活性代謝物
↑ “On the assessment of drug metabolism by assays of codeine and its main metabolites”. Therapeutic Drug Monitoring 22 (3): 258–65. (June 2000). doi:10.1097/00007691-200006000-00005. PMID 10850391.
↑ Raffa RB (July 1996). “A novel approach to the pharmacology of analgesics”. The American Journal of Medicine 101 (1A): 40S–46S. doi:10.1016/s0002-9343(96)00137-4. PMID 8764759.
1 2 “Substrates, inducers, inhibitors and structure-activity relationships of human Cytochrome P450 2C9 and implications in drug development”.
活性代謝物(かっせいたいしゃぶつ、Active metabolite)は、薬物が代謝作用を受けて生成する、生理活性を有する分子である。