baber/WOPTO huggingface dataset:
Patent CY-1119831-T1 (CY)
Title: Αποτρεπτικα της καταχρησης σκευασματα φαρμακων
Inventor: HIRSH JANE
IPC: A61K9/20
Filed: 2017-12-20
Abstract: Αναπτύχθηκε μια αποτρεπτική της κατάχρησης φαρμακευτική σύνθεση προς μείωση της πιθανότητας ακατάλληλης χορήγησης φαρμάκων, ειδικώς φαρμάκων όπως οπιοειδή. Στην προτιμώμενη ενσωμάτωση, το φάρμακο τροποποιείται για να αυξηθεί η λιποφιλία του διά του σχηματισμού ενός άλατος μεταξύ του φαρμάκου και ενός ή περισσότερων λιπαρών οξέων όπου η συγκέντρωση του ενός ή περισσότερων λιπαρών οξέων είναι μία έως 15 φορές η γραμμομοριακή ποσότητα του ενεργού παράγοντα, κατά προτίμηση δύο έως δέκα φορές η γραμμομοριακή ποσότητα του ενεργού παράγοντα. Σε μια ενσωμάτωση το τροποποιημένο φάρμακο διασπείρεται ομοιογενώς εντός μικροσωματιδίων αποτελούμενων από ένα υλικό που είτε είναι βραδέως διαλυτό είτε μη διαλυτό σε ύδωρ. Σε μερικές ενσωματώσεις τα περιέχοντα φάρμακο μικροσωματίδια ή σωματίδια φαρμάκου επικαλύπτονται με μία ή περισσότερες στιβάδες επικάλυψης, όπου τουλάχιστον μία επικάλυψη είναι αδιάλυτη σε ύδωρ και κατά προτίμηση αδιάλυτη σε οργανικό διαλύτη. Η αποτρεπτική της κατάχρησης σύνθεση παρεμποδίζει την άμεση απελευθέρωση ενός σημαντικού μέρους του φαρμάκου, ακόμη και όταν η φυσική ακεραιότητα του σκευάσματος τίθεται σε κίνδυνο (για παράδειγμα, με τεμαχισμό με μια λεπτίδα ή σύνθλιψη) και το προκύπτον υλικό τοποθετείται σε ύδωρ, εισπνέεται μέσω της μύτης, ή καταπίνεται. Εντούτοις, όταν χορηγείται όπως υποδεικνύεται, το φάρμακο απελευθερώνεται βραδέως από τη σύνθεση καθώς η σύνθεση διασπάται ή διαλύεται βαθμιαία εντός του γαστροεντερικού σωλήνα με έναν συνδυασμό ενζυμικής αποδόμησης, επιφανειοδραστικής δράσης χολικών οξέων, και μηχανικής διάβρωσης.
Patent CY-1121564-T1 (CY)
Title: Σπειρο-ινδολινες για τη θεραπεια και την προφυλαξη απο τη λοιμωξη απο τον αναπνευστικο συγκυτιακο ιο (rsv)
Inventor: COCKERILL STUART
IPC: A61P31/14
Filed: 2019-04-11
Abstract: Βενζιμιδαζόλες του τύπου (I): όπου : το ένα εκ των Χ και Υ είναι άτομο Ν ή υποκατεστημένο άτομο C και το άλλο είναι CH· το L είναι απλός δεσμός, C1-3 αλκυλένιο, C2-3 αλκενυλένιο ή C2-3 αλκυνυλένιο· το R1 είναι C1-6 αλκύλιο, C2-6 αλκενύλιο, C2-6 αλκυνύλιο, κυκλοαλκύλιο 3 έως 10 μελών, ετεροκυκλική ένωση 5 έως 10 μελών ή ετεροαρύλιο 5 έως 12 μελών, καθένα εκ των οποίων είναι μη υποκατεστημένο ή υποκατεστημένο· το Ζ είναι αλογόνο, C1-6 αλοαλκύλιο, άζωτο, -CN, -N(R2)2, -OR2, -SR2, -S(=0)R2 ή -S(=0)2R2· κάθε R2 είναι ανεξαρτήτως υδρογόνο, C1-6 αλκύλιο, C2-6 αλκενύλιο ή C2-6 αλκυνύλιο, όπου οι εν λόγω αλκυλομάδες, αλκενυλομάδες και αλκυνυλομάδες είναι μη υποκατεστημένες ή υποκατεστημένες· και το m είναι 0 ή 1· και τα φαρμακευτικώς αποδεκτά άλατα τους είναι αναστολείς του RSV και μπορούν, επομένως, να χρησιμοποιηθούν για τη θεραπεία ή την πρόληψη της λοίμωξης από RSV.
Patent HR-P20120472-T1 (HR)
Title: Apparatus for fabricating an insulated container
Inventor: GIANFRANCO D AMATO
IPC: B31B50/59
Filed: 2012-06-05
Abstract: The invention relates to a method of fabricating an insulating container (10) for hot drinks or the like. The container includes an inner cup (12) having a generally frusto-conical cup body (22), a generally frusto-conical outer shell (14), a thermo-sealable plastic coating (42) on at least one of the inside of said shell and the outside of said cup body. The cup is seated within said shell so that the coating extends at least along a contact path (3) near the upper edge (9) of the shell along which contact path outer surface of the cup body and inner surface of the shell are in contact and are bonded.
Patent HR-P20120617-T1 (HR)
Title: Method of transmitting and receiving a signal and apparatus for transmitting and receiving a signal
Inventor: HO TAEK HONG
IPC: H04N5/44
Filed: 2012-07-30
Abstract: The present invention relates to method of transmitting and receiving broadcasting signal and a corresponding apparatus. One aspect of the present invention relates to a method of receiving broadcasting signal, wherein a C2 delivery system descriptor including an identifier of a PLP and an identifier of a C2 system in a TS loop of the NIT maps a transport stream to the data PLP in a data slice of the C2 system.
Patent SI-1519709-T1 (SI)
Title: Novel cosmetic applications of polyphenols and derivatives thereof
Inventor: VERCAUTEREN JOSEPH
IPC: A61K8/34
Filed: 2003-07-10
Abstract: The invention concerns cosmetic compositions with skin lightening and/or spot-removing effect. Said compositions contain polyphenols selected from the group consisting of epsilon -viniferin, mixtures of resveratrol and epsilon -viniferin, and mixtures of polyphenolic, in particular stilbene and/or falvonol, oligomers and/or polymers.
Patent SI-1756359-T1 (SI)
Title: High solids fabric crepe process for producing absorbent sheet with in-fabric drying
Inventor: MURRAY FRANK C
IPC: D21F11/00
Filed: 2005-06-17
Abstract: A method of making a fabric-creped absorbent cellulosic sheet is provided which includes dewatering a papermaking furnish and partially drying the web without wet-pressing before applying it to a translating transfer surface moving at a first speed. The process further includes fabric-creping the web from the transfer surface at a consistency of from about 30 to about 60 percent utilizing a creping fabric, the creping step occurring under pressure in a creping nip defined between the transfer surface and the creping fabric wherein the fabric is traveling at a second speed slower than the speed of said transfer surface, the fabric pattern, nip parameters, velocity delta and web consistency being selected such that the web is creped from the surface and redistributed on the creping fabric. After creping, the web is dried, preferably with a plurality of can dryers to a consistency of at least about 90 percent while it is held in the creping fabric.
Patent SI-1579915-T1 (SI)
Title: Mill with replacable beater strip
Inventor: ADAM MARCUS
IPC: B02C13/00
Filed: 2005-03-18
Abstract: The mill with several stages has a cylindrical or truncated cone-form driven rotor (2) with circular discs (4) installed one above the other and circumferentially distributed beating arms (6) with a cylindrical or truncated cone-form stator. The beating arms extend over several and preferably all milling stages. The mill housing on the end face has at least one opening for the equipping of the rotor with exchangeable, plug-in beating arms which can be fitted without additional means of fastening.
Patent SI-1877073-T1 (SI)
Title: Non-cytotoxic protein conjugates
Inventor: FOSTER KEITH
IPC: C07K14/00
Filed: 2005-12-01
Abstract: A single chain, polypeptide fusion protein, comprising: a non-cytotoxic protease, or a fragment thereof, which protease or protease fragment is capable of cleaving a protein of the exocytic fusion apparatus of a nociceptive sensory afferent; a Targeting Moiety that is capable of binding to a Binding Site on the nociceptive sensory afferent, which Binding Site is capable of undergoing endocytosis to be incorporated into an endosome within the nociceptive sensory afferent; a protease cleavage site at which site the fusion protein is cleavable by a protease, wherein the protease cleavage site is located between the non-cytotoxic protease or fragment thereof and the Targeting Moiety; and a translocation domain that is capable of translocating the protease or protease fragment from within an endosome, across the endosomal membrane and into the cytosol of the nociceptive sensory afferent. Nucleic acid sequences encoding the polypeptide fusion proteins, methods of preparing same and uses thereof are also described.
Patent SI-3157967-T1 (SI)
Title: Metallocene catalyzed polyethylene resin
Inventor: VANTOMME AURELIEN
IPC: C08L23/00
Filed: 2015-11-10
Abstract: The present invention relates to a metallocene-catalyzed polyethylene resin comprising at least two metallocene-catalyzed polyethylene fractions A and B, wherein the polyethylene resin comprises: at least 25 % to at most 55 % by weight of polyethylene fraction A based on the total weight of the polyethylene resin, wherein fraction A has a density at least 0.005 g/cm3 higher than the density of the polyethylene resin; and a melt index MI2 of at least 25.0 g/10 min as determined according to ISO 1133, condition D, at 190 °C and under a load of 2.16 kg; and wherein the polyethylene resin has a density of at least 0.938 g/cm3 to at most 0.954 g/cm3 as measured according to ASTM D-1505 at 23 °C; a melt index MI2 of at least 2.5 g/10 min to at most 25.0 g/10 min as determined according to ISO 1133, condition D, at 190 °C and under a load of 2.16 kg and a molecular weight distribution Mw/Mn of at least 2.6 to at most 4.2, with Mw being the weight-average molecular weight and Mn being the number-average molecular weight. The present invention also relates to an article comprising said resin.
Patent DE-3177299-T2 (DE)
Inventor: GABRIEL STEVEN ALLEN
IPC: G06T3/40
Filed: 1981-04-10
Granted: 1993-06-17
Abstract: A predecimation filter which converts input data samples corresponding to picture elements of an image into output data samples arranged in sequence, successive groups ofoutput data samples corresponding to successively smaller fractional sized versions of the image. A filter (708) responds to successive input data samples corresponding to successive picture elements in a given coordinate direction and yields filtered samples which are reduced in number in accordance with the fractional reduction in the image size. The filtered samples are recursively applied to the filter as input samples.
Patent DE-3650221-T2 (DE)
Inventor: SATO MAKOTO
IPC: C07D487/04
Filed: 1986-06-17
Granted: 1995-06-22
Abstract: New derivatives of penem and pharmaceutically acceptable salt thereof are herein disclosed; the compouinds being useful as an antibacterial agent which has a high sensibility to
Patent DE-3685507-T2 (DE)
Inventor: ZOUZOULAS JOHN
IPC: B65H29/18
Filed: 1986-03-07
Granted: 1992-12-24
Abstract: An improved banknote stacker is described which provides a high level of flexibility and a high degree of stacking efficiency with a reduced level of jams and crumpled banknotes. In one embodiment the improved banknote stacker includes upper and lower housings having molded fingers and slots for interconnection with a banknote validator, banknote transport apparatus including a self adjusting belt-pulley arrangement, a prestorage compartment, a banknote pusher having a home sensing arrangement which allows it to be controlled using a simple open-loop control, and a banknote magazine for storing stacked banknotes and providing ready access to the stacked banknotes.
Patent DE-3786351-T2 (DE)
Inventor: KEMENY DAVID MICHAEL
IPC: G01N33/52
Filed: 1987-12-04
Granted: 1993-10-28
Abstract: In a solid phase immunoassay, e.g. RAST or PRIST, the sensitivity can be substantially increased by reducing the volume of liquid in which the indicator (e.g. <125> I anti-IgE) is contained, preferably to the saturation volume of the paper carrier. If the volume of sample is also similarly reduced, the incubation time can be reduced to as little as 5 minutes without loss of sensitivity in comparison with conventional tests. A washing device for the paper carrier is also disclosed, together with immunoassay kits for use in the method of the invention.
Patent DE-3787212-T2 (DE)
Inventor: SHIRASAKI OSAMU OMRON TATEISI
IPC: A61B5/0225
Filed: 1987-06-12
Granted: 1994-04-28
Abstract: An electronic blood pressure meter, equipped with the functions of computing at least a single relative pulse wave amplitude value in relation with a maximum pulse wave amplitude value, computing a blood pressure value from the cuff pressure when an amplitude of the pulse wave signal has coincided with the relative amplitude value during a change in the amplitude value of the pulse wave signal, and using the reference pressure value thus obtained in accordance with a certain arithmetic formula. If desired, a different process may be selected for determining a blood pressure depending on an initial cuff pressure. This electronic blood pressure allows a measurement to be completed in a very short time and minimizes the discomfort of the person whose blood pressure is to measured through reduction of the maximum cuff pressure. Yet the mathematical formula can be reduced to a simple arithmetic algorithm and is therefore easy to implement.
Patent DE-3872193-T2 (DE)
Inventor: GOUBAUD MICHEL
IPC: B21D5/04
Filed: 1988-12-01
Granted: 1992-12-17
Abstract: This relates to a bending machine of the type comprising a fixed support (10) and a blank holder (22) which is rotatably mounted and has a bearing beak-shaped part (23) by which it is capable of applying to the said fixed support (10) a sheet (15) to be formed, while in order to do this being articulated to two links (25) which are themselves articulated to the fixed support (10) by two connecting parts (26). According to the invention, for its articulation to the links (25), the blank holder (22) has two lugs (32) vertically in line with its bearing beak-shaped part (23). Application, especially, to on-site forming operations of zinc- works. <IMAGE>
Patent DE-3878300-T2 (DE)
Inventor: BECK DOMINIQUE
IPC: H01H47/32
Filed: 1988-04-26
Granted: 1993-08-26
Abstract: The circuit is arranged inside the circuit (bb) fed via the network with push-buttons (BP) associated with neon indicator lamps (N), and is connected to the coil (B) of the remote-control apparatus. It comprises a diode bridge (D) associated with a thyristor (Th) and a resistor (R), first means with a resistor R2, a capacitor (C2) in parallel with a Zener diode for disabling the gate transistor (T) after a specified period following the impedance drop caused by operating the push-button, and second means comprising a capacitor (C1) in parallel with the terminals of the bridge (D) for returning the whole to the conductive state. <IMAGE>
Patent DE-3886766-T2 (DE)
Inventor: PUCKETTE THOMAS
IPC: C07F9/50
Filed: 1988-10-31
Granted: 1994-07-28
Abstract: A process is disclosed for preparing bidentate ligands of the formula:   <IMAGE>   wherein: each Ar is independently selected from aromatic ring compounds having 6 up to 14 carbon atoms, e.g., phenyl, naphthyl, phenanthryl and anthracenyl; the x bonds and the y bonds are attached to adjacent carbon atoms on the ring structures; each R, when present as a substituent, is independently selected from alkyl, alkoxy, aryloxy, aryl, aralyky, alkaryl, alkoxyalky, cycloaliphatic, halogen, alkanoyl, alkanoyloxy, alkoxycarbonyl, carboxyl, cyano or formyl radicals; n is a whole number in the range of 0-4 where Ar is phenyl; 0-6 where Ar is naphthyl; and 0-8 where Ar is phenanthryl or anthracenyl; each R1 and R2 is independently selected from alkyl, aryl, aralkyl, alkaryl or cycloaliphatic radicals, or substituted derivatieves thereof; each R3 and R4 is independently selected from hydrogen and the R1 substituents; each of the above alkyl groups or moieties is straight or branched chain of 1-20 carbons; each aryl group contains 6-10 ring carbons; each cycloaliphatic group contains from 4-8 ring carbons; substituted derivatives include others, amines, amides, sulfonic acids, esters, hydroxyl groups and alkoxy groups. The invention process comprises coupling two molecules of a reactant of the formula:   <IMAGE>  wherein X is halogen, by maintaining a redox reaction system comprising said reactant, a polar aprotic solvent, a nickel compound and a reducing agent at a temperature and for a time sufficient to form the desired bidentate ligand.
Patent DE-3889743-T2 (DE)
Inventor: MATTILA TIMO
IPC: B07C5/12
Filed: 1988-02-09
Granted: 1994-10-20
Abstract: The invention concerns a bottle receiving means comprising a transport apparatus for transporting bottles, an identifying means with data processing unit for identifying and accepting bottles having certain given shapes, and a recording means for recording accepted bottles. The identifying means (2) comprises a mainly stationary illuminating means (5) for illuminating the bottle, a detector (6) for examining the bottle, and a conveyor (7) for moving the bottle past the detector. Between the illuminating means and the detector has been interposed a mirror system (44,45,46,47) by the aid of which the optical length of the system can be increased without increasing the structural dimensions of the means.
Patent SI-0779233-T2 (SI)
Title: Traction sheave elevator
Inventor: AULANKO ESKO
IPC: B66B7/00
Filed: 1994-06-27
Abstract: The traction sheave elevator comprises an elevator car (1) moving along elevator guide rails (10), a counterweight (2) moving along counterweight guide rails (11), a set of hoisting ropes (3) on which the elevator car and the counterweight are suspended, and a drive machine unit (6) comprising a traction sheave (7) driven by the drive machine and engaging the hoisting ropes (3). The drive machine unit (6) of the elevator is placed in the top part of the elevator shaft (15) and in the horizontal cross-section of the shaft between the vertical projection of the cabin and the shaft wall, whereby the drive machine unit is fixed to a wall or the ceiling of the elevator shaft.
Patent TR-199900500-T2 (TR)
Inventor: SIFFERT WINFRIED
IPC: C12N15/09
Filed: 1997-08-29
Abstract: Insan G-proteininin Beta-3 alt-birimi olup en fazla alti WD tekrar motifinden  olusur.
Patent TR-199903126-T2 (TR)
Inventor: TZY ANDR S G
IPC: G09F19/14
Filed: 1997-04-23
Abstract: The equipment comprises a broadsheet (1) placed by the side of the road and provided with advertising element(s), especially text(s) and/or picture(s). In front of the broadsheet (1), in the direction of cars nearing the broadsheet (1) on the road, at least one modifying part (2, 9, 9a, 13) freeing and/or covering said advertising elements at least partly, is fixed at a distance creating an impression of movement for persons sitting in the cars.
Patent DE-60005207-T2 (DE)
Inventor: VIRAGH LAJOS
IPC: B61D47/00
Filed: 2000-10-18
Granted: 2004-07-01
Abstract: An apparatus operative to perform at least one of lifting and moving containers. A base structure is provided with wheels, counter-weight and supports on both sides. Transverse beams are arranged on the on the base structure parallel with axles of the wheels. The beams include container moving units. The base structure includes two base cars arranged antimerically to and movable synchronously with each other, both base cars include container moving units having upper and lower container grips. The container moving units include at least one of traveling lower and upper lifting beams bearing at least a part of the container grips.
Patent DE-60008851-T2 (DE)
Inventor: ROCHON SYLVAIN
IPC: H01H13/52
Filed: 2000-12-22
Granted: 2005-02-10
Abstract: The invention provides an electrical switch of the type comprising a support (10, 12) carrying contacts (30, 34), which delimits a housing (22) in the bottom (26) of which are arranged at least two fixed electrical contacts (30, 34) and which receives a tripping member (36) which can deform elastically in a vertical direction (V) substantially perpendicular to the bottom (26) of the housing (22), and of the type comprising an actuating pusher (44) mounted so as to slide (10, 12) in a lateral direction (H), in order to act on the tripping member (36) via mechanical means (48) which convert the actuation force exerted on the pusher (44) into a perpendicular force applied to the tripping member (36), characterized in that it comprises an actuating lever (48) mounted so as to pivot with respect to the support (10, 12) about an axis (X-X) parallel to the bottom (26) of the housing (22) and in that the lever (48) is returned elastically to its rest position. <IMAGE>
Patent DE-60014748-T2 (DE)
Inventor: GORI C O UNIVERSITA DI ROMA TO
IPC: F01P1/06
Filed: 2000-04-19
Granted: 2006-02-16
Abstract: A supercharged internal-combustion engine (1) comprising a turbocharger (3), a supercharging duct (7) connecting an outlet of the turbocharger (3) to an intake manifold of the engine (1), an intercooler (8) in series with the supercharging duct (7) for cooling the supercharging air of the engine, and a forced-ventilation device (14) for cooling the supercharging duct (7); the device (14) comprises at least one ducting (18,19) having an inlet aperture (20) facing a fan (10) and an outlet aperture (21) facing a portion (16,17) of the supercharging duct (7). <IMAGE>
Patent DE-60015437-T2 (DE)
Inventor: POST VAN DER MOLEN MICHIEL
IPC: F16B2/20
Filed: 2000-05-16
Granted: 2005-11-24
Abstract: A clip for fixing a part on a bar (1), said clip comprising a first clip part (2) which is substantially form-retaining and comprises a bracket (4) slidable along the bar, a bracket arm (6) being connected to the bracket (4), the clip comprising a second clip part (3) having a flexible spring arm (7) whose first end (7a) is connected to a free end (6a) of the bracket arm (6) remote from the bracket, the spring arm (7) having such a length that in a clamping position, it is subjected to pressure and whose second end presses against the bar (1), so that the bracket (4) is not slidable along the bar (1), while the spring arm (7) can be bent by means of an operating lever (8), so that the bracket (4) is slidable along the bar (1).  <IMAGE>
Patent DE-60017725-T2 (DE)
Inventor: FONTAINE MARC
IPC: B26F1/24
Filed: 2000-03-20
Granted: 2006-01-12
Abstract: A flexible sheet material of thickness less than half a millimeter for making tensioned structures such as false ceilings, in particular, the material including microprojections formed by displacing the material from which it is made, said material presenting an acoustic absorption coefficient which is higher than that of the same material without said projections.
Patent DE-60022395-T2 (DE)
Inventor: FOX ROD THOMAS
IPC: C11D3/00
Filed: 2000-12-21
Granted: 2006-06-29
Abstract: Cleaning compositions including a photocatalytic material and a sensitiser employ a photocatalytic material and a sensitiser at a locus, for example on a surface. The residue combats soils and/or undesired microorganisms at the locus.
Patent DE-60026318-T2 (DE)
Inventor: NAKATANI MASAO
IPC: A01P13/00
Filed: 2000-08-09
Granted: 2006-08-10
Abstract: The isoxazoline derivative of the present invention is represented by the following general formula ÄIÜ: <CHEM> Äwherein Q is a group represented by -S(O)n-(CR5R6)m- (wherein n is an integer of 0 to 2, m is an integer of 1 to 3, and R5 and R6 are a hydrogen atom, a cyano group, an alkoxycarbonyl group, an alkyl group or the like); R1 and R2 are a hydrogen atom, an optionally substituted alkyl group, an alkoxycarbonyl group, an optionally substituted phenyl group or the like; R3 and R4 are a hydrogen atom, an optionally substituted alkyl group, a cycloalkyl group or the like; Y is a hydrogen atom, an alkoxycarbonyl group, a carboxyl group, an alkenyl group, an optionally substituted alkyl group or an optionally substituted phenyl groupÜ. The herbicide of the present invention contains the above isoxazoline derivative as the active ingredient.
Patent DE-60026469-T2 (DE)
Inventor: BURDGICK STEVEN SEBASTIAN
IPC: F02C7/18
Filed: 2000-12-07
Granted: 2006-11-16
Abstract: A gas turbine nozzle segment (10) has outer and inner bands (12, 14) and vanes (16) therebetween. Each band includes a side wall (40), a cover (20) and an impingement plate (22) between the cover and nozzle wall defining two cavities (24, 26) on opposite sides of the impingement plate. Cooling steam is supplied to one cavity (24) for flow through apertures (30) of the impingement plate to cool the nozzle wall. The side wall of the band and inturned flange define with the nozzle wall an undercut region (44). Slots (60) are formed through the inturned flange along the nozzle side wall. A plate (58) having through-apertures extending between opposite edges thereof is disposed in each slot, the slots and plates being angled such that the cooling medium exiting the apertures in the second cavity lie close to the side wall for focusing and targeting cooling medium onto the side wall. <IMAGE>
Patent DE-60028450-T2 (DE)
Inventor: HALLOCK JOHN SCOTT
IPC: C08K5/098
Filed: 2000-05-03
Granted: 2006-12-28
Abstract: A composition suitable for scavenging oxygen is disclosed which comprises a carrier having a combination of a hydroxosulfitometalate and a transition metal ion source.