baber/WOPTO huggingface dataset:
Patent NZ-709248-A (NZ)
Title: Substituted pyridine-2-carboxamide compounds as apoptosis signal-regulating kinase inhibitors
Inventor: NOTTE GREGORY
IPC: C07D417/14
Filed: 2013-12-20
Abstract: The present invention relates to compounds of Formula (I) wherein variables are as defined above. The compounds have apoptosis signal-regulating kinase (”ASKl”) inhibitory activity, and are thus useful in the treatment of ASKl -mediated conditions, including autoimmune disorders, inflammatory diseases, cardiovascular diseases, diabetes, diabetic nephropathy, cardio-renal diseases, including kidney disease, fibrotic diseases, respiratory diseases, COPD, idiopathic pulmonary fibrosis, acute lung injury, acute and chronic liver diseases, and neurodegenerative diseases.
Patent NZ-714519-A (NZ)
Title: Thieno[3,2-d]pyrimidines derivatives for the treatment of viral infections
Inventor: RABOISSON PIERRE JEAN-MARIE BERNARD
IPC: C07D495/04
Filed: 2014-07-29
Abstract: This invention relates to thieno[3,2-d]pyrimidine derivatives of formula (I), processes for their preparation, pharmaceutical compositions, and their use in treating viral infections.
Patent NZ-716218-A (NZ)
Title: Water-resistant composition for adsorbing volatile organic compounds
Inventor: SMITH ANDREW WILLIAM JOHN
IPC: C08L29/04
Filed: 2014-06-25
Abstract: The present invention provides a water-resistant composition for adsorbing volatile organic compounds (VOCs) derived from organic matter comprising: a) palladium doped hydrogen-ZSM-5, wherein the Si:AI ratio of the hydrogen-ZSM-5 is less than or equal to 200:1; and b) at least one water-soluble binder, wherein the water-soluble binder is selected from the group consisting of: at least one polyvinyl alcohol having a Mw from 80,000 to 215,000 and a degree of hydrolysis ≥ 80% or having a Mw of 27,000 and a degree of hydrolysis of 98%. The invention also provides the use of the water-resistant composition for adsorbing volatile organic compounds (VOCs) derived from organic matter, such as where fruit, vegetables, plants and/or cut flowers are contained in a storage container or package.
Patent NZ-717504-A (NZ)
Title: Methods of treatment of cancer by continuous infusion of coenzyme q10
Inventor: NARAIN NIVEN
IPC: A61K9/107
Filed: 2014-09-04
Abstract: The invention provides regimens and methods for the treatment of cancer comprising continuous infusion of coenzyme QIO. The coenzyme QIO may be administered as a monotherapy, or in combination with an additional agent, such as an anticancer agent, a chemotherapeutic agent, or an anti- angiogenic agent. The coenzyme QIO may be administered at two or more different rates. A specific embodiment requires use of a composition comprising a therapeutically effective amount of coenzyme Q10 in the manufacture of a medicament for treating cancer in a subject, wherein the composition comprising coenzyme Q10 is to be administered to the subject by continuous intravenous infusion for at least 48 hours. A further embodiment requires use of a composition comprising a therapeutically effective amount of coenzyme Q10 in the manufacture of a medicament for increasing therapeutic index of intravenously administered coenzyme Q10 in the treatment of cancer, wherein time of infusion of a dose of coenzyme Q10 is increased from no more than 6 hours to a continuous intravenous infusion for at least 48 hours.
Patent NZ-718490-A (NZ)
Title: Acylated glucagon analogues
Inventor: TOLBORG JAKOB LIND
IPC: C07K14/605
Filed: 2014-10-17
Abstract: The invention provides materials and methods for the treatment of obesity and excess weight, diabetes, and other associated metabolic disorders. In particular, the invention provides novel acylated glucagon analogue peptides effective in such methods. The peptides may mediate their effect by having increased selectivity for the GLP-1 receptor as compared to human glucagon. In particular, the acylated glucagon analogues are modified at a particular residue by addition of a side chain comprising a fatty acid having a polar group at one end, connected to the peptide backbone via a spacer.
Patent NZ-724064-A (NZ)
Title: Functionally-modified oligonucleotides and subunits thereof
Inventor: HANSON GUNNAR
IPC: C07H21/00
Filed: 2012-11-15
Abstract: Disclosed herein are functionally-modified oligonucleotide analogues of formula I where the substituents are as defined herein, comprising modified intersubunit linkages and/or modified 3’ and/or 5’-end groups. The disclosed compounds are useful for the treatment of diseases where inhibition of protein expression or correction of aberrant mRNA splice products produces beneficial therapeutic effects.
Patent NZ-730730-A (NZ)
Title: Novel carboxylic acid compounds useful for inhibiting microsomal prostaglandin e2 synthase-1
Inventor: FISHER MATTHEW JOSEPH
IPC: A61P29/00
Filed: 2015-10-22
Abstract: The present invention provides compounds of Formula 1, or a pharmaceutically acceptable salts, thereof, where R, X, A, E, and G are as described herein, methods of preparing the compounds, and use of the compounds to treat pain and/or inflammation.
Patent NZ-741042-A (NZ)
Title: Method and apparatus for emergency braking performance testing, evaluation and/or driver training
Inventor: HARDY CHRISTOPHER
IPC: G01L5/28
Filed: 2016-09-21
Abstract: The present invention relates to the evaluation of drivers of motorised wheeled vehicles including a system for evaluation of driver braking performance under emergency conditions, comprising: a driver measuring unit including a force measuring means and a communication means, the driver measuring unit adapted for attachment to a road vehicle brake applicator interface and generating force measurement data representative of force applied by the driver to the brake applicator during an evaluation period and transmit the force measurement data using the communications means; a vehicle measuring unit, carried by the vehicle, having a motion measuring means adapted to determine vehicle measurements comprising one or more of the vehicle acceleration, velocity and position, and a communication means, the vehicle measuring means generating vehicle measurement data during an evaluation period and transmit the vehicle measurement data using the communications means; and a processor unit having a display screen, and communications means, wherein the processor unit receiving via the communications means the force measurement data generated by the driver measuring unit and the vehicle measurement data generated by the vehicle measuring unit, and generate brake test result metrics therefrom for display on the display screen; the force measurement data provides a timing trigger for the evaluation period; the motion measuring means combines an inertial measurement unit for determining acceleration/deceleration measurements and a GPS receiver configured for determining one or a combination of distance/positional measurements and velocity measurements based on the Doppler-effect on a GPS carrier signal; and the processor unit enables selection of braking test parameters and provides signals to the driver during a braking test procedure for the driver to act upon the provided signals and the braking test result metrics comprise one or a combination of: driver reaction time; vehicle stop time; vehicle stop distance; brake pedal force; vehicle acceleration/deceleration; and, vehicle speed.
Patent NZ-772299-A (NZ)
Title: Boundary block partitioning in video coding
Inventor: CHEN JIANLE
IPC: H04N19/70
Filed: 2019-06-27
Abstract: A partitioning method comprises determining whether a current block of a picture is a boundary block and whether the size of the current block is larger than a minimum allowed quadtree leaf node size; and if the current block is the boundary block and the size of the current block is not larger than the minimum allowed quadtree leaf node size (MinQTSize), applying forced binary tree (BT) partitioning to the current block. A method comprises making a determination that a current block of a picture is a boundary block and that a size of the current block is less than or equal to a minimum allowed quadtree (QT) leaf node size (MinQTSize); and applying, in response to the determination, forced binary tree (BT) partitioning to the current block.
Patent PT-117287-A (PT)
Title: Biodispositivo biomimético inteligente e seu uso
Inventor: ARTUR JORGE DOS SANTOS MATEUS
IPC: A61M5/00
Filed: 2021-06-14
Abstract: A PRESENTE INVENÇÃO FAZ REFERÊNCIA A UM BIODISPOSITIVO BIOMIMÉTICO INTELIGENTE (18), O QUAL É CONFIGURADO PARA SE COMUNICAR E ATIVAR, POR MEIO DE ESTÍMULO ELÉTRICO E MAGNÉTICO, PARTÍCULAS INCORPORADAS EM MODELOS TRIDIMENSIONAIS (19) QUE APRESENTAM PROPRIEDADES QUE VARIAM DE ACORDO COM O USO PRETENDIDO. O REFERIDO BIODISPOSITIVO (18) É UTILIZADO NA PREVENÇÃO E NO TRATAMENTO DE DOENÇAS ASSOCIADAS AO SISTEMA ESQUELÉTICO, POR MEIO DA ATIVAÇÃO DAS PARTÍCULAS E DA LIBERTAÇÃO DOS AGENTES TERAPÊUTICOS. AINDA, É ÚTIL NO ACOMPANHAMENTO DA EVOLUÇÃO DO PROCESSO DE REGENERAÇÃO, PELA MONITORIZAÇÃO DE INDICADORES ESPECÍFICOS (TAIS COMO FORÇA, PH, OXIGÉNIO, TEMPERATURA E / OU BIOMARCADORES). A INVENÇÃO SURGE COMO UMA ALTERNATIVA TERAPÊUTICA PARA O TRATAMENTO DE ENFERMIDADES ASSOCIADAS À DEGENERAÇÃO ÓSSEA E, AINDA, RESOLVE OS PROBLEMAS REFERENTES À NECESSIDADE DE MONITORIZAÇÃO E / OU CONTROLO EM TEMPO REAL DO TRATAMENTO ESCOLHIDO PARA A ENFERMIDADE A SER TRATADA.
Patent RU-94009883-A (RU)
Inventor: OKUNEV G KH
IPC: B64C25/50
Filed: 1994-03-22
Abstract: FIELD: landing gear control devices. SUBSTANCE: device has actuating mechanism 2 and control unit having housing 3 where distributing device 7, safety valves 8, replenishing check valves 9 and sleeve 10 are mounted. Spring-loaded spool valve 11 of change-over valve is mounted in sleeve 10. Control unit is provided with adjustable stop 13 of spool valve 11 of change-over valve mounted in housing 3 and used for motion of spool valve 11 relative to sleeve 10. EFFECT: enhanced efficiency of dampening wheel shimmy and facilitated manufacture of landing gear legs.
Patent RU-94012932-A (RU)
Inventor: POL G SERUDZHI
IPC: B29C55/08
Filed: 1994-04-18
Abstract: FIELD: metallurgy, apparatus for material motion inside furnaces. SUBSTANCE: each nozzle has fixed part and at least one telescopic part, that is moved sliding inside fixed part. Contact of metal to metal is prevented, that allows nozzles to operate under high temperatures. Nozzle outlet hole configuration is changeable easily to produce air cutter depending on separate needs. Each nozzle does not depend on others. It allows to simplify process of furnaces fitting with nozzles and operation of each nozzle. EFFECT: simplified operation of each nozzle and fitting furnaces with nozzles.
Patent RU-94013555-A (RU)
Inventor: GINKULOV G V
IPC: F03B17/00
Filed: 1994-04-13
Abstract: FIELD: year-round source of mechanical energy at any depth of river in construction of damless hydroelectric stations for rotating generator rotors. SUBSTANCE: propeller consists on one part which may be cut or stamped from flexible material, for example, rubberized cord or synthetic cloth. Form of part is presented in Fig. 2. When this part is in folded state, turbine is formed with three ladle-shaped blades located at an angle of 120 deg relative to one another and pressure of water flow acting on one blade and reflecting from it acts simultaneously on blade in front of it, thus providing for considerable resulting torque of propeller. But this torque may be increased by "n" times if "n" number of such propellers form string (by two ropes) which is actually drive shaft rotating the rotor of high-power generator for damless hydroelectric station. EFFECT: low-cost electric power, enhanced efficiency and reduced usage of materials for manufacture of propellers.
Patent RU-94024388-A (RU)
Inventor: DVORJANKOV V A
IPC: A23L17/50
Filed: 1994-06-29
Abstract: FIELD: fish industry, in particular, preparing of semi-finished product from marine products in public catering enterprises and enterprises using invalid diet as well as food for people living in radioactive contaminated zones. SUBSTANCE: method involves preparing stuffing in two stages; mincing product at the first stage and holding minced mass in refrigeration chamber at temperature not below -5 C until crystallization process is initiated; introducing additives into minced mass at the second stage and repeatedly cooling cutlet mass at temperature ranging from 0 C to -3 C for 6-12 hours; effectuating dewatering by forced blowing of basic raw material with countercurrent air flows; conducting thermal treatment of formed products by blanching in water-salt solution for 2-2.5 min and freezing formed products. EFFECT: improved quality and wider range of products of medicated and prophylactic action and those satisfying human being requirements for microelements.
Patent RU-94025750-A (RU)
Inventor: ZHENCHEVSKIJ R A
IPC: A61B17/00
Filed: 1994-07-11
Abstract: FIELD: medicine; surgery. SUBSTANCE: method involves slanting cross dissection of the empty intestine, low placement of the anastomosis, fixation of the intestine on the back wall of the stomach stump, and positioning the anastomosis horizontally level with the duodenum. EFFECT: more favorable physiological conditions for passage of food chyme; reflux into stomach stump.
Patent RU-94026967-A (RU)
Inventor: PAVLENKO G I
IPC: B05B7/00
Filed: 1994-07-15
Abstract: FIELD: heating engineering, method and apparatus are used in process of watered fuel sprays burning in particular. SUBSTANCE: method of liquid mediums preparations for spraying provides for pressurized liquid medium feeding and its gas impregnation before spraying. New thing in the method is the fact, that liquid medium gas impregnation is exercised by electrolysis of its components disintegrated for gas-shaped components. In the case as liquid medium they use watered fuel, gas impregnation of which is exercised by electrolytic disintegration, of water being component of the liquid medium. For example, water-coal suspension or water residual oil emulsion are used as watered fuel. Apparatus for realization of method of liquid mediums preparation for spraying has body, branch pipe to feed liquid medium and liquid medium gas impregnation block. New thing in the method is that structure of liquid medium gas impregnation block is made in the form of two pipes coaxially mounted inside body and connected to direct current source. EFFECT: method allows to decrease production costs, to increase reliability of apparatus.
Patent RU-94029671-A (RU)
Inventor: RAJNER KHANS TRABER
IPC: D06L4/30
Filed: 1994-08-19
Abstract: FIELD: textile industry. SUBSTANCE: reducing bleaching composition not containing phosphate contains reducing bleacher and bleaching stabilizer taken from citric acid derivative, homo-or copolymer of ethylene-saturated mono-or dicarbonic acids, water-soluble magnesium salt and tetraborate of alkali metal. Bleaching composition is suitable for reducing bleaching of fibers of vegetable and animal origin or synthetic fibers, and also of paper. EFFECT: higher degree of whiteness and provision of safety for environment.
Patent RU-94031173-A (RU)
Inventor: IVANOV V I
IPC: G06F1/16
Filed: 1994-08-15
Abstract: FIELD: computer engineering. SUBSTANCE: device has (m+1) identical processors, m memory units, (m+1) commutators for information input and output, comparison unit with input commutator and control unit. (m- 2) identical processors, (m-2) memory units, (m-3) commutators for information input and output are introduced to accomplish the goal of invention. One additional processor in each clock cycle is connected to subsequent memory unit and operates in parallel with processor which is assigned to this memory unit. When results of processing differ for pair of mutually checked processors, storage of information to memory unit is locked and output of new instructions from memory unit is also locked. Operations of the same pair of processors are repeated again. Device may be used in design of fault-tolerant computing systems using lesser number of additional processors due to elimination of restriction of redundant processors and control units in redundant groups of two basic and one additional processors. EFFECT: decreased number of redundant units while reliability level remains same, increased validity of operations when short interrupts occurs and built-in check of processors has low validity.
Patent RU-94032465-A (RU)
Inventor: FEDOSOV A A
IPC: B06B1/16
Filed: 1994-09-06
Abstract: FIELD: creation of artificial vibrations for vibration packing, withdrawal of models in moulding, pressing mixtures, construction of roads, road-rollers. SUBSTANCE: vibrator has drive and hollow unbalanced mass connected with it; hollow unbalanced mass is divided into chambers and is partially filled with liquid; chambers are brought in communication through holes provided in partitions; area of these holes may be adjusted. Device for control of vibrator has buttons for manual start and stop and vibration sensor whose normally open contact is connected to control circuit so that vibrator should be automatically switched off upon completion of vibration. Mode of operation machine may be changed without attendance every time when vibrator is switched on. EFFECT: enhanced reliability. 3 cl, 3 dwg
Patent RU-94033705-A (RU)
Inventor: GOMOZOV V V
IPC: F25J3/04
Filed: 1994-09-15
Abstract: FIELD: separation of gas mixtures. SUBSTANCE: method may be used for production of pure nitrogen and enriched air at concentration of oxygen satisfying the requirements of customer at minimum power requirements. Liquid products of separation of air (oxygen or nitrogen) may be also obtained in small amounts. Production of pure nitrogen under pressure by single-stage rectification provides for reduction of power requirements as compared with type A-8 scheme due to introduction of additional condenser-evaporator which reduces amount of circulating gas. Evaporation of enriched air is effected due to condensing of part of air directed for separation from main heat exchange unit. Expansion turbine and refrigerant compressor may be mounted on common shaft. Such version may be used for serial production of new generation of air separation plants, type A-8 (or A-6) at saving of power up to 10 percent. New air separation plants for production of enriched air and pure nitrogen will be based on single scheme at nearly complete unification of equipment. EFFECT: enhanced reliability and improved quality.
Patent RU-94037763-A (RU)
Inventor: DEHVID S UAJT
IPC: D21C9/10
Filed: 1992-04-24
Abstract: FIELD: device and method for bleaching of highly consistent lignocellulose pulp with use of ozone as component of ozone-containing gas. SUBSTANCE: the offered reactor device is essentially a cylindrical vessel 42A, 42B with rotating shaft 48B from which blades 52B or some other transmitting members are arranged in radial direction so as to minimize dispersion of pulp in axial direction and to attain maximum dispersing in radial direction and to provide passing the flow through the reactor of dispersed in radial direction pulp in plug mode in the presence of ozone with the aim to produce, essentially, the uniformly bleached pulp. EFFECT: higher efficiency. 1 dwg
Patent RU-94039343-A (RU)
Inventor: REBROV A K
IPC: F04F9/02
Filed: 1994-10-14
Abstract: FIELD: pump engineering. SUBSTANCE: pump has cylindrical housing and steam pipe line with an active Laval nozzle. The housing and steam pipe line are axially alined. The outer wall is converging in the direction to the nozzle exit. A cooled shield is mounted concentrically and with a spaced relation to the nozzle. The shield is protected from the top by a hot screen to exclude molecular flow in the housing from the slot between the nozzle wall and shield and from the surface of the shield as well. EFFECT: expanded functional capabilities.
Patent RU-94040143-A (RU)
Inventor: GANS VEBER
IPC: C08G18/66
Filed: 1994-11-03
Abstract: FIELD: production of cellular polyurethane mold articles. SUBSTANCE: interaction of polyisocyanate component (content of isocyanate groups in it being 18-33.6 weight %) with polyol component (its average hydroxyl functionality being 2-3) and with at least one bifunctional compound having molecular weight 62-1999 is carried out. Quantity of mentioned above third component is 2-15 % of said second component. At least one polyisocyanate or mixture of polyisocyanates of diphenylmethane series which is modified if it is necessary is used as mentioned above polyisocyanate component. At least one polyether polyol having molecular weight 2000-10000 and/or one polyester polyol having molecular weight 2000-10000 is used as mentioned above polyol component. Interaction of these components is carried out in the presence of blowing agent or other means. Carbamates having common formulawhere Ris hydrogen, alkyl with 1-5 carbon atoms or residue having common formulawhere Rand Rbeing the same or different are hydrogen or alkyl with 1-3 carbon atoms, and n is integer 2-6 are used as mentioned above blowing agents. EFFECT: improves efficiency of the method.
Patent RU-94042363-A (RU)
Inventor: CHUPROV V P
IPC: E21B47/12
Filed: 1994-11-29
Abstract: FIELD: well logging; particularly, measurement of downhole parameters in the course of well drilling. SUBSTANCE: system includes drill string, body supply unit, measuring modules, transmitting device modules, electric separator and downhole motor. Diameters of body of measuring modules and power supply unit are smaller than the internal radius of drill string and length l of modules is made equal to, where R is minimum radius of wellbore path; h is half of difference of internal diameter of measuring modules body. Electric separator is made in the form of separate subinstalled directly above downhole motor. Power supply unit, measuring and transmitting modules are interconnected by means of links flexible in radial direction and rigid in longitudinal direction. Links between modules may be in form of flexible in radial direction metal pipes with diameter smaller than diameters of module bodies. Electric cable is located inside pipes and centralizers are installed at ends of pipes. To provide for retrieval of downhole telemetering system from the drill string in emergency situations, electric contact with bottom of drill string is made sliding. EFFECT: higher reliability of well sinking and investigation of well with minor curvature radius, particularly, slim wells.
Patent RU-95101150-A (RU)
Inventor: AJDINOV A M
IPC: C21D1/76
Filed: 1995-01-26
Abstract: FIELD: metallurgy and mechanical engineering; applicable in annealing of electrical steels. SUBSTANCE: method for utilization of atmosphere in tower-type furnaces includes supply of fresh protective atmosphere to heating chambers and holding, withdrawal of used atmosphere and selection of a part of used atmosphere for cleaning, cooling and compression. The part of used atmosphere is selected from gas bleeder of holding chamber and it is returned to heating chamber in the definite amount. Supply of fresh protective atmosphere to heating chamber is discontinued. Total consumption of protective atmosphere is reduced in tower-type furnace by 10-12%. In so doing, potential of used atmosphere fed to heating chamber provides for decarbonization of transformer steel down to preset values by the technology and equalling $$$-0.003-0.004 mas.% upon completion of annealing process (at furnace outlet). EFFECT: higher efficiency.
Patent RU-95103119-A (RU)
Inventor: LEVIN V M
IPC: G09F9/30
Filed: 1995-02-28
Abstract: FIELD: advertising, road signs, stained-glass panels, interiors. SUBSTANCE: device has displaying screen, set of light guides and light source. additional panel is located between displaying screen and light source. One terminals of light guides are connected to light source, another terminal are connected to additional panel, which is located in parallel to displaying screen and spaced from it by 0-150 mm. EFFECT: increased functional capabilities. 1 dwg