/76
Filed: 2007-04-09
Abstract: sistema de circulação (1) para extensões de água (2). em um conjunto de modalidades, para extensões de água maiores, são providos modelos modificados da chapa horizontal (20, 20?), na entrada (7) da mangueira de sucção (5). os modelos de chapa têm seções (22, 22?) que giram no sentido para baixo quando a plataforma flutuante (3) e a mangueira de sucção pendente (5) são rapidamente elevadas nas condições de ondas altas para deixar a água escapar no sentido para baixo, para fora da mangueira (5). adaptação para as bóias (9) para os braços alongados (31) da plataforma (3) também são feitas para essencialmente eliminar a geração de quaisquer torques que causem dano aos mesmos a partir das ondas altas. outro conjunto de modalidades é particularmente adaptado para sistemas menores em tanques municipais de água (41) para misturação completa da água (2) e tratamento para exterminar bactérias indesejáveis de oxidação de amônia e prevenir, ou ao menos inibir, o crescimento das mesmas.
Patent BR-122019023345-B1 (BR)
Title: Sistema de codificação de áudio, decodificador de áudio, método de codificação de áudio e método de decodificação de áudio
Inventor: JONAS LEIF SAMUELSSON
IPC: G10L19/00
Filed: 2008-12-30
Abstract: A presente invenção refere-se a um sistema de codificação de áudio inédito que pode codificar bem sinais tanto de áudio geral quanto de fala em baixas taxas de bit. Um sistema de codificação de áudio proposto compreende a unidade de predição linear para filtrar um sinal de entrada com base em um filtro adaptativo; uma unidade de transformação, para transformar um quadro do sinal de entrada filtrado em um domínio transformado; e uma unidade de quantização para quantizar o sinal do domínio transformado. A unidade de quantização decide, com base nas características do sinal inserido, codificar o sinal do domínio transformado com um quantizador baseado em modelo ou um quantizador não baseado em modelo. Preferivelmente, a decisão é baseada na duração do quadro aplicada pela unidade de transformação.
Patent CS-200207-B2 (CS)
Title: Method of preparing alkylene-dioxy-piperazine derivatives
Inventor: CYRUS RICHARD
IPC: A61K31/495
Filed: 1977-02-03
Abstract: Alkylenedioxy piperazine compounds of the formula   <IMAGE>   and salts thereof with physiologically tolerated acids, useful for the treatment of vascular and cardiac diseases, are disclosed, as are methods for making the compounds and pharmaceutical compositions containing the compounds.
Patent CS-195714-B2 (CS)
Title: Method of producing antimicrobially active derivatives of amoniglycoside
Inventor: ROSS BARRY C
IPC: A61P31/04
Filed: 1977-02-25
Abstract: 1529243 Oxazolidinones and oxazinones PFIZER Ltd 22 Feb 1977 [25 Feb 1976] 07529/76 Heading C2C Novel oxazolidinones and oxazinones of the general Formula III wherein R<SP>4</SP> is H or OH, R<SP>7</SP> is H, C 1-4  alkyl or benzyl, n is 0 or 1, except that n is not O when R<SP>4</SP> is OH, and X is O or (OH) 2 , are prepared by oxidation of the corresponding compound in which -CHX is replaced by or Aminoglycosides of the general formula wherein R is H or C 1-4  alkyl, R<SP>1</SP> is H or methyl, R<SP>2</SP> is OH or NH 2 , each R 3  is H or OH, one of R<SP>5</SP> and R<SP>6</SP> is H and the other is H or glycosyl and the broken line is an optional second bond when each R<SP>3</SP> is H, are prepared by reacting an amine of the general formula in which one or more of the free amino groups, other than the 1-amino group, may optionally be protected, with the oxazolidinone or oxazinone (III), reducing the product to form a substituted amine of the general formula in which one or more of the primary amino groups may optionally be protected, hydrolysing the cyclic urethane group and, if necessary, removing any amino-protecting groups and optionally removing the group R<SP>7</SP>, when R<SP>7</SP> is a benzyl group; by hydrogenation.
Patent CS-198297-B2 (CS)
Title: Method of producing derivatives of urea
Inventor: MAKISUMI YASUO
IPC: C07D263/48
Filed: 1978-04-28
Abstract: Urea derivatives of the formula   <IMAGE>   (wherein Ar represents a residue of 5- or 6-membered heteroaromatic ring; R represents a hydrogen atom or a C1-C6 alkyl group; R1 represents a C1-C6 alkyl group; and R2 represents a C1-C6 alkyl, C2-C6 alkenyl, or C1-C6 alkoxy group) are produced by reacting an amine of the formula Ar-NH-R (wherein Ar and R have the significance given above) with a carbamoyl halogenide of the formula   <IMAGE>  (wherein X represents a halogen atom, and R1 and R2 have the significance given above) in the presence of a Lewis acid in an inert solvent.
Patent CS-216203-B2 (CS)
Title: Method of controlling the pull tension at winding up the material bands on the roll and device for performing the same
Inventor: KATAOKA HIROSHI
IPC: B65H23/195
Filed: 1973-07-16
Abstract: 1429565 Winding webs KATAOKA MACHINE PRODUCT CO Ltd 17 July 1973 [17 July 1972] 33899/73 Heading B8R A method of controlling the tension in a wound web roll comprises the steps of continuously detecting the radius of a wound web roll, calculating the tension based on a theoretical equation and on the detected radius and applying the calculated tension to a comparison unit which stores a preset tension value to produce an output signal corresponding to the difference of the tensions compared in the unit for the purpose of controlling the winding torque applied to the wound web roll. In operation a required tension value F 0  and a tension gradient # are applied to a setting unit 10, Fig. 1, whose output forms the preset value stored in the comparison unit 11. The stored value is compared with a signal corresponding to a detected radius and emitted by detecting means 15 associated with the web roll spindle 14. The comparison unit 11 emits the torque controlling signal which is amplified in an amplifier unit 12 in turn producing an output signal which is applied to a torque actuator 13 which controls the torque applied to the spindle 14. The winding apparatus may include a plurality of web roll stands 78, Fig. 11, each supporting a plurality of pivotal arms 79 carrying respective spindles 83 on which are wound the web rolls 94. Web rolls 94 are formed from a wide web 30, fed over guide rollers 97, 98, 100, 95 and slit into a plurality of webs by a slitter 99. The arms 79 are biased by power cylinders 82 to control the nip pressure between web rolls 94 and the presser roller 95. The spindles 83 are driven by motors 90 and torque actuators 84 over belt drives 92, 89, 87 and gears 86, whereby the torque is controlled by radius detectors 81, connected to the pivotal shafts 80 of the arms 79 by endless chains 93 to indicate the angular displacement of the arms as a function of changing web roll radius.
Patent CS-241007-B2 (CS)
Inventor: STOLL KURT
IPC: F16L33/00
Filed: 1976-09-17
Abstract: Přípojná spojovací součást pro rychlé spojování
a rozpojování vedení z ohebného materiálu,
zejména pro vedení tlakového vzduchu,
s násuvným hrdlem a na druhé straně
s hrdlem závitovým, kde násuvné hrdlo je
vytvořeno pomocí podélných štěrbin jako
kleština a má kónickou oblast, alespoň zčásti
uspořádanou v ohjasti kleštiny, s prestavitelným
bezpečnostním kroužkem, má podstatu
v tom, že části se závitovým i nasouvacím
hrdlem jsou vzájemně nezávislé, oddělené,
vzájemně rozebíratelně zasunuté do
sebe, kde stupňovité vrtání části, tvořící zá­
vitové hrdlo, má na straně závitu koncový
průměr rovný vnitřnímu průměru vedení,
střední průměr rovný vnitřnímu průměru
nasouvacího hrdla a vnějšímu průměru konce
vedení, a největší průměr na vnějším
koncovém úseku, v němž je uložen těsnicí
kroužek.
Patent CS-264343-B2 (CS)
Title: Process for cleavaging perfluorpolyethers
Inventor: CAPORICCITO GERARDO
IPC: C08G65/32
Filed: 1986-11-20
Abstract: A process is disclosed for cracking high molecular weight perfluoropolyethers having neutral end groups obtained from the photooxidation of perfluoroolefins or the fluorination of hydrogenated polyalkylene oxides or by polymerization with opening of the partially fluorinated oxetane ring, said process being carried out in the presence of catalysts composed of fluorides, oxyfluorides or oxides of transi­tion metals or of Al, Sn, Sb at temperatures of from 150 to 380°C. The cracking process leads to the formation of low molecular weight perfluoropolyethers having neutral and acid end groups. The perfluoropolyether acids may be converted to functionalized perfluoropolyethers and are useful to produce new polymers.
Patent JP-2681073-B2 (JP)
IPC: A61N5/06
Filed: 1989-01-17
Granted: 1997-11-19
Abstract: This invention relates to a laser beam emitting probe suitably used for incision, transpiration, and coagulation of animal tissues or thermotherapy as the probe is kept in contact therewith, and a method of manufacturing such a probe. The laser beam emitting probe has a scattering surface at the free end portion thereof, which is bent to one direction on a longitudinal section thereof. In order to manufacture this probe, a laser beam transmitting member at least the free end portion of which is convergent is bent at the same portion thereof, and the resultant probe semiproduct is brought into contact with a liquid containing at least laser beam-absorptive powder, light scattering powder the refractive index of which is higher than that of the laser beam transmitting member, and laser beam transmitting powder the melting point of which is equal to or lower than that of the laser beam transmitting member, to bake the semiproduct at a temperature higher than the melting point of the laser beam transmitting powder but not higher than a level at which the laser beam transmitting member can no longer retain the shape thereof.
Patent AU-703636-B2 (AU)
Title: Tryptase polyclonal antibody and purification method for use in human tryptase immunoassay
Inventor: NILES ANDREW L
IPC: G01N33/543
Filed: 1996-10-31
Granted: 1999-03-25
Abstract: The disclosure describes highly specific tryptase polyclonal antibodies, and a method to purify the antibodies. Specifically, the invention relates to polyclonal antibodies which have the capacity to capture tryptase out of solution, a process to generate the antibodies, and an enzyme-linked immunosorbent assay (ELISA) for human tryptase which utilizes the antibodies.
Patent AU-760160-B2 (AU)
Title: Stable, high glycerol liquids comprising N-acyl amino acids and/or salts
Inventor: MASAAKI ARAI
IPC: A61K8/40
Filed: 2000-11-13
Granted: 2003-05-08
Abstract: The present invention describes high content glycerol liquid compositions comprising N-acyl amino acids and/or salts and defined sulfosuccinic acid monoesters. Although large amounts of glycerin normally destabilizes such compositions, inclusion of dialkylene glycol has been found to enhance stability. A method of enhancing stability of high content glycerin compositions comprising N-acyl amino acids or salts thereof and sulfosuccinic acid monoesters is also described.
Patent AU-599291-B2 (AU)
Title: Rearview mirror assembly with mounting arrangement including integrally molded dual axis pivot means
Inventor: FISHER ROBERT JAMES
IPC: B60R1/072
Filed: 1988-04-12
Granted: 1990-07-12
Abstract: A rearview mirror assembly (10) including an exteriorly convex shell (12) has a concave interior opening rearwardly when the shell is mounted on the side of a vehicle. A power operated assembly (14) is fixed secured to the shell (12) for mounting and moving a mirror assembly (16) for pivotal movement within the open rear of the shell about first and second intersecting pivotal axes normal to one another. The power operated assembly (14) includes a molded plastics member (20) of a size to fit within the concave interior of the shell (12) so as to extend inwardly of and generally across the open rear thereof. The plastics member (20) has spaced portions (22,24) fixedly secured with spaced portions (26,28) of the concave interior of the shell so that the molded plastics member serves as a strengthening strut for the open rear of the shell. The plastics member (20) has a dual axis pivot element (54) molded integrally on the central portion thereof which extends rearwardly therefrom and integral first and second surfaces (62) for engaging and supporting one fore and aft half of first and second power operated moving mechanisms (18) respectively of the power operated assembly. The other fore and aft half of the first and second power operated moving mechanisms (18) respectively is supported by a pair of separate substantially identical casing members (60).
Patent AU-689841-B2 (AU)
Title: Low molecular weight hyaluronic acid with peptide or protein
Inventor: JEDERSTROM GUSTAV
IPC: A61P17/00
Filed: 1995-01-10
Granted: 1998-04-09
Abstract: The invention relates to freeze-dried soft, flexible and continous matrix of low-molecular weight hyaluronic acid or salt thereof, in which the molecular weight of the hyaluronic acid is preferably between 50 000 and 200 000 Da, containing at least one peptide or protein. It also relates to a pharmaceutical composition in the form of a layer which is characterised by this freeze-dried low-molecular weight hyaluronic acid containing at least one peptide or protein. The drug is preferably chosen from at least one of GH, IGF-I, IGF-II and/or EGF and could be mixtured with an antibiotic agent. The process for the manufacture of this matrix and the use of the pharmaceutical composition for the manufacturing of a drug for wound healing is claimed. The invention discloses a method for accurately obtaining a predetermined dosage of a topically administerable drug which is characterised by freeze-drying a water solution of low-molecular weight hyaluronic acid and the peptide or protein to form a layer.
Patent AU-564930-B2 (AU)
Title: Imidazole and triazole fungicides
Inventor: KRAMER WOLFGANG
IPC: C07D405/06
Filed: 1983-06-29
Granted: 1987-09-03
Abstract: Substituted azoyl-ketones and -alcohols of the formula   <IMAGE>   in which A is a nitrogen atom or the CH group, B is CO or CH(OH), R1 is alkyl, alkenyl, alkinyl, optionally substituted phenylalkyl, optionally substituted cycloalkyl or optionally substituted cycloalkylalkyl, R2 is optionally substituted cycloalkyl or the grouping -C(CH3)2R3, and R3 is alkyl having more than 2 carbon atoms, alkenyl, alkinyl or the -CH=O group or a derivative thereof, or addition products thereof with acids or metal salts, exhibit plant growth regulating and fungicidal properties, several intermediates therefor are new.
Patent AU-690644-B2 (AU)
Title: A method for screening for the presence of a genetic defect associated with thrombosis and/or poor anticoagulant response to activated protein C
Inventor: BERTINA ROGIER MARIA
IPC: C12Q1/6883
Filed: 1995-02-14
Granted: 1998-04-30
Abstract: Method for screening for the presence of a genetic defect associated with thrombosis and/or poor anticoagulant response to activated protein C (APC). The method is directed at detecting one or more mutations at one or more of the cleavage and/or binding sites for APC of Factor V and/or Factor Va or at Factor VIII and/or Factor VIIIa at either nucleic acid or protein level or both.
Patent AU-656590-B2 (AU)
Title: High production laser welding assembly and method
Inventor: NEIHEISEL GARY LOUIS
IPC: B23K26/00
Filed: 1992-06-17
Granted: 1995-02-09
Abstract: A method for butt welding metallic sheets along a relatively long common seam line by providing a plurality of laser welding devices aligned above the common seam line, and effectively spaced from one another along a longitudinal axis. In a preferred embodiment, each welding device is independently adjustable in a direction parallel to a transverse axis which is perpendicular to the longitudinal axis. The metallic sheets are aligned on the upper surface in abutting relationship along the seam line and clamped for welding. Each laser welds only a portion of the sheets along the seam line, and the length of the relative movement between the welding devices and the sheets is greater than the effective spacing distance between welding devices to insure that a continuous weld bead is provided along the common seam line. <IMAGE>
Patent AU-730319-B2 (AU)
Title: Dihydrobenzofuran and related compounds useful as anti-inflammatory agents
Inventor: SCHERZ MICHAEL WIARD
IPC: A61P19/02
Filed: 1997-01-30
Granted: 2001-03-01
Abstract: A compound having the structure:   <IMAGE>   wherein (a) n is from 1 to about 3; (b) X is selected from the group consisiting of O, S, SO, or SO2; (c) Y is independently hydrogen or straight, branched or cyclic alkyl having from 1 to about 4 carbon atoms, or the Y's are bonded together to form an alkanyl ring having from 3 to about 7 atoms; (d) Z is hydrogen or straight, branched or cyclic alkyl having from 3 to about 10 atoms other than hydrogen; (e) W is O or S; and (f) R1, R2 and R3 are independently hydrogen, straight, branched or cyclic alkyl having from 1 to 10 carbon atoms, aryl, heterocyclyl, heteroaryl, hydroxy, or alkoxy; or R1, R2 or R3 may be bonded to form one or more rings each ring having from 3 to about 7 atoms wherein from 1 to 3 atoms may be heteroatoms. pharmaceutical compositions comprising such compounds, and methods of treating inflammation or pain using such compounds.
Patent AU-652259-B2 (AU)
Title: Base station for a radio system with arrangement for monitoring quality of radio-transmission channels
Inventor: HANNINEN JOUNI
IPC: H04B17/00
Filed: 1992-06-05
Granted: 1994-08-18
Abstract: PCT No. PCT/FI92/00176 Sec. 371 Date Feb. 5, 1993 Sec. 102(e) Date Feb. 5, 1993 PCT Filed Jun. 5, 1992 PCT Pub. No. WO92/22963 PCT Pub. Date Dec. 23, 1992.The base station includes for monitoring the quality of a radio link between the base station and mobile stations, a generator (1, 2, 3) for generating a square wave signal (CK) having a monitoring signal frequency; and a filter (4) for generating a monitoring signal (CS) from the square wave signal (CK). The frequency of the monitoring signal is set by a control (12) having two modes of operation; in the first mode of operation, the control controls the generator to transmit an analog monitoring signal by maintaining the frequency of the square wave signal (CK) at a constant value throughout the duration of the monitored radio link, and in the second mode of operation, the control controls the generator (1, 2, 3) to transmit a digital monitoring signal by varying the frequency during the monitored radio link in response to changes in the logical state of the monitoring signal between a first frequency corresponding to the first logical state and a second frequency corresponding to the second logical state.
Patent AU-565525-B2 (AU)
Title: Pivotable clay gun for sealing the tapholes of blast furnaces
Inventor: COOPER ARTHUR WILLIAM
IPC: C21B7/12
Filed: 1984-04-19
Granted: 1987-09-17
Abstract: A shaft furnace plugging apparatus is presented which occupies very little space and sweeps out a relatively low and comparatively flat continuous trajectory between an inoperative position and an operative position. The plugging apparatus includes a clay gun pivotably mounted on a first end of a jib, the jib being rotatable about a support column. The apparatus also includes a pair of hydraulic cylinders, the first hydraulic cylinder being pivotably attached between a second end of the jib and an intermediate pivotable frame and the second hydraulic cylinder which is operative between the intermediate pivotable frame and a fixed support frame.
Patent AU-562506-B2 (AU)
Title: Prostacyclin derivatives
Inventor: SKUBALLA WERNER
IPC: A61K31/335
Filed: 1984-06-22
Granted: 1987-06-11
Abstract: 1. 5-Cyanoprostacyclines of the general formula I   see diagramm : EP0130142,P10,F2   wherein A represents a _t_r_a_n_s-CH = CH- or -C -= C- group, W represents a hydroxymethylene, acetoxymethylene,   see diagramm : EP0130142,P10,F3   wherein the OH or acetoxy group may have the alpha- or b¢eta-configuration, D and E together represent a direct bond or D represents a straight-chained alkylene group having from 1 to 5 C atoms or a branched alkylene group having from 2 to 5 C atoms, E represents an oxygen atom, a -C -= C- bond or a direct bond, R2 represents a C1 -C7 -alkyl group or phenyl, R1 represents a hydroxy or acetoxy group and R3 represents the acetal radicals   see diagramm : EP0130142,P11,F1
Patent AU-688952-B2 (AU)
Title: Thrombin inhibitors
Inventor: LUMMA WILLIAM C
IPC: A61K31/50
Filed: 1995-07-18
Granted: 1998-03-19
Abstract: Compounds of the invention have the following structure:   <IMAGE>   for example   <IMAGE>   These compounds inhibit thrombin and associated thrombosis.
Patent AU-622164-B2 (AU)
Title: Fixing-piece with guide-collar
Inventor: JOCHUM PETER
IPC: F16B19/14
Filed: 1989-04-12
Granted: 1992-04-02
Abstract: The fastener (1), having a head (2), shank (3) and tip (4), is provided with a thread (5) in the rearward end region of the shank (3). Onto the thread (5), at a distance (A) from the head (2), there is screwed a guide washer (10) which is designed in the manner of a dome and has a wall region (13) extending in a conical shape from the base (11) in the insertion direction. The guide washer (10) can be deformed, thus braking the insertion process. 
<IMAGE>