1-苄基-1,2,3-三唑

1-苄基-1,2,3-三唑是一种有机化合物，化学式为C9H9N3，它是1H-1,2,3-三唑的氮上的氢被苄基取代的产物。它可由1,2,3-三唑和溴化苄反应制得，Jérémie Doiron; et al. Synthesis and structure–activity relationship of 1- and 2-substituted-1,2,3-triazole letrozole-based analogues as aromatase inhibitors. European Journal of Medicinal Chemistry, 2011. 46 (9): 4010-4024. .或由叠氮化苄和乙炔在碘化亚铜和三乙胺存在下反应得到。Wu L, Yan B, Yang G, et al. Green synthesis of 1-monosubstituted 1,2,3-triazoles via ‘click chemistry’ in water. Heterocyclic Communications, 2013, 19 (6): 397-400. 它和碘甲烷在乙腈中反应，可以得到1-苄基-3-甲基三唑𬭩碘化物。M.C. Casanova; Y. Zhao; S. Hutter; et al. N,N′-bridged heterocyclic bis-iminium salts as potent antimalarial agents against multi-resistant Plasmodium falciparum. European Journal of Medicinal Chemistry, 2025. 292. 117633. . Supp. Info., pp. 5.

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Category:三唑