3-Hydroxyphenazepam

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3-Hydroxyphenazepam bụ benzodiazepine nwere ikike hypnotic, sedative, anxiolytic, na anticonvulsant. Ọ bụ metabolite na-arụ ọrụ nke phenazepam, yana metabolite na'arụ ọrụ nke benzodiazepine prodrug cinazepam. N'ihe gbasara phenazepam, 3-hydroxyphenazepam belatara ihe onwunwe myorelaxant, mana ọ fọrọ nke nta ka ọ bụrụ ihe ha nhata n'ọtụtụ ihe ndị ọzọ. Dị ka benzodiazepines ndị ọzọ, 3-hydroxyphenazepam na-akpa ndị mmadụ n'ihe ndị mere n'oge gara maka nsogbụ ndị na eme àgwà dị ka modulator allosteric dị mma nke ebe benzodiazepine nke onye na-anabata GABAA na uru EC50 nke 10.3 nM. A na-ere ya n'ịntanetị dị ka ọgwụ mmepụta.

 Hụkwa 

 Lorazepam, ọgwụ nwere ikike
 Nifoxipam
 Nitemazepam

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