baber/WOPTO huggingface dataset:
Patent ES-512441-A0 (ES)
IPC: C07D309/12
Filed: 1982-05-21
Abstract: Compounds of Formula I    <IMAGE>  I  wherein X is oxygen or CH2; A is CH2-CH2, trans-CH=CH or C 3BOND C; W is free or functionally modified hydroxymethylene or free or functionally modified   <IMAGE> and the OH groups may be in the  alpha - or the  beta -position; D is straight chain or branched, saturated or unsaturated hydrocarbon aliphatic of from 1 to 10 carbon atoms, which may be substituted by fluorine; E is C 3BOND C or CR3=CR4, R3 and R4 being different and being hydrogen or alkyl of 1 to 5 carbon atoms; R1 is free or functionally modified hydroxy; and R2 is alkyl, cycloalkyl, optionally substituted aryl or heterocyclic, have valuable pharmacological properties, e.g., hypotensive and bronchodilatory characteristics. They can furthermore be used for prophylaxis and therapy of coronary infarct and as a treatment for stroke. They are produced by means of reduction of the corresponding 1-carbonic acid derivatives.
Patent ES-524907-A0 (ES)
IPC: C07D405/06
Filed: 1983-08-12
Abstract: Compounds of the formula:   <IMAGE>   wherein R1, R2, R3, R4 and R5 each represent a hydrogen atom, a halogen atom, a (C1-4)alkoxy radical, a (C1-4)alkylthio radical, a halogeno(C1-4)alkyl radical, a (C1-4)alkyl radical or a cycloalkyl-alkoxy-alkoxy radical or two of the adjacent R symbols together form a methylenedioxy or ethylenedioxy radical, R6 represents a hydrogen atom, a (C1-4)alkyl radical, a (C3-6)cycloalkyl radical or a (C3-6)cycloalkyl-(C1-4)alkyl radical, and R7, R8 and R9 each represent a hydrogen atom or a methoxy radical, are new compounds possessing pharmacological properties; they are useful as calcium antagonists and as antihypertensives.
Patent ES-532031-A0 (ES)
IPC: B01J31/02
Filed: 1984-04-28
Abstract: The invention relates to a new process for the preparation of 21-hydroxy-20-keto-steroids from 17-(isocyano-sulfonylmethylene)-steroids whereby simultaneously an unsaturated bond is introduced between C16 and C17. Furthermore the invention relates to new intermediate compounds formed in this process nad their preparation and to the ultimately formed 21-hydroxy-20-keto-delta<1><6>-steroids, as far as these latter compounds are new.
Patent ES-541501-A0 (ES)
IPC: H04N9/83
Filed: 1985-03-22
Abstract: The recording apparatus comprises a luminance signal processing circuit (16) for generating a frequency-modulated signal (Yf), a chrominance signal processing circuit (15) for generating a frequency-converted chrominance signal (Cc) with a frequency band lower than the frequency deviation range of the frequency-modulated luminance signal, and an audio signal processing circuit (1-13) for generating a frequency-modulated audio signal including a succession of alternately first and second segments of frequency-modulated signals obtained in response to respectively one and the other of two-channel audio signals; a mixed signal (Sm) obtained by causing the frequency-modulated audio signal (Af min ) to be located between the frequency bands of the frequency-modulated luminance and frequency-converted chrominance signals (Yf, Cc) is supplied to a rotary magnetic head (18a, 18b) to be recorded on a magnetic tape; in the reproducing mode, the audio signal obtained from the magnetic tape is demodulated to produce demodulated outputs of the first and second segments alternately, and the demodulated outputs of the first and second segments are separated from each other and for producing the two-channel audio signals.
Patent ES-544642-A0 (ES)
IPC: C07D517/06
Filed: 1985-06-27
Abstract: A benzoselenino[4, 3, 2-cd] indazole compound having in free base form the following general formula <CHEM>  amd the pharmaceutically acceptable salts thereof, wherein: R7, R8, R9 and R10 independently represent hydrogen, hydroxy or alkoxy of from one to four carbon atoms; R2 is ANR  min R sec  in which A is a straight or branched alkylene chain of from two to five carbon atoms, optionally substituted with hydroxyl and in which R min  and R sec  are independently a hydrogen, a straight or branched alkyl of from one to four carbon atoms, optionally substituted with hydroxyl or R min  and R sec  when taken together, represent the bifunctional radical <CHEM> in which n and m are each, independently, the integer 2 or 3 and B is a direct bond or O, S or NR''' wherein R''' is hydrogen or straight or branched alkyl of from one to four carbon atoms, optionally substituted with hydroxyl; and R5 is nitro, NH2, NHR2 or NHR''' min  wherein R''' min  is a one to four carbon atom acyl radical, a chloroacetyl radical,   -@-Z-NRxRy wherein Z is a straight or branched alkylene chain of from one to four carbon atoms and wherein Rx and Ry are each hydrogen, or a straight or branched alkyl of from one to four carbon atoms optionally substituted with hydroxy, R''' min  is the group <CHEM> Also disclosed are methods for their production and pharmaceutical compositions comprising the compounds. Compounds of the invention have pharmacological properties and are useful antibacterial agents, antifungal agents, and antitumor agents.
Patent ES-545006-A0 (ES)
IPC: A61P25/28
Filed: 1985-07-09
Abstract: 1. Phenylethylaminopropiophenone derivatives of the general formula (I)  see diagramm : EP0167945,P10,F4  in which R**1 represents hydrogen, lower alkyl which is optionally substituted by fluorine, or halogen, R**2 denotes hydrogen or lower alkyl and R**3 denotes hydrogen, alkoxy or halogen, and their physiologically acceptable salts with inorganic or organic acids.
Patent ES-547785-A0 (ES)
IPC: C08K5/37
Filed: 1985-10-11
Abstract: Elastomer/filler interface agents for filled vulcanizable matrices, e.g., natural or synthetic rubber, comprise the amido reaction products of tetraethylene pentamine ("TEPA") with amide-forming organosulfur compounds.
Patent ES-552238-A0 (ES)
IPC: H01H50/44
Filed: 1986-02-20
Abstract: A circuit breaker including a housing, coil connector screws and associated connection rails within the housing, a module in a casing received in a recess of the housing, the module being adapted to limit or attenuate voltage peaks, the module having electrical connectors for electrically connecting the module to the connection rails otherwise than through the coil connector screws, the electrical connectors being a pair of metallic leaf springs each in contact with one of the connection rails, the case being of a generally rectangular configuration with a corner recess at two corners thereof, and each corner recess mating with a projection of the housing and being snap-connected thereto.
Patent FI-834315-A0 (FI)
Inventor: CAIGNARD DANIEL HENRI
IPC: C07D413/12
Filed: 1983-11-24
Abstract: The invention relates to compounds of the formula:   <IMAGE>   in which R represents hydrogen or a lower alkyl radical and R1 and R2 separately represent hydrogen, a lower alkyl, cycloalkyl or benzyl radical, or represent, together with the nitrogen atom to which they are bonded, a heterocyclic radical such as a morpholino, 4-(pyrimidin-2-yl)-piperazinyl or 4-phenylpiperazinyl the phenyl radical of which being optionally substituted by halogen, lower alkoxy or trifluoromethyl, having CNS activity and particularly hypnotic properties. Moreover the compounds in which R1 and R2 are hydrogen can be used in the treatment of heart failure.
Patent FI-881658-A0 (FI)
Inventor: GLEMET MICHEL
IPC: B29C48/154
Filed: 1988-04-08
Abstract: The invention is a process for the manufacture of sections of thermoplastic resin reinforced with continuous fibers and the equipment for carrying out the process. The process consists of coating rovings, having their fibers previously arranged in the form of a sheet, in a coating zone fed with a molten thermoplastic, then, to ensure impregnation of each of the fibers of the rovings, the coated rovings are passed into a forced impregnation zone prior to passing into the channel for shaping the final product.
Patent FI-881815-A0 (FI)
Inventor: SCHIMANEK KARL
IPC: B29D30/54
Filed: 1988-04-19
Abstract: PCT No. PCT/EP87/00459 Sec. 371 Date Jun. 21, 1988 Sec. 102(e) Date Jun. 21, 1988 PCT Filed Aug. 18, 1987 PCT Pub. No. WO88/01228 PCT Pub. Date Feb. 25, 1988.A spreadable ring for sealing an envelope at the bead of the tire to be retreaded during the pressure and heat treatment in an autoclave. The ring is spread with the aid of cut-outs (a lap joint) or by forming the ends on both sides of the opened section into a tongue-in-groove joint. In both cases a joint is generated which runs in the circumferential direction. Depending on the bead shape the sealing surface is cylindrical or tapered whereby lateral end stops or rims facilitate the positioning. The spreading is accomplished manually by the inherent tensioning force of the ring or with the aid of tensioning cylinders.
Patent FI-884385-A0 (FI)
Inventor: ZDAREK DRAHOSLAV
IPC: H01F27/32
Filed: 1988-09-23
Abstract: 1. Transformer, especially for a switching power supply. 2.1. In a transformer for a switching power supply, which operates at an elevated frequency of, for example, 32 kHz, the skin effect is noticeable in an interfering manner. In parallel circuits having a plurality of winding strands for reducing the skin effect, compensating currents occur. 2.2 The compensating currents are avoided by each winding strand being split into winding segments (1, 2) and these winding segments having radial distances from the core (K), which are differently offset in a manner such that they cross. 2.3 Especially a transformer for a switching power supply for a television set. <IMAGE>
Patent FI-885783-A0 (FI)
Inventor: ROSATI ROBERT LOUIS
IPC: C07D207/34
Filed: 1988-12-14
Abstract: Simple amides and derivatives thereof useful for inhibiting the angiotensinogen-cleaving action of the enzyme renin of the formula: <CHEM> wherein R1 is (C6-C8)cycloalkyl or i-propyl; R2 is (C3-C5)alkyl, phenyl, methylvinyl, dimethylvinyl, halovinyl, hydroxy(C1-C3)alkyl or amino(C1-C4)alkyl; R3 is (C1-C6)alkyl or morpholinoethyl; and Het is defined to include certain mono and bicyclic nitrogen-containing heterocyclic rings or heterocyclylalkyl groups.
Patent FI-892540-A0 (FI)
Inventor: SCHMITT URBAN
IPC: G01N33/543
Filed: 1989-05-24
Abstract: To determine an immunologically detectable substance on the principle of the heterogeneous immunoassay using a solid phase to which one of the immunologically active reactants is bound, the solid phase used is a reaction vessel to whose inner surface streptavidin or avidin is bound in an amount such that 0.1 to 2.5  mu g are present per ml of reaction volume. A reaction vessel suitable for this purpose has opposite optically transparent wall regions and, moreover, is coated, at least partially in the region of the inner wall provided to receive liquid, with streptavidin or avidin, where the interior of the container intended to receive liquid, and the streptavidin or avidin content of the coating are matched with one another so that 0.1 to 2.5  mu g of streptavidin or avidin are present per ml of reaction volume. <IMAGE>
Patent FI-892622-A0 (FI)
Inventor: CAMUS MICHEL
IPC: G09F3/02
Filed: 1989-05-30
Abstract: The invention relates to a self-adhesive safety support (1) intended to be placed on a substrate. It consists of at least one printable planar structure, coated with a layer of adhesive, the planar structure and the adhesive being such that the layer of adhesive is partially absorbed into the thickness of the planar structure. The planar structure is preferably a sheet of natural and/or synthetic fibres whose degree of print writing adhesive bonding is 5. Application especially as means preventing the falsification of passports. <IMAGE>
Patent FI-905179-A0 (FI)
Inventor: KURONO MASAYASU
IPC: A61K31/35
Filed: 1990-10-19
Abstract: A pharmaceutical composition showing an inhibition to aldose reductase enzymes is disclosed. In the composition, a hydantoin derivative known per se is uniformly dispersed in a high molecular carrier for the hydantoin derivative. The composition may further contains a water soluble high molecular substance. The composition is administered to prevent or cure a complication due to diabetes.
Patent FI-905958-A0 (FI)
Inventor: CAPRATHE BRADLEY WILLIAM
IPC: A61P25/18
Filed: 1990-12-03
Abstract: Substituted cyclohexanols and cyclohexylamines and derivatives thereof of the formula I <CHEM> as well as methods for the preparation and pharmaceutical composition of same, which are useful as central nervous system agents and are particularly useful as dopaminergic, antipsychotic, and antihypertensive agents as well as for treating hyperprolactinaemia-related conditions and central nervous system disorders.
Patent FI-910763-A0 (FI)
Inventor: COX STEVEN WAYNE
IPC: D06B11/00
Filed: 1991-02-18
Abstract: A control system for a patterning device which provides a method for sequentially loading look-up tables, representing pattern conversion values for different patterns to be printed in sequence, into a patterning device in real time. The system also provides a method for reloading a particular look-up table or group of look-up tables in a prioritized sequence as necessary in order to change the characteristics of the pattern or patterns represented by the table or tables. <IMAGE>
Patent FI-911386-A0 (FI)
Inventor: FRAZZA MARK STEPHEN
IPC: C08F/
Filed: 1991-03-21
Abstract: A process for making uniformly sized polymer particles, having a final particle size of 1-50 micron, comprises (a) combining sufficient free-radical-polymerisable, water-insoluble monomer, or mixt thereof, with an aq dispersion of seed polymer particles, at a rate such that the amt of monomer(s) equal to the total initial wt of the seed polymer particles is combined with the dispersion over 45-120 (pref 60-90) mins, in the presence of a dispersion stabiliser and an oil-soluble, free-radical polymsn initiator. The temp is at least high enough to activate the initiator, and (b) maintaining the temp until polymsn is complete. Opt these steps are repeated until the required final particle size is achieved
Patent FI-911507-A0 (FI)
Inventor: ALBIZZATI ENRICO
IPC: C08F4/658
Filed: 1991-03-27
Abstract: Catalyst components for the polymerization of olefins comprising a titanium halide or alkoxyhalide and an electron-donor compound selected from ethers having two or more ether groups and containing at least one heteroatom selected from the group consisting of N, S, P, Si, non-ether O and halogen atoms or at least one double bond, or both at least one heteroatom and at least one double bond, supported on a magnesium halide in active form. Catalysts obtained from said catalyst components and an Al-alkyl compound.
Patent FI-911758-A0 (FI)
Inventor: SUSSMAN MARK L
IPC: C12Q1/04
Filed: 1991-04-11
Abstract: A method for rapidly identifying microorganisms by determining the rates of enzymatic hydrolysis of a plurality of substrates in the presence of at least one enzyme activity affecting agent, called an "affector" is provided. The substrates are selected from fluorogenic and chromogenic substrates to create a characteristic pattern of enzymatic cleavage rates by enzymes expressed by the unidentified microorganism. This characteristic pattern of enzymatic cleavage rates is a "fingerprint" of the unidentified microorganism when in the presence of the affector. The pattern of enzymatic cleavage rates for the unidentified microorganism is compared to a pattern of enzymatic cleavage rates of the same substrates in the presence of the same affector for one or more identified classes or subclasses of microorganisms. The unidentified microorganism is then identified as belonging to a class or subclasses of the known microorganisms which most closely matches the pattern of enzymatic cleavage rates in the presence of the affector.
Patent FI-913884-A0 (FI)
Inventor: BATE FREDERICK DOUGLAS CLAVELL
IPC: B65B11/02
Filed: 1991-08-16
Abstract: PCT No. PCT/GB90/00266 Sec. 371 Date Aug. 9, 1991 Sec. 102(e) Date Aug. 9, 1991 PCT Filed Feb. 16, 1990 PCT Pub. No. WO90/09316 PCT Pub. Date Aug. 23, 1990.Packaging of articles or sets of articles (31) uses both of helical wrapping material (17) and incorporated longitudinal material (18). Helical wrapping station (14) in a gap (16) between infeed (12) and outfeed (13) conveyors passes helical wrapping material (17) transversely of the direction of travel of the article (31). The longitudinal band(s) of material (18) can serve for positively transporting the articles (31) across the gap (16).
Patent FI-920425-A0 (FI)
Inventor: BOHLMANN ROLF
IPC: C07D409/06
Filed: 1992-01-30
Abstract: The disclosure relates to cycloalkylene azoles of general Formula I    <IMAGE>  (I)  wherein    <IMAGE>     is a carbocyclic or carbopolycyclic group optionally carrying at least on a alkyl substituent, X is a grouping   <IMAGE>     an oxygen or sulfur atom, and Y and Z, independently of each other, are   <IMAGE>     or a nitrogen atom, as well as their pharmaceutically compatible addition salts with acids as well as processes for production thereof. The compounds possess strongly aromatase-inhibiting activity and are suitable for the preparation of medicinal agents. Methods for treating estrogen induced or stimulated tumors, male infertility, and impending cardiac infarction with these compounds are also provided as well as methods for inhibiting female fertility.
Patent FI-921088-A0 (FI)
Inventor: CRISTENSEN FINN
IPC: H04N/
Filed: 1992-03-13
Abstract: This invention relates to interfaces between facsimile machines and cellular telephone systems (including both cellular subscriber terminals and the fixed part of the system, such as the mobile switching center and the interworking function). The cellular radio telephone system could for example be GSM. To prevent two different facsimile machine timers (specified in the CCITT T.30 recommendation) from expiring during the communication between two such machines connected to the GSM environment, a timer reset command (e.g. a command repeat signal) is automatically sent by the interface (12 or 15) to the facsimile machine on receipt of the command from the facsimile machine, for causing the machine to repeat its command so as to allow time for receipt of a response from the other machine. Instead of sending this response only if a command is not recognized (as recommended in T.30), it is used as the default response whenever the GSM environment receives a command from a facsimile machine. If necessary this response can be used twice.
Patent FI-932153-A0 (FI)
Inventor: HJERTMAN BIRGER
IPC: A61M5/32
Filed: 1993-05-12
Abstract: PCT No. PCT/SE92/00596 Sec. 371 Date May 3, 1993 Sec. 102(e) Date May 3, 1993 PCT Filed Aug. 31, 1992 PCT Pub. No. WO93/05835 PCT Pub. Date Apr. 1, 1993.A device for limiting the penetration of an injection needle when an injection is administered from an injection apparatus comprises an exterior sleeve (1) arranged around the front part of the injection apparatus (2). In its foremost position, the sleeve (1) surrounds the needle (8) completely, and it may be displaced rearwards while overcoming a spring force (6), to expose the needle (8).
Patent FI-942353-A0 (FI)
Inventor: HAGENAH GERHARD
IPC: E01C5/06
Filed: 1994-05-20
Abstract: PCT No. PCT/EP92/02670 Sec. 371 Date May 19, 1994 Sec. 102(e) Date May 19, 1994 PCT Filed Nov. 20, 1992 PCT Pub. No. WO93/10310 PCT Pub. Date May 27, 1993.Paving stone set and process and device for the manufacture thereof. In the case of lawn-paving blocks formed from paving stones (10) spaced at a considerable distance apart, these are joined together, against relative displacements, by a holding grid (11) embedded in the paving stones (10) and comprising tension-resistant strands. The said holding grid allows the transfer of traction forces and hence the reciprocal safeguarding of the paving stones (10) within a paving stone set held together by the holding grid (11). The manufacture of the paving stone sets is effected in a concrete stone mold which is conventional in its principle. A flask (19) disposed on a molding plate (28) and a drawing sheet (29) is divided in the horizontal plane (33), creating a top part-flask (34) and a bottom part-flask (35). The holding grid (11) is clamped between the two part-flasks during pouring of the concrete. Following the completion of a paving stone set, the bottom part-flask (35) is withdrawn from the concrete stone mold. Demolding can now be carried out in the usual manner.
Patent FI-942560-A0 (FI)
Inventor: GRUBER PATRICK RICHARD
IPC: D04H1/42
Filed: 1994-05-31
Abstract: A nonwoven fabric comprised of a lactide polymer. The lactide polymer comprises a plurality of poly(lactide) polymer chains, residual lactide in concentration of less than about 2 percent and water in concentration of less than about 2000 parts-per-million. A process for manufacturing a nonwoven fabric with the lactide polymer composition is also disclosed.
Patent FI-944613-A0 (FI)
Inventor: SMITH JAMES W
IPC: B03D1/02
Filed: 1994-10-03
Abstract: Components, usually but not exclusively gaseous components, are removed in a liquid medium from gas streams and chemically converted into an insoluble phase or physically removed. Specifically, hydrogen sulfide may be removed from gas streams by oxidation in aqueous chelated transition metal solution in a modified agitated flotation cell. The same principle may be employed with other procedures in which a gaseous phase is dispersed in a liquid phase to effect an interaction between components present in such phases. A gas-liquid contact apparatus, generally a combined chemical reactor and solid product separation device, comprising such modified agitated flotation cell also is described. In order to effect efficient mass transfer and rapid reaction, gas bubbles containing hydrogen sulfide and oxygen are formed by rotating an impeller at a blade tip velocity of at least about 350 in/sec. to achieve the required shear. To assist in the reaction, a surrounding shroud has a plurality of openings, generally of aspect ratio of approximately 1, of equal diameter and arranged in uniform pattern, such as to provide a gas flow therethrough less than about 0.02 lb/min/opening in the shroud. In general, the gas velocity index of gas through the openings in the shroud is at least about 18 per second per opening, preferably at least about 24 per second per opening. Each of the openings has an area corresponding to an equivalent diameter less than about one inch.
Patent FI-945626-A0 (FI)
Inventor: BRITTON THOMAS CHARLES
IPC: C07F7/18
Filed: 1994-11-29
Abstract: A process for preparing 2,2-difluoroketene silyl acetals and  alpha , alpha -difluoro- beta -silyloxy-1,3-dioxolane-4-propanoic acid esters using these acetals.
Patent FI-952022-A0 (FI)
Inventor: WEISS SAMUEL
IPC: C12N5/02
Filed: 1995-04-27
Abstract: Methods are described for increasing the number of neural stem cells that differentiate into astrocytes, oligodendrocytes, or neurons. The methods comprise proliferating isolated neural stem cells in a culture medium having a first growth factor to produce precursor cells. The precursor cells are then differentiated into astrocytes, oligodendrocytes, or neurons in a second culture medium, EGF-free and containing a differentiation-inducing growth factor.
Patent FI-952209-A0 (FI)
Inventor: FIDO PETER MARK
IPC: B63H25/52
Filed: 1995-05-08
Abstract: PCT No. PCT/GB93/02277 Sec. 371 Date Jun. 30, 1995 Sec. 102(e) Date Jun. 30, 1995 PCT Filed Nov. 4, 1993 PCT Pub. No. WO94/11294 PCT Pub. Date May 26, 1994A device (10) for orientating a load to be suspended and moved by a crane includes a flywheel (11) mounted for rotation in a housing (14). A turntable (17) is pivotally connected to the housing (14) and is drivable relative to the housing using a driven worm gear (23) meshing with an annular set of teeth (22) on the turntable (17). The turntable has an axle (18) to which loads can be attached. When the flywheel (11) is spinning at high speed, it resists movement out of its plane of rotation so as to stabilize the cable in winds, etc. The flywheel (11) also allows the worm gear to react against it so as to turn the load relative to the flywheel (11). Maneuvering of the load is therefore made easier.