baber/WOPTO huggingface dataset:
Patent IL-138563-A0 (IL)
Title: Novel cephalotaxane derivatives and process for their preparation
IPC: C07C69/732
Filed: 1999-03-17
Abstract: The present invention concerns a new general process for asymmetric hemisynthesis of harringtonines and their analogs, that are alkaloids used in chemotherapy. This process comprises direct esterification of a natural cephalotaxine with an acylating compound constituted of a side chain precursor which backbone and functionalization are entirely preformed. The invention also concerns a natural, synthetic or semi-synthetic harringtonines including their tautomeric forms and their salts of the following formula: wherein n=2 (i.e. harringtonine) or n=3 (i.e. homoharringtonine), in which the total content of impurities, possibly including enantiomeric forms, is lower than 1%, and/or the content of the major impurity is lower than 0.9%, and/or the chromatographic assay exhibits a harringtonines content higher than 97.5%.
Patent IL-144229-A0 (IL)
Title: Novel 2-(n-cyanoimion) thiazolidin-4-one derivatives
IPC: C07D417/12
Filed: 1999-11-12
Abstract: This invention provides novel 2-(N-cyanoimino)thiazolidin-4-one derivatives represented by formula I or a pharmaceutically acceptable salt or solvate thereof: <CHEM> wherein ring A represents a benzene ring, a condensed ring or a heterocyclic ring, each of which may be substituted by one or more substituents selected from a straight or branched C1 - C4 alkyl group, a haloalkyl group, a halogen atom or -OR<5>,   R<1> represents a single bond, an oxygen atom, a sulfur atom, a methyne group, a straight or branched C1 - C4 alkylene or alkenylene group optionally substituted by a phenyl group, R<6>-X X-R<6>, X-R<6>-X R<6>-X-R<6>, -C(=O)-NR<7>- or -NR<7>-C(=O)-, R<2> and R<3> are the same or different and each represents a hydrogen atom, a C1 - C4 alkyl group, -OR<8> or a halogen atom,   R<4> represents a hydrogen atom or a C1 - C4 alkyl group,   R<5> represents a hydrogen atom or a C1 - C4 alkyl group, R<6> represents a straight or branched C1 - C4 alkylene or alkenylene group,   R<7> represents a hydrogen atom or a C1 - C4 alkyl group, R<8> represents a hydrogen atom, a C1 - C4 alkyl group or an aralkyl group,   X represents an oxygen atom or a sulfur atom.   They have excellent activities of lowering triglyceride and cholesterol levels, and are useful for preventing from and/or treating hyperlipidemia and related complications.
Patent IL-144681-A0 (IL)
Title: Method and device for executing method steps
IPC: B41F33/00
Filed: 2001-08-01
Abstract: The method employs a master computer exercising overall control of a first device and of a number of sub-systems representing the process steps. The master computer has two way communication with slave computers controlling the sub-systems through which it monitors the current control state of those systems to prevent commands being executed unless the correct conditions prevail.
Patent IL-148150-A0 (IL)
Title: Method for the qualitative improvement of the products of the tobacco plant
IPC: A24B15/22
Filed: 2000-03-07
Abstract: The method belongs to the field of electronic science and is applied to the field of the manufacture of products deriving from the tobacco plant, such as cigarettes, cigars, pipe tobacco, tobacco in general, and achieves their qualitative improvement. The qualitative improvement is achieved with the pulsatory emission of electromagnetic waves (6) towards the tobacco products, which are produced by electromechanical or electronic devices (3), are pre-programmed, cover wide ranges of wavelengths from 1 mm to 11,000 Km, together with their harmonic frequencies, which are produced by the device and which are emitted either at all wavelengths from 1 mm to 11,000 Km, or at one or more parts of particular areas, with controlled potency, controlled application time and controlled application result. It is applied in industries, manufacturing and commercial enterprises of final or not tobacco products, which are either at the processing stage, or after the completion of their manufacture, or during their storage, regardless of the way or the materials they are packaged with. <IMAGE>
Patent IL-150349-A0 (IL)
Title: Rapid onset formulation
IPC: A61K9/28
Filed: 2001-06-21
Abstract: A new enterically-coated pyridoxine HCl and doxylamine succinate (DS-P) rapid onset formulation comprises disintegrating agent. The formulation has a dissolution profile of at least 40%, 70%, 80% and 90% after 30, 60, 90 and 120 minutes respectively when measured in 1000 ml phosphate buffer at pH 6.8 and 37[deg]C in a type 2 dissolution apparatus at 100 revolutions per minute (rpm). ACTIVITY : Antiemetic. No biological data given. MECHANISM OF ACTION : None given.
Patent IL-152225-A0 (IL)
Title: A process for the preparation of decahydro-2a,4a,6a,8a-tetraazacyclopent [fg] acenaphthylene and functionalized derivatives
IPC: C07D487/22
Filed: 2001-04-10
Abstract: A process for the preparation of compound of formula (I A), decahydro-2a,4a,6a,8a-tetraazacyclopent[fg]accnaphthylene and the corresponding functionalized compounds of general formula (I), intermediates for the preparation of 1,4,7,10-tetraazacyclododecane (II A) and corresponding derivatives (II), by preparation of compounds of general formula (III) and subsequent reduction thereof.
Patent IL-152852-A0 (IL)
Title: Edge lit illumination devices
IPC: F21Y103/00
Filed: 2001-05-04
Abstract: An edge lit illumination device is described. The device has at least one light source and a light transmission element having at least one light output surface and at least one light ingress edge substantially perpendicular to said surface. The light source is located adjacent to the light ingress edge so that light from the light source enters the transmission element via the said edge and propagates through the element. The light output surface is uniformly roughened across the output surface. The roughening is sufficiently fine to give an average Ra value across the surface of less than 1.0 mum/mm thickness of the element or drop-off of light output across the surface of less than 5000 lux.
Patent IL-154844-A0 (IL)
Title: Composition, method and device for pressuring a fuel tank
IPC: F02K9/50
Filed: 2001-09-21
Abstract: The invention concerns a composition for pressurising a fuel tank. It also concerns the use of said composition for pressurising a fuel tank, a method for supplying a propulsion system with fuel by pressurising said fuel contained in a tank using said composition, and a feed tank for implementing said method. The composition for pressurising a tank supplying a propulsion system with fuel is characterised in that said composition consists of a system having a saturating vapour pressure higher than about 5 x 10<5> to 22 x 10<5> Pa at a temperature of 10 to 50  DEG C partly in liquid form.
Patent IL-161181-A0 (IL)
Title: Therapeutically useful triethyleneglycol cholesteryl oligonucleotides
IPC: A61K45/00
Filed: 2002-10-03
Abstract: The present invention provides a composition comprising a 5'-OH, 3'-TEG cholesteryl synthetic sequence wherein the sequence is SEQ ID NO:5, SEQ ID NO:6, SEQ ID NO:7, SEQ ID NO:8. The present invention provides methods of using this composition for induction of response in a cell, including but not limited to inhibition of cellular proliferation, induction of cell cycle arrest, induction of caspase activation, cleavage of poly(ADP-ribose) polymerase, induction of apoptosis or modulation of extracellular matrix-cell interactions, or combinations thereof, in cancer cells or synovial cells, and methods of using this composition for treating disease.
Patent IL-176155-A0 (IL)
Title: Polycyclic agents for the treatment of respiratory syncytial virus infections
IPC: A61K31/4188
Filed: 2006-06-06
Abstract: Compounds of formula I   
salts, and pharmaceutically acceptable derivatives thereof, wherein: A, together with the atoms to which it is attached, represents an optionally substituted phenyl ring; B-C is an optionally substituted link of the formula -CH 2 -(CH 2 ) z -, where z is 1-4; X and Y are independently selected from O, S and NR 6 , where R 6  is independently selected from hydrogen, C 1-6 alkyl, hydroxy and C 1-6 alkoxy; and R 1  and R 2 ;are as defined herein; are described. The compounds are useful as antiviral agents in particular the treatment of infections involving viruses of the  Pneumovirinae  subfamily.
Patent IL-182534-A0 (IL)
Title: Method of executing handover in broadband wireless access system
IPC: H04W36/14
Filed: 2007-04-12
Abstract: The primitives between an upper management layer and the MAC layer within a mobile station and a base station are defined in order to specify and clarify the operations within the protocol stack layers in a broadband wireless access system to allow a mobile station to execute handover. Media Independent Handover (MIH) procedures can be achieved because the NCMS and MIH layer can communicate through use of these primitives.
Patent IL-185758-A0 (IL)
Title: Process for the production of monoliths by means of the sol-gel process
Filed: 2007-09-06
Abstract: Process for the production of monoliths by means of the sol-gel process, comprising the following steps:  a. hydrolysis of an alkoxide in aqueous solution to form a hydrolysate and optionally evaporation to optimum concentration of the same,  b. addition of an oxide prepared by the pyrogenic route,  c. mixing of the hydrolysate of the alkoxide with the oxide prepared by the pyrogenic route to form a colloidal sol,  d. optional removal of coarse contents from the colloidal sol,  e. gelling of the colloidal sol in a mould,  f. optional replacement of the water contained in the resulting aerogel by an organic solvent,  g. drying of the aerogel,  h. heat treatment of the dried aerogel, the coarse content being removed from the colloidal sol.
Patent RO-125879-A0 (RO)
Title: Kit for driving skills training, testing and checking in real time
Inventor: CATANĂ EUSEBIU
IPC: G09B9/04
Filed: 2010-07-16
Abstract: The invention relates to a kit for driving skills training, testing and checking in real time. According to the invention, the kit is meant to be mounted on a vehicle and comprises a system of sensors (A) to detect motion and measure some parameters, comprising some sensors (1 and 2) mounted on the vehicle accelerator control pedal and brake control pedal, respectively, a pressure sensor (3) adapted to the braking system for measuring braking force and momentum, a speed counter (4) located within the driving system of the vehicle, a rotation sensor (5) located on the steering wheel and meant to determine the running direction, a speed sensor (6) as well as three sensors (7, 8 and 9) for determining longitudinal, lateral and vertical vehicle movement and two video cameras (10 and 11) for viewing the path and the vehicle driver, respectively, all those elements resulting in the real-time determination of the driving manner, driver's response as signals integrated in a data acquisition board (B) connected to a computer (C) where there takes place the real-time processing by means of a specialized software and display of results.
Patent RO-127180-A0 (RO)
Title: Mould and process for carrying out the same
Inventor: IVĂNESCU SEBASTIAN MIHAIL
IPC: B29D15/00
Filed: 2011-11-09
Abstract: The invention relates to an open mould meant to manufacture small- or mid-scale unique parts of epoxy or polyester resins for the motor vehicle industry, such as hoods, and to a process for applying the same. According to the invention, the mould consists of a base plate () made of oriented wood fibres, an extruded polystyrene block (), a layer () of epoxy resin, two layers () of fibre glass fabric impregnated with epoxy resin, some resistors (), an epoxy resin layer () of controlled thickness and a gelcoat layer (). According to the invention, the process for carrying out the mould consists in assembling a block () by adhering with epoxy resin some semifinished products of expanded polystyrene, adhering a block () resulting on the base plate () of oriented wood fibres with epoxy resin, milling the upper surface of the block () according to the pattern of the part to be manufactured by the mould, applying onto the milled surface a layer () of epoxy resin, applying two layers () of glass fibre fabric impregnated with epoxy resin onto the layer (), fixing some electric resistors () on the layers (), applying a layer () of epoxy resin of controlled thickness embedding the electric resistors () onto the layers (), milling the layer () to the shape and dimensions of the part to be manufactured by the mould, applying a gelcoat layer () onto the layer () of epoxy resin and polishing the gelcoat layer ().
Patent IE-910297-A1 (IE)
Title: Optical fibre telecommunications line with separate service channels
Inventor: GRASSO GIORGIO
IPC: H04B10/29
Filed: 1991-01-29
Abstract: The invention refers to an optical fibre transmission line which comprises means (9, 10) for injecting and means (9, 10) for extracting optical service signals from the line' s optical fibre (3), where said means comprise emission and/or reception units (10) of optical service signals, suitable for receiving from the optical line (3) and/or emitting towards the line itself service signals in the form of optical signals having a wavelength which is substantially different from the wavelength of the telecommunications signals, each of which units (10) is associated with a corresponding optical coupler (9) inserted along the line (3), suitable for coupling within the line fibre and/or for extracting from it the optical service signals.
Patent MA-19404-A1 (MA)
Inventor: ADOLPHE MARIE DOUWES
IPC: C07C239/00
Filed: 1982-03-05
Abstract: A process for the preparation of urea at elevated temperatures and pressures in which ammonium carbamate is decomposed into ammonia and carbon dioxide and separated from the urea product stream in at least two pressure stages. The product urea stream having reduced ammonium carbamate content leaving the first high pressure stage is reduced in pressure to a level intermediate the pressure of the high pressure stage and the next pressure stage in a pressure reducing device in which the energy released by the pressure reduction is converted into kinetic energy by means of which a gaseous mixture of ammonia and carbon dioxide resulting from the carbamate decomposition in a further pressure stage or recovered the process condensate formed in a concentrating stage is compressed to the intermediate pressure. The resulting compressed mixture is thereafter condensed, and the condensate thus formed is pumped to the high pressure stage.
Patent MA-23403-A1 (MA)
Inventor: FRISH GERHALD
IPC: A01N25/04
Filed: 1994-12-20
Abstract: PCT No. PCT/EP94/04141 Sec. 371 Date Aug. 29, 1996 Sec. 102(e) Date Aug. 29, 1996 PCT Filed Dec. 14, 1994 PCT Pub. No. WO95/17087 PCT Pub. Date Jun. 29, 1995The present invention relates to oil-in-water emulsions containing 0.001-70% by weight of at least one active substance from the group consisting of phosphates, thiophosphates and/or carbamates, 0.001-30% by weight of one or more surfactant compounds from the group consisting of nonionic surfactant compounds or phosphorylated surfactant compounds or sulfated surfactant compounds or sulfonated surfactant compounds, and also, if desired, adjuvants, and, water to make up 100% by weight.
Patent MA-37172-A1 (MA)
Title: Champs de concentrations solaires à héliostats –adaptation à plusieurs applications : chauffage, solaire climatisation solaire, dessalement
Inventor: BOUKDIR YOUSSEF
IPC: F24S50/20
Filed: 2014-07-01
Abstract: L’invention concerne un système de concentration solaire pour la production d’énergie thermique à l’aide d’une solution complète et autonome (autonome: fonctionnalité automatisée qui permet de collecter l’énergie solaire et de suivre le soleil toute l’année sans une intervention externe).Il s’agit d’un champ de concentrateurs solaire à héliostats de petites échelles (taille dc la surface d'un bâtiment). Cette invention exploite le principe de tracking solaire à deux axes et le principe de concentration solaire dans des petites applications tel que la satisfaction des besoins de l'eau chaude sanitaire dans un bâtiment, l’extraction des huiles essentielles par distillation à la vapeur d'eau, le refroidissement solaire, séchoir solaire, générateur de vapeur etc.
Patent MA-37693-A1 (MA)
Inventor: IVACHTCHENKO ALEXANDRE VASILIEVICH
IPC: A61K31/137
Filed: 2013-07-05
Abstract: يتعلق الاختراع بمجال المستحضرات الصيدلانية, على وجه الخصوص, إلى تركيب صيدلي صلب يحتوي 2—امينو—2—[2—(4—اوكتيل فينيل)اثيل] بروبان—1 ,3—دايول او ملحه المقبول صيدليا, مثبت, مادة حشوة, و بطريقة لتحضير التركيب الصيدلي, و بأدوية لتثبيط المناعة و المعالجة التصلب المتعدد. يمثل 2—امينو—2—[2—(4—اوكتيل فينيل)اثيل] بروبان—1 ,3—دايول مغير مناعي الدي يسبب اعادة توزيع الخلايا اللمفاوية من مجرى الدم إلى الانسجة اللمفاوية الثانوية التي تؤدي إلى تثبيط المناعة. و طرح الاختراع توزيع موحد و متجانس للمعامل الفعال في تركيب الصلب, قابلية ثبات عالية و سيولة محسنة للتركيب الصيدلي الصلب. نظرا لسيولتها محسنة يمكن استخدام التركيب المقترحة في الاختراع في المعادات الالية.
Patent MA-38430-A1 (MA)
Title: Compositions pharmaceutiques comprenant de l'évérolimus
Inventor: DIEDERICH ANKE
IPC: A61K31/00
Filed: 2014-03-19
Abstract: La présente invention concerne une formulation pharmaceutique comprenant de la 40-o-(2-hydroxy)éthyl-rapamycine dans une partie à charge de médicament élevée et une partie à libération immédiate. De plus, l'invention concerne une formulation comprenant de la 40-o-(2-hydroxy)éthyl-rapamycine dans une première couche et un tensioactif dans une couche au-dessous de la première couche. La composition pharmaceutique est particulièrement adaptée pour utilisation en tant que médicament.
Patent UY-23556-A1 (UY)
Title: Metodo para la extraccion de esencia de vainas de vainilla
IPC: C11B9/00
Filed: 1993-03-25
Abstract: La presente invención se refiere a un método para la extracción de esencia de vainas de vainilla que consiste en someter el material de vainilla sin curar a un tratamiento enzimático en un medio acuoso, separando opcionalmente el material sólido de la vaina y recuperando el material de la esencia con un solvente orgánico, tratamiento enzimático que incluye la incubación con una glucosidasa y una proteasa. Preferentemente, el proceso se realiza en un medio acuoso que contiene por cada 100 partes (peso seco) de vainas entre 200 y 5000 partes en peso de agua.
Patent UY-26085-A1 (UY)
Title: N-[-(4-aminofenil)-2,3-dihidro-1,4-benzodioxina-2-metanamina su preparacion y su aplicacion en terapeutica
Inventor: EVANNO ANTONIO ALMARIO GARCIA
IPC: A61P25/22
Filed: 2000-03-29
Abstract: Compuestos de fórmula general I.Aplicación en terapéutica.
Patent UY-31607-A1 (UY)
Title: Derivados bicíclicos de carboxamidas aza-bicíclicas, su preparación y su aplicación terapéutica
Inventor: CATHERINE GILLE
IPC: A61K31/404
Filed: 2009-01-22
Abstract: La invención se refiere a derivados bicíclicos de carboxamidas aza-bicíclicas de fórmula general (I) en forma de base o de sal de adición de ácido, así como en forma de hidrato o de solvato, en la que los sustituyentes e índices son tales como se especifican en la memoria descriptiva y en las reivindicaciones. Se divulgan también los procedimiento de preparación y aplicación en terapéutica en las patologías donde que están implicados los receptores de tipo TRPV1
Patent ZW-12684-A1 (ZW)
Title: Externalization of products of bacteria
Inventor: MARTIN ROSENBERG
IPC: C12N15/73
Filed: 1984-08-08
Abstract: A bacterial product is made by transforming a temperature sensitive lysogen with a DNA molecule which codes, directly or indirectly, for the product, culturing the transformant under permissive conditions and externalizing the product by raising the temperature to induce phage encoded functions.
Patent ES-173819-A1 (ES)
Title: PROCEDIMIENTO PARA LA APLICACIoN DE COLORANTES DESTINABLES A MATERIALES TEXTILES EN FORMA DE MECHAS O PAQUETES
Filed: 1946-05-31
Abstract: Procedimiento para la aplicación de colorantes tinables a materiales textiles en forma de mechas o paquetes, caracterizándose porque se hace circular a través del paquete o mecha una suspensión de un colorante tinable no reducido que contiene un agente de dispersión disuelto en él; añadiéndose gradualmente a la suspensión una cantidad suficiente de una sal inorgánica acuosoluble para dar lugar a la deposición prácticamente completa del colorante de la suspensión en el material del paquete, y después reducir y subsiguientemente oxidar el colorante tinable por cualquier método usual.
Patent ES-174266-A1 (ES)
Title: Mejoras en la manufactura de empaquetaduras.
Filed: 1946-07-11
Abstract: Mejoras introducidas en la manufactura de empaquetaduras caracterizadas porque entre la empaquetadura del recipiente y la del cojinete de un árbol que conduce a un recipiente se deja por lo menos una cámara hueca en la cual reine una presión menor que la del recipiente y del cojinete y porque el árbol tanto en la cámara de cojinete como en la intermedia está provisto de anillos centrifugadores que rechazan del árbol los líquidos a sus vapores.
Patent ES-179401-A1 (ES)
Title: FUNCIONAMIENTOS EN LOS DISPOSITIVOS INDICADORES DE CAMBIOS EN LOS FACTORES FiSICOS
Filed: 1947-08-20
Abstract: Perfeccionamientos en los dispositivos indicadores de cambios en los factores físicos, que incluyen un método para indicar una variación apreciable en un factor físico con la que está relacionada una variación apreciable del valor de la constante dieléctrica, en una tira de material que se precisa tenga una variación despreciable de dicho factor físico en toda su longitud, que comprende las etapas de hacer pasar la tira, o una sección longitudinal escogida de la misma, entre las placas de un condensador de prueba, de utilizar el cambio en la capacidad del condensador de prueba resultante de la variación apreciable del valor de la constante dieléctrica del material de la tira que lo atraviesa para influenciar el funcionamiento de un circuito de control electrónico, y de aprovechar una variación resultante en dicho circuito de control electrónico para dar lugar al funcionamiento de medios indicadores adecuados.
Patent ES-188132-A1 (ES)
Title: SISTEMA RECTIFICADOR ELECTROMECáNICO
Filed: 1949-05-07
Abstract: Sistema de rectificador electromecánico caracterizado por un circuito en el que se establecen una o más válvulas de las características de la reivindicada en la solicitud de patente nº 188.106 accionadas por un motor sincronizado y la disposición del filtraje que consiste en un condensador y una impedancia que a la salida de la válvula tienen por objeto uniformar la corriente contínua pulsatoria que se obtiene en la rectificación para utilizarla en el aparato consumidor.
Patent ES-193913-A1 (ES)
Title: UN PROCEDIMIENTO DE PRODUCCIoN DE CEMENTO METALuRGICO
Filed: 1950-07-14
Abstract: Un procedimiento para la producción de cemento metalúrgico en el cual escoria granulada de alto horno se tritura por vía húmeda en ausencia de catalizador que pueda provocar el fraguado para formar una pasta que luego se seca; caracterizado porque se reduce lo bastante el contenido de agua de la pasta por ejemplo quitando el agua en exceso de 20% aproximadamente para obtener una pasta consistente propia para moldearla se forman ladrillos u objetos análogos de esta pasta consistente se dejan secar los ladrillos o similares hasta la reducción suficiente de su contenido de agua por ejemplo hasta un 5% aproximadamente o menos y después la pulverización de los ladrillos o análogos puede hacerse en cualquier momento deseado.