TRPV1
リファレンス

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↑  “Irritant-evoked activation and calcium modulation of the TRPA1 receptor”. Nature 585 (7823):  141–145. (September 2020). Bibcode: 2020Natur.585..141Z. doi:10.1038/s41586-020-2480-9. PMC 7483980. PMID 32641835. https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7483980/.
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↑  “Low-cost functional plasticity of TRPV1 supports heat tolerance in squirrels and camels”. Proceedings of the National Academy of Sciences of the United States of America 113 (40):  11342–11347. (October 2016). Bibcode: 2016PNAS..11311342L. doi:10.1073/pnas.1604269113. PMC 5056056. PMID 27638213. https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5056056/.
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↑  “TRPV1 receptors in the CNS play a key role in broad-spectrum analgesia of TRPV1 antagonists”. The Journal of Neuroscience 26 (37):  9385–9393. (September 2006). doi:10.1523/JNEUROSCI.1246-06.2006. PMC 6674601. PMID 16971522. https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6674601/.
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↑  “Regulation of Ca2+-dependent desensitization in the vanilloid receptor TRPV1 by calcineurin and cAMP-dependent protein kinase”. The Journal of Biological Chemistry 280 (14):  13424–13432. (April 2005). doi:10.1074/jbc.M410917200. PMID 15691846.
1 2  “Functional Role of Transient Receptor Potential Channels in Immune Cells and Epithelia”. Frontiers in Immunology 9:  174. (2018). doi:10.3389/fimmu.2018.00174. PMC 5808302. PMID 29467763. https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5808302/.
1 2 3 4 5  “TRPV1 Channels in Immune Cells and Hematological Malignancies”. Ion Channels Down Under. Ion Channels DownUnder. 79. Academic Press. (2017-01-01). 173–198. doi:10.1016/bs.apha.2017.01.002. ISBN 9780128104132. PMID 28528668
1 2 3 4  “Inflammation, Cancer and Immunity-Implication of TRPV1 Channel”. Frontiers in Oncology 9:  1087. (2019-10-16). doi:10.3389/fonc.2019.01087. PMC 6805766. PMID 31681615. https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6805766/.
1 2 3  “Modulation of neuroinflammation: Role and therapeutic potential of TRPV1 in the neuro-immune axis”. Brain, Behavior, and Immunity 64:  354–366. (August 2017). doi:10.1016/j.bbi.2017.03.007. PMID 28342781.
↑  Boonen, Brett; Startek, Justyna B.; Talavera, Karel (2016-01-01). Chemical Activation of Sensory TRP Channels. Topics in Medicinal Chemistry. Springer Berlin Heidelberg. pp. 1–41.  doi:10.1007/7355_2015_98.
↑  “Capsaicin (TRPV1 Agonist) therapy for pain relief: farewell or revival?”. The Clinical Journal of Pain 24 (2):  142–154. (February 2008). doi:10.1097/AJP.0b013e318158ed9e. PMID 18209521.
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1 2  “Effects of cannabinoids and cannabinoid-enriched Cannabis extracts on TRP channels and endocannabinoid metabolic enzymes”. British Journal of Pharmacology 163 (7):  1479–1494. (August 2011). doi:10.1111/j.1476-5381.2010.01166.x. PMC 3165957. PMID 21175579. https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3165957/.
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↑  “A FAAH-regulated class of N-acyl taurines that activates TRP ion channels”. Biochemistry 45 (30):  9007–9015. (August 2006). doi:10.1021/bi0608008. PMID 16866345.
1 2 3 4 5 6 7  “Novel endogenous N-acyl amides activate TRPV1-4 receptors, BV-2 microglia, and are regulated in brain in an acute model of inflammation”. Frontiers in Cellular Neuroscience 8:  195. (2014-08-01). doi:10.3389/fncel.2014.00195. PMC 4118021. PMID 25136293. https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4118021/.
↑  “TRPV1 channels as a newly identified target for vitamin D”. Channels 15 (1):  360–374. (December 2021). doi:10.1080/19336950.2021.1905248. PMC 8032246. PMID 33825665. https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8032246/.
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1 2  “TRPV1 channels mediate long-term depression at synapses on hippocampal interneurons”. Neuron 57 (5):  746–759. (March 2008). doi:10.1016/j.neuron.2007.12.027. PMC 2698707. PMID 18341994. https://www.ncbi.nlm.nih.gov/pmc/articles/PMC2698707/.
↑  “Primary afferent activation of thermosensitive TRPV1 triggers asynchronous glutamate release at central neurons”. Neuron 65 (5):  657–669. (March 2010). doi:10.1016/j.neuron.2010.02.017. PMC 2837850. PMID 20223201. https://www.ncbi.nlm.nih.gov/pmc/articles/PMC2837850/.
↑  “Structural determinant of TRPV1 desensitization interacts with calmodulin”. Proceedings of the National Academy of Sciences of the United States of America 100 (13):  8002–8006. (June 2003). Bibcode: 2003PNAS..100.8002N. doi:10.1073/pnas.1337252100. PMC 164702. PMID 12808128. https://www.ncbi.nlm.nih.gov/pmc/articles/PMC164702/.
1 2  “Regulated exocytosis contributes to protein kinase C potentiation of vanilloid receptor activity”. The Journal of Biological Chemistry 279 (24):  25665–25672. (June 2004). doi:10.1074/jbc.M311515200. PMID 15066994.
1 2  “Cannabinoid-induced cell death in endometrial cancer cells: involvement of TRPV1 receptors in apoptosis”. Journal of Physiology and Biochemistry 74 (2):  261–272. (May 2018). doi:10.1007/s13105-018-0611-7. PMID 29441458.
1 2  “"TRPV1 is a component of the atrial natriuretic signaling complex, and using orally delivered antagonists, presents a valid therapeutic target in the longitudinal reversal and treatment of cardiac hypertrophy and heart failure"”. Channels 13 (1):  1–16. (December 2019). doi:10.1080/19336950.2018.1547611. PMC 6298697. PMID 30424709. https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6298697/.
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↑  “The capsaicin receptor: a heat-activated ion channel in the pain pathway”. Nature 389 (6653):  816–824. (October 1997). Bibcode: 1997Natur.389..816C. doi:10.1038/39807. PMID 9349813.