baber/WOPTO huggingface dataset:
Patent BG-64420-B1 (BG)
Title: 2,3-diaryl-pyrazolo[1.5-b]pyridines derivatives, method for their preparation, pharmaceutical composition and usage theof
Inventor: BESWICK PAUL
IPC: C07D487/04
Filed: 2000-03-28
Abstract: The invention relates to 2,3-diarylpyrazolo[1,5-B] pyridazine compounds and to their pharmaceutically acceptable derivatives. They are potent and selective inhibitors of COX-2 and are of use in the treatment of pain, fever and inflammations of a variety of conditions and diseases. The compounds have the general formula wherein R0 is halogen, C1-6 alkyl, C1-6 alkoxy, C1-6 alkoxy substituted by one or more fluorine atoms, or O(CH2)nNR4R5; R1 and R2 are independently selected from H, C1-6 alkyl, C1-6 alkyl substituted by one or more fluorine atoms, C1-6 alkoxy, C 1-6 hydroxyalkyl, SC1-6 alkyl, C(O)H, C(O)C1-6 alkyl, C1-6 alkylsulphonyl, C1-6 alkoxy, substituted by one or more fluorine atoms, O(CH2)nCO2C1-6 alkyl, O(CH2)n SC1-6alkyl, (CH2)nNR4R5, (CH2)nSC1-6 alkyl or C(O)NR4R5; with the proviso that when R0 is at the 4-position and is halogen, at least one of R1 or R2 is C1-6 alkylsulphonyl, C1-6 alkoxy, substituted by one or more fluorine atoms, O(CH2)nCO2C1-6 alkyl, O(CH2)nSC1-6 alkyl, (CH2)n NR4R5 or (CH2)nSC1-6 alkyl, C(O)-NR4R5; R3 is C1-6 alkyl or NH2; R4 and R5 are independently selected from H, or C1-6 alkyl or, together with the nitrogen atom to which they are attached, form a 4-8 membered saturated ring; and n has the value of from 1 to 4.
Patent BG-66255-B1 (BG)
Title: Natural language formalization
Inventor: POPOV IVAYLO
IPC: G06F17/28
Filed: 2007-11-14
Abstract: The formalization finds application in machine translation. It helps achieve synonymous interpretation of the natural language. Under the method, the basic concepts are determined of the essences named by the natural language
Patent CH-700946-B1 (CH)
Title: Tool revolver for use in turning machine, has cutting tool with output shaft aligned with or parallel to output shaft of electric drive motor arranged in tool disk, where output shaft of tool is driven perpendicular to longitudinal axis
Inventor: SAUTER, REINER
IPC: B23B29/32
Filed: 2007-07-06
Abstract: The revolver has a housing (10) connected with a machining tool, and a tool disk (14) pivotably mounted along a longitudinal axis (34) with respect to the housing and fixable in selective angular positions. The tool disk has a holder (16) for holding a rotary cutting tool (18) that is mounted on an output shaft (30) that is driven perpendicular to the longitudinal axis by an electric drive motor (28) that is arranged in the tool disk. An output shaft (24) of the cutting tool is aligned with or parallel to the output shaft (30) of the motor.
Patent CH-700112-B1 (CH)
Title: Schuh.
Inventor: CHUANG-CHUAN CHEN
IPC: B29D35/00
Filed: 2007-08-24
Abstract: Schuh mit einem Verbindungsrahmen (230), welcher die Verbindung des Blatts mit der Laufsohle (240) des Schuhs verbessert, wobei der Schuh aufweist: ein Blatt mit einem Seitenblatt (210) und einem Sohlenblatt (220), einen Verbindungsrahmen, der eine erste Aussenfläche, die das Seitenblatt umläuft, eine zweite Aussenfläche, die an die erste Aussenfläche angeschlossen ist und sich nach aussen erstreckt, eine dritte Aussenfläche, die an die zweite Aussenfläche angeschlossen ist, und sich abwärts erstreckt, und eine vierte Aussenfläche aufweist, die an die dritte Aussenfläche angeschlossen ist und sich einwärts erstreckt, wobei die zweite Aussenfläche eine Mehrzahl von Löchern aufweist; und eine Laufsohle, die den Verbindungsrahmen und das Sohlenblatt umgibt, wobei eine Lücke zwischen der vierten Aussenfläche des Verbindungsrahmens und dem Sohlenblatt und die Löcher in der zweiten Aussenfläche mit einem Material ausgefüllt sind, von welchem die Laufsohle ausgebildet wird.
Patent CH-714455-B1 (CH)
Title: Elektrischer Verteilerkasten zur Bereitstellung von elektrischem Strom.
Inventor: DIRK SANER
IPC: H02B1/52
Filed: 2017-12-15
Abstract: Die erfindung betrifft einen elektrischen Verteilerkasten (1) zur Bereitstellung von elektrischem Strom, der Verteilerkasten (1) umfassend einen Versorgungsanschluss (11) zum Verbinden des Verteilerkastens (1) an ein Stromversorgungsnetz, mindestens eine Steckdose (12a, 12b) zum Anschliessen eines Verbrauchers, ein Kommunikationsmodul (14), welches eingerichtet ist, einen Schaltbefehl von einer computerisierten Verwaltungsvorrichtung zu empfangen, eine Steuerung (15), welche mit dem Kommunikationsmodul (14) verbunden ist, und eingerichtet ist, in Abhängigkeit des Schaltbefehls ein Schaltsignal zu erzeugen, ein Schaltmodul (13), welches mit der Steuerung (15) verbunden ist, und eingerichtet ist, in Abhängigkeit des Schaltsignals die mindestens eine Steckdose (12a, 12b) mit dem Versorgungsanschluss (11) zu verbinden oder vom Versorgungsanschluss (11) zu trennend Darüber hinaus betrifft die erfindung ein Verfahren zum bereitstellen von elektrischen strom mit einem derartigen Verteilerkasten.
Patent CU-24004-B1 (CU)
Title: Peptidomiméticos de smac útiles como inhibidores de proteínas de apoptosis (iap)
Inventor: CHAREST MARK
IPC: C07K5/06
Filed: 2011-02-02
Abstract: La presente invención se refiere a un compuesto de la fórmula (I); o sales farmacéuticamente aceptables del mismo útiles para el tratamiento de enfermedades proliferativas, tales como cáncer, en mamíferos. ESPACIO PARA LA FÓRMULA
Patent DD-239044-B1 (DD)
Title: Feuchtebestimmungsvorrichtung fuer loses, flockiges textilgut
Inventor: HOTZ MICHAEL
IPC: G01N27/04
Filed: 1985-07-02
Abstract: Die Erfindung bezieht sich auf eine Feuchtebestimmungsvorrichtung für loses, flockiges Textilgut am Siebtrommeltrockner und beinhaltet, daß sich mehrere quer zur Transportrichtung des Textilgutes und geringem Abstand zum Textilgut angeordnete, sich nicht berührende Meßwertaufnehmer (I, - 1"), die an die am Ausgang des Trockners befinliche Siebtrommel (0) andrückbar sind, befinden. Die Meßwertaufnehmer (1, - 1,) sind kabelmäßig verbunden mit einem Widerstandsnetzwerk (2), Operationsverstärker (3), Leistungsverstärker (4), Analog-Digital-Wandler (5), Mikrorechner (6) und Meßwertanzeige (7). Damit kann ein repräsentativer Feuchtewert pro Zeiteinheit erhalten werden, so daß verschiedene Prozeßgrößen des Trockners geregelt werden können.
Patent EP-1060762-B1 (EP)
Inventor: NAPPHOLZ TIBOR
IPC: A61N1/37
Filed: 2000-04-20
Granted: 2006-08-30
Abstract: The method involves pre amplifying the sampling signals using two preamplifiers (7,8). The pre amplified sampling signals are compared using a comparator (9). The sampling signals (CARD) and interference signals (EMI) are discriminated between by a phase-sensitive evaluation of the comparator output signal. The comparator output signal is fed back to the gain control of the preamplifier so that while an interference signal is detected, the comparator output signal is minimized. To select interference signals, the comparator output signal is monitored for step function signals. An apparatus for performing the method is also claimed.
Patent EP-1112832-B1 (EP)
Inventor: MAENNER HANS-PETER
IPC: B29C45/30
Filed: 2000-09-06
Granted: 2004-11-10
Abstract: Needle (2) is mounted slidably in the inner side of nozzle (1). A gap is formed between needle end (3) and inflow opening (4). The needle is pulled inwardly to enlarge the gap between needle end and inflow opening. Reciprocation of the needle is made by drive unit selected from piston drive unit (6), locating motor, piezoelectric actuator. The drive unit acts on the extension (5) of needle. The gap formed between the needle end and inflow opening is controlled to large size during starting of molding after which gap is reduced. The position of the needle is adjusted from starting to finishing of post pressure application process. The nozzle is slid to ingate opening before removal from mold.
Patent EP-1029663-B1 (EP)
Inventor: BALDUIN MICHAEL
IPC: B32B37/00
Filed: 2000-01-26
Granted: 2009-12-30
Abstract: Two rigid glass plates and a bonding layer are loosely placed together to create a preform. The preform is then subjected to a pressure below atmospheric and simultaneously heated and pressed together using flexible press parts. Pressure on the laminate is then increased to atmospheric.  An Independent claim is made for the process plant which includes an inlet sluice(4), an evacuated heating chamber(7), an evacuatable press chamber(9) with press parts(11,12), an outlet sluice(16), closures(6,15) for dividing the inlet and outlet sluices from the heating and pressing chamber and conveyers(2,8,10,17) for moving laminating materials through the process chambers.
Patent EP-1150999-B1 (EP)
Inventor: MUTTER MANFRED
IPC: A61K38/13
Filed: 2000-02-07
Granted: 2006-06-21
Abstract: The invention relates to cyclosporin derivatives, whereby the peptide chain thereof comprises at least one pseudo-proline type non-natural amino acid radical. The invention also relates to a method for the production of said derivatives.
Patent EP-1151233-B1 (EP)
Inventor: THOMAS DONALD S
IPC: F26B21/06
Filed: 2000-01-11
Granted: 2005-04-06
Abstract: A process and apparatus for removing moisture from a material, without spoiling the processed product, through the implementation of microwave irradiation heating, drying, dehydration, curing, disinfection, pasteurization, sterilization or vaporization or any combination thereof. The process and apparatus provide for a controlled processing of planar material, a combination of materials organic or inorganic, in natural or processed form, in sheet leaf, granular, prepared or transportable planar form.
Patent EP-1152915-B1 (EP)
Inventor: BRAND WERNER
IPC: B60L5/28
Filed: 2000-01-28
Granted: 2003-03-19
Abstract: A device for determining the pressure between a contact wire and a pantograph of an electrically-powered vehicle is provided with a measuring device for the static pressure that is determined from the distance between two elastically-connected components, the distance being a function of the static pressure, the device further having an acceleration sensor, which is coupled with the pantograph for determining the pantograph accelerations occurring in the direction of the pressure. The output signal of the acceleration sensor is linked with the output signal of the measuring device for calculating the pressure. The acceleration sensor is embodied to include a seismic mass (3) that is resiliently mounted to the pantograph (6) and whose respective position relative to the pantograph is optically detected, and a corresponding light signal is transmitted to an optoelectrical converter that is potential-isolated from the pantograph (6).
Patent EP-1072090-B1 (EP)
Inventor: MOERS PAULUS LOUIS GUIDO
IPC: H03J1/00
Filed: 2000-02-11
Granted: 2005-04-20
Abstract: L'invention concerne un procédé de traitement de données émetteur et programme dans un récepteur FM RDS, ainsi que le récepteur exécutant ledit procédé, comprenant une recherche par balayage de bande afin de détecter des émetteurs FM RDS dépassant un niveau de qualité de réception prédéterminé. Afin d'améliorer l'efficacité du traitement de données et l'utilisation de la capacité de stockage, les données émetteur, y compris les données de mise au point, sont mémorisées séparément des données programme RDS. Pour chaque émetteur détecté, un facteur de qualité indiquant la qualité de réception est assigné à chaque émetteur RDS détecté et mémorisé dans un premier bloc de mémoire, avec les données de mise au point pertinentes. Pour chaque code d'identification de programme acheminé dans les données RDS des émetteurs ainsi détectés, des données programme FM RDS sont mémorisées dans un second bloc de mémoire, un code de liaison définissant l'adresse de stockage dans le second bloc de mémoire contenant les données programme portées par l'émetteur FM RDS pertinent assigné aux données émetteur de chaque émetteur FM RDS et mémorisé dans le premier bloc de mémoire.
Patent EP-1139837-B1 (EP)
Inventor: KARKOS JOHN F JR
IPC: F25C5/12
Filed: 2000-01-11
Granted: 2002-12-04
Abstract: A magnetic induction drive for a rotatable driven member in a sealed housing, in particular, a shaft-mounted blade in a blender cup or a shaft-mounted blade in an ice shaver, uses a comparatively thin circular drive plate of a magnetizable material with circumferentially arrayed poles enclosed within a housing secured to a drive shaft. A brushless d.c. motor in a base separate from the housing has a rotor formed as an array of pie-shaped permanent magnet regions that interact with an electronically controlled, rotating electromagnetic field produced by a ring of stator coils. A second such permanent magnet is coupled to rotate coaxially and in unison with the rotor, with poles of opposite polarity aligned and adjacent one another. A steel disc is sandwiched between and bonded to the rotor and the second permanent magnet. The magnetic field (lines of flux) of the second magnet extends axially away from the rotor to induce magnetic poles of opposite polarity in the drive plate. This second magnet-to-plate magnetic coupling operates across a closely-spaced gap that includes the bottom wall of the base, the upper wall of the housing, and air gaps between these walls, and the plate and the second magnet. A gear train assembly can be coupled to the drive shaft to increase or decrease the amount of torque transmitted from the drive plate to the driven member.
Patent EP-1169115-B1 (EP)
Inventor: MORDUE GEORGE S
IPC: C21C5/46
Filed: 2000-04-07
Granted: 2006-03-29
Abstract: A coupling mechanism for a molten metal processing system includes an elongated shaft having an upper axial end and a lower axial end. A passage having a torque facilitating shape extends through at least a portion of the shaft. The upper end of the shaft tapers inwardly and forms a tapered seat. At least one channel is machined into an outer surface of the upper end of the shaft. The channel has a first portion extending longitudinally downward from a top surface of the shaft and a second portion extending from the first portion at an angle greater than 90° relative to the first portion. A coupling member, for coupling the shaft to a drive system forming a bayonet coupling. The cavity of the coupling member tapers outwardly forming a mouth which engages the tapered seat of the shaft in a sealing relationship.
Patent EP-1244851-B1 (EP)
Inventor: JAEKAERAE JUKKA
IPC: D21H11/16
Filed: 2000-06-14
Granted: 2003-05-07
Abstract: The invention relates to a method for treating mechanical pulp so that aliphatic percarboxylic acid in the amount of 0.5 - 5 kg/ton of pulp is added to the pulp to improve the opacity.
Patent EP-1109644-B1 (EP)
Inventor: KOPRAS ROBERT K
IPC: B23B45/00
Filed: 2000-06-12
Granted: 2007-08-01
Abstract: An angle attachment of a hand-held power tool, such as a spiral cutting tool, includes an angle attachment housing having an open first end adapted to be attached to the motor housing of the power tool. An alignment bearing is mounted in the angle attachment housing and adapted to receive and support a first shaft having a first shaft gear mounted thereon. An attachment shaft is mounted in the angle attachment housing at an angle, e.g., a right angle, to the first shaft. The attachment shaft includes an attachment shaft gear mounted thereon which is engaged with the first shaft gear. One or more attachment shaft bearings are mounted in the angle attachment housing to support the attachment shaft for rotational movement thereof. The first shaft is coupled to a motor shaft of the power tool before the angle attachment housing is attached to the power tool motor housing. Rotation of the first shaft by the power tool motor causes rotation of attachments attached to the attachment shaft mounted at an angle to the first shaft by means of the gear mechanism formed by the engaged first shaft gear and attachment shaft gear.
Patent EP-1194898-B1 (EP)
Inventor: RIGG RICHARD TYSON
IPC: G06T11/00
Filed: 2000-06-09
Granted: 2003-03-05
Abstract: A method and apparatus is provided for virtual color makeover of a customer's face. A digital image is taken of the customer's face. Natural skin color is determined by a differential analysis among at least two different sites along the face to identify an area without color. The identified area without color is then used as a basis for projecting the customer's face with the natural skin color. Consultant's choice of preprogrammed color palettes matching the measured natural skin color is then projected on the facial image. A customer's personal choice such as fashion, natural or go-to-work looks can be registered for modifying the consultant's choice color palette. The selected color palette can then be identified as a set of color cosmetic products which are provided to the customer.
Patent EP-1200208-B1 (EP)
Inventor: STOCCHI GABRIELE
IPC: B67C3/24
Filed: 2000-06-28
Granted: 2005-09-07
Abstract: A machine for treating objects having a series of stations ( 12 ) whereof each includes a system for gripping ( 16 ) a container ( 11 ) in a loading point of the path, wherein, between the loading and unloading points, the container ( 11 ) is displaced from an initial loading position to at least a treating position then to a final unloading position following the circular path. Each station is provided with a gripping unit ( 14 ) comprising at least two grip systems ( 16 ), and the gripping unit ( 14 ) is mobile relative to the station between at least two positions and, between the loading and unloading of an object, the path followed by the latter has a number of cycles of the circuit ranging between the number of grip systems ( 16 ) of each grip unit ( 14 ) and the next lower integer.
Patent EP-1211242-B1 (EP)
Inventor: SATO FUMIE
IPC: C07C405/00
Filed: 2000-09-08
Granted: 2010-01-13
Abstract: A prostaglandin derivative represented by the formula: <CHEM> wherein X is a halogen atom in the  alpha - or  beta -position, Y is an ethylene group, a vinylene group or an ethynylene group, A is a group represented by the formula: O(CH2)n, S(O)p(CH2)n, O(CH2)qO(CH2)r, O(CH2)qS(O)p(CH2)r, S(O)p(CH2)qS(O)p(CH2)r or S(O)p(CH2)qO(CH2)r (wherein n is an integer of 1 to 5, p is 0, 1 or 2, q is an integer of 1 to 3, and r is 0 or 1), R<1> is a C3-10 cycloalkyl group, a C1-4 alkyl-C3-10 cycloalkyl group, a C3-10 cycloalkyl-C1-4 alkyl group, a C5-10 alkyl group, a C5-10 alkenyl group, a C5-10 alkynyl group or a bridged cyclic hydrocarbon group, R<2> is a hydrogen atom, a C1-10 alkyl group or a C3-10 cycloalkyl group, and m is 0, 1 or 2Ü, a pharmaceutically acceptable salt thereof or a hydrate thereof. The present invention is to provide novel PG derivatives having an excellent PGD2-like agonistic activity and a sleep-inducing action.
Patent EP-1330938-B1 (EP)
Inventor: WIDMER CHRISTOPH
IPC: H04R25/00
Filed: 2000-09-25
Granted: 2004-05-12
Abstract: Appareil auditif dans la coque duquel (79) est intégré le conducteur acoustique (81) raccordé à l'entrée d'un transducteur acoustique / électrique ou électrique / acoustique.
Patent EP-1223998-B1 (EP)
Inventor: MUNK JENS
IPC: A61M5/24
Filed: 2000-09-29
Granted: 2007-10-10
Abstract: The present invention relates to an electronic injection device wherein an electronic circuit is designed to work in two alternative modes: an air shot mode and a dose injection mode. When working in the air shot mode a small predetermined air shot dose is pressed out from the ampoule when the injection button is actuated. When working in the injection mode, a dose set by operation of the dose setting means is injected by operation of the injection button. The electronic injection device is normally working in the air shot mode but shifts to work in the dose injection mode when it receives a signal indicating that the dose setting means has been operated. The circuit returns to its air shot mode when receiving a signal indicating that the set dose has been injected. This signal can originate either from a switch indicating that the protection cap is mounted or from a switch indicating that the injection button has been pressed.
Patent EP-1225943-B1 (EP)
Inventor: GENOSAR AMIR
IPC: A61M15/00
Filed: 2000-11-01
Granted: 2007-01-24
Abstract: A metered dose inhaler for use with a pressurized aerosol canister includes a housing defining a conduit with a mouthpiece, and an actuator with a nozzle discharge orifice arranged to discharge aerosol into the conduit. Vortex generators positioned within the wall of the conduit and in fluid communication with air inlets for receiving ambient outside air, provide the inner wall of the conduit with a circumferential-swirling turbulent boundary layer flow to minimize impaction of medication on the inner surfaces of the conduit.
Patent EP-1150105-B1 (EP)
Inventor: SANDER DIETMAR DR
IPC: B01L3/02
Filed: 2001-04-23
Granted: 2010-04-07
Abstract: The micro dosing system has a liquid reservoir (1) with a storage space (1') for the liquid to be dosed and a gas displacement system with a micropump (2), coupled to a dosing control (7) for providing a reduced or raised pressure for the liquid reservoir upon operation of the micropump, for drawing liquid into the storage space or ejecting it from the storage space.
Patent EP-1152506-B1 (EP)
Inventor: KNAB JOSEF
IPC: H02B1/01
Filed: 2001-04-19
Granted: 2003-10-01
Abstract: The frame has transverse profiles, depth profiles and vertical profiles connected by corner joints (5) with three plug-in fittings (7-9) onto which transverse, depth and vertical profiles can be fitted and fixed with the aid of a clamping part (10) with clamping arms (13-15) for holding the profiles and a connecting element for fixing onto the corner joint.
Patent EP-1179408-B1 (EP)
Inventor: DANTLGRABER JOERG
IPC: B29C33/20
Filed: 2001-04-28
Granted: 2007-07-04
Abstract: An electric motor (27) drives a initial cross-member (30) in a straight line in the direction of the motor axis to operate a lever mechanism connected to the moving platen (18). The lever mechanism comprises a lever (32) divided into short (40) and a long (39) arm sections. The long arm is connected to the initial cross-member and the short arm is perpendicular to platen movement and is connected to the platen. Preferred Features: The lever is either an extended lever where the long arm (39) is also perpendicular to the platen movement or an angled lever which, during tool closure, makes an angle of NOTGREATER  90 degrees with the direction of platen movement.
Patent EP-1148136-B1 (EP)
Inventor: WILSON C RON
IPC: C07K14/40
Filed: 1999-09-10
Granted: 2012-12-05
Abstract: Novel genes have been isolated which encode cytochrome P450 and NADPH reductase enzymes of the ω-hydroxylase complex of C. tropicalis 20336. Vectors including these genes, transfected host cells and transformed host cells are provided. Methods of producing of cytochrome P450 and NADPH reductase enzymes are also provided which involve transforming a host cell with a gene encoding these enzymes and culturing the cells. Methods of increasing the production of a dicarboxylic acid and methods of increasing production of the aforementioned enzymes are also provided which involve increasing in the host cell the number of genes encoding these enzymes. A method for discriminating members of a gene family by quantifying the expression of genes is also provided.