Patent Document ID: 20020065265
Application ID: 09951137
Patent Flag: 0

Claim One:
1. A compound represented by A: 51 X represents C(R 3 ) 2, O, S, SO, SO 2, NR 2, NC(O)R 1, NC(O)OR 2, NS(O) 2 R 1, or C&boxH;O; Z represents N or CR; m is 0, 1, 2, 3 or 4; n is 1 or 2; p is 1, 2, or 3; y is 0, 1, or 2; R represents H, alkyl, cycloalkyl, aryl, heteroaryl, aralkyl, or heteroaralkyl; R 1 represents NR 2, alkyl, cycloalkyl, aryl, heteroaryl, aralkyl, or heteroaralkyl; R and R 1 may be connected through a covalent bond; R 2 represents independently for each occurrence H, alkyl, fluoroalkyl, aryl, heteroaryl, or cycloalkyl; R 3 represents independently for each occurrence H, alkyl, aryl, OR 2, OC(O)R 2, CH 2 OR 2, or CO 2 R 2 ; wherein any two instances of R 3 may be connected by a covalent tether whose backbone consists of 1, 2, 3, or 4 carbon atoms; R 4 represents independently for each occurrence H, alkyl, aryl, heteroaryl, alkenyl, or cycloalkyl; R 5 and R 6 are selected independently for each occurrence from the group consisting of H, alkyl, (CH 2 ) p Y, aryl, heteroaryl, F, OR 2, and OC(O)R 2 ; or an instance of CR 5 R 6 taken together is C(O); R 8 and R 9 are selected independently for each occurrence from the group consisting of H, alkyl, (CH 2 ) p Y, aryl, heteroaryl, F, OR 2, and OC(O)R 2 ; or an instance of CR 8 R 9 taken together is C(O); Y represents independently for each occurrence OR 2, N(R 2 ) 2, SR 2, S(O)R 2, S(O) 2 R 2, or P(O)(OR 2 ) 2 ; any two instances of R 2 may be connected through a covalent bond; a covalent bond may connect R 4 and an instance of R 5 or R 6 ; any two instances of R 5 and R 6 may be connected through a covalent bond; any two geminal or vicinal instances of R 8 and R 9 may be connected through a covalent bond; and the stereochemical configuration at any stereocenter of a compound represented by A is R, S, or a mixture of these configurations.