baber/WOPTO huggingface dataset:
Patent IL-149904-A0 (IL)
Title: Amycomycin, a process for its production and its use as a pharmaceutical
IPC: A61K31/4015
Filed: 2000-11-25
Abstract: A compound named Amycomycin of the formula: <CHEM> and its pharmaceutically acceptable salts and derivatives, in all their stereoisomeric and tautomeric forms is obtainable by cultivation of the microorganism Amycolatopsis sp., ST101170 (DSM 12216) and finds use a pharmaceutical, particularly as an antibiotic.
Patent IL-153980-A0 (IL)
Title: Process for the preparation of 2-(6-substituted-1,3-dioxane-4-yl) acetic acid derivatives
IPC: C07D309/30
Filed: 2001-07-12
Abstract: The invention relates to the preparation of 2-(6-substituted-1,3-dioxane-4-yl)acetic acid derivatives of formula 1, where X stands for a leaving group, and R 1 , R 2 , and R 3  each independently stand for an alkyl group with 1-3 carbon atoms from 4-hydroxy-6-X-substituted-methyl-tetrahydropyran-2-one compounds, where X is as defined above, with the aid of an acetalization agent, in the presence of an acid catalyst.  The invention also relates to the novel compounds of formula 1 as well as salts and acids to be prepared from these, with the OR 3  group in formula 1 being replaced by an OY group, where X, R 1  and R 2  have the meanings defined above and where Y stands for an alkaline (earth) metal or a substituted or unsubstituted ammonium group or stands for hydrogen, and to the novel compounds of formula 2.  The products concerned are, after conversion into the t-butyl ester of 2-(6-hydroxymethyl-1,3-dioxane-4-yl)acetic acid, important as intermediary products in the preparation of statins.
Patent IL-159711-A0 (IL)
Title: System for directional angle aiming of weapon
IPC: F41A27/08
Filed: 2002-07-15
Abstract: A traverse laying system for a weapon integral with a frame articulated in traverse with respect to a support providing a large traverse range around a first axis of rotation. The system includes positioning device for the weapon integral with the frame in order to ensure a small lateral range of the weapon around a second axis of rotation passing through the centre of gravity and perpendicular respectively to the longitudinal axis of the weapon and the traverse orientation axis. The first axis of rotation is located to the rear of the weapon's centre of gravity and the lateral range around the second axis may be of around 2°.
Patent IL-160323-A0 (IL)
Title: Droplet deposition apparatus
IPC: B41J2/17
Filed: 2002-09-05
Abstract: An ink supply system for a droplet deposition apparatus wherein the pressure at the nozzle is controlled by a remote point, said remote point being positioned in parallel with said print head. The flow restrictions in the printhead arm and the pressure control arm of the circuit being selected to achieve this.
Patent IL-166704-A0 (IL)
Title: Regulated gas supply system
IPC: F41A33/06
Filed: 2005-02-06
Abstract: A removable gas supply for a weapon simulator, wherein the gas system cycles the bolt or slide of the firearm to provide recoil, actuate a hammer/trigger mechanism and provide realism of the original weapon functions. The weapon simulator has a housing defining a piston chamber and a piston positioned in said chamber and connected to the bolt. The simulator also includes a valve chamber in the housing connected with said regulated gas supply and said bolt, and a recoil valve positioned in the valve chamber to control the release of gas from said regulated gas supply to said piston chamber to generate recoil in the weapon simulator.
Patent IL-174960-A0 (IL)
Title: Process for the preparation of (3r,3as,6ar)-hexahydrofuro [2,3-b] furan-3-yl (1s,2r)-3-[[(4-aminophenyl) sulfonyl] (isobutyl) amino]-1-benzyl-2-hydroxypropylcarbamate
IPC: C07D493/04
Filed: 2006-04-11
Abstract: The present invention relates to a process for the preparation of (3R,3aS,6aR)­-hexahydrofuro [2,3-b] furan-3-yl (1S,2R)-3-[[(4-aminophenyl) sulfonyl] (isobutyl) amino]-1-benzyl-2-hydroxypropylcarbamate as well as intermediates for use in said process. More in particular the invention relates to processes for the preparation of (3R,3aS,6aR)-hexahydrofuro [2,3-b] furan-3-yl (1S,2R)-3-[[(4-aminophenyl) sulfonyl] (isobutyl) amino]-1-benzyl-2-hydroxypropylcarbamate which make use of 4-amino-N­ ((2R,3S)-3-amino-2-hydroxy-4-phenylbutyl)-N-(isobutyl)benzene sulfonamide intermediate, and to processes amenable to industrial scaling up. (3R,3aS,6aR)-hexahydrofuro [2,3-b] furan-3-yl (1S,2R)-3-[[(4-aminophenyl) sulfonyl] (isobutyl) amino]-1-benzyl-2-hydroxypropylcarbamate is particularly useful as HIV protease inhibitors.
Patent IL-189325-A0 (IL)
Title: Moldable fabric with variable constituents
IPC: B32B7/027
Filed: 2008-02-06
Abstract: A woven mat fabric with fused layers containing a plurality of woven layers, where each woven layer contains a plurality of warp elements interwoven with a plurality of weft elements. The warp and weft elements contain polymeric strips which have a core layer disposed in layered relation with at least one surface layer. The core layer contains a first strain oriented polymer composition and having a first softening point and the surface layer contains a second polymer composition having a softening point lower than the first softening point. The weft and warp elements within each layer are fused to one another, but the weft and warp elements of one layer are not consolidated to the weft and warp elements of the adjacent layers.
Patent IL-211035-A0 (IL)
Title: Container having a lid
Filed: 2011-02-03
Abstract: The invention relates to a lidded container for storing and transporting in particular hazardous liquid fill goods, including an outer container body, an upper container lid and an inserted thin-walled inliner. The container lid has at least one filling and emptying opening that can be closed in a gas and liquid tight manner and that, for example, can be attached by means of a U-shaped tension ring closure or without tension ring as a snap cover by means of snap closure or a screw cap by means of screw closure on the upper container opening of the container body on a correspondingly designed flange edge. The thin-walled inliner (26) is fixed on the bottom side of the container lid (14) in the outer peripheral region in a gas and liquid tight manner, wherein the container lid (14) and inliner (26) form a gas and liquid tight hollow body unit. The container body, which can be used multiple times, is only provided as a support and protection unit for the inliner.
Patent RO-131229-A0 (RO)
Title: Composition for fireproofing textiles
Inventor: FLORIŢA ŞERBAN-MIHAI
IPC: D01F1/07
Filed: 2016-01-06
Abstract: The invention relates to a composition for fireproofing textiles. According to the invention, the composition is an antipyrene aqueous solution containing a homogeneous phase consisting of ammonium or polyammonium metaphosphate, orthophosphate, pyrophosphate or polyphosphate, a polyamide, preferably carbodiamide, boric acid and/or an alkaline polyborate; two hydrosoluble alkaline salts, A and B, preferably lithium chloride and potassium chloride, and a disperse phase consisting of a phosphoric acid/carbodiamide adduct doped with ammonium vanadate and silicon dioxide nanocrystals, where the elements: nitrogen from the ammonium ion : amide nitrogen : phosphorus : boron : alkaline cation in A : alkaline cation in B : silicon : vanadium are in a ratio of 15...16 : 17.1...18.2 : 8.3...8.9 : 0.5...2 : 0.8...1 : 0.9...1.1 : 0.1...0.5 : 0.05...0.15 and the concentration of the aqueous solution components, in the homogeneous phase and the disperse phase, is of 12...22% by weight.
Patent RO-134158-A0 (RO)
Title: Rotary shears for harvesting biomass from forestry and agricultural crops
Inventor: TUDOSOIU CĂTĂLIN
IPC: A01D34/64
Filed: 2020-01-20
Abstract: The invention relates to a rotary shear for harvesting biomass from forestry and/or agricultural crops, driven by a general purpose power tiller or a low capacity universal tractor. According to the invention, the shear consists of a moulded housing (1) in which a main shaft (2) is mounted longitudinally, in the extension of which is arranged a non-detachable stiffened conical toothed pinion (3), which engages an upper conical toothed pinion (8), assembled on a vertical inner shaft (7), transmitting it a direction of rotation and engaging further a lower conical toothed pinion (15), detachably assembled on a vertical outer shaft (14), transmitting it a rotation direction opposite to the upper pinion (8), the concentricity and equidistance during the opposite rotation of the outer shaft (14) and inner shaft (7) being carried out by means of some rolling bearings (20), which transmit the rotational movement to an upper rotary knife (23), and the rotational movement, in the opposite direction, to a lower knife (24), respectvely, the shafts (7 and 14) in rotational movement being protected by means of a protective guard (27), the knives (23 and 24) being driven into a shearing process carried out in a plane parallel with the plane determined by the ground, cutting the lignified vegetation between the two knives (23 and 24) which rotate in opposite directions.
Patent RO-137739-A0 (RO)
Title: Food product based on yoghurt, pollen and honey and preparation process thereof
Inventor: COJOCARU AURELIAN- COSMIN
IPC: A23L2/00
Filed: 2023-01-26
Abstract: The invention relates to a food product rich in nutritive substances, vitamins and minerals, with body regenerative and energizing properties, based on pollen, honey and bio yoghurt and to a process for preparing the same. According to the invention, the food product is a mixture made of 3 parts of raw pollen granules, 7 parts of non-thermally treated honey, and 90 parts of creamy bio yoghurt with 4% fat, the parts being expressed by weight, the resulted mixture being a viscous fluid of white-yellowish colour in which the whole pollen granules can be seen. The claimed preparation process consists in introducing the pollen granules into a sterilized glass container, over which the honey is poured, and, by vibration and slight rotation of the container, the whole pollen granules complete incorporation and sealing into the honey is aimed, afterwards the creamy bio yoghurt of 4% fat is poured over the resulted mixture, while slowly stirring only until the mixture becomes slightly yellowish and the whole pollen granules can still be seen.
Patent AP-2000001856-A0 (AP)
Title: Prodrugs of aspartyl protease inhibitors.
Inventor: TUNG ROGER D
IPC: C07F9/655
Filed: 1998-12-23
Abstract: The present invention relates to prodrugs of a class of sulfonamides which are aspartyl protease inhibitors. In one embodiment, this invention relates to a novel class of prodrugs of hiv aspartyl protease inhibitors characterized by favorable aqueous solubility, high oral bioavailability and facile in vivo generation of the active ingredient. This invention also relates to pharmaceutical compositions comprising these prodrugs. The prodrugs and pharmaceutical compositions of this invnetion are particularly well suited for decreasing the pill burden and increasing patient compliance. This invention also relates to methods of treating mammals with these prodrugs and pharmaceutical compositions.
Patent AP-2001002192-A0 (AP)
Title: Substituted bicyclic derivatives for the treatment of abnormal cell growth.
Inventor: KATH JOHN CHARLES
IPC: A61P5/28
Filed: 2001-06-14
Abstract: The invention relates to compounds of the formula 1 and pharmaceutically acceptable salts, prodrugs and solvates thereof, wherein r1, r3, r4, r5, r11, m and p ae as defined herein. The invention also relates to methods of treating abnormal cel growth in mammals by administering the compounds of formula 1 and to pharmaceutical compositions for treating such disorders which contain the compounds of formula 1. The invention also relates to methods of preparing the compounds of formula 1.
Patent IE-910047-A1 (IE)
Title: The diastereoselective preparation of phosphinate esters
Inventor: SEDERGRAN THOMAS C
IPC: A61P9/12
Filed: 1991-01-07
Abstract: An increase in the diastereoselectivity resulting from the reaction of a phosphinic acid ester of the formula <CHEM>  with the halo ester of the formula <CHEM> is achieved by carrying out the reaction in the presence of 4-methylmorpholine, diazabicyclooctane, quinuclidine, 1-methylpyrolidine, or cinchonidine. After removal of the R3 protecting group and fractional crystallization, the resulting desired diastereomeric pair can be resolved, and the desired isomer can be coupled to 4-substituted L-proline to give compounds possessing angiotensin converting enzyme inhibition activity. In particular, the process is useful in producing the antihypertensive agent fosinopril sodium in increased yields.
Patent LU-87941-A1 (LU)
Title: Damper unit for shoes
Inventor: MOYA MARIANO BERNABEU
IPC: A43B21/28
Filed: 1991-05-22
Abstract: The absorbent, for general use and esp. as bedding for animals, is treated with a poly-hydroxylated organic cpd. which acts as a binder for residual fine particles with size below ASTM 400 mesh. The granular absorbent obtained does not release powder during pouring, decanting, etc. The fraction below 400 mesh is less than 0.2%.***.
Patent MA-21342-A1 (MA)
Inventor: CHEE-HWAY TSAI
IPC: A23L1/304
Filed: 1988-07-29
Abstract: Beverages and beverage concentrates nutritionally supplemented with significant levels of solubilized calcium and containing low levels of sulfate, preferably in combination with low levels of chloride, are disclosed. These beverages and concentrates also contain specified levels of edible acids selected from phosphoric acid, citric acid, malic acid, fumaric acid, adipic acid, gluconic acid, and lactic acid, as well as mixtures of these acids. The particular acid systems are selected to provide the desired flavor and sourness character for the beverages and concentrates. Inclusion of low levels of sulfate/chloride in these beverages and concentrates provides a quicker onset of sourness, prevents or reduces aftertaste effects and improves the solubility of the calcium, particularly when high levels of phosphoric acid or citric acid are used. Inclusion of sulfate/chloride also prevents or reduces the precipitation and deposition of calcium salts on equipment surfaces during the pasteurization or sterilization of calcium-containing fruit juice beverages.
Patent MA-23688-A1 (MA)
Inventor: GREGORY P BIDINGER
IPC: C09D133/06
Filed: 1995-10-09
Abstract: A method for polymerizing predominantly one or more acrylate and/or vinyl acetate monomers in the presence of a latex results in high solids dispersions of polymer particles with lower viscosities than traditionally observed. A significant wt. % of added monomers can be present in large particles, having nonspherical shapes. Some of the original latex particles are retained during the polymerization and these increase the solids content and lower the viscosity by packing in the interstices between large particles. The total polymer solids content can easily be varied from 70 to 92 or more wt. % which are higher than achieved in any previously reported aqueous polymerizations. The viscosities at very high solids contents become paste-like but the materials still are stable to storage and further handling without breaking the dispersion into an agglomerated polymer portion and released water. The dispersions are useful to form sealants, membranes, etc., either with or without other additives. A preferred use is as an acrylate water-based caulking compound where the high solids and thixotropy of the dispersion allows for formation of a water-based caulk with low shrinkage.
Patent MA-26744-A1 (MA)
Title: Polymorphes d'un chlorhydrate d'azo-bicyclo-2,2,2-oct-3-ylamine cristallins et compositions pharmaceutiques les contenant
Inventor: DOUGLAS JOHN MELDRUM ALLEN
IPC: C07D453/02
Filed: 2000-06-21
Abstract: DEUX FORMES POLYMORPHES CRISTALLINES DU DICHLORHYDRATE DIHYDRATÉ DE LA (2 - BENZHYDRYL - 1- AZO - BICYCLO  [ 2 ,  2 ,  2 ]  OCT - 3 - YL )  -  ( 5 -ISOPROPYL - 2 - MÉTHOXYBENZYL ) - AMINE SONT LA FORME  I  ET LA FORME II.  LA COMPOSITION  PHARMACEUTIQUE COMPRENANT AU MOINS L'UN DE CES POLYMORPHES  PRÉSENTE UNE STABILKITÉ AVANTAGEUSE  POUR LA FORMULAYION EN VUE DU TRAITEMENT DE L'ÉMèSE CHEZ DES PATIENTS SOUMIS  à UNE CHIMIOTHARAPIE.  L'ADMINISTRATION DE CETTE COMPOSITION PHARMACEUTIQUE S'EFFECTUE DE FAÇON CLASSIQUE PAR VOIE ORALE,  AVANTAGESEMENT SOUS FORMES DE COMPRIMÉS OU GÉLULES,  OU PAR VOIE INTRAVEINEUSES.  UN PROCÉDÉ DE PRODUCTION DES FORMES I ET II  EST ÉGALEMENT PROPOSÉ.
Patent MA-20150044-A1 (MA)
Inventor: BOURZEIX FRANÇOIS
IPC: G06T7/20
Filed: 2013-07-08
Abstract: يقدم هذا الاختراع نظاما لتقدير سرعة العربات بالإعتماد على حساب السرعة المجسمية، يتالف هذا الاختراع من كاميرتين (105 و 110) متصلتين بحاسوب مزود ببطاقة للحساب يسمح بتقدير السرعة على عكس الأجهزة المزوة بكاميرا واحدة فهذا النظام لا يحتاج الى اي تعديل و لا ضبط للصورة و قد تم انجاز هذا الجهاز بالإعتماد على تقنية تصوير ثلاثي الأبعاد باستعمال كاميرتين مثنتتين افقيا موجهتين نحو نفس الهدف و المعلومات التي يتم استخلاسها من الصور تسمح بتحديد المسافة بين الشيئين
Patent MA-20150250-A1 (MA)
Inventor: ABDELLATIF BENABDELLAH
IPC: A61J9/00
Filed: 2013-11-25
Abstract: Afin d’éviter les accidents de brulures chez les nourrissons, nous proposons une nouvelle conception d’un biberon intelligent. L\/luni d’un systeme de verrouillage constitué d’un diaphragme ia base d’un alliage a mémoire de forme amf. Cet alliage est concu de telle sorte que sa température critique tc soit d'environs 40 °c. Des que tc est atteinte, l'alliage se déforme et active le diaphragme situé juste en dessous de la tétine et bloque le liquide chaud de sortir. Le diaphragme s'ouvre a l'aide de l’a|vlf par retour a son état initial une fois la temperature atteint un niveau inférieur a tc.
Patent MA-38251-A1 (MA)
Title: Element de construction et procede de montage d'un tel element de construction
Inventor: LARAKI MOHAMED
IPC: E04B5/08
Filed: 2015-07-08
Abstract: L'invention concerne un élément de construction comprenant au moins deux poutrelles (2) et au moins un entrevous (6) agencés entre lesdites poutrelles. Selon l'invention, chaque entrevous a une section transversale rectangulaire de sorte que des coins opposés de chaque entrevous soient logés dans des coins correspondants des poutrelles, les poutrelles étant constituées d'un ou de deux profilés, les profilés des différentes poutrelles étant au moins solidarisés deux par deux par au moins un organe de connexion appartenant à l'élément de construction. L'invention concerne également un procédé de montage d'un tel élément de construction.
Patent UY-27018-A1 (UY)
Title: Derivados de la pirimidina
Inventor: DAUTZENBERG F
IPC: A61K31/337
Filed: 2001-11-09
Abstract: Compuestos de la fórmula (I), así como los esteres y las sales farmacéuticamente utilizables de los mismos, en donde R1,R2,R3,R4,A1 y A2 tienen el significado dado en la reivindicación 1, que se pueden usar en forma de preparaciones farmacéuticas para el tratamiento o prevención de artritis, diabetes, trastornos alimentarios y obesidad.
Patent UY-31064-A1 (UY)
Title: Vacuna
Inventor: POOLMAN JAN DR
IPC: A61K38/16
Filed: 2008-04-30
Abstract: La presente invención se refiera al campo de las vacunas y en particular a vacunas combinadas y calendarios de administración conjunta. Los presentes inventores describen que el uso excesivo de CRM en las vacunas pediátricas puede provocar interferencia inmunitaria inespecífica con ciertos anfígenos y proporcionan soluciones a este problema.
Patent UY-31215-A1 (UY)
Title: Compuestos de morfolino pirimidina, procesos para su preparacion, composiciones farmacéuticas conteniéndolos y su uso en terapia.
Inventor: PIKE KURT GORDON
IPC: A61K31/506
Filed: 2008-07-09
Abstract: Un compuesto de formula (I) o una sal farmacéuticamente aceptable del mismo, procesos para su preparacion, composiciones farmacéuticas que los contienen y su uso en terapia, por ejemplo en el tratamiento de una enfermedad proliferativa tal como el cáncer y particularmente en una enfermedad mediada por una mTOR y7/o una o más enzimas PI3K.
Patent ES-179088-A1 (ES)
Title: UN APARATO PLANEADOR AUTOMáTICO
Filed: 1947-07-14
Abstract: Un aparato planeador automático que funciona por la acción de la gravedad que esencialmente se caracteriza en que el descenso rotativo del brazo porta-aviones tiene lugar a lo largo de un árbol vertical constituido por espiras helicoidales en las cuales toma apoyo un agujero ovalado que a modo de tuerca presenta el citado brazo siendo dicho brazo porta-aviones retenido al fina de su carrera de descenso por un resorte o muelle llevado por el zócalo del aparato resorte o muelle que si interesa sirve igualmente para el remontado del citado brazo.
Patent ES-190754-A1 (ES)
Title: Un procedimiento para fabricar azul de ultramar
Filed: 1949-12-10
Abstract: Procedimiento para fabricar azul de ultramar caracterizado por el hecho de calentar una mezcla que contiene un silicato de aluminio o una o más sustancias capaces de reaccionar a la temperatura de operación para formar un silicato de aluminio azufre y una sal orgánica de un metal alcalino o alcalino terroso en ausencia de condiciones oxidantes a una temepratura superior a los 600ºC. preferiblemente del orden de 750 a 900ºC. desde 20 minutos a 3 horas cambiando el ambiente para conseguir una atmósfera de condiciones oxidantes continuando el calentamiento bajo dichas condiciones oxidantes a una temperatura del orden de 450 a 600º C. durante un periodo entre media hora y tres horas y enfriando y lavando el producto resultante.
Patent ES-253742-A1 (ES)
Title: Improvements in or relating to the preparation of beverages
IPC: A23L2/06
Filed: 1959-11-26
Abstract: Whole citrus fruit, e.g. oranges, is comminuted, the comminuted fruit is agitated in a quantity of a hot liquid, such as sugar syrup, to effect rapid extraction of the fruit and the resultant dispersion, whilst still hot, is mixed with a substantial volume of a cold or chilled liquid. The process is described with reference to apparatus described and claimed in Specification 866,689. A formulation for orangeade is given.
Patent ES-257195-A1 (ES)
Title: Improvements in or relating to incandescent lamps
IPC: H01K1/46
Filed: 1960-04-07
Abstract: A hollow cylinder of an insulating foam producing composition consisting of novolak, hexamethylene tetramine and a filler such as calcium carbonate woodmeal or gypsum is inserted into the cap of an incandescent lamp and converted to foam during the cementing operation for securing the cap to the bulb. In an example, a mixture of 5 parts novolak, 1 part hexamethylene tetramine, 8 parts dolomite and 0,5 parts woodmeal is used.ALSO:A hollow cylinder of an insulating foam producing composition consisting of Novolak, hexamethylene tetramine and a filler such as calcium carbonate, woodmeal or gypsum is inserted into the cap of an incandescent lamp and converted to foam during the cementing operation for securing the cap to the bulb. In an example, a mixture of 5 parts Novolak, 1 part hexamethylene tetramine, 8 parts dolomite and 0,5 parts woodmeal is used.