baber/WOPTO huggingface dataset:
Patent CZ-308800-B6 (CZ)
Title: Heterocyclic nitrogenous derivatives of purine, pharmaceutical preparations containing these derivatives and their use in neuroprotection
Inventor: GONZALES GABRIEL
IPC: C07D473/16
Filed: 2019-02-12
Abstract: The invention relates to formula I heterocyclic purine derivatives with nitrogen-containing substituents, their use in medical applications and preparations containing these derivatives. The new generation of compounds has selective antineurodegenerative properties on nerve cells and tissues and can be advantageously used in treating and prophylaxis of neurodegenerative diseases, in particular in the treatment and prophylaxis of Parkinson's disease.
Patent CZ-286323-B6 (CZ)
Title: Device for suspension mountaineering
Inventor: HRUS MIROSLAV ING CSC
IPC: A63B29/00
Filed: 1996-09-24
Abstract: The invented device for suspension mountaineering is formed by a floor slap (1) with continuously performed slot (2) passing vertically through said floor slab (1) profile and in which the securing element (6, 7) of the mountaineer is guided.
Patent CZ-286065-B6 (CZ)
Title: Isopropyl-(2-methoxyethyl)-4-(2-chloro-3-cyanophenyl)-1,4-dihydro-2,6-dimethylpyridine-3,5-dicarboxylate, process of its preparation, medicaments in which this substance is comprised, use of this compound and 2-chloro-3-cyanobenzaldehyde as intermediate employed during preparation of this compound
Inventor: MEIER HEINRICH DR
IPC: C07D211/90
Filed: 1994-12-08
Abstract: In the present invention there are disclosed rac-isopropyl-(2-methoxyethyl)-4-(2-chloro-3-cyano-phenyl)-1,4-dihydro -2,6-dimethylpyridine-3,5-dicarboxylate of the general formula I and pure enantiomers thereof, further processes of their preparation and their use as medicaments intended particularly for treating cerebral and  neuronal diseases, as well as an intermediate for preparing the above indicated compound.
Patent SK-283143-B6 (SK)
Title: Pharmaceutical preparation for controlled release
Inventor: MILLER RONALD BROWN
IPC: A61K31/137
Filed: 1994-05-10
Abstract: Pharmaceutical preparation for controlled release in the form of tablet or capsule containing multi-particles of size 0.1 to 3 mm and comprising tramadol or pharmaceutically acceptable salt thereof in the form of hydrochloride tramadol in the matrix of pharmaceutically acceptable bearer. The matrix contains substantially hydrophobic meltable material. The production method of the pharmaceutical preparation contains processing of the tramadol mixture or pharmaceutically acceptable salt thereof in the form of powder in the high-speed mixer and powdered hydrophobic meltable material with a total amount of the active substance 10 to 90 wt. % related to the weight of the final product, processing of the active substance in the high-speed mixer, the mixture is molten or softens with the production of agglomerates, which are subsequently broken with the production of the mixture of powder and small particles and repeatedly the mechanic processing in the high-speed mixer continues to the production of the particles of the size 0.1 to 3.0 mm, which are filled into the capsules or pressed into the tablets, whilst each capsule or tablet contains 50 to 800 mg of the active ingredient.
Patent SK-281313-B6 (SK)
Title: Preparation of halogenated alcohols
Inventor: BOWDEN MARTIN CHARLES
IPC: C07C29/38
Filed: 1994-05-25
Abstract: The invention discloses a process for the preparation of a halogenated alcohol of formula: CF3-CXCl-CH(OH)-CH=C(CH3)2 wherein X is bromo or chloro which comprises reacting a compound of formula: CF3CHXCl with 3-methylbut-2-en-1-al in the presence of a strong base and an inert solvent. The products are useful intermediates for the manufacture of insecticides.
Patent SK-284047-B6 (SK)
Title: Process for producing L-lysine by fermentation
Inventor: KOJIMA HIROYUKI
IPC: C12N9/88
Filed: 1996-03-14
Abstract: A process for producing L-lysine which comprises culturing in an appropriate medium a bacterium belonging to the genus Serratia, which has been transformed by introducing a DNA encoding a dihydrodipicolinic acid synthetase originating in a bacterium belonging to the genus Escherichia or Serratia having a mutation of releasing the feedback inhibition by L-lysine and another DNA encoding an aspartokinase originating in a bacterium belonging to the genus Escherichia or Serratia having a mutation of releasing the feedback inhibition by L-lysine into the cells, and harvesting the L-lysine thus accumulated in the culture.
Patent CZ-300389-B6 (CZ)
Title: Derivate of aminoethylphenoxyacetic acid and pharmaceutical composition containing thereof
Inventor: TAMAI TETSURO
IPC: C07C/
Filed: 1998-07-15
Abstract: In the present invention, there is disclosed a derivate of aminoethylphenoxyacetic acid of the general formula I, wherein Ri1 represents a hydrogen atom or an alkyl group containing 1 to 6 carbon atoms, which is optionally substituted with a phenyl group or a naphthyl group and Ri2 represents a hydrogen or halogen atom, wherein the carbon atom designated as (R) signifies a carbon atom with (R) configuration and the carbon atom designated as (S) signifies a carbon atom with (S) configuration, or its pharmaceutically acceptable salt and its medical applications. There is also disclosed a pharmaceutical composition for reducing pain and support for bladder stones removal during urolithiasis containing the above-described derivative.
Patent CZ-297198-B6 (CZ)
Title: Preparation for inhibiting further growth of cancer tumor of prostate in mammals
Inventor: DIONNE CRAIG A
IPC: A61K38/04
Filed: 1998-08-13
Abstract: A method of treating prostate cancer by co-administering a tyrosine kinase inhibitor such as an indolocarbazole and a chemical castration agent is disclosed. A composition containing a tyrosine kinase inhibitor and a chemical castration agent is also disclosed.
Patent CZ-301784-B6 (CZ)
Title: Detector system for a corpuscular beam apparatus and corpuscular beam apparatus with such a detector system
Inventor: DREXEL VOLKER
IPC: G01N23/225
Filed: 2001-03-13
Abstract: The present invention relates to a detector system for a corpuscular beam apparatus, particularly scanning electron microscope, having a target structure (5) arranged in a beam path of said corpuscular beam apparatus, wherein said target structure (5) comprises a central region (6) adjacent to optical axis (25) of the corpuscular beam apparatus and near to the axis. The central region (6) is of a material strongly converting the electrons. It further comprises a region (7) remote from said optical axis (25) as well as a detection system for detection of conversion electrons emitted from said region (6) of electron-converting material. Said region (28) remote from said optical axis (25) is performed as a half ring and said region (29) near said optical axis (25) is made as a bridge connecting ends of said half ring region (28) remote from said optical axis (25).
Patent CZ-301574-B6 (CZ)
Title: Apparatus for pedal detachment in the course of vehicle frontal collision
Inventor: LEKSA LIBOR
IPC: B60R99/00
Filed: 2004-05-28
Abstract: n the present invention, there is disclosed a pedal release device in a motor vehicle in case of a front impact comprising a transmission arm (6), connected to a swiveling pedal leg (5) through an axial coupling (7) in the pedal leg (5) turning axis. Said transmission arm (6) is in contact with a controlled member being represented by a brake power assist unit or a main brake or coupling hydraulic cylinder. A pressure spring (4) and a disengaging member (10) are assigned to said axial coupling (7). A first part (8) of the axial coupling (7) is fixedly coupled with the pedal leg (5) while the second part (9) thereof is coupled with said transmission arm (6). The disengaging member (10) abut a vehicle frame (12) at a point that is farther from the point of the vehicle front impact if compared with the point of the pedal leg (5) rotatable mounting. The disengaging member (10) is provided with a wedge-shaped portion that reaches between the axial coupling (7) parts (8, 9) and further with a support (11) serving as driver side abutment for the pedal leg (5) when the disengaging member (10) disengages the axial coupling (7).
Patent CZ-299687-B6 (CZ)
Title: Process for preparing controlled layers of fibrin on solid surfaces
Inventor: BACAKOVA LUCIE
IPC: C12N11/082
Filed: 2006-12-21
Abstract: The present invention relates to a process for preparing controlled layers of fibrin on solid surfaces for cultivation of cells wherein the preparation process is characterized in that fibrinogen, preferably in concentration of 2 to 200 Ág/ml is adsorbed by adsorption from a solution on a solid surface in the first step, so treated surface is then subjected in the second step to the action of a thrombin solution preferably exhibiting activity of 0.1 to 10 U/ml, whereupon in the third step the surface is treated with a solution containing fibrinogen, preferably in concentration of 200 Ág/ml or greater and a thrombin inhibitor antithrombin or antithrombin in combination with heparin or heparinized blood plasma, whereby the phase of the thrombin solution treatment and subsequent treatment with the solution containing fibrinogen and antithrombin can be carried out repeatedly. Said fibrinogen solution in the first step can be represented by anti-coagulated blood plasma.
Patent CZ-306879-B6 (CZ)
Title: A biocomposite with a PLA matrix and banana fibres
Inventor: LENFELD PETR
IPC: C08L99/00
Filed: 2012-10-25
Abstract: This is a composite with a targeted composition of the PLA matrix and the fibrous filler based on natural materials in order to improve the final and useful properties of plastic parts with ecologically much lower loadability compared to 100% synthetic products, wherein the essence of the solution lies in the fact that the composite comprises from 50 to 90 wt% of a PLA polymer and from 10 to 50 wt% of natural banana fibres (the fibre length ranges from 0.2 to 3 mm) with the possibility of other additives.
Patent CZ-307636-B6 (CZ)
Title: Tažný vozík pro stolici na tažení trubek
Inventor: DVOŘÁK JOSEF
IPC: B21C1/28
Filed: 2017-05-31
Abstract: Tažný vozík je tvořen tělesem (1) vozíku pojíždějícím po dráze (6) s průvlakovou deskou (7). Těleso (1) vozíku je opatřeno pneumatickými ovládacími ventily (5) pneumatického obvodu pro ovládání pneumatických válců (2) s upínacími čelistmi (3) trubek (9). Pneumatické ovládací ventily (5) jsou ve výchozí poloze "A" tělesa (1) vozíku ve styku s pneumatickým válcem (12) s pohyblivým dorazem, uloženým na dráze (6) za průvlakovou deskou (7) stolice. V koncové poloze "B" tělesa (1) vozíku jsou pneumatické ovládací ventily (5) ve styku s pneumatickým válcem (11) s výklopným dorazem, uloženým na druhé straně dráhy (6). Na dráhu (6) navazuje výklopný stůl (8), pro zachycení trubek (9), který je upevněn na stolici (10).
Patent CZ-309095-B6 (CZ)
Title: Passive system with increased reliability for residual heat removal from a nuclear reactor and doing it
Inventor: Hájek Petr
IPC: G21C15/26
Filed: 2020-12-08
Abstract: A passive system with increased reliability for removing residual heat from a nuclear reactor comprising a heat exchanger (11), a chimney (12) formed by a two-channel pipeline and a flow redirection device (2) with an internal channel (21) with a valve, which separates the channel segment (21) on the (3) side of the reactor from the channel segment (21) on the (1) side of the heat exchanger (11), and an outer channel (22) with at least one valve in the baffle which separates the channel segment (22) on the reactor side (3) from the channel segment (22) on the heat exchanger (11) side (1). The channel segment (21) on the (1) side of the heat exchanger (11) is connected to the channel segment (22) on the reactor side (3) by at least one connecting channel and the channel segment (22) on the (1) side of the heat exchanger (11) is connected by at least one connecting channel to the channel segment (21) on the reactor side (3), each of the connecting channels have at least one valve.
Patent SK-287051-B6 (SK)
Title: Workpiece clamping device
Inventor: FRIES KARL
IPC: B25B23/10
Filed: 2002-02-22
Abstract: A workpiece clamping device including a handle and a holder. Both part (1, 3) intended for fixing against each another have matched surfaces (4, 5) bearing in working position against each other and being clamped against each another through the mediation of fixing means extending transversely or in the right angle to a contact plane of these matched surfaces (4, 5). Matching projections (9) preventing mutual shift of the parts (1, 3) coupled to each another transversely to the fixing means, optionally inside the contact surface of the matched surfaces (4, 5), are additionally arranged on the fixing place to the matching surfaces (4, 5) fixing mutual position. These projections (9) exactly center both the parts (1, 3) transversely to the contact plane at least in the direction (X) and in the direction (Y). At the same time, the matching projections (9) are arranged on one of the parts (3) between the matched surfaces (4, 5), and the other part (1), intended for connection therewith has in the corresponding points a matching recess (10) that engage with the projection when the parts are fastened to each another. Said matching projections (9) are arranged in a region (11) of the part (3) that can deflect or is elastic in axial direction against deformation force applied thereto.
Patent SK-286153-B6 (SK)
Title: Flame arrester
Inventor: READE CHARLES OSBORN
IPC: A62C4/02
Filed: 1999-11-09
Abstract: A flame arrester (10) comprising a flow passage (16) in which is disposed a two dimensional array of adjacent circular section rods (24, 25), each being generally co-aligned and arranged transverse to the flow direction (F), such that fluids flowing in the passage must pass between the roads (24). The roads are arranged in rows and are of solid material.
Patent CZ-298571-B6 (CZ)
Title: Method for reprocessing waste oils and producing high-grade base oils
Inventor: POEHLER JOACHIM
IPC: C10G21/20
Filed: 1999-11-11
Abstract: Method for reprocessing waste oils and production of high-grade base oils, comprising the following steps: A) distillation of the waste oil for removal of low boiling organic fractions and removal of water, wherein the waste oil to be reprocessed is treated with concentrated aqueous potassium hydroxide solution during the distillation step; B) distillation under vacuum of the waste oil obtained according to step A) for segregation of fuel oil and diesel fractions with boiling cut of about 170 to 385 degC in the form of high grade fuel oils; C) non-destructive distillation of the distillation residue from step B) by means of thin film evaporation in vacuum to obtain a lubricating oil fraction, which can be separated, as needed, via a subsequent distillative fractioning step, optionally under vacuum, into boiling cuts of different viscosity states; D) if appropriate, non-destructive distillation of the bottom product from step C) in order to obtain a lubricating oil fraction of kinematic viscosity at 40 degC in the range of 60 to 120 mme2/s, which can be segregated, as needed, optionally under vacuum, by means of a subsequent distillative fractioning step; E) extraction of the fraction or fractions in the form of lubricating oil fractions or boiling cuts of different viscosity states from step C) and optionally D) with N-methyl-2-pyrrolidone (NMP) and/or N-formylmorpholine (NMF) as extraction medium in order to obtain very high grade base oils.
Patent CZ-302941-B6 (CZ)
Title: Tricyclic compound and pharmaceutical composition containing thereof
Inventor: WEBBER STEPHEN EVAN
IPC: C07D221/00
Filed: 2000-01-10
Abstract: In the present invention, there is disclosed a tricyclic compound of the general formula A, which is are poly(ADP-ribosyl)transferase (PARP) inhibitor, and which is useful as therapeutic in the treatment of tumors and the amelioration of the effects of stroke, head trauma, and neurodegenerative disease. As tumor therapeutic, the compound of the present invention may be used, for instance in combination with cytotoxic agents and/or ionizing radiation.
Patent CZ-293103-B6 (CZ)
Title: Composition for combating wood damaging fungi
Inventor: RUSSEL PHILIP ERIC
IPC: A01P3/00
Filed: 2000-10-17
Abstract: In the present invention, there is disclosed the use of a compound of the general formula I, in which R represents the group of the general formula a or b, in which each substituent Re1, which may be the same or different, represents an alkyl group containing 1 to 4 carbon atoms, an alkoxy group having 1 to 4 carbon atoms, a trifluoromethyl group or a halogen atom and n is a number of 0 to 3, for controlling wood damaging fungi such as Coriolus versicolor, Poria placenta, Lentinus lepideus, Trametes versicolor, Serpula lacrymans, Coniophora puteana and Gloeophyllum trabeum.
Patent CZ-293498-B6 (CZ)
Title: Safety equipment, particularly a safe and process for producing thereof
Inventor: WIENKE JURGEN WIENKE JURGEN
IPC: E05G1/00
Filed: 2002-05-20
Abstract: The present invention relates to safety equipment, particularly a safe. Such safe wall (1) consists of filler elements (4) and reinforcing steel sections or another armoring. The walls (1) are made as a compact and single layer flat section of concrete (2), whereby the armoring is arranged within the concrete (2) in the wall (1) along with the filler elements (4). Process for producing such safe is characterized in that firs armoring is arranged within a mold whereupon a quick-setting concrete (2) is poured along with another filler material formed by the reinforcing elements (3) of recycled material and a dyestuff (8) therein.
Patent CZ-301700-B6 (CZ)
Title: Installation arrangement for solenoid controlled handle operation in a door lock
Inventor: RAATIKAINEN JUHA
IPC: E05B59/00
Filed: 2002-01-17
Abstract: The present invention relates to an installation arrangement for a solenoid controlled handle operation in a door lock in which force transmission from an operation axis (3) for a handle or the like to a follower (4) acting on a bolt (12) of the lock is arranged by means of a movable coupling member (6, 6'), which receives its guidance from a solenoid arrangement. The follower (4) is provided with two separate torsion units (13, 14) which are installed on the operation axis (3) on different sides of the follower (4) and are rotatably supported to it and which can be selectively coupled by means of said coupling member (6, 6') to be in force transmission connection with the follower (4). Said operation axis (3) is arranged such that a spindle (17) of the handle arranged on the operation axis (3) is in direct connection for force transmission with the follower (4) wherein the arrangement includes an adapting member (16), which is arranged to be installed in a spindle (17) aperture (13a, 14a) of either one of the torsion units to thereby prevent a spindle (17) of the handle from directly connecting with the follower (4), so that the spindle (17) of the handle is in force transmission connection with the torsion unit (13,1 4) in question. A door lock is provided with the above-described installation arrangement.
Patent CZ-301297-B6 (CZ)
Title: Plasma arc torch, plasma arc torch electrode and method for operating such plasma arc torch
Inventor: CONWAY CHRISTOPHER J
IPC: B23K9/29
Filed: 2003-04-07
Abstract: In the present invention, there is disclosed a plasma arc torch, which comprises a cathode element (22, 22a), which forms a perimeter surface (227), an electrode (100, 100a) constructed for electrical contact with the cathode element (22, 22a) and a fluid passage between the cathode element (22, 22a) and the electrode (100, 100a), whereas the electrode (100, 100a) forms a perimeter surface (223) adjacent to the perimeter surface (227) of the cathode element (22, 22a) and these adjacent perimeter surfaces (225, 227) provide an electrical contact and fluid passage. There is also disclosed an electrode (100, 100a) and a method for operating the above-described plasma torch.
Patent BR-PI0116208-B8 (BR)
Inventor: KARIN HOFFMANN
IPC: A61K31/00
Filed: 2001-12-14
Abstract: The invention provides novel water-free medical skin care formulations comprising micronized urea dispersed in a fatty phase. The fatty phase consists essentially of hydrocarbons and is essentially free from ingredients with known allergenic potential such as perfumes or perfume substitutes (fragrances), preservatives, colorings, plant extracts, PEGs, cetylstearyl alcohol, lanolin alcohols, lower alcohols, and proteins, thus being particularly suitable for patients with highly sensitive skin. The formulations of the invention have favorable sensorial properties and are stable for an extended period of time. The formulations are suitable for medical skin care, such as for the treatment of severely affected dry, sensitive skin and for the therapy or therapy support of ichthyosis, psoriasis, and eczema. The invention also provides methods of manufacturing such water-free skin care formulations.
Patent CH-703591-B8 (CH)
Title: Strahlpumpeninspektionsvorrichtung.
Inventor: DOROSKO ROBERT K
IPC: G21C17/00
Filed: 2011-08-02
Abstract: Die vorliegende Erfindung betrifft eine Strahlpumpeninspektionsvorrichtung, die einen Sondenantrieb (14) enthält, der mit einem Führungstrichter (10) gekoppelt ist. Gemäss der vorliegenden Erfindung sind ein Sondenantrieb (14a–f), der so ausgebildet ist, dass er eine axiale Bewegung einer in die Vorrichtung einführbaren Sonde entlang einer Länge der Vorrichtung bewirkt, und der Führungstrichter (10), der so ausgebildet ist, dass er die Sonde bis auf eine gegebene Tiefe in die Vorrichtung einführt, am Korpus (101) der Vorrichtung angeordnet. So wird die für eine Inspektion benötigte Zeit verringert, wodurch das Personal einer geringeren radioaktiven Kontaminierung ausgesetzt wird.
Patent EP-1198701-B8 (EP)
Inventor: KAUPPILA JARMO
IPC: G01M99/00
Filed: 2000-07-06
Granted: 2010-07-28
Abstract: A method of monitoring the condition of apparatuses wherein the condition of the apparatus is measured from one or more rotating objects by means of a fixedly mounted condition monitoring system during the operation of the apparatus when it operates at its normal operating speed. In the method, at least one signal indicating the condition of the apparatus and the steadiness of the operation is measured during the change in the operating speed of the apparatus and desired characteristic values and/or functions are calculated from each signal measured in this manner as a function of measured time and/or rotational speed.
Patent EP-1728770-B8 (EP)
Inventor: RAINER THOMAS DR
IPC: B41M5/26
Filed: 2006-04-27
Granted: 2008-10-15
Abstract: A process for marking the surface of an object, comprises locating a carrier element so it is in contact or at a distance from the surface. The element has an embedded metal layer, and the layers form a low E layer system. A laser is directed against the layer system, and material is transferred to the object surface and adheres to it as a matrix of metallic nano particles.. The matrix is formed from the substances in the layer system.
Patent EP-1093457-B8 (EP)
Inventor: RUBEN STEVEN M
IPC: A61K31/711
Filed: 1999-03-05
Granted: 2011-02-02
Abstract: The present invention relates to a novel human protein called Cytokine Receptor Common Gamma Chain Like, and isolated polynucleotides encoding this protein. Also provided are vectors, host cells, antibodies, and recombinant methods for producing this human protein. The invention further relates to diagnostic and therapeutic methods useful for diagnosing and treating disorders related to this novel human protein.
Patent BR-PI0509150-B8 (BR)
Title: compostos para a inibição de angiogênese e uso destes
Inventor: FRANK OSTERKAMP
IPC: C07D405/14
Filed: 2005-03-24
Abstract: compostos para a inibição de angiogênese e uso destes. a presente invenção invenção refere-se aos compostos de estrutura (i). particularmente esta invenção é direcionada aos compostos de estrutura (viii) em que as variáveis são definidas como na descrição. estes compostos são inibidores de integrina e são úteis no tratamento de doenças nas quais uma inibição de angiogênese é desejada.