baber/WOPTO huggingface dataset:
Patent HU-212263-B (HU)
Title: Process for producing pyridine derivatives and pharmaceutical compositions containing them
Inventor: BREWSTER ANDREW GEORGE
IPC: A61K31/46
Filed: 1989-10-16
Abstract: The invention concerns novel, pharmaceutically useful 1,3-dioxane alkenoic acid derivatives of the formula I containing a pyridyl moiety at position 4 of the dioxane ring and in which the groups at positions 2, 4 and 5 have cis-relative stereochemistry, X is hydrogen, alkoxy or hydroxy, Y is vinylene, n is 1 or 2, A<1> is alkylene, the substituents R<1> and R<2> at position 2 of the dioxane ring have a variety of values defined hereinafter, and R<4> is hydroxy, a physiologically acceptable alcohol residue or alkanesulphonamido, and the pharmaceutically acceptable salts thereof. The invention also includes processes for the manufacture and use of the acid derivatives as well as pharmaceutical compositions for therapeutic use in one or more of a variety of diseases such as ischaemic heart disease, cerebrovascular disease, asthmatic disease and/or inflammatory disease. <CHEM> l
Patent LV-13816-B (LV)
Title: Hybrid composite cable
Inventor: ROCENS KARLIS
IPC: D07B1/00
Filed: 2008-09-16
Abstract: The essence of invention expresses the structure of hybrid composite cable (1), which consists from the high strength composite material load-bearing core component, carbon fiber reinforced plastic for example, and external steel component. One variant of the suggested hybrid composite cable with the variable by the length cross-sectional areas is shown in Fig.1., where 1-1, 2-2, 3-3 and 4-4 cross-sections, which are differed by the area of steel component cross-section; (2) - leveling layer of the glue, which join together all the elements of the cable by it edges; (6), (7) - high strength composite material load-bearing layers of core components, carbon fiber reinforced plastic, for example; (3), (4), (5), (8), (9), (10) - layers of steel strands; (11) - additional fasteners, which provide invariability of cross-sectional shape by the cable's length; (12) - weldings which provide joint work of steel strands. The suggested hybrid composite cable can be used in structures, where load-bearing elements are straight, as the anchors of several structures, for example, concaved down as in saddle-shaped cable roofs and cable bridges, or concaved up as stressing structural elements. The task of suggested hybrid composite cable is taking up of the loads, acting in the cases, when high strength composite material loose it load-bearing capacity and steel strands are able to take up the forces, which just sufficiently decreased due to the yielding deformation of steel strands and corresponding elongation of the cable.
Patent LV-14054-B (LV)
Title: Fin of hydrodynamic vibro- propulsive device
Inventor: CIFANSKIS SEMJONS
IPC: B63H1/00
Filed: 2009-10-15
Abstract: The present invention pertains to the field of water transport actuators, and it can be used for motion excitation of ships, underwater robotic fishes, motorboats, etc. The objective of the invention is to increase tractive characteristics, velocity of motion and efficiency of floating vehicle. The proposed fin of hydrodynamic vibration propulsive device is made in the form of rectangular plate. Ratio of fin's (5) length (a) to its height (b) is taken within the interval from 1.9 till 2.1. Besides, fin (5) is mounted in the plane, which is perpendicular to liquid surface, and fin's greater side is perpendicular to the vector of velocity of floating vehicle.
Patent LV-10440-B (LV)
Title: A novel sulphonyl urea
Inventor: BEAT JAU
IPC: C07D521/00
Filed: 1993-02-19
Abstract: The invention relates to compounds of formula (I) in which E is -CH= or -N=, and with the proviso that a) at least one of the radicals R3, R4, R5, R6 and R7 is C1-C4 alkyl, b) E is -CH= when X is halogen and c) E is -CH= when X or Y are -OCHF2 or -SCHF2, and in which the meanings of the other substituents are given in the description, and to their use for controlling weeds, or for regulating and inhibiting the growth of plants.
Patent LV-11490-B (LV)
Title: Wrapping  process for warmth-keeping of the external wall
Inventor: LAPSA VIDEVUDS
IPC: E04B1/76
Filed: 1996-04-26
Abstract: The area of usage of this method is construction of insulated buildings and reconstruction. In relation to this, the lagging plates are first joined together, for example, glued with finish plates made of a hard substance and then in this joined manner they are attached to the surface of a building. Commeasure of plates can be created with splice of finish materials over edges of the plates attached previously. This method allows the use of soft and relatively cheaper materials for heat insulation of vertical plane of buildings such as glass- or mineral-wool and peat.
Patent MX-172373-B (MX)
Title: Mejoras a acondicionadores de enjuague del cabello con una sensacion de cabello seco superior y un alto lustre de cabello
Inventor: MARSCHNER FRANK W
IPC: A61K8/86
Filed: 1986-12-23
Abstract: La presente invención se refiere a mejoras a composición acondicionaodra de enjuague para el cabello capaz de proporcionar propiedades de sensación de sequedad superior y de alto lustre que comprende por peso, una mezcla ternaria de 0.5 a 15 por ciento del copolímero de polivinil pirrolidona/acetato de vinilo; 0.1 a 10 por ciento de por lo menos una sal de amonio cuaternario catiónico hidrofílico el cual está libre de radicales de alquilo o alquenilo conteniendo por lo menos 8 átomos de carbono en la molecula, la proporción por peso de dicho compuesto cuaternario al copolímero estando en la gama de 1:5 a 20:1; y de 0.1 a 4 por ciento de un polímero de celulosa no iónico soluble en agua en 71 a 99.3 por ciento de un medio acuoso, la composición tiene un pH en la gama de 3 a 6.
Patent NO-152673-B (NO)
Title: Elastisk festeanordning for bleie-bukser, samt kontinuerlig fremgangsmaate ved fremstilling derav
Inventor: LAPLANCHE PIERRE
IPC: C09J7/02
Filed: 1982-02-18
Abstract: Elastisk festeanordning for bleie-bukser, som omfatter en strekkbar sentraldel, og to ikke strekkbare sidedeler. De to sidedelene består av et stykke i form av et bærebånd utstyrt med en perforeringslinje som av-deles i anvendelsesøyeblikket.Feste for deler av klær, underklær, og spesielt for bleie-bukser til babyer.
Patent NO-149904-B (NO)
Inventor: LEGERIUS BENGT EFRAIM
IPC: F16L5/02
Filed: 1982-12-20
Abstract: PCT No. PCT/SE82/00133 Sec. 371 Date Dec. 15, 1982 Sec. 102(e) Date Dec. 15, 1982 PCT Filed Apr. 23, 1982 PCT Pub. No. WO82/03951 PCT Pub. Date Nov. 11, 1982.A method and tool for sealingly inserting an elastic body in a cavity in a wall in which the cavity has a smaller size than the initial size of the body. A first tubular end portion of the tool is inserted into the cavity and an elastic body is accommodated in a second larger tubular end portion of the tool such that the elastic body rests on a tapered portion which joins the tubular end portions. The second tubular end portion is then closed and pressure fluid is supplied into the second tubular end portion to compress the elastic body and cause it to pass from the second tubular portion into the first tubular portion and then to exit from the first tubular portion into the cavity. The elastic body expands as it exits from the first tubular portion to tightly engage the wall around the cavity and to expel the first tubular end portion from the cavity.
Patent NO-172833-B (NO)
Inventor: TOIVIO ILKKA
IPC: A47C27/10
Filed: 1988-06-20
Abstract: The invention relates to an air mattress (1) comprising a number of successive, elongate and bag-like elements, which can be filled with gas such as air or with some other flowing medium. The elements are arranged transversally with respect to the lengthwise axis (D - D) of the mattress and/or the bed, and are connected to each other successively in a band-like fashion. The successive elements (2, 2 min ) are arranged so that the lenghtwise seam joints (6; 6b) of the elementes are located at given intervals in the bottom part (1b) of the mattress, and that the areas between these seam joints are arranged to form structures which are directed upwards from the bottom part (1b) of the mattress. The invention also relates to a method for adjusting an air mattress or the like. The elements (2, 2 min ; 9, 10) of the mattress are partly filled with for instance air, so that the mattress pressure corresponds to the pressure of the surroundings when the mattress elements are not subjected to a weight load, but the mattress pressure grows in a known fashion according to the weight load of the human body or part thereof, so that the mattress elements conform to the contours of the body or part thereof, and simultaneously the surface pressure against the body or part thereof is distributed evenly over the whole body or part thereof.
Patent NO-169958-B (NO)
Inventor: SENTER PETER D
IPC: A61K47/00
Filed: 1988-11-22
Abstract: There is disclosed a drug-monoclonal antibody conjugate wherein the antibody is linked to a antitumor drug using disulfide benzyl carbamate or carbonate as the linker. The conjugate is used for delivering an active antitumor drug to the site of tumor cells in a mammal by administering the drug-monoclonal antibody conjugate.
Patent NO-174392-B (NO)
Inventor: VON BORSTEL REID WARREN
IPC: A61K8/00
Filed: 1989-06-26
Abstract: Use of acyl derivatives of deoxyribonucleosides in manufacture of a medicament for enhancing haematopoesis or enhancing healing of bone marrow. <IMAGE>
Patent NO-178127-B (NO)
Inventor: OKADA SATORU
IPC: G06F9/06
Filed: 1990-01-09
Abstract: A hand-held electronic game machine includes a computer (22) accommodated in a case and a liquid crystal display (LCD) panel (14). When an external memory (16) is inserted to a receiving port (68), a first character data being set in advance in the computer (22) is compared with a second character data stored in a predetermined area of the external memory (16). Prior to such comparison, the computer displays the characters represented by the second character data on the LCD panel. If the first and second character data are coincident with each other, the computer (22) can access to the external memory (16).
Patent YU-47121-B (YU)
Inventor: STERZYCKI Z R
IPC: A61K31/7042
Filed: 1988-11-04
Abstract: There are disclosed novel 2 min ,3 min -dideoxy-2 min -fluoronucleosides and 2 min -3 min -dideoxy-2 min ,3 min -didehydro-2 min -fluoronucleosides and processes for their preparation. The compounds so produced exhibit therapeutically useful antiviral and, more particularly, anti-HIV effects.
Patent RS-51343-B (RS)
Inventor: LILLIOTT NICOLA JANE
IPC: A61K31/4439
Filed: 2000-11-16
Abstract: Farmaceutska kompozicija, naznačena time, što sadrži tiazolidindion, kao stoje 5-[4-[2-(N-metil-N-(2-piridil)amino)etoksi]benzil]tiazolidin -2,4-dion (Jedinjenje (I), njegovu farmaceutski prihvatljivu so, metformin hidrohlorid i farmaceutski prihvatljiv nosač, pri čemu su, u farmaceutskoj kompoziciji, tiazolidindion i metformin hidrohlorid dispergovani svaki u svom farmaceutski prihvatljivom nosaču.Prijava sadrži još 21 zavisni patentni zahtev.
Patent RS-49680-B (RS)
Inventor: MARKHOFF KLAUS
IPC: G05B19/41
Filed: 2000-12-05
Abstract: Uređaj za obradu boce za gas kojim se optimizuje njen oblik i čvrstoća zidova ima motor za upravljano obrtanje boce 1 oko podužne ose i za upravljanje upravljačkom jedinicom 8, naznačen time, što je na vođici (2) i pogonskom vratilu (3) klizno postavljen nosač (4) nadzvučnog senzora (5) za merenje graničnih površina (10, 11) zida (9) i nosač (6) alata (7) za obradu skidanjem strugotine koji je povezan sa upravljačkom jedinicom 88) za numeričko upravljanje. Prijava sadrži još 1 nezavisan i 5 zavisnih patentnih zahteva.
Patent RS-52091-B (RS)
Inventor: NAKATANI MASAO
IPC: A01N43/828
Filed: 2002-02-07
Abstract: Izoksazolinski derivat predstavljen sledećom opštom formulom $I] ili njena farmaceuski prihvatljiva so:gde R1 i R2 mogu biti isti ili različiti i oba predstavljaju atom vodonika, C1 do C10 alkil grupu, C3 do C8 cikloalkil grupu ili C3 do C8 cikloalkil C1 do C3 alkil grupu koja može biti supstituisana sa atomom halogena ili sa C1 do C3 alkil grupom, ili R1 i R2 mogu biti vezani jedan za drugi da bi se formirao C3 do C7 spiro prsten zajedno sa ugljenikovim atomima za koje su vezani;R3 i R4 mogu biti isti ili različiti i oba su atom vodonika, C1 do C10 alkil grupa ili C3 do C8 cicloalkil grupa; ili R3 i R4 mogu biti vezani jedan za drugi dajući C3 do C7 spiro prsten zajedno sa ugljenikovim atomima za koje su vezani; ili R1, R2, R3 i R4 mogu formirati 5- do 8-očlani prsten zajedno sa ugljenikovim atomima za koje su vezani; R5 i R6 mogu biti isti ili različiti i oba predstavljaju vodonikov atom ili C1 do C10 alkil grupu; gde n predstavlja ceo broj od 0 do 2;gde je Y pirazol-4-il grupa i pirazolski prsten je supstituisan u položaju 3 i 5 sa supstituentskom grupom α i u položaju 1 sa atomom vodonika, C1 do C10 alkil grupom, C1do C10 alkil grupom mono-supstituisanom sa grupom odabranom iz grupe supstituenata (β, C1 do C4 haloalkil grupa, C3 do C8 cikloalkil grupa, C2 do C6 alkenil grupa, C2 do C6 alkinil grupe, C1 do C10 alkilsulfinil grupe, C1 do C10 alkilsulfonil grupe, C1 do C10 alkilsulfonil grupe mono-supstituisane sa grupom odabranom od supstituisane grupe γ, C1 do C4 haloalkilsul-fonil grupe, fenil grupa koja može biti supstituisana sa grupama koje su odabrane od supstituenta ε, aromatična heterociklična grupa koja može biti supstituisana sa grupama koje su odabrane od supstituentne grupe ε, fenilsulfonil grupa koja može biti supstituisana sa grupama odabranim od supstituentne grupe ε; aromatična heterociklična sulfonil grupa koja može biti supstituisana sa grupama koje su odabrane od supstituentne grupe ε; C2 do C5 acil grupa, C1 do C4 haloalkilkar-bonil grupa, benzilkarbonil grupa koja može biti supstituisana sa grupom(ama) odabranim od supstituenta ε; benzoil grupa koja može biti supstituisana sa grupom(ama) odabranim od supstituenta ε; C1 do C10 alkoksikarbonil grupa, benziloksikarbonil grupa koja može biti supstituisana sa grupom(ama) odabranim od supstituenta e, fenoksi-karbonil grupa koja može biti supstituisana sa grupom (ama) odabranim od supstituenta ε, karbamoil grupa (čiji atom azota može biti supstituisan sa istim ili različitim grupama odabranim među C1 do C10 alkil grupama i fenil grupe koja može biti supstituisana sa grup(ama) odabranim od supstituenta e), ili amino grupa (čiji atom azota može biti supstituisan sa istim ili različitim grupama odabranim među C1 do C10 alkil gr
Patent RS-51746-B (RS)
Title: Atorvastatin calcium in a pharmaceutical form, composition thereof, and pharmaceutical formulation comprising atorvastatin calcium
Inventor: KERC JANEZ
IPC: A61K9/08
Filed: 2002-03-13
Abstract: Atorvastatin calcium, the substance known by the chemical name (R-(R*,R*))-2-(4-fluorophenyl)-²,´-dihydroxy-5-(1-methylethyl)-3-phenyl-((phenylamino)carbonyl)-1H-pyrrole-1-heptanoic acid hemi calcium salt is known as HMG-CoA reductase inhibitor and is used as an antihypercholesterolemic agent. Atorvastatin in the pharmaceutical compositions available in the market, is usually prepared as its calcium salt since it enables atorvastatin to be conveniently formulated in the pharmaceutical formulations, for example, in tablets, capsules, powders and the like for oral administration. Atorvastatin calcium can exist in an amorphous form or in one of the at least four known crystalline forms (Form I, Form II, Form III and Form IV). Atorvastatin calcium is the substance which is sparingly soluble in water, with pKa 4,5, and it has been found that the crystalline forms are less soluble than the amorphous form, which may cause problems in bioavailability of atorvastatin in the body.  The present invention solves the problem of providing therapeutic equivalence of atorvastatin pharmaceutical formulation regardless the form (crystalline, amorphous, mixture of both) of atorvastatin calcium used for its preparation.
Patent ZA-793861-B (ZA)
Title: N-substituted nitrogen-containing heterocyclic compounds
Inventor: FUEGNER A
IPC: C07D239/88
Filed: 1979-07-27
Abstract: Compounds of the formula   <IMAGE>   wherein Het is   <IMAGE>  +TR <IMAGE>  n is an integer from 1 to 4, inclusive, preferably 2 or 3, R1 is H or acyl, R2 is H, R1O, -NHSO2R7, -NHCOR8, -NHCONHR8, -NH-CH2-C6H4-R9, -CH2OH, -CH2SO2R7, -CONHR8, halogen or -CN, R3 is H, halogen, R7 or -OR7, R2 and R3 together with each other are <IMAGE>  R4 is H, -CH3 or -C2H5, R5 and R6 are each H or -CH3, R7 is C1-C4 alkyl, R8 is H or C1-C4 alkyl, R9 is H, C1-C4 alkyl or C1-C4 alkoxy optionally interrupted by oxygen, R10 and R12 are each H, CH3, Cl or OCH3, or together methylenedioxy, X is   <IMAGE>   or N, and Z is -CH2 or -CO; in the form of racemates, enantiomers, diastereoisomeric antipode pairs, and non-toxic, pharmacologically acceptable acid addition salts thereof. The compounds as well as the salts are useful as bronchospasmolytics, spasmolytics, muscle-relaxants, antiallergics and hypotensives.
Patent ZA-817696-B (ZA)
Title: N-substituted omega-(2-oxo-4-imidazolin-1-yl)alcanoic acids,salts and esters thereof,process for producing the same and these active agents containing pharmaceutical compounds
Inventor: LAUTENSCHLAEGER HANS HEINER
IPC: A61P7/02
Filed: 1981-11-06
Abstract: The present invention refers to N-substituted  omega -(2-oxo-4-imidazolin-1-yl) alcanoic acids as well as salts and esters thereof having the general formula I   <IMAGE> I
Patent ZA-825969-B (ZA)
Title: Aseptic filling station
Inventor: ANDERSON IAN MCARTHUR
IPC: B67C7/00
Filed: 1982-08-17
Abstract: A method and system for aseptic filling of containers. The flexible containers (1) are presterilized and a rupturable membrane (41) covers the inlet to the container. The filling head (20) includes a recess (46) below the outlet valve (24) and this recess is closed by the rupturable membrane (41) when the container inlet is aligned with the filling head. After alignment sterilizing fluid is introduced into the recess to sterilize the outer surface of the membrane and the internal surfaces of the recess. Following sterilization the valve membrane (22) moves towards the rupturable membrane (41) allowing the piercing tool (25) to rupture said membrane. The outlet valve (24) of the filling head is opened and the liquid is allowed to flow into the container. Subsequent to completion of the filling cycle the inlet to the container is sealed and the sealed and filled container (1) is then removed from the filling head (20).
Patent ZA-837922-B (ZA)
Title: 3-amino-1-phenoxy-2-propanol derivatives
Inventor: LAFON LOUIS
IPC: A61K31/138
Filed: 1983-10-25
Abstract: 1. Claims for the contracting states : BE, CH, DE, FR, GB, IT, LI, LU, NL, SE : 3-amino-1-phenoxy-2-propanol derivative, characterized in that it is selected from the group constituted by (i) the 3-alkylamino-1-(2-chloro-3,5-dimethoxyphenoxy)-2- propanols responding to the general formula  see diagramm : EP0110746,P12,F1 in which R is CH(CH3 )2 or C(CH3 )3 ; and (ii) their addition salts. 1. Claims for the contracting state : AT Use of a 3-amino-1-phenoxy-2-propanol derivative, selected from the group constituted by (i) the 3-alkylamino-1-(2-chloro-3,5-dimethoxyphenoxy)- 2-propanols responding to the general formula :  see diagramm : EP0110746,P13,F1 in which R is CH(CH3 )2 or C(CH3 )3 ; and (ii) their non toxic addition salts for manufacturing a drug.
Patent ZA-842536-B (ZA)
Title: Compact apparatus for plugging the tapholes of shaft furnaces
Inventor: COOPER ARTHUR WILLIAM
IPC: C21B7/12
Filed: 1984-04-04
Abstract: A shaft furnace plugging apparatus is presented which occupies very little space and sweeps out a relatively low and comparatively flat continuous trajectory between an inoperative position and an operative position. The plugging apparatus includes a clay gun pivotably mounted on a first end of a jib, the jib being rotatable about a support column. The apparatus also includes a pair of hydraulic cylinders, the first hydraulic cylinder being pivotably attached between a second end of the jib and an intermediate pivotable frame and the second hydraulic cylinder which is operative between the intermediate pivotable frame and a fixed support frame.
Patent ZA-849117-B (ZA)
Title: Detergent composition
Inventor: CLEMENTS ANTHONY HENRY
IPC: C11D3/39
Filed: 1984-11-22
Abstract: Improved fabric washing detergent composition especially but not exclusively designed for washing mixed coloured fabrics comprising from 0.5 to 25 % by weight of a peracid compound selected from the group consisting of organic peracids, peracid salts and peracid precursors which generate peracids by hydrolysis or perhydrolysis, and from 0.002 to 2.5 % by weight of copper, in the absence or substantial absence of a powerful sequestrant which complexes strongly with copper. The composition is effective in minimizing dye transfer but is non-effective or substantially non-effective with respect to direct fabric dye or stain bleaching.
Patent ZA-853559-B (ZA)
Title: A thermosetting,free radical curable unsaturated polymer resin composition and a method of reducing gas generation in curing thermosetting,free radical curable unsaturated polymer resin compositions
Inventor: MESSICK VIRGINIA B
IPC: C08F290/00
Filed: 1985-05-10
Abstract: A thermosetting, free radical curable unsaturated polymer resin composition and a method of curing thermosetting, free radical curable, unsaturated polymer resin compositions having a pH greater than 4.5 measured as a 10 weight percent methanol solution and containing a tertiary amine as an esterification catalyst and/or an accelerator, such resin being admixed with a copolymerizable monomer, wherein a curing system of a ketone peroxide and a redox active metal salt is employed. An effective amount of an organic sulfonic acid is added to the resin prior to curing, whereby by gas generation upon curing is reduced.
Patent ZA-862259-B (ZA)
Title: 5-(6-imidazo(1,2-a)pyridyl)pyridine derivative
Inventor: YAMANAKA MOTOSUKE
IPC: C07D471/04
Filed: 1986-03-26
Abstract: 5-(6-Imidazo[1,2-a]pyridyl)pyridine derivatives represented by general formula: wherein X represents hydrogen atom or methyl group; Y represents cyano group, carboxamido group, hydrogen atom, amino group or a halogen atom; Z represents hydrogen atom or a lower alkyl group; W represents hydrogen atom or a lower alkyl group; R' represents hydrogen atom, a lower alkyl group, phenyl group, a group shown by formula: -CH<sub>2</sub>R<sup>4</sup> in which R<sup>4</sup> is a lower alkoxy group, or a group shown by formula:in which R<sup>5</sup> and R<sup>6</sup> are hydrogen atom or a lower alkyl group; R<sup>2</sup> represents hydrogen atom or a halogen atom; and R<sup>3</sup> represents hydrogen atom, a lower alkyl group or a halogen atom; or a tautomer thereof; and pharmacologically acceptable salts thereof are disclosed. The 5-(6-imidazo[1,2-a]-pyridyl) pyridine derivatives are effective for treating congestive heart failures.
Patent ZA-875356-B (ZA)
Title: Sorting and orienting apparatus
IPC: B65G47/24
Filed: 1987-07-21
Abstract: Apparatus for selecting elongate containers from a mass of randomly-disposed containers such as capsules open at one end and at least partially closed at the other and depositing them with their open ends aligned for receiving a charge of material. The apparatus including first and second rotors, the first rotor including radially-disposed bores for receiving the containers and the second rotor including radially-disposed spokes for receiving containers with open ends toward the spokes. The first and second rotors including operable elements for removing the containers from the bores or spokes for transfer of the containers to a receiving device with the containers in the same orientation.