drug_name stringlengths 5 40 | target_gene stringlengths 2 363 | evidence_score float64 1 13 | source stringclasses 10
values | is_moa bool 2
classes |
|---|---|---|---|---|
(s)-nicardipine | CACNA1D|CACNA1C | 1 | drugcentral:DRUG LABEL | true |
(s)-nitrendipine | CACNA1C | 1 | drugcentral:SCIENTIFIC LITERATURE | true |
(s)-nitrendipine | CACNA1D | 8.4 | drugcentral:IUPHAR | true |
(s)-nitrendipine | CACNA1F | 6 | drugcentral:IUPHAR | false |
(s)-nitrendipine | KCNN4 | 7.6 | drugcentral:IUPHAR | false |
abaloparatide | PTH1R | 9.7 | drugcentral:SCIENTIFIC LITERATURE | true |
abametapir | CCR1 | 4.8 | drugcentral:CHEMBL | false |
abametapir | CCR5 | 5.64 | drugcentral:CHEMBL | false |
abametapir | CCR8 | 5.12 | drugcentral:CHEMBL | false |
abarelix | GNRHR | 9.49 | drugcentral:IUPHAR | true |
abatacept | CD80 | 7.92 | drugcentral:IUPHAR | true |
abatacept | CD86 | 7.92 | drugcentral:IUPHAR | true |
abciximab | ITGB3|ITGA2B | 1 | drugcentral:DRUG LABEL | true |
abemaciclib | CDK1 | 5.82 | drugcentral:CHEMBL | false |
abemaciclib | CDK4 | 9.222 | drugcentral:SCIENTIFIC LITERATURE | true |
abemaciclib | CDK6 | 8.62 | drugcentral:SCIENTIFIC LITERATURE | true |
abemaciclib | CDK7 | 6.52 | drugcentral:CHEMBL | false |
abemaciclib | CDK9 | 7.24 | drugcentral:CHEMBL | false |
abemaciclib | KCNH2 | 4.96 | drugcentral:CHEMBL | false |
abiraterone acetate | AR | 4.77 | drugcentral:CHEMBL | false |
abiraterone acetate | CYP11B1 | 5.79 | drugcentral:CHEMBL | false |
abiraterone acetate | CYP11B2 | 5.76 | drugcentral:CHEMBL | false |
abiraterone acetate | CYP17A1 | 8.54 | drugcentral:CHEMBL | true |
abiraterone acetate | CYP3A4 | 5.57 | drugcentral:CHEMBL | false |
acalabrutinib | BMX | 7.337 | drugcentral:SCIENTIFIC LITERATURE | false |
acalabrutinib | BTK | 8.292 | drugcentral:SCIENTIFIC LITERATURE | true |
acalabrutinib | ERBB2 | 8.13 | drugcentral:CHEMBL | false |
acalabrutinib | ERBB4 | 7.796 | drugcentral:SCIENTIFIC LITERATURE | false |
acalabrutinib | LYN | 6 | drugcentral:IUPHAR | false |
acalabrutinib | TEC | 7.032 | drugcentral:SCIENTIFIC LITERATURE | false |
acalabrutinib | TXK | 6.434 | drugcentral:SCIENTIFIC LITERATURE | false |
acamprosate | GABRA1|GABRG2|GABRB3 | 1 | drugcentral:WOMBAT-PK | true |
acamprosate | GRIN2D|GRIN3B|GRIN1|GRIN2A|GRIN2B|GRIN2C|GRIN3A | 1 | drugcentral:CHEMBL | true |
acarbose | AMY1A | 6 | drugcentral:CHEMBL | false |
acarbose | AMY2A | 1 | drugcentral:CHEMBL | true |
acarbose | GAA | 5.3 | drugcentral:CHEMBL | false |
acarbose | MGAM | 5.697 | drugcentral:WOMBAT-PK | true |
acarbose | SI | 6.609 | drugcentral:SCIENTIFIC LITERATURE | false |
acebutolol | ADRB1 | 7.3 | drugcentral:WOMBAT-PK | true |
acebutolol | ADRB2 | 6.4 | drugcentral:WOMBAT-PK | false |
aceclidine | CHRM1 | 5 | drugcentral:IUPHAR | false |
aceclidine | CHRM2 | 5.7 | drugcentral:IUPHAR | false |
aceclidine | CHRM3 | 5.1 | drugcentral:IUPHAR | false |
aceclidine | CHRM4 | 4.8 | drugcentral:IUPHAR | false |
aceclidine | CHRM5 | 5.1 | drugcentral:IUPHAR | false |
aceclofenac | MAPK1 | 5.227 | drugcentral:DRUG MATRIX | false |
aceclofenac | PTGS2 | 1 | drugcentral:DRUG LABEL | true |
aceclofenac | TTR | 5.92 | drugcentral:CHEMBL | false |
acefylline | ADORA2B | 4.56 | drugcentral:CHEMBL | false |
acemetacin | GLO1 | 4.89 | drugcentral:CHEMBL | false |
acemetacin | PTGS1 | 1 | drugcentral:KEGG DRUG | true |
acemetacin | PTGS2 | 1 | drugcentral:KEGG DRUG | true |
acenocoumarol | VKORC1 | 6.114 | drugcentral:SCIENTIFIC LITERATURE | true |
acepromazine | DRD1 | 1 | drugcentral:DRUGBANK | true |
acepromazine | DRD2 | 1 | drugcentral:DRUGBANK | true |
acepromazine | PRNP | 5.3 | drugcentral:CHEMBL | false |
aceprometazine | HRH1 | 1 | drugcentral:DRUG LABEL | true |
acetanilide | NAPRT | 9 | drugcentral:CHEMBL | false |
acetazolamide | AQP1 | 1 | drugcentral:WOMBAT-PK | false |
acetazolamide | CA1 | 7.92 | drugcentral:CHEMBL | true |
acetazolamide | CA11 | 8.24 | drugcentral:CHEMBL | false |
acetazolamide | CA12 | 8.6 | drugcentral:CHEMBL | true |
acetazolamide | CA12|CA1|CA2|CA3|CA4|CA6|CA5A|CA7|CA9|CA13|CA14|CA5B | 9.1 | drugcentral:CHEMBL | false |
acetazolamide | CA13 | 8.24 | drugcentral:CHEMBL | false |
acetazolamide | CA14 | 7.39 | drugcentral:CHEMBL | false |
acetazolamide | CA2 | 8.48 | drugcentral:CHEMBL | true |
acetazolamide | CA3 | 8.51 | drugcentral:CHEMBL | false |
acetazolamide | CA4 | 7.96 | drugcentral:CHEMBL | true |
acetazolamide | CA5A | 7.22 | drugcentral:CHEMBL | false |
acetazolamide | CA5A|CA5B | 8.74 | drugcentral:CHEMBL | false |
acetazolamide | CA5B | 7.27 | drugcentral:CHEMBL | false |
acetazolamide | CA6 | 7.96 | drugcentral:CHEMBL | false |
acetazolamide | CA7 | 8.6 | drugcentral:CHEMBL | false |
acetazolamide | CA9 | 8.05 | drugcentral:CHEMBL | false |
acetic acid | FFAR2 | 4.6 | drugcentral:IUPHAR | false |
acetic acid | FFAR3 | 4.92 | drugcentral:CHEMBL | false |
acetic acid | FYN | 6.05 | drugcentral:CHEMBL | false |
acetic acid | LCK | 6.19 | drugcentral:CHEMBL | false |
acetohexamide | ABCC8|KCNJ11 | 4.639 | drugcentral:SCIENTIFIC LITERATURE | true |
acetohydroxamic acid | CA2 | 4.33 | drugcentral:CHEMBL | false |
acetophenazine | DRD2 | 1 | drugcentral:DRUGBANK | true |
acetoxolone | CES1 | 4.3 | drugcentral:CHEMBL | false |
acetoxolone | CES2 | 4.39 | drugcentral:CHEMBL | false |
acetoxolone | HSD11B1 | 6.1 | drugcentral:CHEMBL | false |
acetoxolone | HSD11B2 | 6.7 | drugcentral:CHEMBL | false |
acetoxolone | HSD17B1 | 4.73 | drugcentral:CHEMBL | false |
acetoxolone | HSD17B2 | 5.42 | drugcentral:CHEMBL | false |
acetylcholine | CHRM1 | 6.11 | drugcentral:CHEMBL | false |
acetylcholine | CHRM2 | 6.5 | drugcentral:IUPHAR | false |
acetylcholine | CHRM3 | 6.66 | drugcentral:CHEMBL | true |
acetylcholine | CHRM4 | 5.6 | drugcentral:IUPHAR | false |
acetylcholine | CHRM5 | 6.1 | drugcentral:CHEMBL | false |
acetylcholine | CHRNA7 | 5.1 | drugcentral:CHEMBL | false |
acetylcholine | CHRNB2|CHRNA4 | 5.8 | drugcentral:CHEMBL | false |
acetylcysteine | CYCS | 1 | drugcentral:WOMBAT-PK | false |
acetylcysteine | GSS | 1 | drugcentral:DRUGBANK | false |
acetylcysteine | SLC7A11 | 1 | drugcentral:SCIENTIFIC LITERATURE | false |
acetylcysteine | SOD2 | 1 | drugcentral:WOMBAT-PK | false |
acetylcysteine | VEGFA | 1 | drugcentral:WOMBAT-PK | false |
acetyldigitoxin | ATP1A1|ATP1B1|ATP1A3|ATP1B2|ATP1A2|ATP1B3|FXYD2|ATP1A4 | 1 | drugcentral:CHEMBL | true |
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