baber/WOPTO huggingface dataset:
Patent HU-T65820-A (HU)
Title: Process for prepearing compounds to inhibit hiv-protease
Inventor: HUI KWAN YUK
IPC: C07C237/08
Filed: 1993-12-20
Abstract: The present invention provides novel HIV protease inhibitors, of formula I <CHEM>  wherein:   Z   is hydrogen, formyl, carbamoyl, C2-C6 alkanoyl, C1-C4 alkoxycarbonyl, -C(O)CF3 or -S(O)2-R, where R   is C1-C6 alkyl, amino, trifluoromethyl, C1-C4 alkylamino, di(C1-C4)alkylamino, aryl, aryl(C1-C4)alkyl, heterocycle, unsaturated heterocycle or C5-C7 cycloalkyl; R<1>   is aryl, C5-C7 cycloalkyl or -S-R<1x>, where R<1x> is aryl or C5-C7 cycloalkyl; R<2>   is an amino acid side chain, -(CH2)y-X-R<2a>, cyano(C1-C4)alkyl or -(CH2)y-S(O)w-[1-N(R<2c>)-tetrazol-5-yl], where        y is 0, 1, 2 or 3; X is a bond, divalent(C2-C4)alkenyl, divalent(C2-C4)alkynyl, -C(O)-O-, -O-C(O)-, -C(O)-NR<2b>-, -NR<2b>-C(O)-, -NR<2b>-, -C(O)-, -O-, -S(O)w-;        w is 0, 1 or 2; R<2a> is C1-C6 alkyl, aryl, unsaturated heterocycle, heterocycle, aryl(C1-C4)alkyl, unsaturated heterocycle(C1-C4)alkyl or heterocycle(C1-C4)alkyl;        R<2b> is hydrogen or C1-C4 alkyl; R<2c> is hydrogen, C1-C6 alkyl, aryl, unsaturated heterocycle, aryl(C1-C4)alkyl or unsaturated heterocycle(C1-C4)alkyl; Y   is aryl or unsaturated heterocycle; R<3>   is a group having the structure: <CHEM>   <CHEM>   <CHEM>   <CHEM>   <CHEM>   <CHEM>  where:        p is 4 or 5;        l is 3, 4 or 5; R<4> at each occurrence is independently hydrogen, C1-C6 alkyl or hydroxy(C1-C4)alkyl; R<5> and R<6> are independently selected from hydrogen, hydroxy, C1-C6 alkyl, C1-C6 alkoxy, amino, C1-C4 alkylamino, hydroxy(C1-C4)alkyl, carboxy, C1-C4 alkoxycarbonyl, carbamoyl, N-(C1-C4)alkylcarbamoyl, aryl, heterocycle or unsaturated heterocycle; o
Patent HU-T73200-A (HU)
Title: Solid polymeric product, method of making thereof and a treating process
Inventor: ALLEN ADRIAN SWINBURN
IPC: C02F1/52
Filed: 1995-02-10
Abstract: PCT No. PCT/GB95/00282 Sec. 371 Date Oct. 11, 1995 Sec. 102(e) Date Oct. 11, 1995 PCT Filed Feb. 10, 1995 PCT Pub. No. WO95/21796 PCT Pub. Date Aug. 17, 1995A flocculant, viscosifier or other water soluble or water swellable particulate polymer is formulated as a block having a dimension of at least 10 mm and which comprises a wax matrix in which the polymer particles are dispersed. The block can be made by blending polymer powder with the molten wax matrix and cooling and solidifying it. The block is of particular value for releasing flocculant into a flowing stream of suspension.
Patent HU-T74734-A (HU)
Title: Use of biphenyl methyl imidazole derivatives for producing pharmaceutical compositions having ocular tension derpessant activity
Inventor: HOSOKAWA TSUNEMICHI
IPC: A61K31/41
Filed: 1995-03-16
Abstract: Use, in the manufacture of a medicament suitable for local application to the eyes for use in combination with a  beta -blocker for the treatment of ocular hypertension and/or glaucoma, of a compound of general formula (I): <CHEM>  wherein:   R<1> represents alkyl, alkenyl or a group of formula R<5>-A-B- (R<5> represents hydrogen, alkyl, cycloalkyl or aliphatic acyl, A represents oxygen or sulfur, and B represents a single bond or alkylene); R<2> represents alkyl, alkenyl or a group of formula -C(R<6>)(R<7>)(R<8>) (R<6> represents hydroxyl or alkoxy, and R<7> and R<8> represent hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, aryl or aralkyl); R<3> represents carboxyl or a group of formula -CON(R<9>)(R<10>) (R<9> and R<10> represent hydrogen or alkyl optionally substituted by 1 to 3 substituents from Substituent group (I)); and optionally substituted by 1 to 3 substituents from Substituent group (I)); and   R<4> represents carboxyl, carboxycarbonyl or tetrazol-5-yl; substituent group (I): aryl, 5- or 6-membered heteroaromatic ring group, halogen, hydroxyl, alkoxy, carboxyl, alkoxycarbonyl, amino, aliphatic acylamide and aromatic acylamide.
Patent IL-58256-A (IL)
Title: N-pyrrolyl-pyridazineamines,process for their manufacture and antihypertensive compositions containing them
IPC: A61K31/535
Filed: 1979-09-17
Abstract: New N-pyrrolyl-3-pyridazine-amines having a further aminic substituent in the 6 position of the formula (I), <CHEM> wherein R, R1, R2 and R3 are hydrogen or lower alkyl, R4 is e.g. hydrogen or lower alkyl, R5 and R6 are e.g. lower alkyl or taken together with the adjacent nitrogen atom represent a saturated 5 - 6 membered heterocyclic ring which may contain a further heteroatom, R7 and R8 represent hydrogen or, taken together, a 1,3-butadienylene radical forming a benzo system fused with the pyridazine ring, for example N-2,5-dimethyl-1H-pyrrol-1-yl)- 6-morpholino-3-pyridazineamine or N-(2,5-dimethyl-1H-pyrrol- 1-yl)-4-(4-hydroxypiperidino)-1-phthalazineamine, and their pharmaceutically acceptable salts are made e.g. by contacting a hydrazino derivate of the formula (II), wherein the substituents have the same meaning as above or an acid addition salt thereof with a dicarbonyl compound of the formula (III), wherein the substituents have the same meaning as above, or a functional derivative thereof in the presence of an acid catalyst at a temperature between 15 DEG C and 120 DEG C. The new compounds can be used as antihypertensive agents.
Patent IL-64432-A (IL)
Title: Applicator having a special shape for use with nose-clip
IPC: A61D7/00
Filed: 1981-12-01
Abstract: 1. A nose-clip with a bow (7), with means for receiving applicators (5) free from active substance, equipped with the applicators (5) which have a nearly triangular outline, and with reservoirs fixed thereon and containing active substance wherein the bow (7) is fixed near of one edge of each applicator whereby the sides of the triangle directed towards the bow (7) form an angle alpha of at least 40 degrees.
Patent IL-73800-A (IL)
Title: Parenteral parasiticidal compositions containing ivermectin and their preparation
IPC: A61K47/00
Filed: 1984-12-11
Abstract: Ivermectin, an antiparasitic agent which is insoluble and unstable in water, and other avermectin and milbemycin compounds, are formulated in glycerol formal and propylene glycol or in water and propylene glycol. These liquid formulations are suitable for parenteral administration for the treatment of parasitic infections and demonstrate improved efficacy and a broadened spectrum over previous formulations.
Patent IL-82659-A (IL)
Title: Bis(azolylmethyl)-aralkanols,their preparation and pharmaceutical compositions containing them
IPC: A61K31/41
Filed: 1987-05-27
Abstract: Heterocyclic compounds of the formula:- <CHEM> wherein X and Y, which may be the same or different, are each a =N- or =CH- group and R is a phenyl radical which optionally bears one or more substituents selected from halogen atoms, amino, cyano, carbamoyl, hydroxy and nitro radicals, 1-6C alkyl, halogenoalkyl, alkoxy, halogenoalkoxy and alkylamino radicals, di(1-6C alkyl)amino and 2-6C alkoxycarbonyl radicals, and n is 1 to 6, but excluding the compound wherein X and Y are each =N-, R is 2,4-dichlorophenyl and n is 1; and the pharmaceutically or veterinarily acceptable acid addition salts thereof; processes for their manufacture; and pharmaceutical and veterinary compositions containing them.
Patent JP-S55103658-A (JP)
Title: Diagnostic system
Inventor: KANAMARU KOUICHI
IPC: G06F11/00
Filed: 1979-01-31
Abstract: PURPOSE: To perform diagnosis without addition of a diagnostic hard circuit by utilizing features of a processing unit to diagnose the data buffer, the data bus, etc., of the processing unit.  
     CONSTITUTION: For execution of memory-memory-data instruction MOVE to transfer and write data of a designated address in main memory 3 to another address, data to be stored temporarily in write data buffer 12 is stored temporarily in one unused buffer of the first and the second read data buffers 1 and 2. After execution of instruction MOVE, corresponding data of buffers 1 and 2 is read selectively according to indication of point registers 6 and 7 and is supplied to respective input ends of comparator circuit 8. Then, circuit 8 compares data to decide on a basis of the coincidence decision whether buffers 1 and 2, buffer 12, etc., specially, of the processing unit are normal or not. Similar data comparison is repeated by movement of the indication position of registers 6 and 7. 
     COPYRIGHT: (C)1980,JPO&Japio
Patent JP-S62169482-A (JP)
Title: Manufacture of semiconductor device
Inventor: INOMATA HIRONORI
IPC: H01L21/338
Filed: 1986-01-22
Abstract: PURPOSE:To reduce a parasitic capacity between an Si substrate and a wiring electrode by a method wherein an insulating film is selectively formed on the Si substrate and the wiring electrode is formed n a GaAs layer region laminated on the insulating film. CONSTITUTION:An SiO2 film 2 is grown on the whole surface of an Si substrate 1 by a CVD method and the SiO2 film 2 at the programming region for forming an active layer is selectively etched to form an aperture 3 for exposing the Si substrate 1. A GaAs layer is grown using an MOCVD method to laminate a poly GaAs layer 4 on the SiO2 film 2 and to laminate a single crystal GaAs layer 5 on the substrate 1 in the aperture 3. Moreover, an impurity-doped GaAs layer is epitaxially grown n the single crystal GaAs layer 5 to form an N-type channel region 6. A gate electrode 7 is formed on the region 6, a source electrode 9 connected to the substrate through a contact hole 8 and a drain electrode 10 are formed and a wiring electrode 11 is formed on the poly GaAs layer 4 from the drain electrode 10 and the gate electrode 7.
Patent JP-H08294508-A (JP)
Title: Shade glasses
Inventor: KIN TOUSHIYU
IPC: G02C7/16
Filed: 1996-01-24
Abstract: PROBLEM TO BE SOLVED: To promote controlling power in the pupils of eyes due to the difference in light intensity, psychologically give an emotional relief and mentally concentrate by forming eye-shade to shield the light around the eyes by providing eye-shade spectacles main body which is made of a paper-made case foldable back and forth or up and down around periphery of the eyeballs while the front and back openings remain as a natural space. SOLUTION: A paper-made case forming a square or an oval cylinder-shape space is positioned before eyes to promote a view increasing effect obtained from light intensity by certainly forming eye-shade to shield the four sides around the eyes. In the eye-shade spectacles main body constructed by the paper-made case of the square cylinder-shape of which front and back surfaces are penetrated, four corners 11, 11', 11", 11''' can be folded or opened, and foldable center lines 2, 2' on right and left sides are formed thereon. The eye- shade spectacles main body 1 of the square cylinder-shape can be used in such a manner that a spectacle suspension or a band 5 for wearing it on the head is attached to the right and the left sides of the backward opening side of the square cylinder. A nose suspension groove may be preferably formed at a region attached to the nose.
Patent JP-S62171861-A (JP)
Title: Paper sheet accumulating apparatus
Inventor: NAGASAWA YUTAKA
IPC: B65H29/40
Filed: 1986-01-22
Abstract: PURPOSE:To certainly accumulate the paper sheets having the sufficient softness by arranging a paper sheet feeding means which compulsorily pushes the paper sheets into between the vanes of two vane wheels arranged in parallel so as to be retracted inside the vanes. CONSTITUTION:The transported paper money B is nipped between pulleys 4A, 5A, and 8A and sent towards the vane wheels 1 arranged in parallel and inserted into between the vanes 1A. Since a belt 8C is positioned at the inwardly retracted position opposed to the vane 1A, the paper money B is compulsorily shifted towards between the vanes 1A, and can be certainly pushed in. Even if the paper money having breakage or folds generated is inserted into between the vanes 1A, the paper money can be certainly guided into the vanes 1A by the belt 8C and can be pushed in. Therefore, even if the paper money having the sufficient softness or the paper money having folds or breakage is supplied, said paper money can be certainly taken into the vanes,and the reliability of accumulation can be improved.
Patent JP-S5294152-A (JP)
Title: Optical detector
Inventor: AKITA KIMIO
IPC: H01H47/24
Filed: 1976-02-04
Abstract: PURPOSE: To provide a reflection plate on a light path and to interrupt emitted by a light emitting device at least twice by the material to be detected so that the reduction quentity of light volume at the detector device is increased to permit even semitransparent materials to be detected. 
     COPYRIGHT: (C)1977,JPO&Japio
Patent JP-H11215204-A (JP)
Title: Data transmitter and its method
Inventor: MAEDA YASUYORI
IPC: H04L12/70
Filed: 1998-01-22
Abstract: PROBLEM TO BE SOLVED: To attain high speed processing that divides terminal data, adds protocol control information to the data and that generates packets while using a main memory. SOLUTION: A transmission terminal data memory means 21 stores terminal data. A divided data selection means 22 selects sequentially divided data that are to be transmitted. A divided data packet processing means 23 generates protocol control information of the selected divided data and writes the information in front of a head of the divided data or behind an end of the divided data in the transmission terminal data memory means 21 to generate packets. Data that are destroyed by the write of the protocol control information are read before the write and saved in a save data memory means 25 and restored to the original data position later. A packet transmission means 24 reads the protocol control information and the divided data in the lump from the transmission terminal data memory means 21 as one packet and sends them to a transmission line.
Patent JP-S62168481-A (JP)
Title: Video signal processor
Inventor: TAKAYAMA MAKOTO
IPC: H04N5/04
Filed: 1986-01-20
Abstract: PURPOSE:To facilitate a noise-countermeasure in the processing of a video signal by counting horizontal synchronizing signals or signals synchronized with them, comparing the counting value of said counting with a prescribed value to detect the noise, and thereby providing an accurate detecting of the noise. CONSTITUTION:The horizontal synchronizing signal 1 and a vertical synchronizing signal 2 are inputted to a counter 6, and the counter 6 counts the number of the horizontal synchronizing signals during the period of the vertical synchronizing signal 2. The output of the counter 6 is inputted to a memory 7 and a comparator 8. Since the result of the counter 6 preceding one-field is stored in the memory 7, the comparator 8 detects the coincidence between the output of the counter 6 preceding one-field and the current output of the counter 6. In case the detection result is in dissidence, the comparator 8 outputs an error output 9 indicating that there is an influence of noise. In this way, an accurage detection of the noise is made possible.
Patent JP-S63177989-A (JP)
Title: Work positioning device
Inventor: FUJIKOSHI NOZOMI
IPC: B23K26/02
Filed: 1987-01-20
Abstract: PURPOSE:To improve the accuracy in positioning by providing the work positioning jig movable in parallel in the coordinate axial direction for a work table and arranging the NC control device performing the storage of the movement amt. of the jig and the reading of an original coordinate as well. CONSTITUTION:The work positioning jigs 6, 7 moving in parallel in X axial direction and Y axial direction respectively on a work table 1 are provided and the NC control device storing the moving amt. of the jigs 6, 7 and capable of reading the original coordinate of a work 5 as the intersection point thereof is provided as well. In case of performing the positioning of the work 5 a work head is first moved to an original point. The jigs 7, 6 are then moved and after storing the movement amt. to a control device moved to a refuge position. The work head is thereafter moved to the stored original point 8 of the jigs 6, 7 to process the work 5 according to the program. Owing to the positioning at the work starting point becoming correct the positioning accuracy is improved.
Patent JP-H09204383-A (JP)
Title: Client, server terminal connection method and client terminal equipment
Inventor: ASADA JUNICHI
IPC: H04L12/28
Filed: 1996-01-25
Abstract: PROBLEM TO BE SOLVED: To use the server of lightest loads on a LAN and to introduce a batch processing. SOLUTION: A client terminal 1 gathers load information from server terminals 20, 21 and 22 by a load information gathering means 2, obtains the average load rates of the respective server terminals from the information by a calculation means 3, selects the server terminal of the lightest loads by a comparison and selection means 4 and connects the server terminal. As a result, an effect capable of executing an application faster is provided. Also, the presence/absence of the space of an application execution licence is checked by an application execution information gathering means 6 from the connected server terminal 21, and when no space is present in the licence, the batch processing is set and the application is executed. As a result, the need of an operation manually repeatedly executed before until the licence becomes free is eliminated.
Patent JP-H02189247-A (JP)
Title: Outer mirror for automobile
Inventor: OGASAWARA MORIHIKO
IPC: F16H25/20
Filed: 1989-01-18
Abstract: PURPOSE:To obtain such a transfer that is stable in driving force by forming a driving force transfer thread part in an operating screw shaft, and engaging an engaging member, where a nut member being rotated by a driver is engaged, with this thread part, in a device which tilts a mirror holder by longitudinal motion of the operating screw shaft. CONSTITUTION:A mirror holder 1 supporting a mirror body is supported free of tilting motion around a horizontal and vertical tilting center axis to a mirror case, and a heat part 4b at a tip of a leg part 4a of an operating screw shaft 4 installed free of longitudinal motion in the mirror case in the axial direction is attached to the mirror holder 1 free of tilting motion. Then, a nut member 7 being rotated by a driver in the mirror cases is engaged with the leg part 4a of the operating screw shaft 4 via an engaging member 10 and thereby this operating screw shaft 4 is made so as to do longitudinal motion in the axial direction, but at this time, a driving force transfer thread part 4d is formed in a specified spot on an outer circumferential surface of the leg part 4a of the operating screw shaft 4, and only this thread part 4d is made so as to be fitted in the engaging member 10.
Patent JP-H03215891-A (JP)
Title: Information input device
Inventor: ISHII TOSHIYUKI
IPC: G06F3/048
Filed: 1990-01-21
Abstract: PURPOSE:To enable a user to grasp the operation state of an equipment main body instinctively by displaying guide characters on the same display screen with interactive display elements when the interactive display elements are displayed to the user by using the display screen. CONSTITUTION:The information input device which prompts the user to responding operation by displaying the interactive display elements AR1 and AR3 indicating the operation state of the electronic equipment main body 3 on display screens 4A and 6A is provided with a character display means 8 which displays personified guide characters CH indicating operation or expression corresponding to the display contents of the interactive display elements AR1 and AR3 at the positions in the display screens 4A and 6A corresponding to the interactive display elements AR1 and AR3. When the interactive display elements AR1 and AR3 are displayed to the user, the guide characters CH showing the operation or expression corresponding to the display contents are displayed, so the user can grasp the operation state of the electronic equipment main body 3 instinctively with easy with the guide characters CH.
Patent JP-H07222245-A (JP)
Title: Radio communication system
Inventor: YANO MOTOMITSU
IPC: H04W72/04
Filed: 1994-02-02
Abstract: PURPOSE:To enable high-quality data transmission without necessity to previously grasp conditions such as traffic. CONSTITUTION:At each radio communication terminal, the list of service areas, to which the terminal itself can belong, is prepared when turning on a power source and moving between the service areas, that list is stored in the memory of a service area control part 31, afterwards, the state of the belonging service area is decided by monitoring a packet collision rate or a bit error rate and when it is judged that the transmission quality can not be mainstained, based on this list, the service area at the belonging destination is switched to the next candidate.
Patent JP-S54105608-A (JP)
Title: Exhaust gas purifier for internal combustion engine
Inventor: TSUJI RIICHI
IPC: F01N3/10
Filed: 1978-02-04
Abstract: PURPOSE: To enable a secondary air flow control in a skipping manner in an internal combustion engine by constituting an exhaust gas purifier therefor such that a negative pressure control valve is provided with, in addition to a first diaphragm, a second spring-urged diaphragm so that a negative pressure control chamber can be changed over to communicate alternatively to the atmospheric air and negative pressure of the exhaust system in synchronism with operations of a negative pressure change-over valve.  
     CONSTITUTION: A negative pressure control mechanism 70 has a negative pressure chamber 76 of a constant volume below a diaphragm 74 which is urged downwardly by a spring 72. A spacing 75 above the diaphram 74 is changed over to communicate alternatively to the atmospheric air and negative pressure by means of a second negative pressure change-over valve 80. When skipping increase of secondary air supply is required, a signal is transmitted from a control circuit 64 to the valve 80 so that a common port 84 is communicated to a first change-over port 88. As a result, a negative pressure signal is introduced into the spacing 75 through a pipe 86, the ports 88, 84, and another pipe 82 so that the volume of the skipping control chamber 76 is rapidly increased to thereby move a valve body 30 instantaneously. Thus, a skipping increase feature of secondary air flow from an air chamber 24 to a nozzle 25 through a chamber 26 can be attained thereby. 
     COPYRIGHT: (C)1979,JPO&Japio
Patent JP-S56109097-A (JP)
Title: Diaphragm plate for speaker and its manufacture
Inventor: YAMAMOTO TOORU
IPC: H04R7/02
Filed: 1980-01-31
Abstract: PURPOSE:To enable to continuously manufacture a diaphragm plate of sandwich construction in high speed and to foam uniformly the foaming sheet, by laminating a surface member on the surface of a core made of foaming sheet. CONSTITUTION:When the surface member sheet 1 passes between rollers 3, 3' heated to about 120 deg.C wrapped on the surface of the core sheet 2, the both sheets 1, 2 are molten. The composite sheet 6 made of laminated core sheet 2 and surface  member sheet 1 with the heat of the rollers 3, 3' is heated for several seconds at  about 180 deg.C with the heaters 4, 4'. Since the foaming member in the core sheet 2 is  heated more than foaming start temperature with the heat of the heaters 4, 4', it is  foamed and polyethylene short fibers in the surface member sheet 1 and polyethylene being the base material of the core sheet 2 are molten. The composite sheet  6 foamed and softened with the heaters 4, 4' is cold-pressed with metal molds 5, 5'  and formed into the shape of diaphragm plate.