mhurhangee/ep-ind-claims huggingface dataset:
A process for producing a cyclopentaquinazoline of general formula (VIII) wherein R 1 is independently selected from hydrogen, amino, C 1-4 alkyl, C 1-4 alkoxy, fluoroC 1-4 alkyl, hydroxyC 1-4 alkyl and protected hydroxyC 1-4 alkyl R 2 is C 3-4 alkynyl Ar is independently selected from C 5-20 arylene optionally substituted on the ring with one or two substituents selected from halogeno, hydroxyl, amino, nitro, cyano, trifluoromethyl, C 1-4 alkyl and C 1-4 alkoxy from a 5-amino-6-haloindanone of formula IX wherein X is a halide comprising the steps of: (a) acylation of the 5-amino group; (b) cyanide displacement of the 6-halo group; (c) hydrolysis of the nitrile group produced in step (b); and (d)cyclisation of the 5-(N-acylamino)-6-amidoindanone to form a cyclopentaquinazoline ring system characterised in that the process further comprises steps (e) reduction of the cyclopentaquinazoline keto group to produce an indanol of general formula and (f) coupling of an amine nucleophile to the indanol produced in step (e) wherein coupling comprises conversion of the hydroxy group of the indanol into a leaving group, followed by reaction with the amine nucleophile, wherein the amine nucleophile is an amine of general formula wherein R' is hydrogen, or a protecting group. R 1 is independently selected from hydrogen, amino, C 1-4 alkyl, C 1-4 alkoxy, fluoroC 1-4 alkyl, hydroxyC 1-4 alkyl and protected hydroxyC 1-4 alkyl R 2 is C 3-4 alkynyl Ar is independently selected from C 5-20 arylene optionally substituted on the ring with one or two substituents selected from halogeno, hydroxyl, amino, nitro, cyano, trifluoromethyl, C 1-4 alkyl and C 1-4 alkoxy (a) acylation of the 5-amino group; (b) cyanide displacement of the 6-halo group; (c) hydrolysis of the nitrile group produced in step (b); and (d)cyclisation of the 5-(N-acylamino)-6-amidoindanone to form a cyclopentaquinazoline ring system characterised in that the process further comprises steps (e) reduction of the cyclopentaquinazoline keto group to produce an indanol of general formula and (f) coupling of an amine nucleophile to the indanol produced in step (e) wherein coupling comprises conversion of the hydroxy group of the indanol into a leaving group, followed by reaction with the amine nucleophile, wherein the amine nucleophile is an amine of general formula wherein R' is hydrogen, or a protecting group.
A wireless communication device comprising: a reception unit; and a transmission unit configured to transmit or to stop transmitting data on a basis of a first threshold value set in association with a second threshold value, characterized in that the first threshold value, which is a signal detection level at which a signal transported by an electric wave is detected by the reception unit of the wireless communication device, is a threshold value that changes in accordance with a change of the second threshold value, and wherein the second threshold value is a reception determination level set on a basis of a transmission power of a signal, the signal being transmitted from a second wireless communication device that belongs to a second wireless communication network that is different from a first wireless communication network to which the wireless communication device belongs, and the signal being detected by the reception unit of the wireless communication device. a reception unit; and a transmission unit configured to transmit or to stop transmitting data on a basis of a first threshold value set in association with a second threshold value, characterized in that the first threshold value, which is a signal detection level at which a signal transported by an electric wave is detected by the reception unit of the wireless communication device, is a threshold value that changes in accordance with a change of the second threshold value, and wherein the second threshold value is a reception determination level set on a basis of a transmission power of a signal, the signal being transmitted from a second wireless communication device that belongs to a second wireless communication network that is different from a first wireless communication network to which the wireless communication device belongs, and the signal being detected by the reception unit of the wireless communication device.
A method in a first network element (1, 3, 5, 90) of a telecommunications network for determining a quality of an uplink from a second network element (1, 3, 5, 90) to the first network element(1, 3, 5, 90), the method comprising: monitoring an amount of data received from the second network element (1, 3, 5, 90), the amount of data received providing a first value, Mrx; characterized in that the method further comprises the steps of: receiving a second value, Xtx, from the second network element (1, 3, 5, 90), the second value, Xtx, corresponding to a first time period during which the second network element (1, 3, 5, 90) has been transmitting data to the first network element (1, 3, 5, 90); and wherein the method further comprises determining the quality of the uplink by determining a throughput of the uplink from the second network element (1, 3, 5, 90) to the first network element (1, 3, 5, 90) using the first value, Mrx, and the second value, Xtx. monitoring an amount of data received from the second network element (1, 3, 5, 90), the amount of data received providing a first value, Mrx; characterized in that the method further comprises the steps of: receiving a second value, Xtx, from the second network element (1, 3, 5, 90), the second value, Xtx, corresponding to a first time period during which the second network element (1, 3, 5, 90) has been transmitting data to the first network element (1, 3, 5, 90); and wherein the method further comprises determining the quality of the uplink by determining a throughput of the uplink from the second network element (1, 3, 5, 90) to the first network element (1, 3, 5, 90) using the first value, Mrx, and the second value, Xtx. receiving a second value, Xtx, from the second network element (1, 3, 5, 90), the second value, Xtx, corresponding to a first time period during which the second network element (1, 3, 5, 90) has been transmitting data to the first network element (1, 3, 5, 90); and wherein the method further comprises determining the quality of the uplink by determining a throughput of the uplink from the second network element (1, 3, 5, 90) to the first network element (1, 3, 5, 90) using the first value, Mrx, and the second value, Xtx.
A method of making an ion-conductive polymer film for an electrochromic device, wherein the method comprises: (a) mixing one or more monomers capable of forming a thermoplastic polymer, a plasticizer, a salt which is soluble in the plasticizer, a UV stabilizer, and a polymer-forming catalyst to form a mixture; (b) polymerizing during a first polymerization the mixture to obtain a formulation containing a thermoplastic polymer; and (c) extruding or casting the formulation to form said ion-conductive polymer film characterized in that the mixture prior to the first polymerization further contains at least one additional monomer which does not participate in the formation of the thermoplastic polymer, and which is polymerized after the polymer film has been formed by irradiating the polymer film after step (c). (a) mixing one or more monomers capable of forming a thermoplastic polymer, a plasticizer, a salt which is soluble in the plasticizer, a UV stabilizer, and a polymer-forming catalyst to form a mixture; (b) polymerizing during a first polymerization the mixture to obtain a formulation containing a thermoplastic polymer; and (c) extruding or casting the formulation to form said ion-conductive polymer film characterized in that the mixture prior to the first polymerization further contains at least one additional monomer which does not participate in the formation of the thermoplastic polymer, and which is polymerized after the polymer film has been formed by irradiating the polymer film after step (c).
Method for access control, in particular in buildings, in which a bidirectional data transmission takes place between an electronic key and an access control device, said data transmission including the transmission of identification data from the electronic key to the access control device, wherein the identification data are evaluated in the access control device for determining access authorization and a blocking member for selectively authorizing or blocking the access is activated as a function of the determined access authorization, wherein the data transmission is effected at least partially via a capacitive coupling between the electronic key and the access control device, wherein a portion of the data transmitted between the electronic key and the access control device is transferred via a capacitive coupling and a portion of the data is transferred via radio waves, characterized in that the bidirectional data transmission comprises the emission of a presence control signal by the access control device, said presence control signal being emitted via radio waves with a range of less than 2m, preferably less than 1m.
Apparatus for replacing an exhausted transmission fluid of an automatic gear shift of a motor vehicle with a fresh transmission fluid, comprising: a first tube and a second tube, respectively connectable to two different access points of said automatic gear shift; a first tank containing the fresh transmission fluid; a second tank configured to receive the exhausted transmission fluid; a first three-way electro valve configured to establish a selective communication between said first tube and said first tank or between said first tube and said second tank; a second three-way electro valve configured to establish a selective communication between said second tube and said first tank or between said second tube and said second tank; a first pressure gauge and a second pressure gauge which are operatively active respectively on the first tube and on the second tube so as to detect the pressure of the transmission fluid, the apparatus comprises an oleodynamic manifold in turn comprising a box-like casing housing said three-way electro valves (14, 15) and said pressure gauges (8, 9), and a first calibrated throttling is present between said first gauge and said first three-way electro valve and a second calibrated throttling is present between said second gauge and said second three-way electro valve. a first tube and a second tube, respectively connectable to two different access points of said automatic gear shift; a first tank containing the fresh transmission fluid; a second tank configured to receive the exhausted transmission fluid; a first three-way electro valve configured to establish a selective communication between said first tube and said first tank or between said first tube and said second tank; a second three-way electro valve configured to establish a selective communication between said second tube and said first tank or between said second tube and said second tank; a first pressure gauge and a second pressure gauge which are operatively active respectively on the first tube and on the second tube so as to detect the pressure of the transmission fluid, the apparatus comprises an oleodynamic manifold in turn comprising a box-like casing housing said three-way electro valves (14, 15) and said pressure gauges (8, 9), and a first calibrated throttling is present between said first gauge and said first three-way electro valve and a second calibrated throttling is present between said second gauge and said second three-way electro valve.
Exterior aircraft light unit, comprising: a plurality of LEDs, a support plate for supporting the plurality of LEDs, the support plate having a main plane of extension, and a reflector, characterized in that the support plate has a curved, concave LED support surface, substantially orthogonal to the main plane of extension, the plurality of LEDs are arranged along the curved, concave LED support surface, and the reflector faces the plurality of LEDs and is shaped to reflect light from the plurality of LEDs past the support plate towards an outside of the exterior aircraft light unit. a plurality of LEDs, a support plate for supporting the plurality of LEDs, the support plate having a main plane of extension, and a reflector, characterized in that the support plate has a curved, concave LED support surface, substantially orthogonal to the main plane of extension, the plurality of LEDs are arranged along the curved, concave LED support surface, and the reflector faces the plurality of LEDs and is shaped to reflect light from the plurality of LEDs past the support plate towards an outside of the exterior aircraft light unit. the support plate has a curved, concave LED support surface, substantially orthogonal to the main plane of extension, the plurality of LEDs are arranged along the curved, concave LED support surface, and the reflector faces the plurality of LEDs and is shaped to reflect light from the plurality of LEDs past the support plate towards an outside of the exterior aircraft light unit.
Bone mill (20; 20') for comminuting grinding material in the form of bone or bone material, comprising a receiving chamber for the grinding material, a comminuting device and an advancing element for moving the grinding material in the receiving chamber in the direction towards the comminuting device, wherein the receiving chamber has an exit opening covered at least partially by the comminuting device, wherein the receiving chamber is movable relative to the comminuting device and wherein the receiving chamber is rotatable about an axis of rotation relative to the comminuting device, characterized in that the receiving chamber has an inner wall section curved convexly in relation to the axis of rotation.
Composition comprising, HFO-1234yf, HCC-40 and at least one compound chosen from HFO-1234ze, HFC-134a, HCFC-115, HFC-152a and HFO-1243zf; said composition comprising at least 99% by weight of HFO-1234yf and at most 1% by weight of all of the additional compounds.
A system, comprising: a resonant air gap transfer transformer having a primary side resonant LC circuit and a secondary side resonant LC circuit; a power generating section that provides a first square wave through a first DC blocking capacitor and a first Thevenin inductor to a summing node of the primary side resonant LC circuit; a reactance generating section that provides a second square wave through a second DC blocking capacitor and a second Thevenin inductor to the summing node of the primary side resonant LC circuit, wherein phase and amplitude differences between said first square wave and said second square wave produce a current into the summing node of the primary side resonant LC circuit, wherein the reactance generating section provides an effective impedance that is adjusted by adjusting the phase and/or the magnitude of the first and second square waves; and a rectifier-filter load circuit connected to said secondary side resonant LC circuit. a resonant air gap transfer transformer having a primary side resonant LC circuit and a secondary side resonant LC circuit; a power generating section that provides a first square wave through a first DC blocking capacitor and a first Thevenin inductor to a summing node of the primary side resonant LC circuit; a reactance generating section that provides a second square wave through a second DC blocking capacitor and a second Thevenin inductor to the summing node of the primary side resonant LC circuit, wherein phase and amplitude differences between said first square wave and said second square wave produce a current into the summing node of the primary side resonant LC circuit, wherein the reactance generating section provides an effective impedance that is adjusted by adjusting the phase and/or the magnitude of the first and second square waves; and a rectifier-filter load circuit connected to said secondary side resonant LC circuit.
A dairy bacterial strain with clumping and/or chaining properties, preferably when cultured under liquid conditions, preferably without a substantial amount of a clumping agent, wherein the clumping property results in clumps of at least 20 bacteria per average clump and wherein the chaining property results in chains of at least 8 bacteria per average chain and wherein said strain comprises an increased amount of expression product of a pilin gene cluster, such expression product comprising pilin, and wherein the amount of expression product is increased in view of Lactococcus lactis subsp cremoris NCDO712 when cultured under identical conditions and wherein the pilin gene cluster has a nucleotide sequence that has at least 90% sequence identity with SEQ ID NO: 1 and wherein said dairy bacterial strain is a lactic acid bacterial strain.
A computer-implemented method comprising: implementing, on a client computing device, a client-side application that communicates with an online content management system to sync data stored locally on the client computing device with data stored at the online content management system; running a local web server on the client computing device, the local web server being configured to communicate with the client-side application to interact with at least a portion of the data stored locally, wherein the data stored locally is synced with the data stored at the online content management system; running a web browser on the client computing device; accessing the local web server running on the client computing device via the web browser; initiating a request, simultaneously with respect to the online content management system and the local web server, to access data stored on the online content management system and on the local web server, wherein the request is satisfied by the online content management system if the online content management system responds first and the request is satisfied by the local web server if the local web server responds first, and wherein the data stored on the online content management system and the data stored on the local web server are synched; and interacting with the at least a portion of the data stored locally when the local web server responds first, wherein the interacting with the at least a portion of the data stored locally is based, at least in part, on the accessing of the local web server via the web browser. implementing, on a client computing device, a client-side application that communicates with an online content management system to sync data stored locally on the client computing device with data stored at the online content management system; running a local web server on the client computing device, the local web server being configured to communicate with the client-side application to interact with at least a portion of the data stored locally, wherein the data stored locally is synced with the data stored at the online content management system; running a web browser on the client computing device; accessing the local web server running on the client computing device via the web browser; initiating a request, simultaneously with respect to the online content management system and the local web server, to access data stored on the online content management system and on the local web server, wherein the request is satisfied by the online content management system if the online content management system responds first and the request is satisfied by the local web server if the local web server responds first, and wherein the data stored on the online content management system and the data stored on the local web server are synched; and interacting with the at least a portion of the data stored locally when the local web server responds first, wherein the interacting with the at least a portion of the data stored locally is based, at least in part, on the accessing of the local web server via the web browser.
An underwater vehicle comprising: a longitudinal body that defines a longitudinal axis and is rotatable about the longitudinal axis between a forward orientation and a sideways orientation; a wing attached to the longitudinal body wherein the wing is moveable between a vertically extending wing orientation when the longitudinal body is in the forward orientation and a horizontally extending wing orientation when the longitudinal body is in the sideways orientation, wherein the wing includes at least two sensors (44, 46) including a first sensor arranged at an end of the wing and a second sensor arranged at an opposite end of the wing relative to the first sensor; a propulsion system (28, 30) having a front propulsion device and a rear propulsion device that is arranged rearwardly along the longitudinal axis relative to the front propulsion device, the propulsion system providing thrust in a perpendicular direction relative to the longitudinal axis; and an after-propulsion system arranged at a rear end of the longitudinal body that provides thrust along the longitudinal axis, wherein the longitudinal body includes at least one moveable mass that moves the longitudinal body between the forward orientation and the sideward orientation and maintains a buoyancy of the longitudinal body. a longitudinal body that defines a longitudinal axis and is rotatable about the longitudinal axis between a forward orientation and a sideways orientation; a wing attached to the longitudinal body wherein the wing is moveable between a vertically extending wing orientation when the longitudinal body is in the forward orientation and a horizontally extending wing orientation when the longitudinal body is in the sideways orientation, wherein the wing includes at least two sensors (44, 46) including a first sensor arranged at an end of the wing and a second sensor arranged at an opposite end of the wing relative to the first sensor; a propulsion system (28, 30) having a front propulsion device and a rear propulsion device that is arranged rearwardly along the longitudinal axis relative to the front propulsion device, the propulsion system providing thrust in a perpendicular direction relative to the longitudinal axis; and an after-propulsion system arranged at a rear end of the longitudinal body that provides thrust along the longitudinal axis, wherein the longitudinal body includes at least one moveable mass that moves the longitudinal body between the forward orientation and the sideward orientation and maintains a buoyancy of the longitudinal body.