mhurhangee/ep-ind-claims huggingface dataset:
A compound having the formula: wherein: L is -NHCO- or -CONH-; and R 1 and R 2 are both heteroaryl, wherein at least one of R 1 and R 2 is unsubstituted and one of R 1 and R 2 is optionally mono-, di-, or tri-substituted independently with alkyl, alkoxy, halogen, cyano, nitro, trifluoroalkyl, amino, alkylamino, dialkylamino, acyl, aryl, heteroaryl, heterocyclyl, heterocyclyl-R 3, -NHR 3, -N(alkyl)R 3, -C NHR 3, -C N(alkyl)R 3, -NHC R 3, -N(alkyl)C R 3, - OH or -OR 3, wherein: R 3 is C 1 -C 6 alkyl or C 1 -C 6 cycloalkyl, which is optionally substituted with halogen, -CN, -NH 2, - NH(C 1 -C 3 alkyl), -N(C 1 -C 3 alkyl) 2, C 1 -C 3 alkylheterocyclyl, C 1 -C 3 alkylcarbamate, -C NH(C 1 -C 3 alkyl), -C N(C 1 -C 3 alkyl) 2, -NHC -C 1 -C 3 alkyl, -N(C 1 -C 3 alkyl)-C -C 1 -C 3 alkyl, OH, or -O-C 1 -C 6 alkyl; or a pharmaceutically acceptable salt thereof. L is -NHCO- or -CONH-; and R 1 and R 2 are both heteroaryl, wherein at least one of R 1 and R 2 is unsubstituted and one of R 1 and R 2 is optionally mono-, di-, or tri-substituted independently with alkyl, alkoxy, halogen, cyano, nitro, trifluoroalkyl, amino, alkylamino, dialkylamino, acyl, aryl, heteroaryl, heterocyclyl, heterocyclyl-R 3, -NHR 3, -N(alkyl)R 3, -C NHR 3, -C N(alkyl)R 3, -NHC R 3, -N(alkyl)C R 3, - OH or -OR 3, wherein: R 3 is C 1 -C 6 alkyl or C 1 -C 6 cycloalkyl, which is optionally substituted with halogen, -CN, -NH 2, - NH(C 1 -C 3 alkyl), -N(C 1 -C 3 alkyl) 2, C 1 -C 3 alkylheterocyclyl, C 1 -C 3 alkylcarbamate, -C NH(C 1 -C 3 alkyl), -C N(C 1 -C 3 alkyl) 2, -NHC -C 1 -C 3 alkyl, -N(C 1 -C 3 alkyl)-C -C 1 -C 3 alkyl, OH, or -O-C 1 -C 6 alkyl; or a pharmaceutically acceptable salt thereof. R 3 is C 1 -C 6 alkyl or C 1 -C 6 cycloalkyl, which is optionally substituted with halogen, -CN, -NH 2, - NH(C 1 -C 3 alkyl), -N(C 1 -C 3 alkyl) 2, C 1 -C 3 alkylheterocyclyl, C 1 -C 3 alkylcarbamate, -C NH(C 1 -C 3 alkyl), -C N(C 1 -C 3 alkyl) 2, -NHC -C 1 -C 3 alkyl, -N(C 1 -C 3 alkyl)-C -C 1 -C 3 alkyl, OH, or -O-C 1 -C 6 alkyl; or a pharmaceutically acceptable salt thereof.
A concentrated power-distribution member for a concentrated winding motor, comprising: a ring-shaped busbar having a center axis; and a coil connection terminal formed in one-piece with the busbar to hold a coil winding end positioned in an inner side of the busbar, wherein the coil connection terminal comprises: an erected portion that extends from the busbar in parallel with the center axis, the erected portion having a leading end; a pair of arms extending from the leading end toward the center axis, the pair of arms being constituted by a pair of wing portions that extends from the leading end of the erected portion to both sides of a tangential direction of the busbar and are bent toward the center axis along a bending line parallel to the center axis; and a coil end holding portion provided in the leading ends of the pair of arms, characterised in that a narrow portion is formed by deforming a middle part of the pair of arms to adjoin each other to cause the coil end holding portion to be provided in a leading end side of the pair of arms from the narrow portion and form a fork-shape. a ring-shaped busbar having a center axis; and a coil connection terminal formed in one-piece with the busbar to hold a coil winding end positioned in an inner side of the busbar, wherein the coil connection terminal comprises: an erected portion that extends from the busbar in parallel with the center axis, the erected portion having a leading end; a pair of arms extending from the leading end toward the center axis, the pair of arms being constituted by a pair of wing portions that extends from the leading end of the erected portion to both sides of a tangential direction of the busbar and are bent toward the center axis along a bending line parallel to the center axis; and a coil end holding portion provided in the leading ends of the pair of arms, characterised in that a narrow portion is formed by deforming a middle part of the pair of arms to adjoin each other to cause the coil end holding portion to be provided in a leading end side of the pair of arms from the narrow portion and form a fork-shape. an erected portion that extends from the busbar in parallel with the center axis, the erected portion having a leading end; a pair of arms extending from the leading end toward the center axis, the pair of arms being constituted by a pair of wing portions that extends from the leading end of the erected portion to both sides of a tangential direction of the busbar and are bent toward the center axis along a bending line parallel to the center axis; and a coil end holding portion provided in the leading ends of the pair of arms, characterised in that a narrow portion is formed by deforming a middle part of the pair of arms to adjoin each other to cause the coil end holding portion to be provided in a leading end side of the pair of arms from the narrow portion and form a fork-shape.
A system for energy recovery for zootechnical plants, which comprises - a first circuit of water to be cooled, which has a duct for drawing well water at a first temperature and a duct for discharging said well water at a temperature that is lower than said first temperature in a first accumulation vat for the water that arrives from said discharge duct - a duct for conveying milk from a milking plant to a low-temperature milk storage tank, there being, along said milk conveyance duct, at least one first exchanger that uses, for cooling said milk, the water stored in said first accumulation vat for the water that arrives from said discharge duct characterized in that the system further comprises: - a geothermal heat pump - a second circuit of water to be heated in order to be stored in at least one first hot water accumulation tank, said geothermal heat pump being provided with a device for heat exchange between said said first circuit and said second circuit, - a milk refrigeration unit - a second exchanger connected functionally to said milk refrigeration unit, said second exchanger being provided along said milk conveyance duct, said milk refrigeration unit comprising a chilled water accumulation vat connected, by way of a cooling circuit, to said second exchanger said milk refrigeration unit being connected functionally to a second hot water accumulation tank, which is connected to the first hot water accumulation tank by way of an exchanger circuit. - a first circuit of water to be cooled, which has a duct for drawing well water at a first temperature and a duct for discharging said well water at a temperature that is lower than said first temperature in a first accumulation vat for the water that arrives from said discharge duct - a duct for conveying milk from a milking plant to a low-temperature milk storage tank, there being, along said milk conveyance duct, at least one first exchanger that uses, for cooling said milk, the water stored in said first accumulation vat for the water that arrives from said discharge duct - a geothermal heat pump - a second circuit of water to be heated in order to be stored in at least one first hot water accumulation tank, said geothermal heat pump being provided with a device for heat exchange between said said first circuit and said second circuit, - a milk refrigeration unit - a second exchanger connected functionally to said milk refrigeration unit, said second exchanger being provided along said milk conveyance duct,
A polymer fibre comprising a thermoplastic polymer comprising the following building blocks A and B: -O-(CH 2 -CH 2 -O) n - -O-[CH 2] y -O- n indicating a repeating unit and being an integer of 10-400, and y being an integer in the range of 2 to 16, wherein: • A is present in an amount of 15-30 mole%, • B is present in an amount of 20-40 mole%, wherein building blocks A and B are linked by the following linking group C: -[(C=O)-NH-CH 2 -CH 2 -CH 2 -CH 2 -CH 2 -CH 2 -NH-(C=O)]- wherein • C is present in an amount of 45-55 mole%. • A is present in an amount of 15-30 mole%, • B is present in an amount of 20-40 mole%, • C is present in an amount of 45-55 mole%.
A method of controlling a wind turbine having a rotor and a generator for producing power, the wind turbine being erected on a location and designed for a nominal load, the method comprising: - defining a plurality of sectors each specifying a range of wind directions towards the wind turbine, - defining, for each sector, an expected wind load from the specified directions and a sector control strategy which is based on a predetermined comparison between the expected wind load and the nominal load; and. - determining a current wind direction and controlling the wind turbine in accordance with the sector control strategy defined for the sector to which the current wind direction corresponds. - defining a plurality of sectors each specifying a range of wind directions towards the wind turbine, - defining, for each sector, an expected wind load from the specified directions and a sector control strategy which is based on a predetermined comparison between the expected wind load and the nominal load; and. - determining a current wind direction and controlling the wind turbine in accordance with the sector control strategy defined for the sector to which the current wind direction corresponds.
A reversible airway device comprising: a tubular guide having a distal end portion, a proximal end portion, and a first passageway extending between the distal and proximal end portions; a laryngeal mask attached to the distal end portion of the tubular guide, the laryngeal mask including an opening in fluid communication with the first passageway; an endotracheal tube slidably disposed within the first passageway, the endotracheal tube having a second passageway that is disposed within the first passageway; and a sealing mechanism disposed within the first passageway for occluding the flow of a gas through the first passageway; characterised in that the tubular guide includes a longitudinal slot partially extending between the distal and proximal end portions thereof. a tubular guide having a distal end portion, a proximal end portion, and a first passageway extending between the distal and proximal end portions; a laryngeal mask attached to the distal end portion of the tubular guide, the laryngeal mask including an opening in fluid communication with the first passageway; an endotracheal tube slidably disposed within the first passageway, the endotracheal tube having a second passageway that is disposed within the first passageway; and a sealing mechanism disposed within the first passageway for occluding the flow of a gas through the first passageway; characterised in that the tubular guide includes a longitudinal slot partially extending between the distal and proximal end portions thereof.
A vehicle window plate protection sheet which is suitable to be applied to a window plate of a vehicle to protect the window plate, comprising a substrate and a pressure-sensitive adhesive layer provided to one face of the substrate, wherein the pressure-sensitive adhesive layer comprises a base polymer and an application aider, the base polymer being an acrylic polymer, wherein the acrylic polymer is a copolymer of a monomer mixture comprising: 30% by weight or greater of a monomer (a) represented by the following formula: CH 2 =C(R 1)COOR 2 in which R 1 is a hydrogen atom or a methyl group and R 2 is an C 6-16 acyclic alkyl group; 30% by weight or greater of a monomer (b) represented by the following formula: CH 2 =C(R 3)COOR 4 in which R 3 is a hydrogen atom or a methyl group and R 4 is an C 1-3 acyclic alkyl group; and 2 to 20 parts by weight of a hydroxy group-containing monomer to 100 parts by weight of all alkyl (meth)acrylate; the application aider content being higher than 0 parts by weight and up to 10 parts by weight to 100 parts by weight of the base polymer, wherein the application aider is selected from anionic surfactants, nonionic surfactants, cationic surfactants, hydrophilic polymers and a combination thereof, and wherein the protection sheet satisfies the following conditions: having a 30-minute peel strength of less than 0.10 N/20mm; and having a 48-hour peel strength of 0.05 N/20mm or greater, wherein the 30-minute peel strength and the 48-hour peel strength are determined according to methods disclosed in the specification. 30% by weight or greater of a monomer (a) represented by the following formula: CH 2 =C(R 1)COOR 2 in which R 1 is a hydrogen atom or a methyl group and R 2 is an C 6-16 acyclic alkyl group; 30% by weight or greater of a monomer (b) represented by the following formula: CH 2 =C(R 3)COOR 4 in which R 3 is a hydrogen atom or a methyl group and R 4 is an C 1-3 acyclic alkyl group; and 2 to 20 parts by weight of a hydroxy group-containing monomer to 100 parts by weight of all alkyl (meth)acrylate; the application aider content being higher than 0 parts by weight and up to 10 parts by weight to 100 parts by weight of the base polymer, wherein the application aider is selected from anionic surfactants, nonionic surfactants, cationic surfactants, hydrophilic polymers and a combination thereof, and wherein the protection sheet satisfies the following conditions: having a 30-minute peel strength of less than 0.10 N/20mm; and having a 48-hour peel strength of 0.05 N/20mm or greater, having a 30-minute peel strength of less than 0.10 N/20mm; and having a 48-hour peel strength of 0.05 N/20mm or greater,
Component of a kitchen appliance with a coupling for fastening a tool and a pot-shaped sieve part with a pot base provided with through openings and a pot casing surrounding the pot base in the manner of a flange, wherein the sieve part has sharp cutting edges on an interior, which are aligned essentially radially to an axis of the coupling, wherein the cutting edges are distributed non-uniformly or uniformly on the interior of the sieve part, so that the cutting edges divide the pot base in a fan-shaped manner into segments which are twisted with respect to one another, wherein the cutting edges are configured to catch and break up the item to be processed and to convey it through the through openings in the pot base and cut-outs in the pot casing onto an exterior of the sieve part, characterised in that the sharp cutting edges on the interior of the sieve part are formed in the injection moulding method.
Magnetic trip device of a thermal magnetic circuit breaker, wherein the magnetic trip device has at least - an armature locator moveable arranged around a pin in order to adjust a magnetic field area, - an armature element fixed on a lower surface of said armature locator in order to interact with a yoke, which is arranged near a current conductive element for conducting electric energy, wherein the magnetic trip device has an adjustment element arranged between a spring element and the yoke, wherein the spring element surrounding at least a part of the pin is arranged between the armature element and the yoke, characterized in that the adjustment element has at least one protrusion (80.1) of the current conductive element, and a contacting area (60.2) extending at least partially rectangular from the protrusion area (60.1). - an armature locator moveable arranged around a pin in order to adjust a magnetic field area, - an armature element fixed on a lower surface of said armature locator in order to interact with a yoke, which is arranged near a current conductive element for conducting electric energy, wherein the magnetic trip device has an adjustment element arranged between a spring element and the yoke, wherein the spring element surrounding at least a part of the pin is arranged between the armature element and the yoke,
System for automatic determination of welding parameters for automated friction stir welding are variants thereof, comprising a welding conditions assessing device and a welding parameters determining device in data communication with each other, characterized in that said welding conditions assessing device comprises - joint thickness measuring means, - base material properties determining means, comprising a chemical composition determining device, a hardness test device for assessing the metallurgical state of said base material, - at least one data processing means for receiving a manual data entering of the joint type and weld path and for processing the latter data and the information from said joint thickness measuring means and said base material properties determining means in order to obtain the mechanical properties of said base material to be welded and send the information to said welding parameters determining device and wherein said welding parameters determining device comprises electronic means to compute and output suitable welding parameters for welding said base material. - joint thickness measuring means, - base material properties determining means, comprising a chemical composition determining device, a hardness test device for assessing the metallurgical state of said base material, - at least one data processing means for receiving a manual data entering of the joint type and weld path and for processing the latter data and the information from said joint thickness measuring means and said base material properties determining means in order to obtain the mechanical properties of said base material to be welded and send the information to said welding parameters determining device
A method for manufacturing a spider silk thread on basis of a spider silk filament in the manufacture of cosmetic, medical, textile or industrial applications, comprising the steps of: providing spider silk filament derived from genetically modified organisms; treating of the spider silk filament with at least one component selected from the group consisting of vitamins, hormones, antioxidants, chelating agents, antibiotics, preserving agents, fragrances, dyes, pigments, magnetic nanoparticles, nanocrystals, cell adhesion enhancers, thermal insulators, shrinkage agents and cosmetic, medical or dermatological active substances; characterised, in that for obtaining a better bonding of the proteins in the spider silk filament the spider silk filament is treated with a 0.4 wt.% potassium aluminum sulfate KAl(SO 4) 2 ·12H 2 O solution, wherein the treatment comprises the following subsequent steps: bringing the potassium aluminum sulfate solution to its boiling point, cooling the potassium aluminum sulfate solution to a temperature of 21 °C, immersing the spider silk filament in the potassium aluminum sulfate solution for 24 hours, rinsing the spider silk filament thoroughly with water of 21 °C, passing the spider silk filament through a physiological saline solution 0.9 wt.% NaCl, drying the spider silk filament; twining, cabling or braiding of two or more spider silk filaments into the spider silk thread. providing spider silk filament derived from genetically modified organisms; treating of the spider silk filament with at least one component selected from the group consisting of vitamins, hormones, antioxidants, chelating agents, antibiotics, preserving agents, fragrances, dyes, pigments, magnetic nanoparticles, nanocrystals, cell adhesion enhancers, thermal insulators, shrinkage agents and cosmetic, medical or dermatological active substances; bringing the potassium aluminum sulfate solution to its boiling point, cooling the potassium aluminum sulfate solution to a temperature of 21 °C, immersing the spider silk filament in the potassium aluminum sulfate solution for 24 hours, rinsing the spider silk filament thoroughly with water of 21 °C, passing the spider silk filament through a physiological saline solution 0.9 wt.% NaCl, drying the spider silk filament; twining, cabling or braiding of two or more spider silk filaments into the spider silk thread.
A method for bundling acknowledgement/negative acknowledgment, ACK/NACK, feedback in a time division duplex long-term evolution, LTE, system, comprising bundling acknowledgement/negative acknowledgment, ACK/NACK, feedback determined for a plurality of subframes within a time window into at least two sets of feedback information based on differently timed bundling windows defined based on subframe types, characterised in that one bundling window covers system information block 1 configured downlink subframes or system information block 1 configured downlink subframes and special subframes and where another bundling window covers other downlink subframes.
A method for preparing a security or value document comprising a card body consisting of a plurality of plastic layers having a high softening temperature, in which is provided at least one cavity for later embedding at least one further module, wherein a) at least at one position between the plastic layers, a separating layer is arranged, the separating layer consisting of a silicone oil-containing ink, and the separating layer not being extended up to the border of the document, b) the plastic layers and the separating layer are laminated together, and c) thereafter, precisely above the separating layer, the desired cavity is produced by punching out, characterized by that at least one plastic layer is made of polycarbonate or polyethylene terephthalate. a) at least at one position between the plastic layers, a separating layer is arranged, the separating layer consisting of a silicone oil-containing ink, and the separating layer not being extended up to the border of the document, b) the plastic layers and the separating layer are laminated together, and c) thereafter, precisely above the separating layer, the desired cavity is produced by punching out, characterized by that at least one plastic layer is made of polycarbonate or polyethylene terephthalate.
A lyophilized daptomycin formulation comprising from 200mg to 600mg of daptomycin and the additive citric acid which, upon reconstitution in a pharmaceutically acceptable diluent, leads to a daptomycin concentration of from 20mg/mL to 100mg/mL and a citric acid concentration of from 25mM to 75mM.