baber/WOPTO huggingface dataset:
Patent UA-121227-C2 (UA)
Title: ЗАСТОСУВАННЯ ГІДРОБРОМІДУ 1-(4<sup>1</sup>-ЦИКЛОГЕКСИЛФЕНІЛ)-2-[(5,6-ДИГІДРО-4H-[1,3]ТІАЗИН-2-ІЛ)-(4<sup>2</sup>-ЕТИЛФЕНІЛ)АМІНО]ЕТАНОНУ ЯК СПОЛУКИ, ЩО МАЄ ПРОТИПУХЛИННІ ВЛАСТИВОСТІ
Filed: 2017-06-21
Abstract: Гідробромід 1-(41-циклогексилфеніл)-2-[5,6-дигідро-4H-[1,3]тіазин-2-іл)-(42-етилфеніл)аміно]етанону, що має протипухлинні властивості. Винахід належить до органічної, фармацевтичної хімії та медицини. Визначення протипухлинної активності заявленої сполуки проведено in vitro на 60 лініях ракових клітин при дії речовини в концентрації 10-5 моль/л та у градієнті концентрацій 10-4-10-8 M за стандартною процедурою оцінки мітотичної активності, виконаних в Національному інституті раку США (National Cancer Institute of Health, USA) в рамках Development Therapeutic Program. Сполука є ефективною відносно клітин меланоми, лейкемії, дрібноклітинного раку легенів, раку товстого кишечнику, пухлин кори головного мозку, яєчників, простати, молочної залози та нирок і виявила більш високу протипухлинну активність, ніж препарат порівняння - 5-флуороурацил. Так, заявлена сполука виявилася відносно всіх клітин лейкемії CCRF-СЕМ, НL-60(ТВ), К-562, МОLT-4 та RPMI-8226 із значенням -3.76 %, -55.48 %, -13.40 %, -24.41 % та -37.55 % відповідно. Від'ємні значення свідчать про те, що досліджувана сполука не тільки затримує ріст пухлини, але і знищує зазначені лінії ракових клітин). Заявлена сполука знищує клітини дрібноклітинного раку легенів HОР-92, NCI-H460 та NCI-H522 на -17.44 %, -73.50 % та -23.31 % відповідно. Найбільш активною заявлена сполука виявилась проти клітин меланоми LOX IМVI та SK-MHL-5 із значеннями -90.06 % та -86.39 % відповідно.
Patent UA-124028-C2 (UA)
Title: Широкозахватна посівна машина
Filed: 2019-06-24
Abstract: Широкозахватна посівна машина, що містить центральну секцію з задніми приводними колесами, оснащеними механізмами приводу висівних апаратів, та передніми самоустановними колесами, закріпленими на кінцях поперечної шарнірної балки, з'єднаної з поздовжнім брусом рами центральної секції за допомогою горизонтального шарніра, і бокові секції, з'єднані з центральною секцією за допомогою проміжних опор з горизонтальними і вертикальними шарнірами, висівні апарати з валами приводу. Відповідно до винаходу, задні приводні колеса центральної секції виконані самоустановними, оснащені фіксаторами робочого і транспортного положень, а бокові секції з'єднані з центральною секцією горизонтальними шарнірами, приводні вали висівних апаратів виконані телескопічними і оснащені шарнірами Гука, осі яких перетинаються з осями горизонтальних шарнірів. Таке конструктивне виконання широкозахватної посівної машини спрощує її конструкцію, полегшує переведення у транспортне (робоче) положення, зменшує транспортну ширину.
Patent UA-127033-C2 (UA)
Title: Мобільна радіолокаційна станція контрбатарейної боротьби малої дальності
Filed: 2019-07-11
Abstract: Винахід належить до галузі радіоелектронної техніки. Мобільна радіолокаційна станція контрбатарейної боротьби малої дальності включає елементи, в яких до складу кожної з матриць підсумовування НВЧ-сигналів, що входять до складу НВЧ-панелей для випромінювання і прийому НВЧ-сигналів, додатково введені перший керований фазообертач, другий керований фазообертач та регулятор електричної довжини мікросмужкових ліній, до складу програмного комплексу управління променями РЛС додатково введена підпрограма управління нахилом вертикальних променів, до складу приймального пристрою додатково введено модуль цифрової обробки сигналів, до складу якого входять аналого-цифровий перетворювач та блок цифрової обробки сигналів. Винахід забезпечує усунення впливу підстильної поверхні землі на характеристики виявлення цілі, тобто зменшує помилки визначення координат цілі.
Patent UA-126977-C2 (UA)
Title: Delayed release deferiprone tablets and methods of using the same
Inventor: SHERMAN BERNARD CHARLES (DECEASED)
Filed: 2018-10-25
Abstract: The invention is directed to pharmaceutical compositions such as tablets that exhibit delayed release properties when administered as either whole or half tablets. The invention is also directed to delayed release tablets comprising deferiprone for oral administration, for which twice daily administration is bioequivalent to the same daily dose of an immediate release tablet administered thrice daily. The invention is also directed to methods of making and using the same.
Patent UA-125989-C2 (UA)
Title: Спосіб одержання (1r,2s)-1-(6-бром-2-метоксихінолін-3-іл)-4-диметиламіно-2-(1-нафтил)-1-фенілбутан-2-олу та його фармацевтично прийнятної солі
Inventor: KIM YONG JIK
Filed: 2021-06-11
Abstract: Винахід стосується способу одержання (1R,2S)-1-(6-бром-2-метоксихінолін-3-іл)-4-диметиламіно-2-(1-нафтил)-1-фенілбутан-2-олу або його фармацевтично прийнятних солей, де спосіб включає виділення (1R,2S)-1-(6-бром-2-метоксихінолін-3-іл)-4-диметиламіно-2-(1-нафтил)-1-фенілбутан-2-олу, який можна виготовляти масово шляхом здійснення економічного способу одержання і з високим виходом.
Patent DE-19602888-C5 (DE)
Title: Bremsbacke, insbesondere für Nutzfahrzeug-Scheibenbremsen
Inventor: KUEHNE VIKTOR
IPC: F16D65/00
Filed: 1996-01-29
Granted: 2004-05-27
Abstract: Bremsbacke (1), insbesondere für Nutzfahrzeug-Scheibenbremsen, die ein Belagmaterial (3) und einen Belagträger (2) mit Abstützflächen (4) aufweist und zum Eingriff in einen Bremsträger (6) ausgelegt ist, wobei in den Belagträger (2) zur Geräuschdämmung ein elastisch verformbares Abstützelement (5) eingesetzt ist, welches im Belagträger (2) und am Bremsträger (6) abgestützt ist sowie über die Abstützflächen (4) hinausragt, und das Abstützelement (5) als Verbundteil ausgestaltet ist, das einen im wesentlichen federnden und/oder dämpfenden Bereich – Elastoelement (51) – und einen im wesentlichen festen, reibungsarmen Bereich – Gleitelement (52) – aufweist, dadurch gekennzeichnet, daß das Abstützelement (5) in Richtung des Bremsmomentes und/oder in Richtung der Auflagekraft der Bremsbacke (1) begrenzt elastisch verformbar ist, wobei die Abstützfläche (4) die Begrenzung der elastischen Verformung des Abstützelementes (5) nach Art eines Festanschlages bildet, derart, daß nach dem vollen Verformungsweg des Abstützelementes (5) die Abstützfläche (4) des Belagträgers (2) mit dem Bremsträger (6) in Wirkung steht, wobei...
Patent DE-50203783-C5 (DE)
Inventor: PIZZUTO GIANFRANCO
IPC: A01B33/10
Filed: 2002-10-07
Granted: 2010-02-11
Abstract: A milling tooth body for a comminution machine has a working side, oriented in a working direction; a flange side detachably connected to a milling tooth holder of the comminution machine; a tooth tip on the side of a recess; and a base at an end of the tooth body facing away from the tooth tip. A cutter device is in the recess. The flange side on the tooth body is opposite the working side. An entire side of the tooth body, which is oriented in the working direction, is the working side. The tooth tip projects away from the flange side in the direction of a longitudinal axis of the tooth body, perpendicular to the working direction. A first section of the tooth body projects away from the flange side in a direction parallel to and opposite the working direction.
Patent DE-60040799-C5 (DE)
Inventor: SVENSSON OLA
IPC: H04W36/00
Filed: 2000-10-20
Granted: 2020-03-05
Abstract: A method for conveying measurement information from a mobile terminal in a first communication system to a second communication system is disclosed, whereby the measurement information related to the first communication system is conveyed to the second communication system on a control channel which can function in a non-stealing mode. For example, Universal Mobile Telecommunication System (UMTS) measurement information can be conveyed from a mobile terminal to a Base Station Controller (BSC) in a Global System for Mobile Communications (GSM) network, in a GSM message on a Slow Associated Control Channel (SACCH). In this way, the UMTS measurement information can be conveyed effectively between the two mobile communication systems without sacrificing the quality of speech information being conveyed. Moreover, handovers between the two mobile communication systems can be effectively performed.
Patent RU-2574522-C9 (RU)
Title: Способ регистрации малоконтрастных точечных объектов
Inventor: Zdor Stanislav Evgenevich
IPC: H04N5/30
Filed: 2014-10-17
Granted: 2016-06-10
Abstract: Способ регистрации малоконтрастных точечных объектов использует астрономический или иной оптико-электронный прибор, объектив которого формирует оптические изображения точечных объектов на светочувствительной поверхности матричного приемника излучения, которая состоит из множества пикселей, образующих столбцы и строки матричного приемника излучения. Эти изображения многократно экспонируют и считывают с бинированием пикселей, когда соседние пиксели матричного приемника излучения группируют в один бинируемый массив. При каждом новом экспонировании и считывании в данном способе бинируемый массив смещают по строке или столбцу матричного приемника излучения по отношению к предыдущему положению. Технический результат - повышение вероятности правильной регистрации малоконтрастных точечных объектов. 5 ил., 4 табл.
Patent DK-28589-D0 (DK)
Inventor: RASMUSSEN JAN KROEYER
IPC: A01K1/02
Filed: 1989-01-23
Abstract: In order to be able to keep pigs in an expedient manner, this must be effected in such a way that the pigs are given living and growing conditions which correspond substantially to their natural behavior. According to the invention, for this purpose there can be used a pigpen unit comprising a piggery (1) and an enclosed yard (2), neither of which have a floor, and an external feeding place (3). These sections can be separated and assembled in such a manner that it is easy to move the pigpen unit for a crop rotation. In order to facilitate the feeding and the operation, the unit has a straight side wall (4, 12, 15) which faces out towards the road (25), and from which through a door (13) there is access into the yard (2) and through an opening (27) fodder can be introduced into a trough.
Patent DK-78090-D0 (DK)
Inventor: SOELBECK PETER
IPC: F16B5/00
Filed: 1990-03-27
Abstract: PCT No. PCT/DK91/00092 Sec. 371 Date Sep. 4, 1992 Sec. 102(e) Date Sep. 4, 1992 PCT Filed Mar. 25, 1991 PCT Pub. No. WO91/14842 PCT Pub. Date Oct. 3, 1991.For the fastening of a protecting or shielding cover, in particular a tarpaulin, to a scaffolding, a fastening member is provided which has an anchor pin to be arranged on the external surface of the tarpaulin, a flexible strap being firmly connected with the anchor pin and having a slit or opening through which the free end of the strap may be pushed and a toothing to prevent the strap from being retracted. The slit or opening is provided in a clamping member at the opposite end of the strap in relation to the insertion end and the anchor pin is connected with the strap at a distance from the clamping member conforming to the dimensions of a frame member of the scaffolding, while the distance of the anchor pin from the insertion end is substantially larger. For mounting the fastening member use is made of a tool in which a hollow piston axially displaceable in a holder has a pointed cutting end and is designed to receive the anchor pin of the pin being pressed out of the hollow piston by use of a slide accommodated in the piston.
Patent DK-149283-D0 (DK)
Inventor: CREMER JOSEF
IPC: A23K20/26
Filed: 1983-03-30
Abstract: 1. Process for making a granulated animal feed phosphate consisting of the phosphates of sodium, magnesium and calcium by introducing phosphoric acid, dolomite and sodium hydroxide solution into an elongated reaction zone, wherein the dolomite consisting of particles with a size of less than 0.1 mm and phosphoric acid are introduced into the head portion of the reaction zone and sodium hydroxide solution is added to said mixture at a point in the reaction zone the mixture of dolomite and phosphoric acid reaches after 0.5-3 minutes, and wherein the dolomite, phosphoric acid and sodium hydroxide solution are passed through the reaction zone with continuous agitation, and reacted, characterized in that a) the phosphoric acid presents a concentration of 50 to 70 weight% P2 O5 and the sodium hydroxide solution presents a concentration of 50 to 80 weight% NaOH, b) the phosphoric acid is introduced into the reaction zone at a temperature of 50 to 120 degrees C and the sodium hydroxide solution is introduced there into at a temperature of 60 to 140 degrees C, c) the sodium hydroxide solution is added to the mixture of dolomite and phosphoric acid along a path of at most 5% the length of the reaction zone, and d) granules with a particle size of 0.5 to 2.5 mm are sieved off.
Patent DK-208789-D0 (DK)
Inventor: MOHRS KLAUS
IPC: C07D215/14
Filed: 1989-04-28
Abstract: alpha -Substituted 4-(quinolin-2-ylmethoxy)phenylacetic acids and esters can be prepared by reaction of appropriate phenols with 2-halomethylquinolines or by reaction of appropriately substituted quinoline with halides. The novel compounds can be employed as active substances in medicaments.
Patent DK-252286-D0 (DK)
Inventor: BENAVIDES JESUS
IPC: C07C233/11
Filed: 1986-05-29
Abstract: Amides of formula:    <IMAGE>  I  in which A is   <IMAGE>  V and W are H, halogen, alkyl (1-3C), alkoxy (1-3C), NO2 or CF3, Z is bound in the ortho or para position with respect to B and is phenyl, optionally substituted, thienyl or pyridyl, the chain X-(CH2)n-(CHR)m-CO-NR1R2 is bound in the ortho or para position with respect to B, R is H or alkyl (1-3C), R1 and R2 are alkyl (1-6C), cycloalkyl (3-6C), phenyl, phenylalkyl, cycloalkylalkyl, alkenyl (3-6C), R1 and R2 can also form, with the nitrogen atom to which they are attached, a pyrrolidine, piperidine, morpholine or thiomorpholine ring, X is >CH-R3, >N-R4, >SO, >SO2, >O or >S, R3 is H, alkyl (1-3C), R4 is alkyl (1-3C) m=0 or 1 and n=0, 1 or 2, provided that, if X is >SO, >SO2 or >N-R4, the sum m+n is equal to at least 1, that, when A and B are N and Z is in the para position with respect to B, X cannot denote the group >CH-R3 and that when A is CH, B is N, Z is in the ortho position with respect to B, X is an oxygen atom, and R is a hydrogen atom, the sum m+n is other than 1, and excluding 2-phenyl-4-quinolyl N,N-dimethylcarbamate, have useful pharmacological activity, e.g. as anxiolytics, anticonvulsants and antiangina agents.
Patent DK-286684-D0 (DK)
Inventor: JESCHKE WILLI
IPC: B41F33/00
Filed: 1984-06-12
Abstract: A device for controlling, by a measuring technique, the dampening medium guidance zonewise in an inking unit of an offset printing machine includes a measuring roller engaging an ink applicator roller of the inking unit and having interfaced oleophilic and hydrophilic surface regions, and an optoelectronic measuring device disposed adjacent to the measuring roller and operating thereon over the entire width thereof at a spaced distance therefrom, and wherein at least the oleophilic surface regions of the measuring roller is formed as a screen.
Patent DK-481889-D0 (DK)
Inventor: MATSON STEPHEN L
IPC: C12P17/12
Filed: 1989-09-29
Abstract: This invention relates to novel methods for facilitating the enzymatic resolution of racemic mixtures of esters, which are derivatized with groups which enhance the esters' aqueous solubility, in an extractive member reactor where the enzyme is placed alternatively either (1) in the aqueous phase, (2) in association with the membrane, or (3) in the aqueous phase and in association with the membrane, wherein the aqueous ester phase is contacted with one side of the membrane, and where an organic extractive phase is contacted with the other side of the membrane, wherein the extractive phase serves to remove the resolving reaction product. Of particular significance regarding this invention is its use of water soluble esters that are derivatized with groups which enhance their aqueous solubility and their reactivity with enzymatic resolving methods which are mediated in an aqueous environment. Novel methods were utilized to prepare these esters, for use in this invention's methods for enzymatically resolving the racemic mixtures of the esters, to produce the separate chiral isomers of the racemic mixture. The importance of the resolution of the separate chiral isomers of the racemic mixtures resides in the isolation of the isomers which frequently have different biological activities.
Patent DK-491187-D0 (DK)
Inventor: PETERSEN FLEMMING OLUF
IPC: E04D13/02
Filed: 1987-09-18
Abstract: The vertical breast wall (4) forming the rear wall of a balcony installed in an inclined roof comprises a hinged door (5) which is completed to full height by a top-hinged window (6) which in its closed position flushes with the roof surface and at is lower edge fits tightly against the top edge of the door.
Patent DK-510788-D0 (DK)
Inventor: AUHORN WERNER
IPC: D21H19/58
Filed: 1988-09-14
Abstract: Process for improving the printability of paper by a single- or two-sided application of aqueous coating materials consisting of
 a) 100 parts by weight of a finely dispersed pigment
 b) 5 to 70 parts by weight (based on solids) of a cationic aqueous polymer dispersion of a paper size and
 c) 0.01 to 10 parts by weight of a surfactant which interferes with the formation of the surface sizing and/or of a polymeric dispersant
 to the surface of the paper in a quantity of 0.5 to 4 g/m<2> and drying the coated paper.
Patent DK-688687-D0 (DK)
Inventor: VANERDEN DONALD L
IPC: B65D33/20
Filed: 1987-12-28
Abstract: A bag (80) has wall panels (81) defining a receptacle space (82) and providing a bag mouth arrangement between upper end portions of the wall panels (81). A tamper evident, and if desired hermetic seal, non-reclosable closure (90) adjacent to a reclosable zipper (85) and located adjacently below upper end portions of the wall panels is accessible to be opened when the zipper (85) is open. The zipper (85) is arranged for intermittent opening and closing of the bag (80). The non-reclosable (90) closure is a peel seal. <IMAGE>
Patent HU-904426-D0 (HU)
Title: 8-alpha-acyl-amino-ergoline derivatives and their utilization as medicament
Inventor: SAUER GERHARD
IPC: C07D457/12
Filed: 1990-05-10
Abstract: 8 alpha -acylamino ergolines are useful dopamine agonists.
Patent HU-905348-D0 (HU)
Title: Telescopic casing
Inventor: WEHLER HERBERT
IPC: B23Q11/08
Filed: 1990-08-27
Abstract: The subject matter of the invention is a telescopic covering with a number of cover boxes (A, B, C, D) which can telescope one inside the other, consisting of a top wall (1), two side walls (2) and a rear wall (3), in which arrangement a part projecting beyond the top wall (1) in the plane of the rear wall (3) forms a stop for carrying the next larger cover box. For improved support and guidance of the cover boxes (A, B, C, D) on one another and against one another, it is proposed to arrange a corner profile (9) between the top wall (1) and the two side walls (2) of each cover box, and to support the cover boxes on one another with these corner profiles (9). 
<IMAGE>
Patent IT-9009482-D0 (IT)
Inventor: BEDENDO ARMANDO
IPC: G01N21/78
Filed: 1990-09-05
Abstract: The apparatus for field or process colorimetric analyses of water or other samples with a discontinuous on-line system comprises: an open colorimetric cell (9) with means of charging the sample from the base and discharge of the excess sample over the spill rim. The cell is combined with means for producing a precise amount of the sample, in particular by the use of a magnetically driven two-speed stirrer (26) which at a first speed produces the precise amount by discharging through forced overflow and at a second speed stirs the sample treated with appropriate reagents introduced through suitable metering means (30, 32, 34, 36). <IMAGE>
Patent NO-880360-D0 (NO)
Inventor: DELAYE JEAN-LUC
IPC: B02C13/18
Filed: 1988-01-28
Abstract: The rotor of the crusher receives the stones at its centre. It comprises three blades (20, 21) which, except on the ejecting edges (22), are protected against internal wear by their hollow shape which retains a protective layer of stones. These edges are protected from impacts by protecting plates (24) arranged radially in front of them.   <IMAGE>
Patent NO-883592-D0 (NO)
Inventor: GILLIGAN JAMES P
IPC: C12N11/00
Filed: 1988-08-12
Abstract: The present invention provides a method for the production of an alpha-amidating enzyme comprising the steps of providing a DNA sequence capable of coding for an alpha-amidating enzyme, ligating said DNA sequence into an expression vector, inducing transformation of said expression vector into a host cell capable of expressing said DNA sequence, and preferentially selecting host cells having and expressing said DNA sequence and a genetically engineered microorganism comprising at least one preferentially selected host cell by such a method.
Patent NO-893628-D0 (NO)
Inventor: CHARLES JEMIN
IPC: A01N43/80
Filed: 1989-09-11
Abstract: Biocide compositions comprising 5-chloro-2-methyl-4-isothiazolin-3-one-and 2-methyl-4-isothiazolon-3-one- in a weight ratio 1.2 to 25.4 : 74.6 to 98.8 demonstrate synergism and decreased sensitization potential.
Patent NO-902552-D0 (NO)
Inventor: FLYNN KATHY M
IPC: H05K3/28
Filed: 1990-06-08
Abstract: A photoimageable composition for forming a solder mask has a photopolymerizable acrylate chemical system which renders exposed portions insolvable to alkaline aqueous developers and an epoxy chemical system which hardens the composition after exposure and development. The acrylate chemical system comprises acrylate monomers, epoxy-acrylate oligomers and a photoinitiator. The epoxy chemical system comprises an epoxy resin and a curative therefore. The composition further comprises a cross-linking agent which is reactive with hydroxyl groups of the acrylate and epoxy chemical systems.
Patent NO-903694-D0 (NO)
Inventor: HEINEMEYER BEN WILLIAM
IPC: C08G59/14
Filed: 1990-08-22
Abstract: Advanced resin compositions are prepared from a compound having an average of more than one vicinal epoxide group per molecule and an epoxide equivalent weight of from 170 to 200 and a compound having an average of more than one aromatic hydroxyl group per molecule wherein the resultant advanced resin has an epoxide or aromatic hydroxyl equivalent weight of from 200 to 50,000.
Patent NO-911230-D0 (NO)
Inventor: JONES DAVID RUSSEL
IPC: C08G101/00
Filed: 1991-03-26
Abstract: A foam formulation, useful in the preparation of water-blown heat-insulating material, comprising (i) one or more polyols, (ii) one or more organic polyisocyanates, (iii) water, and (iv) auxiliary materials known in the art, characterized in that the polyol or polyol mixture has an average functionality (Fn) varying from 2.7 to 4.3; a hydroxyl value (OHv) of 325 to 500 mg KOH/g, and a viscosity measured at 20  DEG C of between 350 mPa.s and 2300 mPa.s; the use of said polyol or polyol mixture as softening point improver in a process of preparing water-blown heat-insulating material, and the water-blown heat-insulating material so prepared.
Patent NO-912541-D0 (NO)
Inventor: BAADER EKKEHARD
IPC: A61K31/44
Filed: 1991-06-27
Abstract: 2,4- and 2,5-substituted pyridine N-oxides which have fibrosuppressive and immunosuppressive activity are presented. The said compounds are likewise suitable for the treatment of disturbances of the metabolism of collagen and collagen-like substances and of the biosynthesis of C1q.