baber/WOPTO huggingface dataset:
Patent CZ-91897-A3 (CZ)
Title: Derivatives of n-substituted piperidinyl bicyclic benzoates
Inventor: VAN DAELE GEORGES HENRI PAUL
IPC: C07D405/14
Filed: 1995-09-19
Abstract: The present invention is concerned with novel benzoate derivatives having formula (I), the N-oxide forms, the salts and the stereochemically isomeric forms thereof, wherein: R<1> is halo or C1-6alkylsulfonylamino; A represents a bivalent radical of formula -CH2-CH2- (a), -CH2-CH2-CH2- (b), -CH=CH- (c), in the radicals (a), (b) and (c) one or two hydrogen atoms may be replaced by a C1-6alkyl; R<2> is hydrogen or C1-6alkyloxy; L is a radical of formula: -Alk-R<4> (d), -Alk-O-R<5> (e), -Alk-NR<6>R<7> (f), Alk is C1-12alkanediyl; R<4> is hydrogen; cyano; C1-6alkylcarbonyl; C1-6alkyloxycarbonyl; C3-7cycloalkyl; C1-6alkylsulfinyl; C1-6alkylsulfonyl; phenyl or phenyl substituted with halo, C1-6alkyl or C1-6alkyloxy; tetrahydrofuran; dioxolane; dioxolane substituted with C1-6alkyl; dioxane; dioxane substituted with C1-6alkyl; pyridine; pyridine substituted with halo or C1-6alkyl; pyridazine; pyridazine substituted with one or two substituents selected from halo, C1-6alkyl, hydroxy or an optionally substituted benzimidazolone or an optionally substituted imidazolone; R<5> is hydrogen; C1-6alkyl; hydroxyC1-6alkyl; C1-6alkylcarbonyl; phenyl or phenyl substituted with up to three substituents selected from halo, C1-6alkyl, C1-6alkyloxy; R<6> is hydrogen or C1-6alkyl; R<7> is hydrogen; C1-6alkyl; C1-6alkylcarbonyl; C1-6alkyloxycarbonyl; pyridazine; pyridazine substituted with one or two substituents selected from halo, C1-6alkyl, hydroxy; pyrazine; pyrazine substituted with one or two substituents selected from halo, C1-6alkyl, hydroxy. Pharmaceutical compositions comprising said compounds, processes for preparing compounds and compositions as well as the use as a medicine, in particular for the treatment of gastrointestinal disorders involving a decreased colon motility are described.
Patent SK-75096-A3 (SK)
Title: Panel radiator
Inventor: SEIDL NIKOLAUS
IPC: F28F9/26
Filed: 1994-12-16
Abstract: The invention describes a panal radiator with built-in valve and connection fitting (3) which is equipped with a control valve (5) situated at the side and near the top of the radiator, mounted to the radiator panel supply connection (6), and which comprises connecting pipes (13, 14) that run from the control valve (5) and from a radiator panel return connection (10) to screwed joints (12) at the bottom of the radiator that can be loosened on the radiator side. The screwed joints (12) are situated in the center of the underside (4c) of the radiator (1); from these screwed joints one connecting pipe (13) fixed inside the radiator leads to the control valve (5), and another connecting pipe (14) fixed inside the radiator (1) leads to a radiator panel return connection (10) mounted at the bottom of the radiator (1) in the half of the radiator opposite the control valve (5). These connecting pipes (13, 14) are preferably made of steel.
Patent SK-79797-A3 (SK)
Title: Piperazine derivatives, medicaments containing the same, their use and process for preparing the same
Inventor: PIEPER HELMUT
IPC: C07D211/34
Filed: 1995-12-19
Abstract: Piperazine derivatives have the general formula (I), in which Ra, Y1 to Y3 and E have the definitions given in the first claim. Also disclosed are their tautomers, their stereoisomers, including their mixtures and their salts, in particular their physiologically tolerable salts with inorganic or organic acids or bases, having valuable pharmacological properties, preferably aggregation-inhibiting effects, medicaments containing these compounds, their use and a process for preparing the same.
Patent SK-90798-A3 (SK)
Title: Side wall for closing casting space of the twin roll continuous casting machine for casting thin metal strip
Inventor: DAMASSE JEAN-MICHEL
IPC: B21B1/46
Filed: 1998-07-01
Abstract: A lateral face (4) is claimed for closing the casting space of a continuous casting installation for the production of metal strip (7) between two rolls (1, 1') counter- rotating closely together on their horizontal axes, of the type incorporating a lower part (10) made of a first refractory material with an elevated hardness in the zone where the lower part (10) is in contact with the sides (5, 5') of the rolls (1, 1') or with the liquid metal (3) or with an edge of the solidified strip (7). The lower part (10) incorporates, on its face destined to be turned in the direction of the casting space, a recess filled with a refractory material. Preferably this refractory material enclosed by the recess is a material presenting a lower hardness than that of the first refractory material and with elevated thermal insulating properties.
Patent CH-617056G-A3 (CH)
IPC: G04B37/10
Filed: 1976-07-26
Abstract: A water-proof watch which comprises a composite watch case and a movement therein, said case consisting of a transparent plastic face crystal having overmolded therein a generally opaque plastic body portion to which can be fitted a plastic closure portion sealable after the movement is placed in the watch. At least a zone of the case or of the closure portion is flexible in order to provide control of the winding and regulating mechanism of the movement.
Patent CZ-135892-A3 (CZ)
Title: Process and apparatus for determining dependence of polarizing potential capacity with exclusion of conductivity
Inventor: MATTAUSCH PAVEL ING
IPC: G01R27/26
Filed: 1992-05-05
Abstract: The invented process for determining dependence of capacitance or inductance on polarization potential or current is characterized in that the capacitance dependence on polarization potential is determined differentially with simultaneous suppression of affect of parasitic conductance being parallel-connected thereto and when this conductance can also be determined. Capacitance and parasitic conductance are of non-linear character. Analogously also dependence of series connection of inductance and parasitic resistance on polarization current is determined. Capacitance is determined in a measurement period (30), when in its first measuring time interval (31) and the second measuring time interval (32) the capacitance and the parasitic conductance are excited by a first linearly incrementing voltage potential (41) of a first slope of potential growth and by a second linearly incrementing voltage potential (42) of a second slope of potential growth which induce a first passing current (51) and a second passing current (52) whose magnitudes are at the same exciting voltage potential (60) that is the polarization potential of both capacitance and parasitic conductance, are the magnitudes of a first instantaneous passing current (70) and a second instantaneous passing current (72). The capacitance is evaluated from a relationship for instantaneous current which passes through the capacitance and which is determined as a difference of the first instantaneous passing current (70) and the second instantaneous passing current (72). The apparatus for determining dependence of capacitance or inductance on polarization potential or current consists of excitation, reference, integrator, connection, mode switching, current measurement, current determination, control circuits, timing, filter and evaluation unit.
Patent CS-387991-A3 (CS)
Title: Short peptides with insulin activity
Inventor: MULLNER STEFAN DR
IPC: A61K38/08
Filed: 1991-12-18
Abstract: Short peptides of the formula I X-Y-A-B-C-Cys-D-E (I> in which A and B are an amino acid or a covalent bond, C and D are an amino acid or a substituted amino acid, E is a modified or unmodified amino acid or a covalent bond, X is a radical or hydrogen and Y is leucine or a covalent bond, or dimers of the peptides of the formula I with cystine as dimerisation component, the stereoisomeric forms thereof where appropriate or their physiologically tolerated salts, the preparation thereof, and their use for the treatment of diabetes mellitus are described.
Patent CZ-114193-A3 (CZ)
Title: Rivetting tool
Inventor: WIHAN JOSEF
IPC: B25C5/00
Filed: 1993-06-11
Abstract: A riveting tool includes a tool body having a hydraulic controlled rivet shank clamping assembly and a rivet suction system. A control valve is provided for directing a flow of pressurized air to the rivet clamping assembly and the rivet suction system. The control valve includes a valve rod having a valve rod piston on an upper end and a plurality of radial steps arranged on an outer surface of a lower end. A trigger is mounted slidably in a trigger transverse guide in the tool body and a spring is located within the trigger transverse guide such that pressure applied to the trigger causes the valve rod to move within the control valve from a first to a second position. When the valve rod is in the first position, pressurized air is guided to the rivet suction system. When the valve rod is in the second position, pressurized air is guided to a space below a pneumatic piston. A space above the pneumatic piston is connected to the hydraulic cylinder of the hydraulic controlled rivet shank clamping assembly.
Patent CZ-137096-A3 (CZ)
Title: Device for air flow distribution
Inventor: SCHWARZ STEFAN
IPC: F24F13/075
Filed: 1995-09-18
Abstract: The proposed air diffuser device contains front horizontal deflecting fins (L1-L5) and rear vertical deflecting fins (L6-L10), the fins in each set being interconnected by respective coupling rods (K1, K2), and the fins can articulate about a nozzle housing (GH). The front and rear deflecting fins can be adjusted by an adjusting element (B) extending along a front deflecting fin (L3). To ensure that the front deflecting fins and rear deflecting fins can be adjusted independently of each other, the adjusting element (B) is connected at its rear face via a ball joint (B3; V1) with a connection-adjusting element (V) which is itself hinged on the rear deflecting fins vertically in relation to their pivoting axis so as to be moveable longitudinally.
Patent CZ-166198-A3 (CZ)
Title: Composition containing plastic material and additive as well as use of the additive in the plastic material
Inventor: DE BRABANDER-VAN DEN BERG ELLE
IPC: C08L77/00
Filed: 1996-11-15
Abstract: The invention relates to a composition comprising a plastic and an additive, the additive being present in a dendrimer having functional end groups, said functional end groups being provided, at least in part, with a modifying group, which modifiying group is compatible with the plastic. The additive remains trapped in the dendrimer and, owing to the presence of the modifying group on the dendrimer, cannot migrate or bleed from the plastic.
Patent CZ-171095-A3 (CZ)
Title: Novel steroidal derivatives specific for colon or ilium
Inventor: BRATTSAND RALPH LENNART
IPC: C07J71/00
Filed: 1993-12-17
Abstract: Novel compounds which are a glucocorticosteroid (GCS) chemically bound to a sugar, having the general formula GCS1-O-Sugar1 for colon- or ileum-specific delivery of the GCS to inflamed bowel mucosa, as well as processes for their preparation, pharmaceutical preparations containing the compounds and the use of said compounds in therapy.
Patent CZ-180199-A3 (CZ)
Title: Apparatus for utilization of geothermal power
Inventor: MOE PER H
IPC: E21B43/30
Filed: 1997-11-24
Abstract: A plant for exploiting geothermal energy by circulating water through a geological formation (1) at a substantial depth below the earth surface (2), comprises at least one supply hole (3) leading from the surface (2) down to said formation (1) and at least one return hole (4) for transporting heated water from the formation to the surface. The supply and return holes (3, 4) are interconnected by a plurality of heat absorbing holes (5) which are spaced more than 50 m apart. The heat absorbing holes (5) have a total length of many kilometers but a relatively small diameter in the order of 10 cm. A method for designing the plant involving determining the dimensions of the heat transfer holes (5) is also disclosed.
Patent CZ-9402000-A3 (CZ)
Title: Recyclable moulded thermoplastic structures reinforced by high-molecular fibers and process for preparing thereof
Inventor: FISHER JOHN MICHAEL
IPC: B29K101/10
Filed: 1992-02-21
Abstract: A process is provided for preparing recyclable reinforced composite structures having enhanced surface appearance by heating a self-supporting porous batt comprised of an intimate homogenous blend of high modulus reinforcing fibers and thermoplastic resin fibers to a temperature sufficient to melt the resin component and convert the batt into moldable form, placing the moldable batt into a heated mold to flow, solidify and substantially crystallize the resin component, introducing a thermosetting resin-containing coating material into the mold adjacent at least one surface of the crystallized structure to provide a coating on the one surface and dwelling the coated structure in the mold for a time sufficient to set the coating material.
Patent CZ-200223-A3 (CZ)
Title: Method for inspecting grouting quality and apparatus for making the same
Inventor: PROCHAZKA MARTIN RNDR
IPC: G01N27/76
Filed: 2002-01-03
Abstract: The proposed method for inspecting quality of a grouting being carried out for the purpose to seal and/or consolidation of a solid rock mass is characterized in that a recess with diameter of at least 7.5 centimeter and 50 centimeter in length is executed in the object to be inspected and in the area of said recess a well logging is conducted, whereby said consists in measurement of magnetic susceptibility, calliper looping and measurement of resistance by employing a method of diluting the indicated liquid and a method of constant pouring of the consolidated solid rock mass after grouting. The well logging is preferably carried out prior and after grouting in order to compare state prior grouting with changes caused by grouting. Apparatus for well logging consists of a set of at least three surface panels (3) and at least three measuring probes (4) for measuring magnetic susceptibility, calliper looping and measurement of resistance. The well logging apparatus is preferably built-in an off-road vehicle and consists of a winch section (1) with a special cable (2), at least three surface panels (3) and at least three measuring probes (4) recording various physical parameters of conditions inside the well; the probes are connected through the mediation of a coupling (5) to the special cable (2) terminal with the surface panels (3).
Patent CZ-200247-A3 (CZ)
Title: Computer with illuminator for keyboard
Inventor: TAKAHASHI TOMOYUKI
IPC: F21Y101/02
Filed: 2000-07-03
Abstract: In a portable computer (100), an LED holder (150) is provided in the upper portion of an LCD (109) and an LED is attached inside the LED holder (150). Light emitted from the LED passes through an aperture provided in the bottom portion of the LED holder (150) and illuminates a keyboard (103).
Patent CZ-202321-A3 (CZ)
Title: Ohniště spalovacího zdroje na pevná paliva, zejména zplyňovacího teplovodního kotle na dřevo
Inventor: BENDA LEOPOLD
IPC: F23H17/00
Filed: 2023-01-20
Abstract: Ohniště spalovacího zdroje na pevná paliva obsahuje roštovou část (1) s roštem (2) a spalovací komoru (4). Roštová část (1), která je zhotovena z materiálu o teplotní odolnosti převyšující 700 °C, je propojena kanály (3) situovanými po stranách dna roštové části (1) do spalovací komory (4), která je pod roštovou částí (1). Spalovací komora (4) je zhotovena z materiálu o teplotní odolnosti převyšující 500 °C. Plocha příčných průřezů kanálů (3) je minimálně 3 cm2 na kW jmenovitého výkonu spalovacího zdroje. Spalovací komora (4) má objem minimálně 800 cm3 na 1 kW jmenovitého výkonu spalovacího zdroje. Pod spalovací komoru (4) je umístěna dohořívací komora (5) o objemu maximálně 80 % objemu spalovací komory (4). Obě komory jsou propojeny spojovacími průduchy (6) o ploše alespoň 30 % minimální plochy kanálů (3).
Patent CZ-247797-A3 (CZ)
Title: N alpha-2-(4-nitrophenylsulfonyl)ethoxycarbonyl amino acids, process of their preparation as well as synthesis process of peptides
Inventor: SAMUKOV VLADIMIR VASILYEVICH
IPC: C07C317/18
Filed: 1996-01-27
Abstract: Protected amino acid derivatives of general formula (I) wherein R1 represents hydrogen atom, and R2 represents hydrogen, methyl, isopropyl, 1-methylpropyl, 2-methylpropyl, tert-butoxymethyl, 1-tert-butoxyethyl, 2-methylthioethyl, benzyl, carboxamidomethyl, 2-carboxamidoethyl, tert-butoxycarbonylmethyl, 2-(tert-butoxycarbonyl)ethyl, 4-(tert-butoxycarbamido)butyl, 4-tert-butoxybenzyl, indolyl-3-methyl, S(triphenylmethyl)thiomethyl, 1-(triphenylmethyl)imidazolyl-4-methyl, 3-(N<G>-mesitylenesulfonyl)guanidinopropyl, N-xanthylcarboxamidomethyl, 2-(N-xanthylcarboxamido)ethyl or S-(acetamidomethyl)thiomethyl; or R1 and R2 together represent propylene radical. Methods for the preparation of said derivatives are provided, and a process for solid phase peptide synthesis using said derivatives is described.
Patent CZ-282894-A3 (CZ)
Title: Substituted 1,2,3,4-tetrahydroisoquinolines as such and for treating diseases, pharmaceutical preparations based thereon and intermediates for their preparation
Inventor: BLANKLEY CLIFTON JOHN
IPC: C07C43/23
Filed: 1993-04-19
Abstract: This invention relates to novel substituted 1,2,3,4-tetrahydroisoquinolines which are useful the treatment of vascular restenosis, various disorders of the central nervous system, in the regulation of female reproductive functions, in cognitive enhancement, in atherosclerosis and in treating excessive AVP secretory disorders. Novel intermediates useful in the preparation of the compounds are also disclosed. Methods of using the compounds and pharmaceutical compositions containing them are disclosed.
Patent CZ-291195-A3 (CZ)
Title: Electric hand-held cutting tool with a potentiometer and potentiometer setting method
Inventor: KRAENZLER ERNST
IPC: H01C10/14
Filed: 1995-03-24
Abstract: In prior art electric hand tools, it is necessary to adjust the power-control potentiometer so that, when the potentiometer is adjusted to a particular position, the required resistance is provided by the potentiometer. The invention aims to simplify manufacture by ensuring that the potentiometer can be adjusted without the need for additional components and without the need for costly additional equipment. The potentiometer (20) has a resistance track (21) with which a sliding contact (22) is in electrical contact. The sliding contact (22) can be operated by hand by means of an adjustment element (15). Both sliding contact (22) and adjustment element (15) include means (26) for the adjustment of their relative  positions following insertion into the housing (11) of the power tool.
Patent CZ-291599-A3 (CZ)
Title: Disubstituted bicyclic heterocyclic derivatives
Inventor: HAUEL NORBERT
IPC: A61K31/454
Filed: 1998-02-16
Abstract: The invention relates to new disubstituted bicyclic heterocycles of the general formula (I): Ra-A-Het-B-Ar-E, in which A, B, Ar, Het and Ra are defined as in claim 1. The invention also relates to their tautomers, their stereoisomers, their mixtures, and their salts, which have valuable properties. The compounds of the above general formula (I), in which E is a cyano group, thus represent valuable intermediate products for the production of the other compounds of the general formula (I). Furthermore, the compounds of the above general formula (I), in which E stands for a RbNH-C(=NH)-group, have valuable pharmacological properties, in particular in inhibiting thrombin and prolonging thrombin time.
Patent CZ-293497-A3 (CZ)
Title: Mercapto and seleno derivatives as inhibitors of nitrogen(ii) oxide synthase
Inventor: SOUTHAN GARRY J
IPC: A61K31/425
Filed: 1996-03-22
Abstract: This invention is directed to a pharmacologically acceptable composition for inhibiting nitric oxide synthase in a mammal, which includes a mercapto or seleno derivative and a pharmaceutically acceptable carrier. The invention also concerns a method of inhibiting nitric oxide synthase, selectively inhibiting the inducible isoform of nitric oxide synthase, and treating various conditions where there is an advantage in inhibiting nitric oxide biosynthesis. The method includes the step of administering to a mammal a mercapto or seleno derivative in pure form or in a pharmaceutically acceptable carrier.
Patent CZ-308995-A3 (CZ)
Title: The use of nonapeptides and decapeptides for preparing a medicament against aids
Inventor: ENGEL JURGEN PROF DR
IPC: C07K7/23
Filed: 1994-04-02
Abstract: PCT No. PCT/EP94/01037 Sec. 371 Date Dec. 18, 1995 Sec. 102(e) Date Dec. 18, 1995 PCT Filed Apr. 2, 1994 PCT Pub. No. WO95/00168 PCT Pub. Date Jan. 5, 1995Described are LHRH-antagonistic and bombesin-antagonistic nona- and decapeptides suitable for use in the preparation of a drug for the treatment of AIDS and ARC as well as for use in the preparation of an immunostimulation drug.
Patent CZ-326494-A3 (CZ)
Title: Process and apparatus for collecting and packaging of permanent containers, the use of such apparatus and packaging system
Inventor: GREINER CHRISTOPH DIPL ING
IPC: B65D6/16
Filed: 1994-12-21
Abstract: A device (10) is described for holding a multi-pack (20) of low rigidity for collecting and packaging reusable packagings for filter material. It is characterised in that a holding device (30), connected to the side parts (1 to 6), is provided for attaching the multi-pack (20) to the erected side parts (1 to 6), the side parts (1, 2, 6; 3, 4, 5) are divided into one or more side-part groups (A, B), the side parts (1, 2, 6; 3, 4, 5) being connected to one another in an articulated manner in each of the side-part groups (A; B), and the side parts (1, 2, 6; 3, 4, 5) being connected to one another in an articulated manner in one or more side-part groups (A, B) in such a way that one or more side parts (2, 3; 5, 6) of one or more side-part groups (A, B) can be pivoted outwards, away from the multi-pack (20), in such a way that the multi-pack (20) can be removed from the device (10) laterally or at an end face. A device is furthermore described for holding the multi-pack (20), the device (10) having a side part or a plurality of erectable side parts (1 to 6) which, erected outside the multi-pack (20), delimit a space for accommodating the multi-pack (20) and surround the multi-pack (20) or, erected inside the multi-pack (20), are arranged in such a way that they delimit the largest possible space inside the multi-pack (20) and are surrounded by the multi-pack (20), and having a holding device (30), connected to the side part or parts (1 to 6), for attaching the multi-pack (20) to the erected side part or parts (1 to 6). Further subjects of the invention are an appropriate method and packaging system. <IMAGE>
Patent CZ-347895-A3 (CZ)
Title: Butter and process for preparing thereof butter and process for preparing thereof
Inventor: NORTON IAN TIMOTHY NORTON IAN
IPC: A23L29/231
Filed: 1994-06-07
Abstract: A fat-continuous spread comprising: (A) from 0.1 to 10 wt% of gelatin; (B) from 0.1 to 7 wt% of a gelled polysaccharide not being starch; and (C) from 10 to 60 wt% of fat. The balance of the above being traditional constituents of spreads.
Patent CZ-350496-A3 (CZ)
Title: Process for preparing ketals of steroidal compounds
Inventor: BRANDS FRANCISCUS THEODORUS LE
IPC: C07J75/00
Filed: 1996-11-29
Abstract: The invention relates to a method of the preparation of a steroid derivative ketal according to the general formula I:
         wherein
     R 1  is CH 3  or C 2 H 5 ;   R 2  is OH;   R 3  is H, CH 3 ; C≡CH, CH 2 Hal,, or CH 2 CN; or R 2  and R 3  together are O;   R 4  is (2-5C) alkylene; and   Hal is Cl, Br or I,       characterized in that the compound of formula II:
         wherein R 1 , R 2  and R 3  have the previously given meanings, is treated in the presence of an orthoester of formula III:
         or an orthoester of formula IV:
         wherein R 4  has the previously indicated meaningor a mixture thereof 
   with an alcohol according to the general formula HOR 4 OH, wherein R 4  has the previously given meaning.