baber/WOPTO huggingface dataset:
Patent EA-018917-B1 (EA)
Title: 6-o-substituted benzoxazole and benzothiazole compounds and methods of inhibiting csf-1r signaling
Inventor: SUTTON JAMES C
IPC: A61K31/44
Filed: 2007-04-18
Abstract: Benzoxazole and benzothiazole compounds and the stereoisomers, tautomers, solvates, oxides, esters, and prodrugs thereof and pharmaceutically acceptable salts thereof are disclosed. Compositions of the compounds, either alone or in combination with at least one additional therapeutic agent, with a pharmaceutically acceptable carrier, and uses of the compounds, either alone or in combination with at least one additional therapeutic agent are also disclosed. The embodiments are useful for inhibiting cellular proliferation, inhibiting the growth and/or metathesis of tumors, treating or preventing cancer, treating or preventing degenerating bone diseases such as rheumatoid arthritis, and/or inhibiting molecules such as CSF-1R.
Patent EA-018669-B1 (EA)
Title: Transport vehicle for personnel conveyance
Inventor: PEJSAROV VALERIJ NISANOVICH
IPC: B60P3/14
Filed: 2009-08-06
Abstract: A transport vehicle for personnel conveyance comprises a cab 1, an engine 2 and a chassis comprising a front frame 3 and a rear frame 4. The cab 1 with a steering wheel, the engine 2 with a hydromechanical gear 5 and a front driving axle 6 are mounted on the front frame, wherein a rear driving axle 7, a manrider 11 with four doorways on both sides of the rear driving axle 7 are mounted on the rear frame 4. The frames 3, 4 are pivotally connected by hinges 8, 9 coaxially arranged one above the other. Hydro cylinders 16,17 of the vehicle turn are pivotally fixed by sleeves on the rear frame 4 and pivotally connected by rods to the front axle 3. The engine 2 is connected to the front axle 6 by a propeller shaft 10 and to the rear axle by two serially connected propeller shafts 12,13. A dosing pump 14 is connected to a common hydraulic tank 23, gear feed pump 18 and to two hydro cylinders 16,17 via six line and three line distributors 24, 25, wherein the latter is connected to a braking hydro system comprising three hydropneumatic accumulators 26 connected to brake cavities 27 via distributors 28,29,30. The invention results in widening the range of turn angles of the front frame relative to the rear frame, and angles of ascent, increasing permissible load capacity and permissible angle of vehicle incline during running and stop, safety, stability, durability and reliability of the vehicle are enhanced, the maneuvering and control abilities in restricted conditions are broadened, layout and distribution of operation loads are optimized, raising the operation efficiency.
Patent EA-015792-B1 (EA)
Title: Shock absorber for transport vehicle
Inventor: TIKHONENKO OLEG OLEGOVICH
IPC: F16F5/00
Filed: 2010-12-03
Abstract: The invention relates to mechanical engineering and can be used in manufacturing and operation of shock absorbers. The invention is aimed at improving shock absorber damping properties, the shock absorber of a transport vehicle comprises a bushing, a piston cover, a rod cover, a rod piston with seal, the bushing is embodied so that in a zone/zones adjoining the shock absorber covers, the inner bushing cavity comprises along the bushing length at least two sections and at each of the sections the bushing inner diameter along the section length (in the direction from the piston cover to the rod cover) decreases to the length of the minimum bushing inner diameter at this section and increases to the value of bushing maximum inner diameter at this section. The technical result is a substantial increase of force counteracting the piston motion in the bushing in sections adjoining the shock absorbers covers; operating two lateral sealing surfaces when moving the piston in said sections.
Patent EA-019986-B1 (EA)
Title: Installation for the extraction of fluid from an expanse of water and method for disconnecting same
Inventor: CROME TIMOTHY JOHN
IPC: B63B21/50
Filed: 2009-06-09
Abstract: This installation comprises an upper structure (12), and a flexible hose (16) capable of moving through the expanse of water (11B) between an upper connected configuration and a lower disconnected configuration. The installation comprises a lower structure (14) having a base (60) extending at a distance from the bottom (11A) of the expanse of water (11B). The upper structure (12) is capable of moving relative to the lower structure (14) between an extraction position and an evacuation position. The base (60) defines a passage (68) for travel of the flexible hose (16) as it moves between the upper connected configuration and the lower disconnected configuration and a stop (74) for retaining a connection head (92) of the hose (14), disposed in the travel passage (68), to keep the connection head (92) at a distance from the bottom (11A) of the expanse of water (11B) in the lower disconnected configuration.
Patent EA-019901-B1 (EA)
Title: Carbamoyl derivatives of bicyclic carbonylamino-pyrazoles as prodrugs
Inventor: POLUCCI PAOLO
IPC: A61K31/416
Filed: 2009-05-14
Abstract: There are provided bicyclic carbonylamino-pyrazoles of formula (I), wherein the variables are as specified in the claims, for use as medicament, in particular for the treatment of diseases due to the malfunctioning of protein kinases (PKs), such as cancer, pharmaceutical compositions comprising such carbamoyl derivatives, and their use as prodrugs of therapeutically active agents. Method of treatment and some new bicyclic carbonylamino-pyrazoles are also object of the present invention.
Patent EA-020675-B1 (EA)
Title: Ventilation insert for clothing that protects against blood-sucking and stinging insects
Inventor: CHEPIK ALIAKSEI ANDREEVICH
IPC: A41D31/02
Filed: 2010-11-25
Abstract: The invention relates to elements of protective clothing and can be used to protect a person against blood-sucking and stinging insects. In particular, the invention may be widely used for protecting beekeepers against bee stings while they work. The ventilation insert for clothing that protects against blood-sucking and stinging insects is in the form of an insulating system having a thickness greater than the length of the proboscis or the sting of an insect, and is comprised of three layers. The outside layer and the inside lining and anchoring layer are made of a mesh material; the middle layer is made up of cells in the shape of prisms, the area of the bases of which is greater than the area of a cell of the mesh of the outside layer. Using the claimed design for a ventilation insert in clothing that protects against blood-sucking and stinging insects makes it possible to improve the reliability, durability and ventilation efficiency of such clothing and provide for the easy manufacture, repair, use and storage thereof as well as a reduction in its cost.
Patent EA-022690-B1 (EA)
Title: Imidazopyridine derivatives, process for the preparation thereof and therapeutic use thereof
Inventor: ALCOUFFE CHANTAL
IPC: C07D471/04
Filed: 2011-07-04
Abstract: The invention relates to compounds corresponding to formula (I)in which Rand Rtogether form, with the carbon atoms of the phenyl nucleus to which they are attached, a 6-membered nitrogenous heterocycle corresponding to one of formulae (A), (B) or (C) belowin which the wavy lines represent the phenyl nucleus to which Rand Rare attached. The invention also relates to a preparation process and therapeutic use of the compounds.
Patent EA-035973-B1 (EA)
Title: Amino acid sequences directed against il-17a, il-17f and/or il-17a/f and polypeptides comprising the same
Inventor: ROMMELAERE HEIDI
IPC: C07K16/46
Filed: 2012-05-04
Abstract: The present invention relates to a polypeptide which specifically binds to human IL-17A, human IL-17F and/or human IL-17A/F, to the use of such polypeptide, to a method of treating a disease and to a pharmaceutical composition comprising the same. The polypeptide is useful in treating a disease selected from the group consisting of systemic lupus erythematosis, rheumatoid arthritis, osteoarthritis, juvenile chronic arthritis, spondyloarthropathies, systemic sclerosis, idiopathic inflammatory myopathies, Sjogren's syndrome, systemic vasculitis, sarcoidosis, autoimmune hemolytic anemia, autoimmune thrombocytopenia, thyroiditis, diabetes mellitus, immune-mediated renal diseases, demyelinating diseases of the central and peripheral nervous systems such as multiple sclerosis, idiopathic demyelinating polyneuropathy or Guillain-Barre syndrome and chronic inflammatory demyelinating polyneuropathy, hepatobiliary diseases such as infectious autoimmune chronic active hepatitis, primary biliary cirrhosis, granulomatous hepatitis and sclerosing cholangitis, inflammatory bowel disease, gluten-sensitive enteropathy and Whipple's disease, autoimmune or immune-mediated skin diseases including bullous skin diseases, erythema multiforme and contact dermatitis, psoriasis, allergic diseases such as asthma, allergic rhinitis, atopic dermatitis, food hypersensitivity and urticaria, immunologic diseases of the lung such as eosinophilic pneumonia, idiopathic pulmonary fibrosis and hypersensitivity pneumonitis, transplantation associated diseases including graft rejection and graft-versus-host-disease.
Patent EA-026848-B1 (EA)
Title: Antiviral compounds
Inventor: RANDOLPH JOHN T
IPC: C07D405/14
Filed: 2010-06-10
Abstract: Compounds effective in inhibiting replication of Hepatitis C virus ("HCV") are described This invention relates to processes of making such compounds, compositions comprising such compounds, and methods of using such compounds to treat HCV infection.
Patent EA-025531-B1 (EA)
Title: Dimethyl-benzoic acids
Inventor: BLANCO-PILLADO MARIA-JESUS
IPC: C07D401/04
Filed: 2013-06-20
Abstract: Described is a compound of the Formula IIwherein A isRis CH, CF, or F; Ris H, CH, or F; Ris CH, OCH, OH, F; Ris OH or CHOH; and X is CH or N; or a pharmaceutically acceptable salts thereof.
Patent EA-028261-B1 (EA)
Title: Combustion process for fuel containing vanadium compounds
Inventor: MALAVASI MASSIMO PIETRO
IPC: F23L7/00
Filed: 2013-07-22
Abstract: A process of fuel combustion in the presence of catalyst for producing energy wherein low ranking gaseous, liquid, solid, optionally solid melting hydrocarbon fractions are used as fuels, having a vanadium content in the amount by weight from 50 to 500 ppm or higher, and alkaline metals Ma in the amount from 20 to 10,000 ppm, wherein magnesium is added as oxide, or as a magnesium compound forming MgO in the combustion process, or a mixture thereof and a silico-aluminate is added wherein the molar ratio SiO:AlOis from 2:1 to 6:1; the combustor being refractored, isotherm or quasi-isotherm, flameless, working at a temperature 1,250-1,450°C and under pressurized conditions, wherein the oxidant is used in admixture with water or steam, the ratio by moles oxidant:(water/steam) being between about 1:0.4 and about 1:3, or the oxidant is used in admixture with flue gases recycled from the flue gases outletting the energy recovery equipments, wherein the water/steam amount is higher than 30% by volume, optionally adding water to the recycled flue or combustion gases wherein the molar ratio oxidant:(water/steam) in flue gases is from about 1:0.4 to about 1:3; the hydrocarbon fraction being fed in admixture with water or steam, the amount of water/steam being at least 30 wt.% with respect to the hydrocarbon fraction.
Patent EA-034447-B1 (EA)
Title: Method for producing beverages by acid removal
Inventor: DONALDSON IAIN
IPC: A23L2/38
Filed: 2013-06-28
Abstract: The present invention relates to methods for producing beverages with low levels of acids, cations and/or sugars. The methods comprise the step of removing acidic ions through an AX-REED membrane stack and optionally removing cations through a CX-REED membrane stack. In certain embodiments, the AX-REED and the CX-REEF membrane stacks are operated in parallel. The methods may also comprise a step of converting sugar to organic acid, while simultaneously removing the generated organic acid through the AX-REED membrane stack. The sugar may for example be converted with the aid of enzymes and/or microorganisms.
Patent EA-033675-B1 (EA)
Title: System and method for automated conversion of interactive sites and applications to support mobile and other display environments
Inventor: BEN-AHARON RONI
IPC: G06F40/143
Filed: 2014-09-11
Abstract: A system and a method for convertion of a website page layout in a website building system having at least one processor to process instructions, a preprocessor including a receiver to receive a website page from a website building system, the page having a source layout for a source display area and the page having an object model representation of components, and orderers to determine an order and set of relationships among the components and to create a target layout of the website page for a target display area, the target layout being based on a semantic analysis and reconciliation of the determined order and set of relationships and where the source display area has different attributes than the target display area.
Patent EA-035798-B1 (EA)
Title: Method to treat or prevent cataract
Inventor: ZHANG KANG
IPC: A61K31/56
Filed: 2015-08-24
Abstract: The present invention relates to pharmacology, namely to treating ophthalmic diseases. Provided is a method of treating or preventing cataract in a subject in need thereof, comprising administering in the eye of said subject a composition comprising a pharmaceutically acceptable carrier and a pharmaceutically effective amount of lanosterol. Lanosterol inhibits crystallin protein aggregation or dissolves crystallin protein aggregate.
Patent EA-039738-B1 (EA)
Title: Method and device for executing an e-vaping device operating system, e-vaping programming language, and e-vaping application programming interface
Inventor: JUSTER BERNARD C
IPC: A24F40/90
Filed: 2015-11-25
Abstract: An electronic vaping device includes a housing extending in a longitudinal direction, the housing including a mouth-end and a connection-end, a reservoir containing a pre-vapor formulation, the reservoir in the housing, a heating element in the housing, the heating element in fluid communication with the reservoir, the heating element configured to generate a vapor, and a rechargeable battery configured to power at least the heating element and any other potential power consuming element(s) such as electronic circuits. The electronic vaping device also includes a first memory having stored thereon computer readable instructions relating to an electronic vaping operating system (OS), and at least one processor configured to execute the OS computer readable instructions to execute the operating system, the operating system including a real-time kernel configured to operate the electronic vaping device, and execute object code related to electronic vaping device functionality.
Patent EA-037569-B1 (EA)
Title: Salts of monobactam antibiotic and use thereof
Inventor: AUBIN ERIC
IPC: A61K31/427
Filed: 2016-09-20
Abstract: The invention relates to a disodium and double (L)-arginine salt of 1-(((Z)-(1-(2-aminothiazol-4-yl)-2-oxo-2-(((3S,4R)-2-oxo-4-((2-oxooxazolidin-3-yl)methyl)-1-sulfoazetidin-3-yl)amino)ethylidene)amino)oxy)cyclopropanecarboxylic acid (referred to herein as compound X), as well as pharmaceutical compositions comprising these materials and the use thereof in treating a Gram-negative bacterial infection.
Patent ES-2169665-B1 (ES)
Title: Procedimiento para la reparacion de pistas de deporte.
Inventor: LLEWELLYN BUNNELL ROGER
IPC: E01C13/06
Filed: 2000-05-16
Granted: 2003-06-01
Abstract: Procedimiento para la reparación de pistas de deporte. Comprende limpiar la capa superficial con medios mecánicos; aplicar una capa de imprimación de poliuretano [I]; aplicar una capa de un poliuretano de dos componentes [P(2)C]; estando en estado líquido, aplicar un granulado de EPDM de diferente granulometría [EPDM]; dejar secar; y recuperar el granulado no adherido. Alternativamente, puede prepararse una mezcla de poliuretano y EPDM, que se proyecta, primero, en un ángulo; y después, en el ángulo opuesto. Cuando la capa base está muy deteriorada, es decir presenta una adherencia inferior a 0,2 N/mm2, se procede al arranque de dicha capa base; se aplica una capa de imprimación de poliuretano monocomponente en el asfalto y superficie perimetral; y se aplica una capa base de dureza semejante a la zona no afectada. La capa superficial se aplica de acuerdo con lo descrito más arriba.
Patent ES-2161654-B1 (ES)
Title: Armario frigorifico de absorcion.
Inventor: SCHWARZPAUL UWE
IPC: F25B49/04
Filed: 2000-06-05
Granted: 2002-07-01
Abstract: Armario frigorífico de absorción, que comprende: - un circuito 7 cerrado de enfriamiento para el enfriamiento de una cámara 3 frigorífica, circuito 7 que posee un evaporador 9 dispuesto en la cámara 3 frigorífica, -un dispositivo 23 de mando para suministrar al circuito 7 cerrado de enfriamiento un valor P de potencia. - un sensor 27 de temperatura para suministrar al dispositivo 23 de mando un valor v{sub,e} de medida de la temperatura, - un temporizador 29 para suministrar al dispositivo 23 de mando un primer intervalo t{sub,1}, t{sub,2} de tiempo prefijado y un segundo intervalo t{sub,3}, t{sub,4} de tiempo prefijado - el dispositivo 23 de mando suministra unos primero (P{sub,1}) y segundo (P{sub,2}) valores de potencia, - y el dispositivo 23 de mando registra al comienzo t{sub,3} del segundo intervalo de tiempo un primer valor v{sub,1} de temperatura y al final t{sub,4} del segundo intervalo de tiempo registra un segundo valor v{sub,2} de temperatura y genera en caso necesario una señalS de avería.
Patent ES-2172451-B1 (ES)
Title: Mueble para usos multiples.
Inventor: SORIO VELA JOAQUIN
IPC: A47B85/00
Filed: 2000-12-14
Granted: 2003-12-16
Abstract: Mueble para usos múltiples. El mueble comprende un armazón de asiento, dotado de ruedas giratorias inferiores y que delimitan un volumen utilizable para disponer objetos y presentando asociadas con los montantes de su respaldo, sendas guías verticales alargadas destinadas a recibir los pivotes de guiado de una tabla de plancha, susceptible en la posición de desplazamiento vertical máximo, de bascular horizontalmente, quedando apoyada por su parte media en topes adyacentes a los extremos superiores de las guías y por su parte delantera, en el extremo libre de la placa constitutiva del asiento que es basculante alrededor de un eje situado en la parte frontal del armazón.
Patent ES-2193877-B1 (ES)
Title: Lampara decorativa.
Inventor: DE LA BARRERA-MONTENEGRO MENDE
IPC: B44F1/06
Filed: 2002-04-15
Granted: 2005-03-01
Abstract: La lámpara decorativa está constituida por un receptáculo, principalmente una esfera (2), translúcido o transparente en el que se genera una figura poligonal bidimensional o tridimensional mediante un haz láser generado por un puntero emisor (3). El haz o bien es reflejado mediante espejos (6) situados en los vértices de la poligonal que conforma la figura o bien es refractado mediante prismas (5) capaces de dividir el haz en dos o más aristas. El haz o los haces que han completado su recorrido son eliminados mediante la inclusión de esferas (8). Es posible el cambio de color en un punto intermedio mediante el uso de filtros (7) y la visualización del haz láser se consigue con una atmósfera controlada que contiene partículas (9) en suspensión movidas por un ventilador (4) o bien con un líquido.
Patent ES-2198225-B1 (ES)
Title: Proceso de mecanizado de precision para diametros interiores de orificios en cigueñales y maquina para dicho proceso.
Inventor: GABILONDO PENALBA JOSE JUAN
IPC: B23C3/02
Filed: 2002-07-12
Granted: 2005-04-01
Abstract: Proceso de mecanizado de precisión para diámetros interiores de orificios en cigüeñales y máquina para dicho proceso, en el que el cigüeñal es sujetado, por un extremo, por medios que originan a su vez el giro del cigüeñal sobre el eje Z y por su otro extremo por una luneta dispuesta en las cercanías de la brida; disponiéndose enfrentada a la brida según el eje Z una unidad de mecanizado con un cabezal de fresar con un husillo portador de una fresa que dispone al menos de movimiento longitudinal según los ejes (X, Z) ó (Y, Z); procediéndose a girar el cigüeñal a menos de 50 rpm. con una primera fase con arranque de viruta según el eje X ó Y con la fresa girando sobre su eje sin desplazamiento longitudinal de la fresa; y una segunda fase con arranque de viruta con la fresa girando sobre su eje y con desplazamiento longitudinal según el eje Z. De aplicación en máquinas herramientas.
Patent ES-2220186-B1 (ES)
Title: Cetarea portatil.
Inventor: GONZALEZ Y DAVID MAR
IPC: A01K63/02
Filed: 2002-08-02
Granted: 2006-05-16
Abstract: Cetárea portátil que consiste en un recipiente compartimentado interiormente mediante filtros (4) que actúan de soporte de los envases (10), presentando una pluralidad de canalizaciones (2) con boquillas (3) para la entrada del agua reciclada al interior, impulsada por una bomba (6) y contando con un depósito (5) para la incorporación de los residuos extraídos.
Patent ES-2224866-B1 (ES)
Title: Dispositivo para la formacion de juntas en obras de hormigon.
Inventor: VAZQUEZ RUIZ DEL ARBOL JOSE RA
IPC: E01C11/04
Filed: 2003-07-17
Granted: 2007-04-16
Abstract: Dispositivo para la formación de juntas de retracción en obras de hormigón constituido por una pluralidad de bandejas de un material separador del hormigón montadas en elementos lineales rígidos de manera alternada a un lado y otro de la línea superficial de fisura en la cara superior de la superficie hormigonada y dejando espacios libres entre ellas para permitir la fisuración. El dispositivo propicia el empotramiento de las losas contiguas formadas por la junta de retracción con la consiguiente mejora del comportamiento resistente. Es de aplicación en obras de hormigón in situ tales como carreteras, canales, explanadas, colectores, túneles, ferrocarriles, diques y otras.
Patent ES-2229948-B1 (ES)
Title: Preparacion de monoesteres de acidos grasos.
Inventor: CORMA CANOS AVELINO
IPC: C07C67/03
Filed: 2003-10-14
Granted: 2006-07-01
Abstract: Preparación de monoésteres de ácidos grasos. En la presente invención se describe un procedimiento para la obtención de selectiva de monoésteres de ácidos grasos y alcoholes polihidroxílicos por transesterificación entre alcoholes polihidroxílicos, preferentemente glicerina, y triglicéridos de origen animal o vegetal (aceites de colza, palma, coco, girasol etc) o ésteres metílicos derivados de ácidos grasos que poseen entre 10 y 32 átomos de carbono. Los catalizadores básicos heterogéneos que se utilizan en este proceso son óxidos mixtos de un metal trivalente y un metal monovalente, óxidos mixtos de un metal trivalente y un metal divalente que se someten a un proceso de rehidratación previo a su utilización como catalizadores básicos, y alúmina impregnada con sales de metales alcalinos que tras su calcinación dan lugar al óxido correspondiente soportado sobre la alúmina.
Patent ES-2221815-B1 (ES)
Title: Composicion insecticida microencapsulada.
Inventor: INUI KEIICHIRO
IPC: A01N25/28
Filed: 2003-11-07
Granted: 2006-03-01
Abstract: Una composición insecticida microencapsulada, que comprende una piretrina encapsulada en una pared formada por un polímero sintético y que tiene un diámetro medio de partícula de 5 a 100 {mi}m y tiene un espesor de 0,03 a 1 {mi}m, es eficaz para control de insectos.