mhurhangee/ep-ind-claims huggingface dataset:
Process for the preparation of a compound of general formula or a salt thereof, said process comprising: a) reacting an indanone of general formula with a compound of general formula, so as to provide a compound of general formula; b) converting said compound of general formula into a compound of general formula; wherein: - R 1 is selected from the group consisting of -CN and 1,2,4-oxadiazole, said 1,2,4-oxadiazole being attached to the bicycle via carbon 3 and optionally substituted in position 5 with a 3'-cyano-4'-isopropoxyphenyl group; - one of the dashed lines indicates a single bond and the other one a double bond, and when the dashed line linked to R 2 is a double bond R 2 is N, and when the dashed line linked to R 2 is a single bond R 2 is NH; - R 10 is selected from the group consisting of -CH 2 OH, -CH 2 OPg and -CO 2 R 12; - R 12 is selected from the group consisting of H, a linear or branched C1-C8 alkyl or a linear or branched C1-C8 alkyl substituted with a C6-C10 aryl; - Pg is an oxygen protecting group; and - the * indicates a stereogenic center; said process being characterized in that step a) is carried out in the absence of titanium alkoxides. a) reacting an indanone of general formula with a compound of general formula, so as to provide a compound of general formula; b) converting said compound of general formula into a compound of general formula; wherein: - R 1 is selected from the group consisting of -CN and 1,2,4-oxadiazole, said 1,2,4-oxadiazole being attached to the bicycle via carbon 3 and optionally substituted in position 5 with a 3'-cyano-4'-isopropoxyphenyl group; - one of the dashed lines indicates a single bond and the other one a double bond, and when the dashed line linked to R 2 is a double bond R 2 is N, and when the dashed line linked to R 2 is a single bond R 2 is NH; - R 10 is selected from the group consisting of -CH 2 OH, -CH 2 OPg and -CO 2 R 12; - R 12 is selected from the group consisting of H, a linear or branched C1-C8 alkyl or a linear or branched C1-C8 alkyl substituted with a C6-C10 aryl; - Pg is an oxygen protecting group; and - the * indicates a stereogenic center; - R 1 is selected from the group consisting of -CN and 1,2,4-oxadiazole, said 1,2,4-oxadiazole being attached to the bicycle via carbon 3 and optionally substituted in position 5 with a 3'-cyano-4'-isopropoxyphenyl group; - one of the dashed lines indicates a single bond and the other one a double bond, and when the dashed line linked to R 2 is a double bond R 2 is N, and when the dashed line linked to R 2 is a single bond R 2 is NH; - R 10 is selected from the group consisting of -CH 2 OH, -CH 2 OPg and -CO 2 R 12; - R 12 is selected from the group consisting of H, a linear or branched C1-C8 alkyl or a linear or branched C1-C8 alkyl substituted with a C6-C10 aryl; - Pg is an oxygen protecting group; and - the * indicates a stereogenic center;
Device for removing the coating from a pipe end of a brake or fuel line, which is coated with a plastic coating, which has a metal pipe core, characterized in that the device comprises at least one pressure element, that is capable of removing the plastic coating from the pipe core through a mechanical deformation process, in which the plastic coating is subjected alternately to compression and pressure release.
A method of regenerating superabsorbent polymers which have been inactivated by an acid into superabsorbent recycled polymers which have a predetermined absorption property, the method comprising: a preparation step of preparing the superabsorbent polymers having an acid group and having been inactivated by the acid, a superabsorbent recycled polymer formation step of forming wet-state superabsorbent recycled polymers from the superabsorbent polymers which have been inactivated by the acid, by adding an alkali metal ion supply source which is capable of supplying an alkali metal ion to an aqueous solution for regeneration which includes the superabsorbent polymers which have been inactivated by the acid, and a drying step of forming the superabsorbent recycled polymers which have the predetermined absorption property by drying the wet-state superabsorbent recycled polymers, wherein the predetermined absorption property is adjusted by controlling a pH of the aqueous solution for regeneration. a preparation step of preparing the superabsorbent polymers having an acid group and having been inactivated by the acid, a superabsorbent recycled polymer formation step of forming wet-state superabsorbent recycled polymers from the superabsorbent polymers which have been inactivated by the acid, by adding an alkali metal ion supply source which is capable of supplying an alkali metal ion to an aqueous solution for regeneration which includes the superabsorbent polymers which have been inactivated by the acid, and a drying step of forming the superabsorbent recycled polymers which have the predetermined absorption property by drying the wet-state superabsorbent recycled polymers, wherein the predetermined absorption property is adjusted by controlling a pH of the aqueous solution for regeneration.
A method of coating a surface with a water and oil repellant polymer layer, the method comprising the steps of: - providing a substrate with a surface, - exposing said surface to a monomer compound, - exposing said surface to a continuous plasma having a plasma power provided by a plasma circuit, wherein said plasma circuit is impedance-adjusted so that a forward power is slightly higher than a reflected power and during the exposition of said surface to said continuous plasma, said plasma power is reduced from an initial higher plasma power to a final lower plasma power, said final lower plasma power being less than 30% of said initial higher plasma power, thus applying an even polymer layer exhibiting a water contact angle of more than 110°. - providing a substrate with a surface, - exposing said surface to a monomer compound, - exposing said surface to a continuous plasma having a plasma power provided by a plasma circuit,
A rotating machining device for machining a work piece comprising: 1) a support housing adapted to be mounted on a work piece; 2) a headstock rotatably mounted on the support housing; 3) at least one tool module mounted to the headstock and including a tool feed system having a tool holder and a feed mechanism operatively connected to the tool holder; and 4) a tripper pin assembly mounted on the support housing and arranged to collide with the feed mechanism for advancement of the tool holder relative to the work piece; wherein the tripper pin assembly collides with the feed mechanism at a collision point radially positioned inside of an outer diameter of the headstock, characterized by the radial position of the collision point being adjustable relative to the at least one tool module such that the collision point is repositionable independent of the at least one tool module. 1) a support housing adapted to be mounted on a work piece; 2) a headstock rotatably mounted on the support housing; 3) at least one tool module mounted to the headstock and including a tool feed system having a tool holder and a feed mechanism operatively connected to the tool holder; and 4) a tripper pin assembly mounted on the support housing and arranged to collide with the feed mechanism for advancement of the tool holder relative to the work piece; wherein the tripper pin assembly collides with the feed mechanism at a collision point radially positioned inside of an outer diameter of the headstock, characterized by the radial position of the collision point being adjustable relative to the at least one tool module such that the collision point is repositionable independent of the at least one tool module.
An artificial stone for covering a supporting surface, comprising: a base portion having a flat bottom for placement on the supporting surface, the base portion being shaped as a right regular prism, for patterned, fitting arrangement of the stone with like stones to produce a surface covering, the base portion having a regular base contour which is polygonal and a side wall for each side of the polygonal base contour; a top portion with a facing surface, the facing surface having an irregularly shaped top contour; and an intermediate portion connecting the top portion with the base portion, the intermediate portion having an inclined wall extending between the top portion and a sidewall of the base portion, the irregularly shaped top contour of the facing surface being different from the base contour for generating visible joints of irregular width and outline between adjacent like stones in an installed condition, the top contour being shifted or rotated relative to the polygonal cross-section or footprint of the base contour, wherein the top contour fits within the base contour, characterized in that the top portion has a depending rim along the top contour, the rim and the sidewall of the base portion being oriented perpendicular to the flat bottom. a base portion having a flat bottom for placement on the supporting surface, the base portion being shaped as a right regular prism, for patterned, fitting arrangement of the stone with like stones to produce a surface covering, the base portion having a regular base contour which is polygonal and a side wall for each side of the polygonal base contour; a top portion with a facing surface, the facing surface having an irregularly shaped top contour; and an intermediate portion connecting the top portion with the base portion, the intermediate portion having an inclined wall extending between the top portion and a sidewall of the base portion, the irregularly shaped top contour of the facing surface being different from the base contour for generating visible joints of irregular width and outline between adjacent like stones in an installed condition, the top contour being shifted or rotated relative to the polygonal cross-section or footprint of the base contour, wherein the top contour fits within the base contour, characterized in that the top portion has a depending rim along the top contour, the rim and the sidewall of the base portion being oriented perpendicular to the flat bottom.
An oil pressure controller for an automatic transmission, the oil pressure controller producing a pre-charge shelf pressure (Pa) supplied to a starter clutch by rapidly-decreasing a command hydraulic pressure to the starter clutch after temporarily rapidly increasing the command hydraulic pressure and also producing a capacity adjustment pressure (Pb1, Pb2) of the starter clutch by gradually increasing the command hydraulic pressure after decreasing the pre-charge shelf pressure (Pa) when a selecting operation is made from a neutral range to a drive range, the oil pressure controller comprising: a brake state detecting unit that detects a brake-operating/nonoperating state of a vehicle mounting the automatic transmission, and the command hydraulic pressure in the brake-nonoperating state being set to be higher than the command hydraulic pressure in the brake-operating state, characterized in that the capacity adjustment pressure in the brake-nonoperating state is a pressure obtained by adding a predetermined offset hydraulic pressure amount (Of) to the capacity adjustment pressure in the brake-operating state, wherein, when a brake is changed from the brake-operating state to the brake-nonoperating state during the progress of production of the capacity adjustment pressure on the basis of the selecting operation from the neutral range to the drive range, the capacity adjustment pressure in the brake-nonoperating state being produced by adding the offset hydraulic pressure amount (Of) to the capacity adjustment pressure In the brake-operating state while gradually increasing the offset hydraulic pressure amount (Of). a brake state detecting unit that detects a brake-operating/nonoperating state of a vehicle mounting the automatic transmission, and the command hydraulic pressure in the brake-nonoperating state being set to be higher than the command hydraulic pressure in the brake-operating state, characterized in that the capacity adjustment pressure in the brake-nonoperating state is a pressure obtained by adding a predetermined offset hydraulic pressure amount (Of) to the capacity adjustment pressure in the brake-operating state, wherein, when a brake is changed from the brake-operating state to the brake-nonoperating state during the progress of production of the capacity adjustment pressure on the basis of the selecting operation from the neutral range to the drive range, the capacity adjustment pressure in the brake-nonoperating state being produced by adding the offset hydraulic pressure amount (Of) to the capacity adjustment pressure In the brake-operating state while gradually increasing the offset hydraulic pressure amount (Of).
A processing apparatus comprising a processor, wherein: the processor comprises a plurality of deferred-push processor registers; the processor comprises processor-register control circuitry (220, 222, 224, 226, 228); the processor-register control circuitry comprises a plurality of status registers, each status register corresponding to a different respective deferred-push register; the processor-register control circuitry (220, 222, 224, 226, 228) is configured to detect a write of a new value to a register of the deferred-push registers; the processor-register control circuitry (220, 222, 224, 226, 228) is configured, in response to said detection, to determine whether the status register for the deferred-push register has a first value, indicative of an unsaved status for the deferred-push register; and the processor-register control circuitry (220, 222, 224, 226, 228) is configured, when the status register is determined to have the first value, to: read a current value from the deferred-push register before the writing of the new value to the deferred-push register completes; write the current value to a memory; and set the status register for the deferred-push register to a second value, indicative of a saved status for the deferred-push register. the processor comprises a plurality of deferred-push processor registers; the processor comprises processor-register control circuitry (220, 222, 224, 226, 228); the processor-register control circuitry comprises a plurality of status registers, each status register corresponding to a different respective deferred-push register; the processor-register control circuitry (220, 222, 224, 226, 228) is configured to detect a write of a new value to a register of the deferred-push registers; the processor-register control circuitry (220, 222, 224, 226, 228) is configured, in response to said detection, to determine whether the status register for the deferred-push register has a first value, indicative of an unsaved status for the deferred-push register; and the processor-register control circuitry (220, 222, 224, 226, 228) is configured, when the status register is determined to have the first value, to: read a current value from the deferred-push register before the writing of the new value to the deferred-push register completes; write the current value to a memory; and set the status register for the deferred-push register to a second value, indicative of a saved status for the deferred-push register.
A method for high-spatial and temporal resolution imaging of microvessels using an ultrasound system, the steps of the method comprising: (a) accessing ultrasound data with a computer system, the ultrasound data having been acquired with the ultrasound system from a region-of-interest in a subject in which a microbubble contrast agent was present when the ultrasound data were acquired; (b) generating microbubble signal data with the computer system by separating microbubble signals in the ultrasound data from other signals in the ultrasound data; (c) determining a point spread function for the ultrasound system used to acquire the ultrasound data; (d) generating (350,360) a cross-correlation map by: determining a first Nth power of the microbubble signal data, wherein N for the first Nth power is an integer greater than 1; determining a second Nth power of the PSF of the ultrasound system, wherein N for the second Nth power is an integer greater than 1; and generating the cross-correlation map between the first Nth power of the microbubble signal data and the second Nth power of the point spread function of the ultrasound system; and (e) producing a high spatial and temporal resolution microvessel image based at least in part on the generated cross-correlation map. (a) accessing ultrasound data with a computer system, the ultrasound data having been acquired with the ultrasound system from a region-of-interest in a subject in which a microbubble contrast agent was present when the ultrasound data were acquired; (b) generating microbubble signal data with the computer system by separating microbubble signals in the ultrasound data from other signals in the ultrasound data; (c) determining a point spread function for the ultrasound system used to acquire the ultrasound data; (d) generating (350,360) a cross-correlation map by: determining a first Nth power of the microbubble signal data, wherein N for the first Nth power is an integer greater than 1; determining a second Nth power of the PSF of the ultrasound system, wherein N for the second Nth power is an integer greater than 1; and generating the cross-correlation map between the first Nth power of the microbubble signal data and the second Nth power of the point spread function of the ultrasound system; and determining a first Nth power of the microbubble signal data, wherein N for the first Nth power is an integer greater than 1; determining a second Nth power of the PSF of the ultrasound system, wherein N for the second Nth power is an integer greater than 1; and generating the cross-correlation map between the first Nth power of the microbubble signal data and the second Nth power of the point spread function of the ultrasound system; and (e) producing a high spatial and temporal resolution microvessel image based at least in part on the generated cross-correlation map.
A method for wireless communications, comprising: receiving multiple feedback aspects of a channel for the wireless communications; determining multiple codewords (W 1, W 2) based on the multiple feedback aspects; determining a final precoding matrix based on the multiple codewords (W 1, W 2); enforcing at least one codebook property in the final precoding matrix, wherein enforcing the at least one codebook property comprises quantizing the final precoding matrix, wherein quantizing the final precoding matrix comprises quantizing each element in the final precoding matrix to a nearest value in a finite alphabet; applying the final precoding matrix to a plurality of spatial streams to form precoded spatial streams; and transmitting the precoded spatial streams. receiving multiple feedback aspects of a channel for the wireless communications; determining multiple codewords (W 1, W 2) based on the multiple feedback aspects; determining a final precoding matrix based on the multiple codewords (W 1, W 2); enforcing at least one codebook property in the final precoding matrix, wherein enforcing the at least one codebook property comprises quantizing the final precoding matrix, wherein quantizing the final precoding matrix comprises quantizing each element in the final precoding matrix to a nearest value in a finite alphabet; applying the final precoding matrix to a plurality of spatial streams to form precoded spatial streams; and transmitting the precoded spatial streams.
An isolated nucleic acid molecule that encodes a cytochrome P450 polypeptide wherein said nucleic acid molecule comprises or consists of a nucleotide sequence selected from the group consisting of: i) a nucleotide sequence as represented by the sequence in Figure 1c, 1d or 3c; ii) a nucleotide sequence wherein said sequence is degenerate as a result of the genetic code to the nucleotide sequence defined in (i); iii) a nucleic acid molecule the complementary strand of which hybridizes to nucleotide sequences with at least 90% identity under very stringent hybridization conditions to the sequence in Figure 1c 1d or 3c wherein said nucleic acid molecule encodes a cytochrome P450 polypeptide; iv) a nucleotide sequence that encodes a polypeptide comprising an amino acid sequence as represented in Figure 4c; v) a nucleotide sequence that encodes a polypeptide comprising an amino acid sequence wherein said amino acid sequence is modified by addition deletion or substitution of at least one amino acid residue as represented in iv) above and has at least 85% sequence identity to the full length sequence represented in Figure 4c which has retained cytochrome P450 activity. i) a nucleotide sequence as represented by the sequence in Figure 1c, 1d or 3c; ii) a nucleotide sequence wherein said sequence is degenerate as a result of the genetic code to the nucleotide sequence defined in (i); iii) a nucleic acid molecule the complementary strand of which hybridizes to nucleotide sequences with at least 90% identity under very stringent hybridization conditions to the sequence in Figure 1c 1d or 3c wherein said nucleic acid molecule encodes a cytochrome P450 polypeptide; iv) a nucleotide sequence that encodes a polypeptide comprising an amino acid sequence as represented in Figure 4c; v) a nucleotide sequence that encodes a polypeptide comprising an amino acid sequence wherein said amino acid sequence is modified by addition deletion or substitution of at least one amino acid residue as represented in iv) above and has at least 85% sequence identity to the full length sequence represented in Figure 4c which has retained cytochrome P450 activity.
Storage assembly for a vehicle, the assembly comprising: • a storage body delimiting a storage area accessible via an opening; • a cover that is movable in relation to the storage body between an open position, in which the opening is detached, and a closed position, in which the cover closes the opening; and • a locking device arranged to lock the cover in relation to the storage body comprising a lever connected to the storage body and a locking member fastened to the cover; characterised in that the lever is movable in relation to the storage body between a locking position, in which the lever cooperates with the locking member to block the cover in closed position in order to prevent it from moving towards its open position, and a release position, in which the cover is free to move in relation to the storage body from its closed position to its open position; and in that: • a bistable spring of the locking device stresses the lever selectively towards the locking position or towards the release position. • a storage body delimiting a storage area accessible via an opening; • a cover that is movable in relation to the storage body between an open position, in which the opening is detached, and a closed position, in which the cover closes the opening; and • a locking device arranged to lock the cover in relation to the storage body comprising a lever connected to the storage body and a locking member fastened to the cover; characterised in that the lever is movable in relation to the storage body between a locking position, in which the lever cooperates with the locking member to block the cover in closed position in order to prevent it from moving towards its open position, and a release position, in which the cover is free to move in relation to the storage body from its closed position to its open position; and in that: • a bistable spring of the locking device stresses the lever selectively towards the locking position or towards the release position.