baber/WOPTO huggingface dataset:
Patent SI-2178858-T1 (SI)
Title: Novel heterocyclic compounds as mglu5 antagonists
Inventor: LEONARDI AMEDEO
IPC: A61K31/00
Filed: 2008-08-01
Abstract: This invention relates to novel heterocyclic compounds having selective affinity for the mGlu5 subtype of metabotropic receptors, pharmaceutical compositions thereof and uses for such compounds and compositions in the treatment of lower urinary tract disorders, such as neuromuscular dysfunction of the lower urinary tract, and in the treatment of migraine and gastroesophagael reflux disease (GERD).
Patent SI-3083655-T1 (SI)
Title: A process for the production of 19-norpregn-4-en-3,20-dione-17.alpha.-ol (gestonorone) and intermediates therefor.
Inventor: CSORGEI JANOS
IPC: C07J51/00
Filed: 2014-12-15
Abstract: The present invention relates to a new stereoselective process for the synthesis of 17(α)-17-acetyl-17-hydroxy-estr-4-en-3-one of formula (I), as well as to the new intermediates of the process. The 17(α)-17-acetyl-17-hy droxy-estr-4-en-3 -one (gestonorone) is an important intermediate in the synthesis of the active ingredients having progestogen activity - such as gestonorone capronate and nomegestroi acetate. Formulas (I), (II) and (III).
Patent TR-200101873-T1 (TR)
Title: Termoplastik reineler iin darbe snmleyici.
Inventor: TAKAKI AKIRA
IPC: C08L27/06
Filed: 2000-10-18
Abstract: Bir vinil klorür reçineye uygulanabilecek mükemmel darbe sönümleyici bulunmuçtur. Bu mükemmel darbe sönümleyici olarak, aG rl kça %60 ila %100 oran nda bir (met) akrilat bileçiGi, bir aromatik vinil bileçiGi, bir vinil siyanür bileçiGi ve vinil klorürden oluçan gruptan seçilen en az bir vinil monomerin, monomerin aG rl kça %10 ile %70'inin ve aG rl kça %0 ila %40 oran nda, bu monomerle kopolimerize edilebilecek bir baçka monomerin, cam geçiç  s s  Tg en çok 0°C ve lateks halde boçluk oran  %3 ila %90 olan ve aG rl kça 100 k s m toplam kauçuk bileçeni monomeri baz nda 0.1 ila 5 k s m miktarda bir çapraz baGlant  maddesi içeren, aG rl kça %30 ila %90 gözenekli kauçuk parçac G  varl G nda polimerize edilmesi suretiyle haz rlanan bir kopolimer kullan lmaktad r.
Patent TR-201111169-T1 (TR)
Title: Işık çıkartan pürüzlü bir yapıya sahip olan ledi cihazı ve bunun üretim metotları.
Inventor: YEN JUI-KANG
IPC: F21V5/00
Filed: 2010-05-10
Abstract: Bu buluş, ışık çıkartan pürüzlü bir yapıya sahip olan bir ışık yayan diyot cihazı ve bunun üretim metotları ile ilgili olup, içerisinde ışık çıkartan pürüzlü yapı, ve ışık yayan diyotun ışık çıkartma verimliliğini ve homojenliğini arttırmak için mikron ölçeğinde bir pürüzlülüğe sahiptir.
Patent TR-201704471-T1 (TR)
Title: Pankreatin İhtiva Eden İyileştirilmiş Güvenlik Profiline Sahip Bileşimlerin Üretilmesi İçin Prosesler Ve Farmasötik Kullanıma Uygun Bileşimler
Inventor: GEORGE SHLIEOUT
IPC: A61P1/18
Filed: 2015-11-05
Abstract: Katı veya yarı-katı bileşimler, özellikle farmasötik kullanıma yönelik katı oral bileşimler üretmek için, lipaz aktivitesine sahip olan ve bir sürfaktan-bileşen ihtiva eden bir enzim veya enzim-karışımının belirli proses parametrelerinde işlenmesini kapsayan prosesler tarif edilmiştir. Söz konusu prosesler, söz konusu enzimin veya enzim-karışımının istenen biyolojik aktivitelerini, ör. enzimatik aktivitelerini korurken, istenmeyen biyolojik kirlenmenin, ör. viral kirlenmenin azaltılması için uygundurlar. Proses endüstriyel kullanım için uygundur. Ayrıca, lipaz aktivitesine sahip olan bir enzim veya enzim-karışımı, bir sürfaktan-bileşen ve bir polimerik katkı ihtiva eden, opsiyonel olarak diğer yardımcı maddeler ihtiva eden katı veya yarı-katı bileşimler tarif edilmiştir. Söz konusu bileşimler tercihen burada tarif edilen prosesler ile elde edilebilirler. Ayrıca burada tarif edilen katı veya yarı-katı bileşimleri ihtiva eden farmasötik bileşimler tarif edilmiştir.
Patent DE-3586830-T2 (DE)
Inventor: HONJO TASUKU
IPC: C12N15/85
Filed: 1985-04-24
Granted: 1993-04-22
Abstract: A method of linking two or more heterogenes of biologically different origins, their introns being eliminated by the splicing technique using a retrovirus vector and a eucaryotic cell.
Patent DE-3687523-T2 (DE)
Inventor: FIESCHKO C
IPC: C12N1/18
Filed: 1986-08-15
Granted: 1993-05-13
Abstract: A method for culturing yeast capable of expressing an exogenous gene product wherein the yeast is cultured at about 25<o>C in a medium including balanced free amino acids at a concentration between about 20 g/l and about 160 g/l. Alternatively, yeast capable of expressing an exogenous gene product (e.g. the product of a gene introduced by the application of recombinant gene technology) may be introduced into a medium including a total carbon source concentration above but maintained as close to zero as possible, and cultured at about 25<o>C. A medium for fermentation of yeast capable of expressing an exogenous gene product includes balanced free amino acids at a concentration between about 20 g/l and about 160 g/l. The culture medium is preferably saturated with oxygen at least 30% of air saturation.
Patent DE-3751893-T2 (DE)
Inventor: ONO YOSHITAKA
IPC: C12R1/91
Filed: 1987-06-26
Granted: 1997-01-16
Abstract: Rat protein kinase C, recombinant DNA containing DNA sequence coding for rat kinase C, a transformant transformed with a vector containing the above recombinant DNA, and the production method of rat kinase C cultivating the transformant are disclosed. Rat kinase C is useful as reagent for studying cellular signal transduction mechanism, as diagnostic and inspection agent for disease, for example tumor, resulting from the trouble of cellular signal transduction mechanism, and as screening agent for a preventive agent or medicine to the disease.
Patent DE-3780299-T2 (DE)
Inventor: BROWN J
IPC: H02J3/00
Filed: 1987-09-16
Granted: 1993-01-07
Abstract: Described herein is an energy management system in which a central unit provides a series of energy managing signals over a medium, such as TV cables, power lines, telephone lines or free space radio frequency transmissions, to a plurality of subscriber units. Within each unit is a transponder which responds to the transmitted central unit signals and provides corresponding signals onto an electric grid, such as the power lines, within the subscribing unit. The appliances to be managed each have associated therewith a responder unit, which is coupled to the electric grid to receive the transponder provided signals. Each of the central unit transmitted signals is encoded to manifest the energy managing dictates of a particular one of a plurality of diffferent schedules and is only provided in conformance with the dictates of the schedule is manifests. Typically, where an appliance is to be turned off as part of the energy management scheme, the encoded signals are provided only when the schedule manifested thereby indicate that a particular appliance is to be turned off. The responder units each have subscriber settable encoding devices associated therewith and the subscriber sets the code of a particular schedule for each responder after referring to series of schedules which is supplied to each user of the energy management system. The responder then responds to only the codes applied thereto conforming to the code set on the settable encoding devices and the appliance with which that responder is associated is then managed in accordance with the selected schedule.
Patent DE-3788884-T2 (DE)
Inventor: GIDDINGS JOHN C
IPC: G01N15/02
Filed: 1987-01-13
Granted: 1994-05-05
Abstract: A thin channel split flow process for particle fractionation which effects a rapid and efficient separation of the particles comprising continuously introducing two or more fluid substreams of different composition into separate inlet ports of a thin enclosed channel having a thickness which is very thin compared to the other two dimensions and bringing the substreams into contact with adjacent substreams so as to collectively form a series of thin laminae flowing parallel to one another in the channel and in contact with one another over a sufficient length of channel to allow a desired level of mass transport between and through laminae, continuously introducing a fluid medium containing the particles to be separated as one or more of the fluid substreams and independently of the particle concentration, varying the fluid composition of the different substreams as needed to realize separation, at the outlet end of the channel splitting the collective streams into another set of substreams so as to permit separate recovery of one or more of the substreams.
Patent DE-3850704-T2 (DE)
Inventor: SCHAD ROBERT D
IPC: B29C45/02
Filed: 1988-02-22
Granted: 1994-12-08
Abstract: Apparatus and method for tri-injecting a plurality of thermoplastic materials to mold an article having a layered wall structure using thermoplastic materials having different optimum processing temperatures including the maintenance of the optimum temperatures in flow paths individual to each material from its source at least to the injection nozzle.
Patent DE-3871905-T2 (DE)
Inventor: CALLUT FRANCOIS J
IPC: B03B9/00
Filed: 1988-11-11
Granted: 1992-12-10
Abstract: Particulate material such as coal of a size inferior to 1 mm is recovered by being entrained in a liquid medium and being fed through an apparatus comprising a plurality of cyclone separators (104, 112, 118, 125) connected in series, the cyclone angle of the separators decreasing in the direction of flow. The cyclone angle  alpha  2 of a cyclone separator in the series is within +/- 5% of the angle calculated according to the formula <MATH> where  alpha  2 is the cyclone angle of a cyclone separator following a separator with angle  alpha  1 and O1 and O2 represent the geometric mean particle size of the cut of successive separators with these angles.
Patent DE-3872330-T2 (DE)
Inventor: TERVAMAEKI JUKKA
IPC: B67D7/58
Filed: 1988-02-17
Granted: 1992-12-03
Abstract: PCT No. PCT/FI88/00024 Sec. 371 Date Oct. 13, 1988 Sec. 102(e) Date Oct. 13, 1988 PCT Filed Feb. 17, 1988 PCT Pub. No. WO88/06138 PCT Pub. Date Aug. 25, 1988.Dosage equipment, which includes a peristaltic pump for the dosage of liquid. The set of hoses (17) of the peristaltic pump includes an upper piece (18) and a lower piece (19). The body of the pump includes an attaching piece (13), to which the upper piece and the lower piece can be attached.
Patent DE-3873200-T2 (DE)
Inventor: YOSHIHAMA MAKOTO
IPC: A61K31/565
Filed: 1988-02-05
Granted: 1993-02-25
Abstract: Androst-4-ene-3,17-diones of formula (I) are new; where X is =O or beta-OR; Y is H or OH; Z is H or OH; and R is H, acetyl, propionyl, isobutyryl or pivaloyl. Pref. 14alpha-hydroxyandrost-4-ene -3,6,17-trione; 6beta,11alpha-dihydroxyandrost -4-end-3,17-dione; 6beta,14alpha-dihydroxyandrost -4-ene-3,17-dione; 6beta-acetoxy-14alpha-hydroxyandrost -4-ene-3,17-dione; 14alpha-hydroxy-6beta-propionyloxy androst-4-ene-3,17-dione; 14alpha-hydroxy- 6beta-isobutyryloxyandrost -4-end-3,17-dione and 14alpha-hydroxy-6beta pivaloyloxyandrost-4-ene-3,17-dione. Prepn. comprises culturing Acremonium species (esp. A.strictum NN-106; FERM P-9143) in the presence of androst-4-ene-3,17-dione gives (I, X = beta-OH) which may be oxidised to (I, X = =O) or acylated (e.g. with an acid anhydride).
Patent DE-3880938-T2 (DE)
Inventor: HENSLER PAUL LEONARD
IPC: C01B25/41
Filed: 1988-08-08
Granted: 1993-09-02
Abstract: The method of prodycing sodium tripolyphosphate hexahydrate powder which comprises hydrating anhydrous sodium tripolyphosphates having a particle size such that at least 85% by weight is less than 150  mu m with sufficient water to provide not more than 105% of the theoretical amount of water to form the hexahydrate, drying the sodium tripolyphosphate hexahydrate to remove substantially all of the uncombined water and maintaining said hydrating and drying steps at less than 80% thereby producing a sodium tripolyphosphate hexahydrate powder such that at least 50% by weight is less than 150 mu m. It is particularly useful for use as a builder in a heavy duty detergent.
Patent DE-3882868-T2 (DE)
Inventor: STORAY CRAIG FRANCIS
IPC: B62B1/00
Filed: 1988-04-12
Granted: 1994-03-10
Abstract: A hand trolley for lifting and moving an object comprises a support frame for the object and a wheel assembly coupled to the support frame by means of a link arm (33) on each side of the trolley. Each link arm is connected at one end to the axle (31) of the wheel assembly and pivotally connected at the other end to the support frame. In a carry position of the trolley, at which the object is supported on the wheel assembly, the link arms (33) are located in a locked position so as to lock together the wheel assembly and the support frame when an operator pulls the trolley rearwardly over an obstacle
Patent TR-199900202-T2 (TR)
Inventor: KAFKA BERNARD
IPC: C08L95/00
Filed: 1997-07-17
Abstract: Ziftin özelliklerini iyilestirmek için kullanilan mineral lifli katkilar açiklanmaktadir. Erimis zift için bir mineral lifli katki tedarik edilmektedir.Bu katkidaki lifler ziftin içine eklenmeden önce küçük bogumlar halinde biraraya getirilmektedir. Sözü edilen katki, su ve isi karsisinda özelliklerini koruyan ve önceden bir isitici ajan ile islemden geçirilerek lifleri zift ile islatilan bir baglayici da içermektedir. Su ve isi karsisinda özelliklerini koruyan bu baglayici tercihen, genellikle cam ya da tas yönünden yapilmis yalitici hasirlarin üretilmesinde kullanilan cinsten fenolik reçineden olusmaktadir.
Patent DE-60000036-T2 (DE)
Inventor: DE NANTEUIL GUILLAUME
IPC: C07D401/12
Filed: 2000-05-02
Granted: 2002-07-18
Abstract: 2,3-methano amino acid derivatives (I), their isomers, their acid and base addition salts, their preparation, and pharmaceut compositions are new. The new compounds are of formula (I) n = 2 or 3; R1 = 3-8C cycloalkyl, phenyl (optionally substituted), 1-6c alkyl (optionally substituted by one or more halogens, 3-8C cycloalkyl, or phenyl, itself optionally substituted); R2 = amino, amidino (optionally substituted by one or more alkyl or OH groups), guanidino (optionally substituted by alkyl), or isothioureido (optionally substituted by 1-6C alkyl); Ar = aryl or nitrogen monocyclic heteroaryl; X1 = OH, amino, or -NHR3; R3 = propargyl, iminomethyl, 1-6C alkylsulfonyl, arylalkyl sulfonyl, -CONR'3R3 or 1-6C alkyl (optionally substituted by -COOR'3, -CONR'3R3, heterocycle, aminosulfonyl, aryl, or heteroaryl,; R'3 and R3 = H, 1-6C alkylsulfonyl, aryl, alkyl (optionally substituted by carboxy, alkoxycarbonyl, or carbamoyl), or together with the N atom they form a heterocycle.
Patent DE-60001120-T2 (DE)
Inventor: MEYN PIETER
IPC: A22C21/00
Filed: 2000-02-03
Granted: 2003-11-13
Abstract: An apparatus for suspending poultry by the feet from an overhead conveyor has pairs (12,34) of cooperating strings for gripping the poultry by the feet in an upside-down hanging position in order to supply them to the overhead conveyor respectively in preparation of that. Check means (6,9) are applied to check the position of the feet with respect to the strings in the hanging position of the poultry, and to provide a control signal that depends thereon. <IMAGE>
Patent DE-60002672-T2 (DE)
Inventor: ZENTI MAXIMILIANO
IPC: A01C1/04
Filed: 2000-02-23
Granted: 2004-03-25
Abstract: A sod of cultivation soil, complete with lawn grass seeds, fertilizers, selective herbicide and a bonding agent for the cohesion of the various elements contained therein. The sod has the conventional geometric shapes of paving tiles and allows to cover continuously, i.e. without gaps, the soil to be revegetated. A method for producing the sod makes it possible to store it and subsequent reuse it while obtaining optimum and rapid growth, of lawns, grassy layers, flowers and the like.
Patent DE-60003526-T2 (DE)
Inventor: PATUREAUX THIERRY
IPC: B65B1/06
Filed: 2000-01-27
Granted: 2004-04-29
Abstract: The invention relates to a method for facilitating the filling of a vertical tube (1) with the aid of a solid material in a particulate state, whereby the particles move downwards in said tube as a result of gravity and encounter obstacles along the path thereof, whereby said obstacles are supported by at least one cable or similar that is vertically suspended in the tube. According to the invention, the particles encounter at least three obstacles during the fall thereof, whereby said obstacles are disposed in the tube at different levels and are supported by at least two cables (4) that are laterally offset in relation to the axis of the tube.
Patent DE-60003682-T2 (DE)
Inventor: HESS JOSEPH
IPC: B05B12/00
Filed: 2000-08-30
Granted: 2004-05-27
Abstract: The smart fragrance dispensing device (1) comprises an airless fragrance reservoir (1a) containing a principal medium (8), a flow channel (3) for receiving said principal medium (8), a liquid spray dispenser (2) connected to said reservoir (1a) for dispensing said principal medium (8) as a spray into said flow channel (3), a programmable driving circuit (5) for operating said liquid spray device so as to create said spray consisting of monodispersive droplets, a memory device (4) carrying and communicating identification information about at least said principal medium (8), its dispensing and diffusing characteristics, said liquid spray dispenser (2) and said reservoir (1a), and a programmable control and communication micro-controller unit (7) linked to said reservoir (1a), said programmable, driver circuit (5), and said flow channel (3), and controlling the programmable driver circuit (5) and the flow channel (3) in such a manner that flow is started in time before the driver circuit (5) is activated and stopped in time after the driver circuit (5) is activated and otherwise as a function of information read from said memory device (4), said information being used to adapt to the individual perception of a user by means of adjusting to a desired level and memorising said level. <IMAGE>
Patent DE-60006999-T2 (DE)
Inventor: COLLINS IAN RALPH
IPC: C09K23/00
Filed: 2000-11-09
Granted: 2004-05-27
Abstract: A method of treating a subterranean formation, the method comprising: (A) injecting down a well bore into the formation an admixture of (a) an emulsion having an internal aqueous phase comprising a water-soluble oil or gas field chemical or an aqueous dispersion of a water-dispersible oil or gas field chemical and an external oil phase comprising a liquid hydrocarbon and an oil-soluble surfactant and (b) a demulsifier comprising a solution of a surfactant having a cloud point temperature of above 40° C.; or (B) separately injecting down a well bore into the formation emulsion (a) and demulsifier (b) and generating an admixture of emulsion (a) and demulsifier (b) within the formation.
Patent DE-60010237-T2 (DE)
Inventor: KENDALL K
IPC: C07C17/02
Filed: 2000-02-15
Granted: 2005-04-14
Abstract: This invention relates to the production of an hexabromocyclododecane product, which process comprises brominating cyclododecatriene in the presence of a 1,4-dioxane and water based solvent and from about 0.5 to about 30 wt % bromide ion in the liquid phase of the reaction mass. Optional post-reaction heat treatment in a finishing step increases process yields if needed. The hexabromocyclododecane product is unrecrystallized and contains no more than about 1.5 wt % tetrabromocyclododecene impurities.
Patent DE-60010582-T2 (DE)
Inventor: LE ROUX JEAN-CLAUDE
IPC: B63C9/125
Filed: 2000-07-05
Granted: 2005-05-19
Abstract: The sea rescue harness has an exterior envelope (3) and an inner inflatable bag (4) formed separately. The strap (5) is attached to the envelope and the bag is of inverted U-shape with the branches (4a,b) attached to the strap. The envelope is formed by two flaps (3a,b) with their outer sides attached by straps (6,7) with hooks and loops to allow opening of the envelope during inflation of the bag.
Patent DE-60011387-T2 (DE)
Inventor: VAN GANSBERGHE FREDERIC M
IPC: E03F5/06
Filed: 2000-04-04
Granted: 2005-06-16
Abstract: The cleaner, especially for drains covered by gratings, consists of a mobile head (16) with rollers (22) to guide it along the edges of the gratings, and angled pipes (18) for projecting a fluid under pressure between the bars (14) of the gratings. The mobile head is moved either manually or automatically along the grating following the slope upwards as the pressure fluid is delivered to its angled pipes (18) from a reservoir and through a coupling (20).
Patent DE-60015655-T2 (DE)
Inventor: PARENT HUGUES
IPC: F24D3/10
Filed: 2000-06-20
Granted: 2005-07-28
Abstract: Part of fluid flowing in main pipe (3) is diverted and introduced into expansion vessel through inlet pipe (4). Fluid is withdrawn from expansion vessel and introduced through evacuation pipe (5) into main pipe downstream of inlet pipe water intake. Main pipe houses a valve (6) between water intake (A) of inlet pipe (4) and outlet (B) of evacuation pipe (5). Inlet pipe (4) also houses valve (7). Isolating valve (13) temporarily seals inlet and outlet pipes and purge tap (14) empties contents of vessel.
Patent DE-60015667-T2 (DE)
Inventor: DUMOULIN-WHITER ROGER J
IPC: A61B17/00
Filed: 2000-08-08
Granted: 2005-11-24
Abstract: A method is provided for treating a patient having a disorder, wherein the method includes irradiating a tissue surface of the patient with at least one laser beam, automatically monitoring the tissue, and automatically controlling the at least one laser beam to adjust and/or terminate the treatment in a therapeutically effective manner. The method noninvasively determines in real-time the irradiance and/or radiant exposure of a target tissue at a predetermined depth below the tissue surface by detecting the radial dependence of light remitted from the tissue surface. Preferably, the method employs a near-infrared light laser beam and a visible laser light beam in combination. An apparatus for performing the method is also provided.  <IMAGE>
Patent DE-60017353-T2 (DE)
Inventor: QUINN PATRICK
IPC: F24C3/12
Filed: 2000-01-20
Granted: 2006-03-02
Abstract: The gas cooker has a burner connected to a gas conduit with a metering control for the gas. The burner has an injector (8) for pilot flame supply and a burner (7) for cooking. The control has a first valve (4) with a push button (12) and a second valve (5) placed downstream of the first. The first valve is connected to the injector (8) for the pilot gas supply. The second valve is connected to the burner and has a control lever (6). The first valve can be controlled by a thermocouple in the pilot flame to control the valve.
Patent DE-60019425-T2 (DE)
Inventor: HASSINEN REIJO
IPC: D21G3/00
Filed: 2000-02-01
Granted: 2006-03-09
Abstract: The invention relates to a doctor assembly in a paper machine, which is intended to clean, e.g., a roll, and which includes a surface against which a doctor blade is set, a blade support for supporting the doctor blade, a frame, a jointed bearing assembly, which supports the doctor blade and is itself supported from the frame, and which is parallel to the doctor blade, and extends essentially over the entire width of the roll, and loading devices between the blade support and the frame for turning the doctor blade in relation to the frame and for pressing the doctor blade against the surface with a selected pressure. Due to the continuous support, there is essentially no deflection in the doctor assembly, when it is attached by its frame directly to the structures of the paper machine.