baber/WOPTO huggingface dataset:
Patent ES-2204303-B2 (ES)
Inventor: ARMENGOL ASPARO MONTSERRAT
IPC: C07D249/08
Filed: 2002-08-07
Granted: 2004-12-16
Abstract: In particular, rizatriptan or a pharmaceutically acceptable salt thereof, which includes a) Preparation of the diazonium salt of aniline hydrochloride (II); followed by reduction and acidification to give the hydrazine (III); b) reaction in situ of the hydrazine hydrochloride (III) with alpha-keto-delta-valerolactone, to give the hydrazone (IV); c) Fischer indole reaction of the hydrazone (IV), to give the pyranoindolone (V), optionally followed by a hydrolysis reaction to give (VI); d) Transesterification of (V) or esterification of its hydrolysis product (VI), to give (VII), where R means straight or branched C1-C4 alkyl chain; e) Conversion of the hydroxyl group of (VII) into dimethylamino, to give the indolecarboxylate (VIII), where R has the meaning defined above; f) Saponification of the 2-carboalkoxy group of (VIII) to give indolecarboxylic acid (IX); and g) Decarboxylaton of the indolecarboxylic acid (IX) to give rizatriptan and, eventually, to obtain a pharmaceutically acceptable salt thereof. The invention also relates to synthesis intermediates to obtain rizatriptan.
Patent ES-2281274-B2 (ES)
Title: Peptidos ciclicos antimicrobianos.
Inventor: BARDAJI RODRIGUEZ EDUARD
IPC: A01N37/44
Filed: 2005-12-21
Granted: 2008-07-16
Abstract: La presente invención se refiere a nuevos péptidos cíclicos que tienen propiedades antimicrobianas. Dichos péptidos tienen un número par de aminoácidos comprendido entre 4 y 10, y un contenido molar de lisina comprendido entre el 40% y el 60%. La invención describe la síntesis y la utilización de los mencionados péptidos como agentes antimicrobianos frente a bacterias y hongos patógenos para plantas. También se refiere a composiciones que comprenden dichos péptidos y un agente auxiliar, y a un método para prevenir y tratar infecciones y enfermedades de las plantas provocadas por bacterias y hongos patógenos.
Patent ES-2577881-B2 (ES)
Title: Sistema inalámbrico distribuido y procedimiento para la clasificación y localización de faltas en una red de distribución eléctrica subterránea
Inventor: LEON DE MORA CARLOS
IPC: H04W88/00
Filed: 2015-01-16
Granted: 2016-11-03
Abstract: Sistema inalámbrico distribuido y procedimiento para la clasificación y localización de faltas en una red de distribución eléctrica subterránea. El sistema comprende dispositivos sensores (3), conformando una red de sensores inalámbricos (2), distribuidos en la red de distribución eléctrica subterránea (1) y acoplados a conductores (7) de la red (1) de forma que todos los tramos de conductores entre bifurcaciones tienen asociados un dispositivo sensor (3). Los dispositivos sensores (3) comprenden medios de medición de la corriente (34) que circula por el conductor (7), estando sincronizados entre sí y configurados para identificar el tipo de falta originada y la localización de la misma mediante el intercambio de mensajes, entre los distintos dispositivos sensores (3), con información de las medidas de corriente sincronizadas y mediante el análisis de la información fasorial de dichas medidas de corriente sincronizadas, teniendo en cuenta la topología de la red.
Patent ES-2625739-B2 (ES)
Title: Procedimiento para la desoxigenación de N-óxidos de piridina, quinolina e isoquinolina.
Inventor: SANZ DÍEZ ROBERTO
IPC: C07D215/60
Filed: 2016-01-20
Granted: 2018-02-15
Abstract: La presente invención se refiere a un procedimiento para la desoxigenación catalítica de N-óxidos de piridina, quinolina e isoquinolina a los correspondientes compuestos heterocícicos derivados de piridina, quinolina e isoquinolina, mediante la utilización de pinacol (2,3-dimetil-2,3-butanodiol) como agente reductor en presencia de un catalizador de molibdeno (VI), en un disolvente orgánico, a presión atmosférica y a una temperatura de 130ºC o, alternativamente, por irradiación en un horno microondas monomodo a una potencia máxima de 150 W y a una temperatura de 130°C, generando como principales subproductos agua y acetona.
Patent AU-2000258008-B2 (AU)
Title: Method for the assembly of a mobile radio network base station and connection of the base station to the network
Inventor: RITTER RUDOLF
IPC: H04B3/54
Filed: 2000-07-26
Granted: 2005-09-01
Abstract: The invention relates to a method for the assembly of a mobile radio network base station comprising a mobile service switching centre (MSC) and one or more base station controllers (BSC) each with one or more base stations (BTS). The invention in particular comprises a method for the assembly of a base station of a public mobile radio network (PLMN), the connection of the base station with the public mobile radio network and the arrangement of a corresponding mobile radio network. The base stations are installed in existing constructions on public, open ground, said constructions having a mains electrical supply. The signal transmission of the radio frequency transmission occurs bi-directionally between base station and the base station controller by means of the mains electrical supply.
Patent AU-2001265669-B2 (AU)
Title: Device for directly reducing ore fine and installation for carrying out said method
Inventor: ROSSMANN GOTTFRIED
IPC: C22B1/10
Filed: 2001-06-27
Granted: 2004-12-16
Abstract: The invention relates to a method for directly reducing, by way of a fluidized bed method, ore fine that comprises at least one ore component from the group of the magnetite, hydrated, carbonate or sulfide ores. The ore fine is heated in a heating fluidized bed zone which is operated with a heating medium, and said heating medium is combusted. The ore is then transferred to at least one reducing fluidized bed zone in which the synthesis gas is fed as the reducing gas to the ore fine in a counter-current and is removed as a top gas, the ore fine being reduced in said zone to sponge iron. In the heating fluidized bed zone the ore fine is specifically heated up by combustion of the heating medium while oxygen or an oxygen-containing gas is additionally fed to adjust oxidizing conditions, and the hydrate, carbonate and/or sulfide groups are removed and/or converted to hematite. At least a part of the top gas is used as a recycled reducing gas for the direct reduction in the reducing fluidized bed zone.
Patent AU-2001274771-B2 (AU)
Title: Human site-1 protease promoter
Inventor: FORSGREN MARGARETA
IPC: C12N9/64
Filed: 2001-06-19
Granted: 2007-01-04
Abstract: The present invention relates to an isolated human Site-1 Protease promoter region. The invention also relates to screening methods for agents decreasing the expression of Site-1 protease and thereby being potentially useful for the treatment of medical conditions related to obesity and/or diabetes.
Patent AU-2002233537-B2 (AU)
Title: Mechanical handling device for golf balls at a driving range
Inventor: GAGER PHILIP
IPC: A63B47/00
Filed: 2002-02-22
Granted: 2007-01-11
Abstract: A mechanical handling device for golf balls at a driving range, comprising a pivotally mounted balance or lever arm provided at one end with a tee adapted, in use, to receive and support a golf ball from a supply source, and provided at its other end with a weight sensitive transducer whereby, from a neutral start position, the arm/tee is initially pivoted downwardly under the influence of the weight of a ball arriving at the tee, such initial movement being sensed by the transducer to activate control means causing the arm/tee to be pivoted to an elevated, striking position, and loss of ball weight at the tee, after striking of the ball, also being sensed by the transducer to activate control means to cause the arm/tee to be pivotally returned to its neutral position. The invention also includes a driving range tee provided with a device.
Patent AU-2002253698-B2 (AU)
Title: Clathrate of azithromycin hydrate with 1,2-propyleneglycol, method for the manufacture thereof and pharmaceutical composition comprising same
Inventor: KIM GI JEONG
IPC: A61K31/7052
Filed: 2002-04-25
Granted: 2005-12-08
Abstract: The present invention relates to a clathrate of azithromycin hydrate with 1,2-propyleneglycol of formula (I), a method for the manufacture thereof, and a pharmaceutical composition containing same. The inventive compound is much less hygroscopic than azithromycin hydrate or crystals known in the art, therefore, it can be useful for the preparation of a medicine for treating various microbial infections. wherein m ranges from 1 to 2 and n, from 0.30 to 0.45.
Patent AU-2002257666-B2 (AU)
Title: Method, computer program product and computer system for modifying roles that trigger application services
Inventor: BITTNER PETER
IPC: G06F15/00
Filed: 2002-03-15
Granted: 2005-07-07
Abstract: The present invention discloses a method, computer program product and system for adjusting roles in a computer system (100) that launch application services (301-307) by a first user who is assigned to at least one role. A first role (110) calls a second role (150) by reference (111). Both roles comprise representations of applications services (101, 102, 103) and (104, 105). When representations in the second role are modified, for example, application services are added (106, 107), a delta list (112) for the first reference is automatically created to conditionally prevent the first role (110) from referencing to at least some of the modified representations of the second role (150). This is achieved by using a rule database (118) containing rules about application services that are mutually exclusive and checking for conflicts between the representations of the first role and modified, second role. A second user, e.g. a system administrator, can accept or reject automatically created delta entries (114) in the delta list (112). <IMAGE>
Patent AU-2002342210-B2 (AU)
Title: Dual input AC/DC/battery operated power supply
Inventor: PIATETSKY ALEXEI A
IPC: H02M3/155
Filed: 2002-10-30
Granted: 2005-06-02
Abstract: A dual input battery assisted power converter (10) which provides a continuous, regulated DC voltage output to a user-connected mobile device, such as, a laptop computer or a cell phone, for example. The power converter (10) comprises a power supply circuit (12) and a separate, detachable power storage circuit comprising a battery pack (14) having a re-chargeable battery (36). The power supply (12) is adapted to deliver a pair of regulated DC output voltages, of opposite voltage potentials, to a pair of respective output terminals. Preferably these output voltages are derived from two external input voltages: an AC input voltage and a DC input voltage. Advantageously, if both of the external input voltages are temporarily removed, the battery pack (14) will advantageously serve as a substitute DC input power source, thereby allowing the power supply (12) to deliver the same regulated DC output voltage to the user-connected mobile device without interruption. Moreover, once either of the external input voltages are again re-established, the battery pack (14) automatically taps the output terminal of the power supply (12) at a node to recharge the battery pack (14).
Patent AU-2002354766-B2 (AU)
Title: Multi-phase headset for pilots
Inventor: MCDONALD THOMAS K
IPC: A62B7/14
Filed: 2002-05-31
Granted: 2007-08-09
Abstract: A multi-phase headset ( 50 ) for aircraft crew members is provided which includes an inflatable gas mask unit ( 54 ) and a visor unit ( 56 ), supported on the head of a user ( 60 ) by mounting assembly ( 52 ). The overall headset ( 50 ) also has a selectively and/or automatically operable motive and control assembly ( 60 ). Preferably; the mounting assembly ( 52 ) includes a pair of ear pieces ( 62, 64 ) and a strap assembly ( 66 ) to allow positioning of the headset ( 50 ) on the user's head, with the mask and visor units ( 54, 56 ) adjacent the crown of the user's head. In the event of an emergency, the mask unit ( 54 ) is lowered and the mask body ( 124 ) is inflated for delivery of breathable gas to the user ( 60 ). Also, the visor unit ( 56 ) may be lowered to a use position atop mask unit ( 54 ). The pneumatically or electrically operated motive and control assembly ( 60 ) serves to move the mask and visor units ( 54, 56 ) between their retracted and deployed position. In order to prevent ingress of smoke, physical seals or air curtain passageways ( 144, 286 ) may be provided along the upper and lower margins of the visor and mask units ( 56, 54 ).
Patent AU-2002356077-B2 (AU)
Title: Residue Guard for nozzle groups of an ink jet printhead
Inventor: SILVERBROOK KIA
IPC: B41J2/045
Filed: 2002-08-21
Granted: 2005-11-10
Abstract: A nozzle guard 80 for an ink jet printer printhead with an array 14 of nozzles 10. The nozzle guard 80 has an array of apertures 84 individually corresponding to the nozzle array 14.The ink droplets are ejected through the apertures 84 and onto the media to be printed. A wiper blade 143 sweeps dust and residual ink 144 stuck to the exterior surface 142 of the nozzle guard 80 characterized in that the exterior surface has one or more recesses 146 encompassing a group, or pod, of the apertures 84 to prevent the wiper blade 143 from engaging the exterior surface 142 immediately adjacent any of the apertures 84 in the pod.
Patent AU-2003275046-B2 (AU)
Title: OXIDATION OF NOx'S WITH SODIUM CHLORITE IN COMBINATION WITH A THERMAL NOX REMOVAL PROCESS
Inventor: KNIGHT DAVID G
IPC: B01D53/56
Filed: 2003-05-09
Granted: 2009-02-12
Abstract: A process for reducing NOx concentrations in waste gas streams by contacting the waste gas stream with a reducing agent selected from ammonia and urea and then oxidizing the lower NOx's present in the waste gas streams to higher oxides with chlorine dioxide.
Patent AU-2003287922-B2 (AU)
Title: 1,2,4-triaminobenzene derivatives useful for treating disorders of the central nervous system
Inventor: RITZEN ANDREAS
IPC: C07D333/20
Filed: 2003-12-18
Granted: 2009-12-10
Abstract: The present invention concerns 1,2,4-triaminobenzene derivatives of the general formula I or pharmaceutically acceptable salts thereof and the use thereof.
Patent AU-2003304518-B2 (AU)
Title: Telecommunication loose tube optical cable with reduced diameter
Inventor: GINOCCHIO ALESSANDRO
IPC: G02B6/44
Filed: 2003-09-30
Granted: 2010-09-09
Abstract: An optical fiber cable has a highly reduced diameter. The cable has a central strength member; a number of tubes containing loosely arranged optical fibers, each tube having a thickness, and each optical fiber having a coating; and a protective outer jacket, wherein the filling coefficient of optical fibers in at least one loose tube is >=45°/0. The tubes are made of a material having an elasticity modulus >=700 MPa; and the optical fibers are SM-R fibers having a microbending sensitivity <=4.0 DB.KM<SUP>-1</SUP>/g.mm<SUP>-1 </SUP>at a temperature of about -30° C. to +60° C. at about 1550 nm.
Patent AU-2004220730-B2 (AU)
Title: Washer and washing cycle control method thereof
Inventor: KIM SEONG SIK
IPC: D06F39/00
Filed: 2004-10-14
Granted: 2010-11-11
Abstract: The present invention provides a washer and washing cycle control method thereof, by which a laundry amount of a laundry can be measured prior to a water supply despite a dry state of the laundry and by which the waste of power consumption and unnecessary use of water can be prevented. The present invention includes a drum holding a laundry therein, a motor rotating the drum, and a control unit executing a sub-routine for measuring a laundry amount of the laundry prior to a water supply to the drum. The sub-routine includes the steps of applying a ramp drive voltage to the motor during an acceleration section to measure a motor RPM amount and a drive voltage amount during the acceleration section, stopping supplying the ramp drive voltage to the motor to measure a motor RPM amount of a deceleration section, and measuring a laundry amount of the laundry using the motor RPM amount of acceleration section, the drive voltage amount of the acceleration section, and the motor RPM amount of the deceleration section
Patent AU-2004233869-B2 (AU)
Title: Solid drug formulation and device for storage and controlled delivery thereof
Inventor: PRESCOTT JAMES H
IPC: A61F2/82
Filed: 2004-04-26
Granted: 2010-08-12
Abstract: Devices and methods are provided for the storage and controlled release of a solid form of a drug. The device comprises a body portion; one or more reservoirs located in and defined by the body portion; a solid matrix which comprises a drug and which is contained in each of the one or more reservoirs; and one or more excipient materials dispersed throughout pores or interstices within the solid matrix and substantially filling any space not otherwise occupied by the solid matrix within each of the one or more reservoirs, wherein the excipient material enhances stability of the drug while stored in the one or more reservoirs or enhances release of the drug from each reservoir. In an alternative embodiment, the device provides for the storage and controlled exposure of a chemical sensor material.
Patent AU-2004269838-B2 (AU)
Title: Device for administering an injectable product, comprising an anti-release safety device
Inventor: SCHERER BENJAMIN
IPC: A61M5/24
Filed: 2004-09-08
Granted: 2009-02-19
Abstract: A device for administering an injectable product includes a drive unit for driving a drive member in an administering direction, a release mechanism for releasing the drive unit and a locking mechanism which, when locked, prevents the release mechanism from being operated, wherein the locking mechanism is displaceable generally along the longitudinal axis of the device from a locked to an unlocked position and the release mechanism can be moved generally radially with respect to the longitudinal axis for releasing purposes when the locking mechanism is in the unlocked position.
Patent AU-2004308955-B2 (AU)
Title: Amino substituted diaryl[a,d]cycloheptene analogs as muscarinic agonists and methods of treatment of neuropsychiatric disorders
Inventor: JORGEN OHLSSON
IPC: A61K31/554
Filed: 2004-12-21
Granted: 2011-08-04
Abstract: Disclosed herein are analogs of clozapine and pharmaceutically acceptable salts, esters, amides, or prodrugs thereof; methods of synthesizing the analogs; and methods of using the analogs for treating neuorpsychiatric disorders. In some embodiments, the analogs are amino substituted diaryl[a,d]cycloheptenes.
Patent AU-2005228716-B2 (AU)
Title: Anionic hydrogel matrices with pH dependent modified release as drug carriers
Inventor: GIAMMONA GAETANO
IPC: A61K9/19
Filed: 2005-02-16
Granted: 2010-07-15
Abstract: Compositions with pH-dependent modified release are described, consisting of hydrogel matrices containing one or more active ingredients, in which said matrices are suitable for releasing said active ingredients in a prolonged manner in given sites of the body.
Patent AU-2005239725-B2 (AU)
Title: Underground mine tire
Inventor: JACOB FRANK MAURICE
IPC: B60C9/00
Filed: 2005-12-02
Granted: 2011-08-18
Abstract: UNDERGROUND MINE TIRE An underground mine tire (20) having a nominal bead diameter of 20.0 inches or s less has a carcass (21), a tread (25) and a pair of rubber sidewalls (23), each extending along the outer periphery of the carcass (21) below the tread (25). The tire 20 has a nominal bead width (D) greater than 8.50 inches and an overall diameter of less than 55 inches. The carcass (21) has at least one radial steel cord reinforced ply (24). FIG- 1
Patent AU-2005249137-B2 (AU)
Title: Method and apparatus for providing enhanced messages on common control channel in wireless communication system
Inventor: KIM MYEONG-CHEOL
IPC: H04W84/00
Filed: 2005-05-11
Granted: 2008-03-20
Abstract: A method and apparatus for providing new configurations for transmitting control information between a mobile terminal and a network using a common control channel (CCCH) logical channel/transport channel. The new configurations enable messages to be sent that are larger than currently allowed and the availability of the new configurations is indicated such that mobile terminals that do not support the new configurations are not impacted.
Patent AU-2005280419-B2 (AU)
Title: Composition and method for improved bioavailability and enhanced brain delivery of 5,5-diphenyl barbituric acid
Inventor: MOROS DANIEL
IPC: A61K31/515
Filed: 2005-08-10
Granted: 2010-09-23
Abstract: The present invention relates to a composition and a method of delivering a barbituric acid derivative to the central nervous system of a mammal in need of treatment for neurological conditions. In particular, the present invention relates to a method of administering an oral dosage form of a sodium salt of 5,5-diphenyl barburtic acid to enhance the bioavailability of 5,5-diphenyl barbituric acid and brain delivery of same.
Patent AU-2005318464-B2 (AU)
Title: Prevention of thrombus formation and/or stabilization
Inventor: NIESWANDT BERNHARD
IPC: A61K39/395
Filed: 2005-12-20
Granted: 2012-02-23
Abstract: The present invention relates to the use of at least one antibody and/or one inhibitor for inhibiting factor XII and preventing the formation and/or the stabilization of threedimensional thrombi. It also relates to a pharmaceutical formulation and the use of factor XII as an anti-thrombotic target.
Patent AU-2005329319-B2 (AU)
Title: Sealing arrangement
Inventor: ZELAZO PAAVO
IPC: B60J10/00
Filed: 2005-12-21
Granted: 2009-07-23
Abstract: In order to easily permit functionally correct mounting of a sealing strip ( 3 ) which is intended for use on the frame structure of a vehicle opening, a sealing arrangement is proposed which is composed of an attachment section ( 4 ) and a sealing section ( 5 ), wherein aids are provided which are intended for carrying out uniquely determined positioning on a section ( 2 ) of the aforesaid frame structure. These aids are a groove ( 7 ) which is configured to receive a frame part of the frame structure and which extends along the entire length of the sealing strip ( 3 ) and whose maximum insertion depth signals the precise positioning of the sealing strip on the aforesaid frame part. These aids can also be a bead ( 15 ) which is integrally formed on the attachment section ( 4 ) and which performs the function of a spacing element in relation to a stop surface of the aforesaid frame structure and is connected to the attachment section in a releasable, in particular tear-off connection. Such a sealing arrangement can be mounted easily and quickly, in particular under service conditions.
Patent AU-2006214097-B2 (AU)
Title: Radio link protocols for multi-link communication systems
Inventor: AGASHE PARAG A
IPC: H04J99/00
Filed: 2006-02-16
Granted: 2010-03-04
Abstract: Embodiments disclosed herein relate to a new set of radio link protocols (RLPs) configured to provide for efficient data transmission in a multi-link communication system. In an embodiment, an upper-layer packet is segmented into link-layer packets to be transmitted over a plurality of communication links, each including a first sequence number in accordance with a predetermined order. A second sequence number is further added to each link-layer packet to be transmitted for the first time. The second sequence number is configured to be in a sequence space associated with a particular communication link, and may be used for detection of missing packets.
Patent AU-2006231929-B2 (AU)
Title: Substituted oxazole derivatives and their use as tyrosine kinase inhibitors
Inventor: MOUSSY ALAIN
IPC: C07D417/12
Filed: 2006-04-04
Granted: 2012-09-06
Abstract: The present invention relates to novel compounds selected from substituted oxazole derivatives of formula (I) that selectively modulate, regulate, and/or inhibit signal transduction mediated by certain native and/or mutant tyrosine kinases implicated in a variety of human and animal diseases such as cell proliferative, metabolic, allergic, and degenerative disorders. More particularly, these compounds are potent and selective c-kit, bcr-abl and Fit- 3 inhibitors.