Compound ID,Target,Assay (Percent degradation),DOI,DC50,Dmax,Assay (DC50/Dmax),PROTAC to Target
1,BRD7,20/12 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in HeLa cells after 4/16 h treatment at 1 μM
1,BRD9,19/30 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in HeLa cells after 4/16 h treatment at 1 μM
2,BRD7,19/27 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in HeLa cells after 4/16 h treatment at 1 μM
2,BRD9,5/21 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in HeLa cells after 4/16 h treatment at 1 μM
3,BRD9,94/93 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in HeLa cells after 4/16 h treatment at 1 μM
4,BRD9,81/89 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in HeLa cells after 4/16 h treatment at 1 μM
5,BRD9,0/19 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in HeLa cells after 4/16 h treatment at 1 μM
5,BRD7,0/14 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in HeLa cells after 4/16 h treatment at 1 μM
6,BRD9,0/14 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in HeLa cells after 4/16 h treatment at 1 μM
6,BRD7,19/14 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in HeLa cells after 4/16 h treatment at 1 μM
7,BRD7,0 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in HeLa cells after 4 h treatment at 1 μM
7,BRD9,23 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in HeLa cells after 4 h treatment at 1 μM
8,BRD7,0 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in HeLa cells after 4 h treatment at 1 μM
8,BRD9,57 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in HeLa cells after 4 h treatment at 1 μM
9,BRD7,0 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in HeLa cells after 4 h treatment at 1 μM
9,BRD9,7 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in HeLa cells after 4 h treatment at 1 μM
10,BRD9,26 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in HeLa cells after 4 h treatment at 1 μM
10,BRD7,5 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in HeLa cells after 4 h treatment at 1 μM
11,BRD7,3 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in HeLa cells after 4 h treatment at 1 μM
11,BRD9,,10.1021/acs.jmedchem.8b01413,560,80,Degradation of BRD9 in HeLa cells after 4 h treatment,
12,BRD7,12 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in HeLa cells after 4 h treatment at 1 μM
12,BRD9,50 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in HeLa cells after 4 h treatment at 1 μM
13,BRD7,11 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in HeLa cells after 4 h treatment at 1 μM
13,BRD9,9 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in HeLa cells after 4 h treatment at 1 μM
14,BRD7,0 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in HeLa cells after 4 h treatment at 1 μM
14,BRD9,32 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in HeLa cells after 4 h treatment at 1 μM
15,BRD9,1 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in HeLa cells after 4 h treatment at 1 μM
15,BRD7,5 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in HeLa cells after 4 h treatment at 1 μM
16,BRD9,8 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in HeLa cells after 4 h treatment at 1 μM
16,BRD7,0 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in HeLa cells after 4 h treatment at 1 μM
17,BRD7,37 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in RI-1 cells after 2 h treatment at 1 μM
17,BRD9,37 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in RI-1 cells after 2 h treatment at 1 μM
18,BRD9,6 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in RI-1 cells after 2 h treatment at 1 μM
18,BRD7,2 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in RI-1 cells after 2 h treatment at 1 μM
19,BRD7,0 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in RI-1 cells after 2 h treatment at 1 μM
19,BRD9,0 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in RI-1 cells after 2 h treatment at 1 μM
20,BRD7,0 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in RI-1 cells after 2 h treatment at 1 μM
20,BRD9,0 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in RI-1 cells after 2 h treatment at 1 μM
21,BRD7,0 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in RI-1 cells after 2 h treatment at 1 μM
21,BRD9,0 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in RI-1 cells after 2 h treatment at 1 μM
22,BRD9,,10.1021/acs.jmedchem.8b01413,1.76,95,Degradation of BRD9 in RI-1 cells after 8 h treatment,
22,BRD7,,10.1021/acs.jmedchem.8b01413,34.5,,Degradation of HiBiT-BRD7 in HEK293 cells after 24 h treatment using CRISPR/Cas9,
22,BRD7,,10.1021/acs.jmedchem.8b01413,4.5,95,Degradation of BRD7 in RI-1 cells after 8 h treatment,
22,BRD9,,10.1021/acs.jmedchem.8b01413,2/8,,Degradation of BRD9 in EOL-1/A-204 cells after 18 h treatment on a WES capillary electrophoresis instrument,
22,BRD9,,10.1021/acs.jmedchem.8b01413,4,,Degradation of HiBiT-BRD9 in HEK293 cells after 24 h treatment using CRISPR/Cas9,
23,BRD9,35 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in RI-1 cells after 2 h treatment at 1 μM
23,BRD7,35 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in RI-1 cells after 2 h treatment at 1 μM
24,BRD9,31 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in RI-1 cells after 2 h treatment at 1 μM
24,BRD7,17 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in RI-1 cells after 2 h treatment at 1 μM
25,BRD7,0 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in RI-1 cells after 2 h treatment at 1 μM
25,BRD9,11 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in RI-1 cells after 2 h treatment at 1 μM
26,BRD9,0 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in RI-1 cells after 2 h treatment at 1 μM
26,BRD7,0 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in RI-1 cells after 2 h treatment at 1 μM
27,BRD7,0 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in RI-1 cells after 2 h treatment at 1 μM
27,BRD9,1 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in RI-1 cells after 2 h treatment at 1 μM
28,BRD9,5 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in RI-1 cells after 2 h treatment at 1 μM
28,BRD7,8 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in RI-1 cells after 2 h treatment at 1 μM
29,BRD7,0 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in RI-1 cells after 2 h treatment at 1 μM
29,BRD9,0 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in RI-1 cells after 2 h treatment at 1 μM
30,BRD7,2 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in RI-1 cells after 2 h treatment at 1 μM
30,BRD9,11 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in RI-1 cells after 2 h treatment at 1 μM
31,BRD9,5 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in RI-1 cells after 2 h treatment at 1 μM
31,BRD7,15 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in RI-1 cells after 2 h treatment at 1 μM
32,BRD7,30 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in RI-1 cells after 2 h treatment at 1 μM
32,BRD9,32 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in RI-1 cells after 2 h treatment at 1 μM
33,BRD7,0 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in RI-1 cells after 2 h treatment at 1 μM
33,BRD9,0 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in RI-1 cells after 2 h treatment at 1 μM
34,BRD7,0 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in RI-1 cells after 2 h treatment at 1 μM
34,BRD9,8 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in RI-1 cells after 2 h treatment at 1 μM
35,BRD7,3 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD7 degradation in RI-1 cells after 2 h treatment at 1 μM
35,BRD9,6 (WB),10.1021/acs.jmedchem.8b01413,,,,% BRD9 degradation in RI-1 cells after 2 h treatment at 1 μM
36,MCL1,11/37/37/42/0 (WB),10.1021/acs.jmedchem.9b00455,,,,% MCL1 degradation in OPM2 cells after 48 h treatment at 25/100/250/500/1000 nM
37,MDM2,50/70/90 (WB),10.1021/acs.jmedchem.8b00909,,,,% MDM2 degradation in RS4;11 cells after 2 h treatment at 3/10/30 nM
38,MDM2,80/90/93 (WB),10.1021/acs.jmedchem.8b00909,,,,% MDM2 degradation in RS4;11 cells after 2 h treatment at 3/10/30 nM
39,MDM2,0/10 (WB),10.1021/acs.jmedchem.8b00909,,,,% MDM2 degradation in RS4;11 cells after 2 h treatment at 100/300 nM
40,MDM2,50/60 (WB),10.1021/acs.jmedchem.8b00909,,,,% MDM2 degradation in RS4;11 cells after 2 h treatment at 30/100 nM
41,MDM2,70/70 (WB),10.1021/acs.jmedchem.8b00909,,,,% MDM2 degradation in RS4;11 cells after 2 h treatment at 10/30 nM
42,MDM2,60/80 (WB),10.1021/acs.jmedchem.8b00909,,,,% MDM2 degradation in RS4;11 cells after 2 h treatment at 10/30 nM
43,MDM2,10/40 (WB),10.1021/acs.jmedchem.8b00909,,,,% MDM2 degradation in RS4;11 cells after 2 h treatment at 30/100 nM
44,MDM2,0/30 (WB),10.1021/acs.jmedchem.8b00909,,,,% MDM2 degradation in RS4;11 cells after 2 h treatment at 100/300 nM
45,MDM2,70/60 (WB),10.1021/acs.jmedchem.8b00909,,,,% MDM2 degradation in RS4;11 cells after 2 h treatment at 10/30 nM
46,MDM2,70/60 (WB),10.1021/acs.jmedchem.8b00909,,,,% MDM2 degradation in RS4;11 cells after 2 h treatment at 10/30 nM
47,MDM2,,10.1021/acs.jmedchem.8b00909,,,,
48,MDM2,,10.1021/acs.jmedchem.8b00909,,,,
49,MDM2,60/93/96/98 (WB),10.1021/acs.jmedchem.8b00909,,,,% MDM2 degradation in RS4;11 cells after 2 h treatment at 1/3/10/30 nM
50,MDM2,80/95/98/99 (WB),10.1021/acs.jmedchem.8b00909,,,,% MDM2 degradation in RS4;11 cells after 2 h treatment at 1/3/10/30 nM
51,MDM2,,10.1021/acs.jmedchem.8b00909,,,,
52,MDM2,60/80/70 (WB),10.1021/acs.jmedchem.8b00909,,,,% MDM2 degradation in RS4;11 cells after 2 h treatment at 3/10/30 nM
53,MDM2,60/80/80 (WB),10.1021/acs.jmedchem.8b00909,,,,% MDM2 degradation in RS4;11 cells after 2 h treatment at 3/10/30 nM
54,MDM2,,10.1021/acs.jmedchem.8b00909,,N.D.,,
55,MDM2,,10.1021/acs.jmedchem.8b00909,,N.D.,,
56,MDM2,,10.1021/acs.jmedchem.8b00909,,N.D.,,
57,ER,,10.1021/acs.jmedchem.8b01572,,N.D.,,
58,ER,,10.1021/acs.jmedchem.8b01572,,N.D.,,
59,ER,0/99.4/99.6/33 (WB),10.1021/acs.jmedchem.8b01572,,,,% ER degradation in MCF-7 cells after 4 h treatment at 1/10/100/1000 nM
60,ER,79/99.6/99.7/36 (WB),10.1021/acs.jmedchem.8b01572,,,,% ER degradation in MCF-7 cells after 4 h treatment at 1/10/100/1000 nM
61,ER,37/0/0 (WB),10.1021/acs.jmedchem.8b01572,,,,% ER degradation in MCF-7 cells after 4 h treatment at 1/10/100 nM
62,ER,10/0/8 (WB),10.1021/acs.jmedchem.8b01572,,,,% ER degradation in MCF-7 cells after 4 h treatment at 1/10/100 nM
63,ER,74/34/88 (WB),10.1021/acs.jmedchem.8b01572,,,,% ER degradation in MCF-7 cells after 4 h treatment at 1/10/100 nM
64,ER,68/92/94 (WB),10.1021/acs.jmedchem.8b01572,,,,% ER degradation in MCF-7 cells after 4 h treatment at 1/10/100 nM
115,AR,20/81/97,10.1021/acs.jmedchem.8b01631,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
116,AR,38/80/95,10.1021/acs.jmedchem.8b01631,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
117,AR,18/34/35,10.1021/acs.jmedchem.8b01631,,,,% AR degradation in LNCaP cells after 6 h treatment at 100/1000/10000 nM
118,AR,76/98/99,10.1021/acs.jmedchem.8b01631,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
118,AR,76/>95/>99,10.1021/acs.jmedchem.9b01393,7.2/1,>95/>95,Degradation of AR in LNCaP/VCaP AR+ cells after 6 h treatment,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
119,AR,65/93/78,10.1021/acs.jmedchem.8b01631,,,,% AR degradation in LNCaP cells after 6 h treatment at 100/1000/10000 nM
120,AR,89/99/100,10.1021/acs.jmedchem.8b01631,0.86/0.76/10.4,>95/>95/>95,Degradation of AR in LNCaP/VCaP/22Rv1 cells after 24 h treatment,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
121,AR,76/99/100,10.1021/acs.jmedchem.8b01631,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
122,AR,39/77/99,10.1021/acs.jmedchem.8b01631,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
123,AR,<5/<5/<5,10.1021/acs.jmedchem.8b01631,,,,% AR degradation in LNCaP cells after 6 h treatment at 100/1000/10000 nM
124,AR,<5/<5/<5,10.1021/acs.jmedchem.8b01631,,,,% AR degradation in LNCaP cells after 6 h treatment at 100/1000/10000 nM
125,AR,43/91/96,10.1021/acs.jmedchem.8b01631,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
126,AR,7/20/5,10.1021/acs.jmedchem.8b01631,,,,% AR degradation in LNCaP cells after 6 h treatment at 100/1000/10000 nM
127,AR,2/25/20,10.1021/acs.jmedchem.8b01631,,,,% AR degradation in LNCaP cells after 6 h treatment at 100/1000/10000 nM
128,BRD4,,10.1021/acs.jmedchem.6b01816,,,,
128,BRD2,,10.1021/acs.jmedchem.6b01816,,,,
128,BRD3,,10.1021/acs.jmedchem.6b01816,,,,
129,BRD3,,10.1021/acs.jmedchem.6b01816,,,,
129,BRD2,,10.1021/acs.jmedchem.6b01816,,,,
129,BRD4,,10.1021/acs.jmedchem.6b01816,,,,
130,BRD2,,10.1021/acs.jmedchem.6b01816,,,,
130,BRD3,,10.1021/acs.jmedchem.6b01816,,,,
130,BRD4,,10.1021/acs.jmedchem.6b01816,,,,
131,BRD4,,10.1021/acs.jmedchem.6b01816,,,,
131,BRD2,,10.1021/acs.jmedchem.6b01816,,,,
131,BRD3,,10.1021/acs.jmedchem.6b01816,,,,
132,BRD2,,10.1021/acs.jmedchem.6b01816,,,,
132,BRD4,,10.1021/acs.jmedchem.6b01816,,,,
132,BRD3,,10.1021/acs.jmedchem.6b01816,,,,
133,BRD4,,10.1021/acs.jmedchem.6b01816,,,,
133,BRD2,,10.1021/acs.jmedchem.6b01816,,,,
133,BRD3,,10.1021/acs.jmedchem.6b01816,,,,
134,BRD3,,10.1021/acs.jmedchem.6b01816,,,,
134,BRD4,,10.1021/acs.jmedchem.6b01816,,,,
134,BRD2,,10.1021/acs.jmedchem.6b01816,,,,
135,BRD4,,10.1021/acs.jmedchem.6b01816,,,,
135,BRD3,,10.1021/acs.jmedchem.6b01816,,,,
135,BRD2,,10.1021/acs.jmedchem.6b01816,,,,
136,BRD4,,10.1021/acs.jmedchem.6b01816,,,,
136,BRD2,,10.1021/acs.jmedchem.6b01816,,,,
136,BRD3,,10.1021/acs.jmedchem.6b01816,,,,
137,BRD3,,10.1021/acs.jmedchem.6b01816,,,,
137,BRD2,,10.1021/acs.jmedchem.6b01816,,,,
137,BRD4,,10.1021/acs.jmedchem.6b01816,,,,
138,BRD3,,10.1021/acs.jmedchem.6b01816,,,,
138,BRD2,,10.1021/acs.jmedchem.6b01816,,,,
138,BRD4,,10.1021/acs.jmedchem.6b01816,,,,
139,BRD3,,10.1021/acs.jmedchem.6b01816,,,,
139,BRD2,,10.1021/acs.jmedchem.6b01816,,,,
139,BRD4,,10.1021/acs.jmedchem.6b01816,,,,
140,BRD3,,10.1021/acs.jmedchem.6b01816,,,,
140,BRD4,,10.1021/acs.jmedchem.6b01816,,,,
140,BRD2,,10.1021/acs.jmedchem.6b01816,,,,
141,BRD2,,10.1021/acs.jmedchem.6b01816,,,,
141,BRD4,,10.1021/acs.jmedchem.6b01816,,,,
141,BRD3,,10.1021/acs.jmedchem.6b01816,,,,
142,BRD2,,10.1021/acs.jmedchem.8b00506,,,,
142,BRD2,,10.1021/acs.jmedchem.6b01816,,,,
142,BRD3,,10.1021/acs.jmedchem.6b01816,,,,
142,BRD4,,10.1021/acs.jmedchem.6b01816,,,,
142,BRD3,,10.1021/acs.jmedchem.8b00506,,,,
142,BRD4,,10.1021/acs.jmedchem.8b00506,,,,
142,BRD2,,10.1158/0008-5472.CAN-16-2622,,,,
142,BRD3,,10.1158/0008-5472.CAN-16-2622,,,,
142,BRD4,,10.1158/0008-5472.CAN-16-2622,,,,
143,BRD2,,10.1021/acs.jmedchem.6b01816,,,,
143,BRD3,,10.1021/acs.jmedchem.6b01816,,,,
143,BRD4,,10.1021/acs.jmedchem.6b01816,,,,
144,BRD4,,10.1021/acs.jmedchem.6b01816,,,,
144,BRD2,,10.1021/acs.jmedchem.6b01816,,,,
144,BRD3,,10.1021/acs.jmedchem.6b01816,,,,
145,BRD3,,10.1021/acs.jmedchem.6b01816,,,,
145,BRD2,,10.1021/acs.jmedchem.6b01816,,,,
145,BRD4,,10.1021/acs.jmedchem.6b01816,,,,
146,BRD4,,10.1021/acs.jmedchem.6b01781,490/500,,Degradation of BRD4 in NCI-H661/NCI-H838 cells after 4h treatment,
147,BRD4,,10.1021/acs.jmedchem.6b01781,>5000/130,,Degradation of BRD4 in NCI-H661/NCI-H838 cells after 4h treatment,
148,BRD4,,10.1021/acs.jmedchem.6b01781,>5000/1260,,Degradation of BRD4 in NCI-H661/NCI-H838 cells after 4h treatment,
149,BRD4,,10.1021/acs.jmedchem.6b01781,450/250,,Degradation of BRD4 in NCI-H661/NCI-H838 cells after 4h treatment,
150,BRD4,,10.1021/acs.jmedchem.6b01781,200/150,,Degradation of BRD4 in NCI-H661/NCI-H838 cells after 4h treatment,
151,BRD4,,10.1021/acs.jmedchem.6b01781,59/550,,Degradation of BRD4 in NCI-H661/NCI-H838 cells after 4h treatment,
152,BRD4,,10.1021/acs.jmedchem.6b01781,83/470,,Degradation of BRD4 in NCI-H661/NCI-H838 cells after 4h treatment,
153,BRD4,,10.1021/acs.jmedchem.6b01781,240/1670,,Degradation of BRD4 in NCI-H661/NCI-H838 cells after 4h treatment,
154,BRD4,,10.1021/acs.jmedchem.6b01781,460/3660,,Degradation of BRD4 in NCI-H661/NCI-H838 cells after 4h treatment,
155,BRD4,,10.1021/acs.jmedchem.6b01781,630/2730,,Degradation of BRD4 in NCI-H661/NCI-H838 cells after 4h treatment,
156,SIRT2,,10.1021/acs.jmedchem.6b01872,,,,
157,BRD2,,10.1021/acs.jmedchem.8b00506,,,,
157,BRD3,,10.1021/acs.jmedchem.8b00506,,,,
157,BRD4,,10.1021/acs.jmedchem.8b00506,,,,
158,BRD4,,10.1021/acs.jmedchem.8b00506,,,,
158,BRD2,,10.1021/acs.jmedchem.8b00506,,,,
158,BRD3,,10.1021/acs.jmedchem.8b00506,,,,
159,BRD4,,10.1021/acs.jmedchem.8b00506,,,,
159,BRD3,,10.1021/acs.jmedchem.8b00506,,,,
159,BRD2,,10.1021/acs.jmedchem.8b00506,,,,
160,BRD2,,10.1021/acs.jmedchem.8b00506,,,,
160,BRD4,,10.1021/acs.jmedchem.8b00506,,,,
160,BRD3,,10.1021/acs.jmedchem.8b00506,,,,
161,BRD3,,10.1021/acs.jmedchem.8b00506,,,,
161,BRD4,,10.1021/acs.jmedchem.8b00506,,,,
161,BRD2,,10.1021/acs.jmedchem.8b00506,,,,
162,BRD3,,10.1021/acs.jmedchem.8b00506,,,,
162,BRD4,,10.1021/acs.jmedchem.8b00506,,,,
162,BRD2,,10.1021/acs.jmedchem.8b00506,,,,
163,BRD4,,10.1021/acs.jmedchem.8b00506,,,,
163,BRD2,,10.1021/acs.jmedchem.8b00506,,,,
163,BRD3,,10.1021/acs.jmedchem.8b00506,,,,
164,BRD4,,10.1021/acs.jmedchem.8b00506,,,,
164,BRD2,,10.1021/acs.jmedchem.8b00506,,,,
164,BRD3,,10.1021/acs.jmedchem.8b00506,,,,
165,BRD2,,10.1021/acs.jmedchem.8b00506,,,,
165,BRD4,,10.1021/acs.jmedchem.8b00506,,,,
165,BRD3,,10.1021/acs.jmedchem.8b00506,,,,
166,BRD4,,10.1021/acs.jmedchem.8b00506,,,,
166,BRD3,,10.1021/acs.jmedchem.8b00506,,,,
166,BRD2,,10.1021/acs.jmedchem.8b00506,,,,
167,BRD3,,10.1021/acs.jmedchem.8b00506,,,,
167,BRD2,,10.1021/acs.jmedchem.8b00506,,,,
167,BRD4,,10.1021/acs.jmedchem.8b00506,,,,
168,PARP1,0 (WB),10.1039/c8cc07813k,,,,% PARP1 degradation in MDA-MB-231 cells after 24 h treatment at 10 μM
169,PARP1,0 (WB),10.1039/c8cc07813k,,,,% PARP1 degradation in MDA-MB-231 cells after 24 h treatment at 10 μM
170,PARP1,52 (WB),10.1039/c8cc07813k,,,,% PARP1 degradation in MDA-MB-231 cells after 24 h treatment at 10 μM
171,PARP1,0 (WB),10.1039/c8cc07813k,,,,% PARP1 degradation in MDA-MB-231 cells after 24 h treatment at 10 μM
172,PARP1,0 (WB),10.1039/c8cc07813k,,,,% PARP1 degradation in MDA-MB-231 cells after 24 h treatment at 10 μM
173,CRBN,,10.1039/c8cc09541h,,,,
174,CRBN,,10.1038/s41598-019-56177-5,367.8,85.1,Degradation of CRBN in HEK293T cells after 24h treatment,
175,CRBN,,10.1039/c8cc09541h,,,,
176,CRBN,,10.1039/c8cc09541h,1.5,,Degradation of CRBN in MM1S cells after 24h treatment,
177,CRBN,,10.1039/c8cc09541h,,,,
178,CRBN,,10.1039/c8cc09541h,,,,
179,CRBN,,10.1039/c8cc09541h,,,,
180,CRBN,,10.1039/c8cc09541h,,,,
181,p38alpha,,10.1038/s41467-018-08027-7,40.1,92.6,Degradation of p38alpha in MDA-MB-231 cells,
181,p38delta,,10.1038/s41467-018-08027-7,51.4,81.8,Degradation of p38delta in MDA-MB-231 cells,
182,p38delta,,10.1038/s41467-018-08027-7,91.7,96.7,Degradation of p38delta in MDA-MB-231 cells,
182,p38alpha,,10.1038/s41467-018-08027-7,18.8,99.4,Degradation of p38alpha in MDA-MB-231 cells,
183,p38alpha,,10.1038/s41467-018-08027-7,230,90.1,Degradation of p38alpha in MDA-MB-231 cells,
183,RIPK2,,10.1016/j.chembiol.2017.09.010,,,,
183,p38delta,,10.1016/j.chembiol.2017.09.010,,,,
183,c-Met,,10.1016/j.chembiol.2017.09.010,,,,
183,c-Met,,10.1016/j.chembiol.2017.09.009,,,,
183,p38delta,,10.1038/s41467-018-08027-7,456,54.3,Degradation of p38delta in MDA-MB-231 cells,
183,p38alpha,,10.1016/j.chembiol.2017.09.010,210,91,Degradation of p38alpha in MDA-MB-231 cells after 24 h treatment,
184,p38alpha,,10.1038/s41467-018-08027-7,9.5,99.6,Degradation of p38alpha in MDA-MB-231 cells,
184,p38delta,,10.1038/s41467-018-08027-7,1160,25.1,Degradation of p38delta in MDA-MB-231 cells,
185,p38alpha,,10.1038/s41467-018-08027-7,45.9,34.5,Degradation of p38alpha in MDA-MB-231 cells,
185,p38delta,,10.1038/s41467-018-08027-7,79.2,98.4,Degradation of p38delta in MDA-MB-231 cells,
186,p38delta,,10.1038/s41467-018-08027-7,106,43.5,Degradation of p38delta in MDA-MB-231 cells,
186,p38alpha,,10.1038/s41467-018-08027-7,127,25.3,Degradation of p38alpha in MDA-MB-231 cells,
187,p38alpha,,10.1038/s41467-018-08027-7,760,16.8,Degradation of p38alpha in MDA-MB-231 cells,
187,p38delta,,10.1038/s41467-018-08027-7,1890,78.7,Degradation of p38delta in MDA-MB-231 cells,
188,p38alpha,,10.1038/s41467-018-08027-7,304,19.9,Degradation of p38alpha in MDA-MB-231 cells,
188,p38delta,,10.1038/s41467-018-08027-7,1140,33.5,Degradation of p38delta in MDA-MB-231 cells,
189,CDK6,,10.1021/acs.jmedchem.9b00871,,,,
189,CDK4,,10.1021/acs.jmedchem.9b00871,,,,
190,CDK6,,10.1016/j.bmcl.2019.03.035,,,,
191,CDK6,,10.1016/j.bmcl.2019.03.035,,,,
192,CDK6,,10.1016/j.bmcl.2019.03.035,,,,
193,CDK6,,10.1016/j.bmcl.2019.03.035,,,,
194,BRD2,,10.1021/acs.orglett.9b01326,<0.5,,Degradation of BRD2,
194,BRD3,,10.1021/acs.orglett.9b01326,<0.5,,Degradation of BRD3,
194,BRD4,,10.1021/acs.orglett.9b01326,<0.5,,Degradation of BRD4,
195,ERRalpha,28/50,10.1021/acsmedchemlett.9b00025,,,,% ERRalpha degradation in MDA-MB-231 cells after 4 h treatment at 30/100 nM
196,ERRalpha,58/85,10.1021/acsmedchemlett.9b00025,,,,% ERRalpha degradation in MDA-MB-231 cells after 4 h treatment at 30/100 nM
197,ERRalpha,39/83/96,10.1021/acsmedchemlett.9b00025,,,,% ERRalpha degradation in MDA-MB-231 cells after 4 h treatment at 10/30/100 nM
198,ERRalpha,58/78,10.1021/acsmedchemlett.9b00025,,,,% ERRalpha degradation in MDA-MB-231 cells after 4 h treatment at 30/100 nM
199,ERRalpha,23/71,10.1021/acsmedchemlett.9b00025,,,,% ERRalpha degradation in MDA-MB-231 cells after 4 h treatment at 30/100 nM
200,ERRalpha,3/9,10.1021/acsmedchemlett.9b00025,,,,% ERRalpha degradation in MDA-MB-231 cells after 4 h treatment at 30/100 nM
201,ERRalpha,79/92,10.1021/acsmedchemlett.9b00025,,,,% ERRalpha degradation in MDA-MB-231 cells after 4 h treatment at 30/100 nM
202,ERRalpha,25/63/89,10.1021/acsmedchemlett.9b00025,,,,% ERRalpha degradation in MDA-MB-231 cells after 4 h treatment at 10/30/100 nM
203,ERRalpha,0/15/19,10.1021/acsmedchemlett.9b00025,,,,% ERRalpha degradation in MDA-MB-231 cells after 4 h treatment at 30/100/300 nM
204,ERRalpha,0/4/10,10.1021/acsmedchemlett.9b00025,,,,% ERRalpha degradation in MDA-MB-231 cells after 4 h treatment at 30/100/300 nM
205,BTK,85 (WB),10.1039/c8cc08716d,,,,% BTK degradation in Ramos cells after 16 h treatment at 2 μM
206,BTK,,10.1039/c8cc08716d,,,,
207,BTK,,10.1039/c8cc08716d,,,,
208,BRD4,,10.1158/0008-5472.CAN-18-2918,32,98,Degradation of BRD4 in HCT116 cells after 24 h treatment,
209,BRD4,,10.1158/0008-5472.CAN-18-2918,23.1,89,Degradation of BRD4 in HCT116 cells after 24 h treatment,
210,BTK,,10.1073/pnas.1803662115,,N.D.,,
211,BTK,,10.1073/pnas.1803662115,,N.D.,,
212,BTK,,10.1073/pnas.1803662115,,33/18,,
213,BTK,,10.1073/pnas.1803662115,,34/15,,
214,BTK,,10.1073/pnas.1803662115,1487/(n/a),64/36,Degradation of BTK in Ramos/THP-1 cells after 24 h treatment,
215,BTK,,10.1073/pnas.1803662115,36.9/398.5,85/68,Degradation of BTK in Ramos/THP-1 cells after 24 h treatment,
216,BTK,,10.1073/pnas.1803662115,21.8/469.9,84/63,Degradation of BTK in Ramos/THP-1 cells after 24 h treatment,
217,BTK,,10.1073/pnas.1803662115,4.5/90.5,87/75,Degradation of BTK in Ramos/THP-1 cells after 24 h treatment,
218,BTK,,10.1073/pnas.1803662115,5.9/217.7,85/71,Degradation of BTK in Ramos/THP-1 cells after 24 h treatment,
219,BTK,,10.1073/pnas.1803662115,1.1/37.4,87/80,Degradation of BTK in Ramos/THP-1 cells after 24 h treatment,
220,BTK,,10.1073/pnas.1803662115,9.7/184.1,85/70,Degradation of BTK in Ramos/THP-1 cells after 24 h treatment,
221,BTK,,10.1038/s41589-020-00686-2,182,,Degradation of BTK in THP-1 cells,
221,BTK,45/49/64/85 (WB),10.1073/pnas.1803662115,,,,% BTK degradation in THP-1 cells after 24 h treatment at 0.1/0.3/1/3 μM
222,BTK,27/36/17/33/70 (WB),10.1073/pnas.1803662115,,,,% BTK degradation in THP-1 cells after 24 h treatment at 0.03/0.1/0.3/1/3 μM
223,ALK,,10.1016/j.ejmech.2018.03.071,3/34,,Degradation of NPM-ALK/EML4-ALK in SU-DHL-1/NCI-H2228 cells after 16 h treatment,
224,ALK,,10.1016/j.ejmech.2018.03.071,11/59,,Degradation of NPM-ALK/EML4-ALK in SU-DHL-1/NCI-H2228 cells after 16 h treatment,
225,HDAC6,,10.1016/j.bmcl.2018.05.057,,,,
226,HDAC6,,10.1016/j.bmcl.2018.05.057,,,,
227,HDAC6,47.9/73.5,10.1021/acs.jmedchem.9b00516,9.12,84.07,Degradation of HDAC6 in MM1S cells after 6 h treatment,% HDAC6 degradation in MM1S cells after 6 h treatment at 10/100 nM
227,HDAC6,,10.1016/j.bmcl.2018.05.057,34,70.5,Degradation of HDAC6 in MCF-7 cells after 12 h treatment,
228,HDAC6,,10.1016/j.bmcl.2018.05.057,,,,
229,BRD3,,10.1021/jacs.8b05807,10,,Degradation of BRD3 in HeLa cells after 24 h treatment,
229,BRD2,,10.1021/jacs.8b05807,10,,Degradation of BRD2 in HeLa cells after 24 h treatment,
229,BRD4,,10.1021/jacs.8b05807,1~3,,Degradation of BRD4 in HeLa cells after 24 h treatment,
230,BRD2,,10.1021/jacs.8b05807,3000,,Degradation of BRD2 in HeLa cells after 24 h treatment,
230,BRD3,,10.1021/jacs.8b05807,3000,,Degradation of BRD3 in HeLa cells after 24 h treatment,
230,BRD4,,10.1021/jacs.8b05807,10-30,,Degradation of BRD4 in HeLa cells after 24 h treatment,
231,BRD4,11/36/14 (WB),10.1016/j.ejmech.2019.01.023,,,,% BRD4 degradation in 22RV1 cells after 24 h treatment at 10/100/1000 nM
232,BRD4,13/12/21/63/56 (WB),10.1016/j.ejmech.2019.01.023,,,,% BRD4 degradation in 22RV1 cells after 24 h treatment at 0.1/1/10/100/1000 nM
233,BRD4,,10.1016/j.ejmech.2019.01.023,3.3,,Degradation of BRD4 in 22RV1 cells after 24 h treatment,
234,BRD4,,10.1016/j.ejmech.2019.01.023,0.32,,Degradation of BRD4 in 22RV1 cells after 24 h treatment,
235,BRAF,,10.1016/j.bioorg.2019.03.035,,,,
236,BRAF,71.7/81,10.1016/j.bioorg.2019.03.035,,,,% B-Raf degradation in MCF-7 cells after 24 h treatment at 5000/10000 nM
237,BRAF,,10.1016/j.bioorg.2019.03.035,,,,
238,BRAF,,10.1016/j.bioorg.2019.03.035,,,,
239,CDK4,,10.1002/anie.201901336,,,,
239,CDK6,,10.1016/j.bmcl.2020.127106,13,,Degradation of CDK6 in Jurkat cells after 24 h treatment,
239,CDK6,,10.1021/acs.jmedchem.9b00871,14.3,,Degradation of CDK6 in U251 cells after 24 h treatment,
239,CDK4,,10.1016/j.bmcl.2020.127106,126,,Degradation of CDK4 in Jurkat cells after 24 h treatment,
239,CDK4,,10.1016/j.chembiol.2018.11.006,,,,
239,CDK4,,10.1021/acs.jmedchem.9b00871,>100,,Degradation of CDK4 in U251 cells after 24 h treatment,
239,Wee1,,10.1016/j.cell.2020.10.038,,,,
239,CDK6,,10.1002/anie.201901336,,,,
239,CDK6,,10.1016/j.chembiol.2018.11.006,,,,
240,PDK3,,10.1016/j.cell.2020.10.038,,,,
240,PDK1,,10.1016/j.cell.2020.10.038,,,,
240,BCKDK,,10.1016/j.cell.2020.10.038,,,,
240,CDK6,,10.1002/anie.201901336,,,,
240,CDK6,,10.1016/j.chembiol.2018.11.006,,,,
240,CDK4,,10.1016/j.cell.2020.10.038,,,,
240,Wee1,,10.1016/j.cell.2020.10.038,,,,
240,PDK2,,10.1016/j.cell.2020.10.038,,,,
240,COQ8A,,10.1016/j.cell.2020.10.038,,,,
241,BTK,,10.1038/s41422-018-0055-1,,,,
242,BTK C481S,41/69/78 (WB),10.1038/s41422-018-0055-1,,,,% BTK C481S degradation in HeLa cells after 4 days treatment at 30/100/300 nM
242,BTK,,10.1038/s41422-018-0055-1,8.5/6.3/9.2/11.4,,Degradation of BTK in RAMOS/HBL-1/Mino/IgE MM cells after 48 h treatment,
243,BTK,,10.1038/s41422-018-0055-1,,,,
244,BTK,,10.1038/s41422-018-0055-1,,,,
245,BTK,,10.1038/s41422-018-0055-1,,,,
246,BTK,,10.1038/s41422-018-0055-1,,,,
247,BTK,,10.1038/s41422-018-0055-1,,,,
248,BTK,,10.1038/s41422-018-0055-1,,,,
249,BTK,,10.1038/s41422-018-0055-1,,,,
250,BTK,,10.1038/s41422-018-0055-1,,,,
251,BTK,,10.1038/s41422-018-0055-1,,,,
252,BTK,,10.1038/s41422-018-0055-1,,,,
253,BTK,,10.1038/s41422-018-0055-1,,,,
254,BTK,,10.1038/s41422-018-0055-1,,,,
255,AR,,10.1038/s42003-018-0105-8,,47,,
256,AR,,10.1038/s42003-018-0105-8,15,76,Degradation of AR in VCaP cells after 20 h treatment,
257,AR,,10.1038/s42003-018-0105-8,5,98,Degradation of AR in VCaP cells after 20 h treatment,
258,BCL6,82 (WB),10.1021/acschembio.8b00698,,,,% BTK C481S degradation in OCI-Ly1 cells after 4 h treatment at 1 μM
259,ALK,,10.1016/j.bbrc.2018.09.169,,,,
260,ALK,,10.1016/j.bbrc.2018.09.169,,,,
261,ALK,,10.1016/j.bbrc.2018.09.169,,,,
262,ALK,,10.1016/j.bbrc.2018.09.169,,,,
263,ALK,,10.1016/j.bbrc.2018.09.169,,,,
264,ALK,,10.1016/j.bbrc.2018.09.169,,,,
265,FAK,,10.1021/jacs.8b08008,23.2,99,Degradation of Fak in PC3 cells after 24 h treatment,
266,FAK,,10.1021/jacs.8b08008,7.6,99,Degradation of Fak in PC3 cells after 24 h treatment,
267,FAK,,10.1021/jacs.8b08008,3,99,Degradation of Fak in PC3 cells after 24 h treatment,
268,FAK,,10.1021/jacs.8b08008,4,99,Degradation of Fak in PC3 cells after 24 h treatment,
269,FAK,,10.1021/jacs.8b08008,20.8,99,Degradation of Fak in PC3 cells after 24 h treatment,
270,FAK,,10.1021/jacs.8b08008,48.1,91,Degradation of Fak in PC3 cells after 24 h treatment,
271,FAK,,10.1021/jacs.8b08008,8.2,98,Degradation of Fak in PC3 cells after 24 h treatment,
272,FAK,,10.1021/jacs.8b08008,26.7,99,Degradation of Fak in PC3 cells after 24 h treatment,
273,FAK,,10.1021/jacs.8b08008,<10,87,Degradation of Fak in PC3 cells after 24 h treatment,
274,FLT3,,10.1021/jacs.8b10320,,,,
275,EGFR,,10.1016/j.chembiol.2017.09.009,39.2/736.2,97.6/68.8,Degradation of WT/Exon 20 Ins EGFR in OVCAR8/HeLa cells after 24 h treatment,
275,HER2,,10.1016/j.chembiol.2017.09.009,,,,
276,EGFR,,10.1016/j.chembiol.2017.09.009,11.7/22.3,98.9/96.6,Degradation of Exon 19 del/L858R EGFR in HCC827/H3255 cells after 24 h treatment,
277,EGFR,,10.1016/j.chembiol.2017.09.009,215.8,79.1,"Degradation of L858R, T790M EGFR in H1975 cells after 24 h treatment",
278,EGFR,,10.1016/j.chembiol.2017.09.009,,,,
279,MCL1,,10.1021/acs.jmedchem.9b00455,,,,
280,BTK,,10.1021/acs.biochem.8b00391,80.6,96,Degradation of BTK in NAMALWA cells after 24 h treatment,
281,BTK,,10.1021/acs.biochem.8b00391,90.1,93,Degradation of BTK in NAMALWA cells after 24 h treatment,
282,BTK,,10.1021/acs.biochem.8b00391,68.3,95,Degradation of BTK in NAMALWA cells after 24 h treatment,
283,BTK C481S,,10.1021/acs.biochem.8b00391,14.9,>99,Degradation of C481S BTK in XLA cells after 24 h treatment,
283,BTK,,10.1021/acs.biochem.8b00391,9.1/14.6,>99/(n/a),Degradation of BTK in NAMALWA/XLA cells after 24 h treatment,
283,BTK,,10.1016/j.bmcl.2019.126877,6.2,99,Degradation of BTK in NAMALWA cells after 24 h treatment,
284,BTK,,10.1021/acs.biochem.8b00391,11.6,>99,Degradation of BTK in NAMALWA cells after 24 h treatment,
285,RIPK2,,10.1016/j.chembiol.2017.09.010,,,,
285,MerTK,,10.1016/j.chembiol.2017.09.010,,,,
285,p38delta,,10.1016/j.chembiol.2017.09.010,27,91,Degradation of p38delta in MDA-MB-231 cells after 24 h treatment,
285,c-Met,,10.1016/j.chembiol.2017.09.010,,,,
286,CDK9,,10.1016/j.bioorg.2018.08.028,,,,
287,CDK9,,10.1016/j.bioorg.2018.08.028,,,,
288,CDK9,,10.1016/j.bioorg.2018.08.028,,,,
289,CDK9,,10.1016/j.bioorg.2018.08.028,,,,
290,CDK9,,10.1016/j.bioorg.2018.08.028,,,,
291,CDK9,,10.1016/j.bioorg.2018.08.028,,,,
292,CDK9,,10.1016/j.bioorg.2018.08.028,,,,
293,CDK9,,10.1016/j.bioorg.2018.08.028,,,,
294,GCN5,,10.1021/acschembio.8b00705,<3,,Degradation of GCN5 in THP1 cells after 18 h treatment,
294,PCAF,,10.1021/acschembio.8b00705,<1.5,,Degradation of PCAF in THP1 cells after 18 h treatment,
295,PCAF,27/15/21/34/34 (WB),10.1021/acschembio.8b00705,,,,% PCAF degradation in THP1 cells after 18 h treatment at 0.1/1/10/100/1000 nM
296,CRBN,,10.1021/acschembio.8b00693,,,,
297,CRBN,,10.1021/acschembio.8b00693,,,,
298,CRBN,,10.1021/acschembio.8b00693,,,,
299,CRBN,,10.1021/acschembio.8b00693,,,,
300,CRBN,,10.1021/acschembio.8b00693,,,,
301,CRBN,,10.1021/acschembio.8b00693,,,,
302,CRBN,,10.1021/acschembio.8b00693,,,,
303,CDK9,56/65 (WB),10.1039/c7cc03879h,,,,% CDK9 degradation in HCT116 cells after 6 h treatment at 10/20 μM
304,PI3Kalpha,,10.1016/j.ejmech.2018.03.066,,,,
305,PI3Kalpha,,10.1016/j.ejmech.2018.03.066,,,,
306,PI3Kalpha,,10.1016/j.ejmech.2018.03.066,,,,
307,PI3Kalpha,,10.1016/j.ejmech.2018.03.066,,,,
308,PI3Kalpha,,10.1016/j.ejmech.2018.03.066,,,,
309,PI3Kalpha,,10.1016/j.ejmech.2018.03.066,,,,
310,BRD4,,10.1021/acschembio.9b00092,,,,
310,BRD4,,10.1038/nchembio.2329,,,,
311,BRD4,,10.1038/nchembio.2329,,,,
312,BRD4,,10.1038/nchembio.2329,,,,
313,BRD4,,10.1038/nchembio.2329,,,,
314,BRD4,,10.1038/nchembio.2329,,,,
315,BRD4,,10.1038/nchembio.2329,,,,
316,BCR-ABL,,10.1002/anie.201507634,,,,
317,BCR-ABL,>90/>80 (WB),10.1002/anie.201507634,,,,% c-ABL/BCR-ABL degradation in K562 cells after 24 h treatment at 2.5 μM
318,BCR-ABL,,10.1002/anie.201507634,,,,
319,BCR-ABL,,10.1002/anie.201507634,,,,
320,BCR-ABL,,10.1002/anie.201507634,,,,
321,BCR-ABL,>65 (WB),10.1002/anie.201507634,,,,% c-ABL degradation in K562 cells after 24 h treatment at 1 μM
321,BCR-ABL,0,10.1021/acs.jmedchem.9b01264,,,,% BCR-ABL degradation in K562 cells after 16 h treatment at 10000 nM
322,BCR-ABL,,10.1002/anie.201507634,,,,
323,BCR-ABL,,10.1002/anie.201507634,,,,
324,BCR-ABL,,10.1002/anie.201507634,,,,
325,BCR-ABL,>85/>60 (WB),10.1002/anie.201507634,,,,% c-ABL/BCR-ABL degradation in K562 cells after 24 h treatment at 1 μM
325,BCR-ABL,,10.1021/acs.jmedchem.0c00967,,,,
326,BCR-ABL,,10.1002/anie.201507634,,,,
327,BCR-ABL,,10.1002/anie.201507634,,,,
328,BRD3,,10.1073/pnas.1521738113,<5/<5/<5,,Degradation of BRD3 in 22Rv1/VCaP/LnCaP95 cells after 16 h treatment,
328,BRD4,,10.1073/pnas.1521738113,<5/<5/<5,,Degradation of BRD4 in 22Rv1/VCaP/LnCaP95 cells after 16 h treatment,
328,BRD2,,10.1073/pnas.1521738113,<5/<5/<5,,Degradation of BRD2 in 22Rv1/VCaP/LnCaP95 cells after 16 h treatment,
328,BRD2,,10.1021/acs.jmedchem.8b00506,,,,
328,BRD3,,10.1021/acs.jmedchem.8b00506,,,,
328,BRD4,,10.1021/acs.jmedchem.8b00506,,,,
329,BRD4,,10.1016/j.chembiol.2015.05.009,<1/<1,,Degradation of BRD4 in Namalwa/CA-46 cells after overnight treatment,
329,BRD4,,10.1016/j.ejmech.2019.01.023,0.57,,Degradation of BRD4 in 22RV1 cells after 24 h treatment,
329,BRD4,,10.1021/acs.jmedchem.6b01912,0.6/1,97/100,Degradation of BRD4 short/long in HeLa cells after 24 h treatment,
329,BRD2,,10.1016/j.chembiol.2015.05.009,,,,
329,BRD3,,10.1021/acs.jmedchem.8b00506,,,,
329,BRD2,,10.1021/acs.jmedchem.8b00506,,,,
329,BRD3,,10.1016/j.chembiol.2015.05.009,,,,
329,BRD4,,10.1021/acs.jmedchem.8b00506,,,,
329,BRD2,,10.1021/acs.jmedchem.6b01912,6,83,Degradation of BRD2 in HeLa cells after 24 h treatment,
329,BRD3,,10.1021/acs.jmedchem.6b01912,0.8,98,Degradation of BRD3 in HeLa cells after 24 h treatment,
330,BRD3,,10.1021/acs.jmedchem.8b00506,,,,
330,BRD4,,10.1021/acs.orglett.9b01326,,,,
330,BRD4,,10.1126/science.aab1433,430,,Degradation of BRD4 in SUM149 cells after 18 h treatment,
330,BRD4,,10.1038/s41589-018-0055-y,500/1000,,Degradation of BRD4 BD1/2 assessed by EGFP/mCherry reporter assay,
330,BRD4,,10.1002/anie.202108848,5.27/2.9,,Degradation of BRD4 in MV4-11 cells after 12/24 h treatment,
330,BRD4,,10.1002/anie.202108848,230,,Degradation of BRD4 in HD-MB03 cells after 12 h treatment,
330,BRD4,,10.1021/acs.jmedchem.8b00506,,,,
330,BRD2,,10.1021/acs.orglett.9b01326,,,,
330,BRD3,,10.1021/acs.orglett.9b01326,,,,
330,BRD2,,10.1126/science.aab1433,,,,
330,BRD3,,10.1126/science.aab1433,,,,
330,BRD2,,10.1021/acs.jmedchem.6b01816,,,,
330,BRD3,,10.1021/acs.jmedchem.6b01816,,,,
330,BRD4,,10.1021/acs.jmedchem.6b01816,,,,
330,BRD2,,10.1021/acs.jmedchem.8b00506,,,,
331,FKBP12,50/83/95/73 (WB),10.1126/science.aab1433,,,,% FKBP12 degradation in MV4;11 cells after 18 h treatment at 0.01/0.1/1/10 μM
332,FKBP12,60/81/93/74 (WB),10.1126/science.aab1433,,,,% FKBP12 degradation in MV4;11 cells after 18 h treatment at 0.01/0.1/1/10 μM
333,ERRalpha,,10.1038/nchembio.1858,100,86,Degradation of ERRalpha in MCF-7 cells after 8 h treatment,
334,RIPK2,,10.1038/nchembio.1858,1.4,95,Degradation of RIPK2 in THP-1 cells after 16 h treatment,
334,RIPK2,,10.1038/s42003-020-0868-6,2,,Degradation of RIPK2 in THP-1 cells after 18 h treatment,
335,BRD3,,10.1038/nchembio.2329,,,,
335,BRD2,,10.1038/nchembio.2329,,,,
335,BRD4,,10.1021/jacs.8b05807,,,,
335,BRD3,,10.1021/jacs.8b05807,,,,
335,BRD2,,10.1021/jacs.8b05807,,,,
335,BRD4,,10.1021/acschembio.5b00216,,,,
335,BRD3,,10.1021/acschembio.5b00216,,,,
335,BRD2,,10.1021/acschembio.5b00216,,,,
335,BRD3,,10.1038/s41589-019-0294-6,,,,
335,BRD3,,10.1021/acschembio.9b00092,,,,
335,BRD4,,10.1038/s41589-019-0294-6,,,,
335,BRD4,,10.1021/acschembio.9b00092,,,,
335,BRD2,,10.1021/acs.jmedchem.6b01912,40,98,Degradation of BRD2 in HeLa cells after 24 h treatment,
335,BRD2,,10.1038/s41589-019-0294-6,,,,
335,BRD4,,10.1038/nchembio.2329,,,,
335,BRD2,,10.1021/acschembio.9b00092,,,,
335,BRD4,,10.1021/acs.jmedchem.6b01912,8/3,98/100,Degradation of BRD4 short/long in HeLa cells after 24 h treatment,
335,BRD3,,10.1021/acs.jmedchem.6b01912,100,100,Degradation of BRD3 in HeLa cells after 24 h treatment,
336,BRD3,,10.1021/acs.jmedchem.6b01912,316,99,Degradation of BRD3 in HeLa cells after 24 h treatment,
336,BRD4,,10.1021/acs.jmedchem.6b01912,4/10,99/100,Degradation of BRD4 short/long in HeLa cells after 24 h treatment,
336,BRD2,,10.1021/acs.jmedchem.6b01912,200,97,Degradation of BRD2 in HeLa cells after 24 h treatment,
337,BRD2,,10.1021/acschembio.5b00216,,,,
337,BRD3,,10.1021/acschembio.5b00216,,,,
337,BRD4,,10.1021/acschembio.5b00216,,,,
338,AR,,10.1016/j.bmcl.2008.07.114,,,,
339,BRD3,,10.1038/s41589-018-0055-y,,,,
339,BRD4,,10.1038/s41589-018-0055-y,10/50,,Degradation of BRD4 BD1/2 assessed by EGFP/mCherry reporter assay,
339,BRD4,,10.1021/acschembio.1c00376,6,97,Degradation of BRD4 in HEK293T cells after 3 h treatment,
339,BRD2 BD2,,10.1038/s41589-018-0055-y,,,,
340,BRD4,,10.1038/s41589-018-0055-y,50/>1000,,Degradation of BRD4 BD1/2 assessed by EGFP/mCherry reporter assay,
341,BRD4,,10.1038/s41589-018-0055-y,,,,
342,BRD3 BD1,,10.1038/s41589-018-0055-y,,,,
342,BRD4 BD1,,10.1038/s41589-018-0055-y,500,,Degradation of BRD4 BD1 assessed by EGFP/mCherry reporter assay,
343,BRD4,,10.1038/s41589-018-0055-y,5/5,,Degradation of BRD4 BD1/2 assessed by EGFP/mCherry reporter assay,
344,BRD4,,10.1038/s41589-018-0055-y,,,,
345,BRD4 BD1,,10.1038/s41589-018-0055-y,,,,
346,BRD4,,10.1038/s41589-018-0055-y,,,,
347,BRD4,,10.1038/s41589-018-0055-y,,,,
348,BRD4 BD1,,10.1038/s41589-018-0055-y,,,,
349,BRD4 BD1,,10.1038/s41589-018-0055-y,,,,
350,BRD4 BD1,,10.1038/s41589-018-0055-y,5,,Degradation of BRD4 BD1 assessed by EGFP/mCherry reporter assay,
351,MCL1,,10.1021/acs.jmedchem.9b00455,,,,
352,MCL1,,10.1021/acs.jmedchem.9b00455,,,,
353,MCL1,,10.1021/acs.jmedchem.9b00455,,,,
354,AR,68/>95/>99,10.1021/acs.jmedchem.9b01393,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
355,AR,81/>95/>99,10.1021/acs.jmedchem.9b01393,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
356,AR,45/76/>95,10.1021/acs.jmedchem.9b01393,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
357,AR,85/>95/>99,10.1021/acs.jmedchem.9b01393,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
358,AR,92/>95/>99,10.1021/acs.jmedchem.9b01393,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
359,AR,62/72/>99,10.1021/acs.jmedchem.9b01393,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
360,AR,8/11/17,10.1021/acs.jmedchem.9b01393,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
361,AR,6/68/86,10.1021/acs.jmedchem.9b01393,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
362,AR,21/67/68,10.1021/acs.jmedchem.9b01393,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
363,AR,90/>95/>99,10.1021/acs.jmedchem.9b01393,0.5/1/0.2,>99/>95/>95,Degradation of AR in LNCaP/VCaP/22Rv1 cells after 6 h treatment,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
364,AR,48/>95/>99,10.1021/acs.jmedchem.9b01393,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
365,AR,40/>95/>99,10.1021/acs.jmedchem.9b01393,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
366,AR,38/>95/>99,10.1021/acs.jmedchem.9b01393,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
367,AR,<5/>95/>99,10.1021/acs.jmedchem.9b01393,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
368,AR,56/>95/>99,10.1021/acs.jmedchem.9b01393,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
369,AR,62/>95/>99,10.1021/acs.jmedchem.9b01393,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
370,AR,85/>95/>99,10.1021/acs.jmedchem.9b01393,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
371,AR,31/>95/>99,10.1021/acs.jmedchem.9b01393,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
372,AR,80/>95/>99,10.1021/acs.jmedchem.9b01393,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
373,AR,76/>95/>99,10.1021/acs.jmedchem.9b01393,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
374,AR,<5/<5/<5,10.1021/acs.jmedchem.9b01393,,,,% AR degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
375,CDK4,,10.1021/acs.jmedchem.9b00871,,,,
375,CDK6,,10.1021/acs.jmedchem.9b00871,,,,
376,CDK4,,10.1021/acs.jmedchem.9b00871,,,,
376,CDK6,,10.1021/acs.jmedchem.9b00871,,,,
377,CDK6,,10.1021/acs.jmedchem.9b00871,,,,
377,CDK4,,10.1021/acs.jmedchem.9b00871,,,,
378,CDK4,,10.1021/acs.jmedchem.9b00871,,,,
378,CDK6,,10.1021/acs.jmedchem.9b00871,,,,
379,CDK4,,10.1021/acs.jmedchem.9b00871,>100,,Degradation of CDK4 in U251 cells after 24 h treatment,
379,CDK6,,10.1021/acs.jmedchem.9b00871,1.1,,Degradation of CDK6 in U251 cells after 24 h treatment,
380,CDK4,,10.1021/acs.jmedchem.9b00871,>100,,Degradation of CDK4 in U251 cells after 24 h treatment,
380,CDK6,,10.1021/acs.jmedchem.9b00871,24.2,,Degradation of CDK6 in U251 cells after 24 h treatment,
381,CDK4,,10.1021/acs.jmedchem.9b00871,>100,,Degradation of CDK4 in U251 cells after 24 h treatment,
381,CDK6,,10.1021/acs.jmedchem.9b00871,31,,Degradation of CDK6 in U251 cells after 24 h treatment,
382,CDK4,,10.1021/acs.jmedchem.9b00871,>100,,Degradation of CDK4 in U251 cells after 24 h treatment,
382,CDK6,,10.1021/acs.jmedchem.9b00871,2.1,,Degradation of CDK6 in U251 cells after 24 h treatment,
383,CDK4,,10.1021/acs.jmedchem.9b00871,,,,
383,CDK6,,10.1021/acs.jmedchem.9b00871,,,,
384,CDK6,,10.1021/acs.jmedchem.9b00871,5.3,,Degradation of CDK6 in U251 cells after 24 h treatment,
384,CDK4,,10.1021/acs.jmedchem.9b00871,>100,,Degradation of CDK4 in U251 cells after 24 h treatment,
385,CDK6,,10.1021/acs.jmedchem.9b00871,10.6,,Degradation of CDK6 in U251 cells after 24 h treatment,
385,CDK4,,10.1021/acs.jmedchem.9b00871,>100,,Degradation of CDK4 in U251 cells after 24 h treatment,
386,CDK6,,10.1021/acs.jmedchem.9b00871,1.6,,Degradation of CDK6 in U251 cells after 24 h treatment,
386,CDK4,,10.1021/acs.jmedchem.9b00871,>50,,Degradation of CDK4 in U251 cells after 24 h treatment,
387,CDK6,,10.1021/acs.jmedchem.9b00871,1.7,,Degradation of CDK6 in U251 cells after 24 h treatment,
387,CDK4,,10.1021/acs.jmedchem.9b00871,>50,,Degradation of CDK4 in U251 cells after 24 h treatment,
388,CDK4,,10.1021/acs.jmedchem.9b00871,,,,
388,CDK6,,10.1021/acs.jmedchem.9b00871,,,,
389,CDK4,,10.1021/acs.jmedchem.9b00871,,,,
389,CDK6,,10.1021/acs.jmedchem.9b00871,,,,
390,CDK4,,10.1021/acs.jmedchem.9b00871,,,,
390,CDK6,,10.1021/acs.jmedchem.9b00871,,,,
391,CDK6,,10.1021/acs.jmedchem.9b00871,,,,
391,CDK4,,10.1021/acs.jmedchem.9b00871,,,,
392,CDK4,,10.1021/acs.jmedchem.9b00871,>100,,Degradation of CDK4 in U251 cells after 24 h treatment,
392,CDK6,,10.1021/acs.jmedchem.9b00871,81.6,,Degradation of CDK6 in U251 cells after 24 h treatment,
393,CDK6,,10.1021/acs.jmedchem.9b00871,86.8,,Degradation of CDK6 in U251 cells after 24 h treatment,
393,CDK4,,10.1021/acs.jmedchem.9b00871,>100,,Degradation of CDK4 in U251 cells after 24 h treatment,
394,CDK4,,10.1021/acs.jmedchem.9b00871,>500,,Degradation of CDK4 in U251 cells after 24 h treatment,
394,CDK6,,10.1021/acs.jmedchem.9b00871,8.6,,Degradation of CDK6 in U251 cells after 24 h treatment,
395,CDK4,,10.1021/acs.jmedchem.9b00871,>500,,Degradation of CDK4 in U251 cells after 24 h treatment,
395,CDK6,,10.1021/acs.jmedchem.9b00871,129.7,,Degradation of CDK6 in U251 cells after 24 h treatment,
396,CDK6,,10.1021/acs.jmedchem.9b00871,271.9,,Degradation of CDK6 in U251 cells after 24 h treatment,
396,CDK4,,10.1021/acs.jmedchem.9b00871,>500,,Degradation of CDK4 in U251 cells after 24 h treatment,
397,CDK6,,10.1021/acs.jmedchem.9b00871,145.5,,Degradation of CDK6 in U251 cells after 24 h treatment,
397,CDK4,,10.1021/acs.jmedchem.9b00871,>500,,Degradation of CDK4 in U251 cells after 24 h treatment,
398,BTK,,10.1073/pnas.1803662115,,N.D.,,
399,BTK,,10.1073/pnas.1803662115,,N.D.,,
400,BCR-ABL,,10.1002/anie.201507634,,N.D.,,
401,BCR-ABL,,10.1002/anie.201507634,,N.D.,,
402,BCR-ABL,,10.1002/anie.201507634,,N.D.,,
403,BCR-ABL,,10.1002/anie.201507634,,N.D.,,
404,BCR-ABL,,10.1002/anie.201507634,,N.D.,,
405,BCR-ABL,,10.1002/anie.201507634,,N.D.,,
406,BCR-ABL,,10.1002/anie.201507634,,N.D.,,
407,BCR-ABL,,10.1002/anie.201507634,,N.D.,,
408,BCR-ABL,,10.1002/anie.201507634,,N.D.,,
409,BCR-ABL,,10.1002/anie.201507634,,N.D.,,
410,BCR-ABL,,10.1002/anie.201507634,,N.D.,,
411,BCR-ABL,,10.1002/anie.201507634,,N.D.,,
412,BRD4,,10.1038/s41589-018-0055-y,,N.D.,,
412,BRD3,,10.1038/s41589-018-0055-y,,N.D.,,
412,BRD2,,10.1038/s41589-018-0055-y,,N.D.,,
413,CDK4,,10.1021/acs.jmedchem.9b00871,,N.D.,,
413,CDK6,,10.1021/acs.jmedchem.9b00871,,N.D.,,
414,CDK4,,10.1021/acs.jmedchem.9b00871,,N.D.,,
414,CDK6,,10.1021/acs.jmedchem.9b00871,,N.D.,,
415,CDK6,,10.1021/acs.jmedchem.9b00871,,N.D.,,
415,CDK4,,10.1021/acs.jmedchem.9b00871,,N.D.,,
416,CDK6,,10.1021/acs.jmedchem.9b00871,,N.D.,,
416,CDK4,,10.1021/acs.jmedchem.9b00871,,N.D.,,
417,CDK6,,10.1021/acs.jmedchem.9b00871,,N.D.,,
417,CDK4,,10.1021/acs.jmedchem.9b00871,,N.D.,,
418,CDK6,,10.1021/acs.jmedchem.9b00871,,N.D.,,
418,CDK4,,10.1021/acs.jmedchem.9b00871,,N.D.,,
419,CDK4,,10.1021/acs.jmedchem.9b00871,,N.D.,,
419,CDK6,,10.1021/acs.jmedchem.9b00871,,N.D.,,
420,CDK4,,10.1021/acs.jmedchem.9b00871,,N.D.,,
420,CDK6,,10.1021/acs.jmedchem.9b00871,,N.D.,,
421,CDK6,,10.1021/acs.jmedchem.9b00871,,N.D.,,
421,CDK4,,10.1021/acs.jmedchem.9b00871,,N.D.,,
422,CDK4,,10.1021/acs.jmedchem.9b00871,,N.D.,,
422,CDK6,,10.1021/acs.jmedchem.9b00871,,N.D.,,
423,CDK6,,10.1021/acs.jmedchem.9b00871,,N.D.,,
423,CDK4,,10.1021/acs.jmedchem.9b00871,,N.D.,,
424,CDK6,,10.1021/acs.jmedchem.9b00871,,N.D.,,
424,CDK4,,10.1021/acs.jmedchem.9b00871,,N.D.,,
425,CDK4,,10.1021/acs.jmedchem.9b00871,,N.D.,,
425,CDK6,,10.1021/acs.jmedchem.9b00871,,N.D.,,
426,CDK6,,10.1021/acs.jmedchem.9b00871,,N.D.,,
426,CDK4,,10.1021/acs.jmedchem.9b00871,,N.D.,,
427,MEK1,90/94,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
427,MEK2,,10.1021/acs.jmedchem.9b00810,,,,
428,MEK1,91/96,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
428,MEK2,,10.1021/acs.jmedchem.9b00810,,,,
429,MEK1,72/95,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
429,MEK2,,10.1021/acs.jmedchem.9b00810,,,,
430,MEK1,77/96,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
431,MEK1,47/94,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
432,MEK1,46/97,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
433,MEK1,18/48,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
434,MEK1,35/48,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
435,MEK1,67/91,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
436,MEK1,87/96,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
437,MEK1,16/39,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
438,MEK1,29/47,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
439,MEK1,3/38,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
440,MEK1,5/57,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
441,MEK1,30/65,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
442,MEK1,23/86,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
443,MEK1,8/57,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
444,MEK1,33/87,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
445,MEK1,41/88,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
446,MEK1,28/65,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
447,MEK1,45/47,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
448,MEK1,16/87,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
449,MEK1,57/93,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
450,MEK1,14/29,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
451,MEK1,30/81,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
452,MEK1,18/89,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
453,MEK1,42/94,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
454,MEK1,24/90,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
455,MEK1,55/96,10.1021/acs.jmedchem.9b00810,,,,% MEK1 degradation in A375 cells after 16 h treatment at 1000/10000 nM
456,BCR-ABL,0,10.1021/acs.jmedchem.9b01264,,,,% BCR-ABL degradation in K562 cells after 16 h treatment at 10000 nM
457,BCR-ABL,0,10.1021/acs.jmedchem.9b01264,,,,% BCR-ABL degradation in K562 cells after 16 h treatment at 10000 nM
458,BCR-ABL,0,10.1021/acs.jmedchem.9b01264,,,,% BCR-ABL degradation in K562 cells after 16 h treatment at 10000 nM
459,BCR-ABL,0,10.1021/acs.jmedchem.9b01264,,,,% BCR-ABL degradation in K562 cells after 16 h treatment at 10000 nM
460,BCR-ABL,0,10.1021/acs.jmedchem.9b01264,,,,% BCR-ABL degradation in K562 cells after 16 h treatment at 10000 nM
461,BCR-ABL,0,10.1021/acs.jmedchem.9b01264,,,,% BCR-ABL degradation in K562 cells after 16 h treatment at 10000 nM
462,BCR-ABL,0,10.1021/acs.jmedchem.9b01264,,,,% BCR-ABL degradation in K562 cells after 16 h treatment at 10000 nM
463,BCR-ABL,0,10.1021/acs.jmedchem.9b01264,,,,% BCR-ABL degradation in K562 cells after 16 h treatment at 10000 nM
464,BCR-ABL,,10.1021/acs.jmedchem.9b01264,10.1,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
465,BCR-ABL,,10.1021/acs.jmedchem.9b01264,37.9,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
466,BCR-ABL,,10.1021/acs.jmedchem.9b01264,8.5,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
467,BCR-ABL,,10.1021/acs.jmedchem.9b01264,17.9,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
468,BCR-ABL,,10.1021/acs.jmedchem.9b01264,34.7,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
469,BCR-ABL,,10.1021/acs.jmedchem.9b01264,40.2,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
470,BCR-ABL,,10.1021/acs.jmedchem.9b01264,611.4,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
471,BCR-ABL,0,10.1021/acs.jmedchem.9b01264,,,,% BCR-ABL degradation in K562 cells after 16 h treatment at 10000 nM
472,BCR-ABL,0,10.1021/acs.jmedchem.9b01264,,,,% BCR-ABL degradation in K562 cells after 16 h treatment at 10000 nM
473,BCR-ABL,0,10.1021/acs.jmedchem.9b01264,,,,% BCR-ABL degradation in K562 cells after 16 h treatment at 10000 nM
474,BCR-ABL,0,10.1021/acs.jmedchem.9b01264,,,,% BCR-ABL degradation in K562 cells after 16 h treatment at 10000 nM
475,STAT3,,10.1021/acs.jmedchem.9b01530,2630,,Degradation of total STAT3 and p-STAT3Y705 proteins in Molm-16 cells after 4 h treatment,
476,STAT3,,10.1021/acs.jmedchem.9b01530,260,,Degradation of total STAT3 and p-STAT3Y705 proteins in Molm-16 cells after 4 h treatment,
477,STAT3,,10.1021/acs.jmedchem.9b01530,60/28,,Degradation of total STAT3 and p-STAT3Y705 proteins in Molm-16/SU-DHL-1 cells after 4/16 h treatment,
478,STAT3,,10.1021/acs.jmedchem.9b01530,90,,Degradation of total STAT3 and p-STAT3Y705 proteins in Molm-16 cells after 4 h treatment,
479,STAT3,,10.1021/acs.jmedchem.9b01530,150,,Degradation of total STAT3 and p-STAT3Y705 proteins in Molm-16 cells after 4 h treatment,
480,STAT3,,10.1021/acs.jmedchem.9b01530,650/919,,Degradation of total STAT3 and p-STAT3Y705 proteins in Molm-16/SU-DHL-1 cells after 4/16 h treatment,
481,STAT3,,10.1021/acs.jmedchem.9b01530,240/49,,Degradation of total STAT3 and p-STAT3Y705 proteins in Molm-16/SU-DHL-1 cells after 4/16 h treatment,
482,STAT3,,10.1021/acs.jmedchem.9b01530,50/11,,Degradation of total STAT3 and p-STAT3Y705 proteins in Molm-16/SU-DHL-1 cells after 4/16 h treatment,
483,STAT3,,10.1021/acs.jmedchem.9b01530,180,,Degradation of total STAT3 and p-STAT3Y705 proteins in Molm-16 cells after 4 h treatment,
484,STAT3,,10.1021/acs.jmedchem.9b01530,250,,Degradation of total STAT3 and p-STAT3Y705 proteins in Molm-16 cells after 4 h treatment,
485,STAT3,,10.1021/acs.jmedchem.9b01530,180,,Degradation of total STAT3 and p-STAT3Y705 proteins in Molm-16 cells after 4 h treatment,
486,STAT3,,10.1021/acs.jmedchem.9b01530,2470,,Degradation of total STAT3 and p-STAT3Y705 proteins in Molm-16 cells after 4 h treatment,
487,STAT3,,10.1021/acs.jmedchem.9b01530,380,,Degradation of total STAT3 and p-STAT3Y705 proteins in Molm-16 cells after 4 h treatment,
488,STAT3,,10.1021/acs.jmedchem.9b01530,160,,Degradation of total STAT3 and p-STAT3Y705 proteins in Molm-16 cells after 4 h treatment,
489,STAT3,,10.1021/acs.jmedchem.9b01530,90,,Degradation of total STAT3 and p-STAT3Y705 proteins in Molm-16 cells after 4 h treatment,
490,STAT3,,10.1021/acs.jmedchem.9b01530,3540/>10000,,Degradation of total STAT3 and p-STAT3Y705 proteins in Molm-16/SU-DHL-1 cells after 4/16 h treatment,
491,STAT3,,10.1021/acs.jmedchem.9b01530,410,,Degradation of total STAT3 and p-STAT3Y705 proteins in Molm-16 cells after 4 h treatment,
492,STAT3,,10.1021/acs.jmedchem.9b01530,360,,Degradation of total STAT3 and p-STAT3Y705 proteins in Molm-16 cells after 4 h treatment,
493,STAT3,,10.1021/acs.jmedchem.9b01530,220/55,,Degradation of total STAT3 and p-STAT3Y705 proteins in Molm-16/SU-DHL-1 cells after 4/16 h treatment,
494,STAT3,,10.1021/acs.jmedchem.9b01530,640/890,,Degradation of total STAT3 and p-STAT3Y705 proteins in Molm-16/SU-DHL-1 cells after 4/16 h treatment,
495,STAT3,,10.1021/acs.jmedchem.9b01530,>10000,,Degradation of total STAT3 and p-STAT3Y705 proteins in Molm-16 cells after 4 h treatment,
496,STAT3,,10.1021/acs.jmedchem.9b01530,>10000,,Degradation of total STAT3 and p-STAT3Y705 proteins in Molm-16 cells after 4 h treatment,
497,STAT3,,10.1021/acs.jmedchem.9b01530,4450/>10000,,Degradation of total STAT3 and p-STAT3Y705 proteins in Molm-16/SU-DHL-1 cells after 4/16 h treatment,
498,BCL2,0/0 (WB),10.1021/acs.jmedchem.9b00919,,,,% BCL2 degradation in HeLa cells after 12 h treatment at 1/10 μM
498,MCL1,0/0 (WB),10.1021/acs.jmedchem.9b00919,,,,% MCL1 degradation in HeLa cells after 12 h treatment at 1/10 μM
499,MCL1,0/10 (WB),10.1021/acs.jmedchem.9b00919,,,,% MCL1 degradation in HeLa cells after 12 h treatment at 1/10 μM
499,BCL2,0/0 (WB),10.1021/acs.jmedchem.9b00919,,,,% BCL2 degradation in HeLa cells after 12 h treatment at 1/10 μM
500,MCL1,,10.1021/acs.jmedchem.9b00919,700,,Degradation of MCL1 in HeLa cells after 12 h treatment,
500,BCL2,10/0/10/0/20 (WB),10.1021/acs.jmedchem.9b00919,,,,% BCL2 degradation in HeLa cells after 12 h treatment at 0.1/0.3/1/3/10 μM
501,BCL2,0/10 (WB),10.1021/acs.jmedchem.9b00919,,,,% BCL2 degradation in HeLa cells after 12 h treatment at 1/10 μM
501,MCL1,0/10 (WB),10.1021/acs.jmedchem.9b00919,,,,% MCL1 degradation in HeLa cells after 12 h treatment at 1/10 μM
502,MCL1,10 (WB),10.1021/acs.jmedchem.9b00919,,,,% MCL1 degradation in HeLa cells after 12 h treatment at 10 μM
502,BCL2,,10.1021/acs.jmedchem.9b00919,3000,,Degradation of BCL2 in HeLa cells after 12 h treatment,
503,MCL1,0/0 (WB),10.1021/acs.jmedchem.9b00919,,,,% MCL1 degradation in HeLa cells after 12 h treatment at 1/10 μM
503,BCL2,10/10 (WB),10.1021/acs.jmedchem.9b00919,,,,% BCL2 degradation in HeLa cells after 12 h treatment at 1/10 μM
504,BCL2,0/0 (WB),10.1021/acs.jmedchem.9b00919,,,,% BCL2 degradation in HeLa cells after 12 h treatment at 1/10 μM
504,MCL1,0/0 (WB),10.1021/acs.jmedchem.9b00919,,,,% MCL1 degradation in HeLa cells after 12 h treatment at 1/10 μM
505,BCL2,0/0 (WB),10.1021/acs.jmedchem.9b00919,,,,% BCL2 degradation in HeLa cells after 12 h treatment at 1/10 μM
505,MCL1,10/20 (WB),10.1021/acs.jmedchem.9b00919,,,,% MCL1 degradation in HeLa cells after 12 h treatment at 1/10 μM
506,MCL1,10/20 (WB),10.1021/acs.jmedchem.9b00919,,,,% MCL1 degradation in HeLa cells after 12 h treatment at 1/10 μM
506,BCL2,0/0 (WB),10.1021/acs.jmedchem.9b00919,,,,% BCL2 degradation in HeLa cells after 12 h treatment at 1/10 μM
507,BCL2,0/0 (WB),10.1021/acs.jmedchem.9b00919,,,,% BCL2 degradation in HeLa cells after 12 h treatment at 1/10 μM
507,MCL1,0/0 (WB),10.1021/acs.jmedchem.9b00919,,,,% MCL1 degradation in HeLa cells after 12 h treatment at 1/10 μM
508,BCL2,0/0 (WB),10.1021/acs.jmedchem.9b00919,,,,% BCL2 degradation in HeLa cells after 12 h treatment at 1/10 μM
508,MCL1,0/0 (WB),10.1021/acs.jmedchem.9b00919,,,,% MCL1 degradation in HeLa cells after 12 h treatment at 1/10 μM
509,ALK,,10.1016/j.ejmech.2020.112190,,,,
510,ALK,,10.1016/j.ejmech.2020.112190,,,,
511,ALK,,10.1016/j.ejmech.2020.112190,,,,
512,ALK,,10.1016/j.ejmech.2020.112190,,,,
513,ALK,,10.1016/j.ejmech.2020.112190,>50,,Degradation of ALK in SR cells after 16 h treatment,
514,ALK,,10.1016/j.ejmech.2020.112190,15,,Degradation of ALK in SR cells after 16 h treatment,
515,ALK,,10.1016/j.ejmech.2020.112190,>50,,Degradation of ALK in SR cells after 16 h treatment,
516,ALK,,10.1016/j.ejmech.2020.112190,,,,
517,ALK,,10.1016/j.ejmech.2020.112190,,,,
518,ALK,,10.1016/j.ejmech.2020.112190,,,,
519,ALK,,10.1016/j.ejmech.2020.112190,,,,
520,ALK,,10.1016/j.ejmech.2020.112190,9.1,,Degradation of ALK in SR cells after 16 h treatment,
521,ALK,,10.1016/j.ejmech.2020.112190,20.9,,Degradation of ALK in SR cells after 16 h treatment,
522,ALK,,10.1016/j.ejmech.2020.112190,7.2,,Degradation of ALK in SR cells after 16 h treatment,
523,ALK,,10.1016/j.ejmech.2020.112190,7,,Degradation of ALK in SR cells after 16 h treatment,
523,ALK G1202R,,10.1016/j.ejmech.2020.112190,<200,,Degradation of G1202R ALK in 293T cells,
524,ALK,,10.1016/j.ejmech.2020.112190,,,,
525,ALK,,10.1016/j.ejmech.2020.112190,,,,
526,ALK,,10.1016/j.ejmech.2020.112190,,,,
527,ALK,,10.1016/j.ejmech.2020.112190,,,,
528,ALK,,10.1016/j.ejmech.2020.112190,11.4,,Degradation of ALK in SR cells after 16 h treatment,
529,ALK,,10.1016/j.ejmech.2020.112190,25.1,,Degradation of ALK in SR cells after 16 h treatment,
530,ALK,,10.1016/j.ejmech.2020.112190,7.5,,Degradation of ALK in SR cells after 16 h treatment,
531,ALK,,10.1016/j.ejmech.2020.112190,,,,
532,ALK,,10.1016/j.ejmech.2020.112190,,,,
533,ALK,,10.1016/j.ejmech.2020.112190,,,,
534,ALK,,10.1016/j.ejmech.2020.112190,,,,
535,ALK,,10.1016/j.ejmech.2020.112190,,,,
536,ALK,,10.1016/j.ejmech.2020.112190,,,,
537,ALK,,10.1016/j.ejmech.2020.112190,,,,
538,ALK,,10.1016/j.ejmech.2020.112190,,,,
539,ALK,,10.1016/j.ejmech.2020.112190,,,,
540,ALK,,10.1016/j.ejmech.2020.112190,,,,
541,ALK,,10.1016/j.ejmech.2020.112190,,,,
542,ALK,,10.1016/j.ejmech.2020.112190,,,,
543,AURKA,,10.1021/acs.jmedchem.7b01655,,,,
543,FAK,,10.1021/acs.jmedchem.7b01655,,,,
543,FER,,10.1021/acs.jmedchem.7b01655,,,,
543,RPS6KA1,,10.1021/acs.jmedchem.7b01655,,,,
543,ALK,,10.1021/acs.jmedchem.7b01655,10/180/50,,Degradation of ALK in H3122/Karpas 299/Kelly cells 16 h treatment,
544,AURKA,,10.1021/acs.jmedchem.7b01655,,,,
544,FAK,,10.1021/acs.jmedchem.7b01655,,,,
544,FER,,10.1021/acs.jmedchem.7b01655,,,,
544,RPS6KA1,,10.1021/acs.jmedchem.7b01655,,,,
544,ALK,,10.1021/acs.jmedchem.7b01655,10/40/50,,Degradation of ALK in H3122/Karpas 299/Kelly cells 16 h treatment,
545,MDM2,,10.1016/j.ejmech.2019.05.046,,,,
546,MDM2,,10.1016/j.ejmech.2019.05.046,,,,
547,MDM2,,10.1016/j.ejmech.2019.05.046,,,,
548,MDM2,,10.1016/j.ejmech.2019.05.046,,,,
549,MDM2,,10.1016/j.ejmech.2019.05.046,,,,
550,MDM2,,10.1016/j.ejmech.2019.05.046,,,,
551,MDM2,,10.1016/j.ejmech.2019.05.046,,,,
552,MDM2,,10.1016/j.ejmech.2019.05.046,,,,
553,MDM2,,10.1016/j.ejmech.2019.05.046,,,,
554,MDM2,,10.1016/j.ejmech.2019.05.046,,,,
555,MDM2,,10.1016/j.ejmech.2019.05.046,,,,
556,MDM2,,10.1016/j.ejmech.2019.05.046,23,90,Degradation of MDM2 in RS4; 11 cells after 24 h treatment,
557,MDM2,,10.1016/j.ejmech.2019.05.046,,,,
558,MDM2,,10.1016/j.ejmech.2019.05.046,,,,
559,EGFR,,10.1016/j.ejmech.2020.112061,45.2,87,Degradation of EGFR in HCC827 cells,
560,EGFR,,10.1016/j.ejmech.2020.112061,,,,
561,EGFR,,10.1016/j.ejmech.2020.112061,,,,
562,EGFR,,10.1016/j.ejmech.2020.112061,,,,
563,EGFR,,10.1016/j.ejmech.2020.112061,,,,
564,EGFR,,10.1016/j.ejmech.2020.112061,,,,
565,EGFR,,10.1016/j.ejmech.2020.112061,,,,
566,EGFR,,10.1016/j.ejmech.2020.112061,,,,
567,EGFR,,10.1016/j.ejmech.2020.112061,34.8,98,Degradation of EGFR in HCC827 cells,
568,EGFR,,10.1016/j.ejmech.2020.112061,,,,
569,EGFR,,10.1016/j.ejmech.2020.112061,,,,
570,EGFR,,10.1016/j.ejmech.2020.112061,,,,
571,EGFR,,10.1016/j.ejmech.2020.112061,,,,
572,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112199,>2000,,Degradation of EGFR L858R/T790M in H1975 cells after 16h treatment,
572,EGFR,,10.1016/j.ejmech.2020.112199,>2000,,Degradation of EGFR in A431 cells after 16 h treatment,
573,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112199,>2000,,Degradation of EGFR L858R/T790M in H1975 cells after 16h treatment,
573,EGFR,,10.1016/j.ejmech.2020.112199,>2000,,Degradation of EGFR in A431 cells after 16 h treatment,
574,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112199,263.8,,Degradation of EGFR L858R/T790M in H1975 cells after 16h treatment,
574,EGFR,,10.1016/j.ejmech.2020.112199,>2000,,Degradation of EGFR in A431 cells after 16 h treatment,
575,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112199,>2000,,Degradation of EGFR L858R/T790M in H1975 cells after 16h treatment,
575,EGFR,,10.1016/j.ejmech.2020.112199,>2000,,Degradation of EGFR in A431 cells after 16 h treatment,
576,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112199,312.9,,Degradation of EGFR L858R/T790M in H1975 cells after 16h treatment,
576,EGFR,,10.1016/j.ejmech.2020.112199,>2000,,Degradation of EGFR in A431 cells after 16 h treatment,
577,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112199,25.3,,Degradation of EGFR L858R/T790M in H1975 cells after 16h treatment,
577,EGFR,,10.1016/j.ejmech.2020.112199,50.3,,Degradation of EGFR in A431 cells after 16 h treatment,
578,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112199,77,,Degradation of EGFR L858R/T790M in H1975 cells after 16h treatment,
578,EGFR,,10.1016/j.ejmech.2020.112199,>2000,,Degradation of EGFR in A431 cells after 16 h treatment,
579,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112199,>2000,,Degradation of EGFR L858R/T790M in H1975 cells after 16h treatment,
579,EGFR,,10.1016/j.ejmech.2020.112199,>2000,,Degradation of EGFR in A431 cells after 16 h treatment,
580,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112199,>2000,,Degradation of EGFR L858R/T790M in H1975 cells after 16h treatment,
580,EGFR,,10.1016/j.ejmech.2020.112199,>2000,,Degradation of EGFR in A431 cells after 16 h treatment,
581,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112199,69,,Degradation of EGFR L858R/T790M in H1975 cells after 16h treatment,
581,EGFR,,10.1016/j.ejmech.2020.112199,>2000,,Degradation of EGFR in A431 cells after 16 h treatment,
582,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112199,235,,Degradation of EGFR L858R/T790M in H1975 cells after 16h treatment,
582,EGFR,,10.1016/j.ejmech.2020.112199,>2000,,Degradation of EGFR in A431 cells after 16 h treatment,
583,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112199,>2000,,Degradation of EGFR L858R/T790M in H1975 cells after 16h treatment,
583,EGFR,,10.1016/j.ejmech.2020.112199,>2000,,Degradation of EGFR in A431 cells after 16 h treatment,
584,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112199,132,,Degradation of EGFR L858R/T790M in H1975 cells after 16h treatment,
584,EGFR,,10.1016/j.ejmech.2020.112199,>2000,,Degradation of EGFR in A431 cells after 16 h treatment,
585,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112199,466,,Degradation of EGFR L858R/T790M in H1975 cells after 16h treatment,
585,EGFR,,10.1016/j.ejmech.2020.112199,>2000,,Degradation of EGFR in A431 cells after 16 h treatment,
586,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112199,5.9,,Degradation of EGFR L858R/T790M in H1975 cells after 16h treatment,
586,EGFR,,10.1016/j.ejmech.2020.112199,>2000,,Degradation of EGFR in A431 cells after 16 h treatment,
587,EGFR,,10.1016/j.ejmech.2020.112199,>2000,,Degradation of EGFR in A431 cells after 16 h treatment,
587,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112199,>2000,,Degradation of EGFR L858R/T790M in H1975 cells after 16h treatment,
588,EGFR L858R,,10.1021/acs.jmedchem.9b01566,,,,
588,EGFR e19d,,10.1021/acs.jmedchem.9b01566,,,,
589,EGFR e19d,,10.1021/acs.jmedchem.9b01566,,,,
589,EGFR L858R,,10.1021/acs.jmedchem.9b01566,,,,
590,EGFR e19d,,10.1021/acs.jmedchem.9b01566,,,,
590,EGFR L858R,,10.1021/acs.jmedchem.9b01566,,,,
591,EGFR e19d,,10.1021/acs.jmedchem.9b01566,,,,
591,EGFR L858R,,10.1021/acs.jmedchem.9b01566,,,,
592,EGFR e19d,,10.1021/acs.jmedchem.9b01566,,,,
592,EGFR L858R,,10.1021/acs.jmedchem.9b01566,,,,
593,EGFR L858R,,10.1021/acs.jmedchem.9b01566,3.3,,Degradation of EGFR L858R in H3255 cells after 16 h treatment,
593,EGFR e19d,,10.1021/acs.jmedchem.9b01566,5,,Degradation of EGFR e19d in HCC-827 cells after 16 h treatment,
594,EGFR L858R,,10.1021/acs.jmedchem.9b01566,,,,
594,EGFR e19d,,10.1021/acs.jmedchem.9b01566,,,,
595,EGFR L858R,,10.1021/acs.jmedchem.9b01566,,,,
595,EGFR e19d,,10.1021/acs.jmedchem.9b01566,,,,
596,EGFR L858R,,10.1021/acs.jmedchem.9b01566,,,,
596,EGFR e19d,,10.1021/acs.jmedchem.9b01566,,,,
597,EGFR e19d,,10.1021/acs.jmedchem.9b01566,11,,Degradation of EGFR e19d in HCC-827 cells after 16 h treatment,
597,EGFR L858R,,10.1021/acs.jmedchem.9b01566,25,,Degradation of EGFR L858R in H3255 cells after 16 h treatment,
598,CDK9,,10.1016/j.ejmech.2019.111952,,N.D.,,
598,CDK2,,10.1016/j.ejmech.2019.111952,,N.D.,,
599,CDK9,,10.1016/j.ejmech.2019.111952,,,,
599,CDK2,,10.1016/j.ejmech.2019.111952,,,,
600,CDK9,,10.1016/j.ejmech.2019.111952,,N.D.,,
600,CDK2,,10.1016/j.ejmech.2019.111952,,N.D.,,
601,CDK9,,10.1016/j.ejmech.2019.111952,,N.D.,,
601,CDK2,,10.1016/j.ejmech.2019.111952,,N.D.,,
602,CDK2,,10.1016/j.ejmech.2019.111952,,N.D.,,
602,CDK9,,10.1016/j.ejmech.2019.111952,,N.D.,,
603,CDK2,,10.1016/j.ejmech.2019.111952,,N.D.,,
603,CDK9,,10.1016/j.ejmech.2019.111952,,N.D.,,
604,CDK2,,10.1016/j.ejmech.2019.111952,,N.D.,,
604,CDK9,,10.1016/j.ejmech.2019.111952,,N.D.,,
605,CDK9,,10.1016/j.ejmech.2019.111952,,N.D.,,
605,CDK2,,10.1016/j.ejmech.2019.111952,,N.D.,,
606,CDK2,,10.1016/j.ejmech.2019.111952,,,,
606,CDK9,,10.1016/j.ejmech.2019.111952,,N.D.,,
607,CDK9,,10.1016/j.ejmech.2019.111952,,N.D.,,
607,CDK2,,10.1016/j.ejmech.2019.111952,,N.D.,,
608,CDK2,,10.1016/j.ejmech.2019.111952,,,,
608,CDK9,,10.1016/j.ejmech.2019.111952,,,,
609,CDK2,,10.1016/j.ejmech.2019.111952,,,,
609,CDK9,,10.1016/j.ejmech.2019.111952,,,,
610,CDK9,,10.1016/j.ejmech.2019.111952,33,,Degradation of CDK9 in PC-3 cells after 24 h treatment,
610,CDK2,,10.1016/j.ejmech.2019.111952,62,,Degradation of CDK2 in PC-3 cells after 24 h treatment,
611,CDK2,,10.1016/j.ejmech.2019.111952,,,,
611,CDK9,,10.1016/j.ejmech.2019.111952,,,,
612,CDK9,,10.1016/j.ejmech.2019.111952,,,,
612,CDK2,,10.1016/j.ejmech.2019.111952,,N.D.,,
613,CDK2,,10.1016/j.ejmech.2019.111952,,N.D.,,
613,CDK9,,10.1016/j.ejmech.2019.111952,,,,
614,CDK2,,10.1016/j.ejmech.2019.111952,,N.D.,,
614,CDK9,,10.1016/j.ejmech.2019.111952,,N.D.,,
615,CDK2,,10.1016/j.ejmech.2019.111952,,N.D.,,
615,CDK9,,10.1016/j.ejmech.2019.111952,,N.D.,,
616,CDK2,,10.1016/j.ejmech.2019.111952,,N.D.,,
616,CDK9,,10.1016/j.ejmech.2019.111952,,,,
617,CDK2,,10.1016/j.ejmech.2019.111952,,N.D.,,
617,CDK9,,10.1016/j.ejmech.2019.111952,,N.D.,,
618,BCL-xL,4 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 100 nM
619,BCL-xL,8 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 100 nM
620,BCL-xL,18 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 100 nM
621,BCL-xL,48 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 100 nM
622,BCL-xL,68 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 100 nM
623,BCL-xL,39 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 100 nM
624,BCL-xL,,10.1016/j.ejmech.2020.112186,93,,Degradation of BCL-xL in MOLT-4 cells after 16 h treatment,
625,BCL-xL,38 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 100 nM
626,BCL-xL,22 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 100 nM
627,BCL-xL,38 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 100 nM
628,BCL-xL,21 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 100 nM
629,BCL-xL,52 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 100 nM
630,BCL-xL,28 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 100 nM
631,BCL-xL,45 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 100 nM
632,BCL-xL,22 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 100 nM
633,BCL-xL,25 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 100 nM
634,BCL-xL,40 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 100 nM
635,BCL-xL,,10.1016/j.ejmech.2020.112186,71,,Degradation of BCL-xL in MOLT-4 cells after 16 h treatment,
636,BCL-xL,54 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 100 nM
637,BCL-xL,51 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 100 nM
638,BCL-xL,38 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 100 nM
639,BCL-xL,76 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 100 nM
640,BCL-xL,67 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 100 nM
641,BCL-xL,67 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 100 nM
642,BCL-xL,56 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
643,BCL-xL,19 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
644,BCL-xL,37 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
645,BCL-xL,0 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
646,BCL-xL,11 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
647,BCL-xL,70 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
648,BCL-xL,80 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
649,BCL-xL,55 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
650,BCL-xL,80 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
651,BCL-xL,79 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
652,BCL-xL,89 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
653,BCL-xL,73 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
654,BCL-xL,24 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
655,BCL-xL,80 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
656,BCL-xL,87 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
657,BCL-xL,,10.1016/j.ejmech.2020.112186,4.5,,Degradation of BCL-xL in MOLT-4 cells after 16 h treatment,
658,BCL-xL,34 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
659,BCL-xL,33 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
660,BCL-xL,72 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
661,BCL-xL,71 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
662,BCL-xL,,10.1016/j.ejmech.2020.112186,6.3,,Degradation of BCL-xL in MOLT-4 cells after 16 h treatment,
663,BCL-xL,76 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
664,BCL-xL,,10.1016/j.ejmech.2020.112186,10.6,,Degradation of BCL-xL in MOLT-4 cells after 16 h treatment,
665,BCL-xL,60 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
666,BCL-xL,53 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
667,BCL-xL,27 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
668,BCL-xL,6 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
669,BCL-xL,89 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
670,BCL-xL,,10.1016/j.ejmech.2020.112186,2.5,,Degradation of BCL-xL in MOLT-4 cells after 16 h treatment,
671,BCL-xL,95 (WB),10.1016/j.ejmech.2020.112186,,,,% BCL-xL degradation in MOLT-4 cells after 16 h treatment at 50 nM
672,CYP1B1,,10.1016/j.ejmech.2019.112028,,,,
673,CYP1B1,,10.1016/j.ejmech.2019.112028,,,,
674,CYP1B1,,10.1016/j.ejmech.2019.112028,,,,
675,CYP1B1,,10.1016/j.ejmech.2019.112028,,,,
676,eIF4E,,10.1016/j.ejmech.2019.01.080,,,,
677,eIF4E,,10.1016/j.ejmech.2019.01.080,,,,
678,eIF4E,,10.1016/j.ejmech.2019.01.080,,,,
679,eIF4E,,10.1016/j.ejmech.2019.01.080,,,,
680,eIF4E,,10.1016/j.ejmech.2019.01.080,,,,
681,eIF4E,,10.1016/j.ejmech.2019.01.080,,,,
682,eIF4E,,10.1016/j.ejmech.2019.01.080,,,,
683,eIF4E,,10.1016/j.ejmech.2019.01.080,,,,
684,eIF4E,,10.1016/j.ejmech.2019.01.080,,,,
685,eIF4E,,10.1016/j.ejmech.2019.01.080,,,,
686,eIF4E,,10.1016/j.ejmech.2019.01.080,,,,
687,eIF4E,,10.1016/j.ejmech.2019.01.080,,,,
688,eIF4E,,10.1016/j.ejmech.2019.01.080,,,,
689,eIF4E,,10.1016/j.ejmech.2019.01.080,,,,
690,eIF4E,,10.1016/j.ejmech.2019.01.080,,,,
691,eIF4E,,10.1016/j.ejmech.2019.01.080,,,,
692,eIF4E,,10.1016/j.ejmech.2019.01.080,,,,
693,eIF4E,,10.1016/j.ejmech.2019.01.080,,,,
694,CRABP-II,,10.1021/ja100691p,,,,
694,CRABP-I,,10.1021/ja100691p,,,,
695,CRABP-II,,10.1021/ja100691p,,,,
695,CRABP-I,,10.1021/ja100691p,,,,
696,CRABP-I,,10.1021/ja100691p,,,,
696,CRABP-II,,10.1021/ja100691p,,,,
697,BCL-xL,,10.1038/s41591-019-0668-z,63/>3000,90.8/26,Degradation of BCL-xL in MOLT-4/platelets cells after 16 h treatment,
697,BCL-xL,,10.1016/j.ejmech.2020.112186,53,,Degradation of BCL-xL in MOLT-4 cells after 16 h treatment,
698,CDK4,,10.1002/anie.201901336,,,,
698,CDK6,,10.1002/anie.201901336,,,,
699,CDK4,,10.1002/anie.201901336,,,,
699,CDK6,,10.1002/anie.201901336,,,,
700,CDK6,,10.1182/blood.2019003604,,,,
700,CDK4,,10.1182/blood.2019003604,,,,
701,CDK6,,10.1016/j.bmcl.2020.127106,0.8,,Degradation of CDK6 in Jurkat cells after 24 h treatment,
701,Wee1,,10.1016/j.cell.2020.10.038,,,,
701,CDK6,,10.1002/anie.201901336,,,,
701,CDK4,,10.1002/anie.201901336,,,,
701,CDK4,,10.1016/j.bmcl.2020.127106,10,,Degradation of CDK4 in Jurkat cells after 24 h treatment,
702,CDK4,,10.1002/anie.201901336,,,,
702,PDK1,,10.1016/j.cell.2020.10.038,,,,
702,Wee1,,10.1016/j.cell.2020.10.038,,,,
702,CDK6,,10.1002/anie.201901336,,,,
703,CDK6,,10.1002/anie.201901336,,,,
703,CDK4,,10.1002/anie.201901336,,,,
704,CDK4,,10.1182/blood.2019003604,,,,
704,CDK6,,10.1002/anie.201901336,,,,
704,CDK6,,10.1182/blood.2019003604,,,,
704,CDK4,,10.1002/anie.201901336,,,,
705,CDK4,,10.1002/anie.201901336,,,,
705,CDK6,,10.1002/anie.201901336,,,,
706,CDK6,,10.1002/anie.201901336,,,,
706,CDK4,,10.1002/anie.201901336,,,,
707,CDK6,,10.1002/anie.201901336,,,,
707,CDK4,,10.1002/anie.201901336,,,,
708,CDK4,,10.1002/anie.201901336,,,,
708,CDK6,,10.1002/anie.201901336,,,,
709,COQ8A,,10.1016/j.cell.2020.10.038,,,,
709,PDK3,,10.1016/j.cell.2020.10.038,,,,
709,PDK2,,10.1016/j.cell.2020.10.038,,,,
709,PDK1,,10.1016/j.cell.2020.10.038,,,,
709,CDK6,,10.1016/j.cell.2020.10.038,,,,
709,BCKDK,,10.1016/j.cell.2020.10.038,,,,
709,CDK4,,10.1002/anie.201901336,,,,
710,CDK4,,10.1002/anie.201901336,,,,
710,CDK6,,10.1002/anie.201901336,,,,
711,CDK6,,10.1002/anie.201901336,,,,
711,CDK9,,10.1002/anie.201901336,,,,
711,CDK4,,10.1002/anie.201901336,,,,
712,PDEdelta,,10.1002/anie.201913904,,,,
713,PDEdelta,,10.1002/anie.201913904,,,,
714,PDEdelta,,10.1002/anie.201913904,48,83.4,Degradation of PDEdelta in Panc Tu-I cells after 24 h treatment,
715,PDEdelta,,10.1002/anie.201913904,,,,
716,BCL-xL,,10.1039/c9cc07217a,,,,
717,BCL-xL,,10.1039/c9cc07217a,50,,Degradation of BCL-xL in MOLT-4 cells after 16 h treatment,
718,BCL-xL,,10.1039/c9cc07217a,,,,
719,CDK4,,10.1039/c9cc00163h,12.9,,Degradation of CDK4 in MDA-MB-231 cells after 18 h treatment,
719,CDK6,,10.1039/c9cc00163h,34.1,,Degradation of CDK6 in MDA-MB-231 cells after 18 h treatment,
720,CDK6,,10.1039/c9cc00163h,,,,
720,CDK4,,10.1039/c9cc00163h,,,,
721,CDK6,,10.1039/c9cc00163h,300,,Degradation of CDK6 in MDA-MB-231 cells after 18 h treatment,
721,CDK4,,10.1039/c9cc00163h,97,,Degradation of CDK4 in MDA-MB-231 cells after 18 h treatment,
722,CDK4,,10.1039/c9cc00163h,,,,
722,CDK6,,10.1039/c9cc00163h,,,,
723,HDAC6,,10.1039/c9cc08509b,3.2,,Degradation of HDAC6 in MM.1S cells after 24 h treatment,
724,HDAC6,,10.1039/c9cc08509b,,,,
725,HDAC6,,10.1039/c9cc08509b,,,,
726,HDAC6,,10.1039/c9cc08509b,,,,
727,HDAC1,,10.1039/d0cc01485k,,,,
727,HDAC3,,10.1039/d0cc01485k,,,,
727,HDAC2,,10.1039/d0cc01485k,,,,
728,HDAC3,,10.1039/d0cc01485k,,,,
728,HDAC1,26/5/23/62 (WB),10.1039/d0cc01485k,,,,% HDAC1 degradation in HCT116 cells after 24 h treatment at 0.01/0.1/1/10 μM
728,HDAC2,10/0/0/40 (WB),10.1039/d0cc01485k,,,,% HDAC2 degradation in HCT116 cells after 24 h treatment at 0.01/0.1/1/10 μM
729,HDAC1,,10.1039/d0cc01485k,,,,
729,HDAC2,,10.1039/d0cc01485k,,,,
729,HDAC3,,10.1039/d0cc01485k,,,,
730,HDAC1,25/36/52/85 (WB),10.1039/d0cc01485k,,,,% HDAC1 degradation in HCT116 cells after 24 h treatment at 0.01/0.1/1/10 μM
730,HDAC2,21/22/60/76 (WB),10.1039/d0cc01485k,,,,% HDAC2 degradation in HCT116 cells after 24 h treatment at 0.01/0.1/1/10 μM
730,HDAC3,0/27/52/63 (WB),10.1039/d0cc01485k,,,,% HDAC3 degradation in HCT116 cells after 24 h treatment at 0.01/0.1/1/10 μM
731,RAR,,10.1016/j.bmc.2011.09.041,,,,
732,ER,,10.1016/j.bmc.2011.09.041,,,,
733,AR,,10.1016/j.bmc.2011.09.041,,,,
734,CRABP-II,,10.1016/j.bmc.2011.03.057,,,,
735,BRD4,,10.1016/j.bmc.2019.115181,,,,
736,BRD4,,10.1016/j.bmc.2019.115181,,,,
737,BRD3,,10.1016/j.bmc.2019.115181,,,,
737,BRD4,,10.1016/j.bmc.2019.115181,,,,
737,BRD2,,10.1016/j.bmc.2019.115181,,,,
738,BRD4,,10.1016/j.bmc.2019.115181,,,,
739,BRD4,,10.1016/j.bmc.2019.115181,,,,
740,CDK4,,10.1016/j.bmcl.2020.127106,25,,Degradation of CDK4 in Jurkat cells after 24 h treatment,
740,CDK6,,10.1016/j.bmcl.2020.127106,4,,Degradation of CDK6 in Jurkat cells after 24 h treatment,
741,CDK6,,10.1016/j.bmcl.2020.127106,20,,Degradation of CDK6 in Jurkat cells after 24 h treatment,
741,CDK6,,10.1039/d0sc00167h,1.7,,Degradation of CDK6 in MM.1S cells after 16 h treatment,
741,CDK4,,10.1039/d0sc00167h,32,,Degradation of CDK4 in MM.1S cells after 16 h treatment,
741,CDK4,,10.1016/j.bmcl.2020.127106,631,,Degradation of CDK4 in Jurkat cells after 24 h treatment,
742,CDK6,,10.1016/j.bmcl.2020.127106,200,,Degradation of CDK6 in Jurkat cells after 24 h treatment,
742,CDK4,,10.1016/j.bmcl.2020.127106,2512,,Degradation of CDK4 in Jurkat cells after 24 h treatment,
743,CDK6,,10.1016/j.bmcl.2020.127106,5,,Degradation of CDK6 in Jurkat cells after 24 h treatment,
743,CDK4,,10.1016/j.bmcl.2020.127106,20,,Degradation of CDK4 in Jurkat cells after 24 h treatment,
744,CDK4,,10.1016/j.bmcl.2020.127106,79,,Degradation of CDK4 in Jurkat cells after 24 h treatment,
744,CDK6,,10.1016/j.bmcl.2020.127106,16,,Degradation of CDK6 in Jurkat cells after 24 h treatment,
745,CDK6,,10.1016/j.bmcl.2020.127106,1585,,Degradation of CDK6 in Jurkat cells after 24 h treatment,
745,CDK4,,10.1016/j.bmcl.2020.127106,5012,,Degradation of CDK4 in Jurkat cells after 24 h treatment,
746,CDK6,,10.1016/j.bmcl.2020.127106,5,,Degradation of CDK6 in Jurkat cells after 24 h treatment,
746,CDK4,,10.1016/j.bmcl.2020.127106,50,,Degradation of CDK4 in Jurkat cells after 24 h treatment,
747,BCR-ABL,0/19 (WB),10.1016/j.bmcl.2016.09.041,,,,% BCR-ABL degradation in K562 cells after 24 h treatment at 30/100 μM
748,BCR-ABL,76/97 (WB),10.1016/j.bmcl.2016.09.041,,,,% BCR-ABL degradation in K562 cells after 24 h treatment at 30/100 μM
749,BCR-ABL,86/92 (WB),10.1016/j.bmcl.2016.09.041,,,,% BCR-ABL degradation in K562 cells after 24 h treatment at 30/100 μM
750,BTK,,10.1016/j.bmcl.2019.126877,374,49,Degradation of BTK in NAMALWA cells after 24 h treatment,
751,BTK,,10.1016/j.bmcl.2019.126877,162,50,Degradation of BTK in NAMALWA cells after 24 h treatment,
752,BTK,,10.1016/j.bmcl.2019.126877,>1000,,Degradation of BTK in NAMALWA cells after 24 h treatment,
753,BTK,,10.1016/j.bmcl.2019.126877,8.3,91,Degradation of BTK in NAMALWA cells after 24 h treatment,
754,BTK,,10.1016/j.bmcl.2019.126877,7.9,95,Degradation of BTK in NAMALWA cells after 24 h treatment,
755,JAK2,,10.1016/j.bmc.2020.115326,,,,
755,JAK1,,10.1016/j.bmc.2020.115326,,,,
756,JAK2,,10.1016/j.bmc.2020.115326,,,,
756,JAK1,,10.1016/j.bmc.2020.115326,,,,
757,JAK1,,10.1016/j.bmc.2020.115326,,N.D.,,
757,JAK2,,10.1016/j.bmc.2020.115326,,N.D.,,
758,JAK2,,10.1016/j.bmc.2020.115326,,,,
758,JAK1,,10.1016/j.bmc.2020.115326,,,,
759,JAK2,,10.1016/j.bmc.2020.115326,,N.D.,,
759,JAK1,,10.1016/j.bmc.2020.115326,,N.D.,,
760,JAK1,,10.1016/j.bmc.2020.115326,,N.D.,,
760,JAK2,,10.1016/j.bmc.2020.115326,,N.D.,,
761,JAK1,,10.1016/j.bmc.2020.115326,,,,
761,JAK2,,10.1016/j.bmc.2020.115326,,,,
762,JAK2,,10.1016/j.bmc.2020.115326,,,,
762,JAK1,,10.1016/j.bmc.2020.115326,,,,
763,JAK2,,10.1016/j.bmc.2020.115326,,,,
763,JAK1,,10.1016/j.bmc.2020.115326,,,,
764,JAK2,,10.1016/j.bmc.2020.115326,,,,
764,JAK1,,10.1016/j.bmc.2020.115326,,,,
765,JAK1,,10.1016/j.bmc.2020.115326,,N.D.,,
765,JAK2,,10.1016/j.bmc.2020.115326,,N.D.,,
766,JAK1,,10.1016/j.bmc.2020.115326,,,,
766,JAK2,,10.1016/j.bmc.2020.115326,,,,
767,JAK1,,10.1016/j.bmc.2020.115326,,,,
767,JAK2,,10.1016/j.bmc.2020.115326,,,,
768,JAK1,,10.1016/j.bmc.2020.115326,,,,
768,JAK2,,10.1016/j.bmc.2020.115326,,,,
769,JAK1,,10.1016/j.bmc.2020.115326,,,,
769,JAK2,,10.1016/j.bmc.2020.115326,,,,
770,JAK2,,10.1016/j.bmc.2020.115326,,,,
770,JAK1,,10.1016/j.bmc.2020.115326,,,,
771,JAK1,,10.1016/j.bmc.2020.115326,,,,
771,JAK2,,10.1016/j.bmc.2020.115326,,,,
772,JAK1,,10.1016/j.bmc.2020.115326,,N.D.,,
772,JAK2,,10.1016/j.bmc.2020.115326,,N.D.,,
773,JAK1,,10.1016/j.bmc.2020.115326,,,,
773,JAK2,,10.1016/j.bmc.2020.115326,,,,
774,JAK1,,10.1016/j.bmc.2020.115326,,N.D.,,
774,JAK2,,10.1016/j.bmc.2020.115326,,N.D.,,
775,JAK2,,10.1016/j.bmc.2020.115326,,N.D.,,
775,JAK1,,10.1016/j.bmc.2020.115326,,N.D.,,
776,JAK2,,10.1016/j.bmc.2020.115326,,,,
776,JAK1,,10.1016/j.bmc.2020.115326,,,,
777,JAK2,,10.1016/j.bmc.2020.115326,,,,
777,JAK1,,10.1016/j.bmc.2020.115326,,,,
778,JAK2,,10.1016/j.bmc.2020.115326,,,,
778,JAK1,,10.1016/j.bmc.2020.115326,,,,
779,BRD4,,10.1016/j.bmc.2019.115228,,,,
780,BRD4,,10.1016/j.bmc.2019.115228,,,,
781,BRD4,,10.1016/j.bmc.2019.115228,,,,
782,BRD4,,10.1016/j.bmc.2019.115228,,,,
783,BRD4,,10.1016/j.bmc.2019.115228,,,,
784,BRD4,,10.1016/j.bmc.2019.115228,,,,
785,BRD4,,10.1016/j.bmc.2019.115228,,,,
786,BRD4,,10.1016/j.bmc.2019.115228,,,,
787,BRD4,,10.1016/j.bmc.2019.115228,,,,
788,BRD4,,10.1016/j.bmc.2019.115228,,,,
789,BRD4,,10.1016/j.bmc.2019.115228,,,,
790,BRD4,,10.1016/j.bmc.2019.115228,,,,
791,BRD4,,10.1016/j.bmc.2019.115228,,,,
792,BRD4,,10.1016/j.bmc.2019.115228,,,,
793,BRD4,,10.1016/j.bmc.2019.115228,,,,
794,BRD4,,10.1016/j.bmc.2019.115228,,,,
795,BRD4,,10.1016/j.bmc.2019.115228,,,,
796,SMARCA2,,10.1038/s41589-019-0294-6,300,65,Degradation of SMARCA2 in MV-4-11 cells after 18 h treatment,
796,PBRM1,,10.1038/s41589-019-0294-6,,,,
796,SMARCA4,,10.1038/s41589-019-0294-6,250,70,Degradation of SMARCA4 in MV-4-11 cells after 18 h treatment,
797,SMARCA2,,10.1038/s41589-019-0294-6,,,,
797,PBRM1,,10.1038/s41589-019-0294-6,,,,
797,SMARCA4,,10.1038/s41589-019-0294-6,,,,
798,PBRM1,,10.1038/s41589-019-0294-6,32/15.6,,Degradation of PBRM1 in MV-4-11/NCI-H1568 cells after 18 h treatment,
798,SMARCA2,,10.1038/s41589-019-0294-6,6/3.3,,Degradation of SMARCA2 in MV-4-11/NCI-H1568 cells after 18 h treatment,
798,SMARCA4,,10.1038/s41589-019-0294-6,11,,Degradation of SMARCA2 in MV-4-11 cells after 18 h treatment,
799,CDK9,,10.1038/nchembio.2538,,,,
800,CDK9,,10.1038/nchembio.2538,,,,
801,CDK9,,10.1038/nchembio.2538,,,,
802,CDK9,,10.1038/nchembio.2538,,,,
803,CDK9,,10.1038/nchembio.2538,,,,
804,FKBP12,,10.1038/s41589-019-0279-5,,,,
805,FKBP12,,10.1038/s41589-019-0279-5,,,,
806,FKBP12,,10.1038/s41589-019-0279-5,,,,
807,FKBP12,,10.1038/s41589-019-0279-5,,,,
808,BRD4,,10.1038/s41589-019-0279-5,,,,
809,IRAK4,,10.1021/acsmedchemlett.9b00219,,N.D.,,
810,IRAK4,,10.1021/acsmedchemlett.9b00219,,50,,
811,IRAK4,,10.1021/acsmedchemlett.9b00219,,N.D.,,
812,IRAK4,,10.1021/acsmedchemlett.9b00219,,N.D.,,
813,IRAK4,,10.1021/acsmedchemlett.9b00219,,N.D.,,
814,IRAK4,,10.1021/acsmedchemlett.9b00219,,N.D.,,
815,IRAK4,,10.1021/acsmedchemlett.9b00219,259,,Degradation of IRAK4 in PBMC cells after 24 h treatment,
816,IRAK4,,10.1021/acsmedchemlett.9b00219,151/36,,Degradation of IRAK4 in PBMC cells/dermal fibroblast after 24/24 h treatment,
817,PLK1,,10.1016/j.bbrc.2019.11.007,10-20,,Degradation of PLK1 in MV4-11 cells after 24 h treatment,
817,BRD4,,10.1016/j.bbrc.2019.11.007,<5,,Degradation of BRD4 in MV4-11 cells after 24 h treatment,
818,BRD4,,10.1016/j.bbrc.2019.11.007,,,,
818,PLK1,,10.1016/j.bbrc.2019.11.007,,,,
819,CRABP-I,21/21/37/39/55 (WB),10.1021/acschembio.9b00704,,,,% CRABP-I degradation in IMR-32 cells after 24 h treatment at 0.1/0.3/1/3/10 μM
819,CRABP-II,7/42/48/54/55 (WB),10.1021/acschembio.9b00704,,,,% CRABP-II degradation in IMR-32 cells after 24 h treatment at 0.1/0.3/1/3/10 μM
820,CRABP-II,0/4/32 (WB),10.1021/acschembio.9b00704,,,,% CRABP-II degradation in IMR-32 cells after 24 h treatment at 0.1/1/10 μM
820,CRABP-I,3/20/35 (WB),10.1021/acschembio.9b00704,,,,% CRABP-I degradation in IMR-32 cells after 24 h treatment at 0.1/1/10 μM
821,CRABP-I,37/45/51/46/43 (WB),10.1021/acschembio.9b00704,,,,% CRABP-I degradation in IMR-32 cells after 8 h treatment at 0.3/1/3/10/30 μM
821,CRABP-II,29/48/52/47/35 (WB),10.1021/acschembio.9b00704,,,,% CRABP-II degradation in IMR-32 cells after 8 h treatment at 0.3/1/3/10/30 μM
822,BRD4,20/6/0/45 (WB),10.1021/acschembio.9b00704,,,,% BRD4 degradation in MCF7 cells after 24 h treatment at 0.01/0.1/1/10 μM
822,BRD2,6/1/4/34 (WB),10.1021/acschembio.9b00704,,,,% BRD2 degradation in MCF7 cells after 24 h treatment at 0.01/0.1/1/10 μM
822,BRD3,16/45/63/66 (WB),10.1021/acschembio.9b00704,,,,% BRD3 degradation in MCF7 cells after 24 h treatment at 0.01/0.1/1/10 μM
823,ER,,10.1021/acschembio.0c00140,,,,
824,ER,,10.1021/acschembio.0c00140,,,,
825,ER,,10.1021/acschembio.0c00140,7.7/10.3,95/98,Degradation of ERalpha in MCF-7/T47D cells after 6 h treatment,
826,ER,,10.1021/acschembio.0c00140,,,,
827,ER,,10.1021/acschembio.0c00140,,,,
828,ER,,10.1021/acschembio.0c00140,,,,
829,ER,,10.1021/acschembio.0c00140,,,,
830,ER,,10.1021/acschembio.0c00140,,,,
831,ER,,10.1021/acschembio.0c00140,,,,
832,ER,,10.1021/acschembio.0c00140,,,,
833,ER,,10.1021/acschembio.0c00140,,,,
834,ER,,10.1021/acschembio.0c00140,,,,
835,ER,,10.1021/acschembio.0c00140,,,,
836,ER,,10.1021/acschembio.0c00140,,,,
837,ER,,10.1021/acschembio.0c00140,,,,
838,ER,,10.1021/acschembio.0c00140,,,,
839,ER,,10.1021/acschembio.0c00140,,,,
840,ER,,10.1021/acschembio.0c00140,,,,
841,ER,,10.1021/acschembio.0c00140,,,,
842,ER,,10.1021/acschembio.0c00140,,,,
843,ER,,10.1021/acschembio.0c00140,,,,
844,ER,,10.1021/acschembio.0c00140,,,,
845,ER,,10.1021/acschembio.0c00140,,,,
846,ER,,10.1021/acschembio.0c00140,,,,
847,ER,,10.1021/acschembio.0c00140,,,,
848,ER,,10.1021/acschembio.0c00140,,,,
849,ER,,10.1021/acschembio.0c00140,,,,
850,ER,,10.1021/acschembio.0c00140,,,,
851,ER,,10.1021/acschembio.0c00140,,,,
852,ER,,10.1021/acschembio.0c00140,,,,
853,ER,,10.1021/acschembio.0c00140,,,,
854,ER,,10.1021/acschembio.0c00140,,,,
855,ER,,10.1021/acschembio.0c00140,,,,
856,ER,,10.1021/acschembio.0c00140,,,,
857,ER,,10.1021/acschembio.0c00140,,,,
858,ER,,10.1021/acschembio.0c00140,,,,
859,ER,,10.1021/acschembio.0c00140,,,,
860,ER,,10.1021/acschembio.0c00140,5.2,75,Degradation of ERalpha in MCF-7 cells after 6 h treatment,
861,ER,,10.1021/acschembio.0c00140,,,,
862,ER,,10.1021/acschembio.0c00140,,,,
863,ER,,10.1021/acschembio.0c00140,,,,
864,ER,,10.1021/acschembio.0c00140,,,,
865,ER,,10.1021/acschembio.0c00140,,,,
866,ER,,10.1021/acschembio.0c00140,,,,
867,ER,,10.1021/acschembio.0c00140,,,,
868,ER,,10.1021/acschembio.0c00140,,,,
869,ER,,10.1021/acschembio.0c00140,,,,
870,ER,,10.1021/acschembio.0c00140,,,,
871,ER,,10.1021/acschembio.0c00140,,,,
872,ER,,10.1021/acschembio.0c00140,,,,
873,ER,,10.1021/acschembio.0c00140,,,,
874,ER,,10.1021/acschembio.0c00140,,,,
875,ER,,10.1021/acschembio.0c00140,,,,
876,ER,,10.1021/acschembio.0c00140,,,,
877,ER,,10.1021/acschembio.0c00140,,,,
878,ER,,10.1021/acschembio.0c00140,,,,
879,ER,,10.1021/acschembio.0c00140,,,,
880,ER,,10.1021/acschembio.0c00140,,,,
881,ER,,10.1021/acschembio.0c00140,,,,
882,ER,,10.1021/acschembio.0c00140,,,,
883,ER,,10.1021/acschembio.0c00140,,,,
884,ER,,10.1021/acschembio.0c00140,,,,
885,ER,,10.1021/acschembio.0c00140,,,,
886,ER,,10.1021/acschembio.0c00140,,,,
887,ER,,10.1021/acschembio.0c00140,,,,
888,ER,,10.1021/acschembio.0c00140,,,,
889,ER,,10.1021/acschembio.0c00140,,,,
890,ER,,10.1021/acschembio.0c00140,,,,
891,ER,,10.1021/acschembio.0c00140,,,,
892,ER,,10.1021/acschembio.0c00140,,,,
893,ER,,10.1021/acschembio.0c00140,,,,
894,ER,,10.1021/acschembio.0c00140,,,,
895,ER,,10.1021/acschembio.0c00140,,,,
896,ER,,10.1021/acschembio.0c00140,,,,
897,ER,,10.1021/acschembio.0c00140,,,,
898,ER,,10.1021/acschembio.0c00140,,,,
899,ER,,10.1021/acschembio.0c00140,,,,
900,ER,,10.1021/acschembio.0c00140,,,,
901,ER,,10.1021/acschembio.0c00140,,,,
902,ER,,10.1021/acschembio.0c00140,,,,
903,ER,,10.1021/acschembio.0c00140,,,,
904,ER,,10.1021/acschembio.0c00140,,,,
905,ER,,10.1021/acschembio.0c00140,,,,
906,ER,,10.1021/acschembio.0c00140,,,,
907,ER,,10.1021/acschembio.0c00140,,,,
908,ER,,10.1021/acschembio.0c00140,,,,
909,ER,,10.1021/acschembio.0c00140,,,,
910,ER,,10.1021/acschembio.0c00140,,,,
911,ER,,10.1021/acschembio.0c00140,,,,
912,ER,,10.1021/acschembio.0c00140,,,,
913,ER,,10.1021/acschembio.0c00140,,,,
914,ER,,10.1021/acschembio.0c00140,,,,
915,ER,,10.1021/acschembio.0c00140,,,,
916,ER,,10.1021/acschembio.0c00140,,,,
917,ER,,10.1021/acschembio.0c00140,,,,
918,ER,,10.1021/acschembio.0c00140,,,,
919,ER,34/85/94 (WB),10.1021/acschembio.0c00140,,,,% ER degradation in MCF-7 cells after 6 h treatment at 10/100/1000 nM
920,ER,,10.1021/acschembio.0c00140,1.1,98,Degradation of ERalpha in MCF-7 cells after 6h treatment,
921,ER,28/85/94 (WB),10.1021/acschembio.0c00140,,,,% ER degradation in MCF-7 cells after 6 h treatment at 10/100/1000 nM
922,SGK3,23/59/77 (WB),10.1021/acschembio.9b00505,,,,% SGK3 degradation in HEK293 cells after 48 h treatment at 0.1/1/10 μM
923,SGK3,0/3/16 (WB),10.1021/acschembio.9b00505,,,,% SGK3 degradation in HEK293 cells after 48 h treatment at 0.1/1/10 μM
924,SGK3,19/26/30 (WB),10.1021/acschembio.9b00505,,,,% SGK3 degradation in HEK293 cells after 48 h treatment at 0.1/1/10 μM
925,SGK3,0/11/16 (WB),10.1021/acschembio.9b00505,,,,% SGK3 degradation in HEK293 cells after 48 h treatment at 0.1/1/10 μM
926,SGK3,18/8/27/64 (WB),10.1021/acschembio.9b00505,,,,% SGK3 degradation in HEK293 cells after 48 h treatment at 0.01/0.1/1/10 μM
927,SGK3,10/29/56/80 (WB),10.1021/acschembio.9b00505,,,,% SGK3 degradation in HEK293 cells after 48 h treatment at 0.01/0.1/1/10 μM
928,SGK3,20/5/63/71 (WB),10.1021/acschembio.9b00505,,,,% SGK3 degradation in HEK293 cells after 48 h treatment at 0.01/0.1/1/10 μM
929,SGK3,0/66/76/81 (WB),10.1021/acschembio.9b00505,,,,% SGK3 degradation in HEK293 cells after 48 h treatment at 0.01/0.1/1/10 μM
930,SGK3,29/60/89/88 (WB),10.1021/acschembio.9b00505,,,,% SGK3 degradation in HEK293 cells after 48 h treatment at 0.01/0.1/1/10 μM
931,SGK3,24/46/89/91 (WB),10.1021/acschembio.9b00505,,,,% SGK3 degradation in HEK293 cells after 48 h treatment at 0.01/0.1/1/10 μM
932,SGK3,3/59/68/71 (WB),10.1021/acschembio.9b00505,,,,% SGK3 degradation in HEK293 cells after 48 h treatment at 0.01/0.1/1/10 μM
933,SGK3,16/21/68/71 (WB),10.1021/acschembio.9b00505,,,,% SGK3 degradation in HEK293 cells after 48 h treatment at 0.01/0.1/1/10 μM
934,EED,,10.1016/j.chembiol.2019.11.004,,,,
934,EZH2,,10.1016/j.chembiol.2019.11.004,,,,
934,SUZ12,,10.1016/j.chembiol.2019.11.004,,,,
935,EED,,10.1016/j.chembiol.2019.11.004,,,,
935,SUZ12,,10.1016/j.chembiol.2019.11.004,,,,
935,EZH2,,10.1016/j.chembiol.2019.11.004,,,,
936,EED,,10.1016/j.chembiol.2019.11.006,,,,
936,SUZ12,,10.1016/j.chembiol.2019.11.006,,,,
936,EZH2,,10.1016/j.chembiol.2019.11.006,,,,
937,SUZ12,,10.1016/j.chembiol.2019.11.006,(n/a)/590,22/82,Degradation of SUZ12 in HeLa/DB cells after 24 h treatment,
937,EED,,10.1016/j.chembiol.2019.11.006,790/610,92/94,Degradation of EED in HeLa/DB cells after 24 h treatment,
937,EZH2,,10.1016/j.chembiol.2019.11.006,300/670,75/96,Degradation of EZH2 in HeLa/DB cells after 24 h treatment,
938,SUZ12,,10.1016/j.chembiol.2019.11.006,,,,
938,EZH2,,10.1016/j.chembiol.2019.11.006,,,,
938,EED,,10.1016/j.chembiol.2019.11.006,,,,
939,EED,,10.1016/j.chembiol.2019.11.006,,,,
939,SUZ12,,10.1016/j.chembiol.2019.11.006,,,,
939,EZH2,,10.1016/j.chembiol.2019.11.006,,,,
940,SUZ12,,10.1016/j.chembiol.2019.11.006,,,,
940,EED,,10.1016/j.chembiol.2019.11.006,,,,
940,EZH2,,10.1016/j.chembiol.2019.11.006,,,,
941,SUZ12,,10.1016/j.chembiol.2019.11.006,,,,
941,EZH2,,10.1016/j.chembiol.2019.11.006,,,,
941,EED,,10.1016/j.chembiol.2019.11.006,,,,
942,AKT1,,10.1016/j.chembiol.2019.11.014,,,,
942,MAPK6,,10.1016/j.cell.2020.10.038,,,,
942,STK17A,,10.1016/j.cell.2020.10.038,,,,
942,AKT2,,10.1016/j.chembiol.2019.11.014,,,,
942,AKT3,,10.1016/j.chembiol.2019.11.014,,,,
942,CDK4,,10.1016/j.cell.2020.10.038,,,,
943,KRAS G12C,,10.1016/j.chembiol.2019.12.006,,N.D.,,
944,KRAS G12C,,10.1016/j.chembiol.2019.12.006,,N.D.,,
945,KRAS G12C,,10.1016/j.chembiol.2019.12.006,,N.D.,,
946,KRAS G12C,,10.1016/j.chembiol.2019.12.006,,N.D.,,
947,KRAS G12C,,10.1016/j.chembiol.2019.12.006,,N.D.,,
948,KRAS G12C,,10.1016/j.chembiol.2019.12.006,,N.D.,,
949,KRAS G12C,,10.1016/j.chembiol.2019.12.006,,N.D.,,
950,KRAS G12C,,10.1016/j.chembiol.2019.12.006,,N.D.,,
951,KRAS G12C,,10.1016/j.chembiol.2019.12.006,,N.D.,,
952,KRAS G12C,,10.1016/j.chembiol.2019.12.006,,N.D.,,
953,KRAS G12C,,10.1016/j.chembiol.2019.12.006,,N.D.,,
954,KRAS G12C,,10.1016/j.chembiol.2019.12.006,,N.D.,,
955,KRAS G12C,,10.1016/j.chembiol.2019.12.006,,N.D.,,
956,KRAS G12C,,10.1016/j.chembiol.2019.12.006,,N.D.,,
957,KRAS G12C,,10.1016/j.chembiol.2019.12.006,,N.D.,,
958,KRAS G12C,,10.1016/j.chembiol.2019.12.006,,N.D.,,
959,BCR-ABL,,10.1158/0008-5472.CAN-19-1236,2000,85,Degradation of BCR-ABL in K562 cells after 18 h treatment,
960,BCR-ABL,,10.1158/0008-5472.CAN-19-1236,,,,
961,BCR-ABL,,10.1158/0008-5472.CAN-19-1236,340,95,Degradation of BCR-ABL in K562 cells after 18 h treatment,
962,CRBN,9 (WB),10.1016/j.bmc.2019.02.048,,,,% CRBN degradation in HeLa cells after 4 h treatment at 1 μM
963,CRBN,9 (WB),10.1016/j.bmc.2019.02.048,,,,% CRBN degradation in HeLa cells after 4 h treatment at 1 μM
964,CRBN,6 (WB),10.1016/j.bmc.2019.02.048,,,,% CRBN degradation in HeLa cells after 4 h treatment at 1 μM
965,CRBN,14 (WB),10.1016/j.bmc.2019.02.048,,,,% CRBN degradation in HeLa cells after 4 h treatment at 1 μM
966,CRBN,9 (WB),10.1016/j.bmc.2019.02.048,,,,% CRBN degradation in HeLa cells after 4 h treatment at 1 μM
967,CRBN,35 (WB),10.1016/j.bmc.2019.02.048,,,,% CRBN degradation in HeLa cells after 4 h treatment at 1 μM
968,CRBN,,10.1016/j.bmc.2019.02.048,200/230,75/98,Degradation of CRBN in HeLa/HEK293 cells,
969,CRBN,29 (WB),10.1016/j.bmc.2019.02.048,,,,% CRBN degradation in HeLa cells after 4 h treatment at 1 μM
970,CRBN,54 (WB),10.1016/j.bmc.2019.02.048,,,,% CRBN degradation in HeLa cells after 4 h treatment at 1 μM
971,CRBN,5 (WB),10.1016/j.bmc.2019.02.048,,,,% CRBN degradation in HeLa cells after 4 h treatment at 1 μM
972,CRBN,29 (WB),10.1016/j.bmc.2019.02.048,,,,% CRBN degradation in HeLa cells after 4 h treatment at 1 μM
973,CRBN,32 (WB),10.1016/j.bmc.2019.02.048,,,,% CRBN degradation in HeLa cells after 4 h treatment at 1 μM
974,CRBN,19 (WB),10.1016/j.bmc.2019.02.048,,,,% CRBN degradation in HeLa cells after 4 h treatment at 1 μM
975,FKBP12,,10.1038/s41421-018-0079-1,0.27,,Degradation of FKBP12 in Jurkat cells after 12 h treatment,
976,BTK,,10.1038/s41421-018-0079-1,,,,
977,RIPK2,,10.1038/s42003-020-0868-6,0.4,,Degradation of RIPK2 in THP-1 cells after 18 h treatment,
978,RIPK2,,10.1038/s42003-020-0868-6,2.5,,Degradation of RIPK2 in THP-1 cells after 18 h treatment,
979,RIPK2,,10.1038/s42003-020-0868-6,12.6,69.2,Degradation of RIPK2 in hPBMC cells after 24 h treatment,
979,RIPK2,,10.1021/acs.jmedchem.1c01118,,,,
980,RIPK2,,10.1021/acs.jmedchem.1c01118,0.79,,Degradation of RIPK2 in THP1 cells after 18 h treatment,
980,RIPK2,,10.1038/s42003-020-0868-6,0.4,94.3,Degradation of RIPK2 in hPBMC cells after 24 h treatment,
981,Cdc20,,10.1016/j.ebiom.2019.10.013,,,,
982,Cdc20,,10.1016/j.ebiom.2019.10.013,,,,
983,Cdc20,,10.1016/j.ebiom.2019.10.013,,,,
984,Cdc20,,10.1016/j.ebiom.2019.10.013,1600/1600,,Degradation of Cdc20 in MCF7/MDA-MB-231 cells after 10 h treatment,
985,Cdc20,,10.1016/j.ebiom.2019.10.013,,,,
986,Cdc20,,10.1016/j.ebiom.2019.10.013,,,,
987,Cdc20,,10.1016/j.ebiom.2019.10.013,,,,
988,Cdc20,,10.1016/j.ebiom.2019.10.013,,,,
989,Cdc20,,10.1016/j.ebiom.2019.10.013,,,,
990,Cdc20,,10.1016/j.ebiom.2019.10.013,,,,
991,Cdc20,,10.1016/j.ebiom.2019.10.013,,,,
992,Cdc20,,10.1016/j.ebiom.2019.10.013,,,,
993,Cdc20,,10.1016/j.ebiom.2019.10.013,,,,
994,Cdc20,,10.1016/j.ebiom.2019.10.013,,,,
995,Cdc20,,10.1016/j.ebiom.2019.10.013,,,,
996,VHL,88/96 (WB),10.1038/s41467-017-00954-1,,,,% pVHL30 degradation in HeLa cells after 24 h treatment at 1/10 μM
997,VHL,36/38/87/100/100 (WB),10.1038/s41467-017-00954-1,,,,% pVHL30 degradation in HeLa cells after 24 h treatment at 0.001/0.01/0.1/1/10 μM
998,VHL,,10.1038/s41467-017-00954-1,10-100,,Degradation of pVHL30 in HeLa cells after 24 h treatment,
999,VHL,0/7 (WB),10.1038/s41467-017-00954-1,,,,% pVHL30/pVHL19 degradation in HeLa cells after 10 h treatment at 1 μM
1000,VHL,0/3 (WB),10.1038/s41467-017-00954-1,,,,% pVHL30/pVHL19 degradation in HeLa cells after 10 h treatment at 1 μM
1001,VHL,0/11 (WB),10.1038/s41467-017-00954-1,,,,% pVHL30/pVHL19 degradation in HeLa cells after 10 h treatment at 1 μM
1002,VHL,0/0 (WB),10.1038/s41467-017-00954-1,,,,% pVHL30/pVHL19 degradation in HeLa cells after 10 h treatment at 1 μM
1003,TRKC,,10.1021/acs.molpharmaceut.9b00673,100-1000,,Degradation of TrkC in Hs578t cells after 24 h treatment,
1004,TRKC,,10.1021/acs.molpharmaceut.9b00673,,,,
1005,TRKC,,10.1021/acs.molpharmaceut.9b00673,,,,
1006,CRABP-II,,10.1016/j.bmcl.2012.04.134,,,,
1007,HDAC6,,10.1007/s13238-018-0602-z,,,,
1008,HDAC6,,10.1007/s13238-018-0602-z,3.8,,Degradation of HADC6 in MM.1S cells after 24 h treatment,
1009,HDAC6,,10.1007/s13238-018-0602-z,,,,
1010,HDAC6,,10.1007/s13238-018-0602-z,,,,
1011,CRBN,,10.1038/s41598-019-56177-5,44.5,97.1,Degradation of CRBN in HEK293T cells after 24h treatment,
1012,CRBN,,10.1038/s41598-019-56177-5,20.4,99.6,Degradation of CRBN in HEK293T cells after 24h treatment,
1013,CRBN,,10.1038/s41598-019-56177-5,100.6,96.9,Degradation of CRBN in HEK293T cells after 24h treatment,
1014,CRBN,,10.1038/s41598-019-56177-5,28.8,98.4,Degradation of CRBN in HEK293T cells after 24h treatment,
1015,CRBN,,10.1038/s41598-019-56177-5,367.7,82,Degradation of CRBN in HEK293T cells after 24h treatment,
1016,CRBN,,10.1038/s41598-019-56177-5,2546.1,77.9,Degradation of CRBN in HEK293T cells after 24h treatment,
1017,BCR-ABL,,10.1111/cas.13284,100000,,Degradation of BCR-ABL in K562 cells after 6 h treatment,
1018,BCR-ABL,,10.1111/cas.13284,20000,,Degradation of BCR-ABL in K562 cells after 6 h treatment,
1019,BCR-ABL,,10.1111/cas.13284,10000,,Degradation of BCR-ABL in K562 cells after 6 h treatment,
1020,BCR-ABL,,10.1111/cas.13284,>100000,,Degradation of BCR-ABL in K562 cells after 6 h treatment,
1021,BCR-ABL,,10.1111/cas.13284,>100000,,Degradation of BCR-ABL in K562 cells after 6 h treatment,
1022,BCR-ABL,,10.1111/cas.13284,5000,,Degradation of BCR-ABL in K562 cells after 6 h treatment,
1023,BCR-ABL,,10.1111/cas.13284,2000,,Degradation of BCR-ABL in K562 cells after 6 h treatment,
1024,BCR-ABL,,10.1111/cas.13284,300,,Degradation of BCR-ABL in K562 cells after 6 h treatment,
1025,BCR-ABL,,10.1111/cas.13284,10000,,Degradation of BCR-ABL in K562 cells after 6 h treatment,
1026,BCR-ABL,,10.1111/cas.13284,5000,,Degradation of BCR-ABL in K562 cells after 6 h treatment,
1027,BCR-ABL,,10.1111/cas.13284,300,,Degradation of BCR-ABL in K562 cells after 6 h treatment,
1028,BCR-ABL,,10.1111/cas.13284,10,,Degradation of BCR-ABL in K562 cells after 6 h treatment,
1029,BCR-ABL,19/39 (WB),10.1111/cas.13284,,,,% BCR-ABL degradation in K562 cells after 6 h treatment at 10/30 nM
1030,BCR-ABL,11/46 (WB),10.1111/cas.13284,,,,% BCR-ABL degradation in K562 cells after 6 h treatment at 10/30 nM
1031,BCR-ABL,39/65 (WB),10.1111/cas.13284,,,,% BCR-ABL degradation in K562 cells after 6 h treatment at 10/30 nM
1032,BCR-ABL,36/18/19/95 (WB),10.1021/acsmedchemlett.7b00247,,,,% BCR-ABL degradation in K562 cells after 6 h treatment at 10/100/1000/5000 nM
1033,BCR-ABL,28/46/62/72/48 (WB),10.1021/acsmedchemlett.7b00247,,,,% BCR-ABL degradation in K562 cells after 6 h treatment at 10/30/100/300/1000 nM
1034,ER,,10.1016/j.bmcl.2011.11.086,,,,
1035,ER,,10.1016/j.bmcl.2011.11.086,,,,
1036,ER,,10.1016/j.bmcl.2011.11.086,,,,
1037,ER,0/5/13/32 (WB),10.1074/jbc.M116.768853,,,,% ERalpha degradation in MCF-7 cells after 24 h treatment at 3/10/30/100 nM
1038,ER,,10.1074/jbc.M116.768853,3,,Degradation of ERalpha in MCF-7 cells after 6 h treatment,
1038,ER,,10.1074/jbc.RA117.001091,<3/83,,Degradation of ERalpha in MCF-7 cells after 4/48 h treatment,
1039,ER,18/40/53/54 (WB),10.1074/jbc.M116.768853,,,,% ERalpha degradation in MCF-7 cells after 24 h treatment at 3/10/30/100 nM
1040,BRD4,,10.1248/cpb.c18-00567,,,,
1040,BRD4,67/74/30 (WB),10.1074/jbc.M116.768853,,,,% BRD4 degradation in LNCaP cells after 6 h treatment at 10/100/1000 nM
1041,PDE4,62/61/67/43 (WB),10.1074/jbc.M116.768853,,,,% PDE4 degradation in HT1080 cells after 6 h treatment at 1/10/100/1000 nM
1042,ER,0/0/0/13 (WB),10.1074/jbc.M116.768853,,,,% ERalpha degradation in MCF-7 cells after 6 h treatment at 0.01/0.1/1/10 μM
1043,ER,0 (WB),10.1074/jbc.M116.768853,,,,% ERalpha degradation in MCF-7 cells after 6 h treatment at 0.03/0.1/0.3/1 μM
1044,ER,56/65/67/64 (WB),10.1074/jbc.M116.768853,,,,% ERalpha degradation in MCF-7 cells after 6 h treatment at 0.03/0.1/0.3/1 μM
1045,ER,36/61/53/57 (WB),10.1074/jbc.M116.768853,,,,% ERalpha degradation in MCF-7 cells after 6 h treatment at 0.01/0.1/1/10 μM
1046,ER,49/52/53/44 (WB),10.1074/jbc.M116.768853,,,,% ERalpha degradation in MCF-7 cells after 6 h treatment at 0.03/0.1/0.3/1 μM
1047,ER,0/16/36/18 (WB),10.1074/jbc.M116.768853,,,,% ERalpha degradation in MCF-7 cells after 6 h treatment at 0.01/0.1/1/10 μM
1048,ER,8/43/5/42 (WB),10.1074/jbc.M116.768853,,,,% ERalpha degradation in MCF-7 cells after 6 h treatment at 0.01/0.1/1/10 μM
1049,ER,0 (WB),10.1074/jbc.M116.768853,,,,% ERalpha degradation in MCF-7 cells after 6 h treatment at 0.01/0.1/1/10 μM
1050,BRD4,56/67/34/18 (WB),10.1248/cpb.c18-00567,,,,% BRD4 degradation in LNCaP cells after 6 h treatment at 0.01/0.1/1/10 μM
1051,ER,,10.1074/jbc.RA117.001091,>100,,Degradation of ERalpha in MCF-7 cells after 4h treatment,
1052,ER,,10.1074/jbc.RA117.001091,<3/<3,,Degradation of ERalpha in MCF-7 cells after 4/48h treatment,
1053,ER,,10.1074/jbc.RA117.001091,<3/7.7,,Degradation of ERalpha in MCF-7 cells after 4/48h treatment,
1054,ER,,10.1074/jbc.RA117.001091,<3/13.3,,Degradation of ERalpha in MCF-7 cells after 4/48h treatment,
1055,ER,,10.1074/jbc.RA117.001091,>100,,Degradation of ERalpha in MCF-7 cells after 4h treatment,
1056,ER,,10.1074/jbc.RA117.001091,4/15.7,,Degradation of ERalpha in MCF-7 cells after 4/48h treatment,
1057,ER,,10.1074/jbc.RA117.001091,>100,,Degradation of ERalpha in MCF-7 cells after 4h treatment,
1058,ER,,10.1074/jbc.RA117.001091,<3/3.7,,Degradation of ERalpha in MCF-7 cells after 4/48h treatment,
1059,ER,,10.1074/jbc.RA117.001091,36.9,,Degradation of ERalpha in MCF-7 cells after 4h treatment,
1060,ER,,10.1074/jbc.RA117.001091,33.8,,Degradation of ERalpha in MCF-7 cells after 4h treatment,
1061,ER,,10.1074/jbc.RA117.001091,>100,,Degradation of ERalpha in MCF-7 cells after 4h treatment,
1062,ER,,10.1074/jbc.RA117.001091,>100,,Degradation of ERalpha in MCF-7 cells after 4h treatment,
1063,AR,,10.1021/acs.jmedchem.7b00168,21600,,Degradation of AR in 22Rv1 cells after 6 h treatment,
1064,AR,,10.1021/acs.jmedchem.7b00168,>30000,,Degradation of AR in 22Rv1 cells after 6 h treatment,
1065,AR,,10.1021/acs.jmedchem.7b00168,11700,,Degradation of AR in 22Rv1 cells after 6 h treatment,
1066,AR,,10.1021/acs.jmedchem.7b00168,20500,,Degradation of AR in 22Rv1 cells after 6 h treatment,
1067,AR,,10.1021/acs.jmedchem.7b00168,>30000,,Degradation of AR in 22Rv1 cells after 6 h treatment,
1068,AR,0/40/52 (WB),10.1021/acs.jmedchem.7b00168,,,,% AR degradation in 22Rv1 cells after 6 h treatment at 3/10/20 μM
1069,AR,57/62/52 (WB),10.1021/acs.jmedchem.7b00168,,,,% AR degradation in 22Rv1 cells after 6 h treatment at 3/10/30 μM
1070,AR,24/74 (WB),10.1021/acs.jmedchem.7b00168,,,,% AR degradation in 22Rv1 cells after 6 h treatment at 1/3 μM
1071,AR,8/73 (WB),10.1021/acs.jmedchem.7b00168,,,,% AR degradation in 22Rv1 cells after 6 h treatment at 1/3 μM
1072,AR,32/74 (WB),10.1021/acs.jmedchem.7b00168,,,,% AR degradation in 22Rv1 cells after 6 h treatment at 1/3 μM
1073,AR,10/94 (WB),10.1021/acs.jmedchem.7b00168,,,,% AR degradation in 22Rv1 cells after 6 h treatment at 1/3 μM
1074,AR,21/86 (WB),10.1021/acs.jmedchem.7b00168,,,,% AR degradation in 22Rv1 cells after 6 h treatment at 1/3 μM
1075,AR,23/89 (WB),10.1021/acs.jmedchem.7b00168,,,,% AR degradation in 22Rv1 cells after 6 h treatment at 1/3 μM
1076,AR,0/18 (WB),10.1021/acs.jmedchem.7b00168,,,,% AR degradation in 22Rv1 cells after 6 h treatment at 1/3 μM
1077,AR,,10.1021/acs.jmedchem.7b00168,,N.D.,,
1078,AR,,10.1021/acs.jmedchem.7b00168,,N.D.,,
1079,AR,,10.1021/acs.jmedchem.7b00168,,N.D.,,
1080,BRAF V600E,88 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1081,BRAF V600E,91 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1081,BRAF V600E,,10.1038/s41589-020-0609-7,100,65,Degradation of BRAF V600E in A375 cells after 24 h treatment,
1082,BRAF V600E,84 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1083,BRAF V600E,49 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1084,BRAF V600E,36 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1085,BRAF V600E,21 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1086,BRAF V600E,14 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1087,BRAF V600E,33 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1088,BRAF V600E,36 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1089,BRAF V600E,53 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1090,BRAF V600E,56 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1091,BRAF V600E,6 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1092,BRAF V600E,7 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1093,BRAF V600E,11 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1094,BRAF V600E,12 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1095,BRAF V600E,11 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1096,BRAF V600E,16 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1097,BRAF V600E,59 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1098,BRAF V600E,,10.1038/s41589-020-0609-7,15,82,Degradation of BRAF V600E in A375 cells after 24 h treatment,
1098,BRAF V600E,93 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1099,BRAF V600E,95 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1099,BRAF V600E,,10.1038/s41589-020-0609-7,70,82,Degradation of BRAF V600E in A375 cells after 24 h treatment,
1100,BRAF V600E,36 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1101,BRAF V600E,16 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1102,BRAF V600E,41 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1103,BRAF V600E,33 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1104,BRAF V600E,17 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1105,BRAF V600E,24 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1106,BRAF V600E,36 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1106,BRAF V600E,,10.1038/s41589-020-0609-7,100,40,Degradation of BRAF V600E in A375 cells after 24 h treatment,
1107,BRAF V600E,54 (WB),10.1021/acs.jmedchem.9b02083,,,,% BRAF V600 degradation in A375 cells after 16 h treatment at 500 nM
1108,HMGCR,,10.1021/acs.jmedchem.0c00339,>3000,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1109,HMGCR,,10.1021/acs.jmedchem.0c00339,>3000,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1110,HMGCR,,10.1021/acs.jmedchem.0c00339,3000,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1111,HMGCR,,10.1021/acs.jmedchem.0c00339,>3000,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1112,HMGCR,,10.1021/acs.jmedchem.0c00339,>3000,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1113,HMGCR,,10.1021/acs.jmedchem.0c00339,>3000,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1114,HMGCR,,10.1021/acs.jmedchem.0c00339,>3000,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1115,HMGCR,,10.1021/acs.jmedchem.0c00339,>3000,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1116,HMGCR,,10.1021/acs.jmedchem.0c00339,1800,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1117,HMGCR,,10.1021/acs.jmedchem.0c00339,100,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1118,HMGCR,,10.1021/acs.jmedchem.0c00339,400,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1119,HMGCR,,10.1021/acs.jmedchem.0c00339,500,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1120,HMGCR,,10.1021/acs.jmedchem.0c00339,200,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1121,HMGCR,,10.1021/acs.jmedchem.0c00339,>3000,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1122,HMGCR,,10.1021/acs.jmedchem.0c00339,600,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1123,HMGCR,,10.1021/acs.jmedchem.0c00339,,,,
1124,HMGCR,,10.1021/acs.jmedchem.0c00339,400,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1125,HMGCR,,10.1021/acs.jmedchem.0c00339,200,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1126,HMGCR,,10.1021/acs.jmedchem.0c00339,300,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1127,HMGCR,,10.1021/acs.jmedchem.0c00339,400,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1128,HMGCR,,10.1021/acs.jmedchem.0c00339,300,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1129,HMGCR,,10.1021/acs.jmedchem.0c00339,500,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1130,HMGCR,,10.1021/acs.jmedchem.0c00339,>3000,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1131,HMGCR,,10.1021/acs.jmedchem.0c00339,>3000,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1132,HMGCR,,10.1021/acs.jmedchem.0c00339,>3000,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1133,HMGCR,,10.1021/acs.jmedchem.0c00339,300,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1134,HMGCR,,10.1021/acs.jmedchem.0c00339,>3000,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1135,HMGCR,,10.1021/acs.jmedchem.0c00339,>3000,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1136,HMGCR,,10.1021/acs.jmedchem.0c00339,>3000,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1137,HMGCR,,10.1021/acs.jmedchem.0c00339,>3000,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1138,HMGCR,,10.1021/acs.jmedchem.0c00339,>3000,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1139,HMGCR,,10.1021/acs.jmedchem.0c00339,300,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1140,HMGCR,,10.1021/acs.jmedchem.0c00339,200,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1141,HMGCR,,10.1021/acs.jmedchem.0c00339,700,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1142,HMGCR,,10.1021/acs.jmedchem.0c00339,>3000,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1143,HMGCR,,10.1021/acs.jmedchem.0c00339,>3000,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1144,HMGCR,,10.1021/acs.jmedchem.0c00339,>3000,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1145,HMGCR,,10.1021/acs.jmedchem.0c00339,2300,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1146,HMGCR,,10.1021/acs.jmedchem.0c00339,500,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1147,HMGCR,,10.1021/acs.jmedchem.0c00339,600,,Degradation of HMGCR in SRD15 cells after 16 h treatment,
1148,MEK2,,10.1021/acs.jmedchem.9b01528,,,,
1148,MEK1,,10.1021/acs.jmedchem.9b01528,,,,
1149,MEK1,,10.1021/acs.jmedchem.9b01528,,,,
1149,MEK2,,10.1021/acs.jmedchem.9b01528,,,,
1150,MEK1,,10.1021/acs.jmedchem.9b01528,,,,
1150,MEK2,,10.1021/acs.jmedchem.9b01528,,,,
1151,MEK2,,10.1021/acs.jmedchem.9b01528,,,,
1151,MEK1,,10.1021/acs.jmedchem.9b01528,,,,
1152,MEK1,,10.1021/acs.jmedchem.9b01528,,,,
1152,MEK2,,10.1021/acs.jmedchem.9b01528,,,,
1153,MEK1,,10.1021/acs.jmedchem.9b01528,31/31/18,,Degradation of MEK1 in HT-29/SK-MEL-28/COLO 205 cells after 24 h treatment,
1153,MEK2,,10.1021/acs.jmedchem.9b01528,17/9.3/11,,Degradation of MEK2 in HT-29/SK-MEL-28/COLO 205 cells after 24 h treatment,
1154,HDAC6,62.1/81.3,10.1021/acs.jmedchem.9b00516,3.41,88.01,Degradation of HDAC6 in MM1S cells after 6 h treatment,% HDAC6 degradation in MM1S cells after 6 h treatment at 10/100 nM
1155,HDAC6,67.3/84.1,10.1021/acs.jmedchem.9b00516,,,,% HDAC6 degradation in MM1S cells after 6 h treatment at 10/100 nM
1156,HDAC6,64.3/85,10.1021/acs.jmedchem.9b00516,,,,% HDAC6 degradation in MM1S cells after 6 h treatment at 10/100 nM
1157,HDAC6,,10.1021/acsmedchemlett.0c00046,2.2/18,86/45,Degradation of HDAC6 in MM1S/Mouse 4935 cells after 4/6 h treatment,
1157,HDAC6,74.9/82.7,10.1021/acs.jmedchem.9b00516,1.64,86.26,Degradation of HDAC6 in MM1S cells after 6 h treatment,% HDAC6 degradation in MM1S cells after 6 h treatment at 10/100 nM
1158,HDAC6,66.1/77.8,10.1021/acs.jmedchem.9b00516,,,,% HDAC6 degradation in MM1S cells after 6 h treatment at 10/100 nM
1159,HDAC6,49.3/81.8,10.1021/acs.jmedchem.9b00516,,,,% HDAC6 degradation in MM1S cells after 6 h treatment at 10/100 nM
1160,HDAC6,64.8/84.2,10.1021/acs.jmedchem.9b00516,,,,% HDAC6 degradation in MM1S cells after 6 h treatment at 10/100 nM
1161,HDAC6,71.7/79.2,10.1021/acs.jmedchem.9b00516,,,,% HDAC6 degradation in MM1S cells after 6 h treatment at 10/100 nM
1162,HDAC6,70.6/83.1,10.1021/acs.jmedchem.9b00516,2.54,86.3,Degradation of HDAC6 in MM1S cells after 6 h treatment,% HDAC6 degradation in MM1S cells after 6 h treatment at 10/100 nM
1163,HDAC6,45.6/77.3,10.1021/acs.jmedchem.9b00516,,,,% HDAC6 degradation in MM1S cells after 6 h treatment at 10/100 nM
1164,HDAC6,50.9/75.7,10.1021/acs.jmedchem.9b00516,,,,% HDAC6 degradation in MM1S cells after 6 h treatment at 10/100 nM
1165,HDAC6,57.1/81.4,10.1021/acs.jmedchem.9b00516,,,,% HDAC6 degradation in MM1S cells after 6 h treatment at 10/100 nM
1166,HDAC6,60.3/81.2,10.1021/acs.jmedchem.9b00516,,,,% HDAC6 degradation in MM1S cells after 6 h treatment at 10/100 nM
1167,HDAC6,63.3/80.9,10.1021/acs.jmedchem.9b00516,,,,% HDAC6 degradation in MM1S cells after 6 h treatment at 10/100 nM
1168,HDAC6,69.9/84.7,10.1021/acs.jmedchem.9b00516,,,,% HDAC6 degradation in MM1S cells after 6 h treatment at 10/100 nM
1169,HDAC6,70.8/83.5,10.1021/acs.jmedchem.9b00516,,,,% HDAC6 degradation in MM1S cells after 6 h treatment at 10/100 nM
1170,HDAC6,47.2/80.4,10.1021/acs.jmedchem.9b00516,,,,% HDAC6 degradation in MM1S cells after 6 h treatment at 10/100 nM
1171,HDAC6,60.9/81.9,10.1021/acs.jmedchem.9b00516,,,,% HDAC6 degradation in MM1S cells after 6 h treatment at 10/100 nM
1172,HDAC6,,10.1021/acsmedchemlett.0c00046,,,,
1173,HDAC6,,10.1021/acsmedchemlett.0c00046,,,,
1174,HDAC6,,10.1021/acsmedchemlett.0c00046,,,,
1175,HDAC6,,10.1021/acsmedchemlett.0c00046,,,,
1176,HDAC6,,10.1021/acsmedchemlett.0c00046,,,,
1177,HDAC6,,10.1021/acsmedchemlett.0c00046,,,,
1178,HDAC6,,10.1021/acsmedchemlett.0c00046,,,,
1179,HDAC6,,10.1021/acsmedchemlett.0c00046,,,,
1180,HDAC6,,10.1021/acsmedchemlett.0c00046,,,,
1181,HDAC6,,10.1021/acsmedchemlett.0c00046,7.1/4.3,90/57,Degradation of HDAC6 in MM1S/Mouse 4935 cells after 4/6 h treatment,
1182,HDAC6,,10.1021/acsmedchemlett.0c00046,11,89,Degradation of HDAC6 in MM1S cells after 4 h treatment,
1183,HDAC6,,10.1021/acsmedchemlett.0c00046,,,,
1184,HDAC6,,10.1021/acsmedchemlett.0c00046,,,,
1185,HDAC6,,10.1021/acsmedchemlett.0c00046,,,,
1186,HDAC6,,10.1021/acsmedchemlett.0c00046,,,,
1187,BRD9,,10.1002/anie.201611281,,,,
1188,BRD9,,10.1002/anie.201611281,,,,
1189,BRD9,,10.1002/anie.201611281,,,,
1190,BRD9,,10.1002/anie.201611281,,,,
1191,BRD9,,10.1002/anie.201611281,,,,
1192,BRD9,,10.1002/anie.201611281,,,,
1193,BRD9,,10.1002/anie.201611281,,,,
1194,BRD9,,10.1002/anie.201611281,,,,
1195,BRD9,,10.1002/anie.201611281,,,,
1196,BRD7,,10.1002/anie.201611281,,,,
1196,BRD4,,10.1002/anie.201611281,,,,
1196,BRD9,,10.1002/anie.201611281,,,,
1197,BRD9,,10.1002/anie.201611281,,,,
1198,BRD9,,10.1002/anie.201611281,,,,
1199,BRD9,,10.1002/anie.201611281,,,,
1200,BRD9,,10.1002/anie.201611281,,,,
1201,BRD9,,10.1021/acs.jmedchem.8b01413,,,,
1201,BRD9,,10.1002/anie.201611281,,,,
1202,Htt,,10.1002/anie.201706529,,,,
1203,Htt,,10.1002/anie.201706529,,,,
1204,CDK2,,10.1002/anie.202004087,,,,
1205,CDK2,,10.1002/anie.202004087,,,,
1206,CDK2,,10.1002/anie.202004087,,,,
1207,CDK2,,10.1002/anie.202004087,,,,
1208,CDK2,,10.1002/anie.202004087,,,,
1209,CDK2,,10.1002/anie.202004087,,,,
1210,CDK6,,10.1002/anie.202004087,,,,
1210,CDK4,,10.1002/anie.202004087,,,,
1210,CDK12,,10.1016/j.cell.2020.10.038,,,,
1210,CDK2,,10.1002/anie.202004087,,,,
1210,RPS6KA1,,10.1016/j.cell.2020.10.038,,,,
1210,CDK17,,10.1016/j.cell.2020.10.038,,,,
1210,CDK16,,10.1016/j.cell.2020.10.038,,,,
1210,CDK5,,10.1002/anie.202004087,,,,
1210,CDK9,,10.1016/j.cell.2020.10.038,,,,
1210,CDK7,,10.1016/j.cell.2020.10.038,,,,
1210,MAPK9,,10.1016/j.cell.2020.10.038,,,,
1210,MAPK8,,10.1016/j.cell.2020.10.038,,,,
1210,CDK1,,10.1016/j.cell.2020.10.038,,,,
1210,AURKA,,10.1016/j.cell.2020.10.038,,,,
1210,MAPK10,,10.1016/j.cell.2020.10.038,,,,
1211,CDK16,,10.1016/j.cell.2020.10.038,,,,
1211,PRKAA1,,10.1016/j.cell.2020.10.038,,,,
1211,PTK2B,,10.1016/j.cell.2020.10.038,,,,
1211,STK38,,10.1016/j.cell.2020.10.038,,,,
1211,RPS6KA1,,10.1016/j.cell.2020.10.038,,,,
1211,MAP3K11,,10.1016/j.cell.2020.10.038,,,,
1211,AAK1,,10.1016/j.cell.2020.10.038,,,,
1211,AURKB,,10.1016/j.cell.2020.10.038,,,,
1211,STK33,,10.1016/j.cell.2020.10.038,,,,
1211,CDK12,,10.1016/j.cell.2020.10.038,,,,
1211,IRAK3,,10.1016/j.cell.2020.10.038,,,,
1211,TTK,,10.1016/j.cell.2020.10.038,,,,
1211,MAPK8,,10.1016/j.cell.2020.10.038,,,,
1211,MAPK9,,10.1016/j.cell.2020.10.038,,,,
1211,CLK1,,10.1016/j.cell.2020.10.038,,,,
1211,GSK3A,,10.1016/j.cell.2020.10.038,,,,
1211,GSK-3beta,,10.1016/j.cell.2020.10.038,,,,
1211,CDK7,,10.1016/j.cell.2020.10.038,,,,
1211,CDK9,,10.1016/j.cell.2020.10.038,,,,
1211,RPS6KA3,,10.1016/j.cell.2020.10.038,,,,
1211,PRKAA2,,10.1016/j.cell.2020.10.038,,,,
1211,CDK5,,10.1016/j.cell.2020.10.038,,,,
1211,CDK17,,10.1016/j.cell.2020.10.038,,,,
1211,CDK2,,10.1002/anie.202004087,,,,
1211,AURKA,,10.1016/j.cell.2020.10.038,,,,
1211,NUAK1,,10.1016/j.cell.2020.10.038,,,,
1211,CDK1,,10.1016/j.cell.2020.10.038,,,,
1211,FER,,10.1016/j.cell.2020.10.038,,,,
1212,STK33,,10.1016/j.cell.2020.10.038,,,,
1212,AURKB,,10.1016/j.cell.2020.10.038,,,,
1212,RPS6KA1,,10.1016/j.cell.2020.10.038,,,,
1212,FAK,,10.1016/j.cell.2020.10.038,,,,
1212,RPS6KA3,,10.1016/j.cell.2020.10.038,,,,
1212,MAPK9,,10.1016/j.cell.2020.10.038,,,,
1212,MAPK8,,10.1016/j.cell.2020.10.038,,,,
1212,TTK,,10.1016/j.cell.2020.10.038,,,,
1212,CDK1,,10.1016/j.cell.2020.10.038,,,,
1212,AURKA,,10.1016/j.cell.2020.10.038,,,,
1212,CDK5,,10.1002/anie.202004087,,,,
1212,CDK2,,10.1002/anie.202004087,,,,
1213,GSK-3beta,,10.1016/j.cell.2020.10.038,,,,
1213,NEK4,,10.1016/j.cell.2020.10.038,,,,
1213,PRKAA2,,10.1016/j.cell.2020.10.038,,,,
1213,CDK5,,10.1016/j.cell.2020.10.038,,,,
1213,CDK16,,10.1016/j.cell.2020.10.038,,,,
1213,CDK17,,10.1016/j.cell.2020.10.038,,,,
1213,FAK,,10.1016/j.cell.2020.10.038,,,,
1213,PRKAA1,,10.1016/j.cell.2020.10.038,,,,
1213,PTK2B,,10.1016/j.cell.2020.10.038,,,,
1213,STK38,,10.1016/j.cell.2020.10.038,,,,
1213,RPS6KA1,,10.1016/j.cell.2020.10.038,,,,
1213,MAP3K11,,10.1016/j.cell.2020.10.038,,,,
1213,AAK1,,10.1016/j.cell.2020.10.038,,,,
1213,NEK9,,10.1016/j.cell.2020.10.038,,,,
1213,STK35,,10.1016/j.cell.2020.10.038,,,,
1213,AURKB,,10.1016/j.cell.2020.10.038,,,,
1213,NEK1,,10.1016/j.cell.2020.10.038,,,,
1213,STK33,,10.1016/j.cell.2020.10.038,,,,
1213,CDK12,,10.1016/j.cell.2020.10.038,,,,
1213,TBK1,,10.1016/j.cell.2020.10.038,,,,
1213,IRAK3,,10.1016/j.cell.2020.10.038,,,,
1213,RPS6KA3,,10.1016/j.cell.2020.10.038,,,,
1213,CDK9,,10.1016/j.cell.2020.10.038,,,,
1213,CDK7,,10.1016/j.cell.2020.10.038,,,,
1213,NEK3,,10.1016/j.cell.2020.10.038,,,,
1213,GSK3A,,10.1016/j.cell.2020.10.038,,,,
1213,CLK1,,10.1016/j.cell.2020.10.038,,,,
1213,MAPK9,,10.1016/j.cell.2020.10.038,,,,
1213,MAPK8,,10.1016/j.cell.2020.10.038,,,,
1213,TEC,,10.1016/j.cell.2020.10.038,,,,
1213,TTK,,10.1016/j.cell.2020.10.038,,,,
1213,Wee1,,10.1016/j.cell.2020.10.038,,,,
1213,FER,,10.1016/j.cell.2020.10.038,,,,
1213,CDK1,,10.1016/j.cell.2020.10.038,,,,
1213,RPS6KA4,,10.1016/j.cell.2020.10.038,,,,
1213,NUAK1,,10.1016/j.cell.2020.10.038,,,,
1213,AURKA,,10.1016/j.cell.2020.10.038,,,,
1213,CDK2,,10.1002/anie.202004087,,,,
1214,BRD4,,10.1016/j.bioorg.2020.103817,,,,
1215,BRD4,,10.1016/j.bioorg.2020.103817,,,,
1216,BRD4,,10.1016/j.bioorg.2020.103817,,,,
1217,BRD4,,10.1016/j.bioorg.2020.103817,,,,
1218,EGFR,,10.1016/j.bmcl.2020.127167,,,,
1219,EGFR,,10.1016/j.bmcl.2020.127167,,,,
1220,EGFR,,10.1016/j.bmcl.2020.127167,161,68,Degradation of EGFR in PC9 cells after 6 h treatment,
1221,BRD3,,10.1158/0008-5472.CAN-16-2622,,,,
1221,BRD4,,10.1158/0008-5472.CAN-16-2622,,,,
1221,BRD2,,10.1158/0008-5472.CAN-16-2622,,,,
1222,BTK,,10.1182/blood-2018-07-862953,,,,
1222,BTK C481S,,10.1182/blood-2018-07-862953,,,,
1223,BTK C481S,,10.1182/blood-2018-07-862953,,,,
1223,BTK,,10.1182/blood-2018-07-862953,,,,
1224,BTK,,10.1182/blood-2018-07-862953,,,,
1225,SLC9A1,,10.1016/j.chembiol.2020.04.003,,,,
1226,SLC9A4,,10.1016/j.chembiol.2020.04.003,,,,
1226,SLC9A7,,10.1016/j.chembiol.2020.04.003,,,,
1226,SLC9B1,,10.1016/j.chembiol.2020.04.003,,,,
1226,SLC9A1,,10.1016/j.chembiol.2020.04.003,,,,
1226,SLC9A2,,10.1016/j.chembiol.2020.04.003,,,,
1227,SLC9A1,,10.1016/j.chembiol.2020.04.003,,,,
1228,SLC9A1,,10.1016/j.chembiol.2020.04.003,,,,
1229,SLC9A1,,10.1016/j.chembiol.2020.04.003,,,,
1230,MAP4K2,,10.1016/j.cell.2020.10.038,,,,
1230,FLT3,,10.1016/j.chembiol.2017.10.005,,,,
1230,GAK,,10.1016/j.cell.2020.10.038,,,,
1230,LCK,,10.1016/j.cell.2020.10.038,,,,
1230,Src,,10.1016/j.cell.2020.10.038,,,,
1230,FER,,10.1016/j.cell.2020.10.038,,,,
1230,BLK,,10.1016/j.cell.2020.10.038,,,,
1230,IRAK1,,10.1016/j.cell.2020.10.038,,,,
1230,CDK5,,10.1016/j.cell.2020.10.038,,,,
1230,RIPK1,,10.1016/j.cell.2020.10.038,,,,
1230,p38alpha,,10.1016/j.cell.2020.10.038,,,,
1231,FLT3,,10.1016/j.chembiol.2017.10.005,,N.D.,,
1232,FLT3,,10.1016/j.chembiol.2017.10.005,,,,
1233,FLT3,,10.1016/j.chembiol.2017.10.005,,N.D.,,
1234,FLT3,,10.1016/j.chembiol.2017.10.005,,N.D.,,
1235,FLT3,,10.1016/j.chembiol.2017.10.005,,N.D.,,
1236,FLT3,,10.1016/j.chembiol.2017.10.005,,N.D.,,
1237,FLT3,,10.1016/j.chembiol.2017.10.005,,N.D.,,
1238,FLT3,,10.1016/j.chembiol.2017.10.005,,N.D.,,
1239,BTK,,10.1016/j.chembiol.2017.10.005,,,,
1240,BTK,,10.1016/j.chembiol.2017.10.005,,,,
1241,Wee1,,10.1016/j.chembiol.2019.10.013,,,,
1242,Wee1,,10.1016/j.chembiol.2019.10.013,,,,
1243,Wee1,,10.1016/j.chembiol.2019.10.013,,,,
1244,Wee1,,10.1016/j.chembiol.2019.10.013,,,,
1244,TBCK,,10.1016/j.cell.2020.10.038,,,,
1244,COQ8A,,10.1016/j.cell.2020.10.038,,,,
1244,PDK2,,10.1016/j.cell.2020.10.038,,,,
1244,PDK1,,10.1016/j.cell.2020.10.038,,,,
1244,PRKCI,,10.1016/j.cell.2020.10.038,,,,
1244,PAK4,,10.1016/j.cell.2020.10.038,,,,
1244,PDK3,,10.1016/j.cell.2020.10.038,,,,
1244,MKNK2,,10.1016/j.cell.2020.10.038,,,,
1245,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1246,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1247,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1248,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1249,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1250,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1251,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1252,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1253,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1254,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1255,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1256,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1257,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1258,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1259,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1260,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1261,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1262,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1263,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1264,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1265,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1266,PD-L1,21/35 (WB),10.1016/j.ejmech.2020.112377,,,,% PD-L1 degradation in MDA-MB-231 cells after 24 h treatment at 1/10 μM
1267,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1268,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1269,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1270,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1271,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1272,PD-L1,,10.1016/j.ejmech.2020.112377,,,,
1273,BCL-xL,69 (WB),10.1016/j.ejmech.2020.112397,,,,% BCL-xL degradation in MyLa 1929 cells after 16 h treatment at 500 nM
1274,BCL-xL,41 (WB),10.1016/j.ejmech.2020.112397,,,,% BCL-xL degradation in MyLa 1929 cells after 16 h treatment at 500 nM
1275,BCL-xL,40 (WB),10.1016/j.ejmech.2020.112397,,,,% BCL-xL degradation in MyLa 1929 cells after 16 h treatment at 500 nM
1276,BCL-xL,71 (WB),10.1016/j.ejmech.2020.112397,,,,% BCL-xL degradation in MyLa 1929 cells after 16 h treatment at 500 nM
1277,BCL-xL,45 (WB),10.1016/j.ejmech.2020.112397,,,,% BCL-xL degradation in MyLa 1929 cells after 16 h treatment at 500 nM
1278,BCL-xL,20 (WB),10.1016/j.ejmech.2020.112397,,,,% BCL-xL degradation in MyLa 1929 cells after 16 h treatment at 500 nM
1279,BCL-xL,0 (WB),10.1016/j.ejmech.2020.112397,,,,% BCL-xL degradation in MyLa 1929 cells after 16 h treatment at 500 nM
1280,BCL-xL,0 (WB),10.1016/j.ejmech.2020.112397,,,,% BCL-xL degradation in MyLa 1929 cells after 16 h treatment at 500 nM
1281,BCL-xL,84 (WB),10.1016/j.ejmech.2020.112397,,,,% BCL-xL degradation in MyLa 1929 cells after 16 h treatment at 500 nM
1282,BCL-xL,89 (WB),10.1016/j.ejmech.2020.112397,,,,% BCL-xL degradation in MyLa 1929 cells after 16 h treatment at 500 nM
1283,BCL-xL,85 (WB),10.1016/j.ejmech.2020.112397,,,,% BCL-xL degradation in MyLa 1929 cells after 16 h treatment at 500 nM
1284,BCL-xL,90 (WB),10.1016/j.ejmech.2020.112397,,,,% BCL-xL degradation in MyLa 1929 cells after 16 h treatment at 500 nM
1285,BCL-xL,85 (WB),10.1016/j.ejmech.2020.112397,,,,% BCL-xL degradation in MyLa 1929 cells after 16 h treatment at 500 nM
1286,BCL-xL,73 (WB),10.1016/j.ejmech.2020.112397,,,,% BCL-xL degradation in MyLa 1929 cells after 16 h treatment at 500 nM
1287,BCL-xL,27 (WB),10.1016/j.ejmech.2020.112397,,,,% BCL-xL degradation in MyLa 1929 cells after 16 h treatment at 500 nM
1288,BCL-xL,0 (WB),10.1016/j.ejmech.2020.112397,,,,% BCL-xL degradation in MyLa 1929 cells after 16 h treatment at 500 nM
1289,PARP1,,10.1038/s41589-019-0379-2,,N.D.,,
1290,PARP1,,10.1038/s41589-019-0379-2,,N.D.,,
1291,PARP1,,10.1038/s41589-019-0379-2,,,,
1292,PARP1,,10.1038/s41589-019-0379-2,,,,
1293,PARP1,,10.1038/s41589-019-0379-2,,N.D.,,
1294,PARP1,,10.1038/s41589-019-0379-2,,N.D.,,
1295,PARP1,,10.1038/s41589-019-0379-2,,N.D.,,
1296,PARP1,,10.1038/s41589-019-0379-2,,,,
1297,PARP1,,10.1038/s41589-019-0379-2,,,,
1298,PARP1,,10.1038/s41589-019-0379-2,,,,
1299,PARP3,,10.1038/s41589-019-0379-2,,,,
1299,PARP1,,10.1038/s41589-019-0379-2,35.7,90,Degradation of PARP1 in Primary Cardiomyocytes after 24 h treatment,
1300,PARP3,,10.1038/s41589-019-0379-2,,,,
1300,PARP1,,10.1038/s41589-019-0379-2,81.8,92,Degradation of PARP1 in Primary Cardiomyocytes after 24 h treatment,
1301,PARP1,,10.1038/s41589-019-0379-2,,,,
1302,PARP1,,10.1038/s41589-019-0379-2,,,,
1303,PARP1,,10.1038/s41589-019-0379-2,,,,
1304,PARP2,,10.1038/s41589-019-0379-2,,,,
1304,PARP1,,10.1038/s41589-019-0379-2,,N.D.,,
1305,PARP1,,10.1038/s41589-019-0379-2,,N.D.,,
1305,PARP2,,10.1038/s41589-019-0379-2,,,,
1306,PARP2,,10.1038/s41589-019-0379-2,62.8,,Degradation of PARP2 in HeLa cells after 24 h treatment,
1306,PARP1,,10.1038/s41589-019-0379-2,,,,
1307,PARP2,,10.1038/s41589-019-0379-2,,,,
1307,PARP1,,10.1038/s41589-019-0379-2,,,,
1308,PARP1,,10.1038/s41589-019-0379-2,,N.D.,,
1309,PARP1,,10.1038/s41589-019-0379-2,,N.D.,,
1310,PARP1,,10.1038/s41589-019-0379-2,,N.D.,,
1311,PARP1,,10.1038/s41589-019-0379-2,,N.D.,,
1312,PARP1,,10.1038/s41589-019-0379-2,,N.D.,,
1313,PARP1,,10.1038/s41589-019-0379-2,,N.D.,,
1314,PARP1,,10.1038/s41589-019-0379-2,,N.D.,,
1315,PARP1,,10.1038/s41589-019-0379-2,,,,
1316,TRIM24,20/29/2/39/72 (WB),10.1038/s41589-018-0010-y,,,,% TRIM24 degradation in 293FT cells after 24 h treatment at 0.25/0.5/1/2.5/5 μM
1317,TRIM24,16/38/40 (WB),10.1038/s41589-018-0010-y,,,,% TRIM24 degradation in 293FT cells after 24 h treatment at 0.5/5/10 μM
1318,FKBP12 F36V,,10.1038/s41589-018-0021-8,,,,
1319,FKBP12 F36V,,10.1038/s41589-018-0021-8,,,,
1320,FKBP12 F36V,,10.1038/s41589-018-0021-8,,,,
1321,FKBP12 F36V,,10.1038/s41589-018-0021-8,,,,
1322,HDAC6,,10.1016/j.chembiol.2020.04.008,,,,
1323,HDAC6,,10.1016/j.chembiol.2020.04.008,1.94,,Degradation of HDAC6 in MM1S after 6 h treatment by in-cell ELISA analysis,
1324,HDAC6,,10.1016/j.chembiol.2020.04.008,,N.D.,,
1325,HDAC6,,10.1016/j.chembiol.2020.04.008,,,,
1326,HDAC6,,10.1016/j.chembiol.2020.04.008,,,,
1327,HDAC6,,10.1016/j.chembiol.2020.04.008,,,,
1328,HDAC6,,10.1016/j.chembiol.2020.04.008,,,,
1329,HDAC6,,10.1016/j.chembiol.2020.04.008,,,,
1330,HDAC6,,10.1016/j.chembiol.2020.04.008,,,,
1331,Beta-tubulin,,10.3390/cells9051083,,N.D.,,
1331,Alpha-tubulin,,10.3390/cells9051083,,N.D.,,
1332,Beta-tubulin,,10.3390/cells9051083,,N.D.,,
1332,Alpha-tubulin,,10.3390/cells9051083,,N.D.,,
1333,Alpha-tubulin,,10.3390/cells9051083,,N.D.,,
1333,Beta-tubulin,,10.3390/cells9051083,,N.D.,,
1334,Alpha-tubulin,,10.3390/cells9051083,,N.D.,,
1334,Beta-tubulin,,10.3390/cells9051083,,N.D.,,
1335,Alpha-tubulin,,10.3390/cells9051083,,N.D.,,
1335,Beta-tubulin,,10.3390/cells9051083,,N.D.,,
1336,Alpha-tubulin,,10.3390/cells9051083,,N.D.,,
1336,Beta-tubulin,,10.3390/cells9051083,,N.D.,,
1337,Alpha-tubulin,,10.3390/cells9051083,,N.D.,,
1337,Beta-tubulin,,10.3390/cells9051083,,N.D.,,
1338,Beta-tubulin,,10.3390/cells9051083,,N.D.,,
1338,Alpha-tubulin,,10.3390/cells9051083,,N.D.,,
1339,Alpha-tubulin,,10.3390/cells9051083,,N.D.,,
1339,Beta-tubulin,,10.3390/cells9051083,,N.D.,,
1340,Alpha-tubulin,,10.3390/cells9051083,,N.D.,,
1340,Beta-tubulin,,10.3390/cells9051083,,N.D.,,
1341,Alpha-tubulin,,10.3390/cells9051083,,N.D.,,
1341,Beta-tubulin,,10.3390/cells9051083,,N.D.,,
1342,Alpha-tubulin,,10.3390/cells9051083,,N.D.,,
1342,Beta-tubulin,,10.3390/cells9051083,,N.D.,,
1343,Beta-tubulin,,10.3390/cells9051083,,N.D.,,
1343,Alpha-tubulin,,10.3390/cells9051083,,N.D.,,
1344,Tau,,10.7554/eLife.45457,,75/95,,
1345,Rpn13,,10.1038/s41375-019-0467-z,,95,,
1346,Src,,10.3390/molecules25081948,,,,
1346,IGF-1R,,10.3390/molecules25081948,,,,
1347,IGF-1R,,10.3390/molecules25081948,,,,
1347,Src,,10.3390/molecules25081948,,,,
1348,Src,,10.3390/molecules25081948,,,,
1348,IGF-1R,,10.3390/molecules25081948,,,,
1349,Src,,10.3390/molecules25081948,,,,
1349,IGF-1R,,10.3390/molecules25081948,,,,
1350,IGF-1R,,10.3390/molecules25081948,,,,
1350,Src,,10.3390/molecules25081948,,,,
1351,Src,,10.3390/molecules25081948,,,,
1351,IGF-1R,,10.3390/molecules25081948,,,,
1352,IGF-1R,,10.3390/molecules25081948,,,,
1352,Src,,10.3390/molecules25081948,,,,
1353,Src,,10.3390/molecules25081948,,,,
1353,IGF-1R,,10.3390/molecules25081948,,,,
1354,Src,,10.3390/molecules25081948,,,,
1354,IGF-1R,,10.3390/molecules25081948,,,,
1355,IGF-1R,,10.3390/molecules25081948,,,,
1355,Src,,10.3390/molecules25081948,,,,
1356,IGF-1R,,10.3390/molecules25081948,,,,
1356,Src,,10.3390/molecules25081948,,,,
1357,NS3,,10.1038/s41467-019-11429-w,669,,Degradation of NS3 in Huh7.5 cells after 4 h treatment,
1358,NS3,,10.1038/s41467-019-11429-w,489,,Degradation of NS3 in Huh7.5 cells after 4 h treatment,
1359,NS3,,10.1038/s41467-019-11429-w,50,,Degradation of NS3 in Huh7.5 cells after 4 h treatment,
1360,BCL-xL,,10.1038/s41467-020-15838-0,46,96.2,Degradation of BCL-xL in WI38 cells after 16 h treatment,
1361,BTK,,10.1039/c9cc08238g,,,,
1362,BTK,,10.1039/c9cc08238g,,,,
1363,BTK,,10.1039/c9cc08238g,,,,
1364,BTK,,10.1039/c9cc08238g,,,,
1365,BTK,,10.1039/c9cc08238g,,,,
1366,BTK,,10.1039/c9cc08238g,,,,
1367,BTK,,10.1039/c9cc08238g,,,,
1368,BTK,,10.1039/c9cc08238g,,,,
1369,BTK,,10.1039/c9cc08238g,,,,
1370,BTK,,10.1039/c9cc08238g,,,,
1371,BTK,,10.1039/c9cc08238g,,,,
1372,BTK,,10.1039/c9cc08238g,,,,
1373,BLK,,10.1039/c9cc08238g,220,75,Degradation of BLK in Ramos cells after 18 h treatment,
1373,BTK,,10.1039/c9cc08238g,136,88,Degradation of BTK in K562 cells after 18 h treatment,
1374,BTK,,10.1039/c9cc08238g,,,,
1375,BTK,,10.1039/c9cc08238g,,,,
1376,BTK,,10.1039/c9cc08238g,,,,
1377,CDK8,,10.1021/acsmedchemlett.8b00011,,N.D.,,
1378,CDK8,,10.1021/acsmedchemlett.8b00011,,,,
1379,CDK8,,10.1021/acsmedchemlett.8b00011,,N.D.,,
1380,BTK,,10.1021/jacs.9b13907,2.2,97,Degradation of BTK in Mino cells after 24 h treatment,
1381,BTK,,10.1021/jacs.9b13907,8.6,91,Degradation of BTK in Mino cells after 24 h treatment,
1382,BTK,,10.1021/jacs.9b13907,1.9,88,Degradation of BTK in Mino cells after 24 h treatment,
1383,BTK,,10.1021/jacs.9b13907,10,68,Degradation of BTK in Mino cells after 24 h treatment,
1384,BTK,,10.1021/jacs.9b13907,35,66,Degradation of BTK in Mino cells after 24 h treatment,
1385,BTK,,10.1021/jacs.9b13907,6,85,Degradation of BTK in Mino cells after 24 h treatment,
1386,BTK,32 (WB),10.1021/jacs.9b13907,,,,% BTK degradation in Mino cells after 24 h treatment at 1 μM
1387,BTK,19 (WB),10.1021/jacs.9b13907,,,,% BTK degradation in Mino cells after 24 h treatment at 1 μM
1388,BTK,14 (WB),10.1021/jacs.9b13907,,,,% BTK degradation in Mino cells after 24 h treatment at 1 μM
1389,BTK,17 (WB),10.1021/jacs.9b13907,,,,% BTK degradation in Mino cells after 24 h treatment at 1 μM
1390,BTK,68 (WB),10.1021/jacs.9b13907,,,,% BTK degradation in Mino cells after 24 h treatment at 1 μM
1391,BTK,77 (WB),10.1021/jacs.9b13907,,,,% BTK degradation in Mino cells after 24 h treatment at 1 μM
1392,BTK,29 (WB),10.1021/jacs.9b13907,,,,% BTK degradation in Mino cells after 24 h treatment at 1 μM
1393,BTK,9 (WB),10.1021/jacs.9b13907,,,,% BTK degradation in Mino cells after 24 h treatment at 1 μM
1394,BTK,2 (WB),10.1021/jacs.9b13907,,,,% BTK degradation in Mino cells after 24 h treatment at 1 μM
1395,BTK,25 (WB),10.1021/jacs.9b13907,,,,% BTK degradation in Mino cells after 24 h treatment at 1 μM
1396,BRD4,,10.1021/acschembio.8b01083,,,,
1397,c-Met,,10.1021/acschembio.7b00969,,N.D.,,
1398,c-Met,,10.1021/acschembio.7b00969,,N.D.,,
1399,c-Met,,10.1021/acschembio.7b00969,,N.D.,,
1400,c-Met,,10.1021/acschembio.7b00969,,N.D.,,
1401,c-Met,,10.1021/acschembio.7b00969,,N.D.,,
1402,c-Met,,10.1021/acschembio.7b00969,,N.D.,,
1403,c-Met,,10.1021/acschembio.7b00969,,N.D.,,
1404,c-Met,,10.1021/acschembio.7b00969,,N.D.,,
1405,c-Met,,10.1021/acschembio.7b00969,,N.D.,,
1406,c-Met,,10.1021/acschembio.7b00969,,N.D.,,
1407,c-Met,,10.1021/acschembio.7b00969,,N.D.,,
1408,c-KIT,,10.1021/acschembio.7b00969,,N.D.,,
1409,c-KIT,,10.1021/acschembio.7b00969,,N.D.,,
1410,c-KIT,,10.1021/acschembio.7b00969,,N.D.,,
1411,c-KIT,,10.1021/acschembio.7b00969,,N.D.,,
1412,c-KIT,,10.1021/acschembio.7b00969,,N.D.,,
1413,c-KIT,,10.1021/acschembio.7b00969,,N.D.,,
1414,c-KIT,,10.1021/acschembio.7b00969,,N.D.,,
1415,c-KIT,,10.1021/acschembio.7b00969,,N.D.,,
1416,c-KIT,,10.1021/acschembio.7b00969,,N.D.,,
1417,c-KIT,,10.1021/acschembio.7b00969,,N.D.,,
1418,c-KIT,,10.1021/acschembio.7b00969,,N.D.,,
1419,c-KIT,,10.1021/acschembio.7b00969,,N.D.,,
1420,c-KIT,,10.1021/acschembio.7b00969,,N.D.,,
1421,c-KIT,,10.1021/acschembio.7b00969,,N.D.,,
1422,c-KIT,,10.1021/acschembio.7b00969,,N.D.,,
1423,CDK6,,10.1182/blood.2019003604,,,,
1423,CDK4,,10.1182/blood.2019003604,,,,
1424,CDK4,,10.1182/blood.2019003604,,,,
1424,CDK6,,10.1182/blood.2019003604,,,,
1425,CDK6,,10.1182/blood.2019003604,,,,
1425,CDK4,,10.1182/blood.2019003604,,,,
1426,CDK4,,10.1182/blood.2019003604,,,,
1426,CDK6,,10.1182/blood.2019003604,,,,
1427,CDK4,,10.1182/blood.2019003604,,,,
1427,CDK6,,10.1182/blood.2019003604,,,,
1428,CDK6,,10.1182/blood.2019003604,,,,
1428,CDK4,,10.1182/blood.2019003604,,,,
1429,AR,,10.1021/acsmedchemlett.9b00115,<=50/<=50,>=71/51-70,Degradation of AR in LNCaP/VCaP cells after 2-4 h treatment,
1430,AR,,10.1021/acsmedchemlett.9b00115,<=501,51-70,Degradation of AR in LNCaP cells after 2-4 h treatment,
1431,AR,,10.1021/acsmedchemlett.9b00115,<=50,>=71,Degradation of AR in LNCaP cells after 2-4 h treatment,
1432,AR,,10.1021/acsmedchemlett.9b00115,<=50,>=71,Degradation of AR in LNCaP cells after 2-4 h treatment,
1433,AR,,10.1021/acsmedchemlett.9b00115,<=50,>=71,Degradation of AR in LNCaP cells after 2-4 h treatment,
1434,AR,,10.1021/acsmedchemlett.9b00115,<=50,>=71,Degradation of AR in LNCaP cells after 2-4 h treatment,
1435,Tau,,10.3389/fncel.2022.801179,,,,
1436,Tau,,10.3389/fncel.2022.801179,,,,
1437,Tau,,10.3389/fncel.2022.801179,,,,
1438,Tau,,10.3389/fncel.2022.801179,,,,
1439,Tau,,10.3389/fncel.2022.801179,,,,
1440,BRD4,,10.1021/acsmedchemlett.9b00042,,,,
1441,BRD4,,10.1021/acsmedchemlett.9b00042,,,,
1442,AR,,10.1021/acsmedchemlett.9b00424,,,,
1443,AR,,10.1021/acsmedchemlett.9b00424,,,,
1444,BRD4,,10.1021/acsmedchemlett.9b00424,,,,
1445,BRD4,,10.1021/acsmedchemlett.9b00424,,,,
1446,TBK1,,10.1021/acsmedchemlett.9b00424,,,,
1447,TBK1,,10.1021/acsmedchemlett.9b00424,,,,
1448,ERRalpha,,10.1021/acsmedchemlett.9b00424,,,,
1449,BRD4,,10.1021/acsmedchemlett.9b00424,,,,
1450,BRD4,,10.1021/acsmedchemlett.9b00424,,,,
1451,IRAK4,>50/>50/>50,10.1021/acsmedchemlett.9b00423,,,,% IRAK4 degradation in OCILY-10 cells after 4 h treatment at 10/100/1000 nM
1452,IRAK4,>50/>50/>50,10.1021/acsmedchemlett.9b00423,,,,% IRAK4 degradation in OCILY-10 cells after 4 h treatment at 10/100/1000 nM
1453,IRAK4,>50/>50/>50,10.1021/acsmedchemlett.9b00423,,,,% IRAK4 degradation in OCILY-10 cells after 4 h treatment at 10/100/1000 nM
1454,IRAK4,>50/>50/>50,10.1021/acsmedchemlett.9b00423,,,,% IRAK4 degradation in OCILY-10 cells after 4 h treatment at 10/100/1000 nM
1455,IRAK4,20-50/>50/>50,10.1021/acsmedchemlett.9b00423,,,,% IRAK4 degradation in OCILY-10 cells after 4 h treatment at 10/100/1000 nM
1456,IRAK4,>50/>50/>50,10.1021/acsmedchemlett.9b00423,,,,% IRAK4 degradation in OCILY-10 cells after 4 h treatment at 10/100/1000 nM
1457,IRAK4,>50/>50/>50,10.1021/acsmedchemlett.9b00423,,,,% IRAK4 degradation in OCILY-10 cells after 4 h treatment at 10/100/1000 nM
1458,IRAK4,20-50/>50/>50,10.1021/acsmedchemlett.9b00423,,,,% IRAK4 degradation in OCILY-10 cells after 4 h treatment at 10/100/1000 nM
1459,IRAK4,20-50/>50/>50,10.1021/acsmedchemlett.9b00423,,,,% IRAK4 degradation in OCILY-10 cells after 4 h treatment at 10/100/1000 nM
1460,IRAK4,20-50/>50/>50,10.1021/acsmedchemlett.9b00423,,,,% IRAK4 degradation in OCILY-10 cells after 4 h treatment at 10/100/1000 nM
1461,IRAK4,,10.1021/acsmedchemlett.9b00385,<30,>70,Degradation of IRAK4 in MCF7 cells,
1462,IRAK4,,10.1021/acsmedchemlett.9b00385,<30,>70,Degradation of IRAK4 in MCF7 cells,
1463,IRAK4,,10.1021/acsmedchemlett.9b00385,<30,>70,Degradation of IRAK4 in MCF7 cells,
1464,IRAK4,,10.1021/acsmedchemlett.9b00385,<30,50-70,Degradation of IRAK4 in MCF7 cells,
1465,IRAK4,,10.1021/acsmedchemlett.9b00385,<30,50-70,Degradation of IRAK4 in MCF7 cells,
1466,IRAK4,,10.1021/acsmedchemlett.9b00385,30-100,>70,Degradation of IRAK4 in MCF7 cells,
1467,ER,,10.1021/acsmedchemlett.9b00397,0.3,,Degradation of ERalpha in MCF7 cells,
1468,ER,,10.1021/acsmedchemlett.9b00397,0.4,,Degradation of ERalpha in MCF7 cells,
1469,ER,,10.1021/acsmedchemlett.9b00397,0.3,,Degradation of ERalpha in MCF7 cells,
1470,ER,,10.1021/acsmedchemlett.9b00397,0.4,,Degradation of ERalpha in MCF7 cells,
1471,ER,,10.1021/acsmedchemlett.9b00397,0.8,,Degradation of ERalpha in MCF7 cells,
1472,ER,,10.1021/acsmedchemlett.9b00397,0.6,,Degradation of ERalpha in MCF7 cells,
1473,EGFR,,10.1021/acsmedchemlett.9b00283,,,,
1473,EGFR L858R/T790M,,10.1002/anie.202003500,,,,
1474,EGFR L858R/T790M,,10.1002/anie.202003500,,,,
1475,EGFR,,10.1021/acsmedchemlett.9b00283,,,,
1476,EGFR L858R/T790M,24/59/62 (WB),10.1002/anie.202003500,,,,% EGFR degradation in L858R/T790M BaF3 cells after 24 h treatment at 0.01/0.1/1 μM
1476,EGFR L858R/T790M/C797S,74 (WB),10.1002/anie.202003500,,,,% EGFR degradation in L858R/T790M/C797S BaF3 cells after 24 h treatment at 0.1 μM
1476,EGFR L858R/T790M/L718Q,71 (WB),10.1002/anie.202003500,,,,% EGFR degradation in L858R/T790M/L718Q BaF3 cells after 24 h treatment at 0.1 μM
1477,ALK,,10.1021/acsmedchemlett.9b00296,,,,
1478,ALK,,10.1021/acsmedchemlett.9b00296,,,,
1479,ALK,,10.1021/acsmedchemlett.9b00296,,,,
1480,KRAS,<25/>=50/>=50,10.1021/acsmedchemlett.9b00584,,,,% KRAS degradation in H2023 cells at 300/1000/3000 nM
1481,KRAS,<25/>=50/>=50,10.1021/acsmedchemlett.9b00584,,,,% KRAS degradation in H2023 cells at 300/1000/3000 nM
1482,KRAS,<25/25-50/25-50,10.1021/acsmedchemlett.9b00584,,,,% KRAS degradation in H2023 cells at 300/1000/3000 nM
1483,KRAS,<25/25-50/25-50,10.1021/acsmedchemlett.9b00584,,,,% KRAS degradation in H2023 cells at 300/1000/3000 nM
1484,KRAS,<25/25-50/25-50,10.1021/acsmedchemlett.9b00584,,,,% KRAS degradation in H2023 cells at 300/1000/3000 nM
1485,KRAS,<25/<25/<25,10.1021/acsmedchemlett.9b00584,,,,% KRAS degradation in H2023 cells at 300/1000/3000 nM
1486,SHP2,4/0,10.1021/acs.jmedchem.0c00471,,,,% SHP2 degradation in KYSE520 cells after 6 h treatment at 100/1000 nM
1487,SHP2,9/7,10.1021/acs.jmedchem.0c00471,,,,% SHP2 degradation in KYSE520 cells after 6 h treatment at 100/1000 nM
1488,SHP2,13/6,10.1021/acs.jmedchem.0c00471,,,,% SHP2 degradation in KYSE520 cells after 6 h treatment at 100/1000 nM
1489,SHP2,0/3,10.1021/acs.jmedchem.0c00471,,,,% SHP2 degradation in KYSE520 cells after 6 h treatment at 100/1000 nM
1490,SHP2,0/0,10.1021/acs.jmedchem.0c00471,,,,% SHP2 degradation in KYSE520 cells after 6 h treatment at 100/1000 nM
1491,SHP2,20/14,10.1021/acs.jmedchem.0c00471,,,,% SHP2 degradation in KYSE520 cells after 6 h treatment at 100/1000 nM
1492,SHP2,81/80,10.1021/acs.jmedchem.0c00471,,,,% SHP2 degradation in KYSE520 cells after 6 h treatment at 100/1000 nM
1493,SHP2,>95/>95,10.1021/acs.jmedchem.0c00471,,,,% SHP2 degradation in KYSE520 cells after 6 h treatment at 100/1000 nM
1494,SHP2,>95/>95,10.1021/acs.jmedchem.0c00471,,,,% SHP2 degradation in KYSE520 cells after 6 h treatment at 100/1000 nM
1495,SHP2,>95/93,10.1021/acs.jmedchem.0c00471,,,,% SHP2 degradation in KYSE520 cells after 6 h treatment at 100/1000 nM
1496,SHP2,>95/>95,10.1021/acs.jmedchem.0c00471,,,,% SHP2 degradation in KYSE520 cells after 6 h treatment at 100/1000 nM
1497,SHP2,>95/>95,10.1021/acs.jmedchem.0c00471,,,,% SHP2 degradation in KYSE520 cells after 6 h treatment at 100/1000 nM
1498,SHP2,>95/>95,10.1021/acs.jmedchem.0c00471,,,,% SHP2 degradation in KYSE520 cells after 6 h treatment at 100/1000 nM
1499,SHP2,80/>95,10.1021/acs.jmedchem.0c00471,,,,% SHP2 degradation in KYSE520 cells after 6 h treatment at 100/1000 nM
1500,SHP2,32/87,10.1021/acs.jmedchem.0c00471,,,,% SHP2 degradation in KYSE520 cells after 6 h treatment at 100/1000 nM
1501,SHP2,53/>95,10.1021/acs.jmedchem.0c00471,,,,% SHP2 degradation in KYSE520 cells after 6 h treatment at 100/1000 nM
1502,SHP2,85/>95,10.1021/acs.jmedchem.0c00471,,,,% SHP2 degradation in KYSE520 cells after 6 h treatment at 100/1000 nM
1503,SHP2,80/>95,10.1021/acs.jmedchem.0c00471,,,,% SHP2 degradation in KYSE520 cells after 6 h treatment at 100/1000 nM
1504,SHP2,62/90,10.1021/acs.jmedchem.0c00471,,,,% SHP2 degradation in KYSE520 cells after 6 h treatment at 100/1000 nM
1505,SHP2,>95/>95,10.1021/acs.jmedchem.0c00471,6/2.6,,Degradation of SHP2 in KYSE520/MV4;11 cells after 12 h treatment,% SHP2 degradation in KYSE520 cells after 6 h treatment at 100/1000 nM
1506,SHP2,>95/>95,10.1021/acs.jmedchem.0c00471,,,,% SHP2 degradation in KYSE520 cells after 6 h treatment at 100/1000 nM
1507,SHP2,>95/>95,10.1021/acs.jmedchem.0c00471,,,,% SHP2 degradation in KYSE520 cells after 6 h treatment at 100/1000 nM
1508,SHP2,0/82,10.1021/acs.jmedchem.0c00471,,,,% SHP2 degradation in KYSE520 cells after 6 h treatment at 100/1000 nM
1509,FAK,,10.1021/acsmedchemlett.9b00372,0.37/0.04,,Degradation of FAK in LNCaP/Ramos cells after 8 h treatment,
1509,FAK,,10.1021/acsmedchemlett.9b00372,0.31/0.08/0.33,,Degradation of FAK in TM3/PA1/MDA-MB-436 cells after 8 h treatment,
1509,FAK,,10.1007/s13238-020-00732-8,1.3/0.4,,Degradation of Fak in primary Sertoli/germ cells after 8 h treatment,
1510,BCR-ABL,,10.1021/acs.jmedchem.9b02058,391,,Degradation of BCR-ABL in K562 cells,
1511,BCR-ABL,,10.1021/acs.jmedchem.9b02058,114,,Degradation of BCR-ABL in K562 cells,
1512,BCR-ABL,,10.1021/acs.jmedchem.9b02058,62,,Degradation of BCR-ABL in K562 cells,
1513,BCR-ABL,,10.1021/acs.jmedchem.9b02058,>500,,Degradation of BCR-ABL in K562 cells,
1514,BCR-ABL,,10.1021/acs.jmedchem.9b02058,>500,,Degradation of BCR-ABL in K562 cells,
1515,BRD2,,10.1021/acscentsci.9b00713,,,,
1516,BRD3,,10.1126/sciadv.aay5064,,,,
1516,BRD2,,10.1126/sciadv.aay5064,,,,
1516,BRD4,,10.1126/sciadv.aay5064,,,,
1517,BRD3,,10.1126/sciadv.aay5064,,,,
1517,BRD2,,10.1126/sciadv.aay5064,,,,
1517,BRD4,,10.1126/sciadv.aay5064,,,,
1518,BRD3,,10.1126/sciadv.aay5064,,,,
1518,BRD2,,10.1126/sciadv.aay5064,,,,
1518,BRD4,,10.1126/sciadv.aay5064,,,,
1519,BRD3,,10.1126/sciadv.aay5064,,,,
1519,BRD2,,10.1126/sciadv.aay5064,,,,
1519,BRD4,,10.1126/sciadv.aay5064,,,,
1520,BRD3,,10.1126/sciadv.aay5064,,,,
1520,BRD2,,10.1126/sciadv.aay5064,,,,
1520,BRD4,,10.1126/sciadv.aay5064,,,,
1521,BRD3,,10.1126/sciadv.aay5064,,,,
1521,BRD4,,10.1126/sciadv.aay5064,,,,
1521,BRD2,,10.1126/sciadv.aay5064,,,,
1522,BRD2,,10.1126/sciadv.aay5064,,,,
1522,BRD4,,10.1126/sciadv.aay5064,,,,
1522,BRD3,,10.1126/sciadv.aay5064,,,,
1523,BRD3,,10.1126/sciadv.aay5064,,,,
1523,BRD4,,10.1126/sciadv.aay5064,,,,
1523,BRD2,,10.1126/sciadv.aay5064,,,,
1524,BRD4,,10.1126/sciadv.aay5064,,,,
1524,BRD2,,10.1126/sciadv.aay5064,,,,
1524,BRD3,,10.1126/sciadv.aay5064,,,,
1525,BRD4,,10.1126/sciadv.aay5064,,,,
1525,BRD3,,10.1126/sciadv.aay5064,,,,
1525,BRD2,,10.1126/sciadv.aay5064,,,,
1526,BRD3,,10.1126/sciadv.aay5064,,,,
1526,BRD2,,10.1126/sciadv.aay5064,,,,
1526,BRD4,,10.1126/sciadv.aay5064,,,,
1527,BRD4,,10.1126/sciadv.aay5064,,,,
1527,BRD2,,10.1126/sciadv.aay5064,,,,
1527,BRD3,,10.1126/sciadv.aay5064,,,,
1528,BRD3,,10.1126/sciadv.aay5064,,,,
1528,BRD2,,10.1126/sciadv.aay5064,,,,
1528,BRD4,,10.1126/sciadv.aay5064,,,,
1529,FKBP12,,10.1126/sciadv.aay5064,,,,
1530,FKBP12,,10.1126/sciadv.aay5064,,,,
1531,FKBP12,,10.1126/sciadv.aay5064,,,,
1532,FKBP12,,10.1126/sciadv.aay5064,,,,
1533,FKBP12,,10.1126/sciadv.aay5064,,,,
1534,FKBP12,,10.1126/sciadv.aay5064,,,,
1535,BRD2,,10.1002/anie.201914396,>125,,Degradation of BRD2 in HeLa cells after 4/18 h treatment,
1535,BRD3,,10.1002/anie.201914396,>125,,Degradation of BRD3 in HeLa cells after 4/18 h treatment,
1535,BRD4,,10.1002/anie.201914396,25-125,,Degradation of BRD4 in HeLa cells after 4/18 h treatment,
1536,BRD2,,10.1002/anie.201914396,,,,
1536,BRD3,,10.1002/anie.201914396,,,,
1536,BRD4,,10.1002/anie.201914396,,,,
1537,BTK,,10.1021/acs.biochem.8b00391,,N.D.,,
1538,EGFR L858R/T790M,0/2/19 (WB),10.1002/anie.202003500,,,,% EGFR degradation in L858R/T790M BaF3 cells after 24 h treatment at 0.01/0.1/1 μM
1539,BTK,,10.1021/acs.biochem.8b00391,,N.D.,,
1540,EGFR L858R/T790M,17/45/40 (WB),10.1002/anie.202003500,,,,% EGFR degradation in L858R/T790M BaF3 cells after 24 h treatment at 0.01/0.1/1 μM
1541,EGFR L858R/T790M,,10.1002/anie.202003500,,,,
1542,EGFR L858R/T790M,,10.1002/anie.202003500,,,,
1543,EGFR L858R/T790M,,10.1002/anie.202003500,,,,
1544,EGFR L858R/T790M,,10.1002/anie.202003500,,,,
1545,EGFR L858R/T790M,,10.1002/anie.202003500,,,,
1546,EGFR L858R/T790M,,10.1002/anie.202003500,,,,
1547,EGFR L858R/T790M,,10.1002/anie.202003500,,,,
1548,EGFR L858R/T790M,,10.1002/anie.202003500,,,,
1549,EGFR L858R/T790M,,10.1002/anie.202003500,,,,
1550,EGFR L858R/T790M,,10.1002/anie.202003500,,,,
1551,EGFR L858R/T790M,,10.1002/anie.202003500,,,,
1552,EGFR L858R/T790M,,10.1002/anie.202003500,,,,
1553,EGFR L858R/T790M,,10.1002/anie.202003500,,,,
1554,EGFR L858R/T790M,,10.1002/anie.202003500,,,,
1555,EGFR L858R/T790M,,10.1002/anie.202003500,,,,
1556,AR,,10.1021/acsmedchemlett.0c00194,,,,
1557,AR,,10.1021/acsmedchemlett.0c00194,,,,
1558,AR,,10.1021/acsmedchemlett.0c00194,,,,
1559,AR,,10.1021/acsmedchemlett.0c00194,,,,
1560,AR,,10.1021/acsmedchemlett.0c00194,,N.D.,,
1561,AR,,10.1021/acsmedchemlett.0c00194,10,33,Degradation of AR in LNCaP cells after 6 h treatment,
1562,AR,,10.1021/acsmedchemlett.0c00194,,,,
1563,AR,,10.1021/acsmedchemlett.0c00194,,,,
1564,AR,,10.1021/acsmedchemlett.0c00194,,,,
1565,AR,,10.1021/acsmedchemlett.0c00194,,,,
1566,AR,,10.1021/acsmedchemlett.0c00194,,,,
1567,AR,,10.1021/acsmedchemlett.0c00194,,,,
1568,AR,,10.1021/acsmedchemlett.0c00194,,,,
1569,AR,,10.1021/acsmedchemlett.0c00194,,,,
1570,Alpha-syn,,10.1021/acsmedchemlett.0c00192,,,,
1571,Alpha-syn,,10.1021/acsmedchemlett.0c00192,,,,
1572,Alpha-syn,,10.1021/acsmedchemlett.0c00192,,,,
1573,Alpha-syn,,10.1021/acsmedchemlett.0c00192,,,,
1574,Alpha-syn,,10.1021/acsmedchemlett.0c00192,,,,
1575,Alpha-syn,,10.1021/acsmedchemlett.0c00192,,,,
1576,TRKB,,10.1021/acsmedchemlett.0c00235,,,,
1576,TRKA,,10.1021/acsmedchemlett.0c00235,,,,
1576,TRKC,,10.1021/acsmedchemlett.0c00235,,,,
1577,TRKA,,10.1021/acsmedchemlett.0c00235,,,,
1577,TRKB,,10.1021/acsmedchemlett.0c00235,,,,
1577,TRKC,,10.1021/acsmedchemlett.0c00235,,,,
1578,TRKA,,10.1021/acsmedchemlett.0c00235,,,,
1578,TRKB,,10.1021/acsmedchemlett.0c00235,,,,
1578,TRKC,,10.1021/acsmedchemlett.0c00235,,,,
1579,TRKA,,10.1021/acsmedchemlett.0c00235,,,,
1579,TRKB,,10.1021/acsmedchemlett.0c00235,,,,
1579,TRKC,,10.1021/acsmedchemlett.0c00235,,,,
1580,TRKA,,10.1021/acsmedchemlett.0c00235,,,,
1580,TRKB,,10.1021/acsmedchemlett.0c00235,,,,
1580,TRKC,,10.1021/acsmedchemlett.0c00235,,,,
1581,TRKA,,10.1021/acsmedchemlett.0c00235,,,,
1581,TRKB,,10.1021/acsmedchemlett.0c00235,,,,
1581,TRKC,,10.1021/acsmedchemlett.0c00235,,,,
1582,TRKA,,10.1021/acsmedchemlett.0c00235,,,,
1582,TRKB,,10.1021/acsmedchemlett.0c00235,,,,
1582,TRKC,,10.1021/acsmedchemlett.0c00235,,,,
1583,TRKA,,10.1021/acsmedchemlett.0c00235,,,,
1583,TRKB,,10.1021/acsmedchemlett.0c00235,,,,
1583,TRKC,,10.1021/acsmedchemlett.0c00235,,,,
1584,AR,,10.1021/acsmedchemlett.0c00236,<=50/<=50,>=71/51-70,"Degradation of AR in LNCaP/VCaP cells using ELISA assay (DC50: 15min, Dmax: 4h)",
1585,AR,,10.1021/acsmedchemlett.0c00236,<=50/<=50,>=71/51-70,"Degradation of AR in LNCaP/VCaP cells using ELISA assay (DC50: 15min, Dmax: 4h)",
1586,AR,,10.1021/acsmedchemlett.0c00236,<=50/<=50,>=71/51-70,"Degradation of AR in LNCaP/VCaP cells using ELISA assay (DC50: 15min, Dmax: 4h)",
1587,AR,,10.1021/acsmedchemlett.0c00236,<=50/<=50,>=71/>=71,"Degradation of AR in LNCaP/VCaP cells using ELISA assay (DC50: 15min, Dmax: 4h)",
1588,AR,,10.1021/acsmedchemlett.0c00236,<=50/<=50,>=71/>=71,"Degradation of AR in LNCaP/VCaP cells using ELISA assay (DC50: 15min, Dmax: 4h)",
1589,AR,,10.1021/acsmedchemlett.0c00236,<=50/<=50,>=71/>=71,"Degradation of AR in LNCaP/VCaP cells using ELISA assay (DC50: 15min, Dmax: 4h)",
1590,AR,,10.1021/acsmedchemlett.0c00236,<=50/<=50,>=71/>=71,"Degradation of AR in LNCaP/VCaP cells using ELISA assay (DC50: 15min, Dmax: 4h)",
1591,BRD4,,10.1038/s41589-019-0304-8,,,,
1592,BRD4,,10.1038/s41589-019-0304-8,,,,
1593,PDEdelta,,10.1021/acs.jmedchem.0c00929,30000,,Degradation of PDEdelta in SW480 cells after 24 h treatment,
1594,PDEdelta,,10.1021/acs.jmedchem.0c00929,25000,,Degradation of PDEdelta in SW480 cells after 24 h treatment,
1595,PDEdelta,,10.1021/acs.jmedchem.0c00929,22000,,Degradation of PDEdelta in SW480 cells after 24 h treatment,
1596,PDEdelta,,10.1021/acs.jmedchem.0c00929,15000,,Degradation of PDEdelta in SW480 cells after 24 h treatment,
1597,PDEdelta,,10.1021/acs.jmedchem.0c00929,14000,,Degradation of PDEdelta in SW480 cells after 24 h treatment,
1598,PDEdelta,,10.1021/acs.jmedchem.0c00929,3600,,Degradation of PDEdelta in SW480 cells after 24 h treatment,
1599,PDEdelta,,10.1021/acs.jmedchem.0c00929,30000,,Degradation of PDEdelta in SW480 cells after 24 h treatment,
1600,PDEdelta,,10.1021/acs.jmedchem.0c00929,10000,,Degradation of PDEdelta in SW480 cells after 24 h treatment,
1601,PDEdelta,,10.1021/acs.jmedchem.0c00929,5000,,Degradation of PDEdelta in SW480 cells after 24 h treatment,
1602,BCR-ABL,,10.1021/acs.jmedchem.0c00967,>10000,,Degradation of BCR-ABL in K562 cells after 32 h treatment,
1603,BCR-ABL,,10.1021/acs.jmedchem.0c00967,>10000,,Degradation of BCR-ABL in K562 cells after 32 h treatment,
1604,BCR-ABL,,10.1021/acs.jmedchem.0c00967,>10000,,Degradation of BCR-ABL in K562 cells after 32 h treatment,
1605,BCR-ABL,,10.1021/acs.jmedchem.0c00967,>10000,,Degradation of BCR-ABL in K562 cells after 32 h treatment,
1606,BCR-ABL,,10.1021/acs.jmedchem.0c00967,>10000,,Degradation of BCR-ABL in K562 cells after 32 h treatment,
1607,BCR-ABL,,10.1021/acs.jmedchem.0c00967,56,,Degradation of BCR-ABL in K562 cells after 48 h treatment,
1608,BCR-ABL,,10.1021/acs.jmedchem.0c00967,56,,Degradation of BCR-ABL in K562 cells after 48 h treatment,
1609,BCR-ABL,,10.1021/acs.jmedchem.0c00967,20,,Degradation of BCR-ABL in K562 cells after 48 h treatment,
1610,BCR-ABL,,10.1021/acs.jmedchem.0c00967,56,,Degradation of BCR-ABL in K562 cells after 48 h treatment,
1611,BCR-ABL,,10.1021/acs.jmedchem.0c00967,10,,Degradation of BCR-ABL in K562 cells after 32 h treatment,
1612,BCR-ABL,,10.1021/acs.jmedchem.0c00967,>625,,Degradation of BCR-ABL in K562 cells after 32 h treatment,
1613,BCR-ABL,,10.1021/acs.jmedchem.0c00967,400,,Degradation of BCR-ABL in K562 cells after 32 h treatment,
1614,BCR-ABL,,10.1021/acs.jmedchem.0c00967,300,,Degradation of BCR-ABL in K562 cells after 32 h treatment,
1615,BCR-ABL T315I,,10.1021/acs.jmedchem.0c00967,,,,
1615,BCR-ABL,,10.1021/acs.jmedchem.0c00967,200,,Degradation of BCR-ABL in K562 cells after 32 h treatment,
1616,BCR-ABL,,10.1021/acs.jmedchem.0c00967,500,,Degradation of BCR-ABL in K562 cells after 32 h treatment,
1617,BCR-ABL,,10.1021/acs.jmedchem.0c00967,625,,Degradation of BCR-ABL in K562 cells after 32 h treatment,
1618,BCR-ABL,,10.1021/acs.jmedchem.0c00967,70,,Degradation of BCR-ABL in K562 cells after 32 h treatment,
1619,BCR-ABL,,10.1021/acs.jmedchem.0c00967,70,,Degradation of BCR-ABL in K562 cells after 32 h treatment,
1620,BCR-ABL T315I,,10.1021/acs.jmedchem.0c00967,,,,
1620,BCR-ABL V468F,,10.1021/acs.jmedchem.0c00967,,,,
1620,BCR-ABL H396R,,10.1021/acs.jmedchem.0c00967,,,,
1620,BCR-ABL E255K,,10.1021/acs.jmedchem.0c00967,,,,
1620,BCR-ABL,,10.1021/acs.jmedchem.0c00967,20,,Degradation of BCR-ABL in K562 cells after 32 h treatment,
1621,BCR-ABL,,10.1021/acs.jmedchem.0c00967,70,,Degradation of BCR-ABL in K562 cells after 32 h treatment,
1622,BCR-ABL T315I,,10.1021/acs.jmedchem.0c00967,,,,
1623,BCR-ABL,,10.1021/acschembio.0c00348,,,,
1624,BCR-ABL,,10.1021/acschembio.0c00348,,,,
1625,p38alpha,8/0 (WB),10.1016/j.ejmech.2020.112451,,,,% p38alpha degradation in BBL358/T47D cells after 24 h treatment at 10 μM
1626,p38alpha,40/0 (WB),10.1016/j.ejmech.2020.112451,,,,% p38alpha degradation in BBL358/T47D cells after 24 h treatment at 10 μM
1627,p38alpha,60/0 (WB),10.1016/j.ejmech.2020.112451,,,,% p38alpha degradation in BBL358/T47D cells after 24 h treatment at 10 μM
1628,p38alpha,55/0 (WB),10.1016/j.ejmech.2020.112451,,,,% p38alpha degradation in BBL358/T47D cells after 24 h treatment at 10 μM
1629,p38alpha,82/20 (WB),10.1016/j.ejmech.2020.112451,,,,% p38alpha degradation in BBL358/T47D cells after 24 h treatment at 10 μM
1630,p38alpha,78/26 (WB),10.1016/j.ejmech.2020.112451,,,,% p38alpha degradation in BBL358/T47D cells after 24 h treatment at 10 μM
1631,p38alpha,92/41 (WB),10.1016/j.ejmech.2020.112451,,,,% p38alpha degradation in BBL358/T47D cells after 24 h treatment at 10 μM
1632,p38alpha,79/85 (WB),10.1016/j.ejmech.2020.112451,,,,% p38alpha degradation in BBL358/T47D cells after 24 h treatment at 10 μM
1633,p38alpha,0.5/76 (WB),10.1016/j.ejmech.2020.112451,,,,% p38alpha degradation in BBL358/T47D cells after 24 h treatment at 10 μM
1634,p38alpha,67/47 (WB),10.1016/j.ejmech.2020.112451,,,,% p38alpha degradation in BBL358/T47D cells after 24 h treatment at 10 μM
1635,p38alpha,77/82 (WB),10.1016/j.ejmech.2020.112451,,,,% p38alpha degradation in BBL358/T47D cells after 24 h treatment at 10 μM
1636,p38alpha,,10.1016/j.ejmech.2020.112451,2.9/18.4,,Degradation of p38alpha in T47D/MB-MDA-231 cells after 24 h treatment,
1636,p38beta,,10.1016/j.ejmech.2020.112451,35.19/19.1,,Degradation of p38beta in T47D/MB-MDA-231 cells after 24 h treatment,
1637,p38alpha,74/16 (WB),10.1016/j.ejmech.2020.112451,,,,% p38alpha degradation in BBL358/T47D cells after 24 h treatment at 10 μM
1638,p38alpha,0/7 (WB),10.1016/j.ejmech.2020.112451,,,,% p38alpha degradation in BBL358/T47D cells after 24 h treatment at 10 μM
1639,p38alpha,36/42 (WB),10.1016/j.ejmech.2020.112451,,,,% p38alpha degradation in BBL358/T47D cells after 24 h treatment at 10 μM
1640,p38alpha,60/68 (WB),10.1016/j.ejmech.2020.112451,,,,% p38alpha degradation in BBL358/T47D cells after 24 h treatment at 10 μM
1641,p38alpha,40/25 (WB),10.1016/j.ejmech.2020.112451,,,,% p38alpha degradation in BBL358/T47D cells after 24 h treatment at 10 μM
1642,p38alpha,12/40 (WB),10.1016/j.ejmech.2020.112451,,,,% p38alpha degradation in BBL358/T47D cells after 24 h treatment at 10 μM
1643,p38alpha,84/91 (WB),10.1016/j.ejmech.2020.112451,,,,% p38alpha degradation in BBL358/T47D cells after 24 h treatment at 10 μM
1644,p38alpha,74/87 (WB),10.1016/j.ejmech.2020.112451,,,,% p38alpha degradation in BBL358/T47D cells after 24 h treatment at 10 μM
1645,p38alpha,,10.1016/j.ejmech.2020.112451,24/27.2,,Degradation of p38alpha in T47D/MB-MDA-231 cells after 24 h treatment,
1645,p38beta,,10.1016/j.ejmech.2020.112451,48.47/48.9,,Degradation of p38beta in T47D/MB-MDA-231 cells after 24 h treatment,
1646,p38alpha,81/93 (WB),10.1016/j.ejmech.2020.112451,,,,% p38alpha degradation in BBL358/T47D cells after 24 h treatment at 10 μM
1647,p38alpha,0/4 (WB),10.1016/j.ejmech.2020.112451,,,,% p38alpha degradation in BBL358/T47D cells after 24 h treatment at 10 μM
1648,BCR-ABL,,10.1039/d0cc02201b,30,,Degradation of BCR-ABL in K562 cells after 24 h treatment,
1649,BCL-xL,,10.1021/acschembio.0c00266,4.8,76,Degradation of BCL-xL in THP-1 cells after 24 h treatment,
1650,BTK,,10.1073/pnas.1803662115,9.6,,Degradation of BTK in Ramos cells after 24 h treatment,
1651,BRD4,,10.1021/acschembio.9b00092,,,,
1651,BRD2,,10.1021/acs.jmedchem.6b01912,,37,,
1651,BRD2,,10.1021/acschembio.9b00092,,,,
1651,BRD3,,10.1021/acschembio.9b00092,,,,
1651,BRD3,,10.1021/acs.jmedchem.6b01912,158,74,Degradation of BRD3 in HeLa cells after 24 h treatment,
1651,BRD4,,10.1021/acs.jmedchem.6b01912,126/200,94/78,Degradation of BRD4 short/long in HeLa cells after 24 h treatment,
1652,BRD2,,10.1021/acs.jmedchem.6b01912,,43,,
1652,BRD4,,10.1021/acs.jmedchem.6b01912,8/25,98/95,Degradation of BRD4 short/long in HeLa cells after 24 h treatment,
1652,BRD3,,10.1021/acs.jmedchem.6b01912,50,91,Degradation of BRD3 in HeLa cells after 24 h treatment,
1653,BRD4,,10.1021/acs.jmedchem.6b01912,8/32,95/93,Degradation of BRD4 short/long in HeLa cells after 24 h treatment,
1653,BRD3,,10.1021/acschembio.9b00092,,,,
1653,BRD4,,10.1021/acschembio.9b00092,,,,
1653,BRD3,,10.1021/acs.jmedchem.6b01912,20,92,Degradation of BRD3 in HeLa cells after 24 h treatment,
1653,BRD2,,10.1021/acs.jmedchem.6b01912,,26,,
1653,BRD2,,10.1021/acschembio.9b00092,,,,
1654,BRD4,,10.1021/acs.jmedchem.6b01912,100/100,96/97,Degradation of BRD4 short/long in HeLa cells after 24 h treatment,
1654,BRD3,,10.1021/acs.jmedchem.6b01912,316,97,Degradation of BRD3 in HeLa cells after 24 h treatment,
1654,BRD2,,10.1021/acs.jmedchem.6b01912,631,93,Degradation of BRD2 in HeLa cells after 24 h treatment,
1655,FAK,,10.1021/acs.jmedchem.8b01826,158/50/13,79/93/93,Degradation of Fak in HLE/HuH-7/SNU-423 cells after 18 h treatment,
1655,FAK,,10.1021/acs.jmedchem.8b01826,398/3/13,30/95/90,Degradation of Fak in HLF/SNU-398/HUCCT1 cells after 18 h treatment,
1655,FAK,,10.1021/acs.jmedchem.8b01826,27/13/25,95/96/90,Degradation of Fak in A549/Hep3B2.1-7/SNU-387 cells after 18 h treatment,
1655,FAK,,10.1021/acs.jmedchem.8b01826,251/32/32,50/89/89,Degradation of Fak in HUH-1/HepG2/SK-Hep-1 cells after 18 h treatment,
1656,FAK,,10.1021/acs.jmedchem.8b01826,79/631/126,79/65/87,Degradation of Fak in HUH-1/HepG2/SK-Hep-1 cells after 18 h treatment,
1656,FAK,,10.1021/acs.jmedchem.8b01826,243/631/32,80/59/98,Degradation of Fak in A549/Hep3B2.1-7/SNU-387 cells after 18 h treatment,
1656,FAK,,10.1021/acs.jmedchem.8b01826,25/100/79,85/79/87,Degradation of Fak in HLE/HuH-7/SNU-423 cells after 18 h treatment,
1656,FAK,,10.1021/acs.jmedchem.8b01826,40/10/126,66/99/86,Degradation of Fak in HLF/SNU-398/HUCCT1 cells after 18 h treatment,
1657,KRAS G12C,,10.1021/acscentsci.0c00411,,30,,
1658,KRAS G12C,,10.1021/acscentsci.0c00411,250/520,90/40,Degradation of KRAS G12C in NCI-H23/NCI-H358 cells after 24 h treatment,
1658,KRAS G12C,,10.1021/acscentsci.0c00411,590/320/760,80/75/90,Degradation of KRAS G12C in NCI-H2030/MIA PaCa-2/SW1573 cells after 24 h treatment,
1659,KRAS G12C,,10.1021/acscentsci.0c00411,640,85,Degradation of KRAS G12C in NCI-H2030 cells after 24 h treatment,
1660,KRAS G12C,,10.1021/acscentsci.0c00411,880,90,Degradation of KRAS G12C in SW1573 cells after 24 h treatment,
1661,KRAS G12C,,10.1021/acscentsci.0c00411,>10000,50,Degradation of KRAS G12C in SW1573 cells after 24 h treatment,
1662,KRAS G12C,,10.1021/acscentsci.0c00411,,35,,
1663,PARP1,,10.1021/acs.jmedchem.0c00821,,,,
1664,PARP1,,10.1021/acs.jmedchem.0c00821,,,,
1665,PARP1,,10.1021/acs.jmedchem.0c00821,,,,
1666,PARP1,,10.1021/acs.jmedchem.0c00821,,,,
1667,PARP1,,10.1021/acs.jmedchem.0c00821,,,,
1668,PARP1,,10.1021/acs.jmedchem.0c00821,,,,
1669,PARP1,,10.1021/acs.jmedchem.0c00821,,,,
1670,PARP1,,10.1021/acs.jmedchem.0c00821,,,,
1671,PARP1,,10.1021/acs.jmedchem.0c00821,,,,
1672,PARP1,,10.1021/acs.jmedchem.0c00821,,,,
1673,PARP1,3/49/97.9/91.2 (WB),10.1021/acs.jmedchem.0c00821,,,,% PARP1 degradation in MDA-MB-436 cells after 24 h treatment at 0.001/0.01/0.1/1 μM
1674,PARP1,9/98.7/100/99.7 (WB),10.1021/acs.jmedchem.0c00821,,,,% PARP1 degradation in MDA-MB-436 cells after 24 h treatment at 0.001/0.01/0.1/1 μM
1675,PARP1,,10.1021/acs.jmedchem.0c00821,0.578/1.08/0.228,>99/>99/>99,Degradation of PARP1 in PC-3/LNCaP/MDA-MB-231 cells after 24 h treatment,
1675,PARP1,,10.1021/acs.jmedchem.0c00821,0.384/0.512/0.263,>99/>99/>99,Degradation of PARP1 in HCC1937/22RV1/MDA-MB-468 cells after 24 h treatment,
1675,PARP1,,10.1021/acs.jmedchem.0c00821,1.26/6.72/0.509,>99/>99/>99,Degradation of PARP1 in MDA-MB-436/Capan-1/SW620 cells after 24 h treatment,
1676,PARP1,59/99.3/100/99.5 (WB),10.1021/acs.jmedchem.0c00821,,,,% PARP1 degradation in MDA-MB-436 cells after 24 h treatment at 0.001/0.01/0.1/1 μM
1677,PARP1,64/98.9/99.4/98.8 (WB),10.1021/acs.jmedchem.0c00821,,,,% PARP1 degradation in MDA-MB-436 cells after 24 h treatment at 0.001/0.01/0.1/1 μM
1678,PARP1,23/70/90.5/45 (WB),10.1021/acs.jmedchem.0c00821,,,,% PARP1 degradation in MDA-MB-436 cells after 24 h treatment at 0.001/0.01/0.1/1 μM
1679,PARP1,29/90/87/42 (WB),10.1021/acs.jmedchem.0c00821,,,,% PARP1 degradation in MDA-MB-436 cells after 24 h treatment at 0.001/0.01/0.1/1 μM
1680,PARP1,31/91.8/95.6/95.1 (WB),10.1021/acs.jmedchem.0c00821,,,,% PARP1 degradation in MDA-MB-436 cells after 24 h treatment at 0.001/0.01/0.1/1 μM
1681,PARP1,32/93.3/94.7/93.2 (WB),10.1021/acs.jmedchem.0c00821,,,,% PARP1 degradation in MDA-MB-436 cells after 24 h treatment at 0.001/0.01/0.1/1 μM
1682,PARP1,26/92.2/97.5/93.5 (WB),10.1021/acs.jmedchem.0c00821,,,,% PARP1 degradation in MDA-MB-436 cells after 24 h treatment at 0.001/0.01/0.1/1 μM
1683,PARP1,52/96.9/99.7/96 (WB),10.1021/acs.jmedchem.0c00821,,,,% PARP1 degradation in MDA-MB-436 cells after 24 h treatment at 0.001/0.01/0.1/1 μM
1684,PARP1,2/53/97.5/99.1 (WB),10.1021/acs.jmedchem.0c00821,,,,% PARP1 degradation in MDA-MB-436 cells after 24 h treatment at 0.001/0.01/0.1/1 μM
1685,PARP1,,10.1021/acs.jmedchem.0c00821,,,,
1686,PARP1,,10.1021/acs.jmedchem.0c00821,,,,
1687,PARP1,,10.1021/acs.jmedchem.0c00821,,,,
1688,PARP1,,10.1021/acs.jmedchem.0c00821,,,,
1689,TRKA,15/45/93,10.1021/acs.jmedchem.0c01342,,,,% TPM3-TRKA degradation in KM12 cells after 6 h treatment at 0.1/1/10 nM
1690,TRKA,9/15/65,10.1021/acs.jmedchem.0c01342,,,,% TPM3-TRKA degradation in KM12 cells after 6 h treatment at 0.1/1/10 nM
1691,TRKA,12/63/94,10.1021/acs.jmedchem.0c01342,,,,% TPM3-TRKA degradation in KM12 cells after 6 h treatment at 0.1/1/10 nM
1692,TRKA,20/69/93,10.1021/acs.jmedchem.0c01342,,,,% TPM3-TRKA degradation in KM12 cells after 6 h treatment at 0.1/1/10 nM
1693,TRKB,70/70/80/60 (WB),10.1021/acs.jmedchem.0c01342,,,,% AGBL4-TRKB degradation in KM12 cells after 6 h treatment at 19/56/167/500 nM
1693,TRKA,18/65/96,10.1021/acs.jmedchem.0c01342,0.48/1.26,,Degradation of TPM3-TRKA/TRKA in KM12/HEL cells after 6 h treatment,% TPM3-TRKA degradation in KM12 cells after 6 h treatment at 0.1/1/10 nM
1693,TRKC,30/40/60/60 (WB),10.1021/acs.jmedchem.0c01342,,,,% ETV6-TRKC degradation in KM12 cells after 6 h treatment at 19/56/167/500 nM
1694,TRKA,21/23/90,10.1021/acs.jmedchem.0c01342,,,,% TPM3-TRKA degradation in KM12 cells after 6 h treatment at 0.1/1/10 nM
1695,TRKA,20/21/83,10.1021/acs.jmedchem.0c01342,,,,% TPM3-TRKA degradation in KM12 cells after 6 h treatment at 0.1/1/10 nM
1696,TRKB,50/50/50/30 (WB),10.1021/acs.jmedchem.0c01342,,,,% AGBL4-TRKB degradation in KM12 cells after 6 h treatment at 19/56/167/500 nM
1696,TRKA,46/82/96,10.1021/acs.jmedchem.0c01342,0.36/2.23,,Degradation of TPM3-TRKA/TRKA in KM12/HEL cells after 6 h treatment,% TPM3-TRKA degradation in KM12 cells after 6 h treatment at 0.1/1/10 nM
1696,TRKC,20/60/60/60 (WB),10.1021/acs.jmedchem.0c01342,,,,% ETV6-TRKC degradation in KM12 cells after 6 h treatment at 19/56/167/500 nM
1697,TRKA,30/56/95,10.1021/acs.jmedchem.0c01342,,,,% TPM3-TRKA degradation in KM12 cells after 6 h treatment at 0.1/1/10 nM
1698,TRKA,22/28/86,10.1021/acs.jmedchem.0c01342,,,,% TPM3-TRKA degradation in KM12 cells after 6 h treatment at 0.1/1/10 nM
1699,TRKA,22/40/91,10.1021/acs.jmedchem.0c01342,,,,% TPM3-TRKA degradation in KM12 cells after 6 h treatment at 0.1/1/10 nM
1700,IRAK3,,10.1021/acs.jmedchem.0c01125,,,,
1701,IRAK3,,10.1021/acs.jmedchem.0c01125,,,,
1702,IRAK3,,10.1021/acs.jmedchem.0c01125,,,,
1703,IRAK3,,10.1021/acs.jmedchem.0c01125,,,,
1704,IRAK3,,10.1021/acs.jmedchem.0c01125,,,,
1705,IRAK3,,10.1021/acs.jmedchem.0c01125,,,,
1706,IRAK3,,10.1021/acs.jmedchem.0c01125,,,,
1707,IRAK3,,10.1021/acs.jmedchem.0c01125,,,,
1708,IRAK3,,10.1021/acs.jmedchem.0c01125,,,,
1709,IRAK3,,10.1021/acs.jmedchem.0c01125,,,,
1710,IRAK3,,10.1021/acs.jmedchem.0c01125,,,,
1711,IRAK3,,10.1021/acs.jmedchem.0c01125,,,,
1712,IRAK3,,10.1021/acs.jmedchem.0c01125,,,,
1713,IRAK3,,10.1021/acs.jmedchem.0c01125,,,,
1714,IRAK3,,10.1021/acs.jmedchem.0c01125,,,,
1715,IRAK3,,10.1021/acs.jmedchem.0c01125,,,,
1716,IRAK3,,10.1021/acs.jmedchem.0c01125,52,74,Degradation of IRAK3 in THP1 cells after 16 h treatment,
1717,IRAK3,,10.1021/acs.jmedchem.0c01125,2,98,Degradation of IRAK3 in THP1 cells after 16 h treatment,
1718,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1718,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1719,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1719,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1720,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1720,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1721,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1721,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1722,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1722,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1723,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1723,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1724,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1724,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1725,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1725,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1726,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1726,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1727,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1727,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1728,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1728,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1729,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1729,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1730,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1730,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1731,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1731,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1732,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1732,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1733,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1733,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1734,MEK1,,10.1021/acs.jmedchem.0c01609,18/16,,Degradation of MEK1 in HT-29/SK-MEL-28 cells after 24 h treatment,
1734,MEK2,,10.1021/acs.jmedchem.0c01609,8/6,,Degradation of MEK2 in HT-29/SK-MEL-28 cells after 24 h treatment,
1735,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1735,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1736,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1736,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1737,MEK2,,10.1021/acs.jmedchem.0c01609,9/4,,Degradation of MEK2 in HT-29/SK-MEL-28 cells after 24 h treatment,
1737,MEK1,,10.1021/acs.jmedchem.0c01609,18/10,,Degradation of MEK1 in HT-29/SK-MEL-28 cells after 24 h treatment,
1738,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1738,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1739,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1739,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1740,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1740,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1741,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1741,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1742,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1742,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1743,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1743,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1744,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1744,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1745,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1745,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1746,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1746,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1747,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1747,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1748,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1748,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1749,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1749,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1750,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1750,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1751,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1751,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1752,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1752,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1753,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1753,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1754,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1754,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1755,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1755,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1756,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1756,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1757,MEK1,,10.1021/acs.jmedchem.0c01609,,,,
1757,MEK2,,10.1021/acs.jmedchem.0c01609,,,,
1758,MEK2,,10.1021/acs.jmedchem.0c01609,55/38,,Degradation of MEK2 in HT-29/SK-MEL-28 cells after 24 h treatment,
1758,MEK1,,10.1021/acs.jmedchem.0c01609,118/94,,Degradation of MEK1 in HT-29/SK-MEL-28 cells after 24 h treatment,
1759,EZH2,,10.1021/acs.jmedchem.0c02234,,,,
1760,EZH2,,10.1021/acs.jmedchem.0c02234,,,,
1761,EZH2,,10.1021/acs.jmedchem.0c02234,,,,
1762,EZH2,,10.1021/acs.jmedchem.0c02234,,,,
1763,EZH2,,10.1021/acs.jmedchem.0c02234,,,,
1764,EZH2,,10.1021/acs.jmedchem.0c02234,,,,
1765,EZH2,,10.1021/acs.jmedchem.0c02234,,,,
1766,EZH2,,10.1021/acs.jmedchem.0c02234,,,,
1767,EZH2,,10.1021/acs.jmedchem.0c02234,,,,
1768,EZH2,,10.1021/acs.jmedchem.0c02234,,,,
1769,EZH2,,10.1021/acs.jmedchem.0c02234,,,,
1770,EZH2,,10.1021/acs.jmedchem.0c02234,,,,
1771,EZH2,,10.1021/acs.jmedchem.0c02234,,,,
1772,EZH2,,10.1021/acs.jmedchem.0c02234,,,,
1773,EZH2,,10.1021/acs.jmedchem.0c02234,,,,
1774,EZH2,,10.1021/acs.jmedchem.0c02234,,,,
1775,EZH2,,10.1021/acs.jmedchem.0c02234,,,,
1776,EZH2,,10.1021/acs.jmedchem.0c02234,,,,
1777,PRMT5,0/0/0 (WB),10.1021/acs.jmedchem.0c01111,,,,% PRMT5 degradation in MCF-7 cells after 6 d treatment at 0.2/1/5 μM
1778,PRMT5,0/0/0 (WB),10.1021/acs.jmedchem.0c01111,,,,% PRMT5 degradation in MCF-7 cells after 6 d treatment at 0.2/1/5 μM
1779,PRMT5,0/13/19 (WB),10.1021/acs.jmedchem.0c01111,,,,% PRMT5 degradation in MCF-7 cells after 6 d treatment at 0.2/1/5 μM
1780,PRMT5,13/27/14 (WB),10.1021/acs.jmedchem.0c01111,,,,% PRMT5 degradation in MCF-7 cells after 6 d treatment at 0.2/1/5 μM
1781,PRMT5,17/39/67 (WB),10.1021/acs.jmedchem.0c01111,,,,% PRMT5 degradation in MCF-7 cells after 6 d treatment at 0.2/1/5 μM
1782,PRMT5,,10.1021/acs.jmedchem.0c01111,1100,74,Degradation of PRMT5 in MCF-7 cells after 6 d treatment,
1783,BRD4,,10.1021/acs.jmedchem.0c01846,7.5,98,Degradation of BRD4 in PC3-S1 cells after 4 h treatment,
1784,BRD4,,10.1021/acs.jmedchem.0c01846,0.095,96,Degradation of BRD4 in PC3-S1 cells after 4 h treatment,
1785,BRD4,,10.1021/acs.jmedchem.0c01846,180,99,Degradation of BRD4 in PC3-S1 cells after 4 h treatment,
1786,BRD4,,10.1021/acs.jmedchem.0c01846,3.4,98,Degradation of BRD4 in PC3-S1 cells after 4 h treatment,
1787,BRD4,,10.1021/acs.jmedchem.0c01846,2.1,98,Degradation of BRD4 in EOL-1 cells 4 h treatment,
1788,BRD4,,10.1021/acs.jmedchem.0c01846,1.4,100,Degradation of BRD4 in PC3-S1 cells after 4 h treatment,
1789,BRD4,,10.1021/acs.jmedchem.0c01845,>20000,,Degradation of BRD4 in PC3-S1 cells after 4 h treatment,
1790,BRD4,,10.1021/acs.jmedchem.0c01845,930,79,Degradation of BRD4 in PC3-S1 cells after 4 h treatment,
1791,BRD4,,10.1021/acs.jmedchem.0c01845,780,99,Degradation of BRD4 in PC3-S1 cells after 4 h treatment,
1792,BRD4,,10.1021/acs.jmedchem.0c01845,350,100,Degradation of BRD4 in PC3-S1 cells after 4 h treatment,
1793,BRD4,,10.1021/acs.jmedchem.0c01845,85,98,Degradation of BRD4 in PC3-S1 cells after 4 h treatment,
1794,BRD4,,10.1021/acs.jmedchem.0c01845,280,88,Degradation of BRD4 in PC3-S1 cells after 4 h treatment,
1795,BRD4,,10.1021/acs.jmedchem.0c01845,87,100,Degradation of BRD4 in PC3-S1 cells after 4 h treatment,
1796,BRD4,,10.1021/acs.jmedchem.0c01845,6500,100,Degradation of BRD4 in PC3-S1 cells after 4 h treatment,
1797,BRD4,,10.1021/acs.jmedchem.0c01845,7.2,99,Degradation of BRD4 in PC3-S1 cells after 4 h treatment,
1798,IRAK4,,10.1021/acsmedchemlett.0c00474,,,,
1799,IRAK4,,10.1021/acsmedchemlett.0c00474,,,,
1800,IRAK4,,10.1021/acsmedchemlett.0c00474,,,,
1801,IRAK4,,10.1021/acsmedchemlett.0c00474,,,,
1802,IRAK4,,10.1021/acsmedchemlett.0c00474,,,,
1803,IRAK4,,10.1021/acsmedchemlett.0c00474,,,,
1804,IRAK4,,10.1021/acsmedchemlett.0c00474,,,,
1805,IRAK4,,10.1021/acsmedchemlett.0c00474,,,,
1806,FAK,37/71,10.1021/acsmedchemlett.9b00372,,,,% FAK degradation in PA1 cells after 8 h treatment at 1/10 nM
1807,FAK,32/60,10.1021/acsmedchemlett.9b00372,,,,% FAK degradation in PA1 cells after 8 h treatment at 1/10 nM
1808,FAK,5/22,10.1021/acsmedchemlett.9b00372,,,,% FAK degradation in PA1 cells after 8 h treatment at 1/10 nM
1809,FAK,55/81,10.1021/acsmedchemlett.9b00372,,,,% FAK degradation in PA1 cells after 8 h treatment at 1/10 nM
1810,FAK,40/65,10.1021/acsmedchemlett.9b00372,,,,% FAK degradation in PA1 cells after 8 h treatment at 1/10 nM
1811,FAK,10/30,10.1021/acsmedchemlett.9b00372,,,,% FAK degradation in PA1 cells after 8 h treatment at 1/10 nM
1812,FAK,32/90,10.1021/acsmedchemlett.9b00372,,,,% FAK degradation in PA1 cells after 8 h treatment at 1/10 nM
1813,FAK,71/96,10.1021/acsmedchemlett.9b00372,,,,% FAK degradation in PA1 cells after 8 h treatment at 1/10 nM
1814,FAK,35/92,10.1021/acsmedchemlett.9b00372,,,,% FAK degradation in PA1 cells after 8 h treatment at 1/10 nM
1815,FAK,40/92,10.1021/acsmedchemlett.9b00372,,,,% FAK degradation in PA1 cells after 8 h treatment at 1/10 nM
1816,FAK,46/94,10.1021/acsmedchemlett.9b00372,,,,% FAK degradation in PA1 cells after 8 h treatment at 1/10 nM
1817,FAK,30/82,10.1021/acsmedchemlett.9b00372,,,,% FAK degradation in PA1 cells after 8 h treatment at 1/10 nM
1818,FAK,67/93,10.1021/acsmedchemlett.9b00372,,,,% FAK degradation in PA1 cells after 8 h treatment at 1/10 nM
1819,FAK,62/90,10.1021/acsmedchemlett.9b00372,,,,% FAK degradation in PA1 cells after 8 h treatment at 1/10 nM
1820,FAK,62/90,10.1021/acsmedchemlett.9b00372,,,,% FAK degradation in PA1 cells after 8 h treatment at 1/10 nM
1821,FAK,62/90,10.1021/acsmedchemlett.9b00372,,,,% FAK degradation in PA1 cells after 8 h treatment at 1/10 nM
1822,FAK,85/95,10.1021/acsmedchemlett.9b00372,,,,% FAK degradation in PA1 cells after 8 h treatment at 1/10 nM
1823,FAK,62/90,10.1021/acsmedchemlett.9b00372,,,,% FAK degradation in PA1 cells after 8 h treatment at 1/10 nM
1824,FAK,40/85,10.1021/acsmedchemlett.9b00372,,,,% FAK degradation in PA1 cells after 8 h treatment at 1/10 nM
1825,SIRT2,61/47/15 (WB),10.1021/acsmedchemlett.0c00423,,,,% SIRT2 degradation in MCF7 cells after 48 h treatment at 5/10/25 μM
1826,SIRT2,71/38/13 (WB),10.1021/acsmedchemlett.0c00423,,,,% SIRT2 degradation in MCF7 cells after 48 h treatment at 5/10/25 μM
1827,HPGDS,,10.1021/acsmedchemlett.0c00605,,,,
1828,HPGDS,,10.1021/acsmedchemlett.0c00605,,N.D.,,
1829,IDO1,,10.1016/j.apsb.2020.02.010,,N.D.,,
1830,IDO1,,10.1016/j.apsb.2020.02.010,,N.D.,,
1831,IDO1,,10.1016/j.apsb.2020.02.010,,N.D.,,
1832,IDO1,,10.1016/j.apsb.2020.02.010,,N.D.,,
1833,IDO1,,10.1016/j.apsb.2020.02.010,,N.D.,,
1834,IDO1,,10.1016/j.apsb.2020.02.010,2840,93,Degradation of IDO1 in HeLa cells after 24 h treatment,
1835,IDO1,,10.1016/j.apsb.2020.02.010,,N.D.,,
1836,SHP2,,10.1016/j.bioorg.2021.104788,,,,
1837,SHP2,,10.1016/j.bioorg.2021.104788,,,,
1838,SHP2,,10.1016/j.bioorg.2021.104788,,,,
1839,SHP2,,10.1016/j.bioorg.2021.104788,,,,
1840,ADRA1A,,10.1016/j.apsb.2020.01.014,4320,,Degradation of ADRA1A in HEK293 cells after 12 h treatment,
1841,ADRA1A,,10.1016/j.apsb.2020.01.014,,,,
1842,ADRA1A,,10.1016/j.apsb.2020.01.014,2860,94,Degradation of ADRA1A in HEK293 cells after 12 h treatment,
1843,HDAC1,,10.1002/anie.202006725,,,,
1843,HDAC6,,10.1002/anie.202006725,,,,
1843,HDAC2,,10.1002/anie.202006725,,,,
1843,HDAC3,,10.1002/anie.202006725,,,,
1844,CD147,,10.1016/j.bioorg.2020.104453,>40000,,Degradation of CD147 in Sk-Mel-28 cells after 6 h treatment,
1845,CD147,,10.1016/j.bioorg.2020.104453,13850,,Degradation of CD147 in Sk-Mel-28 cells after 6 h treatment,
1846,CD147,,10.1016/j.bioorg.2020.104453,>40000,,Degradation of CD147 in Sk-Mel-28 cells after 6 h treatment,
1847,CD147,,10.1016/j.bioorg.2020.104453,>40000,,Degradation of CD147 in Sk-Mel-28 cells after 6 h treatment,
1848,CD147,,10.1016/j.bioorg.2020.104453,>40000,,Degradation of CD147 in Sk-Mel-28 cells after 6 h treatment,
1849,CD147,,10.1016/j.bioorg.2020.104453,>40000,,Degradation of CD147 in Sk-Mel-28 cells after 6 h treatment,
1850,CD147,,10.1016/j.bioorg.2020.104453,>40000,,Degradation of CD147 in Sk-Mel-28 cells after 6 h treatment,
1851,CD147,,10.1016/j.bioorg.2020.104453,>40000,,Degradation of CD147 in Sk-Mel-28 cells after 6 h treatment,
1852,CD147,,10.1016/j.bioorg.2020.104453,6720,,Degradation of CD147 in Sk-Mel-28 cells after 6 h treatment,
1853,CD147,,10.1016/j.bioorg.2020.104453,>40000,,Degradation of CD147 in Sk-Mel-28 cells after 6 h treatment,
1854,CD147,,10.1016/j.bioorg.2020.104453,>40000,,Degradation of CD147 in Sk-Mel-28 cells after 6 h treatment,
1855,CD147,,10.1016/j.bioorg.2020.104453,>40000,,Degradation of CD147 in Sk-Mel-28 cells after 6 h treatment,
1856,CD147,,10.1016/j.bioorg.2020.104453,>40000,,Degradation of CD147 in Sk-Mel-28 cells after 6 h treatment,
1857,CD147,,10.1016/j.bioorg.2020.104453,16840,,Degradation of CD147 in Sk-Mel-28 cells after 6 h treatment,
1858,CD147,,10.1016/j.bioorg.2020.104453,>40000,,Degradation of CD147 in Sk-Mel-28 cells after 6 h treatment,
1859,HDAC3,,10.1016/j.ejmech.2020.112800,,,,
1860,HDAC3,,10.1016/j.ejmech.2020.112800,,,,
1861,HDAC2,,10.1016/j.ejmech.2020.112800,,,,
1862,HDAC3,,10.1016/j.ejmech.2020.112800,,,,
1863,HDAC3,,10.1016/j.ejmech.2020.112800,,,,
1863,HDAC2,,10.1016/j.ejmech.2020.112800,,,,
1864,HDAC3,,10.1016/j.ejmech.2020.112800,,,,
1865,HDAC3,,10.1016/j.ejmech.2020.112800,320,,Degradation of HDAC3 in RAW 264.7 cells after 24 h treatment,
1866,AR,,10.1016/j.ejmech.2021.113307,,,,
1867,AR,,10.1016/j.ejmech.2021.113307,,,,
1868,AR,,10.1016/j.ejmech.2021.113307,,,,
1869,AR,,10.1016/j.ejmech.2021.113307,,,,
1870,AR,,10.1016/j.ejmech.2021.113307,,,,
1871,AR,,10.1016/j.ejmech.2021.113307,,,,
1872,AR,,10.1016/j.ejmech.2021.113307,,,,
1873,AR,,10.1016/j.ejmech.2021.113307,,,,
1874,AR,,10.1016/j.ejmech.2021.113307,,,,
1875,AR,,10.1016/j.ejmech.2021.113307,,,,
1876,AR,,10.1016/j.ejmech.2021.113307,,,,
1877,AR,,10.1016/j.ejmech.2021.113307,,,,
1878,AR,,10.1016/j.ejmech.2021.113307,,,,
1879,AR,,10.1016/j.ejmech.2021.113307,,,,
1880,AR,,10.1016/j.ejmech.2021.113307,,,,
1881,AR,,10.1016/j.ejmech.2021.113307,,,,
1882,AR,,10.1016/j.ejmech.2021.113307,,,,
1883,AR,,10.1016/j.ejmech.2021.113307,,,,
1884,AR,,10.1016/j.ejmech.2021.113307,,,,
1885,AR,,10.1016/j.ejmech.2021.113307,,,,
1886,AR,,10.1016/j.ejmech.2021.113307,,,,
1887,AR,,10.1016/j.ejmech.2021.113307,,,,
1888,AR,,10.1016/j.ejmech.2021.113307,,,,
1889,AR,,10.1016/j.ejmech.2021.113307,,,,
1890,AR,,10.1016/j.ejmech.2021.113307,,,,
1891,AR,,10.1016/j.ejmech.2021.113307,,,,
1892,AR,,10.1016/j.ejmech.2021.113307,,,,
1893,AR,,10.1016/j.ejmech.2021.113307,,,,
1894,AR,,10.1016/j.ejmech.2021.113307,,,,
1895,AR,,10.1016/j.ejmech.2021.113307,,,,
1896,AR,,10.1016/j.ejmech.2021.113307,,,,
1897,AR,,10.1016/j.ejmech.2021.113307,,,,
1898,GSK-3beta,,10.1016/j.ejmech.2020.112949,,,,
1899,GSK-3beta,,10.1016/j.ejmech.2020.112949,,,,
1900,GSK-3beta,,10.1016/j.ejmech.2020.112949,,,,
1901,GSK-3beta,,10.1016/j.ejmech.2020.112949,,,,
1902,GSK-3beta,,10.1016/j.ejmech.2020.112949,,,,
1903,GSK-3beta,,10.1016/j.ejmech.2020.112949,,,,
1904,GSK-3beta,,10.1016/j.ejmech.2020.112949,,,,
1905,GSK-3beta,,10.1016/j.ejmech.2020.112949,,,,
1906,GSK-3beta,,10.1016/j.ejmech.2020.112949,,,,
1907,GSK-3beta,,10.1016/j.ejmech.2020.112949,,,,
1908,GSK-3beta,,10.1016/j.ejmech.2020.112949,,,,
1909,GSK-3beta,,10.1016/j.ejmech.2020.112949,,,,
1910,GSK-3beta,,10.1016/j.ejmech.2020.112949,,,,
1911,GSK-3beta,,10.1016/j.ejmech.2020.112949,,,,
1912,GSK-3beta,,10.1016/j.ejmech.2020.112949,,,,
1913,GSK-3beta,,10.1016/j.ejmech.2020.112949,,,,
1914,GSK-3beta,,10.1016/j.ejmech.2020.112949,,,,
1915,GSK-3beta,,10.1016/j.ejmech.2020.112949,,,,
1916,GSK-3beta,,10.1016/j.ejmech.2020.112949,,,,
1917,GSK-3beta,,10.1016/j.ejmech.2020.112949,,,,
1918,GSK-3beta,,10.1016/j.ejmech.2020.112949,,,,
1919,EEF2K,,10.1016/j.ejmech.2020.112505,,,,
1920,EEF2K,,10.1016/j.ejmech.2020.112505,,,,
1921,EEF2K,,10.1016/j.ejmech.2020.112505,,,,
1922,EEF2K,,10.1016/j.ejmech.2020.112505,,,,
1923,EEF2K,,10.1016/j.ejmech.2020.112505,,,,
1924,EEF2K,,10.1016/j.ejmech.2020.112505,,,,
1925,EEF2K,,10.1016/j.ejmech.2020.112505,,,,
1926,EEF2K,,10.1016/j.ejmech.2020.112505,,,,
1927,EEF2K,,10.1016/j.ejmech.2020.112505,,,,
1928,EEF2K,,10.1016/j.ejmech.2020.112505,,,,
1929,EEF2K,,10.1016/j.ejmech.2020.112505,,,,
1930,EEF2K,,10.1016/j.ejmech.2020.112505,,,,
1931,EEF2K,,10.1016/j.ejmech.2020.112505,,,,
1932,EEF2K,,10.1016/j.ejmech.2020.112505,,,,
1933,EEF2K,,10.1016/j.ejmech.2020.112505,,,,
1934,EEF2K,,10.1016/j.ejmech.2020.112505,,,,
1935,EEF2K,,10.1016/j.ejmech.2020.112505,,,,
1936,EEF2K,,10.1016/j.ejmech.2020.112505,,,,
1937,EEF2K,,10.1016/j.ejmech.2020.112505,,,,
1938,EEF2K,,10.1016/j.ejmech.2020.112505,,,,
1939,EEF2K,,10.1016/j.ejmech.2020.112505,,,,
1940,EEF2K,,10.1016/j.ejmech.2020.112505,,,,
1941,EEF2K,,10.1016/j.ejmech.2020.112505,,,,
1942,EEF2K,,10.1016/j.ejmech.2020.112505,,56.7,,
1943,VEGFR-2,,10.1016/j.ejmech.2020.112654,,,,
1944,VEGFR-2,,10.1016/j.ejmech.2020.112654,,,,
1945,VEGFR-2,,10.1016/j.ejmech.2020.112654,,,,
1946,VEGFR-2,,10.1016/j.ejmech.2020.112654,,,,
1947,VEGFR-2,,10.1016/j.ejmech.2020.112654,,,,
1948,VEGFR-2,,10.1016/j.ejmech.2020.112654,,,,
1949,CDK6,,10.1016/j.ejmech.2020.112903,,,,
1949,CDK4,,10.1016/j.ejmech.2020.112903,,,,
1949,CDK2,,10.1016/j.ejmech.2020.112903,,,,
1950,CDK6,,10.1016/j.ejmech.2020.112903,,,,
1950,CDK4,,10.1016/j.ejmech.2020.112903,,,,
1950,CDK2,,10.1016/j.ejmech.2020.112903,,,,
1951,CDK6,,10.1016/j.ejmech.2020.112903,,,,
1951,CDK2,,10.1016/j.ejmech.2020.112903,,,,
1951,CDK4,,10.1016/j.ejmech.2020.112903,,,,
1952,CDK2,,10.1016/j.ejmech.2020.112903,,,,
1952,CDK4,,10.1016/j.ejmech.2020.112903,,,,
1952,CDK6,,10.1016/j.ejmech.2020.112903,,,,
1953,CDK4,,10.1016/j.ejmech.2020.112903,,,,
1953,CDK6,,10.1016/j.ejmech.2020.112903,,,,
1953,CDK2,,10.1016/j.ejmech.2020.112903,,,,
1954,CDK6,,10.1016/j.ejmech.2020.112903,,,,
1954,CDK2,,10.1016/j.ejmech.2020.112903,,,,
1954,CDK4,,10.1016/j.ejmech.2020.112903,,,,
1955,CDK4,,10.1016/j.ejmech.2020.112903,,,,
1955,CDK6,,10.1016/j.ejmech.2020.112903,,,,
1955,CDK2,,10.1016/j.ejmech.2020.112903,,,,
1956,CDK6,,10.1016/j.ejmech.2020.112903,,,,
1956,CDK2,,10.1016/j.ejmech.2020.112903,,,,
1956,CDK4,,10.1016/j.ejmech.2020.112903,,,,
1957,CDK4,,10.1016/j.ejmech.2020.112903,,,,
1957,CDK2,,10.1016/j.ejmech.2020.112903,,,,
1957,CDK6,,10.1016/j.ejmech.2020.112903,,,,
1958,CDK4,,10.1016/j.ejmech.2020.112903,,,,
1958,CDK6,,10.1016/j.ejmech.2020.112903,,,,
1958,CDK2,,10.1016/j.ejmech.2020.112903,,,,
1959,CDK4,,10.1016/j.ejmech.2020.112903,,,,
1959,CDK2,,10.1016/j.ejmech.2020.112903,,,,
1959,CDK6,,10.1016/j.ejmech.2020.112903,,,,
1960,CDK4,,10.1016/j.ejmech.2020.112903,,,,
1960,CDK2,,10.1016/j.ejmech.2020.112903,,,,
1960,CDK6,,10.1016/j.ejmech.2020.112903,,,,
1961,CDK4,,10.1016/j.ejmech.2020.112903,,,,
1961,CDK6,,10.1016/j.ejmech.2020.112903,,,,
1961,CDK2,,10.1016/j.ejmech.2020.112903,,,,
1962,CDK4,,10.1016/j.ejmech.2020.112903,,,,
1962,CDK6,,10.1016/j.ejmech.2020.112903,,,,
1962,CDK2,,10.1016/j.ejmech.2020.112903,,,,
1963,CDK2,,10.1016/j.ejmech.2020.112903,,,,
1963,CDK4,,10.1016/j.ejmech.2020.112903,,,,
1963,CDK6,,10.1016/j.ejmech.2020.112903,,,,
1964,CDK2,,10.1016/j.ejmech.2020.112903,,,,
1964,CDK4,,10.1016/j.ejmech.2020.112903,,,,
1964,CDK6,,10.1016/j.ejmech.2020.112903,,,,
1965,CDK6,,10.1016/j.ejmech.2020.112903,,,,
1965,CDK4,,10.1016/j.ejmech.2020.112903,,,,
1965,CDK2,,10.1016/j.ejmech.2020.112903,,,,
1966,CDK4,,10.1016/j.ejmech.2020.112903,,,,
1966,CDK6,,10.1016/j.ejmech.2020.112903,,,,
1966,CDK2,,10.1016/j.ejmech.2020.112903,,,,
1967,CDK6,,10.1016/j.ejmech.2020.112903,,,,
1967,CDK2,,10.1016/j.ejmech.2020.112903,,,,
1967,CDK4,,10.1016/j.ejmech.2020.112903,,,,
1968,CDK6,,10.1016/j.ejmech.2020.112903,,,,
1968,CDK2,,10.1016/j.ejmech.2020.112903,,,,
1968,CDK4,,10.1016/j.ejmech.2020.112903,,,,
1969,CDK2,,10.1016/j.ejmech.2020.112903,,,,
1969,CDK4,,10.1016/j.ejmech.2020.112903,,,,
1969,CDK6,,10.1016/j.ejmech.2020.112903,,,,
1970,ALK,,10.1016/j.ejmech.2020.113150,,,,
1971,ALK,,10.1016/j.ejmech.2020.113150,,,,
1972,ALK,,10.1016/j.ejmech.2020.113150,,,,
1973,ALK,,10.1016/j.ejmech.2020.113150,,,,
1974,ALK,,10.1016/j.ejmech.2020.113150,,,,
1975,ALK,,10.1016/j.ejmech.2020.113150,,,,
1976,ALK,,10.1016/j.ejmech.2020.113150,,,,
1977,ALK,,10.1016/j.ejmech.2020.113150,,,,
1978,ALK,,10.1016/j.ejmech.2020.113150,,,,
1979,ALK,,10.1016/j.ejmech.2020.113150,,,,
1980,ALK,,10.1016/j.ejmech.2020.113150,,,,
1981,ALK,,10.1016/j.ejmech.2020.113150,,,,
1982,ALK,,10.1016/j.ejmech.2020.113150,,,,
1983,ALK,,10.1016/j.ejmech.2020.113150,,,,
1984,ALK,,10.1016/j.ejmech.2020.113150,,,,
1985,ALK,,10.1016/j.ejmech.2020.113150,,,,
1986,ALK,,10.1016/j.ejmech.2020.113150,,,,
1987,ALK,,10.1016/j.ejmech.2020.113150,,,,
1988,ALK,,10.1016/j.ejmech.2020.113150,,,,
1989,ALK,,10.1016/j.ejmech.2020.113150,,,,
1990,ALK,,10.1016/j.ejmech.2020.113150,,,,
1991,ALK,,10.1016/j.ejmech.2020.113150,,,,
1992,ALK,,10.1016/j.ejmech.2020.113150,,,,
1993,EGFR e19d,,10.1016/j.ejmech.2020.112781,,,,
1993,EGFR,,10.1016/j.ejmech.2020.112781,,,,
1993,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112781,,,,
1994,EGFR e19d,,10.1016/j.ejmech.2020.112781,,,,
1994,EGFR,,10.1016/j.ejmech.2020.112781,,,,
1994,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112781,,,,
1995,EGFR e19d,,10.1016/j.ejmech.2020.112781,0.51,80.4,Degradation of EGFR del19 in HCC827 cells after 48 h treatment,
1995,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112781,126.2,90.3,Degradation of EGFR L858R/T790M in H1975 cells after 48 h treatment,
1995,EGFR,,10.1016/j.ejmech.2020.112781,,N.D.,,
1996,EGFR e19d,,10.1016/j.ejmech.2020.112781,3.54,74.8,Degradation of EGFR del19 in HCC827 cells after 48 h treatment,
1996,EGFR,,10.1016/j.ejmech.2020.112781,,,,
1996,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112781,151.2,80.3,Degradation of EGFR L858R/T790M in H1975 cells after 48 h treatment,
1997,EGFR,,10.1016/j.ejmech.2020.112781,,,,
1997,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112781,,,,
1997,EGFR e19d,,10.1016/j.ejmech.2020.112781,,,,
1998,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112781,,,,
1998,EGFR,,10.1016/j.ejmech.2020.112781,,N.D.,,
1998,EGFR e19d,,10.1016/j.ejmech.2020.112781,1.91,82,Degradation of EGFR del19 in HCC827 cells after 48 h treatment,
1999,EGFR e19d,,10.1016/j.ejmech.2020.112781,,,,
1999,EGFR,,10.1016/j.ejmech.2020.112781,,,,
1999,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112781,,,,
2000,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112781,,,,
2000,EGFR e19d,,10.1016/j.ejmech.2020.112781,,,,
2000,EGFR,,10.1016/j.ejmech.2020.112781,,,,
2001,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112781,,,,
2001,EGFR e19d,,10.1016/j.ejmech.2020.112781,,,,
2001,EGFR,,10.1016/j.ejmech.2020.112781,,,,
2002,EGFR,,10.1016/j.ejmech.2020.112781,,,,
2002,EGFR L858R/T790M,,10.1016/j.ejmech.2020.112781,,,,
2002,EGFR e19d,,10.1016/j.ejmech.2020.112781,,,,
2003,CBP,,10.1016/j.chembiol.2020.12.004,,,,
2003,EP300,,10.1016/j.chembiol.2020.12.004,,,,
2004,IRAK4,,10.1016/j.chembiol.2020.08.010,,46,,
2005,IRAK4,,10.1016/j.chembiol.2020.08.010,485,92,Degradation of IRAK4 in HEK293T cells after 24 h treatment,
2006,IRAK4,,10.1016/j.chembiol.2020.08.010,190,93,Degradation of IRAK4 in HEK293T cells after 24 h treatment,
2007,IRAK4,,10.1016/j.chembiol.2020.08.010,293,97,Degradation of IRAK4 in HEK293T cells after 24 h treatment,
2008,IRAK4,,10.1016/j.chembiol.2020.08.010,405,90,Degradation of IRAK4 in HEK293T cells after 24 h treatment,
2009,IRAK4,,10.1016/j.chembiol.2020.08.010,7420,71,Degradation of IRAK4 in HEK293T cells after 24 h treatment,
2010,IRAK4,,10.1016/j.chembiol.2020.08.010,,47,,
2011,IRAK4,,10.1016/j.chembiol.2020.08.010,,30,,
2012,HDAC3,,10.1039/d0cc03243c,,,,
2013,HDAC3,,10.1039/d0cc03243c,,,,
2014,HDAC3,,10.1039/d0cc03243c,,,,
2015,HDAC3,74/72 (WB),10.1039/d0cc03243c,,,,% HDAC3 degradation in MDA-MB-468 cells after 14 h treatment at 0.1/1 μM
2016,HDAC3,72/84 (WB),10.1039/d0cc03243c,,,,% HDAC3 degradation in MDA-MB-468 cells after 14 h treatment at 0.1/1 μM
2017,HDAC3,,10.1039/d0cc03243c,42,,Degradation of HDAC3 in MDA-MB-468 cells after 14 h treatment,
2018,HDAC3,41/56 (WB),10.1039/d0cc03243c,,,,% HDAC3 degradation in MDA-MB-468 cells after 14 h treatment at 0.1/1 μM
2019,CDK6,,10.1039/d0sc00167h,,,,
2019,CDK4,,10.1039/d0sc00167h,,,,
2020,CDK6,,10.1039/d0sc00167h,,,,
2020,CDK4,,10.1039/d0sc00167h,,,,
2021,CDK4,,10.1039/d0sc00167h,,,,
2021,CDK6,,10.1039/d0sc00167h,,,,
2022,CDK4,,10.1039/d0sc00167h,,,,
2022,CDK6,,10.1039/d0sc00167h,,,,
2023,CDK6,,10.1039/d0sc00167h,,,,
2023,CDK4,,10.1039/d0sc00167h,,,,
2024,CDK6,,10.1039/d0sc00167h,,,,
2024,CDK4,,10.1039/d0sc00167h,,,,
2025,CDK6,,10.1039/d0sc00167h,,,,
2025,CDK4,,10.1039/d0sc00167h,,,,
2026,CDK6,,10.1039/d0sc00167h,,,,
2026,CDK4,,10.1039/d0sc00167h,,,,
2027,CDK4,,10.1039/d0sc00167h,,,,
2027,CDK6,,10.1039/d0sc00167h,,,,
2028,CDK6,,10.1039/d0sc00167h,,,,
2028,CDK4,,10.1039/d0sc00167h,,,,
2029,CDK6,97.1/95.9,10.1039/d0sc00167h,,,,% CDK6 degradation in MM.1S cells after 16 h treatment at 100/1000 nM
2029,CDK4,,10.1039/d0sc00167h,,,,
2030,CDK6,,10.1039/d0sc00167h,,,,
2030,CDK4,,10.1039/d0sc00167h,,,,
2031,CDK6,,10.1039/d0sc00167h,,,,
2031,CDK4,,10.1039/d0sc00167h,,,,
2032,CDK6,,10.1039/d0sc00167h,,,,
2032,CDK4,,10.1039/d0sc00167h,,,,
2033,CDK6,,10.1039/d0sc00167h,,,,
2033,CDK4,,10.1039/d0sc00167h,,,,
2034,CDK6,,10.1039/d0sc00167h,,,,
2034,CDK4,,10.1039/d0sc00167h,,,,
2035,CDK6,,10.1039/d0sc00167h,,,,
2035,CDK4,,10.1039/d0sc00167h,,,,
2036,CDK6,,10.1039/d0sc00167h,,,,
2036,CDK4,,10.1039/d0sc00167h,,,,
2037,CDK4,,10.1039/d0sc00167h,,,,
2037,CDK6,,10.1039/d0sc00167h,,,,
2038,CDK4,,10.1039/d0sc00167h,20,,Degradation of CDK4 in MM.1S cells after 16 h treatment,
2038,CDK6,,10.1039/d0sc00167h,5.1,>95,Degradation of CDK6 in MM.1S cells after 16 h treatment,
2039,CDK6,25/82,10.1039/d0sc00167h,,,,% CDK6 degradation in MM.1S cells after 16 h treatment at 100/1000 nM
2039,CDK4,,10.1039/d0sc00167h,,,,
2040,CDK6,0/0,10.1039/d0sc00167h,,,,% CDK6 degradation in MM.1S cells after 16 h treatment at 100/1000 nM
2040,CDK4,0/0,10.1039/d0sc00167h,,,,% CDK4 degradation in MM.1S cells after 16 h treatment at 100/1000 nM
2041,AURKB,,10.1016/j.cell.2020.10.038,,,,
2041,AURKA,62 (WB),10.1038/s41589-020-00652-y,,,,% AURORA-A degradation in AURORA-A in MV4-11 cells after 6 h treatment at 0.1 μM
2041,AURKA,,10.1016/j.cell.2020.10.038,,,,
2042,AURKA,36 (WB),10.1038/s41589-020-00652-y,,,,% AURORA-A degradation in AURORA-A in MV4-11 cells after 6 h treatment at 1 μM
2043,AURKA,30 (WB),10.1038/s41589-020-00652-y,,,,% AURORA-A degradation in AURORA-A in MV4-11 cells after 6 h treatment at 0.1 μM
2044,AURKA,,10.1038/s41589-020-00652-y,28,,Degradation of AURKA in MV4-11 cells after 6 h treatment,
2045,AURKA,40 (WB),10.1038/s41589-020-00652-y,,,,% AURORA-A degradation in AURORA-A in MV4-11 cells after 6 h treatment at 1 μM
2046,AURKA,2 (WB),10.1038/s41589-020-00652-y,,,,% AURORA-A degradation in AURORA-A in MV4-11 cells after 6 h treatment at 0.1 μM
2047,AURKA,0 (WB),10.1038/s41589-020-00652-y,,,,% AURORA-A degradation in AURORA-A in MV4-11 cells after 6 h treatment at 0.1 μM
2048,BRAF V600E,,10.1038/s41589-020-0609-7,90,84,Degradation of BRAF V600E in A375 cells after 24 h treatment,
2049,BRAF V600E,,10.1038/s41589-020-0609-7,45,65,Degradation of BRAF V600E in A375 cells after 24 h treatment,
2050,BRAF V600E,,10.1038/s41589-020-0609-7,100,51,Degradation of BRAF V600E in A375 cells after 24 h treatment,
2051,BRAF V600E,,10.1038/s41589-020-0609-7,,,,
2052,BRAF V600E,,10.1038/s41589-020-0609-7,,,,
2053,BRAF V600E,,10.1038/s41589-020-0609-7,,,,
2054,BRAF V600E,,10.1038/s41589-020-0609-7,,,,
2055,BRAF V600E,,10.1038/s41589-020-0609-7,,,,
2056,BRAF V600E,,10.1038/s41589-020-0609-7,,,,
2057,BRAF V600E,,10.1038/s41589-020-0609-7,,,,
2058,BRAF V600E,,10.1038/s41589-020-0609-7,,,,
2059,BRAF V600E,,10.1038/s41589-020-0609-7,500,50,Degradation of BRAF V600E in A375 cells after 24 h treatment,
2060,BRAF V600E,,10.1038/s41589-020-0609-7,,N.D.,,
2061,BRAF V600E,,10.1038/s41589-020-0609-7,,N.D.,,
2062,BRAF V600E,,10.1038/s41589-020-0609-7,,N.D.,,
2063,BRAF V600E,,10.1038/s41589-020-0609-7,25,71,Degradation of BRAF V600E in A375 cells after 24 h treatment,
2064,BRAF V600E,,10.1038/s41589-020-0609-7,80,72,Degradation of BRAF V600E in A375 cells after 24 h treatment,
2065,BRAF V600E,,10.1038/s41589-020-0609-7,50,74,Degradation of BRAF V600E in A375 cells after 24 h treatment,
2066,BTK,,10.1038/s41589-020-00686-2,,,,
2067,BTK,,10.1038/s41589-020-00686-2,800,,Degradation of BTK in THP-1 cells,
2068,BTK,,10.1038/s41589-020-00686-2,4700,,Degradation of BTK in THP-1 cells,
2069,CDK2,,10.1038/s41589-021-00742-5,,,,
2070,CDK2,,10.1038/s41589-021-00742-5,,,,
2071,CDK2,,10.1038/s41589-021-00742-5,56/13/18,,Degradation of CDK2 in OCI-AML2/OCI-AML3/Ramos cells after 48 h treatment,
2071,CDK2,,10.1038/s41589-021-00742-5,61/12/1,,Degradation of CDK2 in Kasumi-1/NB4/MV-4-11 cells after 48 h treatment,
2071,CDK2,,10.1038/s41589-021-00742-5,43/33/29,,Degradation of CDK2 in Z138/HBL-1/Mino cells after 48 h treatment,
2071,CDK2,,10.1038/s41589-021-00742-5,38/53/11,,Degradation of CDK2 in Jurkat/MOLT-4/U937 cells after 48 h treatment,
2071,CDK2,,10.1038/s41589-021-00742-5,160/4/9,,Degradation of CDK2 in Pfeiffer/DOHH2/K562 cells after 48 h treatment,
2071,CDK2,,10.1038/s41589-021-00742-5,22/8,,Degradation of CDK2 in MM.1S/MDA-MB-231 cells after 48 h treatment,
2072,CDK2,,10.1038/s41589-021-00742-5,,,,
2073,BRAF G466V,,10.1038/s41467-021-21159-7,29/23,80/90,Degradation of BRAF G466V in H1666/CAL-12T cells,
2073,BRAF V600K,,10.1038/s41467-021-21159-7,,,,
2073,BRAF K601E,,10.1038/s41467-021-21159-7,,,,
2073,BRAF G466E,,10.1038/s41467-021-21159-7,,,,
2073,BRAF D594N,,10.1038/s41467-021-21159-7,,,,
2073,BRAF,,10.1038/s41467-021-21159-7,,,,
2073,BRAF G469A,,10.1038/s41467-021-21159-7,15,95,Degradation of BRAF G469A in SK-MEL-246 cells,
2073,BRAF V600E,,10.1038/s41467-021-21159-7,6.8,95,Degradation of BRAF V600E in SK-MEL-28 cells,
2074,BRAF V600K,,10.1038/s41467-021-21159-7,,,,
2074,BRAF K601E,,10.1038/s41467-021-21159-7,,,,
2074,BRAF G469A,,10.1038/s41467-021-21159-7,,,,
2074,BRAF G466E,,10.1038/s41467-021-21159-7,,,,
2074,BRAF V600E,,10.1038/s41467-021-21159-7,,,,
2074,BRAF D594N,,10.1038/s41467-021-21159-7,,,,
2074,BRAF G466V,,10.1038/s41467-021-21159-7,,,,
2074,BRAF,,10.1038/s41467-021-21159-7,,,,
2075,BRAF G466E,,10.1038/s41467-021-21159-7,,,,
2075,BRAF V600E,,10.1038/s41467-021-21159-7,,,,
2075,BRAF V600K,,10.1038/s41467-021-21159-7,,,,
2075,BRAF K601E,,10.1038/s41467-021-21159-7,,,,
2075,BRAF G469A,,10.1038/s41467-021-21159-7,,,,
2075,BRAF D594N,,10.1038/s41467-021-21159-7,,,,
2075,BRAF G466V,,10.1038/s41467-021-21159-7,,,,
2075,BRAF,,10.1038/s41467-021-21159-7,,,,
2076,BTK,,10.1038/s41467-020-17997-6,6.6,,Degradation of BTK in MOLM-14 cells after 24 h treatment,
2077,BTK,,10.1038/s41467-020-17997-6,,,,
2078,BTK,,10.1038/s41467-020-17997-6,,,,
2079,BTK,,10.1038/s41467-020-17997-6,,,,
2080,BTK,,10.1038/s41467-020-17997-6,,,,
2081,BTK,,10.1038/s41467-020-17997-6,,,,
2082,BTK,,10.1038/s41467-020-17997-6,,,,
2083,BTK,,10.1038/s41467-020-17997-6,,,,
2084,BTK,,10.1038/s41467-020-17997-6,,,,
2085,BTK,,10.1038/s41467-020-17997-6,,,,
2086,BTK,,10.1038/s41467-020-17997-6,,,,
2087,BTK,,10.1038/s41467-020-17997-6,,,,
2088,BTK,,10.1038/s41467-020-17997-6,,,,
2089,BTK,,10.1038/s41467-020-17997-6,,,,
2090,BTK,,10.1038/s41467-020-17997-6,,,,
2091,BTK,,10.1038/s41467-020-17997-6,,,,
2092,BTK,,10.1038/s41467-020-17997-6,,,,
2093,BTK,,10.1038/s41467-020-17997-6,,,,
2094,FLT3,,10.1038/s41467-020-17997-6,,,,
2095,FLT3,,10.1038/s41467-020-17997-6,,,,
2096,FLT3,,10.1038/s41467-020-17997-6,,,,
2097,FKBP12 F36V,,10.1038/s41467-020-18377-w,,,,
2098,FKBP12 F36V,,10.1038/s41467-020-18377-w,,,,
2099,PARP1,,10.1080/14756366.2020.1804382,,,,
2100,PARP1,,10.1080/14756366.2020.1804382,5400,,Degradation of PARP1 in SW620 cells after 24 h treatment,
2101,PARP1,,10.1080/14756366.2020.1804382,6200,,Degradation of PARP1 in SW620 cells after 24 h treatment,
2102,AR,,10.1158/1535-7163.MCT-20-0417,2000,,Degradation of AR in 22Rv1 cells after 24 h treatment,
2102,AR-V7,,10.1158/1535-7163.MCT-20-0417,370,,Degradation of AR-V7 in 22Rv1 cells after 24 h treatment,
2103,LRRK2,,10.1002/cmdc.202000872,,N.D.,,
2104,LRRK2,,10.1002/cmdc.202000872,,N.D.,,
2105,LRRK2,,10.1002/cmdc.202000872,,N.D.,,
2106,LRRK2,,10.1002/cmdc.202000872,,N.D.,,
2107,LRRK2,,10.1002/cmdc.202000872,,N.D.,,
2108,LRRK2,,10.1002/cmdc.202000872,,N.D.,,
2109,LRRK2,,10.1002/cmdc.202000872,,N.D.,,
2110,HDAC1,,10.3390/molecules25214991,,,,
2110,HDAC8,,10.3390/molecules25214991,,,,
2110,HDAC6,,10.3390/molecules25214991,,,,
2111,HDAC1,,10.3390/molecules25214991,,,,
2111,HDAC8,,10.3390/molecules25214991,,,,
2111,HDAC6,,10.3390/molecules25214991,,,,
2112,HDAC8,,10.3390/molecules25214991,,,,
2112,HDAC6,,10.3390/molecules25214991,,,,
2112,HDAC1,,10.3390/molecules25214991,,,,
2113,FAK,>85/>85,10.1021/acsmedchemlett.0c00290,,,,% FAK degradation in PA-TU-8988T cells after 4 h treatment at 10/100 nM
2114,PTK2B,,10.1016/j.cell.2020.10.038,,,,
2114,FAK,70-84/>85,10.1021/acsmedchemlett.0c00290,,,,% FAK degradation in PA-TU-8988T cells after 4 h treatment at 10/100 nM
2114,AURKA,,10.1016/j.cell.2020.10.038,,,,
2114,Wee1,,10.1016/j.cell.2020.10.038,,,,
2114,CDK7,,10.1016/j.cell.2020.10.038,,,,
2114,RPS6KA3,,10.1016/j.cell.2020.10.038,,,,
2114,MAPK7,,10.1016/j.cell.2020.10.038,,,,
2114,CDK10,,10.1016/j.cell.2020.10.038,,,,
2114,RPS6KA1,,10.1016/j.cell.2020.10.038,,,,
2114,STK33,,10.1016/j.cell.2020.10.038,,,,
2115,FAK,>85/>85,10.1021/acsmedchemlett.0c00290,,,,% FAK degradation in PA-TU-8988T cells after 4 h treatment at 10/100 nM
2116,FAK,>85/>85,10.1021/acsmedchemlett.0c00290,,,,% FAK degradation in PA-TU-8988T cells after 4 h treatment at 10/100 nM
2116,STK33,,10.1016/j.cell.2020.10.038,,,,
2116,RPS6KA1,,10.1016/j.cell.2020.10.038,,,,
2116,PTK2B,,10.1016/j.cell.2020.10.038,,,,
2116,RPS6KA3,,10.1016/j.cell.2020.10.038,,,,
2116,Wee1,,10.1016/j.cell.2020.10.038,,,,
2116,NUAK1,,10.1016/j.cell.2020.10.038,,,,
2116,AURKA,,10.1016/j.cell.2020.10.038,,,,
2117,FAK,25-49/>85,10.1021/acsmedchemlett.0c00290,,,,% FAK degradation in PA-TU-8988T cells after 4 h treatment at 10/100 nM
2118,FAK,>85/>85,10.1021/acsmedchemlett.0c00290,,,,% FAK degradation in PA-TU-8988T cells after 4 h treatment at 10/100 nM
2119,ER,,10.1021/acsmedchemlett.0c00589,0.5,,Degradation of ERalpha in MCF-7 cells,
2120,ER,,10.1021/acsmedchemlett.0c00589,0.5,,Degradation of ERalpha in MCF-7 cells,
2121,ER,,10.1021/acsmedchemlett.0c00589,0.6,,Degradation of ERalpha in MCF-7 cells,
2122,ER,,10.1021/acsmedchemlett.0c00589,0.6,,Degradation of ERalpha in MCF-7 cells,
2123,ER,,10.1021/acsmedchemlett.0c00589,0.8,,Degradation of ERalpha in MCF-7 cells,
2124,ER,,10.1021/acsmedchemlett.0c00589,0.4,,Degradation of ERalpha in MCF-7 cells,
2125,ER,,10.1021/acsmedchemlett.0c00589,0.4,,Degradation of ERalpha in MCF-7 cells,
2126,ER,,10.1021/acsmedchemlett.0c00589,0.4,,Degradation of ERalpha in MCF-7 cells,
2127,ER,,10.1021/acsmedchemlett.0c00589,0.5,,Degradation of ERalpha in MCF-7 cells,
2128,ER,,10.1021/acsmedchemlett.0c00589,0.4,,Degradation of ERalpha in MCF-7 cells,
2129,ER,,10.1021/acsmedchemlett.0c00589,0.7,,Degradation of ERalpha in MCF-7 cells,
2130,ER,,10.1021/acsmedchemlett.0c00589,0.4,,Degradation of ERalpha in MCF-7 cells,
2131,SMARCA4,,10.1021/acsmedchemlett.0c00347,26,99,Degradation of SMARCA4 in A549 cells,
2131,SMARCA2,,10.1021/acsmedchemlett.0c00347,41,99,Degradation of SMARCA2 in A549 cells,
2132,SMARCA2,,10.1021/acsmedchemlett.0c00347,26,99,Degradation of SMARCA2 in A549 cells,
2132,SMARCA4,,10.1021/acsmedchemlett.0c00347,16,100,Degradation of SMARCA4 in A549 cells,
2133,SMARCA4,,10.1021/acsmedchemlett.0c00347,25,92,Degradation of SMARCA4 in A549 cells,
2133,SMARCA2,,10.1021/acsmedchemlett.0c00347,58,90,Degradation of SMARCA2 in A549 cells,
2134,SMARCA2,,10.1021/acsmedchemlett.0c00347,55,95,Degradation of SMARCA2 in A549 cells,
2134,SMARCA4,,10.1021/acsmedchemlett.0c00347,33,95,Degradation of SMARCA4 in A549 cells,
2135,GSK3A,,10.1016/j.cell.2020.10.038,,N.D.,,
2135,GSK-3beta,,10.1016/j.cell.2020.10.038,,N.D.,,
2136,GSK3A,,10.1016/j.cell.2020.10.038,,N.D.,,
2136,GSK-3beta,,10.1016/j.cell.2020.10.038,,N.D.,,
2137,AURKB,,10.1016/j.cell.2020.10.038,,,,
2137,BMP2K,,10.1016/j.cell.2020.10.038,,,,
2137,NEK9,,10.1016/j.cell.2020.10.038,,,,
2137,AAK1,,10.1016/j.cell.2020.10.038,,,,
2137,MAP4K2,,10.1016/j.cell.2020.10.038,,,,
2137,ITK,,10.1016/j.cell.2020.10.038,,,,
2137,CDK9,,10.1016/j.cell.2020.10.038,,,,
2137,GSK-3beta,,10.1016/j.cell.2020.10.038,,,,
2137,EPHB2,,10.1016/j.cell.2020.10.038,,,,
2137,PAK4,,10.1016/j.cell.2020.10.038,,,,
2137,LATS1,,10.1016/j.cell.2020.10.038,,,,
2137,STK17B,,10.1016/j.cell.2020.10.038,,,,
2137,AURKA,,10.1016/j.cell.2020.10.038,,,,
2137,PLK4,,10.1016/j.cell.2020.10.038,,,,
2138,PAK1,,10.1016/j.cell.2020.10.038,,N.D.,,
2139,CDK19,,10.1016/j.cell.2020.10.038,,N.D.,,
2139,CDK8,,10.1016/j.cell.2020.10.038,,N.D.,,
2140,ULK1,,10.1016/j.cell.2020.10.038,,,,
2140,GAK,,10.1016/j.cell.2020.10.038,,,,
2140,AURKA,,10.1016/j.cell.2020.10.038,,,,
2140,Wee1,,10.1016/j.cell.2020.10.038,,,,
2140,MARK3,,10.1016/j.cell.2020.10.038,,,,
2140,STK17B,,10.1016/j.cell.2020.10.038,,,,
2140,STK17A,,10.1016/j.cell.2020.10.038,,,,
2140,BMP2K,,10.1016/j.cell.2020.10.038,,,,
2140,SNRK,,10.1016/j.cell.2020.10.038,,,,
2140,SIK2,,10.1016/j.cell.2020.10.038,,,,
2140,MARK4,,10.1016/j.cell.2020.10.038,,,,
2140,AURKB,,10.1016/j.cell.2020.10.038,,,,
2140,MARK2,,10.1016/j.cell.2020.10.038,,,,
2140,AAK1,,10.1016/j.cell.2020.10.038,,,,
2140,CDK10,,10.1016/j.cell.2020.10.038,,,,
2140,CDK9,,10.1016/j.cell.2020.10.038,,,,
2141,SNRK,,10.1016/j.cell.2020.10.038,,,,
2141,Wee1,,10.1016/j.cell.2020.10.038,,,,
2141,MARK3,,10.1016/j.cell.2020.10.038,,,,
2141,RPS6KB1,,10.1016/j.cell.2020.10.038,,,,
2141,MARK2,,10.1016/j.cell.2020.10.038,,,,
2141,STK17B,,10.1016/j.cell.2020.10.038,,,,
2141,ULK1,,10.1016/j.cell.2020.10.038,,,,
2141,GAK,,10.1016/j.cell.2020.10.038,,,,
2141,MARK4,,10.1016/j.cell.2020.10.038,,,,
2141,AAK1,,10.1016/j.cell.2020.10.038,,,,
2141,SIK3,,10.1016/j.cell.2020.10.038,,,,
2141,STK17A,,10.1016/j.cell.2020.10.038,,,,
2141,SIK2,,10.1016/j.cell.2020.10.038,,,,
2142,ABL1,,10.1016/j.cell.2020.10.038,,N.D.,,
2143,CSK,,10.1016/j.cell.2020.10.038,,,,
2143,Wee1,,10.1016/j.cell.2020.10.038,,,,
2143,ABL2,,10.1016/j.cell.2020.10.038,,,,
2143,BLK,,10.1016/j.cell.2020.10.038,,,,
2144,ULK3,,10.1016/j.cell.2020.10.038,,,,
2144,BMP2K,,10.1016/j.cell.2020.10.038,,,,
2144,SIK2,,10.1016/j.cell.2020.10.038,,,,
2144,NEK9,,10.1016/j.cell.2020.10.038,,,,
2144,AAK1,,10.1016/j.cell.2020.10.038,,,,
2144,CDK4,,10.1016/j.cell.2020.10.038,,,,
2144,LCK,,10.1016/j.cell.2020.10.038,,,,
2144,STK17B,,10.1016/j.cell.2020.10.038,,,,
2144,ULK1,,10.1016/j.cell.2020.10.038,,,,
2144,PTK2B,,10.1016/j.cell.2020.10.038,,,,
2144,GAK,,10.1016/j.cell.2020.10.038,,,,
2144,CDK6,,10.1016/j.cell.2020.10.038,,,,
2144,LIMK2,,10.1016/j.cell.2020.10.038,,,,
2144,MAPK9,,10.1016/j.cell.2020.10.038,,,,
2144,CDK16,,10.1016/j.cell.2020.10.038,,,,
2144,MAPK8,,10.1016/j.cell.2020.10.038,,,,
2144,Wee1,,10.1016/j.cell.2020.10.038,,,,
2144,EIF2AK2,,10.1016/j.cell.2020.10.038,,,,
2144,FER,,10.1016/j.cell.2020.10.038,,,,
2144,AURKA,,10.1016/j.cell.2020.10.038,,,,
2144,PLK4,,10.1016/j.cell.2020.10.038,,,,
2144,MAP3K11,,10.1016/j.cell.2020.10.038,,,,
2144,CAMKK1,,10.1016/j.cell.2020.10.038,,,,
2144,STK17A,,10.1016/j.cell.2020.10.038,,,,
2145,ULK1,,10.1016/j.cell.2020.10.038,,,,
2145,LATS1,,10.1016/j.cell.2020.10.038,,,,
2145,LCK,,10.1016/j.cell.2020.10.038,,,,
2145,FYN,,10.1016/j.cell.2020.10.038,,,,
2145,YES1,,10.1016/j.cell.2020.10.038,,,,
2145,LYN,,10.1016/j.cell.2020.10.038,,,,
2145,CDK4,,10.1016/j.cell.2020.10.038,,,,
2145,Src,,10.1016/j.cell.2020.10.038,,,,
2145,FER,,10.1016/j.cell.2020.10.038,,,,
2145,CDK11B,,10.1016/j.cell.2020.10.038,,,,
2145,EPHA3,,10.1016/j.cell.2020.10.038,,,,
2145,Wee1,,10.1016/j.cell.2020.10.038,,,,
2145,TTK,,10.1016/j.cell.2020.10.038,,,,
2145,CSK,,10.1016/j.cell.2020.10.038,,,,
2145,TEC,,10.1016/j.cell.2020.10.038,,,,
2145,ABL2,,10.1016/j.cell.2020.10.038,,,,
2145,MAPK8,,10.1016/j.cell.2020.10.038,,,,
2145,MAPK9,,10.1016/j.cell.2020.10.038,,,,
2145,MAPKAPK2,,10.1016/j.cell.2020.10.038,,,,
2145,BLK,,10.1016/j.cell.2020.10.038,,,,
2145,RPS6KA3,,10.1016/j.cell.2020.10.038,,,,
2145,PLK1,,10.1016/j.cell.2020.10.038,,,,
2145,LIMK1,,10.1016/j.cell.2020.10.038,,,,
2145,LIMK2,,10.1016/j.cell.2020.10.038,,,,
2145,MAPK12,,10.1016/j.cell.2020.10.038,,,,
2145,EPHB3,,10.1016/j.cell.2020.10.038,,,,
2145,FAK,,10.1016/j.cell.2020.10.038,,,,
2145,TNK2,,10.1016/j.cell.2020.10.038,,,,
2145,MAP4K2,,10.1016/j.cell.2020.10.038,,,,
2145,MAP3K1,,10.1016/j.cell.2020.10.038,,,,
2145,RIPK1,,10.1016/j.cell.2020.10.038,,,,
2145,PTK2B,,10.1016/j.cell.2020.10.038,,,,
2145,RPS6KA1,,10.1016/j.cell.2020.10.038,,,,
2145,p38beta,,10.1016/j.cell.2020.10.038,,,,
2145,p38alpha,,10.1016/j.cell.2020.10.038,,,,
2145,MAP3K11,,10.1016/j.cell.2020.10.038,,,,
2145,DDR2,,10.1016/j.cell.2020.10.038,,,,
2145,LRRK2,,10.1016/j.cell.2020.10.038,,,,
2145,UHMK1,,10.1016/j.cell.2020.10.038,,,,
2145,MAP4K1,,10.1016/j.cell.2020.10.038,,,,
2145,SIK2,,10.1016/j.cell.2020.10.038,,,,
2145,MKNK2,,10.1016/j.cell.2020.10.038,,,,
2145,MAP3K20,,10.1016/j.cell.2020.10.038,,,,
2145,NLK,,10.1016/j.cell.2020.10.038,,,,
2145,TAOK2,,10.1016/j.cell.2020.10.038,,,,
2145,CDK11A,,10.1016/j.cell.2020.10.038,,,,
2145,MAP4K5,,10.1016/j.cell.2020.10.038,,,,
2145,AURKA,,10.1016/j.cell.2020.10.038,,,,
2145,GAK,,10.1016/j.cell.2020.10.038,,,,
2145,EPHB6,,10.1016/j.cell.2020.10.038,,,,
2145,RIPK2,,10.1016/j.cell.2020.10.038,,,,
2145,BUB1,,10.1016/j.cell.2020.10.038,,,,
2146,SIK2,,10.1016/j.cell.2020.10.038,,,,
2146,MKNK2,,10.1016/j.cell.2020.10.038,,,,
2146,LCK,,10.1016/j.cell.2020.10.038,,,,
2146,YES1,,10.1016/j.cell.2020.10.038,,,,
2146,CDK4,,10.1016/j.cell.2020.10.038,,,,
2146,Src,,10.1016/j.cell.2020.10.038,,,,
2146,FER,,10.1016/j.cell.2020.10.038,,,,
2146,CSK,,10.1016/j.cell.2020.10.038,,,,
2146,MAPK8,,10.1016/j.cell.2020.10.038,,,,
2146,MAPK9,,10.1016/j.cell.2020.10.038,,,,
2146,CLK1,,10.1016/j.cell.2020.10.038,,,,
2146,BLK,,10.1016/j.cell.2020.10.038,,,,
2146,PLK1,,10.1016/j.cell.2020.10.038,,,,
2146,LIMK1,,10.1016/j.cell.2020.10.038,,,,
2146,TNK2,,10.1016/j.cell.2020.10.038,,,,
2146,PTK2B,,10.1016/j.cell.2020.10.038,,,,
2146,UHMK1,,10.1016/j.cell.2020.10.038,,,,
2147,MAPK9,,10.1016/j.cell.2020.10.038,,,,
2147,MAPKAPK2,,10.1016/j.cell.2020.10.038,,,,
2147,BLK,,10.1016/j.cell.2020.10.038,,,,
2147,RPS6KA3,,10.1016/j.cell.2020.10.038,,,,
2147,LIMK1,,10.1016/j.cell.2020.10.038,,,,
2147,TNK2,,10.1016/j.cell.2020.10.038,,,,
2147,MAP3K1,,10.1016/j.cell.2020.10.038,,,,
2147,PTK2B,,10.1016/j.cell.2020.10.038,,,,
2147,RPS6KA1,,10.1016/j.cell.2020.10.038,,,,
2147,p38alpha,,10.1016/j.cell.2020.10.038,,,,
2147,MAP3K11,,10.1016/j.cell.2020.10.038,,,,
2147,PDIK1L,,10.1016/j.cell.2020.10.038,,,,
2147,UHMK1,,10.1016/j.cell.2020.10.038,,,,
2147,MAP4K1,,10.1016/j.cell.2020.10.038,,,,
2147,SIK2,,10.1016/j.cell.2020.10.038,,,,
2147,MAP3K20,,10.1016/j.cell.2020.10.038,,,,
2147,MKNK2,,10.1016/j.cell.2020.10.038,,,,
2147,GAK,,10.1016/j.cell.2020.10.038,,,,
2147,EPHB6,,10.1016/j.cell.2020.10.038,,,,
2147,BUB1,,10.1016/j.cell.2020.10.038,,,,
2147,ULK1,,10.1016/j.cell.2020.10.038,,,,
2147,PAK4,,10.1016/j.cell.2020.10.038,,,,
2147,ABL1,,10.1016/j.cell.2020.10.038,,,,
2147,LCK,,10.1016/j.cell.2020.10.038,,,,
2147,FYN,,10.1016/j.cell.2020.10.038,,,,
2147,YES1,,10.1016/j.cell.2020.10.038,,,,
2147,CDK4,,10.1016/j.cell.2020.10.038,,,,
2147,Src,,10.1016/j.cell.2020.10.038,,,,
2147,FER,,10.1016/j.cell.2020.10.038,,,,
2147,CDK11B,,10.1016/j.cell.2020.10.038,,,,
2147,CSK,,10.1016/j.cell.2020.10.038,,,,
2147,ABL2,,10.1016/j.cell.2020.10.038,,,,
2147,MAPK8,,10.1016/j.cell.2020.10.038,,,,
2148,SIK2,,10.1016/j.cell.2020.10.038,,,,
2148,MAP3K20,,10.1016/j.cell.2020.10.038,,,,
2148,MKNK2,,10.1016/j.cell.2020.10.038,,,,
2148,p38alpha,,10.1016/j.cell.2020.10.038,,,,
2148,PTK2B,,10.1016/j.cell.2020.10.038,,,,
2148,MAP4K2,,10.1016/j.cell.2020.10.038,,,,
2148,TNK2,,10.1016/j.cell.2020.10.038,,,,
2148,LIMK2,,10.1016/j.cell.2020.10.038,,,,
2148,BLK,,10.1016/j.cell.2020.10.038,,,,
2148,MAPK9,,10.1016/j.cell.2020.10.038,,,,
2148,ABL2,,10.1016/j.cell.2020.10.038,,,,
2148,CSK,,10.1016/j.cell.2020.10.038,,,,
2148,FER,,10.1016/j.cell.2020.10.038,,,,
2148,Src,,10.1016/j.cell.2020.10.038,,,,
2148,CDK4,,10.1016/j.cell.2020.10.038,,,,
2148,LCK,,10.1016/j.cell.2020.10.038,,,,
2148,GAK,,10.1016/j.cell.2020.10.038,,,,
2149,GAK,,10.1016/j.cell.2020.10.038,,,,
2149,MAPK7,,10.1016/j.cell.2020.10.038,,,,
2149,RIPK1,,10.1016/j.cell.2020.10.038,,,,
2149,PTK2B,,10.1016/j.cell.2020.10.038,,,,
2149,RPS6KA1,,10.1016/j.cell.2020.10.038,,,,
2149,p38alpha,,10.1016/j.cell.2020.10.038,,,,
2149,MAPKAPK3,,10.1016/j.cell.2020.10.038,,,,
2149,MAP4K3,,10.1016/j.cell.2020.10.038,,,,
2149,PDIK1L,,10.1016/j.cell.2020.10.038,,,,
2149,STK35,,10.1016/j.cell.2020.10.038,,,,
2149,MAP4K1,,10.1016/j.cell.2020.10.038,,,,
2149,SIK2,,10.1016/j.cell.2020.10.038,,,,
2149,MAP3K20,,10.1016/j.cell.2020.10.038,,,,
2149,NLK,,10.1016/j.cell.2020.10.038,,,,
2149,SIK3,,10.1016/j.cell.2020.10.038,,,,
2149,MAP4K5,,10.1016/j.cell.2020.10.038,,,,
2149,MAP4K2,,10.1016/j.cell.2020.10.038,,,,
2149,TNK2,,10.1016/j.cell.2020.10.038,,,,
2149,LIMK1,,10.1016/j.cell.2020.10.038,,,,
2149,RPS6KA3,,10.1016/j.cell.2020.10.038,,,,
2149,BLK,,10.1016/j.cell.2020.10.038,,,,
2149,MAPKAPK2,,10.1016/j.cell.2020.10.038,,,,
2149,MAPK9,,10.1016/j.cell.2020.10.038,,,,
2149,MAPK8,,10.1016/j.cell.2020.10.038,,,,
2149,ABL2,,10.1016/j.cell.2020.10.038,,,,
2149,CSK,,10.1016/j.cell.2020.10.038,,,,
2149,EPHA3,,10.1016/j.cell.2020.10.038,,,,
2149,CDK11B,,10.1016/j.cell.2020.10.038,,,,
2149,FER,,10.1016/j.cell.2020.10.038,,,,
2149,CDK4,,10.1016/j.cell.2020.10.038,,,,
2149,ABL1,,10.1016/j.cell.2020.10.038,,,,
2149,ULK1,,10.1016/j.cell.2020.10.038,,,,
2150,STK35,,10.1016/j.cell.2020.10.038,,,,
2150,CIT,,10.1016/j.cell.2020.10.038,,,,
2150,GAK,,10.1016/j.cell.2020.10.038,,,,
2150,MAP3K7,,10.1016/j.cell.2020.10.038,,,,
2150,ULK1,,10.1016/j.cell.2020.10.038,,,,
2150,ABL1,,10.1016/j.cell.2020.10.038,,,,
2150,LCK,,10.1016/j.cell.2020.10.038,,,,
2150,CDK4,,10.1016/j.cell.2020.10.038,,,,
2150,EPHA3,,10.1016/j.cell.2020.10.038,,,,
2150,CSK,,10.1016/j.cell.2020.10.038,,,,
2150,ABL2,,10.1016/j.cell.2020.10.038,,,,
2150,MAPK9,,10.1016/j.cell.2020.10.038,,,,
2150,MAP4K5,,10.1016/j.cell.2020.10.038,,,,
2150,TAOK2,,10.1016/j.cell.2020.10.038,,,,
2150,MAP3K20,,10.1016/j.cell.2020.10.038,,,,
2150,SIK2,,10.1016/j.cell.2020.10.038,,,,
2150,MAP4K1,,10.1016/j.cell.2020.10.038,,,,
2150,PDIK1L,,10.1016/j.cell.2020.10.038,,,,
2150,MAPKAPK3,,10.1016/j.cell.2020.10.038,,,,
2150,p38alpha,,10.1016/j.cell.2020.10.038,,,,
2150,MAPKAPK2,,10.1016/j.cell.2020.10.038,,,,
2150,RPS6KA1,,10.1016/j.cell.2020.10.038,,,,
2150,PTK2B,,10.1016/j.cell.2020.10.038,,,,
2150,FER,,10.1016/j.cell.2020.10.038,,,,
2150,RIPK1,,10.1016/j.cell.2020.10.038,,,,
2150,MAPK7,,10.1016/j.cell.2020.10.038,,,,
2150,MAP4K2,,10.1016/j.cell.2020.10.038,,,,
2150,TNK2,,10.1016/j.cell.2020.10.038,,,,
2150,LIMK2,,10.1016/j.cell.2020.10.038,,,,
2150,BLK,,10.1016/j.cell.2020.10.038,,,,
2150,CDK11B,,10.1016/j.cell.2020.10.038,,,,
2151,CDK4,,10.1016/j.cell.2020.10.038,,,,
2151,STK17A,,10.1016/j.cell.2020.10.038,,,,
2151,BUB1,,10.1016/j.cell.2020.10.038,,,,
2151,SIK2,,10.1016/j.cell.2020.10.038,,,,
2151,UHMK1,,10.1016/j.cell.2020.10.038,,,,
2151,TNK2,,10.1016/j.cell.2020.10.038,,,,
2151,LIMK2,,10.1016/j.cell.2020.10.038,,,,
2151,BLK,,10.1016/j.cell.2020.10.038,,,,
2151,TEC,,10.1016/j.cell.2020.10.038,,,,
2152,p38alpha,,10.1016/j.cell.2020.10.038,,,,
2153,PLK1,,10.1016/j.cell.2020.10.038,,,,
2153,BCKDK,,10.1016/j.cell.2020.10.038,,,,
2153,AURKA,,10.1016/j.cell.2020.10.038,,,,
2153,CDK1,,10.1016/j.cell.2020.10.038,,,,
2153,CDK4,,10.1016/j.cell.2020.10.038,,,,
2153,EIF2AK2,,10.1016/j.cell.2020.10.038,,,,
2153,CDK2,,10.1016/j.cell.2020.10.038,,,,
2153,CSK,,10.1016/j.cell.2020.10.038,,,,
2153,LIMK1,,10.1016/j.cell.2020.10.038,,,,
2153,LIMK2,,10.1016/j.cell.2020.10.038,,,,
2153,CDK6,,10.1016/j.cell.2020.10.038,,,,
2153,CDK16,,10.1016/j.cell.2020.10.038,,,,
2153,CDK17,,10.1016/j.cell.2020.10.038,,,,
2153,PDK1,,10.1016/j.cell.2020.10.038,,,,
2153,PDK2,,10.1016/j.cell.2020.10.038,,,,
2153,PDK3,,10.1016/j.cell.2020.10.038,,,,
2153,COQ8A,,10.1016/j.cell.2020.10.038,,,,
2153,COQ8B,,10.1016/j.cell.2020.10.038,,,,
2153,TESK2,,10.1016/j.cell.2020.10.038,,,,
2153,MAP3K20,,10.1016/j.cell.2020.10.038,,,,
2153,NLK,,10.1016/j.cell.2020.10.038,,,,
2154,PDK2,,10.1016/j.cell.2020.10.038,,,,
2154,PDK1,,10.1016/j.cell.2020.10.038,,,,
2154,LIMK1,,10.1016/j.cell.2020.10.038,,,,
2154,BCKDK,,10.1016/j.cell.2020.10.038,,,,
2154,COQ8A,,10.1016/j.cell.2020.10.038,,,,
2154,PDK3,,10.1016/j.cell.2020.10.038,,,,
2155,Src,,10.1016/j.cell.2020.10.038,,,,
2155,CSK,,10.1016/j.cell.2020.10.038,,,,
2155,TEC,,10.1016/j.cell.2020.10.038,,,,
2155,BLK,,10.1016/j.cell.2020.10.038,,,,
2155,LCK,,10.1016/j.cell.2020.10.038,,,,
2155,FYN,,10.1016/j.cell.2020.10.038,,,,
2155,ABL2,,10.1016/j.cell.2020.10.038,,,,
2156,LIMK1,,10.1016/j.cell.2020.10.038,,,,
2156,CDK17,,10.1016/j.cell.2020.10.038,,,,
2156,LIMK2,,10.1016/j.cell.2020.10.038,,,,
2157,c-KIT,,10.1016/j.cell.2020.10.038,,N.D.,,
2158,MAP2K5,,10.1016/j.cell.2020.10.038,,,,
2158,CSK,,10.1016/j.cell.2020.10.038,,,,
2158,MAP3K20,,10.1016/j.cell.2020.10.038,,,,
2158,LCK,,10.1016/j.cell.2020.10.038,,,,
2158,LIMK2,,10.1016/j.cell.2020.10.038,,,,
2158,BLK,,10.1016/j.cell.2020.10.038,,,,
2159,SGK3,,10.1016/j.cell.2020.10.038,,,,
2159,PIK3CG,,10.1016/j.cell.2020.10.038,,,,
2159,CLK1,,10.1016/j.cell.2020.10.038,,,,
2159,GSK3A,,10.1016/j.cell.2020.10.038,,,,
2159,GSK-3beta,,10.1016/j.cell.2020.10.038,,,,
2159,CDK9,,10.1016/j.cell.2020.10.038,,,,
2159,CDK11A,,10.1016/j.cell.2020.10.038,,,,
2160,CSK,,10.1016/j.cell.2020.10.038,,,,
2160,BLK,,10.1016/j.cell.2020.10.038,,,,
2161,PTK6,,10.1016/j.cell.2020.10.038,,,,
2161,CDC7,,10.1016/j.cell.2020.10.038,,,,
2161,PLK4,,10.1016/j.cell.2020.10.038,,,,
2161,CHEK1,,10.1016/j.cell.2020.10.038,,,,
2161,AURKA,,10.1016/j.cell.2020.10.038,,,,
2161,GAK,,10.1016/j.cell.2020.10.038,,,,
2161,BUB1B,,10.1016/j.cell.2020.10.038,,,,
2161,ULK1,,10.1016/j.cell.2020.10.038,,,,
2161,RPS6KA4,,10.1016/j.cell.2020.10.038,,,,
2161,CDK1,,10.1016/j.cell.2020.10.038,,,,
2161,FGFR1,,10.1016/j.cell.2020.10.038,,,,
2161,CDK4,,10.1016/j.cell.2020.10.038,,,,
2161,FER,,10.1016/j.cell.2020.10.038,,,,
2161,EPHA1,,10.1016/j.cell.2020.10.038,,,,
2161,CDK2,,10.1016/j.cell.2020.10.038,,,,
2161,Wee1,,10.1016/j.cell.2020.10.038,,,,
2161,ABL2,,10.1016/j.cell.2020.10.038,,,,
2161,CSNK1D,,10.1016/j.cell.2020.10.038,,,,
2161,CDK7,,10.1016/j.cell.2020.10.038,,,,
2161,CDK9,,10.1016/j.cell.2020.10.038,,,,
2161,LIMK2,,10.1016/j.cell.2020.10.038,,,,
2161,CDK6,,10.1016/j.cell.2020.10.038,,,,
2161,FAK,,10.1016/j.cell.2020.10.038,,,,
2161,TNK2,,10.1016/j.cell.2020.10.038,,,,
2161,ITK,,10.1016/j.cell.2020.10.038,,,,
2161,MAP4K2,,10.1016/j.cell.2020.10.038,,,,
2161,PRKAA1,,10.1016/j.cell.2020.10.038,,,,
2161,MAPK7,,10.1016/j.cell.2020.10.038,,,,
2161,MAP4K3,,10.1016/j.cell.2020.10.038,,,,
2161,UHMK1,,10.1016/j.cell.2020.10.038,,,,
2161,STK35,,10.1016/j.cell.2020.10.038,,,,
2161,AURKB,,10.1016/j.cell.2020.10.038,,,,
2161,MARK4,,10.1016/j.cell.2020.10.038,,,,
2161,SIK2,,10.1016/j.cell.2020.10.038,,,,
2161,IRAK4,,10.1016/j.cell.2020.10.038,,,,
2161,CDK12,,10.1016/j.cell.2020.10.038,,,,
2161,CDK13,,10.1016/j.cell.2020.10.038,,,,
2161,MELK,,10.1016/j.cell.2020.10.038,,,,
2161,MAPK6,,10.1016/j.cell.2020.10.038,,,,
2161,AAK1,,10.1016/j.cell.2020.10.038,,,,
2161,PKN3,,10.1016/j.cell.2020.10.038,,,,
2162,ABL1,,10.1016/j.cell.2020.10.038,,N.D.,,
2163,ABL1,,10.1016/j.cell.2020.10.038,,N.D.,,
2164,PDK2,,10.1016/j.cell.2020.10.038,,,,
2164,PDK3,,10.1016/j.cell.2020.10.038,,,,
2164,PDK1,,10.1016/j.cell.2020.10.038,,,,
2165,AKT1,,10.1016/j.cell.2020.10.038,,N.D.,,
2165,AKT2,,10.1016/j.cell.2020.10.038,,N.D.,,
2165,AKT3,,10.1016/j.cell.2020.10.038,,N.D.,,
2166,AKT3,,10.1016/j.cell.2020.10.038,,N.D.,,
2166,AKT2,,10.1016/j.cell.2020.10.038,,N.D.,,
2166,AKT1,,10.1016/j.cell.2020.10.038,,N.D.,,
2167,BCKDK,,10.1016/j.cell.2020.10.038,,,,
2167,AKT1,,10.1016/j.cell.2020.10.038,,,,
2167,AKT2,,10.1016/j.cell.2020.10.038,,,,
2167,AKT3,,10.1016/j.cell.2020.10.038,,,,
2167,PDK1,,10.1016/j.cell.2020.10.038,,,,
2168,AKT3,,10.1016/j.cell.2020.10.038,,N.D.,,
2168,AKT1,,10.1016/j.cell.2020.10.038,,N.D.,,
2168,AKT2,,10.1016/j.cell.2020.10.038,,N.D.,,
2169,AKT2,,10.1016/j.cell.2020.10.038,,N.D.,,
2169,AKT1,,10.1016/j.cell.2020.10.038,,N.D.,,
2169,AKT3,,10.1016/j.cell.2020.10.038,,N.D.,,
2170,LATS1,,10.1016/j.cell.2020.10.038,,,,
2170,STK17A,,10.1016/j.cell.2020.10.038,,,,
2171,Wee1,,10.1016/j.cell.2020.10.038,,,,
2171,AAK1,,10.1016/j.cell.2020.10.038,,,,
2171,BMP2K,,10.1016/j.cell.2020.10.038,,,,
2171,AURKA,,10.1016/j.cell.2020.10.038,,,,
2171,GAK,,10.1016/j.cell.2020.10.038,,,,
2172,AAK1,,10.1016/j.cell.2020.10.038,,,,
2172,AURKA,,10.1016/j.cell.2020.10.038,,,,
2173,GAK,,10.1016/j.cell.2020.10.038,,,,
2173,AAK1,,10.1016/j.cell.2020.10.038,,,,
2174,RPS6KB1,,10.1016/j.cell.2020.10.038,,,,
2174,CDK16,,10.1016/j.cell.2020.10.038,,,,
2174,AAK1,,10.1016/j.cell.2020.10.038,,,,
2174,NEK9,,10.1016/j.cell.2020.10.038,,,,
2174,MARK4,,10.1016/j.cell.2020.10.038,,,,
2174,GAK,,10.1016/j.cell.2020.10.038,,,,
2174,Wee1,,10.1016/j.cell.2020.10.038,,,,
2174,STK17A,,10.1016/j.cell.2020.10.038,,,,
2174,SIK3,,10.1016/j.cell.2020.10.038,,,,
2174,SIK2,,10.1016/j.cell.2020.10.038,,,,
2174,SNRK,,10.1016/j.cell.2020.10.038,,,,
2174,STK17B,,10.1016/j.cell.2020.10.038,,,,
2175,JAK2,,10.1016/j.cell.2020.10.038,,N.D.,,
2176,ABL2,,10.1016/j.cell.2020.10.038,,,,
2176,TYK2,,10.1016/j.cell.2020.10.038,,,,
2176,EPHB2,,10.1016/j.cell.2020.10.038,,,,
2176,SIK2,,10.1016/j.cell.2020.10.038,,,,
2177,CDK13,,10.1016/j.cell.2020.10.038,,,,
2177,CDK4,,10.1016/j.cell.2020.10.038,,,,
2177,LCK,,10.1016/j.cell.2020.10.038,,,,
2177,STK10,,10.1016/j.cell.2020.10.038,,,,
2177,CDK2,,10.1016/j.cell.2020.10.038,,,,
2177,Wee1,,10.1016/j.cell.2020.10.038,,,,
2177,CDK7,,10.1016/j.cell.2020.10.038,,,,
2177,CDK9,,10.1016/j.cell.2020.10.038,,,,
2177,BLK,,10.1016/j.cell.2020.10.038,,,,
2177,LIMK2,,10.1016/j.cell.2020.10.038,,,,
2177,CDK6,,10.1016/j.cell.2020.10.038,,,,
2177,CDK5,,10.1016/j.cell.2020.10.038,,,,
2177,CDK17,,10.1016/j.cell.2020.10.038,,,,
2177,AURKA,,10.1016/j.cell.2020.10.038,,,,
2177,ITK,,10.1016/j.cell.2020.10.038,,,,
2177,PRKAA1,,10.1016/j.cell.2020.10.038,,,,
2177,PTK2B,,10.1016/j.cell.2020.10.038,,,,
2177,AAK1,,10.1016/j.cell.2020.10.038,,,,
2177,BMP2K,,10.1016/j.cell.2020.10.038,,,,
2177,CDK12,,10.1016/j.cell.2020.10.038,,,,
2177,FER,,10.1016/j.cell.2020.10.038,,,,
2178,BUB1B,,10.1016/j.cell.2020.10.038,,,,
2178,STK17A,,10.1016/j.cell.2020.10.038,,,,
2178,PIM2,,10.1016/j.cell.2020.10.038,,,,
2178,RIOK2,,10.1016/j.cell.2020.10.038,,,,
2178,UHMK1,,10.1016/j.cell.2020.10.038,,,,
2178,MAP3K1,,10.1016/j.cell.2020.10.038,,,,
2178,PLK1,,10.1016/j.cell.2020.10.038,,,,
2178,CSNK1A1,,10.1016/j.cell.2020.10.038,,,,
2178,TTK,,10.1016/j.cell.2020.10.038,,,,
2178,Wee1,,10.1016/j.cell.2020.10.038,,,,
2178,CDK4,,10.1016/j.cell.2020.10.038,,,,
2178,NUAK1,,10.1016/j.cell.2020.10.038,,,,
2178,BUB1,,10.1016/j.cell.2020.10.038,,,,
2178,AURKA,,10.1016/j.cell.2020.10.038,,,,
2179,PIK3CG,,10.1016/j.cell.2020.10.038,,,,
2179,CSNK1D,,10.1016/j.cell.2020.10.038,,,,
2179,CSNK1A1,,10.1016/j.cell.2020.10.038,,,,
2179,CDK17,,10.1016/j.cell.2020.10.038,,,,
2179,STK17A,,10.1016/j.cell.2020.10.038,,,,
2179,PIM2,,10.1016/j.cell.2020.10.038,,,,
2179,RIOK2,,10.1016/j.cell.2020.10.038,,,,
2179,UHMK1,,10.1016/j.cell.2020.10.038,,,,
2179,CDK13,,10.1016/j.cell.2020.10.038,,,,
2179,MAP3K1,,10.1016/j.cell.2020.10.038,,,,
2179,CHEK1,,10.1016/j.cell.2020.10.038,,,,
2179,TTK,,10.1016/j.cell.2020.10.038,,,,
2179,Wee1,,10.1016/j.cell.2020.10.038,,,,
2179,CDK14,,10.1016/j.cell.2020.10.038,,,,
2179,STK17B,,10.1016/j.cell.2020.10.038,,,,
2179,ERN1,,10.1016/j.cell.2020.10.038,,,,
2179,CDK4,,10.1016/j.cell.2020.10.038,,,,
2179,BUB1B,,10.1016/j.cell.2020.10.038,,,,
2179,AURKA,,10.1016/j.cell.2020.10.038,,,,
2179,GSK3A,,10.1016/j.cell.2020.10.038,,,,
2179,GSK-3beta,,10.1016/j.cell.2020.10.038,,,,
2179,CDK9,,10.1016/j.cell.2020.10.038,,,,
2179,PLK1,,10.1016/j.cell.2020.10.038,,,,
2179,DAPK1,,10.1016/j.cell.2020.10.038,,,,
2179,BUB1,,10.1016/j.cell.2020.10.038,,,,
2179,CLK1,,10.1016/j.cell.2020.10.038,,,,
2179,NUAK1,,10.1016/j.cell.2020.10.038,,,,
2180,LIMK2,,10.1016/j.cell.2020.10.038,,,,
2180,NEK9,,10.1016/j.cell.2020.10.038,,,,
2180,STK17A,,10.1016/j.cell.2020.10.038,,,,
2180,CDK6,,10.1016/j.cell.2020.10.038,,,,
2180,AURKA,,10.1016/j.cell.2020.10.038,,,,
2180,AAK1,,10.1016/j.cell.2020.10.038,,,,
2180,PTK2B,,10.1016/j.cell.2020.10.038,,,,
2180,ULK1,,10.1016/j.cell.2020.10.038,,,,
2180,ULK3,,10.1016/j.cell.2020.10.038,,,,
2180,STK17B,,10.1016/j.cell.2020.10.038,,,,
2180,CDK4,,10.1016/j.cell.2020.10.038,,,,
2180,Wee1,,10.1016/j.cell.2020.10.038,,,,
2180,CAMKK1,,10.1016/j.cell.2020.10.038,,,,
2181,CDK16,,10.1016/j.cell.2020.10.038,,,,
2181,GAK,,10.1016/j.cell.2020.10.038,,,,
2181,ULK1,,10.1016/j.cell.2020.10.038,,,,
2181,STK17B,,10.1016/j.cell.2020.10.038,,,,
2181,LATS1,,10.1016/j.cell.2020.10.038,,,,
2181,CDK1,,10.1016/j.cell.2020.10.038,,,,
2181,CDK4,,10.1016/j.cell.2020.10.038,,,,
2181,RPS6KB1,,10.1016/j.cell.2020.10.038,,,,
2181,CDK2,,10.1016/j.cell.2020.10.038,,,,
2181,Wee1,,10.1016/j.cell.2020.10.038,,,,
2181,CDK7,,10.1016/j.cell.2020.10.038,,,,
2181,LIMK2,,10.1016/j.cell.2020.10.038,,,,
2181,CDK6,,10.1016/j.cell.2020.10.038,,,,
2181,CDK17,,10.1016/j.cell.2020.10.038,,,,
2181,MAPK6,,10.1016/j.cell.2020.10.038,,,,
2181,AAK1,,10.1016/j.cell.2020.10.038,,,,
2181,MARK2,,10.1016/j.cell.2020.10.038,,,,
2181,MAPKAPK5,,10.1016/j.cell.2020.10.038,,,,
2181,NEK9,,10.1016/j.cell.2020.10.038,,,,
2181,STK35,,10.1016/j.cell.2020.10.038,,,,
2181,MARK4,,10.1016/j.cell.2020.10.038,,,,
2181,SIK2,,10.1016/j.cell.2020.10.038,,,,
2181,MKNK2,,10.1016/j.cell.2020.10.038,,,,
2181,SNRK,,10.1016/j.cell.2020.10.038,,,,
2181,EIF2AK4,,10.1016/j.cell.2020.10.038,,,,
2181,STK17A,,10.1016/j.cell.2020.10.038,,,,
2182,LIMK1,,10.1016/j.cell.2020.10.038,,,,
2182,MAP2K5,,10.1016/j.cell.2020.10.038,,,,
2182,AURKA,,10.1016/j.cell.2020.10.038,,,,
2182,LATS1,,10.1016/j.cell.2020.10.038,,,,
2182,ABL1,,10.1016/j.cell.2020.10.038,,,,
2182,LCK,,10.1016/j.cell.2020.10.038,,,,
2182,FYN,,10.1016/j.cell.2020.10.038,,,,
2182,Src,,10.1016/j.cell.2020.10.038,,,,
2182,CSK,,10.1016/j.cell.2020.10.038,,,,
2182,ABL2,,10.1016/j.cell.2020.10.038,,,,
2182,CSNK1E,,10.1016/j.cell.2020.10.038,,,,
2182,BLK,,10.1016/j.cell.2020.10.038,,,,
2183,FER,,10.1016/j.cell.2020.10.038,,,,
2183,EPHA1,,10.1016/j.cell.2020.10.038,,,,
2183,EPHA2,,10.1016/j.cell.2020.10.038,,,,
2183,ABL2,,10.1016/j.cell.2020.10.038,,,,
2183,BLK,,10.1016/j.cell.2020.10.038,,,,
2183,IRAK1,,10.1016/j.cell.2020.10.038,,,,
2183,CDK6,,10.1016/j.cell.2020.10.038,,,,
2183,CDK5,,10.1016/j.cell.2020.10.038,,,,
2183,CDK17,,10.1016/j.cell.2020.10.038,,,,
2183,MAP4K2,,10.1016/j.cell.2020.10.038,,,,
2183,MAP3K1,,10.1016/j.cell.2020.10.038,,,,
2183,RIPK1,,10.1016/j.cell.2020.10.038,,,,
2183,GAK,,10.1016/j.cell.2020.10.038,,,,
2183,MAP3K7,,10.1016/j.cell.2020.10.038,,,,
2183,RIPK2,,10.1016/j.cell.2020.10.038,,,,
2183,STK10,,10.1016/j.cell.2020.10.038,,,,
2183,CDK14,,10.1016/j.cell.2020.10.038,,,,
2183,ABL1,,10.1016/j.cell.2020.10.038,,,,
2183,LCK,,10.1016/j.cell.2020.10.038,,,,
2183,FYN,,10.1016/j.cell.2020.10.038,,,,
2183,YES1,,10.1016/j.cell.2020.10.038,,,,
2183,LYN,,10.1016/j.cell.2020.10.038,,,,
2183,Src,,10.1016/j.cell.2020.10.038,,,,
2183,p38alpha,,10.1016/j.cell.2020.10.038,,,,
2183,COQ8A,,10.1016/j.cell.2020.10.038,,,,
2183,TAOK3,,10.1016/j.cell.2020.10.038,,,,
2183,MAP3K20,,10.1016/j.cell.2020.10.038,,,,
2183,MAP4K5,,10.1016/j.cell.2020.10.038,,,,
2183,PDK1,,10.1016/j.cell.2020.10.038,,,,
2183,PDK2,,10.1016/j.cell.2020.10.038,,,,
2183,PDK3,,10.1016/j.cell.2020.10.038,,,,
2184,BMP2K,,10.1016/j.cell.2020.10.038,,,,
2184,AURKA,,10.1016/j.cell.2020.10.038,,,,
2184,GSK3A,,10.1016/j.cell.2020.10.038,,,,
2184,GSK-3beta,,10.1016/j.cell.2020.10.038,,,,
2184,AAK1,,10.1016/j.cell.2020.10.038,,,,
2185,ABL2,,10.1016/j.cell.2020.10.038,,,,
2185,NLK,,10.1016/j.cell.2020.10.038,,,,
2185,SIK2,,10.1016/j.cell.2020.10.038,,,,
2185,PKMYT1,,10.1016/j.cell.2020.10.038,,,,
2185,p38alpha,,10.1016/j.cell.2020.10.038,,,,
2185,PDK1,,10.1016/j.cell.2020.10.038,,,,
2185,TNK2,,10.1016/j.cell.2020.10.038,,,,
2185,LIMK2,,10.1016/j.cell.2020.10.038,,,,
2185,BLK,,10.1016/j.cell.2020.10.038,,,,
2185,CSK,,10.1016/j.cell.2020.10.038,,,,
2185,Wee1,,10.1016/j.cell.2020.10.038,,,,
2185,EPHA3,,10.1016/j.cell.2020.10.038,,,,
2185,Src,,10.1016/j.cell.2020.10.038,,,,
2185,YES1,,10.1016/j.cell.2020.10.038,,,,
2185,FYN,,10.1016/j.cell.2020.10.038,,,,
2185,LCK,,10.1016/j.cell.2020.10.038,,,,
2185,ABL1,,10.1016/j.cell.2020.10.038,,,,
2185,EPHB6,,10.1016/j.cell.2020.10.038,,,,
2185,GAK,,10.1016/j.cell.2020.10.038,,,,
2185,AURKA,,10.1016/j.cell.2020.10.038,,,,
2186,TTK,,10.1016/j.cell.2020.10.038,,,,
2186,CDK9,,10.1016/j.cell.2020.10.038,,,,
2186,CDK6,,10.1016/j.cell.2020.10.038,,,,
2186,AAK1,,10.1016/j.cell.2020.10.038,,,,
2186,AURKB,,10.1016/j.cell.2020.10.038,,,,
2186,STK17A,,10.1016/j.cell.2020.10.038,,,,
2186,AURKA,,10.1016/j.cell.2020.10.038,,,,
2186,FGFR2,,10.1016/j.cell.2020.10.038,,,,
2187,CSNK1E,,10.1016/j.cell.2020.10.038,,,,
2187,BLK,,10.1016/j.cell.2020.10.038,,,,
2187,MAP2K5,,10.1016/j.cell.2020.10.038,,,,
2187,LIMK1,,10.1016/j.cell.2020.10.038,,,,
2187,LATS1,,10.1016/j.cell.2020.10.038,,,,
2187,ABL1,,10.1016/j.cell.2020.10.038,,,,
2187,LCK,,10.1016/j.cell.2020.10.038,,,,
2187,FYN,,10.1016/j.cell.2020.10.038,,,,
2187,Src,,10.1016/j.cell.2020.10.038,,,,
2187,CSK,,10.1016/j.cell.2020.10.038,,,,
2187,ABL2,,10.1016/j.cell.2020.10.038,,,,
2188,PTK2B,,10.1016/j.cell.2020.10.038,,,,
2188,AURKA,,10.1016/j.cell.2020.10.038,,,,
2188,LCK,,10.1016/j.cell.2020.10.038,,,,
2188,FER,,10.1016/j.cell.2020.10.038,,,,
2188,CDK2,,10.1016/j.cell.2020.10.038,,,,
2188,Wee1,,10.1016/j.cell.2020.10.038,,,,
2188,CDK7,,10.1016/j.cell.2020.10.038,,,,
2188,CDK9,,10.1016/j.cell.2020.10.038,,,,
2188,BLK,,10.1016/j.cell.2020.10.038,,,,
2188,LIMK2,,10.1016/j.cell.2020.10.038,,,,
2188,CDK5,,10.1016/j.cell.2020.10.038,,,,
2188,CDK17,,10.1016/j.cell.2020.10.038,,,,
2188,ITK,,10.1016/j.cell.2020.10.038,,,,
2188,AAK1,,10.1016/j.cell.2020.10.038,,,,
2188,CDK12,,10.1016/j.cell.2020.10.038,,,,
2189,PTK2B,,10.1016/j.cell.2020.10.038,,,,
2189,ITK,,10.1016/j.cell.2020.10.038,,,,
2189,CDK6,,10.1016/j.cell.2020.10.038,,,,
2189,CDK5,,10.1016/j.cell.2020.10.038,,,,
2189,AURKA,,10.1016/j.cell.2020.10.038,,,,
2189,STK10,,10.1016/j.cell.2020.10.038,,,,
2189,LCK,,10.1016/j.cell.2020.10.038,,,,
2189,CDK4,,10.1016/j.cell.2020.10.038,,,,
2189,FER,,10.1016/j.cell.2020.10.038,,,,
2189,CDK2,,10.1016/j.cell.2020.10.038,,,,
2189,CDK12,,10.1016/j.cell.2020.10.038,,,,
2189,Wee1,,10.1016/j.cell.2020.10.038,,,,
2189,CDK7,,10.1016/j.cell.2020.10.038,,,,
2189,CDK9,,10.1016/j.cell.2020.10.038,,,,
2189,BLK,,10.1016/j.cell.2020.10.038,,,,
2189,LIMK2,,10.1016/j.cell.2020.10.038,,,,
2189,CDK17,,10.1016/j.cell.2020.10.038,,,,
2189,AAK1,,10.1016/j.cell.2020.10.038,,,,
2190,PRAG1,,10.1016/j.cell.2020.10.038,,,,
2190,CDC7,,10.1016/j.cell.2020.10.038,,,,
2190,PLK4,,10.1016/j.cell.2020.10.038,,,,
2190,BCKDK,,10.1016/j.cell.2020.10.038,,,,
2190,AURKA,,10.1016/j.cell.2020.10.038,,,,
2190,GAK,,10.1016/j.cell.2020.10.038,,,,
2190,BUB1,,10.1016/j.cell.2020.10.038,,,,
2190,MAST3,,10.1016/j.cell.2020.10.038,,,,
2190,BUB1B,,10.1016/j.cell.2020.10.038,,,,
2190,ULK1,,10.1016/j.cell.2020.10.038,,,,
2190,STK17B,,10.1016/j.cell.2020.10.038,,,,
2190,CDK14,,10.1016/j.cell.2020.10.038,,,,
2190,LATS1,,10.1016/j.cell.2020.10.038,,,,
2190,ABL1,,10.1016/j.cell.2020.10.038,,,,
2190,LCK,,10.1016/j.cell.2020.10.038,,,,
2190,FYN,,10.1016/j.cell.2020.10.038,,,,
2190,YES1,,10.1016/j.cell.2020.10.038,,,,
2190,CDK4,,10.1016/j.cell.2020.10.038,,,,
2190,Src,,10.1016/j.cell.2020.10.038,,,,
2190,FER,,10.1016/j.cell.2020.10.038,,,,
2190,RPS6KB1,,10.1016/j.cell.2020.10.038,,,,
2190,CDK2,,10.1016/j.cell.2020.10.038,,,,
2190,EPHB2,,10.1016/j.cell.2020.10.038,,,,
2190,Wee1,,10.1016/j.cell.2020.10.038,,,,
2190,AKT2,,10.1016/j.cell.2020.10.038,,,,
2190,TTK,,10.1016/j.cell.2020.10.038,,,,
2190,BMPR1A,,10.1016/j.cell.2020.10.038,,,,
2190,TGFBR1,,10.1016/j.cell.2020.10.038,,,,
2190,CSK,,10.1016/j.cell.2020.10.038,,,,
2190,TEC,,10.1016/j.cell.2020.10.038,,,,
2190,ABL2,,10.1016/j.cell.2020.10.038,,,,
2190,CSNK1D,,10.1016/j.cell.2020.10.038,,,,
2190,CDK7,,10.1016/j.cell.2020.10.038,,,,
2190,CDK9,,10.1016/j.cell.2020.10.038,,,,
2190,BLK,,10.1016/j.cell.2020.10.038,,,,
2190,NEK2,,10.1016/j.cell.2020.10.038,,,,
2190,PLK1,,10.1016/j.cell.2020.10.038,,,,
2190,LIMK1,,10.1016/j.cell.2020.10.038,,,,
2190,LIMK2,,10.1016/j.cell.2020.10.038,,,,
2190,PRKAA2,,10.1016/j.cell.2020.10.038,,,,
2190,EPHB4,,10.1016/j.cell.2020.10.038,,,,
2190,CDK6,,10.1016/j.cell.2020.10.038,,,,
2190,CDK5,,10.1016/j.cell.2020.10.038,,,,
2190,CDK16,,10.1016/j.cell.2020.10.038,,,,
2190,CDK17,,10.1016/j.cell.2020.10.038,,,,
2190,FAK,,10.1016/j.cell.2020.10.038,,,,
2190,CDK18,,10.1016/j.cell.2020.10.038,,,,
2190,TNK2,,10.1016/j.cell.2020.10.038,,,,
2190,ITK,,10.1016/j.cell.2020.10.038,,,,
2190,MAP3K12,,10.1016/j.cell.2020.10.038,,,,
2190,PRKAA1,,10.1016/j.cell.2020.10.038,,,,
2190,MAPK7,,10.1016/j.cell.2020.10.038,,,,
2190,MAP3K1,,10.1016/j.cell.2020.10.038,,,,
2190,TNK1,,10.1016/j.cell.2020.10.038,,,,
2190,PTK6,,10.1016/j.cell.2020.10.038,,,,
2190,CDK13,,10.1016/j.cell.2020.10.038,,,,
2190,PTK2B,,10.1016/j.cell.2020.10.038,,,,
2190,PDK3,,10.1016/j.cell.2020.10.038,,,,
2190,CDK10,,10.1016/j.cell.2020.10.038,,,,
2190,RPS6KA1,,10.1016/j.cell.2020.10.038,,,,
2190,MAP3K11,,10.1016/j.cell.2020.10.038,,,,
2190,MAPK6,,10.1016/j.cell.2020.10.038,,,,
2190,AAK1,,10.1016/j.cell.2020.10.038,,,,
2190,SBK1,,10.1016/j.cell.2020.10.038,,,,
2190,LRRK2,,10.1016/j.cell.2020.10.038,,,,
2190,MAP3K21,,10.1016/j.cell.2020.10.038,,,,
2190,ULK3,,10.1016/j.cell.2020.10.038,,,,
2190,MARK2,,10.1016/j.cell.2020.10.038,,,,
2190,STK32C,,10.1016/j.cell.2020.10.038,,,,
2190,HIPK1,,10.1016/j.cell.2020.10.038,,,,
2190,MAP4K3,,10.1016/j.cell.2020.10.038,,,,
2190,STK40,,10.1016/j.cell.2020.10.038,,,,
2190,COQ8A,,10.1016/j.cell.2020.10.038,,,,
2190,UHMK1,,10.1016/j.cell.2020.10.038,,,,
2190,MAP4K1,,10.1016/j.cell.2020.10.038,,,,
2190,AURKB,,10.1016/j.cell.2020.10.038,,,,
2190,MARK4,,10.1016/j.cell.2020.10.038,,,,
2190,TRPM7,,10.1016/j.cell.2020.10.038,,,,
2190,TRIB3,,10.1016/j.cell.2020.10.038,,,,
2190,RPS6KC1,,10.1016/j.cell.2020.10.038,,,,
2190,RIOK2,,10.1016/j.cell.2020.10.038,,,,
2190,STK33,,10.1016/j.cell.2020.10.038,,,,
2190,SIK2,,10.1016/j.cell.2020.10.038,,,,
2190,MKNK2,,10.1016/j.cell.2020.10.038,,,,
2190,BMP2K,,10.1016/j.cell.2020.10.038,,,,
2190,CDK12,,10.1016/j.cell.2020.10.038,,,,
2190,STK17A,,10.1016/j.cell.2020.10.038,,,,
2190,RPS6KA6,,10.1016/j.cell.2020.10.038,,,,
2190,AKT3,,10.1016/j.cell.2020.10.038,,,,
2191,CDK12,,10.1016/j.cell.2020.10.038,,,,
2191,BMP2K,,10.1016/j.cell.2020.10.038,,,,
2191,AAK1,,10.1016/j.cell.2020.10.038,,,,
2191,RPS6KA1,,10.1016/j.cell.2020.10.038,,,,
2191,CDK6,,10.1016/j.cell.2020.10.038,,,,
2191,CDK5,,10.1016/j.cell.2020.10.038,,,,
2191,CDK17,,10.1016/j.cell.2020.10.038,,,,
2191,ITK,,10.1016/j.cell.2020.10.038,,,,
2191,AURKA,,10.1016/j.cell.2020.10.038,,,,
2191,GAK,,10.1016/j.cell.2020.10.038,,,,
2191,LCK,,10.1016/j.cell.2020.10.038,,,,
2191,CDK4,,10.1016/j.cell.2020.10.038,,,,
2191,PRKAA1,,10.1016/j.cell.2020.10.038,,,,
2191,Src,,10.1016/j.cell.2020.10.038,,,,
2191,CDK13,,10.1016/j.cell.2020.10.038,,,,
2191,FER,,10.1016/j.cell.2020.10.038,,,,
2191,CDK2,,10.1016/j.cell.2020.10.038,,,,
2191,Wee1,,10.1016/j.cell.2020.10.038,,,,
2191,ABL2,,10.1016/j.cell.2020.10.038,,,,
2191,PTK2B,,10.1016/j.cell.2020.10.038,,,,
2191,CDK7,,10.1016/j.cell.2020.10.038,,,,
2191,CDK9,,10.1016/j.cell.2020.10.038,,,,
2191,BLK,,10.1016/j.cell.2020.10.038,,,,
2191,LIMK2,,10.1016/j.cell.2020.10.038,,,,
2192,GAK,,10.1016/j.cell.2020.10.038,,,,
2192,AURKA,,10.1016/j.cell.2020.10.038,,,,
2192,PLK4,,10.1016/j.cell.2020.10.038,,,,
2192,EEF2K,,10.1016/j.cell.2020.10.038,,,,
2192,CDK5,,10.1016/j.cell.2020.10.038,,,,
2192,LIMK2,,10.1016/j.cell.2020.10.038,,,,
2192,LIMK1,,10.1016/j.cell.2020.10.038,,,,
2192,NEK2,,10.1016/j.cell.2020.10.038,,,,
2192,BLK,,10.1016/j.cell.2020.10.038,,,,
2192,CDK9,,10.1016/j.cell.2020.10.038,,,,
2192,CDK7,,10.1016/j.cell.2020.10.038,,,,
2192,CSNK1E,,10.1016/j.cell.2020.10.038,,,,
2192,CSNK1D,,10.1016/j.cell.2020.10.038,,,,
2192,ABL2,,10.1016/j.cell.2020.10.038,,,,
2192,TEC,,10.1016/j.cell.2020.10.038,,,,
2192,BMPR1A,,10.1016/j.cell.2020.10.038,,,,
2192,Wee1,,10.1016/j.cell.2020.10.038,,,,
2192,CDK2,,10.1016/j.cell.2020.10.038,,,,
2192,FLT1,,10.1016/j.cell.2020.10.038,,,,
2192,FER,,10.1016/j.cell.2020.10.038,,,,
2192,Src,,10.1016/j.cell.2020.10.038,,,,
2192,CDK4,,10.1016/j.cell.2020.10.038,,,,
2192,YES1,,10.1016/j.cell.2020.10.038,,,,
2192,LCK,,10.1016/j.cell.2020.10.038,,,,
2192,STK10,,10.1016/j.cell.2020.10.038,,,,
2192,ULK1,,10.1016/j.cell.2020.10.038,,,,
2192,BUB1B,,10.1016/j.cell.2020.10.038,,,,
2192,BUB1,,10.1016/j.cell.2020.10.038,,,,
2192,PRKAA1,,10.1016/j.cell.2020.10.038,,,,
2192,ITK,,10.1016/j.cell.2020.10.038,,,,
2192,TNK2,,10.1016/j.cell.2020.10.038,,,,
2192,CDK17,,10.1016/j.cell.2020.10.038,,,,
2192,CDK6,,10.1016/j.cell.2020.10.038,,,,
2192,STK17A,,10.1016/j.cell.2020.10.038,,,,
2192,NLK,,10.1016/j.cell.2020.10.038,,,,
2192,CDK12,,10.1016/j.cell.2020.10.038,,,,
2192,IRAK4,,10.1016/j.cell.2020.10.038,,,,
2192,SIK2,,10.1016/j.cell.2020.10.038,,,,
2192,RIOK2,,10.1016/j.cell.2020.10.038,,,,
2192,MARK4,,10.1016/j.cell.2020.10.038,,,,
2192,AURKB,,10.1016/j.cell.2020.10.038,,,,
2192,COQ8B,,10.1016/j.cell.2020.10.038,,,,
2192,MAP4K1,,10.1016/j.cell.2020.10.038,,,,
2192,HASPIN,,10.1016/j.cell.2020.10.038,,,,
2192,STK35,,10.1016/j.cell.2020.10.038,,,,
2192,COQ8A,,10.1016/j.cell.2020.10.038,,,,
2192,MAP4K3,,10.1016/j.cell.2020.10.038,,,,
2192,PRAG1,,10.1016/j.cell.2020.10.038,,,,
2192,MARK2,,10.1016/j.cell.2020.10.038,,,,
2192,ULK3,,10.1016/j.cell.2020.10.038,,,,
2192,MAP3K21,,10.1016/j.cell.2020.10.038,,,,
2192,AAK1,,10.1016/j.cell.2020.10.038,,,,
2192,MAPK6,,10.1016/j.cell.2020.10.038,,,,
2192,MAP3K11,,10.1016/j.cell.2020.10.038,,,,
2192,RPS6KA1,,10.1016/j.cell.2020.10.038,,,,
2192,CDK10,,10.1016/j.cell.2020.10.038,,,,
2192,PDK2,,10.1016/j.cell.2020.10.038,,,,
2192,PTK2B,,10.1016/j.cell.2020.10.038,,,,
2192,CDK13,,10.1016/j.cell.2020.10.038,,,,
2192,MAPK7,,10.1016/j.cell.2020.10.038,,,,
2193,MAP3K20,,10.1016/j.cell.2020.10.038,,,,
2193,p38alpha,,10.1016/j.cell.2020.10.038,,,,
2193,LIMK1,,10.1016/j.cell.2020.10.038,,,,
2193,CDK4,,10.1016/j.cell.2020.10.038,,,,
2193,MAST3,,10.1016/j.cell.2020.10.038,,,,
2194,FER,,10.1016/j.cell.2020.10.038,,,,
2194,MARK4,,10.1016/j.cell.2020.10.038,,,,
2194,AURKB,,10.1016/j.cell.2020.10.038,,,,
2194,ULK3,,10.1016/j.cell.2020.10.038,,,,
2194,AAK1,,10.1016/j.cell.2020.10.038,,,,
2194,MAP3K11,,10.1016/j.cell.2020.10.038,,,,
2194,RPS6KA1,,10.1016/j.cell.2020.10.038,,,,
2194,STK38,,10.1016/j.cell.2020.10.038,,,,
2194,CDK13,,10.1016/j.cell.2020.10.038,,,,
2194,PRKAA1,,10.1016/j.cell.2020.10.038,,,,
2194,ITK,,10.1016/j.cell.2020.10.038,,,,
2194,TNK2,,10.1016/j.cell.2020.10.038,,,,
2194,CDK17,,10.1016/j.cell.2020.10.038,,,,
2194,CDK5,,10.1016/j.cell.2020.10.038,,,,
2194,CDK6,,10.1016/j.cell.2020.10.038,,,,
2194,LIMK2,,10.1016/j.cell.2020.10.038,,,,
2194,LIMK1,,10.1016/j.cell.2020.10.038,,,,
2194,BLK,,10.1016/j.cell.2020.10.038,,,,
2194,CDK9,,10.1016/j.cell.2020.10.038,,,,
2194,CDK7,,10.1016/j.cell.2020.10.038,,,,
2194,ABL2,,10.1016/j.cell.2020.10.038,,,,
2194,TEC,,10.1016/j.cell.2020.10.038,,,,
2194,Wee1,,10.1016/j.cell.2020.10.038,,,,
2194,CDK2,,10.1016/j.cell.2020.10.038,,,,
2194,Src,,10.1016/j.cell.2020.10.038,,,,
2194,CDK4,,10.1016/j.cell.2020.10.038,,,,
2194,LCK,,10.1016/j.cell.2020.10.038,,,,
2194,STK10,,10.1016/j.cell.2020.10.038,,,,
2194,ULK1,,10.1016/j.cell.2020.10.038,,,,
2194,BUB1B,,10.1016/j.cell.2020.10.038,,,,
2194,AURKA,,10.1016/j.cell.2020.10.038,,,,
2194,PLK4,,10.1016/j.cell.2020.10.038,,,,
2195,PIP4K2C,,10.1016/j.cell.2020.10.038,,N.D.,,
2195,PIP4K2B,,10.1016/j.cell.2020.10.038,,N.D.,,
2195,PIP4K2A,,10.1016/j.cell.2020.10.038,,N.D.,,
2196,PAK4,,10.1016/j.cell.2020.10.038,,,,
2196,CSNK1A1,,10.1016/j.cell.2020.10.038,,,,
2196,CSNK1D,,10.1016/j.cell.2020.10.038,,,,
2196,CSNK1E,,10.1016/j.cell.2020.10.038,,,,
2196,GSK3A,,10.1016/j.cell.2020.10.038,,,,
2196,GSK-3beta,,10.1016/j.cell.2020.10.038,,,,
2196,LIMK2,,10.1016/j.cell.2020.10.038,,,,
2196,STK4,,10.1016/j.cell.2020.10.038,,,,
2196,MAP3K1,,10.1016/j.cell.2020.10.038,,,,
2196,STK35,,10.1016/j.cell.2020.10.038,,,,
2196,MINK1,,10.1016/j.cell.2020.10.038,,,,
2196,STK17B,,10.1016/j.cell.2020.10.038,,,,
2196,STK10,,10.1016/j.cell.2020.10.038,,,,
2197,GSK3A,,10.1016/j.cell.2020.10.038,,,,
2197,STK4,,10.1016/j.cell.2020.10.038,,,,
2197,NUAK1,,10.1016/j.cell.2020.10.038,,,,
2197,PIM2,,10.1016/j.cell.2020.10.038,,,,
2197,STK17B,,10.1016/j.cell.2020.10.038,,,,
2197,CDK14,,10.1016/j.cell.2020.10.038,,,,
2197,CSNK1D,,10.1016/j.cell.2020.10.038,,,,
2197,GSK-3beta,,10.1016/j.cell.2020.10.038,,,,
2198,BLK,,10.1016/j.cell.2020.10.038,,,,
2198,STK17A,,10.1016/j.cell.2020.10.038,,,,
2198,LIMK1,,10.1016/j.cell.2020.10.038,,,,
2198,LIMK2,,10.1016/j.cell.2020.10.038,,,,
2198,TNK2,,10.1016/j.cell.2020.10.038,,,,
2199,CLK1,,10.1016/j.cell.2020.10.038,,,,
2199,CDK9,,10.1016/j.cell.2020.10.038,,,,
2200,ALK,,10.1016/j.ejmech.2021.113335,,,,
2201,ALK,0/0/4/30/47 (WB),10.1016/j.ejmech.2021.113335,,,,% ALK degradation in SR cells at 0.05/0.5/5/50/500 nM
2202,ALK,,10.1016/j.ejmech.2021.113335,,,,
2202,ALK,77.3/96.9,10.1021/acs.jmedchem.1c00270,,,,% ALK degradation in H3122 cells after 16 h treatment at 100/1000 nM
2203,ALK,4/0/0/7/57 (WB),10.1016/j.ejmech.2021.113335,,,,% ALK degradation in SR cells at 0.05/0.5/5/50/500 nM
2204,ALK,0/7/0/7/49 (WB),10.1016/j.ejmech.2021.113335,,,,% ALK degradation in SR cells at 0.05/0.5/5/50/500 nM
2205,ALK,,10.1016/j.ejmech.2021.113335,,,,
2206,ALK,,10.1016/j.ejmech.2021.113335,,,,
2207,ALK,,10.1016/j.ejmech.2021.113335,,,,
2208,ALK,,10.1016/j.ejmech.2021.113335,,,,
2209,ALK,,10.1021/acs.jmedchem.1c00270,27.4/116.5,,Degradation of ALK in H3122/Karpas 299 cells after 16/48 h treatment,
2209,ALK,,10.1016/j.ejmech.2021.113335,,,,
2210,ALK,,10.1016/j.ejmech.2021.113335,,,,
2210,ALK,77.4/85.9,10.1021/acs.jmedchem.1c00270,,,,% ALK degradation in Karpas 299 cells after 24 h treatment at 100/1000 nM
2211,ALK,,10.1016/j.ejmech.2021.113335,,,,
2211,ALK,55.1/71.6,10.1021/acs.jmedchem.1c00270,,,,% ALK degradation in Karpas 299 cells after 24 h treatment at 100/1000 nM
2212,ALK,,10.1016/j.ejmech.2021.113335,,,,
2213,ALK,,10.1016/j.ejmech.2021.113335,,,,
2214,ALK,,10.1016/j.ejmech.2021.113335,,,,
2215,ALK,0/18/34/45/53 (WB),10.1016/j.ejmech.2021.113335,,,,% ALK degradation in SR cells at 0.05/0.5/5/50/500 nM
2216,ALK,,10.1016/j.ejmech.2021.113335,,,,
2217,ALK,,10.1016/j.ejmech.2021.113335,6.1,87.7,Degradation of ALK in SR cells,
2217,ALK G1202R,,10.1016/j.ejmech.2021.113335,,,,
2218,ALK,,10.1016/j.ejmech.2021.113335,,,,
2219,ALK,,10.1016/j.ejmech.2021.113335,,,,
2220,ALK,,10.1016/j.ejmech.2021.113335,,,,
2221,ALK,,10.1016/j.ejmech.2021.113335,,,,
2222,ALK G1202R,,10.1016/j.ejmech.2021.113335,200,,Degradation of ALK G1202R in 293T cells,
2222,ALK,,10.1016/j.ejmech.2021.113335,3.9,70.3,Degradation of ALK in SR cells,
2223,ALK,,10.1016/j.ejmech.2021.113335,,,,
2224,ALK,0/0/24/33/31 (WB),10.1016/j.ejmech.2021.113335,,,,DC50 of ALK in SR cells (nM)
2225,ALK,,10.1016/j.ejmech.2021.113335,,,,
2226,ALK,,10.1016/j.ejmech.2021.113335,,,,
2227,EGFR e19d,,10.1016/j.ejmech.2021.113328,,,,
2227,EGFR L858R/T790M,,10.1016/j.ejmech.2021.113328,,,,
2228,EGFR L858R/T790M,,10.1016/j.ejmech.2021.113328,,,,
2228,EGFR e19d,,10.1016/j.ejmech.2021.113328,,,,
2229,EGFR L858R/T790M,,10.1016/j.ejmech.2021.113328,,,,
2229,EGFR e19d,,10.1016/j.ejmech.2021.113328,,,,
2230,EGFR L858R/T790M,,10.1016/j.ejmech.2021.113328,,,,
2230,EGFR e19d,,10.1016/j.ejmech.2021.113328,,,,
2231,EGFR L858R/T790M,,10.1016/j.ejmech.2021.113328,30-50/100,,Degradation of EGFR L858R/T790M in H1975/(Ba/F3) cells after 16 h treatment,
2231,EGFR e19d,,10.1016/j.ejmech.2021.113328,100,40,Degradation of EGFR e19d in PC9 cells after 48 h treatment,
2232,EGFR L858R/T790M,,10.1016/j.ejmech.2021.113328,<30/100,,Degradation of EGFR L858R/T790M in H1975/(Ba/F3) cells after 16 h treatment,
2232,EGFR e19d,,10.1016/j.ejmech.2021.113328,30-100,,Degradation of EGFR e19d in PC9 cells after 48 h treatment,
2233,SHP2,,10.1016/j.ejmech.2021.113341,,,,
2234,SHP2,,10.1016/j.ejmech.2021.113341,,,,
2235,SHP2,,10.1016/j.ejmech.2021.113341,,,,
2236,SHP2,,10.1016/j.ejmech.2021.113341,6.02,,Degradation of SHP2 in MV4;11 cells after 12 h treatment,
2237,SHP2,,10.1016/j.ejmech.2021.113341,,,,
2238,SHP2,,10.1016/j.ejmech.2021.113341,,,,
2239,SHP2,,10.1016/j.ejmech.2021.113341,,,,
2240,SHP2,,10.1016/j.ejmech.2021.113341,,,,
2241,SHP2,,10.1016/j.ejmech.2021.113341,,,,
2242,SHP2,,10.1016/j.ejmech.2021.113341,,,,
2243,SHP2,,10.1016/j.ejmech.2021.113341,,,,
2244,SHP2,,10.1016/j.ejmech.2021.113341,,,,
2245,SHP2,,10.1016/j.ejmech.2021.113341,,,,
2246,SHP2,,10.1016/j.ejmech.2021.113341,,,,
2247,PARP14,,10.1002/cbic.202100047,5,,Degradation of PARP14 in KYSE-270 cells after 24 h treatment,
2248,CDK12,,10.1038/s41589-021-00765-y,,,,
2249,CDK12,,10.1038/s41589-021-00765-y,,,,
2250,CDK12,,10.1038/s41589-021-00765-y,,,,
2251,CDK12,,10.1038/s41589-021-00765-y,,,,
2251,CDK12 C1039F,,10.1038/s41589-021-00765-y,,,,
2252,CDK12,,10.1038/s41589-021-00765-y,,,,
2253,CDK12,,10.1038/s41589-021-00765-y,,,,
2254,CDK12,,10.1038/s41589-021-00765-y,,,,
2255,CDK12,,10.1038/s41589-021-00765-y,,,,
2255,CDK12 C1039F,,10.1038/s41589-021-00765-y,,,,
2256,FKBP12,,10.1021/jacs.1c00990,,,,
2257,FKBP12,,10.1021/jacs.1c00990,,,,
2258,AR,,10.1021/jacs.1c00990,,,,
2259,FLT3-ITD,,10.1021/acs.jmedchem.1c00996,8/6.9,,Degradation of FLT3-ITD in MOLM-13/MV-4-11 cells after 24 h treatment,
2260,FLT3-ITD,,10.1021/acs.jmedchem.1c00996,7.4/9.1,,Degradation of FLT3-ITD in MOLM-13/MV-4-11 cells after 24 h treatment,
2261,FLT3-ITD,,10.1021/acs.jmedchem.1c00996,,,,
2262,FLT3-ITD,,10.1021/acs.jmedchem.1c00996,,,,
2263,FLT3-ITD,,10.1021/acs.jmedchem.1c00996,,,,
2264,FLT3-ITD,,10.1021/acs.jmedchem.1c00996,,,,
2265,FLT3-ITD,,10.1021/acs.jmedchem.1c00996,,,,
2266,FLT3-ITD,,10.1021/acs.jmedchem.1c00996,,,,
2267,FLT3-ITD,,10.1021/acs.jmedchem.1c00996,,,,
2268,FLT3-ITD,,10.1021/acs.jmedchem.1c00996,,,,
2269,FLT3-ITD,,10.1021/acs.jmedchem.1c00996,,,,
2270,FLT3-ITD,,10.1021/acs.jmedchem.1c00996,,,,
2271,FLT3-ITD,,10.1021/acs.jmedchem.1c00996,,,,
2272,FLT3-ITD,,10.1021/acs.jmedchem.1c00996,,,,
2273,FLT3-ITD,,10.1021/acs.jmedchem.1c00996,,,,
2274,FLT3-ITD,,10.1021/acs.jmedchem.1c00996,,,,
2275,WDR5,,10.1021/acs.jmedchem.1c00146,,N.D.,,
2276,WDR5,,10.1021/acs.jmedchem.1c00146,,N.D.,,
2277,WDR5,,10.1021/acs.jmedchem.1c00146,,N.D.,,
2278,WDR5,,10.1021/acs.jmedchem.1c00146,,N.D.,,
2279,WDR5,,10.1021/acs.jmedchem.1c00146,,N.D.,,
2280,WDR5,,10.1021/acs.jmedchem.1c00146,,N.D.,,
2281,WDR5,,10.1021/acs.jmedchem.1c00146,,N.D.,,
2282,WDR5,,10.1021/acs.jmedchem.1c00146,,N.D.,,
2283,WDR5,,10.1021/acs.jmedchem.1c00146,,N.D.,,
2284,WDR5,,10.1021/acs.jmedchem.1c00146,625,,Degradation of WDR5-HiBiT in MV4-11 (WDR5-HiBiT) cells after 24 h treatment,
2285,WDR5,,10.1021/acs.jmedchem.1c00146,116,,Degradation of WDR5-HiBiT in MV4-11 (WDR5-HiBiT) cells after 24 h treatment,
2286,WDR5,,10.1021/acs.jmedchem.1c00146,53,,Degradation of WDR5-HiBiT in MV4-11 (WDR5-HiBiT) cells after 24 h treatment,
2287,WDR5,,10.1021/acs.jmedchem.1c00146,920,,Degradation of WDR5-HiBiT in MV4-11 (WDR5-HiBiT) cells after 24 h treatment,
2288,WDR5,,10.1021/acs.jmedchem.1c00146,915,,Degradation of WDR5-HiBiT in MV4-11 (WDR5-HiBiT) cells after 24 h treatment,
2289,WDR5,,10.1021/acs.jmedchem.1c00146,,,,
2290,WDR5,,10.1021/acs.jmedchem.1c00146,,,,
2291,WDR5,,10.1021/acs.jmedchem.1c00146,,,,
2292,WDR5,,10.1021/acs.jmedchem.1c00146,,,,
2293,WDR5,,10.1021/acs.jmedchem.1c00146,,N.D.,,
2294,WDR5,,10.1021/acs.jmedchem.1c00146,1240,,Degradation of WDR5-HiBiT in MV4-11 (WDR5-HiBiT) cells after 24 h treatment,
2295,WDR5,,10.1021/acs.jmedchem.1c00146,,N.D.,,
2296,WDR5,,10.1021/acs.jmedchem.1c00146,,N.D.,,
2297,WDR5,,10.1021/acs.jmedchem.1c00146,,N.D.,,
2298,WDR5,,10.1021/acs.jmedchem.1c00146,,N.D.,,
2299,WDR5,,10.1021/acs.jmedchem.1c00146,,N.D.,,
2300,AR,0/25/63/70,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2301,AR,42/76/55/21,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2302,AR,49/84/89/97,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2303,AR,69/85/77/79,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2304,AR,28/58/79/62,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2305,AR,48/76/82/73,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2306,AR,58/83/79/76,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2307,AR,22/37/54/53,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2308,AR,42/63/84/82,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2309,AR,12/59/85/60,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2310,AR,<5/9/36/38,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2311,AR,10/22/43/48,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2312,AR,<5/23/41/32,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2313,AR,<5/<5/<5/9,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2314,AR,7/40/47/32,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2315,AR,54/77/91/73,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2316,AR,64/96/98/90,10.1021/acs.jmedchem.1c00882,0.15/5.08,,Degradation of AR in VCaP/LNCaP cells after 24 h treatment,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2317,AR,79/93/85/55,10.1021/acs.jmedchem.1c00882,0.76/1.41,,Degradation of AR in VCaP/LNCaP cells after 24 h treatment,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2318,AR,62/94/98/96,10.1021/acs.jmedchem.1c00882,0.28/8.3,,Degradation of AR in VCaP/LNCaP cells after 24 h treatment,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2319,AR,71/83/95/83,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2320,AR,65/92/96/79,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2321,AR,85/97/96/83,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2322,AR,76/97/97/96,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2323,AR,57/93/96/85,10.1021/acs.jmedchem.1c00882,0.12/1.43,,Degradation of AR in VCaP/LNCaP cells after 24 h treatment,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2324,AR,40/96/99/99,10.1021/acs.jmedchem.1c00882,0.38/3.38,,Degradation of AR in VCaP/LNCaP cells after 24 h treatment,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2325,AR,37/78/93/88,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2326,AR,30/82/97/95,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2327,AR,38/80/87/84,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2328,AR,16/56/71/51,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2329,AR,14/38/67/80,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2330,AR,15/48/73/82,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2331,AR,0/16/82/88,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2332,AR,13/30/38/57,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2333,AR,<5/19/75/90,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2334,AR,<5/30/25/39,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2335,AR,<5/15/75/80,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2336,AR,22/45/87/90,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2337,AR,6/12/33/41,10.1021/acs.jmedchem.1c00882,,,,% AR degradation in VCaP cells after 6 h treatment at 1/10/100/1000 nM
2338,BRD3,,10.1021/acs.jmedchem.1c01496,158.5,,Degradation of BRD3 in HEK293 cells after 4 h treatment,
2338,BRD4,,10.1021/acs.jmedchem.1c01496,125.89,,Degradation of BRD4 long in HEK293 cells after 4 h treatment,
2338,BRD2,,10.1021/acs.jmedchem.1c01496,158.5,,Degradation of BRD2 in HEK293 cells after 4 h treatment,
2339,BRD3,,10.1021/acs.jmedchem.1c01496,199.5,,Degradation of BRD3 in HEK293 cells after 4 h treatment,
2339,BRD2,,10.1021/acs.jmedchem.1c01496,251.2,,Degradation of BRD2 in HEK293 cells after 4 h treatment,
2339,BRD4,,10.1021/acs.jmedchem.1c01496,125.89,,Degradation of BRD4 long in HEK293 cells after 4 h treatment,
2340,BRD3,,10.1021/acs.jmedchem.1c01496,199.5,,Degradation of BRD3 in HEK293 cells after 4 h treatment,
2340,BRD4,,10.1021/acs.jmedchem.1c01496,39.81,,Degradation of BRD4 long in HEK293 cells after 4 h treatment,
2340,BRD2,,10.1021/acs.jmedchem.1c01496,125.9,,Degradation of BRD2 in HEK293 cells after 4 h treatment,
2341,BRD3,,10.1021/acs.jmedchem.1c01496,4,,Degradation of BRD3 in HEK293 cells after 4 h treatment,
2341,BRD2,,10.1021/acs.jmedchem.1c01496,1.3,,Degradation of BRD2 in HEK293 cells after 4 h treatment,
2341,BRD4,,10.1021/acs.jmedchem.1c01496,6.31,,Degradation of BRD4 long in HEK293 cells after 4 h treatment,
2342,BRD3,,10.1021/acs.jmedchem.1c01496,100,,Degradation of BRD3 in HEK293 cells after 4 h treatment,
2342,BRD4,,10.1021/acs.jmedchem.1c01496,63.1,,Degradation of BRD4 long in HEK293 cells after 4 h treatment,
2342,BRD2,,10.1021/acs.jmedchem.1c01496,79.4,,Degradation of BRD2 in HEK293 cells after 4 h treatment,
2343,BRD4,,10.1021/acs.jmedchem.1c01496,31.62,,Degradation of BRD4 long in HEK293 cells after 4 h treatment,
2343,BRD3,,10.1021/acs.jmedchem.1c01496,63.1,,Degradation of BRD3 in HEK293 cells after 4 h treatment,
2343,BRD2,,10.1021/acs.jmedchem.1c01496,63.1,,Degradation of BRD2 in HEK293 cells after 4 h treatment,
2344,TTK,,10.1021/acs.jmedchem.1c01768,>1000,,Degradation of TTK in HCT-116 cells after 6 h treatment,
2345,TTK,,10.1021/acs.jmedchem.1c01768,>1000,,Degradation of TTK in HCT-116 cells after 6 h treatment,
2346,TTK,,10.1021/acs.jmedchem.1c01768,>1000,,Degradation of TTK in HCT-116 cells after 6 h treatment,
2347,TTK,,10.1021/acs.jmedchem.1c01768,>1000,,Degradation of TTK in HCT-116 cells after 6 h treatment,
2348,TTK,,10.1021/acs.jmedchem.1c01768,598.7/>1000,28/43,Degradation of TTK in COLO-205/HCT-116 cells after 6 h treatment,
2349,TTK,,10.1021/acs.jmedchem.1c01768,4.97/20.3,76/50,Degradation of TTK in COLO-205/HCT-116 cells after 6 h treatment,
2350,TTK,,10.1021/acs.jmedchem.1c01768,7.05/58.1,84/53,Degradation of TTK in COLO-205/HCT-116 cells after 6 h treatment,
2351,TTK,,10.1021/acs.jmedchem.1c01768,2.25/49.6,87/66,Degradation of TTK in COLO-205/HCT-116 cells after 6 h treatment,
2352,TTK,,10.1021/acs.jmedchem.1c01768,1.75/5.8,88/80,Degradation of TTK in COLO-205/HCT-116 cells after 6 h treatment,
2353,TTK,,10.1021/acs.jmedchem.1c01768,1.55/35,86/61,Degradation of TTK in COLO-205/HCT-116 cells after 6 h treatment,
2354,TTK,,10.1021/acs.jmedchem.1c01768,3.04/663,85/50,Degradation of TTK in COLO-205/HCT-116 cells after 6 h treatment,
2355,TTK,,10.1021/acs.jmedchem.1c01768,5.6/30.2,85/83,Degradation of TTK in COLO-205/HCT-116 cells after 6 h treatment,
2356,TTK,,10.1021/acs.jmedchem.1c01768,3.31/25.4,77/57,Degradation of TTK in COLO-205/HCT-116 cells after 6 h treatment,
2357,TTK,,10.1021/acs.jmedchem.1c01768,3.15/12.4,82/77,Degradation of TTK in COLO-205/HCT-116 cells after 6 h treatment,
2358,TTK,,10.1021/acs.jmedchem.1c01768,7.03/161,84/43,Degradation of TTK in COLO-205/HCT-116 cells after 6 h treatment,
2359,TTK,,10.1021/acs.jmedchem.1c01768,19.09/74.5,87/66,Degradation of TTK in COLO-205/HCT-116 cells after 6 h treatment,
2360,TTK,,10.1021/acs.jmedchem.1c01768,30.28/>1000,64/28,Degradation of TTK in COLO-205/HCT-116 cells after 6 h treatment,
2361,TTK,,10.1021/acs.jmedchem.1c01768,31.35/>1000,72/41,Degradation of TTK in COLO-205/HCT-116 cells after 6 h treatment,
2362,TTK,,10.1021/acs.jmedchem.1c01768,46/496,73/37,Degradation of TTK in COLO-205/HCT-116 cells after 6 h treatment,
2363,TTK,,10.1021/acs.jmedchem.1c01768,21.71/>1000,88/13,Degradation of TTK in COLO-205/HCT-116 cells after 6 h treatment,
2364,RIPK2,,10.1021/acs.jmedchem.1c01118,,,,
2365,RIPK2,,10.1021/acs.jmedchem.1c01118,,,,
2366,RIPK2,,10.1021/acs.jmedchem.1c01118,,,,
2367,RIPK2,,10.1021/acs.jmedchem.1c01118,,,,
2368,RIPK2,,10.1021/acs.jmedchem.1c01118,,,,
2369,RIPK2,,10.1021/acs.jmedchem.1c01118,,,,
2370,RIPK2,,10.1021/acs.jmedchem.1c01118,,,,
2371,RIPK2,,10.1021/acs.jmedchem.1c01118,,,,
2372,RIPK2,,10.1021/acs.jmedchem.1c01118,,,,
2373,RIPK2,,10.1021/acs.jmedchem.1c01118,,,,
2374,RIPK2,,10.1021/acs.jmedchem.1c01118,,,,
2375,RIPK2,,10.1021/acs.jmedchem.1c01118,,,,
2376,RIPK2,,10.1021/acs.jmedchem.1c01118,0.13,,Degradation of RIPK2 in THP1 cells after 18 h treatment,
2377,RIPK2,,10.1021/acs.jmedchem.1c01118,0.16,,Degradation of RIPK2 in THP1 cells after 18 h treatment,
2378,RIPK2,,10.1021/acs.jmedchem.1c01118,0.1,,Degradation of RIPK2 in THP1 cells after 18 h treatment,
2379,RIPK2,,10.1021/acs.jmedchem.1c01118,0.05,,Degradation of RIPK2 in THP1 cells after 18 h treatment,
2380,RIPK2,,10.1021/acs.jmedchem.1c01118,0.16,,Degradation of RIPK2 in THP1 cells after 18 h treatment,
2381,BCL-xL,,10.1021/acs.jmedchem.1c00517,,,,
2382,BCL-xL,,10.1021/acs.jmedchem.1c00517,,,,
2383,BCL-xL,,10.1021/acs.jmedchem.1c00517,,,,
2384,BCL-xL,,10.1021/acs.jmedchem.1c00517,,,,
2385,BCL-xL,,10.1021/acs.jmedchem.1c00517,31.6/22.6,,Degradation of BCL-xL in MOLT-4/RS4;11 cells after 16 h treatment,
2386,BCL-xL,,10.1021/acs.jmedchem.1c00517,,,,
2387,BCL-xL,,10.1021/acs.jmedchem.1c00517,,,,
2388,BCL-xL,,10.1021/acs.jmedchem.1c00517,,,,
2389,BCL-xL,,10.1021/acs.jmedchem.1c00517,127.4/75.2,,Degradation of BCL-xL in MOLT-4/RS4;11 cells after 16 h treatment,
2390,BCL-xL,,10.1021/acs.jmedchem.1c00517,14.3/11.6,,Degradation of BCL-xL in MOLT-4/RS4;11 cells after 16 h treatment,
2391,ALK,,10.1021/acs.jmedchem.1c00373,,,,
2392,ALK,,10.1021/acs.jmedchem.1c00373,,,,
2393,ALK,,10.1021/acs.jmedchem.1c00373,,,,
2394,ALK,,10.1021/acs.jmedchem.1c00373,,,,
2395,ALK,,10.1021/acs.jmedchem.1c00373,,,,
2396,ALK,,10.1021/acs.jmedchem.1c00373,<10,,Degradation of ALK in SR cells after 24 h treatment,
2396,FAK,,10.1021/acs.jmedchem.1c00373,<1/<1/<1,,Degradation of FAK in NCI-H2228/A549/Calu-1 cells after 16 h treatment,
2396,ALK G1202R,,10.1021/acs.jmedchem.1c00373,<100,,Degradation of ALK G1202R in 293T cells after 72 h treatment,
2396,PTK2B,,10.1021/acs.jmedchem.1c00373,<1,,Degradation of PYK2 in SR cells after 24 h treatment,
2396,PTK6,,10.1021/acs.jmedchem.1c00373,<1,,Degradation of PTK6 in MDA-MB-231 cells after 16 h treatment,
2396,EGFR L858R/T790M,,10.1021/acs.jmedchem.1c00373,<100,,Degradation of EGFR L858R/T790M in H1975 cells after 72 h treatment,
2396,FER,,10.1021/acs.jmedchem.1c00373,<10,,Degradation of FER in SR cells after 24 h treatment,
2396,RPS6KA1,,10.1021/acs.jmedchem.1c00373,<100/<100/<100,,Degradation of RSK1 in NCI-H2228/A549/Calu-1 cells after 16 h treatment,
2397,ALK,,10.1021/acs.jmedchem.1c00373,,,,
2398,ALK,,10.1021/acs.jmedchem.1c00373,,,,
2399,ALK,,10.1021/acs.jmedchem.1c00373,,,,
2400,ALK,,10.1021/acs.jmedchem.1c00373,,,,
2401,ALK,,10.1021/acs.jmedchem.1c00373,,,,
2402,EGFR e19d,,10.1016/j.bioorg.2022.105605,,,,
2403,EGFR e19d,,10.1016/j.bioorg.2022.105605,,,,
2404,EGFR e19d,,10.1016/j.bioorg.2022.105605,,,,
2405,EGFR e19d,,10.1016/j.bioorg.2022.105605,,,,
2406,EGFR e19d,,10.1016/j.bioorg.2022.105605,,,,
2407,EGFR e19d,,10.1016/j.bioorg.2022.105605,,,,
2408,EGFR e19d,,10.1016/j.bioorg.2022.105605,,,,
2409,EGFR e19d,,10.1016/j.bioorg.2022.105605,,,,
2410,EGFR e19d,,10.1016/j.bioorg.2022.105605,,,,
2411,EGFR e19d,,10.1016/j.bioorg.2022.105605,7.95,98,Degradation of EGFR del19 in HCC-827 cells after 72 h treatment,
2412,EGFR e19d,,10.1016/j.bioorg.2022.105605,,,,
2413,EGFR e19d,,10.1016/j.bioorg.2022.105605,,,,
2414,EGFR e19d,,10.1016/j.bioorg.2022.105605,3.57,91,Degradation of EGFR del19 in HCC-827 cells after 72 h treatment,
2415,EGFR e19d,,10.1016/j.bioorg.2022.105605,,,,
2416,EGFR e19d,,10.1016/j.bioorg.2022.105605,,,,
2417,EGFR,,10.1021/acs.jmedchem.1c02221,,N.D.,,
2418,EGFR,,10.1021/acs.jmedchem.1c02221,36.51,,Degradation of EGFR in HCC-827 cells after 72 h treatment,
2419,HDAC2,,10.1021/acs.jmedchem.1c02179,,32,,
2419,HDAC1,,10.1021/acs.jmedchem.1c02179,,41,,
2419,HDAC3,,10.1021/acs.jmedchem.1c02179,,3,,
2420,HDAC1,,10.1021/acs.jmedchem.1c02179,,54,,
2420,HDAC3,,10.1021/acs.jmedchem.1c02179,,23,,
2420,HDAC2,,10.1021/acs.jmedchem.1c02179,,37,,
2421,HDAC3,,10.1021/acs.jmedchem.1c02179,,33,,
2421,HDAC1,,10.1021/acs.jmedchem.1c02179,,67,,
2421,HDAC2,,10.1021/acs.jmedchem.1c02179,,43,,
2422,HDAC3,,10.1021/acs.jmedchem.1c02179,,44,,
2422,HDAC2,,10.1021/acs.jmedchem.1c02179,,44,,
2422,HDAC1,,10.1021/acs.jmedchem.1c02179,,63,,
2423,HDAC1,,10.1021/acs.jmedchem.1c02179,,60,,
2423,HDAC3,,10.1021/acs.jmedchem.1c02179,,67,,
2423,HDAC2,,10.1021/acs.jmedchem.1c02179,,57,,
2424,HDAC3,,10.1021/acs.jmedchem.1c02179,640,59,Degradation of HDAC3 in HCT116 cells after 24 h treatment,
2424,HDAC2,,10.1021/acs.jmedchem.1c02179,4190,56,Degradation of HDAC2 in HCT116 cells after 24 h treatment,
2424,HDAC1,,10.1021/acs.jmedchem.1c02179,910,74,Degradation of HDAC1 in HCT116 cells after 24 h treatment,
2425,HDAC2,,10.1021/acs.jmedchem.1c02179,,47,,
2425,HDAC3,,10.1021/acs.jmedchem.1c02179,,39,,
2425,HDAC1,,10.1021/acs.jmedchem.1c02179,,57,,
2426,HDAC1,,10.1021/acs.jmedchem.1c02179,550,77,Degradation of HDAC1 in HCT116 cells after 24 h treatment,
2426,HDAC3,,10.1021/acs.jmedchem.1c02179,530,66,Degradation of HDAC3 in HCT116 cells after 24 h treatment,
2426,HDAC2,,10.1021/acs.jmedchem.1c02179,,52,,
2427,HDAC1,,10.1021/acs.jmedchem.1c02179,,13,,
2427,HDAC2,,10.1021/acs.jmedchem.1c02179,,6,,
2427,HDAC3,,10.1021/acs.jmedchem.1c02179,,24,,
2428,HDAC3,,10.1021/acs.jmedchem.1c02179,,44,,
2428,HDAC2,,10.1021/acs.jmedchem.1c02179,,14,,
2428,HDAC1,,10.1021/acs.jmedchem.1c02179,,29,,
2429,HDAC3,,10.1021/acs.jmedchem.1c02179,,22,,
2429,HDAC1,,10.1021/acs.jmedchem.1c02179,,6,,
2429,HDAC2,,10.1021/acs.jmedchem.1c02179,,5,,
2430,HDAC3,,10.1021/acs.jmedchem.1c02179,,N.D.,,
2430,HDAC2,,10.1021/acs.jmedchem.1c02179,,5,,
2430,HDAC1,,10.1021/acs.jmedchem.1c02179,,4,,
2431,HDAC2,,10.1021/acs.jmedchem.1c02179,,13,,
2431,HDAC3,,10.1021/acs.jmedchem.1c02179,,39,,
2431,HDAC1,,10.1021/acs.jmedchem.1c02179,,41,,
2432,HDAC2,,10.1021/acs.jmedchem.1c02179,,26,,
2432,HDAC1,,10.1021/acs.jmedchem.1c02179,,61,,
2432,HDAC3,,10.1021/acs.jmedchem.1c02179,,51,,
2433,HDAC2,,10.1021/acs.jmedchem.1c02179,,N.D.,,
2433,HDAC3,,10.1021/acs.jmedchem.1c02179,,37,,
2433,HDAC1,,10.1021/acs.jmedchem.1c02179,,11,,
2434,HDAC1,,10.1021/acs.jmedchem.1c02179,,58,,
2434,HDAC3,,10.1021/acs.jmedchem.1c02179,,63,,
2434,HDAC2,,10.1021/acs.jmedchem.1c02179,,23,,
2435,HDAC3,,10.1021/acs.jmedchem.1c02179,,3,,
2435,HDAC2,,10.1021/acs.jmedchem.1c02179,,6,,
2435,HDAC1,,10.1021/acs.jmedchem.1c02179,,6,,
2436,HDAC3,,10.1021/acs.jmedchem.1c02179,,10,,
2436,HDAC2,,10.1021/acs.jmedchem.1c02179,,15,,
2436,HDAC1,,10.1021/acs.jmedchem.1c02179,,26,,
2437,HDAC3,,10.1021/acs.jmedchem.1c02179,,23,,
2437,HDAC1,,10.1021/acs.jmedchem.1c02179,,22,,
2437,HDAC2,,10.1021/acs.jmedchem.1c02179,,15,,
2438,HDAC2,,10.1021/acs.jmedchem.1c02179,,50,,
2438,HDAC3,,10.1021/acs.jmedchem.1c02179,1380,76,Degradation of HDAC3 in HCT116 cells after 24 h treatment,
2438,HDAC1,,10.1021/acs.jmedchem.1c02179,3580,68,Degradation of HDAC1 in HCT116 cells after 24 h treatment,
2439,HDAC2,,10.1021/acs.jmedchem.1c02179,,23,,
2439,HDAC1,,10.1021/acs.jmedchem.1c02179,,45,,
2439,HDAC3,,10.1021/acs.jmedchem.1c02179,440,77,Degradation of HDAC3 in HCT116 cells after 24 h treatment,
2440,HDAC1,,10.1021/acs.jmedchem.1c02179,,53,,
2440,HDAC2,,10.1021/acs.jmedchem.1c02179,,14,,
2440,HDAC3,,10.1021/acs.jmedchem.1c02179,,27,,
2441,HDAC1,,10.1021/acs.jmedchem.1c02179,,38,,
2441,HDAC3,,10.1021/acs.jmedchem.1c02179,,15,,
2441,HDAC2,,10.1021/acs.jmedchem.1c02179,,11,,
2442,EZH2,,10.1021/acs.jmedchem.1c00460,,,,
2443,EZH2,,10.1021/acs.jmedchem.1c00460,,,,
2444,EZH2,,10.1021/acs.jmedchem.1c00460,,,,
2445,EZH2,,10.1021/acs.jmedchem.1c00460,,,,
2446,EZH2,,10.1021/acs.jmedchem.1c00460,,,,
2447,EZH2,,10.1021/acs.jmedchem.1c00460,,,,
2448,EZH2,,10.1021/acs.jmedchem.1c00460,,,,
2449,EZH2,,10.1021/acs.jmedchem.1c00460,,,,
2450,EZH2,,10.1021/acs.jmedchem.1c00460,,,,
2451,EZH2,,10.1021/acs.jmedchem.1c00460,,,,
2452,EZH2,,10.1021/acs.jmedchem.1c00460,,,,
2453,EZH2,,10.1021/acs.jmedchem.1c00460,,,,
2454,EZH2,,10.1021/acs.jmedchem.1c00460,,,,
2455,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2456,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2457,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2458,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2459,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2460,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2461,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2462,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2463,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2464,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2465,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2466,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2467,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2468,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2469,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2470,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2471,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2472,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2473,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2474,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2475,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2476,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2477,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2478,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2479,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2480,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2481,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2482,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2483,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2484,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2485,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2486,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2487,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2488,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2489,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2490,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2491,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2492,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2493,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2494,CDK9,,10.1021/acs.jmedchem.1c01350,,,,
2495,AR,,10.1021/acs.jmedchem.1c00900,1,85,Degradation of AR in VCaP cells after 24 h treatment,
2496,AR,,10.1021/acs.jmedchem.1c00900,1.1,89,Degradation of AR in VCaP cells after 24 h treatment,
2497,AR,,10.1021/acs.jmedchem.1c00900,0.2,95,Degradation of AR in VCaP cells after 24 h treatment,
2498,AR,,10.1021/acs.jmedchem.1c00900,0.6,99,Degradation of AR in VCaP cells after 24 h treatment,
2499,AR,,10.1021/acs.jmedchem.1c00900,0.7,99,Degradation of AR in VCaP cells after 24 h treatment,
2500,AR,,10.1021/acs.jmedchem.1c00900,1.5,97,Degradation of AR in VCaP cells after 24 h treatment,
2501,AR,,10.1021/acs.jmedchem.1c00900,3.2,96,Degradation of AR in VCaP cells after 24 h treatment,
2502,AR,,10.1021/acs.jmedchem.1c00900,>1000,25,Degradation of AR in VCaP cells after 24 h treatment,
2503,AR,,10.1021/acs.jmedchem.1c00900,>1000,42,Degradation of AR in VCaP cells after 24 h treatment,
2504,AR,,10.1021/acs.jmedchem.1c00900,0.8,77,Degradation of AR in VCaP cells after 24 h treatment,
2505,AR,,10.1021/acs.jmedchem.1c00900,2.7,82,Degradation of AR in VCaP cells after 24 h treatment,
2506,AR,,10.1021/acs.jmedchem.1c00900,16.2,67,Degradation of AR in VCaP cells after 24 h treatment,
2507,AR,,10.1021/acs.jmedchem.1c00900,0.9,85,Degradation of AR in VCaP cells after 24 h treatment,
2508,AR,,10.1021/acs.jmedchem.1c00900,0.2,97,Degradation of AR in VCaP cells after 24 h treatment,
2509,AR,,10.1021/acs.jmedchem.1c00900,0.3,88,Degradation of AR in VCaP cells after 24 h treatment,
2510,AR T878A,,10.1021/acs.jmedchem.1c00900,,,,
2510,AR,,10.1021/acs.jmedchem.1c00900,0.2,95,Degradation of AR in VCaP cells after 24 h treatment,
2511,AR T878A,,10.1021/acs.jmedchem.1c00900,,,,
2511,AR,,10.1021/acs.jmedchem.1c00900,0.3,92,Degradation of AR in VCaP cells after 24 h treatment,
2512,AR,,10.1021/acs.jmedchem.1c00900,0.1,76,Degradation of AR in VCaP cells after 24 h treatment,
2513,AR,,10.1021/acs.jmedchem.1c00900,>1000,20,Degradation of AR in VCaP cells after 24 h treatment,
2514,AR,,10.1021/acs.jmedchem.1c00900,>1000,45,Degradation of AR in VCaP cells after 24 h treatment,
2515,AR,,10.1021/acs.jmedchem.1c00900,>1000,54,Degradation of AR in VCaP cells after 24 h treatment,
2516,AR,,10.1021/acs.jmedchem.1c00900,>1000,19,Degradation of AR in VCaP cells after 24 h treatment,
2517,AR,,10.1021/acs.jmedchem.1c00900,>1000,35,Degradation of AR in VCaP cells after 24 h treatment,
2518,AR,,10.1021/acs.jmedchem.1c00900,0.3,78,Degradation of AR in VCaP cells after 24 h treatment,
2519,AR T878A,,10.1021/acs.jmedchem.1c00900,0.3,95,Degradation of AR T878A in LNCaP (AR T878A) cells after 24 h treatment,
2519,AR,,10.1021/acs.jmedchem.1c00900,0.09,99,Degradation of AR in VCaP cells after 24 h treatment,
2520,AR,,10.1021/acs.jmedchem.1c00900,0.1,99,Degradation of AR in VCaP cells after 24 h treatment,
2521,AR,,10.1021/acs.jmedchem.1c00900,1.4,88,Degradation of AR in VCaP cells after 24 h treatment,
2522,AR,,10.1021/acs.jmedchem.1c00900,1.4,93,Degradation of AR in VCaP cells after 24 h treatment,
2523,AR,,10.1021/acs.jmedchem.1c00900,0.5,96,Degradation of AR in VCaP cells after 24 h treatment,
2524,AR T878A,,10.1021/acs.jmedchem.1c00900,0.4,95,Degradation of AR T878A in LNCaP (AR T878A) cells after 24 h treatment,
2524,AR,,10.1021/acs.jmedchem.1c00900,0.1,96,Degradation of AR in VCaP cells after 24 h treatment,
2525,AR,,10.1021/acs.jmedchem.1c00900,0.01,99,Degradation of AR in VCaP cells after 24 h treatment,
2525,AR T878A,,10.1021/acs.jmedchem.1c00900,0.9,99,Degradation of AR T878A in LNCaP (AR T878A) cells after 24 h treatment,
2526,AR,,10.1021/acs.jmedchem.1c00900,0.04,99,Degradation of AR in VCaP cells after 24 h treatment,
2526,AR T878A,,10.1021/acs.jmedchem.1c00900,0.1,98,Degradation of AR T878A in LNCaP (AR T878A) cells after 24 h treatment,
2527,AR T878A,,10.1021/acs.jmedchem.1c00900,1.9,99,Degradation of AR T878A in LNCaP (AR T878A) cells after 24 h treatment,
2527,AR,,10.1021/acs.jmedchem.1c00900,0.1,100,Degradation of AR in VCaP cells after 24 h treatment,
2528,AR,,10.1021/acs.jmedchem.1c00900,0.2,96,Degradation of AR in VCaP cells after 24 h treatment,
2528,AR T878A,,10.1021/acs.jmedchem.1c00900,1.3,64,Degradation of AR T878A in LNCaP (AR T878A) cells after 24 h treatment,
2529,AR,,10.1021/acs.jmedchem.1c00900,>1000,32,Degradation of AR in VCaP cells after 24 h treatment,
2530,AR,,10.1021/acs.jmedchem.1c00900,>1000,14,Degradation of AR in VCaP cells after 24 h treatment,
2531,AR,,10.1021/acs.jmedchem.1c00900,>1000,27,Degradation of AR in VCaP cells after 24 h treatment,
2532,ALK,24.3/50.2,10.1021/acs.jmedchem.1c00270,,,,% ALK degradation in H3122 cells after 16 h treatment at 100/1000 nM
2533,ALK,74.4/81.8,10.1021/acs.jmedchem.1c00270,,,,% ALK degradation in H3122 cells after 16 h treatment at 100/1000 nM
2534,ALK,38.3/75.7,10.1021/acs.jmedchem.1c00270,,,,% ALK degradation in H3122 cells after 16 h treatment at 100/1000 nM
2535,ALK,51.3/75.8,10.1021/acs.jmedchem.1c00270,,,,% ALK degradation in H3122 cells after 16 h treatment at 100/1000 nM
2536,ALK,0/50.6,10.1021/acs.jmedchem.1c00270,,,,% ALK degradation in H3122 cells after 16 h treatment at 100/1000 nM
2537,ALK,47.8/91,10.1021/acs.jmedchem.1c00270,,,,% ALK degradation in H3122 cells after 16 h treatment at 100/1000 nM
2538,ALK,49.9/87,10.1021/acs.jmedchem.1c00270,,,,% ALK degradation in H3122 cells after 16 h treatment at 100/1000 nM
2539,ALK,24.5/77.3,10.1021/acs.jmedchem.1c00270,,,,% ALK degradation in H3122 cells after 16 h treatment at 100/1000 nM
2540,HPGDS,,10.1021/acs.jmedchem.1c01206,,,,
2541,HPGDS,,10.1021/acs.jmedchem.1c01206,,,,
2542,HPGDS,,10.1021/acs.jmedchem.1c01206,,,,
2543,HPGDS,,10.1021/acs.jmedchem.1c01206,,,,
2544,HPGDS,,10.1021/acs.jmedchem.1c01206,0.0263/0.0173,,Degradation of HPGDS in KU812 cells after 6/24 h treatment,
2545,HPGDS,,10.1021/acs.jmedchem.1c01206,,N.D.,,
2546,HPGDS,,10.1021/acs.jmedchem.1c01206,,,,
2547,HPGDS,,10.1021/acs.jmedchem.1c01206,,N.D.,,
2548,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2548,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2548,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2549,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2549,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2549,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2550,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2550,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2550,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2551,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2551,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2551,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2552,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2552,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2552,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2553,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2553,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2553,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2554,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2554,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2554,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2555,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2555,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2555,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2556,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2556,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2556,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2557,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2557,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2557,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2558,AKT1,,10.1021/acs.jmedchem.1c01476,78,,Degradation of total AKT in BT474 cells after 24 h treatment,
2558,AKT2,,10.1021/acs.jmedchem.1c01476,78,,Degradation of total AKT in BT474 cells after 24 h treatment,
2558,AKT3,,10.1021/acs.jmedchem.1c01476,78,,Degradation of total AKT in BT474 cells after 24 h treatment,
2559,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2559,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2559,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2560,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2560,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2560,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2561,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2561,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2561,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2562,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2562,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2562,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2563,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2563,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2563,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2564,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2564,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2564,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2565,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2565,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2565,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2566,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2566,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2566,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2567,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2567,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2567,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2568,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2568,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2568,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2569,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2569,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2569,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2570,AKT2,,10.1021/acs.jmedchem.1c01476,32,,Degradation of total AKT in BT474 cells after 24 h treatment,
2570,AKT1,,10.1021/acs.jmedchem.1c01476,32,,Degradation of total AKT in BT474 cells after 24 h treatment,
2570,AKT3,,10.1021/acs.jmedchem.1c01476,32,,Degradation of total AKT in BT474 cells after 24 h treatment,
2571,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2571,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2571,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2572,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2572,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2572,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2573,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2573,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2573,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2574,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2574,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2574,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2575,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2575,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2575,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2576,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2576,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2576,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2577,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2577,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2577,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2578,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2578,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2578,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2579,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2579,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2579,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2580,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2580,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2580,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2581,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2581,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2581,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2582,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2582,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2582,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2583,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2583,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2583,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2584,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2584,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2584,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2585,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2585,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2585,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2586,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2586,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2586,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2587,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2587,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2587,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2588,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2588,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2588,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2589,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2589,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2589,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2590,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2590,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2590,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2591,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2591,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2591,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2592,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2592,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2592,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2593,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2593,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2593,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2594,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2594,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2594,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2595,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2595,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2595,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2596,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2596,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2596,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2597,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2597,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2597,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2598,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2598,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2598,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2599,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2599,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2599,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2600,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2600,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2600,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2601,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2601,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2601,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2602,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2602,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2602,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2603,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2603,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2603,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2604,AKT1,,10.1021/acs.jmedchem.1c01476,,,,
2604,AKT2,,10.1021/acs.jmedchem.1c01476,,,,
2604,AKT3,,10.1021/acs.jmedchem.1c01476,,,,
2605,EGFR L858R/T790M,<20/<20,10.1021/acs.jmedchem.1c01827,,,,% EGFR L858R/T790M degradation in H1975 cells after 24 h treatment at 100/1000 nM
2605,EGFR e19d,,10.1021/acs.jmedchem.1c01827,,,,
2606,EGFR L858R/T790M,<20/<20,10.1021/acs.jmedchem.1c01827,,,,% EGFR L858R/T790M degradation in H1975 cells after 24 h treatment at 100/1000 nM
2606,EGFR e19d,<20/25,10.1021/acs.jmedchem.1c01827,,,,% EGFR del19 degradation in HCC827 cells after 24 h treatment at 100/1000 nM
2607,EGFR e19d,<20/24,10.1021/acs.jmedchem.1c01827,,,,% EGFR del19 degradation in HCC827 cells after 24 h treatment at 100/1000 nM
2607,EGFR L858R/T790M,<20/<20,10.1021/acs.jmedchem.1c01827,,,,% EGFR L858R/T790M degradation in H1975 cells after 24 h treatment at 100/1000 nM
2608,EGFR L858R/T790M,<20/<20,10.1021/acs.jmedchem.1c01827,,,,% EGFR L858R/T790M degradation in H1975 cells after 24 h treatment at 100/1000 nM
2608,EGFR e19d,<20/25,10.1021/acs.jmedchem.1c01827,,,,% EGFR del19 degradation in HCC827 cells after 24 h treatment at 100/1000 nM
2609,EGFR L858R/T790M,<20/<20,10.1021/acs.jmedchem.1c01827,,,,% EGFR L858R/T790M degradation in H1975 cells after 24 h treatment at 100/1000 nM
2609,EGFR e19d,<20/30,10.1021/acs.jmedchem.1c01827,,,,% EGFR del19 degradation in HCC827 cells after 24 h treatment at 100/1000 nM
2610,EGFR L858R/T790M,<20/<20,10.1021/acs.jmedchem.1c01827,,,,% EGFR L858R/T790M degradation in H1975 cells after 24 h treatment at 100/1000 nM
2610,EGFR e19d,28/34,10.1021/acs.jmedchem.1c01827,,,,% EGFR del19 degradation in HCC827 cells after 24 h treatment at 100/1000 nM
2611,EGFR L858R/T790M,<20/<20,10.1021/acs.jmedchem.1c01827,,,,% EGFR L858R/T790M degradation in H1975 cells after 24 h treatment at 100/1000 nM
2611,EGFR e19d,23/25,10.1021/acs.jmedchem.1c01827,,,,% EGFR del19 degradation in HCC827 cells after 24 h treatment at 100/1000 nM
2612,EGFR L858R/T790M,<20/<20,10.1021/acs.jmedchem.1c01827,,,,% EGFR L858R/T790M degradation in H1975 cells after 24 h treatment at 100/1000 nM
2612,EGFR e19d,<20/<20,10.1021/acs.jmedchem.1c01827,,,,% EGFR del19 degradation in HCC827 cells after 24 h treatment at 100/1000 nM
2613,EGFR L858R/T790M,39/59,10.1021/acs.jmedchem.1c01827,,,,% EGFR L858R/T790M degradation in H1975 cells after 24 h treatment at 100/1000 nM
2613,EGFR e19d,42/57,10.1021/acs.jmedchem.1c01827,,,,% EGFR del19 degradation in HCC827 cells after 24 h treatment at 100/1000 nM
2614,EGFR L858R/T790M,,10.1021/acs.jmedchem.1c01827,,,,
2614,EGFR e19d,,10.1021/acs.jmedchem.1c01827,,,,
2615,EGFR L858R/T790M,,10.1021/acs.jmedchem.1c01827,,,,
2615,EGFR e19d,,10.1021/acs.jmedchem.1c01827,,,,
2616,EGFR L858R/T790M,,10.1021/acs.jmedchem.1c01827,,,,
2616,EGFR e19d,,10.1021/acs.jmedchem.1c01827,,,,
2617,EGFR L858R/T790M,,10.1021/acs.jmedchem.1c01827,,,,
2617,EGFR e19d,,10.1021/acs.jmedchem.1c01827,,,,
2618,EGFR L858R/T790M,<20/<20,10.1021/acs.jmedchem.1c01827,,,,% EGFR L858R/T790M degradation in H1975 cells after 24 h treatment at 100/1000 nM
2618,EGFR e19d,<20/26,10.1021/acs.jmedchem.1c01827,,,,% EGFR del19 degradation in HCC827 cells after 24 h treatment at 100/1000 nM
2619,EGFR L858R/T790M,38/79,10.1021/acs.jmedchem.1c01827,,,,% EGFR L858R/T790M degradation in H1975 cells after 24 h treatment at 10/100 nM
2619,EGFR e19d,65/81,10.1021/acs.jmedchem.1c01827,,,,% EGFR del19 degradation in HCC827 cells after 24 h treatment at 3/30 nM
2620,EGFR L858R/T790M,49/69,10.1021/acs.jmedchem.1c01827,,,,% EGFR L858R/T790M degradation in H1975 cells after 24 h treatment at 10/100 nM
2620,EGFR e19d,62/70,10.1021/acs.jmedchem.1c01827,,,,% EGFR del19 degradation in HCC827 cells after 24 h treatment at 3/30 nM
2621,EGFR L858R/T790M,47/74,10.1021/acs.jmedchem.1c01827,,,,% EGFR L858R/T790M degradation in H1975 cells after 24 h treatment at 10/100 nM
2621,EGFR e19d,69/78,10.1021/acs.jmedchem.1c01827,,,,% EGFR del19 degradation in HCC827 cells after 24 h treatment at 3/30 nM
2622,EGFR L858R/T790M,<20/23,10.1021/acs.jmedchem.1c01827,,,,% EGFR L858R/T790M degradation in H1975 cells after 24 h treatment at 10/100 nM
2622,EGFR e19d,46/60,10.1021/acs.jmedchem.1c01827,,,,% EGFR del19 degradation in HCC827 cells after 24 h treatment at 3/30 nM
2623,EGFR L858R/T790M,<20/<20,10.1021/acs.jmedchem.1c01827,,,,% EGFR L858R/T790M degradation in H1975 cells after 24 h treatment at 10/100 nM
2623,EGFR e19d,63/77,10.1021/acs.jmedchem.1c01827,,,,% EGFR del19 degradation in HCC827 cells after 24 h treatment at 3/30 nM
2624,EGFR L858R/T790M,<20/<20,10.1021/acs.jmedchem.1c01827,,,,% EGFR L858R/T790M degradation in H1975 cells after 24 h treatment at 10/100 nM
2624,EGFR e19d,50/57,10.1021/acs.jmedchem.1c01827,,,,% EGFR del19 degradation in HCC827 cells after 24 h treatment at 3/30 nM
2625,EGFR L858R/T790M,,10.1021/acs.jmedchem.1c01827,1.56,86,Degradation of EGFR L858R/T790M in H1975 cells after 48 h treatment,
2625,EGFR e19d,,10.1021/acs.jmedchem.1c01827,0.49,82,Degradation of EGFR e19d in HCC827 cells after 24 h treatment,
2626,EGFR e19d,69/72,10.1021/acs.jmedchem.1c01827,,,,% EGFR del19 degradation in HCC827 cells after 24 h treatment at 3/30 nM
2626,EGFR L858R/T790M,<20/<20,10.1021/acs.jmedchem.1c01827,,,,% EGFR L858R/T790M degradation in H1975 cells after 24 h treatment at 10/100 nM
2627,SOS1,5.8/30.4,10.1021/acs.jmedchem.1c01774,,,,% SOS1 degradation in NCI-H358 cells after 24 h treatment at 100/1000 nM
2628,SOS1,30.7/79.9,10.1021/acs.jmedchem.1c01774,216.4,,Degradation of SOS1 in NCI-H358 cells after 24 h treatment,% SOS1 degradation in NCI-H358 cells after 24 h treatment at 100/1000 nM
2629,SOS1,27.6/80.9,10.1021/acs.jmedchem.1c01774,150.3,,Degradation of SOS1 in NCI-H358 cells after 24 h treatment,% SOS1 degradation in NCI-H358 cells after 24 h treatment at 100/1000 nM
2630,SOS1,,10.1021/acs.jmedchem.1c01774,104/125/22,,Degradation of SOS1 in SK-LU-1/SW620/A549 cells after 24 h treatment,
2630,SOS1,,10.1021/acs.jmedchem.1c01774,98.4/255/119,,Degradation of SOS1 in NCI-H358/MIA PaCa2/AsPC-1 cells after 24 h treatment,
2631,SOS1,38.5/82,10.1021/acs.jmedchem.1c01774,182.1,,Degradation of SOS1 in NCI-H358 cells after 24 h treatment,% SOS1 degradation in NCI-H358 cells after 24 h treatment at 100/1000 nM
2632,SOS1,31.7/63.2,10.1021/acs.jmedchem.1c01774,,,,% SOS1 degradation in NCI-H358 cells after 24 h treatment at 100/1000 nM
2633,SOS1,33/49,10.1021/acs.jmedchem.1c01774,,,,% SOS1 degradation in NCI-H358 cells after 24 h treatment at 100/1000 nM
2634,SOS1,23.3/24.4,10.1021/acs.jmedchem.1c01774,,,,% SOS1 degradation in NCI-H358 cells after 24 h treatment at 100/1000 nM
2635,SOS1,4.4/14,10.1021/acs.jmedchem.1c01774,,,,% SOS1 degradation in NCI-H358 cells after 24 h treatment at 100/1000 nM
2636,SOS1,15.4/36.6,10.1021/acs.jmedchem.1c01774,,,,% SOS1 degradation in NCI-H358 cells after 24 h treatment at 100/1000 nM
2637,SOS1,0/18.3,10.1021/acs.jmedchem.1c01774,,,,% SOS1 degradation in NCI-H358 cells after 24 h treatment at 100/1000 nM
2638,SOS1,8/12.7,10.1021/acs.jmedchem.1c01774,,,,% SOS1 degradation in NCI-H358 cells after 24 h treatment at 100/1000 nM
2639,SOS1,3.2/0,10.1021/acs.jmedchem.1c01774,,,,% SOS1 degradation in NCI-H358 cells after 24 h treatment at 100/1000 nM
2640,SOS1,13/43.3,10.1021/acs.jmedchem.1c01774,,,,% SOS1 degradation in NCI-H358 cells after 24 h treatment at 100/1000 nM
2641,SOS1,18.1/9.4,10.1021/acs.jmedchem.1c01774,,,,% SOS1 degradation in NCI-H358 cells after 24 h treatment at 100/1000 nM
2642,SOS1,7/11.2,10.1021/acs.jmedchem.1c01774,,,,% SOS1 degradation in NCI-H358 cells after 24 h treatment at 100/1000 nM
2643,BRD3,,10.1016/j.ejmech.2022.114259,,,,
2643,BRD4,,10.1016/j.ejmech.2022.114259,,,,
2643,BRD2,,10.1016/j.ejmech.2022.114259,,,,
2644,BRD3,,10.1016/j.ejmech.2022.114259,,,,
2644,BRD4,,10.1016/j.ejmech.2022.114259,,,,
2644,BRD2,,10.1016/j.ejmech.2022.114259,,,,
2645,BRD3,,10.1016/j.ejmech.2022.114259,,,,
2645,BRD4,,10.1016/j.ejmech.2022.114259,,,,
2645,BRD2,,10.1016/j.ejmech.2022.114259,,,,
2646,BRD3,,10.1016/j.ejmech.2022.114259,,,,
2646,BRD4,,10.1016/j.ejmech.2022.114259,,,,
2646,BRD2,,10.1016/j.ejmech.2022.114259,,,,
2647,BRD3,,10.1016/j.ejmech.2022.114259,,,,
2647,BRD2,,10.1016/j.ejmech.2022.114259,,,,
2647,BRD4,,10.1016/j.ejmech.2022.114259,,,,
2648,BRD2,,10.1016/j.ejmech.2022.114259,,,,
2648,BRD3,,10.1016/j.ejmech.2022.114259,,,,
2648,BRD4,,10.1016/j.ejmech.2022.114259,,,,
2649,BRD3,,10.1016/j.ejmech.2022.114259,,,,
2649,BRD2,,10.1016/j.ejmech.2022.114259,,,,
2649,BRD4,,10.1016/j.ejmech.2022.114259,,,,
2650,BRD4,,10.1016/j.ejmech.2022.114259,,,,
2650,BRD3,,10.1016/j.ejmech.2022.114259,,,,
2650,BRD2,,10.1016/j.ejmech.2022.114259,,,,
2651,BRD3,,10.1016/j.ejmech.2022.114259,,,,
2651,BRD2,,10.1016/j.ejmech.2022.114259,,,,
2651,BRD4,,10.1016/j.ejmech.2022.114259,,,,
2652,BRD3,,10.1016/j.ejmech.2022.114259,,,,
2652,BRD2,,10.1016/j.ejmech.2022.114259,,,,
2652,BRD4,,10.1016/j.ejmech.2022.114259,,,,
2653,BRD3,,10.1016/j.ejmech.2022.114259,,,,
2653,BRD2,,10.1016/j.ejmech.2022.114259,,,,
2653,BRD4,,10.1016/j.ejmech.2022.114259,,,,
2654,BRD3,,10.1016/j.ejmech.2022.114259,,,,
2654,BRD2,,10.1016/j.ejmech.2022.114259,,,,
2654,BRD4,,10.1016/j.ejmech.2022.114259,,,,
2655,BRD3,,10.1016/j.ejmech.2022.114259,,,,
2655,BRD2,,10.1016/j.ejmech.2022.114259,,,,
2655,BRD4,,10.1016/j.ejmech.2022.114259,,,,
2656,BRD3,,10.1016/j.ejmech.2022.114259,,,,
2656,BRD2,,10.1016/j.ejmech.2022.114259,,,,
2656,BRD4,,10.1016/j.ejmech.2022.114259,,,,
2657,BRD3,,10.1016/j.ejmech.2022.114259,,,,
2657,BRD4,,10.1016/j.ejmech.2022.114259,,,,
2657,BRD2,,10.1016/j.ejmech.2022.114259,,,,
2658,eIF4E,,10.1016/j.ejmech.2021.113435,,N.D.,,
2659,eIF4E,,10.1016/j.ejmech.2021.113435,,N.D.,,
2660,eIF4E,,10.1016/j.ejmech.2021.113435,,N.D.,,
2661,eIF4E,,10.1016/j.ejmech.2021.113435,,N.D.,,
2662,eIF4E,,10.1016/j.ejmech.2021.113435,,N.D.,,
2663,eIF4E,,10.1016/j.ejmech.2021.113435,,N.D.,,
2664,TYR,,10.1016/j.ejmech.2021.113850,,N.D.,,
2665,TYR,,10.1016/j.ejmech.2021.113850,,N.D.,,
2666,TYR,,10.1016/j.ejmech.2021.113850,,N.D.,,
2667,TYR,,10.1016/j.ejmech.2021.113850,,N.D.,,
2668,TYR,,10.1016/j.ejmech.2021.113850,,,,
2669,TYR,,10.1016/j.ejmech.2021.113850,,,,
2670,TYR,,10.1016/j.ejmech.2021.113850,,,,
2671,TYR,,10.1016/j.ejmech.2021.113850,,,,
2672,TYR,,10.1016/j.ejmech.2021.113850,50000,61,Degradation of TYR in A375 cells after 24 h treatment,
2673,TYR,,10.1016/j.ejmech.2021.113850,,,,
2674,TYR,,10.1016/j.ejmech.2021.113850,,,,
2675,TYR,,10.1016/j.ejmech.2021.113850,,,,
2676,TYR,,10.1016/j.ejmech.2021.113850,,,,
2677,TYR,,10.1016/j.ejmech.2021.113850,,,,
2678,CDK2,,10.1016/j.ejmech.2021.113849,,,,
2679,CDK2,,10.1016/j.ejmech.2021.113849,100,,Degradation of CDK2 in HEI-OC1 cells after 24 h treatment,
2680,CDK2,,10.1016/j.ejmech.2021.113849,,,,
2681,CDK2,,10.1016/j.ejmech.2021.113849,,,,
2682,BRD4,,10.1016/j.ejmech.2021.113922,,,,
2683,BRD4,,10.1016/j.ejmech.2021.113922,,,,
2684,BRD4,,10.1016/j.ejmech.2021.113922,,,,
2685,BRD4,,10.1016/j.ejmech.2021.113922,,,,
2686,BRD4,,10.1016/j.ejmech.2021.113922,,,,
2687,BRD4,,10.1016/j.ejmech.2021.113922,,,,
2688,BRD4,,10.1016/j.ejmech.2021.113922,,,,
2689,BRD4,,10.1016/j.ejmech.2021.113922,,,,
2690,BRD4,,10.1016/j.ejmech.2021.113922,<1/<1,>99/>99,Degradation of BRD4 in 22Rv1/VCaP cells after 24 h treatment,
2691,BRD4,,10.1016/j.ejmech.2021.113922,,,,
2692,BRD4,,10.1016/j.ejmech.2021.113922,,,,
2693,BRD4,,10.1016/j.ejmech.2021.113922,,,,
2694,BRD4,,10.1016/j.ejmech.2021.113922,,,,
2695,BRD4,,10.1016/j.ejmech.2021.113922,,,,
2696,BRD4,,10.1016/j.ejmech.2021.113922,,,,
2697,BRD4,,10.1016/j.ejmech.2021.113922,,,,
2698,BRD4,,10.1016/j.ejmech.2021.113922,,,,
2699,BCR-ABL,,10.1016/j.ejmech.2021.113645,8.7,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
2700,BCR-ABL,,10.1016/j.ejmech.2021.113645,17.5,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
2701,BCR-ABL,,10.1016/j.ejmech.2021.113645,18.4,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
2702,BCR-ABL,,10.1016/j.ejmech.2021.113645,26.1,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
2703,BCR-ABL,,10.1016/j.ejmech.2021.113645,10.8,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
2704,BCR-ABL,,10.1016/j.ejmech.2021.113645,7.8,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
2705,BCR-ABL,,10.1016/j.ejmech.2021.113645,11,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
2706,BCR-ABL,,10.1016/j.ejmech.2021.113645,9,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
2707,BCR-ABL,,10.1016/j.ejmech.2021.113645,5.6,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
2708,BCR-ABL,,10.1016/j.ejmech.2021.113645,10,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
2709,BCR-ABL,,10.1016/j.ejmech.2021.113645,11.1,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
2710,BCR-ABL,,10.1016/j.ejmech.2021.113645,95.4,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
2711,BCR-ABL,,10.1016/j.ejmech.2021.113645,245.1,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
2712,BCR-ABL T315A,,10.1016/j.ejmech.2021.113645,,,,
2712,BCR-ABL F317V,,10.1016/j.ejmech.2021.113645,,,,
2712,BCR-ABL F317L,,10.1016/j.ejmech.2021.113645,,,,
2712,BCR-ABL V299L,,10.1016/j.ejmech.2021.113645,,,,
2712,BCR-ABL E255V,,10.1016/j.ejmech.2021.113645,,,,
2712,BCR-ABL G250E,,10.1016/j.ejmech.2021.113645,,,,
2712,BCR-ABL,,10.1016/j.ejmech.2021.113645,0.18,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
2713,BCR-ABL,,10.1016/j.ejmech.2021.113645,8.9,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
2714,BCR-ABL,,10.1016/j.ejmech.2021.113645,2.7,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
2715,BCR-ABL,,10.1016/j.ejmech.2021.113645,2.7,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
2716,BCR-ABL,,10.1016/j.ejmech.2021.113645,10.1,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
2717,BCR-ABL,,10.1016/j.ejmech.2021.113645,11.1,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
2718,BCR-ABL,,10.1016/j.ejmech.2021.113645,125,,Degradation of BCR-ABL in K562 cells after 16 h treatment,
2719,HSP90,,10.1016/j.ejmech.2021.114013,,,,
2720,HSP90,,10.1016/j.ejmech.2021.114013,990,83.43,Degradation of HSP90 in MCF-7 cells after 6 h treatment,
2721,HSP90,,10.1016/j.ejmech.2021.114013,,,,
2722,HSP90,,10.1016/j.ejmech.2021.114013,,,,
2723,HSP90,,10.1016/j.ejmech.2021.114013,,,,
2724,HSP90,,10.1016/j.ejmech.2021.114013,,,,
2725,HSP90,,10.1016/j.ejmech.2021.114013,,,,
2726,HSP90,,10.1016/j.ejmech.2021.114013,,,,
2727,HSP90,,10.1016/j.ejmech.2021.114013,,,,
2728,HSP90,,10.1016/j.ejmech.2021.114013,,,,
2729,HSP90,,10.1016/j.ejmech.2021.114013,,N.D.,,
2730,HSP90,,10.1016/j.ejmech.2021.114013,,N.D.,,
2731,HSP90,,10.1016/j.ejmech.2021.114013,,N.D.,,
2732,HSP90,,10.1016/j.ejmech.2021.114013,,N.D.,,
2733,HSP90,,10.1016/j.ejmech.2021.114013,,N.D.,,
2734,HSP90,,10.1016/j.ejmech.2021.114013,,N.D.,,
2735,HSP90,,10.1016/j.ejmech.2021.114013,,N.D.,,
2736,HSP90,,10.1016/j.ejmech.2021.114013,,N.D.,,
2737,HSP90,,10.1016/j.ejmech.2021.114013,,N.D.,,
2738,HSP90,,10.1016/j.ejmech.2021.114013,,N.D.,,
2739,CDK12,,10.1016/j.ejmech.2021.114012,,,,
2740,CDK12,,10.1016/j.ejmech.2021.114012,416/412,,Degradation of CDK12 in Bel-7402/MDA-MB-231 cells after 24 h treatment,
2741,CDK12,,10.1016/j.ejmech.2021.114012,,,,
2742,CDK12,,10.1016/j.ejmech.2021.114012,,,,
2743,GSK-3beta,<5/0,10.1016/j.ejmech.2021.113889,,,,% GSK3B degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2743,GSK3A,<5/0,10.1016/j.ejmech.2021.113889,,,,% GSK3A degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2744,GSK3A,<5/<5,10.1016/j.ejmech.2021.113889,,,,% GSK3A degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2744,GSK-3beta,<5/35.8,10.1016/j.ejmech.2021.113889,,,,% GSK3B degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2745,GSK-3beta,14.5/37.3,10.1016/j.ejmech.2021.113889,,,,% GSK3B degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2745,GSK3A,38.7/76.4,10.1016/j.ejmech.2021.113889,,,,% GSK3A degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2746,GSK3A,<5/<5,10.1016/j.ejmech.2021.113889,,,,% GSK3A degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2746,GSK-3beta,<5/<5,10.1016/j.ejmech.2021.113889,,,,% GSK3B degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2747,GSK-3beta,<5/<5,10.1016/j.ejmech.2021.113889,,,,% GSK3B degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2747,GSK3A,<5/<5,10.1016/j.ejmech.2021.113889,,,,% GSK3A degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2748,GSK-3beta,30.5/39.6,10.1016/j.ejmech.2021.113889,,,,% GSK3B degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2748,GSK3A,46.9/68.9,10.1016/j.ejmech.2021.113889,,,,% GSK3A degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2749,GSK-3beta,29.9/46.6,10.1016/j.ejmech.2021.113889,,,,% GSK3B degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2749,GSK3A,45.4/75.6,10.1016/j.ejmech.2021.113889,,,,% GSK3A degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2750,GSK3A,42.0/79.5,10.1016/j.ejmech.2021.113889,,,,% GSK3A degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2750,GSK-3beta,25.7/65,10.1016/j.ejmech.2021.113889,,,,% GSK3B degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2751,GSK-3beta,28.9/63.8,10.1016/j.ejmech.2021.113889,,,,% GSK3B degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2751,GSK3A,47.4/77.2,10.1016/j.ejmech.2021.113889,,,,% GSK3A degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2752,GSK-3beta,15.2/61.3,10.1016/j.ejmech.2021.113889,,,,% GSK3B degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2752,GSK3A,29.7/75.4,10.1016/j.ejmech.2021.113889,,,,% GSK3A degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2753,GSK-3beta,41.9/79.5,10.1016/j.ejmech.2021.113889,,,,% GSK3B degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2753,GSK3A,61.1/95.2,10.1016/j.ejmech.2021.113889,,,,% GSK3A degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2754,GSK3A,65.0/90.7,10.1016/j.ejmech.2021.113889,,,,% GSK3A degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2754,GSK-3beta,51.6/79.1,10.1016/j.ejmech.2021.113889,,,,% GSK3B degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2755,GSK-3beta,55.9/83.1,10.1016/j.ejmech.2021.113889,,,,% GSK3B degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2755,GSK3A,63.8/91.8,10.1016/j.ejmech.2021.113889,,,,% GSK3A degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2756,GSK-3beta,61.6/81.3,10.1016/j.ejmech.2021.113889,,,,% GSK3B degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2756,GSK3A,68.1/87.8,10.1016/j.ejmech.2021.113889,,,,% GSK3A degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2757,GSK-3beta,55.9/86,10.1016/j.ejmech.2021.113889,,,,% GSK3B degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2757,GSK3A,66.3/93.9,10.1016/j.ejmech.2021.113889,,,,% GSK3A degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2758,GSK-3beta,38.2/88.3,10.1016/j.ejmech.2021.113889,,,,% GSK3B degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2758,GSK3A,70.9/95.1,10.1016/j.ejmech.2021.113889,,,,% GSK3A degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2759,GSK-3beta,54.6/89.7,10.1016/j.ejmech.2021.113889,,,,% GSK3B degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2759,GSK3A,69.3/93.8,10.1016/j.ejmech.2021.113889,,,,% GSK3A degradation in SH-SY5Y cells after 24 h treatment at 1000/10000 nM
2760,GSK-3beta,,10.1016/j.ejmech.2021.113889,110.1,,Degradation of GSK3B in SH-SY5Y cells after 24 h treatment,
2760,GSK3A,,10.1016/j.ejmech.2021.113889,38.2,,Degradation of GSK3A in SH-SY5Y cells after 24 h treatment,
2761,GSK3A,,10.1016/j.ejmech.2021.113889,28.3,,Degradation of GSK3A in SH-SY5Y cells after 24 h treatment,
2761,GSK-3beta,,10.1016/j.ejmech.2021.113889,34.2,,Degradation of GSK3B in SH-SY5Y cells after 24 h treatment,
2762,GSK3A,,10.1016/j.ejmech.2021.113889,40.4,,Degradation of GSK3A in SH-SY5Y cells after 24 h treatment,
2762,GSK-3beta,,10.1016/j.ejmech.2021.113889,66.6,,Degradation of GSK3B in SH-SY5Y cells after 24 h treatment,
2763,GSK3A,,10.1016/j.ejmech.2021.113889,,,,
2763,GSK-3beta,,10.1016/j.ejmech.2021.113889,,,,
2764,GSK3A,,10.1016/j.ejmech.2021.113889,,,,
2764,GSK-3beta,,10.1016/j.ejmech.2021.113889,,,,
2765,GSK3A,,10.1016/j.ejmech.2021.113889,,,,
2765,GSK-3beta,,10.1016/j.ejmech.2021.113889,,,,
2766,GSK-3beta,,10.1016/j.ejmech.2021.113889,,,,
2766,GSK3A,,10.1016/j.ejmech.2021.113889,,,,
2767,GSK3A,,10.1016/j.ejmech.2021.113889,,,,
2767,GSK-3beta,,10.1016/j.ejmech.2021.113889,,,,
2768,GSK-3beta,,10.1016/j.ejmech.2021.113889,,,,
2768,GSK3A,,10.1016/j.ejmech.2021.113889,,,,
2769,GSK3A,,10.1016/j.ejmech.2021.113889,,,,
2769,GSK-3beta,,10.1016/j.ejmech.2021.113889,,,,
2770,GSK-3beta,,10.1016/j.ejmech.2021.113889,,,,
2770,GSK3A,,10.1016/j.ejmech.2021.113889,,,,
2771,GSK3A,,10.1016/j.ejmech.2021.113889,,,,
2771,GSK-3beta,,10.1016/j.ejmech.2021.113889,,,,
2772,GSK-3beta,,10.1016/j.ejmech.2021.113889,,,,
2772,GSK3A,,10.1016/j.ejmech.2021.113889,,,,
2773,AXL,,10.1016/j.ejmech.2022.114253,,,,
2774,AXL,,10.1016/j.ejmech.2022.114253,,,,
2775,AXL,,10.1016/j.ejmech.2022.114253,,,,
2776,AXL,,10.1016/j.ejmech.2022.114253,,,,
2777,AXL,,10.1016/j.ejmech.2022.114253,,,,
2778,AXL,,10.1016/j.ejmech.2022.114253,,,,
2779,AXL,,10.1016/j.ejmech.2022.114253,,,,
2780,AXL,,10.1016/j.ejmech.2022.114253,,,,
2781,AXL,,10.1016/j.ejmech.2022.114253,,,,
2782,AXL,,10.1016/j.ejmech.2022.114253,,,,
2783,AXL,,10.1016/j.ejmech.2022.114253,,,,
2784,AXL,,10.1016/j.ejmech.2022.114253,,,,
2785,AXL,,10.1016/j.ejmech.2022.114253,,,,
2786,AXL,,10.1016/j.ejmech.2022.114253,,,,
2787,AXL,,10.1016/j.ejmech.2022.114253,,,,
2788,AXL,,10.1016/j.ejmech.2022.114253,,,,
2789,AXL,,10.1016/j.ejmech.2022.114253,,,,
2790,AXL,,10.1016/j.ejmech.2022.114253,,,,
2791,AXL,,10.1016/j.ejmech.2022.114253,,,,
2792,AXL,,10.1016/j.ejmech.2022.114253,,,,
2793,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2794,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2795,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2796,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2797,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2798,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2799,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2800,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2801,MDM2,,10.1016/j.ejmech.2021.113425,4.1,,Degradation of MDM2 in RS4;11 cells after 12 h treatment,
2802,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2803,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2804,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2805,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2806,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2807,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2808,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2809,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2810,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2811,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2812,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2813,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2814,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2815,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2816,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2817,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2818,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2819,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2820,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2821,MDM2,,10.1016/j.ejmech.2021.113425,,,,
2822,MDM2,32/81 (WB),10.1016/j.ejmech.2021.113425,,,,% MDM2 degradation in RS4;11 cells at 10/100 nM
2823,MDM2,0/0 (WB),10.1016/j.ejmech.2021.113425,,,,% MDM2 degradation in RS4;11 cells at 10/100 nM
2824,MDM2,91/92 (WB),10.1016/j.ejmech.2021.113425,,,,% MDM2 degradation in RS4;11 cells at 10/100 nM
2825,MDM2,0/0 (WB),10.1016/j.ejmech.2021.113425,,,,% MDM2 degradation in RS4;11 cells at 10/100 nM
2826,MDM2,0/0 (WB),10.1016/j.ejmech.2021.113425,,,,% MDM2 degradation in RS4;11 cells at 10/100 nM
2827,MDM2,31/74 (WB),10.1016/j.ejmech.2021.113425,,,,% MDM2 degradation in RS4;11 cells at 10/100 nM
2828,MDM2,11/84 (WB),10.1016/j.ejmech.2021.113425,,,,% MDM2 degradation in RS4;11 cells at 10/100 nM
2829,KRAS G12C,,10.1016/j.ejmech.2021.114088,3610/4530,,Degradation of KRAS G12C in H358/H23 cells after 24 h treatment,
2830,BTK,0/13.5 (WB),10.1016/j.ejmech.2021.113820,,,,% BTK degradation in JeKo-1 cells at 100/1000 nM
2830,BTK C481S,,10.1016/j.ejmech.2021.113820,,,,
2831,BTK C481S,,10.1016/j.ejmech.2021.113820,,,,
2831,BTK,25.8/69.6 (WB),10.1016/j.ejmech.2021.113820,,,,% BTK degradation in JeKo-1 cells at 100/1000 nM
2832,BTK C481S,,10.1016/j.ejmech.2021.113820,,,,
2832,BTK,33/35 (WB),10.1016/j.ejmech.2021.113820,,,,% BTK degradation in JeKo-1 cells at 100/1000 nM
2833,BTK,,10.1016/j.ejmech.2021.113820,28.5,67.1,Degradation of BTK in JeKo-1 cells after 24 h treatment,
2833,BTK C481S,,10.1016/j.ejmech.2021.113820,,,,
2834,BTK C481S,,10.1016/j.ejmech.2021.113820,52.7,68.6,Degradation of BTK C481S in TMD8 cells after 24 h treatment,
2834,BTK,,10.1016/j.ejmech.2021.113820,9.4,66.5,Degradation of BTK in JeKo-1 cells after 24 h treatment,
2835,BTK C481S,,10.1016/j.ejmech.2021.113820,80.4,88.4,Degradation of BTK C481S in TMD8 cells after 24 h treatment,
2835,BTK,,10.1016/j.ejmech.2021.113820,8.1,72.4,Degradation of BTK in JeKo-1 cells after 24 h treatment,
2836,BTK C481S,,10.1016/j.ejmech.2021.113820,52.3,84.8,Degradation of BTK C481S in TMD8 cells after 24 h treatment,
2836,BTK,,10.1016/j.ejmech.2021.113820,8.3,92.4,Degradation of BTK in JeKo-1 cells after 24 h treatment,
2837,BTK C481S,,10.1016/j.ejmech.2021.113820,,,,
2837,BTK,22.8/33.8 (WB),10.1016/j.ejmech.2021.113820,,,,% BTK degradation in JeKo-1 cells at 100/1000 nM
2838,BTK C481S,,10.1016/j.ejmech.2021.113820,,,,
2838,BTK,7/0 (WB),10.1016/j.ejmech.2021.113820,,,,% BTK degradation in JeKo-1 cells at 100/1000 nM
2839,BTK C481S,,10.1016/j.ejmech.2021.113820,,,,
2839,BTK,22/6 (WB),10.1016/j.ejmech.2021.113820,,,,% BTK degradation in JeKo-1 cells at 100/1000 nM
2840,BTK,,10.1016/j.ejmech.2021.113820,32.3,76.9,Degradation of BTK in JeKo-1 cells after 24 h treatment,
2840,BTK C481S,,10.1016/j.ejmech.2021.113820,30.1,84.3,Degradation of BTK C481S in TMD8 cells after 24 h treatment,
2841,BTK,,10.1016/j.ejmech.2021.113820,12.1,78,Degradation of BTK in JeKo-1 cells after 24 h treatment,
2841,BTK C481S,,10.1016/j.ejmech.2021.113820,37.9,83.5,Degradation of BTK C481S in TMD8 cells after 24 h treatment,
2842,BTK,,10.1016/j.ejmech.2021.113820,41.9,93,Degradation of BTK in JeKo-1 cells after 24 h treatment,
2842,BTK C481S,,10.1016/j.ejmech.2021.113820,42.9,90.7,Degradation of BTK C481S in TMD8 cells after 24 h treatment,
2843,HDAC6,,10.1021/acschembio.1c00681,108.9,88,Degradation of HDAC6 in K562 cells after 8 h treatment,
2844,HDAC6,,10.1021/acschembio.1c00681,,25,,
2845,HDAC6,,10.1021/acschembio.1c00681,,6.3,,
2846,HDAC6,,10.1021/acschembio.1c00681,,17,,
2847,HDAC6,,10.1021/acschembio.1c00681,,42,,
2848,JAK3,72 (WB),10.1021/acsmedchemlett.1c00650,,,,% JAK3 degradation in MHH-CALL-4 cells at 100 nM
2848,JAK2,,10.1021/acsmedchemlett.1c00245,,,,
2848,JAK2,77 (WB),10.1021/acsmedchemlett.1c00650,,,,% JAK2 degradation in MHH-CALL-4 cells at 100 nM
2849,JAK2,40 (WB),10.1021/acsmedchemlett.1c00650,,,,% JAK2 degradation in MHH-CALL-4 cells at 100 nM
2849,JAK3,29 (WB),10.1021/acsmedchemlett.1c00650,,,,% JAK3 degradation in MHH-CALL-4 cells at 100 nM
2850,JAK2,,10.1021/acsmedchemlett.1c00650,21,,Degradation of JAK2 in MHH-CALL-4 cells after 24 h treatment,
2850,JAK3,61 (WB),10.1021/acsmedchemlett.1c00650,,,,% JAK3 degradation in MHH-CALL-4 cells at 100 nM
2851,JAK2,77 (WB),10.1021/acsmedchemlett.1c00650,,,,% JAK2 degradation in MHH-CALL-4 cells at 100 nM
2851,JAK3,58 (WB),10.1021/acsmedchemlett.1c00650,,,,% JAK3 degradation in MHH-CALL-4 cells at 100 nM
2851,JAK2,,10.1021/acsmedchemlett.1c00245,,,,
2852,JAK2,,10.1021/acsmedchemlett.1c00650,14,,Degradation of JAK2 in MHH-CALL-4 cells after 24 h treatment,
2852,JAK3,43 (WB),10.1021/acsmedchemlett.1c00650,,,,% JAK3 degradation in MHH-CALL-4 cells at 100 nM
2853,JAK2,,10.1021/acsmedchemlett.1c00650,17,,Degradation of JAK2 in MHH-CALL-4 cells after 24 h treatment,
2853,JAK3,,10.1021/acsmedchemlett.1c00650,,,,
2854,JAK2,72 (WB),10.1021/acsmedchemlett.1c00650,,,,% JAK2 degradation in MHH-CALL-4 cells at 100 nM
2854,JAK3,54 (WB),10.1021/acsmedchemlett.1c00650,,,,% JAK3 degradation in MHH-CALL-4 cells at 100 nM
2855,JAK2,,10.1021/acsmedchemlett.1c00650,26,,Degradation of JAK2 in MHH-CALL-4 cells after 24 h treatment,
2855,JAK3,42 (WB),10.1021/acsmedchemlett.1c00650,,,,% JAK3 degradation in MHH-CALL-4 cells at 100 nM
2856,JAK2,1/32/69/19 (WB),10.1021/acsmedchemlett.1c00650,,,,% JAK2 degradation in MHH-CALL-4 cells at 1/10/100/1000 nM
2856,JAK3,72 (WB),10.1021/acsmedchemlett.1c00650,,,,% JAK3 degradation in MHH-CALL-4 cells at 100 nM
2857,JAK3,,10.1021/acsmedchemlett.1c00650,11,92,Degradation of JAK3 in PDX SJBALL020589 cells after 24 h treatment,
2857,JAK2,,10.1021/acsmedchemlett.1c00650,14/24,90/82,Degradation of JAK2 in PDX SJBALL020589/MHH-CALL-4 cells after 24 h treatment,
2857,JAK2 R683G,,10.1021/acsmedchemlett.1c00650,74,,Degradation of JAK2 R683G in KOPN49 cells after 24 h treatment,
2858,JAK2,,10.1021/acsmedchemlett.1c00650,,,,
2858,JAK3,,10.1021/acsmedchemlett.1c00650,,,,
2859,JAK2,,10.1021/acsmedchemlett.1c00650,,,,
2859,JAK3,,10.1021/acsmedchemlett.1c00650,,,,
2860,EGFR del19/T790M/C797S,,10.1021/acsmedchemlett.1c00645,,,,
2861,EGFR del19/T790M/C797S,,10.1021/acsmedchemlett.1c00645,,,,
2862,EGFR del19/T790M/C797S,,10.1021/acsmedchemlett.1c00645,,,,
2863,EGFR del19/T790M/C797S,,10.1021/acsmedchemlett.1c00645,,,,
2864,EGFR del19/T790M/C797S,,10.1021/acsmedchemlett.1c00645,,,,
2865,EGFR del19/T790M/C797S,,10.1021/acsmedchemlett.1c00645,,,,
2866,EGFR del19/T790M/C797S,,10.1021/acsmedchemlett.1c00645,,,,
2867,EGFR del19/T790M/C797S,,10.1021/acsmedchemlett.1c00645,8,,Degradation of EGFR del19/T790M/C797S in Ba/F3 cells after 3 h treatment,
2867,EGFR e19d,0/30/30/53/29 (WB),10.1021/acsmedchemlett.1c00645,,,,% EGFR del19 degradation in HCC827 cells at 5/10/50/100/500 nM
2867,EGFR L858R/T790M,10/7/7/27/34 (WB),10.1021/acsmedchemlett.1c00645,,,,% EGFR EGFR L858R/T790M degradation in H1975 cells at 5/10/50/100/500 nM
2868,EGFR del19/T790M/C797S,,10.1021/acsmedchemlett.1c00645,,,,
2869,STAT3,,10.1021/acsmedchemlett.1c00155,120/17/1200,,Degradation of STAT3 in MOLM-16/SU-DHL-1/SUP-M2 cells after 4/14/14 h treatment,
2870,FGFR2,,10.1002/anie.202101328,,,,
2871,FGFR2,,10.1002/anie.202101328,,,,
2872,FGFR2,,10.1002/anie.202101328,,,,
2873,FGFR2,,10.1002/anie.202101328,,,,
2874,FGFR2,,10.1002/anie.202101328,,,,
2875,FGFR2,,10.1002/anie.202101328,,,,
2876,FGFR2,,10.1002/anie.202101328,,,,
2877,FGFR2,,10.1002/anie.202101328,,,,
2878,FGFR2,,10.1002/anie.202101328,70,74,Degradation of FGFR2 in KATO III cells after 6 h treatment,
2878,FGFR1,,10.1002/anie.202101328,4.35,85,Degradation of FGFR1 in CCLP1 cells after 16 h treatment,
2879,FGFR2,,10.1002/anie.202101328,,,,
2880,FGFR2,,10.1002/anie.202101328,,,,
2881,FGFR2,,10.1002/anie.202101328,,,,
2882,FGFR2,,10.1002/anie.202101328,,,,
2883,FGFR2,,10.1002/anie.202101328,,,,
2884,FGFR2,,10.1002/anie.202101328,,,,
2885,FGFR2,,10.1002/anie.202101328,,,,
2886,CCR9,,10.1002/anie.202116782,,,,
2887,FAK,,10.1002/anie.202109237,125.9,,Degradation of FAK in A549 cells after 24 h treatment,
2888,FAK,,10.1002/anie.202109237,20,,Degradation of FAK in A549 cells after 24 h treatment,
2889,FAK,,10.1002/anie.202109237,158.5,,Degradation of FAK in A549 cells after 24 h treatment,
2890,FAK,,10.1002/anie.202109237,31.6,,Degradation of FAK in A549 cells after 24 h treatment,
2891,FAK,,10.1002/anie.202109237,39.8,,Degradation of FAK in A549 cells after 24 h treatment,
2892,FAK,,10.1002/anie.202109237,4,,Degradation of FAK in A549 cells after 24 h treatment,
2893,BRD4,,10.1002/anie.202108848,,,,
2893,BRD2,,10.1002/anie.202108848,,,,
2894,BRD4,,10.1002/anie.202108848,,,,
2894,BRD2,,10.1002/anie.202108848,,,,
2895,BRD2,,10.1002/anie.202108848,,,,
2895,BRD4,,10.1002/anie.202108848,,,,
2896,BRD4,,10.1002/anie.202108848,,,,
2896,BRD2,,10.1002/anie.202108848,,,,
2897,BRD2,,10.1002/anie.202108848,,,,
2897,BRD4,,10.1002/anie.202108848,,,,
2898,BRD4,,10.1002/anie.202108848,0.87/0.16,,Degradation of BRD4 in MV4-11 cells after 12/24 h treatment,
2898,BRD2,,10.1002/anie.202108848,,,,
2898,BRD4,,10.1002/anie.202108848,24,,Degradation of BRD4 in HD-MB03 cells after 12 h treatment,
2899,BRD2,,10.1002/anie.202108848,,,,
2899,BRD4,,10.1002/anie.202108848,,,,
2900,BRD2,,10.1002/anie.202108848,,,,
2900,BRD4,,10.1002/anie.202108848,,,,
2901,MIF,0/16,10.1002/anie.202101864,,,,% MIF degradation in A549 cells after 12 h treatment at 2000/20000 nM
2902,MIF,0/31,10.1002/anie.202101864,,,,% MIF degradation in A549 cells after 12 h treatment at 2000/20000 nM
2903,MIF,0/22,10.1002/anie.202101864,,,,% MIF degradation in A549 cells after 12 h treatment at 2000/20000 nM
2904,MIF,0/50,10.1002/anie.202101864,,,,% MIF degradation in A549 cells after 12 h treatment at 2000/20000 nM
2905,MIF,0/58,10.1002/anie.202101864,,,,% MIF degradation in A549 cells after 12 h treatment at 2000/20000 nM
2906,MIF,0/0,10.1002/anie.202101864,,,,% MIF degradation in A549 cells after 12 h treatment at 2000/20000 nM
2907,MIF,0/61,10.1002/anie.202101864,,,,% MIF degradation in A549 cells after 12 h treatment at 2000/20000 nM
2908,MIF,21/51,10.1002/anie.202101864,,,,% MIF degradation in A549 cells after 12 h treatment at 2000/20000 nM
2909,MIF,,10.1002/anie.202101864,1500,,Degradation of MIF in A549 cells after 12 h treatment,
2910,MIF,55/61,10.1002/anie.202101864,,,,% MIF degradation in A549 cells after 12 h treatment at 2000/20000 nM
2911,MIF,0/40,10.1002/anie.202101864,,,,% MIF degradation in A549 cells after 12 h treatment at 2000/20000 nM
2912,MIF,0/38,10.1002/anie.202101864,,,,% MIF degradation in A549 cells after 12 h treatment at 2000/20000 nM
2913,MIF,,10.1002/anie.202101864,100,90-95,Degradation of MIF in A549 cells after 12 h treatment,
2914,MIF,51/64,10.1002/anie.202101864,,,,% MIF degradation in A549 cells after 12 h treatment at 2000/20000 nM
2915,PI3Kalpha,,10.1016/j.bmc.2022.116707,,,,
2916,PI3Kalpha,,10.1016/j.bmc.2022.116707,,,,
2917,PI3Kalpha,,10.1016/j.bmc.2022.116707,,,,
2918,PI3Kalpha,,10.1016/j.bmc.2022.116707,,,,
2919,PI3Kalpha,,10.1016/j.bmc.2022.116707,,,,
2920,PI3Kalpha,,10.1016/j.bmc.2022.116707,,,,
2921,PI3Kalpha,,10.1016/j.bmc.2022.116707,,,,
2922,PI3Kalpha,,10.1016/j.bmc.2022.116707,,,,
2923,PI3Kalpha,,10.1016/j.bmc.2022.116707,,,,
2924,PI3Kalpha,,10.1016/j.bmc.2022.116707,,,,
2925,PI3Kalpha,,10.1016/j.bmc.2022.116707,,,,
2926,PI3Kalpha,,10.1016/j.bmc.2022.116707,,,,
2927,PI3Kalpha,,10.1016/j.bmc.2022.116707,,,,
2928,FLT3-ITD-D835V,,10.1016/j.bioorg.2021.105508,,,,
2928,FLT3,,10.1016/j.bioorg.2021.105508,,,,
2928,FLT3-ITD,,10.1016/j.bioorg.2021.105508,,,,
2928,FLT3-ITD-F691L,,10.1016/j.bioorg.2021.105508,,,,
2929,FLT3-ITD-D835V,,10.1016/j.bioorg.2021.105508,,,,
2929,FLT3,,10.1016/j.bioorg.2021.105508,,,,
2929,FLT3-ITD,,10.1016/j.bioorg.2021.105508,,,,
2929,FLT3-ITD-F691L,,10.1016/j.bioorg.2021.105508,,,,
2930,FLT3-ITD-D835V,,10.1016/j.bioorg.2021.105508,,,,
2930,FLT3,,10.1016/j.bioorg.2021.105508,,,,
2930,FLT3-ITD,,10.1016/j.bioorg.2021.105508,,,,
2930,FLT3-ITD-F691L,,10.1016/j.bioorg.2021.105508,,,,
2931,FLT3-ITD-D835V,,10.1016/j.bioorg.2021.105508,,,,
2931,FLT3,,10.1016/j.bioorg.2021.105508,,,,
2931,FLT3-ITD,,10.1016/j.bioorg.2021.105508,,,,
2931,FLT3-ITD-F691L,,10.1016/j.bioorg.2021.105508,,,,
2932,FLT3-ITD-F691L,,10.1016/j.bioorg.2021.105508,,,,
2932,FLT3,,10.1016/j.bioorg.2021.105508,,,,
2932,FLT3-ITD,,10.1016/j.bioorg.2021.105508,,,,
2932,FLT3-ITD-D835V,,10.1016/j.bioorg.2021.105508,,,,
2933,FLT3-ITD-F691L,,10.1016/j.bioorg.2021.105508,,,,
2933,FLT3,,10.1016/j.bioorg.2021.105508,,,,
2933,FLT3-ITD,,10.1016/j.bioorg.2021.105508,,,,
2933,FLT3-ITD-D835V,,10.1016/j.bioorg.2021.105508,,,,
2934,FLT3-ITD-D835V,,10.1016/j.bioorg.2021.105508,,,,
2934,FLT3,,10.1016/j.bioorg.2021.105508,,,,
2934,FLT3-ITD,,10.1016/j.bioorg.2021.105508,,,,
2934,FLT3-ITD-F691L,,10.1016/j.bioorg.2021.105508,,,,
2935,FLT3-ITD-D835V,,10.1016/j.bioorg.2021.105508,,,,
2935,FLT3,,10.1016/j.bioorg.2021.105508,,,,
2935,FLT3-ITD,,10.1016/j.bioorg.2021.105508,,,,
2935,FLT3-ITD-F691L,,10.1016/j.bioorg.2021.105508,,,,
2936,FLT3-ITD-D835V,,10.1016/j.bioorg.2021.105508,,,,
2936,FLT3,,10.1016/j.bioorg.2021.105508,,,,
2936,FLT3-ITD,,10.1016/j.bioorg.2021.105508,,,,
2936,FLT3-ITD-F691L,,10.1016/j.bioorg.2021.105508,,,,
2937,FLT3-ITD-D835V,,10.1016/j.bioorg.2021.105508,,,,
2937,FLT3,,10.1016/j.bioorg.2021.105508,,,,
2937,FLT3-ITD,,10.1016/j.bioorg.2021.105508,,,,
2937,FLT3-ITD-F691L,,10.1016/j.bioorg.2021.105508,,,,
2938,FLT3-ITD-D835V,,10.1016/j.bioorg.2021.105508,,,,
2938,FLT3,,10.1016/j.bioorg.2021.105508,,,,
2938,FLT3-ITD,,10.1016/j.bioorg.2021.105508,,,,
2938,FLT3-ITD-F691L,,10.1016/j.bioorg.2021.105508,,,,
2939,FLT3-ITD-D835V,,10.1016/j.bioorg.2021.105508,,,,
2939,FLT3,,10.1016/j.bioorg.2021.105508,,,,
2939,FLT3-ITD,,10.1016/j.bioorg.2021.105508,,,,
2939,FLT3-ITD-F691L,,10.1016/j.bioorg.2021.105508,,,,
2940,FLT3-ITD,,10.1016/j.bioorg.2021.105508,,,,
2940,FLT3,,10.1016/j.bioorg.2021.105508,,,,
2940,FLT3-ITD-F691L,,10.1016/j.bioorg.2021.105508,,,,
2940,FLT3-ITD-D835V,,10.1016/j.bioorg.2021.105508,,,,
2941,FLT3,,10.1016/j.bioorg.2021.105508,,,,
2941,FLT3-ITD,,10.1016/j.bioorg.2021.105508,,,,
2941,FLT3-ITD-D835V,,10.1016/j.bioorg.2021.105508,,,,
2941,FLT3-ITD-F691L,,10.1016/j.bioorg.2021.105508,,,,
2942,FLT3-ITD-D835V,,10.1016/j.bioorg.2021.105508,,,,
2942,FLT3-ITD-F691L,,10.1016/j.bioorg.2021.105508,,,,
2942,FLT3-ITD,,10.1016/j.bioorg.2021.105508,76.7,,Degradation of FLT3-ITD in BaF3 FLT3-ITD cells after 24 h treatment,
2942,FLT3,,10.1016/j.bioorg.2021.105508,,,,
2943,FLT3-ITD,,10.1016/j.bioorg.2021.105508,,,,
2943,FLT3-ITD-F691L,,10.1016/j.bioorg.2021.105508,,,,
2943,FLT3,,10.1016/j.bioorg.2021.105508,,,,
2943,FLT3-ITD-D835V,,10.1016/j.bioorg.2021.105508,,,,
2944,FLT3-ITD,,10.1016/j.bioorg.2021.105508,,,,
2944,FLT3-ITD-F691L,,10.1016/j.bioorg.2021.105508,,,,
2944,FLT3,,10.1016/j.bioorg.2021.105508,,,,
2944,FLT3-ITD-D835V,,10.1016/j.bioorg.2021.105508,,,,
2945,FLT3-ITD,,10.1016/j.bioorg.2021.105508,,,,
2945,FLT3-ITD-F691L,,10.1016/j.bioorg.2021.105508,,,,
2945,FLT3,,10.1016/j.bioorg.2021.105508,,,,
2945,FLT3-ITD-D835V,,10.1016/j.bioorg.2021.105508,,,,
2946,MYC,,10.1016/j.bioorg.2021.105505,,,,
2947,MDM2,,10.1016/j.bioorg.2021.104901,,,,
2948,MDM2,,10.1016/j.bioorg.2021.104901,,,,
2949,MDM2,,10.1016/j.bioorg.2021.104901,,,,
2950,MDM2,,10.1016/j.bioorg.2021.104901,,,,
2951,MDM2,,10.1016/j.bioorg.2021.104901,,,,
2952,MDM2,,10.1016/j.bioorg.2021.104901,,,,
2953,PD-L1,,10.1016/j.bioorg.2021.104833,,,,
2954,PD-L1,,10.1016/j.bioorg.2021.104833,,,,
2955,PD-L1,,10.1016/j.bioorg.2021.104833,,,,
2956,PD-L1,,10.1016/j.bioorg.2021.104833,,,,
2957,PD-L1,,10.1016/j.bioorg.2021.104833,,,,
2958,PD-L1,,10.1016/j.bioorg.2021.104833,,,,
2959,PD-L1,,10.1016/j.bioorg.2021.104833,,,,
2960,PD-L1,,10.1016/j.bioorg.2021.104833,,,,
2961,PD-L1,,10.1016/j.bioorg.2021.104833,,,,
2962,PD-L1,,10.1016/j.bioorg.2021.104833,,,,
2963,PD-L1,,10.1016/j.bioorg.2021.104833,,,,
2964,PD-L1,,10.1016/j.bioorg.2021.104833,,,,
2965,PD-L1,,10.1016/j.bioorg.2021.104833,,,,
2966,PD-L1,,10.1016/j.bioorg.2021.104833,,,,
2967,PD-L1,,10.1016/j.bioorg.2021.104833,,,,
2968,PD-L1,,10.1016/j.bioorg.2021.104833,,,,
2969,PD-L1,,10.1016/j.bioorg.2021.104833,,,,
2970,PD-L1,,10.1016/j.bioorg.2021.104833,,,,
2971,PD-L1,,10.1016/j.bioorg.2021.104833,,,,
2972,KRAS G12C,,10.1016/j.bioorg.2021.105447,,N.D.,,
2973,KRAS G12C,,10.1016/j.bioorg.2021.105447,,N.D.,,
2974,KRAS G12C,,10.1016/j.bioorg.2021.105447,,N.D.,,
2975,KRAS G12C,,10.1016/j.bioorg.2021.105447,,N.D.,,
2976,KRAS G12C,,10.1016/j.bioorg.2021.105447,,N.D.,,
2977,KRAS G12C,,10.1016/j.bioorg.2021.105447,,N.D.,,
2978,KRAS G12C,,10.1016/j.bioorg.2021.105447,,N.D.,,
2979,KRAS G12C,,10.1016/j.bioorg.2021.105447,,N.D.,,
2980,KRAS G12C,,10.1016/j.bioorg.2021.105447,,N.D.,,
2981,KRAS G12C,,10.1016/j.bioorg.2021.105447,,N.D.,,
2982,KRAS G12C,,10.1016/j.bioorg.2021.105447,,,,
2983,KRAS G12C,,10.1016/j.bioorg.2021.105447,,,,
2984,KRAS G12C,,10.1016/j.bioorg.2021.105447,,,,
2985,KRAS G12C,,10.1016/j.bioorg.2021.105447,1250/2500,,Degradation of KRAS G12C in NCI-H358/NCI-H23 cells after 48 h treatment,
2986,KRAS G12C,,10.1016/j.bioorg.2021.105447,,,,
2987,KRAS G12C,,10.1016/j.bioorg.2021.105447,,,,
2988,KRAS G12C,,10.1016/j.bioorg.2021.105447,,,,
2989,KRAS G12C,,10.1016/j.bioorg.2021.105447,,,,
2990,SHP2,,10.1021/acs.biochem.1c00377,,N.D.,,
2991,SHP2,,10.1021/acs.biochem.1c00377,,N.D.,,
2992,SHP2,,10.1021/acs.biochem.1c00377,,N.D.,,
2993,SHP2,,10.1021/acs.biochem.1c00377,,N.D.,,
2994,SHP2,,10.1021/acs.biochem.1c00377,,,,
2994,SHP2 F285S,,10.1021/acs.biochem.1c00377,,,,
2995,SHP2 F285S,,10.1021/acs.biochem.1c00377,,,,
2995,SHP2,,10.1021/acs.biochem.1c00377,,,,
2996,SHP2,,10.1021/acs.biochem.1c00377,,,,
2996,SHP2 F285S,,10.1021/acs.biochem.1c00377,,,,
2997,Wee1,,10.1016/j.bmcl.2022.128636,,,,
2998,Wee1,,10.1016/j.bmcl.2022.128636,,,,
2999,Wee1,,10.1016/j.bmcl.2022.128636,,,,
3000,Wee1,,10.1016/j.bmcl.2022.128636,,,,
3001,Wee1,,10.1016/j.bmcl.2022.128636,,,,
3002,Wee1,,10.1016/j.bmcl.2022.128636,,,,
3003,Wee1,,10.1016/j.bmcl.2022.128636,,,,
3004,Wee1,,10.1016/j.bmcl.2022.128636,,,,
3005,Wee1,,10.1016/j.bmcl.2022.128636,,,,
3006,Wee1,,10.1016/j.bmcl.2022.128636,,,,
3007,Wee1,,10.1016/j.bmcl.2022.128636,,,,
3008,Wee1,,10.1016/j.bmcl.2022.128636,,,,
3009,Wee1,,10.1016/j.bmcl.2022.128636,,,,
3010,Wee1,,10.1016/j.bmcl.2022.128636,,,,
3011,Wee1,,10.1016/j.bmcl.2022.128636,,,,
3012,Wee1,,10.1016/j.bmcl.2022.128636,,,,
3013,Wee1,,10.1016/j.bmcl.2022.128636,,,,
3014,Wee1,,10.1016/j.bmcl.2022.128636,,,,
3015,Wee1,,10.1016/j.bmcl.2022.128636,,,,
3016,Wee1,,10.1016/j.bmcl.2022.128636,,,,
3017,AR-V7,,10.1016/j.bmcl.2021.128448,,N.D.,,
3018,AR-V7,,10.1016/j.bmcl.2021.128448,350,53,Degradation of AR-V7 in 22RV1 cells after 24 h treatment,
3019,AR-V7,,10.1016/j.bmcl.2021.128448,,N.D.,,
3020,AR-V7,,10.1016/j.bmcl.2021.128448,,N.D.,,
3021,AR-V7,,10.1016/j.bmcl.2021.128448,320,67,Degradation of AR-V7 in 22RV1 cells after 24 h treatment,
3022,AR-V7,,10.1016/j.bmcl.2021.128448,,,,
3023,AR-V7,,10.1016/j.bmcl.2021.128448,,,,
3024,AR-V7,,10.1016/j.bmcl.2021.128448,>10000,,Degradation of AR-V7 in 22RV1 cells after 24 h treatment,
3025,AR-V7,,10.1016/j.bmcl.2021.128448,,,,
3026,AR-V7,,10.1016/j.bmcl.2021.128448,,,,
3027,AR-V7,,10.1016/j.bmcl.2021.128448,>10000,,Degradation of AR-V7 in 22RV1 cells after 24 h treatment,
3028,AR-V7,,10.1016/j.bmcl.2021.128448,,,,
3029,AR-V7,,10.1016/j.bmcl.2021.128448,>10000,,Degradation of AR-V7 in 22RV1 cells after 24 h treatment,
3030,AR-V7,,10.1016/j.bmcl.2021.128448,,,,
3031,AR-V7,,10.1016/j.bmcl.2021.128448,,,,
3032,AR-V7,,10.1016/j.bmcl.2021.128448,,,,
3033,AR-V7,,10.1016/j.bmcl.2021.128448,,,,
3034,AR-V7,,10.1016/j.bmcl.2021.128448,,,,
3035,AR-V7,,10.1016/j.bmcl.2021.128448,>10000,,Degradation of AR-V7 in 22RV1 cells after 24 h treatment,
3036,AR-V7,,10.1016/j.bmcl.2021.128448,,,,
3037,AR-V7,,10.1016/j.bmcl.2021.128448,,,,
3038,AR-V7,,10.1016/j.bmcl.2021.128448,,,,
3039,AR-V7,,10.1016/j.bmcl.2021.128448,,,,
3040,AR-V7,,10.1016/j.bmcl.2021.128448,,,,
3041,AR-V7,,10.1016/j.bmcl.2021.128448,,,,
3042,AR-V7,,10.1016/j.bmcl.2021.128448,,,,
3043,AR-V7,,10.1016/j.bmcl.2021.128448,,,,
3044,TACC3,,10.1111/cas.13198,,,,
3045,TACC3,,10.1111/cas.13198,,,,
3046,TACC3,,10.1111/cas.13198,,,,
3047,FGFR3-TACC3,,10.1016/j.bmcl.2022.128584,,,,
3048,FGFR3-TACC3,,10.1016/j.bmcl.2022.128584,,,,
3049,FGFR3-TACC3,,10.1016/j.bmcl.2022.128584,,,,
3050,FGFR3-TACC3,,10.1016/j.bmcl.2022.128584,,,,
3051,FGFR3-TACC3,,10.1016/j.bmcl.2022.128584,,,,
3052,FGFR3-TACC3,,10.1016/j.bmcl.2022.128584,,,,
3053,AR,>=90/>=90,10.1021/acsmedchemlett.1c00498,,,,% AR degradation in Vcap cells after 24 h treatment at 10/100 nM
3054,AR,>=90/>=90,10.1021/acsmedchemlett.1c00498,,,,% AR degradation in Vcap cells after 24 h treatment at 10/100 nM
3055,AR,>=90/>=90,10.1021/acsmedchemlett.1c00498,,,,% AR degradation in Vcap cells after 24 h treatment at 10/100 nM
3056,AR,>=90/>=90,10.1021/acsmedchemlett.1c00498,,,,% AR degradation in Vcap cells after 24 h treatment at 10/100 nM
3057,AR,>=90/>=90,10.1021/acsmedchemlett.1c00498,,,,% AR degradation in Vcap cells after 24 h treatment at 10/100 nM
3058,AR,>=90/>=90,10.1021/acsmedchemlett.1c00498,,,,% AR degradation in Vcap cells after 24 h treatment at 10/100 nM
3059,AR,>=90/>=90,10.1021/acsmedchemlett.1c00498,,,,% AR degradation in Vcap cells after 24 h treatment at 10/100 nM
3060,AR,>=90/>=90,10.1021/acsmedchemlett.1c00498,,,,% AR degradation in Vcap cells after 24 h treatment at 10/100 nM
3061,AR,>=50/>=90,10.1021/acsmedchemlett.1c00498,,,,% AR degradation in Vcap cells after 24 h treatment at 10/100 nM
3062,AR,>=90/>=90,10.1021/acsmedchemlett.1c00498,,,,% AR degradation in Vcap cells after 24 h treatment at 10/100 nM
3063,AR,>=90/>=90,10.1021/acsmedchemlett.1c00498,,,,% AR degradation in Vcap cells after 24 h treatment at 10/100 nM
3064,AR,>=90/>=90,10.1021/acsmedchemlett.1c00498,,,,% AR degradation in Vcap cells after 24 h treatment at 10/100 nM
3065,IRAK1,,10.1021/acsmedchemlett.1c00244,16,95,Degradation of IRAK1 in HEK293T cells after 24 h treatment,
3066,IRAK1,,10.1021/acsmedchemlett.1c00244,3,96,Degradation of IRAK1 in HEK293T cells after 24 h treatment,
3067,IRAK1,,10.1021/acsmedchemlett.1c00244,16,97,Degradation of IRAK1 in HEK293T cells after 24 h treatment,
3068,IRAK1,,10.1021/acsmedchemlett.1c00244,9,90,Degradation of IRAK1 in HEK293T cells after 24 h treatment,
3069,IRAK1,,10.1021/acsmedchemlett.1c00244,13,96,Degradation of IRAK1 in HEK293T cells after 24 h treatment,
3070,IRAK1,,10.1021/acsmedchemlett.1c00244,13,94,Degradation of IRAK1 in HEK293T cells after 24 h treatment,
3071,IRAK1,,10.1021/acsmedchemlett.1c00244,21,96,Degradation of IRAK1 in HEK293T cells after 24 h treatment,
3072,IRAK1,,10.1021/acsmedchemlett.1c00244,,95,,
3073,JAK2,,10.1021/acsmedchemlett.1c00245,,,,
3074,JAK2,,10.1021/acsmedchemlett.1c00245,,,,
3075,JAK2,,10.1021/acsmedchemlett.1c00245,,,,
3076,JAK2,,10.1021/acsmedchemlett.1c00245,,,,
3077,JAK2,,10.1021/acsmedchemlett.1c00245,,,,
3078,JAK2,,10.1021/acsmedchemlett.1c00245,,,,
3079,JAK2,,10.1021/acsmedchemlett.1c00245,,,,
3080,JAK2,,10.1021/acsmedchemlett.1c00245,,,,
3081,JAK2,,10.1021/acsmedchemlett.1c00245,,,,
3082,JAK2,,10.1021/acsmedchemlett.1c00245,,,,
3083,BTK,,10.1021/acsmedchemlett.1c00178,68,,Degradation of BTK in Ramos cells after 16 h treatment by ELISA assay,
3084,BTK,,10.1021/acsmedchemlett.1c00178,78,,Degradation of BTK in Ramos cells after 16 h treatment by ELISA assay,
3085,BTK,,10.1021/acsmedchemlett.1c00178,78,,Degradation of BTK in Ramos cells after 16 h treatment by ELISA assay,
3086,BTK,,10.1021/acsmedchemlett.1c00178,107,,Degradation of BTK in Ramos cells after 16 h treatment by ELISA assay,
3087,BTK,,10.1021/acsmedchemlett.1c00178,34,,Degradation of BTK in Ramos cells after 16 h treatment by ELISA assay,
3088,BTK,,10.1021/acsmedchemlett.1c00178,74,,Degradation of BTK in Ramos cells after 16 h treatment by ELISA assay,
3089,BTK,,10.1021/acsmedchemlett.1c00178,28,,Degradation of BTK in Ramos cells after 16 h treatment by ELISA assay,
3090,BTK,,10.1021/acsmedchemlett.1c00178,2.9,,Degradation of BTK in Ramos cells after 16 h treatment by ELISA assay,
3091,BTK,,10.1021/acsmedchemlett.1c00178,35,,Degradation of BTK in Ramos cells after 16 h treatment by ELISA assay,
3092,BTK,,10.1021/acsmedchemlett.1c00178,17,,Degradation of BTK in Ramos cells after 16 h treatment by ELISA assay,
3093,BTK,,10.1021/acsmedchemlett.1c00178,35,,Degradation of BTK in Ramos cells after 16 h treatment by ELISA assay,
3094,BTK,,10.1021/acsmedchemlett.1c00178,7.2,,Degradation of BTK in Ramos cells after 16 h treatment by ELISA assay,
3095,BRD9,,10.1021/acsmedchemlett.1c00580,1,,Degradation of BRD9 in HEK293A cells after 24 h treatment,
3096,BRD9,,10.1021/acsmedchemlett.1c00580,1,,Degradation of BRD9 in HEK293A cells after 24 h treatment,
3097,BRD9,,10.1021/acsmedchemlett.1c00580,1,,Degradation of BRD9 in HEK293A cells after 24 h treatment,
3098,BRD9,,10.1021/acsmedchemlett.1c00580,1,,Degradation of BRD9 in HEK293A cells after 24 h treatment,
3099,BRD9,,10.1021/acsmedchemlett.1c00580,1,,Degradation of BRD9 in HEK293A cells after 24 h treatment,
3100,BRD9,,10.1021/acsmedchemlett.1c00580,1,,Degradation of BRD9 in HEK293A cells after 24 h treatment,
3101,SMARCA2,,10.1021/acsmedchemlett.1c00657,4,,Degradation of SMARCA2 HiBiT in HT1080 cells after 6 h treatment,
3102,SMARCA2,,10.1021/acsmedchemlett.1c00657,2,,Degradation of SMARCA2 HiBiT in HT1080 cells after 6 h treatment,
3103,SMARCA2,,10.1021/acsmedchemlett.1c00657,2,,Degradation of SMARCA2 HiBiT in HT1080 cells after 6 h treatment,
3104,SMARCA2,,10.1021/acsmedchemlett.1c00657,3,,Degradation of SMARCA2 HiBiT in HT1080 cells after 6 h treatment,
3105,SMARCA2,,10.1021/acsmedchemlett.1c00657,3,,Degradation of SMARCA2 HiBiT in HT1080 cells after 6 h treatment,
3106,SMARCA2,,10.1021/acsmedchemlett.1c00657,3,,Degradation of SMARCA2 HiBiT in HT1080 cells after 6 h treatment,
3107,BRAF V600E,,10.1021/acsmedchemlett.2c00039,26,,Degradation of BRAF V600E in A375 cells after 24 h treatment,
3108,BRAF V600E,,10.1021/acsmedchemlett.2c00039,10,,Degradation of BRAF V600E in A375 cells after 24 h treatment,
3109,BRAF V600E,,10.1021/acsmedchemlett.2c00039,10,,Degradation of BRAF V600E in A375 cells after 24 h treatment,
3110,BRAF V600E,,10.1021/acsmedchemlett.2c00039,20,,Degradation of BRAF V600E in A375 cells after 24 h treatment,
3111,BRAF V600E,,10.1021/acsmedchemlett.2c00039,23,,Degradation of BRAF V600E in A375 cells after 24 h treatment,
3112,BRAF V600E,,10.1021/acsmedchemlett.2c00039,16,,Degradation of BRAF V600E in A375 cells after 24 h treatment,
3113,MDM2,,10.1016/j.apsb.2020.11.022,,,,
3114,MDM2,,10.1016/j.apsb.2020.11.022,,,,
3115,MDM2,,10.1016/j.apsb.2020.11.022,,,,
3116,MDM2,,10.1016/j.apsb.2020.11.022,,,,
3117,MDM2,,10.1016/j.apsb.2020.11.022,,,,
3118,MDM2,,10.1016/j.apsb.2020.11.022,,,,
3119,MDM2,,10.1016/j.apsb.2020.11.022,,,,
3120,MDM2,,10.1016/j.apsb.2020.11.022,1010,>95,Degradation of MDM2 in A549 cells after 24 h treatment,
3121,MDM2,,10.1016/j.apsb.2020.11.022,,,,
3122,MDM2,,10.1016/j.apsb.2020.11.022,,,,
3123,MDM2,,10.1016/j.apsb.2020.11.022,,,,
3124,MDM2,,10.1016/j.apsb.2020.11.022,,,,
3125,MDM2,,10.1016/j.apsb.2020.11.022,,,,
3126,BCR-ABL T315I,,10.1016/j.apsb.2020.11.009,,,,
3127,BCR-ABL T315I,,10.1016/j.apsb.2020.11.009,,,,
3128,BCR-ABL T315I,,10.1016/j.apsb.2020.11.009,,,,
3129,BCR-ABL T315I,,10.1016/j.apsb.2020.11.009,,,,
3130,BCR-ABL T315I,,10.1016/j.apsb.2020.11.009,,,,
3131,BCR-ABL T315I,,10.1016/j.apsb.2020.11.009,,,,
3132,BCR-ABL T315I,,10.1016/j.apsb.2020.11.009,,,,
3133,BCR-ABL T315I,,10.1016/j.apsb.2020.11.009,,,,
3134,BCR-ABL T315I,,10.1016/j.apsb.2020.11.009,,,,
3135,BCR-ABL T315I,,10.1016/j.apsb.2020.11.009,,,,
3136,BCR-ABL T315I,,10.1016/j.apsb.2020.11.009,,,,
3137,BCR-ABL T315I,,10.1016/j.apsb.2020.11.009,,,,
3138,BCR-ABL T315I,,10.1016/j.apsb.2020.11.009,,,,
3139,BCR-ABL T315I,,10.1016/j.apsb.2020.11.009,108.7,,Degradation of BCR-ABL T315I in Ba/F3 cells after 24 h treatment,
3140,BCR-ABL T315I,,10.1016/j.apsb.2020.11.009,,,,
3141,BCR-ABL T315I,,10.1016/j.apsb.2020.11.009,,,,
3142,BCR-ABL T315I,,10.1016/j.apsb.2020.11.009,,,,
3143,BCR-ABL T315I,,10.1016/j.apsb.2020.11.009,,,,
3144,HMGCR,,10.1016/j.apsb.2020.11.001,,,,
3145,HMGCR,,10.1016/j.apsb.2020.11.001,,,,
3146,HMGCR,,10.1016/j.apsb.2020.11.001,,,,
3147,HMGCR,,10.1016/j.apsb.2020.11.001,,,,
3148,HMGCR,,10.1016/j.apsb.2020.11.001,,,,
3149,HMGCR,,10.1016/j.apsb.2020.11.001,120,76,Degradation of HMGCR in HepG2 cells after 16 h treatment,
3150,BRD4,,10.1021/acschembio.1c00376,5,97,Degradation of BRD4 in HEK293T cells after 3 h treatment,
3151,CDK6,,10.1021/acsmedchemlett.1c00368,,,,
3151,CDK4,,10.1021/acsmedchemlett.1c00368,,,,
3152,CDK4,,10.1021/acsmedchemlett.1c00368,,,,
3152,CDK6,,10.1021/acsmedchemlett.1c00368,,,,
3153,CDK4,,10.1021/acsmedchemlett.1c00368,,,,
3153,CDK6,,10.1021/acsmedchemlett.1c00368,,,,
3154,AR,,10.1002/ardp.202100467,,,,
3155,AR,,10.1002/ardp.202100467,,,,
3156,AR,,10.1002/ardp.202100467,,,,
3157,AR,,10.1002/ardp.202100467,,,,
3158,AR,,10.1002/ardp.202100467,,,,
3159,AR,,10.1002/ardp.202100467,,,,
3160,AR,,10.1002/ardp.202100467,,,,
3161,AR,,10.1002/ardp.202100467,,,,
3162,AR,,10.1002/ardp.202100467,,,,
3163,AR,,10.1002/ardp.202100467,,,,
3164,AR,,10.1002/ardp.202100467,,,,
3165,AR,,10.1002/ardp.202100467,,,,
3166,AR,,10.1002/ardp.202100467,,,,
3167,AR,,10.1002/ardp.202100467,,,,
3168,AR,,10.1002/ardp.202100467,,,,
3169,AR,,10.1002/ardp.202100467,,,,
3170,AR,,10.1002/ardp.202100467,,,,
3171,AR,,10.1002/ardp.202100467,75/77,>75/>85,Degradation of AR in A549/LNCaP cells after 24 h treatment,
3172,AR,,10.1002/ardp.202100467,,,,
3173,SF3B1 K400E,,10.1016/j.chembiol.2021.04.018,,,,
3173,SF3B1,,10.1016/j.chembiol.2021.04.018,244,,Degradation of SF3B1 in K562 cells after 24 h treatment,
3174,BTK C481G,,10.1038/s41375-019-0440-x,26,,Degradation of BTK C481G in HeLa cells after 96 h treatment,
3174,BTK C481W,,10.1038/s41375-019-0440-x,41,,Degradation of BTK C481W in HeLa cells after 96 h treatment,
3174,BTK C481A,,10.1038/s41375-019-0440-x,15,,Degradation of BTK C481A in HeLa cells after 96 h treatment,
3174,BTK,,10.1038/s41375-019-0440-x,18,,Degradation of BTK in HeLa cells after 96 h treatment,
3174,BTK C481S,,10.1038/s41375-019-0440-x,29,,Degradation of BTK C481S in HBL-1 cells after 36 h treatment,
3174,BTK C481T,,10.1038/s41375-019-0440-x,38,,Degradation of BTK C481T in HeLa cells after 96 h treatment,
3175,BTK,,10.1038/s41422-021-00533-6,,,,
3176,BTK,,10.1038/s41422-021-00533-6,,,,
3177,BTK,,10.1038/s41422-021-00533-6,,,,
3178,BTK,,10.1038/s41422-021-00533-6,,,,
3179,BTK,,10.1038/s41422-021-00533-6,,,,
3180,BTK,,10.1038/s41422-021-00533-6,,,,
3181,BTK,,10.1038/s41422-021-00533-6,37,,Degradation of BTK in DOHH2 cells after 24 h treatment,
3182,BTK,,10.1038/s41422-021-00533-6,,,,
3183,BTK,,10.1038/s41422-021-00533-6,,,,
3184,BTK,,10.1038/s41422-021-00533-6,,,,
3185,BTK,,10.1038/s41422-021-00533-6,,,,
3186,BTK,,10.1038/s41422-021-00533-6,,,,
3187,BTK,,10.1038/s41422-021-00533-6,,,,
3188,BTK,,10.1038/s41422-021-00533-6,,,,
3189,EGFR e19d,,10.1039/d1cc05715d,,,,
3190,HDAC8,,10.1039/d2cc00272h,,,,
3191,HDAC8,,10.1039/d2cc00272h,,,,
3192,HDAC8,,10.1039/d2cc00272h,702,,Degradation of HDAC8 in Jurkat cells after 24 h treatment,
3193,HDAC8,,10.1039/d2cc00272h,,,,
3194,Tau,,10.3389/fncel.2022.801179,,,,
3195,Tau,,10.3389/fncel.2022.801179,,,,
3196,Tau,,10.3389/fncel.2022.801179,,,,
3197,Tau,,10.3389/fncel.2022.801179,,,,
3198,Tau,,10.3389/fncel.2022.801179,,,,
3199,Tau,,10.3389/fncel.2022.801179,,,,
3200,Tau,,10.3389/fncel.2022.801179,,,,
3201,Tau,,10.3389/fncel.2022.801179,,,,
3202,Tau,,10.3389/fncel.2022.801179,,,,
3203,Tau,,10.3389/fncel.2022.801179,,,,
3204,Tau,,10.3389/fncel.2022.801179,,,,
3205,Tau,,10.3389/fncel.2022.801179,,,,
3206,LXRB,,10.3389/fchem.2021.674967,,,,
3206,LXRA,,10.3389/fchem.2021.674967,,,,
3207,LXRB,,10.3389/fchem.2021.674967,,,,
3207,LXRA,,10.3389/fchem.2021.674967,,,,
3208,LXRB,,10.3389/fchem.2021.674967,,,,
3208,LXRA,,10.3389/fchem.2021.674967,,,,
3209,LXRA,,10.3389/fchem.2021.674967,,,,
3209,LXRB,,10.3389/fchem.2021.674967,,,,
3210,LXRB,,10.3389/fchem.2021.674967,,,,
3210,LXRA,,10.3389/fchem.2021.674967,,,,
3211,LXRA,,10.3389/fchem.2021.674967,,,,
3211,LXRB,,10.3389/fchem.2021.674967,,,,
3212,LXRB,,10.3389/fchem.2021.674967,,,,
3212,LXRA,,10.3389/fchem.2021.674967,,,,
3213,BCL2,,10.1038/s41467-021-27210-x,,47,,
3213,BCL-xL,,10.1038/s41467-021-27210-x,316.2,56,Degradation of BCL-xL in 293T cells after 16 h treatment,
3214,BCL-xL,,10.1038/s41467-021-27210-x,39.9,91,Degradation of BCL-xL in 293T cells after 16 h treatment,
3214,BCL2,,10.1038/s41467-021-27210-x,,47,,
3215,BCL-xL,,10.1038/s41467-021-27210-x,12.8,85,Degradation of BCL-xL in 293T cells after 16 h treatment,
3215,BCL2,,10.1038/s41467-021-27210-x,179.9,79,Degradation of BCL2 in 293T cells after 16 h treatment,
3216,BCL2,,10.1038/s41467-021-27210-x,54,94,Degradation of BCL2 in 293T cells after 16 h treatment,
3216,BCL-xL,,10.1038/s41467-021-27210-x,12.9,94,Degradation of BCL-xL in 293T cells after 16 h treatment,
3217,BCL2,,10.1038/s41467-021-27210-x,316.2,79,Degradation of BCL2 in 293T cells after 16 h treatment,
3217,BCL-xL,,10.1038/s41467-021-27210-x,12.8,96,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL-xL,,10.1038/s41467-021-27210-x,12.1,81,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL2,,10.1038/s41467-021-27210-x,354.8,69,Degradation of BCL2 in 293T cells after 16 h treatment,
3219,BCL2,,10.1038/s41467-021-27210-x,,38,,
3219,BCL-xL,,10.1038/s41467-021-27210-x,,38,,
3220,BCL-xL,,10.1038/s41467-021-27210-x,,,,
3220,BCL2,,10.1038/s41467-021-27210-x,,,,
3221,BCL2,,10.1038/s41467-021-27210-x,48,,Degradation of BCL2 in 293T cells after 16 h treatment,
3221,BCL-xL,,10.1038/s41467-021-27210-x,6,,Degradation of BCL-xL in 293T cells after 16 h treatment,
3222,HDAC1,,10.3390/molecules26237241,,,,
3222,HDAC6,,10.3390/molecules26237241,,,,
3222,HDAC3,,10.3390/molecules26237241,,,,
3223,HDAC1,,10.3390/molecules26237241,,,,
3223,HDAC6,,10.3390/molecules26237241,,,,
3223,HDAC3,,10.3390/molecules26237241,,,,
3224,HDAC1,,10.3390/molecules26237241,,,,
3224,HDAC6,,10.3390/molecules26237241,,,,
3224,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC6,,10.3390/molecules26237241,,,,
3225,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC3,,10.3390/molecules26237241,,,,
3226,HDAC6,,10.3390/molecules26237241,,,,
3227,HDAC1,,10.3390/molecules26237241,,,,
3227,HDAC3,,10.3390/molecules26237241,,,,
3227,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC1,,10.3390/molecules26237241,,,,
3228,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC1,,10.3390/molecules26237241,,,,
3229,HDAC6,,10.3390/molecules26237241,,,,
3230,HDAC3,,10.3390/molecules26237241,,,,
3230,HDAC1,,10.3390/molecules26237241,,,,
3230,HDAC6,,10.3390/molecules26237241,,,,
3231,HDAC3,,10.3390/molecules26237241,,,,
3231,HDAC1,,10.3390/molecules26237241,,,,
3231,HDAC6,,10.3390/molecules26237241,,,,
3232,HDAC3,,10.3390/molecules26237241,,,,
3232,HDAC1,,10.3390/molecules26237241,,,,
3232,HDAC6,,10.3390/molecules26237241,,,,
3233,HDAC3,,10.3390/molecules26237241,,,,
3233,HDAC1,,10.3390/molecules26237241,,,,
3233,HDAC6,,10.3390/molecules26237241,,,,
3234,HDAC3,,10.3390/molecules26237241,,,,
3234,HDAC1,,10.3390/molecules26237241,,,,
3234,HDAC6,,10.3390/molecules26237241,,,,
3235,HSF1,,10.3390/molecules27051655,,,,
3236,HSF1,,10.3390/molecules27051655,,,,
3217,BCL-xL,,10.1038/s41467-021-27210-x,12.8,96,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL-xL,,10.1038/s41467-021-27210-x,12.1,81,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL2,,10.1038/s41467-021-27210-x,354.8,69,Degradation of BCL2 in 293T cells after 16 h treatment,
3219,BCL2,,10.1038/s41467-021-27210-x,,38,,
3219,BCL-xL,,10.1038/s41467-021-27210-x,,38,,
3220,BCL-xL,,10.1038/s41467-021-27210-x,,,,
3220,BCL2,,10.1038/s41467-021-27210-x,,,,
3221,BCL2,,10.1038/s41467-021-27210-x,48,,Degradation of BCL2 in 293T cells after 16 h treatment,
3221,BCL-xL,,10.1038/s41467-021-27210-x,6,,Degradation of BCL-xL in 293T cells after 16 h treatment,
3222,HDAC1,,10.3390/molecules26237241,,,,
3222,HDAC6,,10.3390/molecules26237241,,,,
3222,HDAC3,,10.3390/molecules26237241,,,,
3223,HDAC1,,10.3390/molecules26237241,,,,
3223,HDAC6,,10.3390/molecules26237241,,,,
3223,HDAC3,,10.3390/molecules26237241,,,,
3224,HDAC1,,10.3390/molecules26237241,,,,
3224,HDAC6,,10.3390/molecules26237241,,,,
3224,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC6,,10.3390/molecules26237241,,,,
3225,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC3,,10.3390/molecules26237241,,,,
3226,HDAC6,,10.3390/molecules26237241,,,,
3227,HDAC1,,10.3390/molecules26237241,,,,
3227,HDAC3,,10.3390/molecules26237241,,,,
3227,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC1,,10.3390/molecules26237241,,,,
3228,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC1,,10.3390/molecules26237241,,,,
3229,HDAC6,,10.3390/molecules26237241,,,,
3230,HDAC3,,10.3390/molecules26237241,,,,
3230,HDAC1,,10.3390/molecules26237241,,,,
3230,HDAC6,,10.3390/molecules26237241,,,,
3231,HDAC3,,10.3390/molecules26237241,,,,
3231,HDAC1,,10.3390/molecules26237241,,,,
3231,HDAC6,,10.3390/molecules26237241,,,,
3232,HDAC3,,10.3390/molecules26237241,,,,
3232,HDAC1,,10.3390/molecules26237241,,,,
3232,HDAC6,,10.3390/molecules26237241,,,,
3233,HDAC3,,10.3390/molecules26237241,,,,
3233,HDAC1,,10.3390/molecules26237241,,,,
3233,HDAC6,,10.3390/molecules26237241,,,,
3234,HDAC3,,10.3390/molecules26237241,,,,
3234,HDAC1,,10.3390/molecules26237241,,,,
3234,HDAC6,,10.3390/molecules26237241,,,,
3235,HSF1,,10.3390/molecules27051655,,,,
3236,HSF1,,10.3390/molecules27051655,,,,
3217,BCL-xL,,10.1038/s41467-021-27210-x,12.8,96,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL-xL,,10.1038/s41467-021-27210-x,12.1,81,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL2,,10.1038/s41467-021-27210-x,354.8,69,Degradation of BCL2 in 293T cells after 16 h treatment,
3219,BCL2,,10.1038/s41467-021-27210-x,,38,,
3219,BCL-xL,,10.1038/s41467-021-27210-x,,38,,
3220,BCL-xL,,10.1038/s41467-021-27210-x,,,,
3220,BCL2,,10.1038/s41467-021-27210-x,,,,
3221,BCL2,,10.1038/s41467-021-27210-x,48,,Degradation of BCL2 in 293T cells after 16 h treatment,
3221,BCL-xL,,10.1038/s41467-021-27210-x,6,,Degradation of BCL-xL in 293T cells after 16 h treatment,
3222,HDAC1,,10.3390/molecules26237241,,,,
3222,HDAC6,,10.3390/molecules26237241,,,,
3222,HDAC3,,10.3390/molecules26237241,,,,
3223,HDAC1,,10.3390/molecules26237241,,,,
3223,HDAC6,,10.3390/molecules26237241,,,,
3223,HDAC3,,10.3390/molecules26237241,,,,
3224,HDAC1,,10.3390/molecules26237241,,,,
3224,HDAC6,,10.3390/molecules26237241,,,,
3224,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC6,,10.3390/molecules26237241,,,,
3225,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC3,,10.3390/molecules26237241,,,,
3226,HDAC6,,10.3390/molecules26237241,,,,
3227,HDAC1,,10.3390/molecules26237241,,,,
3227,HDAC3,,10.3390/molecules26237241,,,,
3227,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC1,,10.3390/molecules26237241,,,,
3228,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC1,,10.3390/molecules26237241,,,,
3229,HDAC6,,10.3390/molecules26237241,,,,
3230,HDAC3,,10.3390/molecules26237241,,,,
3230,HDAC1,,10.3390/molecules26237241,,,,
3230,HDAC6,,10.3390/molecules26237241,,,,
3231,HDAC3,,10.3390/molecules26237241,,,,
3231,HDAC1,,10.3390/molecules26237241,,,,
3231,HDAC6,,10.3390/molecules26237241,,,,
3232,HDAC3,,10.3390/molecules26237241,,,,
3232,HDAC1,,10.3390/molecules26237241,,,,
3232,HDAC6,,10.3390/molecules26237241,,,,
3233,HDAC3,,10.3390/molecules26237241,,,,
3233,HDAC1,,10.3390/molecules26237241,,,,
3233,HDAC6,,10.3390/molecules26237241,,,,
3234,HDAC3,,10.3390/molecules26237241,,,,
3234,HDAC1,,10.3390/molecules26237241,,,,
3234,HDAC6,,10.3390/molecules26237241,,,,
3235,HSF1,,10.3390/molecules27051655,,,,
3236,HSF1,,10.3390/molecules27051655,,,,
3217,BCL-xL,,10.1038/s41467-021-27210-x,12.8,96,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL-xL,,10.1038/s41467-021-27210-x,12.1,81,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL2,,10.1038/s41467-021-27210-x,354.8,69,Degradation of BCL2 in 293T cells after 16 h treatment,
3219,BCL2,,10.1038/s41467-021-27210-x,,38,,
3219,BCL-xL,,10.1038/s41467-021-27210-x,,38,,
3220,BCL-xL,,10.1038/s41467-021-27210-x,,,,
3220,BCL2,,10.1038/s41467-021-27210-x,,,,
3221,BCL2,,10.1038/s41467-021-27210-x,48,,Degradation of BCL2 in 293T cells after 16 h treatment,
3221,BCL-xL,,10.1038/s41467-021-27210-x,6,,Degradation of BCL-xL in 293T cells after 16 h treatment,
3222,HDAC1,,10.3390/molecules26237241,,,,
3222,HDAC6,,10.3390/molecules26237241,,,,
3222,HDAC3,,10.3390/molecules26237241,,,,
3223,HDAC1,,10.3390/molecules26237241,,,,
3223,HDAC6,,10.3390/molecules26237241,,,,
3223,HDAC3,,10.3390/molecules26237241,,,,
3224,HDAC1,,10.3390/molecules26237241,,,,
3224,HDAC6,,10.3390/molecules26237241,,,,
3224,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC6,,10.3390/molecules26237241,,,,
3225,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC3,,10.3390/molecules26237241,,,,
3226,HDAC6,,10.3390/molecules26237241,,,,
3227,HDAC1,,10.3390/molecules26237241,,,,
3227,HDAC3,,10.3390/molecules26237241,,,,
3227,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC1,,10.3390/molecules26237241,,,,
3228,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC1,,10.3390/molecules26237241,,,,
3229,HDAC6,,10.3390/molecules26237241,,,,
3230,HDAC3,,10.3390/molecules26237241,,,,
3230,HDAC1,,10.3390/molecules26237241,,,,
3230,HDAC6,,10.3390/molecules26237241,,,,
3231,HDAC3,,10.3390/molecules26237241,,,,
3231,HDAC1,,10.3390/molecules26237241,,,,
3231,HDAC6,,10.3390/molecules26237241,,,,
3232,HDAC3,,10.3390/molecules26237241,,,,
3232,HDAC1,,10.3390/molecules26237241,,,,
3232,HDAC6,,10.3390/molecules26237241,,,,
3233,HDAC3,,10.3390/molecules26237241,,,,
3233,HDAC1,,10.3390/molecules26237241,,,,
3233,HDAC6,,10.3390/molecules26237241,,,,
3234,HDAC3,,10.3390/molecules26237241,,,,
3234,HDAC1,,10.3390/molecules26237241,,,,
3234,HDAC6,,10.3390/molecules26237241,,,,
3235,HSF1,,10.3390/molecules27051655,,,,
3236,HSF1,,10.3390/molecules27051655,,,,
3217,BCL-xL,,10.1038/s41467-021-27210-x,12.8,96,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL-xL,,10.1038/s41467-021-27210-x,12.1,81,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL2,,10.1038/s41467-021-27210-x,354.8,69,Degradation of BCL2 in 293T cells after 16 h treatment,
3219,BCL2,,10.1038/s41467-021-27210-x,,38,,
3219,BCL-xL,,10.1038/s41467-021-27210-x,,38,,
3220,BCL-xL,,10.1038/s41467-021-27210-x,,,,
3220,BCL2,,10.1038/s41467-021-27210-x,,,,
3221,BCL2,,10.1038/s41467-021-27210-x,48,,Degradation of BCL2 in 293T cells after 16 h treatment,
3221,BCL-xL,,10.1038/s41467-021-27210-x,6,,Degradation of BCL-xL in 293T cells after 16 h treatment,
3222,HDAC1,,10.3390/molecules26237241,,,,
3222,HDAC6,,10.3390/molecules26237241,,,,
3222,HDAC3,,10.3390/molecules26237241,,,,
3223,HDAC1,,10.3390/molecules26237241,,,,
3223,HDAC6,,10.3390/molecules26237241,,,,
3223,HDAC3,,10.3390/molecules26237241,,,,
3224,HDAC1,,10.3390/molecules26237241,,,,
3224,HDAC6,,10.3390/molecules26237241,,,,
3224,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC6,,10.3390/molecules26237241,,,,
3225,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC3,,10.3390/molecules26237241,,,,
3226,HDAC6,,10.3390/molecules26237241,,,,
3227,HDAC1,,10.3390/molecules26237241,,,,
3227,HDAC3,,10.3390/molecules26237241,,,,
3227,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC1,,10.3390/molecules26237241,,,,
3228,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC1,,10.3390/molecules26237241,,,,
3229,HDAC6,,10.3390/molecules26237241,,,,
3230,HDAC3,,10.3390/molecules26237241,,,,
3230,HDAC1,,10.3390/molecules26237241,,,,
3230,HDAC6,,10.3390/molecules26237241,,,,
3231,HDAC3,,10.3390/molecules26237241,,,,
3231,HDAC1,,10.3390/molecules26237241,,,,
3231,HDAC6,,10.3390/molecules26237241,,,,
3232,HDAC3,,10.3390/molecules26237241,,,,
3232,HDAC1,,10.3390/molecules26237241,,,,
3232,HDAC6,,10.3390/molecules26237241,,,,
3233,HDAC3,,10.3390/molecules26237241,,,,
3233,HDAC1,,10.3390/molecules26237241,,,,
3233,HDAC6,,10.3390/molecules26237241,,,,
3234,HDAC3,,10.3390/molecules26237241,,,,
3234,HDAC1,,10.3390/molecules26237241,,,,
3234,HDAC6,,10.3390/molecules26237241,,,,
3235,HSF1,,10.3390/molecules27051655,,,,
3236,HSF1,,10.3390/molecules27051655,,,,
3217,BCL-xL,,10.1038/s41467-021-27210-x,12.8,96,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL-xL,,10.1038/s41467-021-27210-x,12.1,81,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL2,,10.1038/s41467-021-27210-x,354.8,69,Degradation of BCL2 in 293T cells after 16 h treatment,
3219,BCL2,,10.1038/s41467-021-27210-x,,38,,
3219,BCL-xL,,10.1038/s41467-021-27210-x,,38,,
3220,BCL-xL,,10.1038/s41467-021-27210-x,,,,
3220,BCL2,,10.1038/s41467-021-27210-x,,,,
3221,BCL2,,10.1038/s41467-021-27210-x,48,,Degradation of BCL2 in 293T cells after 16 h treatment,
3221,BCL-xL,,10.1038/s41467-021-27210-x,6,,Degradation of BCL-xL in 293T cells after 16 h treatment,
3222,HDAC1,,10.3390/molecules26237241,,,,
3222,HDAC6,,10.3390/molecules26237241,,,,
3222,HDAC3,,10.3390/molecules26237241,,,,
3223,HDAC1,,10.3390/molecules26237241,,,,
3223,HDAC6,,10.3390/molecules26237241,,,,
3223,HDAC3,,10.3390/molecules26237241,,,,
3224,HDAC1,,10.3390/molecules26237241,,,,
3224,HDAC6,,10.3390/molecules26237241,,,,
3224,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC6,,10.3390/molecules26237241,,,,
3225,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC3,,10.3390/molecules26237241,,,,
3226,HDAC6,,10.3390/molecules26237241,,,,
3227,HDAC1,,10.3390/molecules26237241,,,,
3227,HDAC3,,10.3390/molecules26237241,,,,
3227,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC1,,10.3390/molecules26237241,,,,
3228,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC1,,10.3390/molecules26237241,,,,
3229,HDAC6,,10.3390/molecules26237241,,,,
3230,HDAC3,,10.3390/molecules26237241,,,,
3230,HDAC1,,10.3390/molecules26237241,,,,
3230,HDAC6,,10.3390/molecules26237241,,,,
3231,HDAC3,,10.3390/molecules26237241,,,,
3231,HDAC1,,10.3390/molecules26237241,,,,
3231,HDAC6,,10.3390/molecules26237241,,,,
3232,HDAC3,,10.3390/molecules26237241,,,,
3232,HDAC1,,10.3390/molecules26237241,,,,
3232,HDAC6,,10.3390/molecules26237241,,,,
3233,HDAC3,,10.3390/molecules26237241,,,,
3233,HDAC1,,10.3390/molecules26237241,,,,
3233,HDAC6,,10.3390/molecules26237241,,,,
3234,HDAC3,,10.3390/molecules26237241,,,,
3234,HDAC1,,10.3390/molecules26237241,,,,
3234,HDAC6,,10.3390/molecules26237241,,,,
3235,HSF1,,10.3390/molecules27051655,,,,
3236,HSF1,,10.3390/molecules27051655,,,,
3217,BCL-xL,,10.1038/s41467-021-27210-x,12.8,96,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL-xL,,10.1038/s41467-021-27210-x,12.1,81,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL2,,10.1038/s41467-021-27210-x,354.8,69,Degradation of BCL2 in 293T cells after 16 h treatment,
3219,BCL2,,10.1038/s41467-021-27210-x,,38,,
3219,BCL-xL,,10.1038/s41467-021-27210-x,,38,,
3220,BCL-xL,,10.1038/s41467-021-27210-x,,,,
3220,BCL2,,10.1038/s41467-021-27210-x,,,,
3221,BCL2,,10.1038/s41467-021-27210-x,48,,Degradation of BCL2 in 293T cells after 16 h treatment,
3221,BCL-xL,,10.1038/s41467-021-27210-x,6,,Degradation of BCL-xL in 293T cells after 16 h treatment,
3222,HDAC1,,10.3390/molecules26237241,,,,
3222,HDAC6,,10.3390/molecules26237241,,,,
3222,HDAC3,,10.3390/molecules26237241,,,,
3223,HDAC1,,10.3390/molecules26237241,,,,
3223,HDAC6,,10.3390/molecules26237241,,,,
3223,HDAC3,,10.3390/molecules26237241,,,,
3224,HDAC1,,10.3390/molecules26237241,,,,
3224,HDAC6,,10.3390/molecules26237241,,,,
3224,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC6,,10.3390/molecules26237241,,,,
3225,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC3,,10.3390/molecules26237241,,,,
3226,HDAC6,,10.3390/molecules26237241,,,,
3227,HDAC1,,10.3390/molecules26237241,,,,
3227,HDAC3,,10.3390/molecules26237241,,,,
3227,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC1,,10.3390/molecules26237241,,,,
3228,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC1,,10.3390/molecules26237241,,,,
3229,HDAC6,,10.3390/molecules26237241,,,,
3230,HDAC3,,10.3390/molecules26237241,,,,
3230,HDAC1,,10.3390/molecules26237241,,,,
3230,HDAC6,,10.3390/molecules26237241,,,,
3231,HDAC3,,10.3390/molecules26237241,,,,
3231,HDAC1,,10.3390/molecules26237241,,,,
3231,HDAC6,,10.3390/molecules26237241,,,,
3232,HDAC3,,10.3390/molecules26237241,,,,
3232,HDAC1,,10.3390/molecules26237241,,,,
3232,HDAC6,,10.3390/molecules26237241,,,,
3233,HDAC3,,10.3390/molecules26237241,,,,
3233,HDAC1,,10.3390/molecules26237241,,,,
3233,HDAC6,,10.3390/molecules26237241,,,,
3234,HDAC3,,10.3390/molecules26237241,,,,
3234,HDAC1,,10.3390/molecules26237241,,,,
3234,HDAC6,,10.3390/molecules26237241,,,,
3235,HSF1,,10.3390/molecules27051655,,,,
3236,HSF1,,10.3390/molecules27051655,,,,
3217,BCL-xL,,10.1038/s41467-021-27210-x,12.8,96,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL-xL,,10.1038/s41467-021-27210-x,12.1,81,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL2,,10.1038/s41467-021-27210-x,354.8,69,Degradation of BCL2 in 293T cells after 16 h treatment,
3219,BCL2,,10.1038/s41467-021-27210-x,,38,,
3219,BCL-xL,,10.1038/s41467-021-27210-x,,38,,
3220,BCL-xL,,10.1038/s41467-021-27210-x,,,,
3220,BCL2,,10.1038/s41467-021-27210-x,,,,
3221,BCL2,,10.1038/s41467-021-27210-x,48,,Degradation of BCL2 in 293T cells after 16 h treatment,
3221,BCL-xL,,10.1038/s41467-021-27210-x,6,,Degradation of BCL-xL in 293T cells after 16 h treatment,
3222,HDAC1,,10.3390/molecules26237241,,,,
3222,HDAC6,,10.3390/molecules26237241,,,,
3222,HDAC3,,10.3390/molecules26237241,,,,
3223,HDAC1,,10.3390/molecules26237241,,,,
3223,HDAC6,,10.3390/molecules26237241,,,,
3223,HDAC3,,10.3390/molecules26237241,,,,
3224,HDAC1,,10.3390/molecules26237241,,,,
3224,HDAC6,,10.3390/molecules26237241,,,,
3224,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC6,,10.3390/molecules26237241,,,,
3225,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC3,,10.3390/molecules26237241,,,,
3226,HDAC6,,10.3390/molecules26237241,,,,
3227,HDAC1,,10.3390/molecules26237241,,,,
3227,HDAC3,,10.3390/molecules26237241,,,,
3227,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC1,,10.3390/molecules26237241,,,,
3228,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC1,,10.3390/molecules26237241,,,,
3229,HDAC6,,10.3390/molecules26237241,,,,
3230,HDAC3,,10.3390/molecules26237241,,,,
3230,HDAC1,,10.3390/molecules26237241,,,,
3230,HDAC6,,10.3390/molecules26237241,,,,
3231,HDAC3,,10.3390/molecules26237241,,,,
3231,HDAC1,,10.3390/molecules26237241,,,,
3231,HDAC6,,10.3390/molecules26237241,,,,
3232,HDAC3,,10.3390/molecules26237241,,,,
3232,HDAC1,,10.3390/molecules26237241,,,,
3232,HDAC6,,10.3390/molecules26237241,,,,
3233,HDAC3,,10.3390/molecules26237241,,,,
3233,HDAC1,,10.3390/molecules26237241,,,,
3233,HDAC6,,10.3390/molecules26237241,,,,
3234,HDAC3,,10.3390/molecules26237241,,,,
3234,HDAC1,,10.3390/molecules26237241,,,,
3234,HDAC6,,10.3390/molecules26237241,,,,
3235,HSF1,,10.3390/molecules27051655,,,,
3236,HSF1,,10.3390/molecules27051655,,,,
3217,BCL-xL,,10.1038/s41467-021-27210-x,12.8,96,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL-xL,,10.1038/s41467-021-27210-x,12.1,81,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL2,,10.1038/s41467-021-27210-x,354.8,69,Degradation of BCL2 in 293T cells after 16 h treatment,
3219,BCL2,,10.1038/s41467-021-27210-x,,38,,
3219,BCL-xL,,10.1038/s41467-021-27210-x,,38,,
3220,BCL-xL,,10.1038/s41467-021-27210-x,,,,
3220,BCL2,,10.1038/s41467-021-27210-x,,,,
3221,BCL2,,10.1038/s41467-021-27210-x,48,,Degradation of BCL2 in 293T cells after 16 h treatment,
3221,BCL-xL,,10.1038/s41467-021-27210-x,6,,Degradation of BCL-xL in 293T cells after 16 h treatment,
3222,HDAC1,,10.3390/molecules26237241,,,,
3222,HDAC6,,10.3390/molecules26237241,,,,
3222,HDAC3,,10.3390/molecules26237241,,,,
3223,HDAC1,,10.3390/molecules26237241,,,,
3223,HDAC6,,10.3390/molecules26237241,,,,
3223,HDAC3,,10.3390/molecules26237241,,,,
3224,HDAC1,,10.3390/molecules26237241,,,,
3224,HDAC6,,10.3390/molecules26237241,,,,
3224,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC6,,10.3390/molecules26237241,,,,
3225,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC3,,10.3390/molecules26237241,,,,
3226,HDAC6,,10.3390/molecules26237241,,,,
3227,HDAC1,,10.3390/molecules26237241,,,,
3227,HDAC3,,10.3390/molecules26237241,,,,
3227,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC1,,10.3390/molecules26237241,,,,
3228,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC1,,10.3390/molecules26237241,,,,
3229,HDAC6,,10.3390/molecules26237241,,,,
3230,HDAC3,,10.3390/molecules26237241,,,,
3230,HDAC1,,10.3390/molecules26237241,,,,
3230,HDAC6,,10.3390/molecules26237241,,,,
3231,HDAC3,,10.3390/molecules26237241,,,,
3231,HDAC1,,10.3390/molecules26237241,,,,
3231,HDAC6,,10.3390/molecules26237241,,,,
3232,HDAC3,,10.3390/molecules26237241,,,,
3232,HDAC1,,10.3390/molecules26237241,,,,
3232,HDAC6,,10.3390/molecules26237241,,,,
3233,HDAC3,,10.3390/molecules26237241,,,,
3233,HDAC1,,10.3390/molecules26237241,,,,
3233,HDAC6,,10.3390/molecules26237241,,,,
3234,HDAC3,,10.3390/molecules26237241,,,,
3234,HDAC1,,10.3390/molecules26237241,,,,
3234,HDAC6,,10.3390/molecules26237241,,,,
3235,HSF1,,10.3390/molecules27051655,,,,
3236,HSF1,,10.3390/molecules27051655,,,,
3217,BCL-xL,,10.1038/s41467-021-27210-x,12.8,96,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL-xL,,10.1038/s41467-021-27210-x,12.1,81,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL2,,10.1038/s41467-021-27210-x,354.8,69,Degradation of BCL2 in 293T cells after 16 h treatment,
3219,BCL2,,10.1038/s41467-021-27210-x,,38,,
3219,BCL-xL,,10.1038/s41467-021-27210-x,,38,,
3220,BCL-xL,,10.1038/s41467-021-27210-x,,,,
3220,BCL2,,10.1038/s41467-021-27210-x,,,,
3221,BCL2,,10.1038/s41467-021-27210-x,48,,Degradation of BCL2 in 293T cells after 16 h treatment,
3221,BCL-xL,,10.1038/s41467-021-27210-x,6,,Degradation of BCL-xL in 293T cells after 16 h treatment,
3222,HDAC1,,10.3390/molecules26237241,,,,
3222,HDAC6,,10.3390/molecules26237241,,,,
3222,HDAC3,,10.3390/molecules26237241,,,,
3223,HDAC1,,10.3390/molecules26237241,,,,
3223,HDAC6,,10.3390/molecules26237241,,,,
3223,HDAC3,,10.3390/molecules26237241,,,,
3224,HDAC1,,10.3390/molecules26237241,,,,
3224,HDAC6,,10.3390/molecules26237241,,,,
3224,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC6,,10.3390/molecules26237241,,,,
3225,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC3,,10.3390/molecules26237241,,,,
3226,HDAC6,,10.3390/molecules26237241,,,,
3227,HDAC1,,10.3390/molecules26237241,,,,
3227,HDAC3,,10.3390/molecules26237241,,,,
3227,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC1,,10.3390/molecules26237241,,,,
3228,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC1,,10.3390/molecules26237241,,,,
3229,HDAC6,,10.3390/molecules26237241,,,,
3230,HDAC3,,10.3390/molecules26237241,,,,
3230,HDAC1,,10.3390/molecules26237241,,,,
3230,HDAC6,,10.3390/molecules26237241,,,,
3231,HDAC3,,10.3390/molecules26237241,,,,
3231,HDAC1,,10.3390/molecules26237241,,,,
3231,HDAC6,,10.3390/molecules26237241,,,,
3232,HDAC3,,10.3390/molecules26237241,,,,
3232,HDAC1,,10.3390/molecules26237241,,,,
3232,HDAC6,,10.3390/molecules26237241,,,,
3233,HDAC3,,10.3390/molecules26237241,,,,
3233,HDAC1,,10.3390/molecules26237241,,,,
3233,HDAC6,,10.3390/molecules26237241,,,,
3234,HDAC3,,10.3390/molecules26237241,,,,
3234,HDAC1,,10.3390/molecules26237241,,,,
3234,HDAC6,,10.3390/molecules26237241,,,,
3235,HSF1,,10.3390/molecules27051655,,,,
3236,HSF1,,10.3390/molecules27051655,,,,
3217,BCL-xL,,10.1038/s41467-021-27210-x,12.8,96,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL-xL,,10.1038/s41467-021-27210-x,12.1,81,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL2,,10.1038/s41467-021-27210-x,354.8,69,Degradation of BCL2 in 293T cells after 16 h treatment,
3219,BCL2,,10.1038/s41467-021-27210-x,,38,,
3219,BCL-xL,,10.1038/s41467-021-27210-x,,38,,
3220,BCL-xL,,10.1038/s41467-021-27210-x,,,,
3220,BCL2,,10.1038/s41467-021-27210-x,,,,
3221,BCL2,,10.1038/s41467-021-27210-x,48,,Degradation of BCL2 in 293T cells after 16 h treatment,
3221,BCL-xL,,10.1038/s41467-021-27210-x,6,,Degradation of BCL-xL in 293T cells after 16 h treatment,
3222,HDAC1,,10.3390/molecules26237241,,,,
3222,HDAC6,,10.3390/molecules26237241,,,,
3222,HDAC3,,10.3390/molecules26237241,,,,
3223,HDAC1,,10.3390/molecules26237241,,,,
3223,HDAC6,,10.3390/molecules26237241,,,,
3223,HDAC3,,10.3390/molecules26237241,,,,
3224,HDAC1,,10.3390/molecules26237241,,,,
3224,HDAC6,,10.3390/molecules26237241,,,,
3224,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC6,,10.3390/molecules26237241,,,,
3225,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC3,,10.3390/molecules26237241,,,,
3226,HDAC6,,10.3390/molecules26237241,,,,
3227,HDAC1,,10.3390/molecules26237241,,,,
3227,HDAC3,,10.3390/molecules26237241,,,,
3227,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC1,,10.3390/molecules26237241,,,,
3228,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC1,,10.3390/molecules26237241,,,,
3229,HDAC6,,10.3390/molecules26237241,,,,
3230,HDAC3,,10.3390/molecules26237241,,,,
3230,HDAC1,,10.3390/molecules26237241,,,,
3230,HDAC6,,10.3390/molecules26237241,,,,
3231,HDAC3,,10.3390/molecules26237241,,,,
3231,HDAC1,,10.3390/molecules26237241,,,,
3231,HDAC6,,10.3390/molecules26237241,,,,
3232,HDAC3,,10.3390/molecules26237241,,,,
3232,HDAC1,,10.3390/molecules26237241,,,,
3232,HDAC6,,10.3390/molecules26237241,,,,
3233,HDAC3,,10.3390/molecules26237241,,,,
3233,HDAC1,,10.3390/molecules26237241,,,,
3233,HDAC6,,10.3390/molecules26237241,,,,
3234,HDAC3,,10.3390/molecules26237241,,,,
3234,HDAC1,,10.3390/molecules26237241,,,,
3234,HDAC6,,10.3390/molecules26237241,,,,
3235,HSF1,,10.3390/molecules27051655,,,,
3236,HSF1,,10.3390/molecules27051655,,,,
3217,BCL-xL,,10.1038/s41467-021-27210-x,12.8,96,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL-xL,,10.1038/s41467-021-27210-x,12.1,81,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL2,,10.1038/s41467-021-27210-x,354.8,69,Degradation of BCL2 in 293T cells after 16 h treatment,
3219,BCL2,,10.1038/s41467-021-27210-x,,38,,
3219,BCL-xL,,10.1038/s41467-021-27210-x,,38,,
3220,BCL-xL,,10.1038/s41467-021-27210-x,,,,
3220,BCL2,,10.1038/s41467-021-27210-x,,,,
3221,BCL2,,10.1038/s41467-021-27210-x,48,,Degradation of BCL2 in 293T cells after 16 h treatment,
3221,BCL-xL,,10.1038/s41467-021-27210-x,6,,Degradation of BCL-xL in 293T cells after 16 h treatment,
3222,HDAC1,,10.3390/molecules26237241,,,,
3222,HDAC6,,10.3390/molecules26237241,,,,
3222,HDAC3,,10.3390/molecules26237241,,,,
3223,HDAC1,,10.3390/molecules26237241,,,,
3223,HDAC6,,10.3390/molecules26237241,,,,
3223,HDAC3,,10.3390/molecules26237241,,,,
3224,HDAC1,,10.3390/molecules26237241,,,,
3224,HDAC6,,10.3390/molecules26237241,,,,
3224,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC6,,10.3390/molecules26237241,,,,
3225,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC3,,10.3390/molecules26237241,,,,
3226,HDAC6,,10.3390/molecules26237241,,,,
3227,HDAC1,,10.3390/molecules26237241,,,,
3227,HDAC3,,10.3390/molecules26237241,,,,
3227,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC1,,10.3390/molecules26237241,,,,
3228,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC1,,10.3390/molecules26237241,,,,
3229,HDAC6,,10.3390/molecules26237241,,,,
3230,HDAC3,,10.3390/molecules26237241,,,,
3230,HDAC1,,10.3390/molecules26237241,,,,
3230,HDAC6,,10.3390/molecules26237241,,,,
3231,HDAC3,,10.3390/molecules26237241,,,,
3231,HDAC1,,10.3390/molecules26237241,,,,
3231,HDAC6,,10.3390/molecules26237241,,,,
3232,HDAC3,,10.3390/molecules26237241,,,,
3232,HDAC1,,10.3390/molecules26237241,,,,
3232,HDAC6,,10.3390/molecules26237241,,,,
3233,HDAC3,,10.3390/molecules26237241,,,,
3233,HDAC1,,10.3390/molecules26237241,,,,
3233,HDAC6,,10.3390/molecules26237241,,,,
3234,HDAC3,,10.3390/molecules26237241,,,,
3234,HDAC1,,10.3390/molecules26237241,,,,
3234,HDAC6,,10.3390/molecules26237241,,,,
3235,HSF1,,10.3390/molecules27051655,,,,
3236,HSF1,,10.3390/molecules27051655,,,,
3217,BCL-xL,,10.1038/s41467-021-27210-x,12.8,96,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL-xL,,10.1038/s41467-021-27210-x,12.1,81,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL2,,10.1038/s41467-021-27210-x,354.8,69,Degradation of BCL2 in 293T cells after 16 h treatment,
3219,BCL2,,10.1038/s41467-021-27210-x,,38,,
3219,BCL-xL,,10.1038/s41467-021-27210-x,,38,,
3220,BCL-xL,,10.1038/s41467-021-27210-x,,,,
3220,BCL2,,10.1038/s41467-021-27210-x,,,,
3221,BCL2,,10.1038/s41467-021-27210-x,48,,Degradation of BCL2 in 293T cells after 16 h treatment,
3221,BCL-xL,,10.1038/s41467-021-27210-x,6,,Degradation of BCL-xL in 293T cells after 16 h treatment,
3222,HDAC1,,10.3390/molecules26237241,,,,
3222,HDAC6,,10.3390/molecules26237241,,,,
3222,HDAC3,,10.3390/molecules26237241,,,,
3223,HDAC1,,10.3390/molecules26237241,,,,
3223,HDAC6,,10.3390/molecules26237241,,,,
3223,HDAC3,,10.3390/molecules26237241,,,,
3224,HDAC1,,10.3390/molecules26237241,,,,
3224,HDAC6,,10.3390/molecules26237241,,,,
3224,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC6,,10.3390/molecules26237241,,,,
3225,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC3,,10.3390/molecules26237241,,,,
3226,HDAC6,,10.3390/molecules26237241,,,,
3227,HDAC1,,10.3390/molecules26237241,,,,
3227,HDAC3,,10.3390/molecules26237241,,,,
3227,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC1,,10.3390/molecules26237241,,,,
3228,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC1,,10.3390/molecules26237241,,,,
3229,HDAC6,,10.3390/molecules26237241,,,,
3230,HDAC3,,10.3390/molecules26237241,,,,
3230,HDAC1,,10.3390/molecules26237241,,,,
3230,HDAC6,,10.3390/molecules26237241,,,,
3231,HDAC3,,10.3390/molecules26237241,,,,
3231,HDAC1,,10.3390/molecules26237241,,,,
3231,HDAC6,,10.3390/molecules26237241,,,,
3232,HDAC3,,10.3390/molecules26237241,,,,
3232,HDAC1,,10.3390/molecules26237241,,,,
3232,HDAC6,,10.3390/molecules26237241,,,,
3233,HDAC3,,10.3390/molecules26237241,,,,
3233,HDAC1,,10.3390/molecules26237241,,,,
3233,HDAC6,,10.3390/molecules26237241,,,,
3234,HDAC3,,10.3390/molecules26237241,,,,
3234,HDAC1,,10.3390/molecules26237241,,,,
3234,HDAC6,,10.3390/molecules26237241,,,,
3235,HSF1,,10.3390/molecules27051655,,,,
3236,HSF1,,10.3390/molecules27051655,,,,
3217,BCL-xL,,10.1038/s41467-021-27210-x,12.8,96,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL-xL,,10.1038/s41467-021-27210-x,12.1,81,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL2,,10.1038/s41467-021-27210-x,354.8,69,Degradation of BCL2 in 293T cells after 16 h treatment,
3219,BCL2,,10.1038/s41467-021-27210-x,,38,,
3219,BCL-xL,,10.1038/s41467-021-27210-x,,38,,
3220,BCL-xL,,10.1038/s41467-021-27210-x,,,,
3220,BCL2,,10.1038/s41467-021-27210-x,,,,
3221,BCL2,,10.1038/s41467-021-27210-x,48,,Degradation of BCL2 in 293T cells after 16 h treatment,
3221,BCL-xL,,10.1038/s41467-021-27210-x,6,,Degradation of BCL-xL in 293T cells after 16 h treatment,
3222,HDAC1,,10.3390/molecules26237241,,,,
3222,HDAC6,,10.3390/molecules26237241,,,,
3222,HDAC3,,10.3390/molecules26237241,,,,
3223,HDAC1,,10.3390/molecules26237241,,,,
3223,HDAC6,,10.3390/molecules26237241,,,,
3223,HDAC3,,10.3390/molecules26237241,,,,
3224,HDAC1,,10.3390/molecules26237241,,,,
3224,HDAC6,,10.3390/molecules26237241,,,,
3224,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC6,,10.3390/molecules26237241,,,,
3225,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC3,,10.3390/molecules26237241,,,,
3226,HDAC6,,10.3390/molecules26237241,,,,
3227,HDAC1,,10.3390/molecules26237241,,,,
3227,HDAC3,,10.3390/molecules26237241,,,,
3227,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC1,,10.3390/molecules26237241,,,,
3228,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC1,,10.3390/molecules26237241,,,,
3229,HDAC6,,10.3390/molecules26237241,,,,
3230,HDAC3,,10.3390/molecules26237241,,,,
3230,HDAC1,,10.3390/molecules26237241,,,,
3230,HDAC6,,10.3390/molecules26237241,,,,
3231,HDAC3,,10.3390/molecules26237241,,,,
3231,HDAC1,,10.3390/molecules26237241,,,,
3231,HDAC6,,10.3390/molecules26237241,,,,
3232,HDAC3,,10.3390/molecules26237241,,,,
3232,HDAC1,,10.3390/molecules26237241,,,,
3232,HDAC6,,10.3390/molecules26237241,,,,
3233,HDAC3,,10.3390/molecules26237241,,,,
3233,HDAC1,,10.3390/molecules26237241,,,,
3233,HDAC6,,10.3390/molecules26237241,,,,
3234,HDAC3,,10.3390/molecules26237241,,,,
3234,HDAC1,,10.3390/molecules26237241,,,,
3234,HDAC6,,10.3390/molecules26237241,,,,
3235,HSF1,,10.3390/molecules27051655,,,,
3236,HSF1,,10.3390/molecules27051655,,,,
3217,BCL-xL,,10.1038/s41467-021-27210-x,12.8,96,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL-xL,,10.1038/s41467-021-27210-x,12.1,81,Degradation of BCL-xL in 293T cells after 16 h treatment,
3218,BCL2,,10.1038/s41467-021-27210-x,354.8,69,Degradation of BCL2 in 293T cells after 16 h treatment,
3219,BCL2,,10.1038/s41467-021-27210-x,,38,,
3219,BCL-xL,,10.1038/s41467-021-27210-x,,38,,
3220,BCL-xL,,10.1038/s41467-021-27210-x,,,,
3220,BCL2,,10.1038/s41467-021-27210-x,,,,
3221,BCL2,,10.1038/s41467-021-27210-x,48,,Degradation of BCL2 in 293T cells after 16 h treatment,
3221,BCL-xL,,10.1038/s41467-021-27210-x,6,,Degradation of BCL-xL in 293T cells after 16 h treatment,
3222,HDAC1,,10.3390/molecules26237241,,,,
3222,HDAC6,,10.3390/molecules26237241,,,,
3222,HDAC3,,10.3390/molecules26237241,,,,
3223,HDAC1,,10.3390/molecules26237241,,,,
3223,HDAC6,,10.3390/molecules26237241,,,,
3223,HDAC3,,10.3390/molecules26237241,,,,
3224,HDAC1,,10.3390/molecules26237241,,,,
3224,HDAC6,,10.3390/molecules26237241,,,,
3224,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC6,,10.3390/molecules26237241,,,,
3225,HDAC3,,10.3390/molecules26237241,,,,
3225,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC1,,10.3390/molecules26237241,,,,
3226,HDAC3,,10.3390/molecules26237241,,,,
3226,HDAC6,,10.3390/molecules26237241,,,,
3227,HDAC1,,10.3390/molecules26237241,,,,
3227,HDAC3,,10.3390/molecules26237241,,,,
3227,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC6,,10.3390/molecules26237241,,,,
3228,HDAC1,,10.3390/molecules26237241,,,,
3228,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC3,,10.3390/molecules26237241,,,,
3229,HDAC1,,10.3390/molecules26237241,,,,
3229,HDAC6,,10.3390/molecules26237241,,,,
3230,HDAC3,,10.3390/molecules26237241,,,,
3230,HDAC1,,10.3390/molecules26237241,,,,
3230,HDAC6,,10.3390/molecules26237241,,,,
3231,HDAC3,,10.3390/molecules26237241,,,,
3231,HDAC1,,10.3390/molecules26237241,,,,
3231,HDAC6,,10.3390/molecules26237241,,,,
3232,HDAC3,,10.3390/molecules26237241,,,,
3232,HDAC1,,10.3390/molecules26237241,,,,
3232,HDAC6,,10.3390/molecules26237241,,,,
3233,HDAC3,,10.3390/molecules26237241,,,,
3233,HDAC1,,10.3390/molecules26237241,,,,
3233,HDAC6,,10.3390/molecules26237241,,,,
3234,HDAC3,,10.3390/molecules26237241,,,,
3234,HDAC1,,10.3390/molecules26237241,,,,
3234,HDAC6,,10.3390/molecules26237241,,,,
3235,HSF1,,10.3390/molecules27051655,,,,
3236,HSF1,,10.3390/molecules27051655,,,,