A process for preparing a compound of Formula (V): comprising the steps of: (a) reacting a compound of Formula (I) and a compound of Formula (II): to provide a compound of Formula (III): and (b) converting said compound of Formula (III) to said compound of Formula (V) by steps (b1), (b2), and (b3), in any order: (b1) forming an indole group by reaction with a compound of Formula (IVa) or a compound of Formula (IVb): (b2) converting said -NR 4 R 5 group to -NH 2 ; and (b3) converting said -OR 3 group to -NH 2 ; wherein: X 1 is halo, -NO 2 , -OS(O) 2 R, or -N 2 + ; X 2 is Cl, Br, I, -OH, -OS(O) 2 R, acyloxy, or trialkylsiloxy; R 1 and R 2 are independently selected from H, benzyl, substituted benzyl, 4-methoxyphenyl, acyl, -S(O) 2 Ar, tert -butoxycarbonyl, or benzyloxycarbonyl; R 3 is H, C 1-8 alkyl, aryl, or heteroaryl; R 4 and R 5 are independently selected from H, benzyl, 4-methoxybenzyl, 4-methoxyphenyl, acyl, -SO) 2 R, tert -butoxycarbonyl, or benzyloxycarbonyl; R 8 is H, C 1-3 alkyl, or aryl; and each R is independently C 1-3 alkyl or aryl. (a) reacting a compound of Formula (I) and a compound of Formula (II): to provide a compound of Formula (III): and (b) converting said compound of Formula (III) to said compound of Formula (V) by steps (b1), (b2), and (b3), in any order: (b1) forming an indole group by reaction with a compound of Formula (IVa) or a compound of Formula (IVb): (b2) converting said -NR 4 R 5 group to -NH 2 ; and (b3) converting said -OR 3 group to -NH 2 ; wherein: X 1 is halo, -NO 2 , -OS(O) 2 R, or -N 2 + ; X 2 is Cl, Br, I, -OH, -OS(O) 2 R, acyloxy, or trialkylsiloxy; R 1 and R 2 are independently selected from H, benzyl, substituted benzyl, 4-methoxyphenyl, acyl, -S(O) 2 Ar, tert -butoxycarbonyl, or benzyloxycarbonyl; R 3 is H, C 1-8 alkyl, aryl, or heteroaryl; R 4 and R 5 are independently selected from H, benzyl, 4-methoxybenzyl, 4-methoxyphenyl, acyl, -SO) 2 R, tert -butoxycarbonyl, or benzyloxycarbonyl; R 8 is H, C 1-3 alkyl, or aryl; and each R is independently C 1-3 alkyl or aryl. (b1) forming an indole group by reaction with a compound of Formula (IVa) or a compound of Formula (IVb): (b2) converting said -NR 4 R 5 group to -NH 2 ; and (b3) converting said -OR 3 group to -NH 2 ; wherein: X 1 is halo, -NO 2 , -OS(O) 2 R, or -N 2 + ; X 2 is Cl, Br, I, -OH, -OS(O) 2 R, acyloxy, or trialkylsiloxy; R 1 and R 2 are independently selected from H, benzyl, substituted benzyl, 4-methoxyphenyl, acyl, -S(O) 2 Ar, tert -butoxycarbonyl, or benzyloxycarbonyl; R 3 is H, C 1-8 alkyl, aryl, or heteroaryl; R 4 and R 5 are independently selected from H, benzyl, 4-methoxybenzyl, 4-methoxyphenyl, acyl, -SO) 2 R, tert -butoxycarbonyl, or benzyloxycarbonyl; R 8 is H, C 1-3 alkyl, or aryl; and each R is independently C 1-3 alkyl or aryl. X 1 is halo, -NO 2 , -OS(O) 2 R, or -N 2 + ; X 2 is Cl, Br, I, -OH, -OS(O) 2 R, acyloxy, or trialkylsiloxy; R 1 and R 2 are independently selected from H, benzyl, substituted benzyl, 4-methoxyphenyl, acyl, -S(O) 2 Ar, tert -butoxycarbonyl, or benzyloxycarbonyl; R 3 is H, C 1-8 alkyl, aryl, or heteroaryl; R 4 and R 5 are independently selected from H, benzyl, 4-methoxybenzyl, 4-methoxyphenyl, acyl, -SO) 2 R, tert -butoxycarbonyl, or benzyloxycarbonyl; R 8 is H, C 1-3 alkyl, or aryl; and each R is independently C 1-3 alkyl or aryl. <EOS>