baber/WOPTO huggingface dataset:
Patent CZ-288971-B6 (CZ)
Title: Redispersible dispersion powder composition, aqueous polymer dispersions prepared therefrom and use thereof
Inventor: FIGGE REINER DR
IPC: C08L33/10
Filed: 1997-01-16
Abstract: The invented redispersible dispersion powder composition contains (a) a water-insoluble base polymer having a glass transition temperature of -60 degC to +80 degC being selected from a group comprising homo- and copolymers of vinyl esters, acrylic acid esters, methacrylic acid esters, styrene and vinyl chloride, or a mixture of the base polymers mentioned, (b) 2 to 40 percent by weight, based on the base polymer, of a water-soluble atomizing protective colloid, and (c) 0 to 30 percent by weight, based on the total weight of polymeric constituents, of an antiblocking agent, wherein the component (b) comprises non-neutralized homo- or copolymers of olefinically unsaturated mono- or dicarboxylic acids or anhydrides thereof, or partly neutralized homopolymers of olefinically unsaturated mono- or dicarboxylic acids or anhydrides thereof or partially neutralized copolymers of olefinically unsaturated mono- or dicarboxylic acids or anhydrides thereof having an acid content greater than 80 mol
Patent CZ-293558-B6 (CZ)
Title: Derivatives of piperidine and piperazine, process of their preparation and use as well as pharmaceutical compositions based thereon
Inventor: BOTTCHER HENNING DR
IPC: C07D405/14
Filed: 1994-09-28
Abstract: In the present invention, there are disclosed derivatives of the general formula I, wherein Ind represents an indol-3-yl radical, which is unsubstituted or mono- or polysubstituted with OH, OA, CN, a halogen, CORe2 or CHi2Re2; Re1 represents benzofuran-5-yl or 2,3-dihydrobenzofuran-5-yl, chroman-6-yl, chroman-4-on-6-yl, 3-chromen-6-yl or chromen-4-on-6-yl, which is unsubstituted or monosubstituted with the CN, CHi2OH, CHi2OA or CORe2 group; Q denotes CimHi2m; Z represents N or CRe3; A denotes alkyl having 1 to 6 carbon atoms; Re2 represents  OH, OA, NHi2, NHA or NAi2; Re3 denotes H, OH or OA; and m is 2, 3 or 4. The above-described derivatives are active on the central nervous system and they are therefore suitable for treating stress, depression and side effects when treating hypertension.
Patent CZ-292482-B6 (CZ)
Title: Process for purifying thrombin-like proteases from snake venom
Inventor: SCHWARZ MARGARETE
IPC: A61K38/00
Filed: 1997-02-18
Abstract: The invented purification process comprises the following steps: a) obtaining a solution comprising the protease; b) loading the protease solution onto an affinity chromatography matrix or an anion exchange resin; c) eluting the protease in an eluate solution from the affinity chromatography matrix or anion exchange resin; d) loading the eluate solution from step c) onto a matrix of glass beads; said glass beads having a pore diameter of from 25 to 35 nm and a particle size of from 30 to 60 micron; said eluate being applied to the matrix of glass beads in a basic solution at a pH value of from 7.5 to 9.0 whereby the glass beads adsorb the thrombin-like protease from snake venom; e) eluting the protease in an eluate solution from the matrix of glass beads; f) loading the eluate solution from step e) onto a size exclusion gel matrix or onto a matrix of glass beads; said glass beads having a pore diameter of from 25 to 35 nm and a particle size of from 30 to 60 micron; said eluate being applied to the matrix of glass beads in an acidic solution; and g) eluting and recovering the purified protease.
Patent CZ-284946-B6 (CZ)
Title: USE OF cGMP PDE PYRAZOLOPYRIMIDINONE INHIBITORS AND GENERAL USE OF THE cGMP PDE PYRAZOLOPYRIMIDINONE INHIBITORS FOR PREPARING MEDICAMENTS
Inventor: ELLIS PETER
IPC: A61K45/00
Filed: 1994-05-13
Abstract: The use of a compound of formula (I) wherein R1 is H; C1-C3 alkyl; C1-C3 perfluomalkyl; or C3-C5 cycloalkyl; R2 is H; optionally substituted C1-C6 alkyl; C1-C3 pefluoroalkyl; or C3-C6 cycloalkyl; R3 is optionally substituted C1-C6 alkyl; C1-C6 perfluoroalkyl; C3-C5 cycloalkyl; C3-C6 alkenyl; or C3-C6 alkynyl; R4 is optionally substituted C1-C4 alkyl, C2-C4 alkenyl, C2-C4 alkanoyl, (hydroxy)C2-C4 alkyl or (C2-C3 alkoxy)C1-C2 alkyl; CONR5R6; CO2R7; halo; NR5R6; NHSO2NR5R6; NHSO2R8; SO2NR9R10; or phenyl, pyridyl, pyrimidinyl, imidazolyl, oxazolyl, thiazolyl, thienyl or triazolyl any of which is optionally substituted with methyl; R5 and R6 are each independently H or C1-C4 alkyl, or together with the nitrogen atom to which they are attached form an optionally substituted pyrrolidinyl, piperidino, morpholino, 4-N(R11)-piperazinyl or imidazolyl group; R7 is H or C1-C4 alkyl; R8 is optionally substituted C1-C3 alkyl; R9 and R10 together with the nitrogen atom to which they are attached form an optionally su
Patent CZ-289483-B6 (CZ)
Title: Semi-finished surface-cladding component
Inventor: BOE HANS PETER
IPC: C04B28/04
Filed: 1997-02-13
Abstract: In the present invention there is disclosed a half-finished product (1) of a construction component for cladding structural surfaces (2), consisting of a glass pane (4) and a layer (5) of bonding mortar on one side of the glass pane (4). Said bonding mortar layer (5) consists of a fine-particle neutral aggregate and cement and is gauged with an aqueous dispersion of a polyacrylic acid derivative, whereby the polyacrylic acid derivative has a maximum logarithmic decrement of torsional vibration damping at temperatures below 0 degC. The bonding mortar on one side of the glass pane (4) is hardened with a deficiency of hydration water, whereby a bond with the surface (2) to be covered can be established through the contact of the bonding mortar layer (5) of the construction component half-finished product (1) with gauged and setting concrete of the surface or with so called tile adhesive.
Patent CZ-291291-B6 (CZ)
Title: Transmission and reception of television programs and other data
Inventor: FURET THIERRY
IPC: G06F21/10
Filed: 1997-04-25
Abstract: In a digital television system, a receiver/decoder (2020) (or "set-up control box") can download one of more of several applications, which can be run by the receiver/decoder (2020) to provide interactivity with the user. These  applications include: an Internet browser application which uses a PSTN connection to make Internet requests and the television signal path to receive Internet responses; a shopping application operable in an "impulse" mode and a "catalogue" mode; a banking application; a quiz application which runs in synchronism with a quiz television program; a magazine browser application; and a weather or traffic application. The user hardware (10) is connected to an application and data service channel (4006) via a switched public telephone network (12). Said application and data service channel (4006) can be connected to the Internet (16) via an interface (14) in a known manner and can communicated with the user hardware (10) via an multiplexer and encoder (2004) a transmitter (2008) a satellite transponder (2014) and a ground receiver (2018).
Patent CZ-292689-B6 (CZ)
Title: Recombinant lectin from dwarf mistletoe
Inventor: LENTZEN HANS
IPC: A61P35/00
Filed: 1996-06-25
Abstract: The present invention relates to nucleic acid molecules encoding preproteins, which after ripening exhibit biological activity of dwarf mistletoe lectin  dimers, further to vectors containing such nucleic acid molecules, hosts transformed by these vectors and polypeptides, optionally polypeptide dimers that  are encoded by these nucleic acid molecules. Polypeptides according to the present invention can be used in many therapeutical applications. The invention further relates to immunotoxins as well as medicaments containing the polypeptides optionally polypeptide dimers, as well as diagnostic kits containing the nucleic acid molecules, the polypeptides, optionally polypeptide dimers according to the present invention or primers, which specifically hybridize with the nucleic acid molecule. In the end, it also relates to plant protection compositions containing the polypeptides optionally polypeptide dimers of said polypeptides.
Patent SK-282134-B6 (SK)
Title: Oxazolidin derivative, method for its preparation and pharmaceutical preparation containing it and use
Inventor: GANTE JOACHIM
IPC: A61P9/08
Filed: 1994-09-19
Abstract: Novel oxazolidinone derivatives of the formula I <IMAGE>  wherein   R<1> is a phenyl radical which is unsubstituted or substituted once by CN, H2N-CH2-, A2N-CH2-, H2N-C(=NH)-, H2N-C(=NH)-NH-, H2N-C(=NH)-NH-CH2-, HO-NH-C(=NH)- or HO-NH-C(=NH)-NH-,   X is O, S, SO, SO2, -NH- or -NA-,   B is <IMAGE>     A is alkyl having 1 to 6 C atoms,   R<2> is H, A, Li, Na, K, NH4 or benzyl,   R<3> is H or (CH2)n-COOR<2>,   E in each case independently of one another is CH or N,   Q is O, S or NH,   m is 1, 2 or 3 and   n is 0, 1, 2 or 3, and their physiologically acceptable salts inhibit the binding of fibrinogen to the corresponding receptor and can be used for the treatment of thromboses, apoplexy, cardiac infarct, inflammations, arteriosclerosis, osteoporosis and tumours.
Patent SK-279344-B6 (SK)
Title: Method and device for panel fulling
Inventor: ZOGG HANS
IPC: B29C67/00
Filed: 1990-07-26
Abstract: In a fulling process, there is at least one panel supported on its upper and lower side in an holding area and then is subjected to fulling on the edge region thereof. The panel is, in the holding area, perpendicularly pressed up to 10 percent of its thickness and is prevented, in the fulling area, from buckling. Fulling is processed in particular phases by application of multiplied strokes of a fulling tool. The number of strokes in the first phase is 20 percent higher than in the second one. From 40 to 45 strokes altogether is applied during the fulling process. Preliminary fulling is carried out over a depth of approximately 6 to 8 and the second fulling up to 11 centimetres. The fulling device consists of at least one fulling tool and a device for securing and moving the mineral fibre panel (11). This device is arranged in the holding area above and below the panel (11) and contains belts (13, 15). The fulling unit, comprising fulling tools (29, 30) used for pre-fulling and panel (11) fulling in the fulling region (23) that is situated by the holding area, is directed transversely to a direction of the panel (11) movement. Above and below the fulling region (23), there are guides (25, 27) with reinforcement (26, 28). The fulling device (29, 30) has a stamp (32) with a convex surface (31).
Patent CZ-295660-B6 (CZ)
Title: Demonstration device modeling a living organism
Inventor: WEINSPACH PAUL-MICHAEL
IPC: G09B23/30
Filed: 1998-09-10
Abstract: The present invention relates to a demonstration device (401), which is a model of a living organism magnified by at least 50 times. Demonstration devices of this type, for example a model of a person lying down, help to explain and to show how the biological processes, which take place in the living organism, are related. The inventive demonstration device (401) has an outer skin (10) and it its interior functional elements (11) representing the organism's organs, vascular system, joints, etc. According to the invention, it is possible to both walk and travel in the demonstration device and its functional elements.
Patent SK-287365-B6 (SK)
Title: Aqueous pesticidal suspension
Inventor: WARRINGTON ROGER PAUL
IPC: A01N25/00
Filed: 2001-08-21
Abstract: Aqueous pesticidal suspensions comprise: (a) 5 to 40 % w/v of (i) a pesticide having a melting point in the range of from 50 to 120 DEG C and a solubility in water of not more than 0.2 % w/v or (ii) a mixture of the pesticide (i) and one or more other pesticides having a melting point of at least 50 DEG C and a solubility in water of not more than 0.2 % w/v in the ratio of at least 1 part by weight of the pesticide (i) to 10 parts by weight of the other pesticide or pesticides, (b) 2.5 to 20 % w/v of a non-ionic alkoxylate surfactant, (c) 0.5 to 5 % w/v of a naphtalene sulphonate-formaldehyde condensate, (d) 0.1 to 5 % w/v of a non-ionic polymethyl methacrylate-polyethylene oxide graft copolymer, (e) 0 to 25 % w/v of other additives, and (f) water in sufficient amount to bring the total composition to 100 % w/v. Pesticidal suspensions formulated in this way show less variation in viscosity.
Patent SK-287012-B6 (SK)
Title: Pharmaceutical composition comprising cyclopeptide, use of the composition or cyclopeptide for the preparation of a medicament and set containing thereof
Inventor: JONCZYK ALFRED
IPC: A61K38/00
Filed: 1999-09-09
Abstract: A pharmaceutical composition comprising cyclo(Arg-Gly-Asp-D- Phe-NMe-Val) and/or its physiologically acceptable salt, and/or angiogenesis inhibitor, and/or its physiologically acceptable salt, wherein a chemotherapeutic agent is selected from the group consisting of a) alkylating agents, b)antibiotics, c) anti metabolites, d) biologika and immune modulators, e) hormones and their antagonists, f) 2,2`-dichloro-diethyl sulphide, g) alkaloids and h) other agents. Use of the pharmaceutical composition or cyclopeptide for the preparation of a medicament for treatment of pathological angiogenic diseases, thromboses, myocardial infarction, coronary heart diseases, arteriosclerosis, tumors, inflammations and infections. Set consists of a) an effective amount of the cyclopeptide and b) an effective amount of the chemotherapeutic agent.
Patent SK-286708-B6 (SK)
Title: Ortho-substituted and meta-substituted bis-aryl compounds, method for the production thereof, their use as a medicament, and pharmaceutical preparations containing these compounds
Inventor: PEUKERT STEFAN
IPC: A61K31/4406
Filed: 2001-11-17
Abstract: The invention relates to ortho- and meta-substituted bis-aryl compounds of formula (I) and to pharmaceutical preparations containing these compounds. These compounds are especially well-suited for use as antiarrhythmic active substances, in particular, for the treatment and prophylaxis of atrial arrhythmias, e. g. atrial fibrillations and atrial flutters.
Patent SK-283904-B6 (SK)
Title: Heterocyclic compounds for inhibition of gastric acid secretion, processes for their preparation and pharmaceutical compositions thereof
Inventor: AMIN KOSRAT
IPC: C07D471/04
Filed: 1998-11-18
Abstract: The present invention relates to heterocyclic compounds of formula (I), in which the phenyl moiety is substituted with lower alkyl in 2- and 6-position, which inhibit exogenously or endogenously stimulated gastric acid secretion and thus can be used in the prevention and treatment of gastrointestinal inflammatory diseases.
Patent CZ-302056-B6 (CZ)
Title: Method for making a puffed food starch product
Inventor: MALFAIT JACQUE L
IPC: A23P30/38
Filed: 2000-07-03
Abstract: In the present invention, there is disclosed a method of making a puffed food starch material product from a bulk amount of food starch material, the method comprising the steps of: providing a puffing chamber having inner surfaces and a chamber volume; placing a bulk amount of the food starch material into the puffing chamber having inner surfaces and a chamber volume; causing a volumetric expansion of the bulk amount of food starch material; and constraining expansion of the bulk amount in at least a first dimension, while permitting unlimited expansion of the bulk amount in at least a second dimension. The present invention also discloses an apparatus for carrying out the above-describe method as well as a puffed food starch product prepared in the above-indicated manner.
Patent CZ-302196-B6 (CZ)
Title: Stable oxaliplatin solution formulation, use of oxaliplatin when obtaining the formulation, method for stabilizing an oxaliplatin aqueous solution, process for preparing the formulation and packaged pharmaceutical composition
Inventor: ANDERSON NICHOLAS HUGH
IPC: A61K33/243
Filed: 1999-02-25
Abstract: The present invention relates to a stable oxaliplatin solution formulation comprising a therapeutically effective amount of oxaliplatin, an effective stabilizing amount of a buffering agent being represented by oxalic acid or an alkali metal salt thereof, and a pharmaceutically acceptable carrier being represented by water. The invention also relates to the use of oxaliplatin when obtaining the above specified formulation in the treatment of cancer tumors, to a method for stabilizing an aqueous solution of oxaliplatin by adding an effective stabilizing amount of a buffering agent to said solution wherein the buffering agent is oxalic acid or an alkali metal salt thereof and to a process for the preparation of such formulation.
Patent CZ-305033-B6 (CZ)
Title: Pharmaceutical composition and its use as inhalation solution
Inventor: DRECHSEL KARIN
IPC: C07D451/02
Filed: 2001-10-24
Abstract: The present invention relates to a liquid, propellant-free pharmaceutical composition comprising at least two combinable active substances containing a tiotropium salt as one of the at least two active substances, in a concentration based on tiotropium of between 0.0005 and 5 percent by weight, a steroid, an antiallergic, an antihistamine, or a leukotriene antagonist as the second of the at least two active substances, and water as a solvent, in which at least the tiotropium salt is dissolved, an acid for achieving a pH between 2.0 and 3.5, a pharmacologically acceptable preservative, and an edetic acid salt in an amount of up to 10 mg/100 ml. The above-described pharmaceutical composition further comprises one or more of a stabilizer, a pharmacologically acceptable co-solvent, a further pharmacologically acceptable adjuvant, and a pharmacologically acceptable additive in addition to the preservative. The invention also relates to the use of the pharmaceutical composition in an inhaler for providing propellant-free aerosols for spraying a defined amount of the pharmaceutical composition through a nozzle at high pressures in order to generate inhalable aerosols.
Patent CZ-293468-B6 (CZ)
Title: Device for locking the end positions of moving points components
Inventor: SCHNEDL KARL SCHNEDL KARL
IPC: B61L5/10
Filed: 2002-01-11
Abstract: The present invention relates to a device for locking the end positions of moving points components, in particular the moving tip (1) of a frog, whereby two pieces, axially displaceable relative to each other, may be moved in at least one displacement direction into a position coupled to each other in an interlocking manner. The pieces that move relative to each other are formed from a tube (5) and a rod (6), running in the tube (5) and are at least partly arranged in a fixed outer tube (4). Locking members (8) co-operate with the pieces (5, 6), which move axially relative to each other and the outer tube (4) and may be moved in the radial direction into a locking position in a recess, or inner annular groove (15, 16), on the outer tube (4). Said device is embodied such that the outer tube (4) comprises two tube pieces (17, 18) which can move axially one within the other and each tube piece (17, 18) comprises at least one recess, optionally an inner annular groove (15, 16).
Patent EP-1272531-B8 (EP)
Inventor: PITHA JOSEF
IPC: A61K31/715
Filed: 2000-11-09
Granted: 2007-02-14
Abstract: Certain mixtures of cyclodextrin derivatives, which were synthesized in mildly basic conditions, can be separated into mixtures that crystallize easily and mixtures of similar composition, which remain amorphous. Thus, it is possible to obtain the particular advantages of crystalline and/or amorphous state components from one reaction product. Both crystalline and amorphous components of the product have good ability to form inclusion complexes.
Patent EP-1456670-B8 (EP)
Inventor: PETYAEV IVAN
IPC: A61K35/66
Filed: 2002-08-22
Granted: 2011-04-27
Abstract: The present invention relates to the identification of lipid oxidising abzymes as a key pathogenic factor in atherosclerotic disorders. Methods and means for the reduction of abzyme mediated lipid oxidation in the vascular system are provided as therapeutic approaches for the treatment of atherosclerotic disorders.
Patent BR-PI0711772-B8 (BR)
Title: método para combater ou controlar insetos, aracnídeos ou nematódeos; método para proteger colheitas e plantas em crescimento do ataque ou infestação de insetos, aracnídeos ou nematódeos; e método para proteger sementes dos insetos de solo e raízes e rebentos das mudas dos insetos de solo; composto e composição agricultural ou veterinária
Inventor: DEBORAH L CULBERTSON
IPC: A01P7/00
Filed: 2007-05-15
Abstract: métodos para combater ou controlar insetos, aracnídeos ou nematódeos, para proteger colheitas e plantas em crescimento do ataque ou infestação de insetos, aracnídeos ou nematódeos, para proteger sementes dos insetos de solo e raízes e rebentos das mudas dos insetos de solo e foliares, e para tratar, controlar, evitar ou proteger animais contra infestação ou infecção por parasitas, composto, composição agricultural ou veterinária, e, semente. a presente invenção refere-se a novos métodos inseticidas de utilizar compostos de 4-arnino-5 -cloro-tieno [2,3 -d] -pirimidina de fórmula (i), em que r^1^, r^2^, r^3^ e a são definidos corno no relatório. a presente invenção refere-se a métodos inseticidas de aplicação de tais compostos de fórmula (i), e a novos derivados de compostos de fórmula (i).
Patent BR-PI0722361-B8 (BR)
Title: métodos para avaliar a concentração de um fármaco imunossupressor em uma amostra de sangue humano, composição de reagente de extração e kit de teste
Inventor: FRANK C GRENIER
IPC: G01N33/53
Filed: 2007-12-19
Abstract: reagente de extração de fármaco imunossupressor para imunoensaios uma composição melhorada de reagente extrativo e método para extrair um fármaco imussupressor, tal como sirolimus, tacrolimus ou ciclosporina, de amostras de sangue ao mesmo tempo em que produz um extrato de amostra de teste que tenha baixa pressão de vapor e que seja compatível com componentes de imunoensaio. a composição inventiva de reagente compreende sulfóxido de dimetila (dmso), pelo menos um sal de metal divalente e água. os extratos das amostras resultantes do uso de cada uma destas combinações têm baixa pressão de vapor e são compatíveis com os ensaios imunoquímicos.
Patent BR-PI0910756-B8 (BR)
Title: distribuidor de turbina para uma turbomáquina, turbina de baixa pressão de turbomáquina e turbomáquina, tal como um turborreator ou um turbopropulsor de avião
Inventor: Bruno marie benjamin jacques richard
IPC: F01D9/04
Filed: 2009-04-17
Abstract: distribuidor de turbina para uma turbomáquina, setor de distribuidor e suporte anular contínuo para um distribuidor, turbina de baixa pressão de turbomáquina e turbomáquina, tal como um turborreator ou um turbopropulsor de avião. distribuidor (112) de turbina para uma turbomáquina, que compreende duas plataformas anulares coaxiais ligadas entre si por pás radiais, a plataforma interna (130) sendo ligada a uma divisória anular (138) recortada ou dentada na qual é afixado uni suporte anular (140) que leva elementos (136) feitos de material abrasivo, esse suporte podendo deslizar circunferencialmente sobre a divisória entre unia posição de montagem/desmontagem e uma posição de bloqueio do suporte sobre a divisória.
Patent BR-PI1009315-B8 (BR)
Title: composto anti-flamatórios e suas composições farmacêuticas
Inventor: C HENRIK HANSEN
IPC: C07D403/10
Filed: 2010-03-16
Abstract: agentes anti-inflamatórios. a invenção refre-se a compostos que são úteis na regulação da expressão de interleucina-6 (il-6) e/ou molécula de adesão celular vascular-1 (vcam-1), e seu uso no tratamento e/ou prevenção de doenças cardiovasculares e inflamatórias e estados de doença relacionados, tal como, por exemplo, aterosclerose, asma, artrite, câncer, esclerose múltipla, psoríase, e doenças do inntestino inflamatórias, e doença(s) autoimune(s). além diss, são descritas composições compreendendo os novos compostos, bem como métodos para sua preparação.