mhurhangee/ep-ind-claims huggingface dataset:
A compound of the formula, or an isomer or pharmaceutically acceptable salt thereof, wherein, n is selected from the group consisting of 1, 2, and 3; R 1 is 4 to 6 membered heterocycloalkyl, which is optionally substituted by 1, 2 or 3 R a; R 2 is C 1-6 alkyl, which is optionally substituted by 1, 2 or 3 R b; R 3 is C 1-6 alkoxy, which is optionally substituted by 1, 2 or 3 R c; X 1 is selected from the group consisting of O, S and -NH-; L 1 is - m -; L 2 is -CRR-; m is selected from the group consisting of 1, 2, 3, and 4; R a, R b and R c are independently selected from the group consisting of H, F, Cl, Br, I, OH, NH 2, CN, and CH 3; each R is independently selected from the group consisting of H, F, Cl, Br, I, OH, NH 2, CN, and CH; the 4 to 6-membered heterocycloalkyl comprises 1, 2, 3 or 4 heteroatoms or heteroatom groups independently selected from the group consisting of -NH -, - O - S- and N; wherein the isomer thereof is a geometric or stereoisomeric isomer; and the sulfur atom with"*" is a chiral sulfur atom, which exists as a or single enantiomer or is riched in one of the enantiomers. n is selected from the group consisting of 1, 2, and 3; R 1 is 4 to 6 membered heterocycloalkyl, which is optionally substituted by 1, 2 or 3 R a; R 2 is C 1-6 alkyl, which is optionally substituted by 1, 2 or 3 R b; R 3 is C 1-6 alkoxy, which is optionally substituted by 1, 2 or 3 R c; X 1 is selected from the group consisting of O, S and -NH-; L 1 is - m -; L 2 is -CRR-; m is selected from the group consisting of 1, 2, 3, and 4; R a, R b and R c are independently selected from the group consisting of H, F, Cl, Br, I, OH, NH 2, CN, and CH 3; each R is independently selected from the group consisting of H, F, Cl, Br, I, OH, NH 2, CN, and CH; the 4 to 6-membered heterocycloalkyl comprises 1, 2, 3 or 4 heteroatoms or heteroatom groups independently selected from the group consisting of -NH -, - O - S- and N; wherein the isomer thereof is a geometric or stereoisomeric isomer; and the sulfur atom with"*" is a chiral sulfur atom, which exists as a or single enantiomer or is riched in one of the enantiomers.
Automatically controlled door arrangement as a floor door of an elevator installation, comprising: at least one door leaf which can be actively moved between an open and a closed position; a drive for moving the door leaf between the open and the closed position; a controller for controlling the drive; a sensor system for detecting people or objects in front of the door leaf; characterised in that the door arrangement comprises further: a data connection for data exchange with an external computer; and wherein the door arrangement is configured to: - receive and process signals from the sensor system in the controller, - send query data to the external computer via the data connection on the basis of the processed signals, - then receive instruction data provided by the external computer, and - control the drive of the door leaf taking into account the instruction data. at least one door leaf which can be actively moved between an open and a closed position; a drive for moving the door leaf between the open and the closed position; a controller for controlling the drive; a sensor system for detecting people or objects in front of the door leaf; characterised in that the door arrangement comprises further: a data connection for data exchange with an external computer; and wherein the door arrangement is configured to: - receive and process signals from the sensor system in the controller, - send query data to the external computer via the data connection on the basis of the processed signals, - then receive instruction data provided by the external computer, and - control the drive of the door leaf taking into account the instruction data. - receive and process signals from the sensor system in the controller, - send query data to the external computer via the data connection on the basis of the processed signals, - then receive instruction data provided by the external computer, and - control the drive of the door leaf taking into account the instruction data.
A leadless ECG measurement system for measuring of bio-potential electrical activity in a patient's body, comprising: at least one multi-contact bio-potential electrode assembly for attachment to the patient's body, said electrode assembly being formed of an electronic patch layer and a disposable electrode layer; said disposable electrode layer having a plurality of contact points for engagement with the patient's body and configuring the plurality of contact points to measure short-lead ECG signals, defined as signals generated from bio-potential measurements across said plurality of contact points, in response to electrical activity in the patient's body; and a processing unit being provided and configured to produce a transfer function which computes estimated long-lead ECG signals, defined as signals generated from bio-potential measurements across any other contact points on the patient's body, based on the measured short-lead ECG signals from said plurality of contact points; characterized in that said processing unit is configured to employ a system identification method for defining said transfer function and that said transfer function is described by a linear state-space model. at least one multi-contact bio-potential electrode assembly for attachment to the patient's body, said electrode assembly being formed of an electronic patch layer and a disposable electrode layer; said disposable electrode layer having a plurality of contact points for engagement with the patient's body and configuring the plurality of contact points to measure short-lead ECG signals, defined as signals generated from bio-potential measurements across said plurality of contact points, in response to electrical activity in the patient's body; and a processing unit being provided and configured to produce a transfer function which computes estimated long-lead ECG signals, defined as signals generated from bio-potential measurements across any other contact points on the patient's body, based on the measured short-lead ECG signals from said plurality of contact points; characterized in that said processing unit is configured to employ a system identification method for defining said transfer function and that said transfer function is described by a linear state-space model.
A fluid pump system comprising: a housing including a first end and a second end, the housing defining a first axis extending between the first end and the second end, characterized by the housing further including a wall extending at least partially around the first axis, the wall at least partially enclosing a chamber; a motor at least partially positioned within the chamber; a fan positioned proximate the first end of the housing, the fan generating air flow through the chamber; and a fluid conduit configured to be in fluid communication with a fluid reservoir, at least a portion of the fluid conduit positioned within the chamber and extending around a portion of the motor. a housing including a first end and a second end, the housing defining a first axis extending between the first end and the second end, characterized by the housing further including a wall extending at least partially around the first axis, the wall at least partially enclosing a chamber; a motor at least partially positioned within the chamber; a fan positioned proximate the first end of the housing, the fan generating air flow through the chamber; and a fluid conduit configured to be in fluid communication with a fluid reservoir, at least a portion of the fluid conduit positioned within the chamber and extending around a portion of the motor.
A WIRELESS FABRIC RECORDING CAP WITH SENSORIAL PROXIMITY AND VOICE CONTROL, characterised in that it comprises: a first removable module, located on the front of the said cap, which incorporates a high resolution micro-camera, a laser pointer, and a coupling LED; wherein the cap further comprises a second removable module, located in the upper part of the cap, where a Wi-Fi system, a battery, for energy storage, and a mini USB connector, for connecting the battery to an external energy source, as well as an internal memory for the storage of images are located; wherein the second removable module also contains a series of red, orange and green LED indicators; and wherein the cap further comprises a proximity sensor, located outside the second removable module and the first removable module. a first removable module, located on the front of the said cap, which incorporates a high resolution micro-camera, a laser pointer, and a coupling LED; wherein the cap further comprises a second removable module, located in the upper part of the cap, where a Wi-Fi system, a battery, for energy storage, and a mini USB connector, for connecting the battery to an external energy source, as well as an internal memory for the storage of images are located; wherein the second removable module also contains a series of red, orange and green LED indicators; and wherein the cap further comprises a proximity sensor, located outside the second removable module and the first removable module.
Method for coding at least one image (IC j) split into blocks, comprising, for a current block (B u) of K pixels to be coded, where K≥1, the steps of: - predicting the current block using at least one predictor block (BP opt) of K pixels, - determining a residual block of K pixels which represents the difference between the predictor block and the current block, - determining a set of Mi data, where i≥1 and 1≤M i <K, - coding the Mi data of the determined set of data, said coding method being characterized in that the set of Mi data is determined on the basis of a group (Gi) of pixel blocks containing a number Mi of blocks of K pixels which each represent a predetermined texture, by calculating pixel-by-pixel products of the residual block determined by each of the M i blocks of K pixels representing a predetermined texture, and then adding the calculated products, the group (Gi) of pixel blocks having been obtained prior to the coding by singular value decomposition or analysis of main components. - predicting the current block using at least one predictor block (BP opt) of K pixels, - determining a residual block of K pixels which represents the difference between the predictor block and the current block, - determining a set of Mi data, where i≥1 and 1≤M i <K, - coding the Mi data of the determined set of data,
Method for controlling a converter of a wind energy installation, which converter is connected to the rotor of a doubly-fed asynchronous generator, connected by its stator to an electrical grid, for feeding electrical power into the electrical grid, with the converter having a generator-side inverter connected to the rotor, a grid-side inverter and at least one converter regulator for controlling the currents emitted from at least one of the inverters, comprising the following method steps: - detection of a change in the electrical voltage which is present, in the emitted real currents and/or the emitted reactive currents at each inverter, - determination of whether the detected change corresponds to a predetermined change, and - changing the nominal values of the real currents to be emitted and/or the reactive currents to be emitted from the respective other inverter, if the detected change corresponds to a predetermined change. - detection of a change in the electrical voltage which is present, in the emitted real currents and/or the emitted reactive currents at each inverter, - determination of whether the detected change corresponds to a predetermined change, and - changing the nominal values of the real currents to be emitted and/or the reactive currents to be emitted from the respective other inverter, if the detected change corresponds to a predetermined change.
A process for the preparation of at least one of S-Rivaroxaban and R-Rivaroxaban comprising reacting, in the presence of a first base, a compound of Formula 9: with a compound of Formula 8: wherein R 4 is selected from the group consisting of: wherein G is OR 1, NR 2 R 3, or CX 3; R 1 is alkyl, substituted alkyl, aryl, substituted aryl, arylalkyl, or substituted aryl alkyl; R 2 and R 3 are either (a) two independent groups or (b) together form a single ring group with the N to which they are bonded; R 2 and R 3, when independent groups, are independently selected from the group consisting of: H, alkyl, substituted alkyl, aryl, substituted aryl, arylalkyl and substituted arylalkyl, R 2 and R 3, when together form a single ring group with the N to which they are bonded, are a heteroaryl ring; X is halogen; and L 2 is a halogen or sulfonyloxy group. R 4 is selected from the group consisting of: wherein G is OR 1, NR 2 R 3, or CX 3; R 1 is alkyl, substituted alkyl, aryl, substituted aryl, arylalkyl, or substituted aryl alkyl; R 2 and R 3 are either (a) two independent groups or (b) together form a single ring group with the N to which they are bonded; R 2 and R 3, when independent groups, are independently selected from the group consisting of: H, alkyl, substituted alkyl, aryl, substituted aryl, arylalkyl and substituted arylalkyl, R 2 and R 3, when together form a single ring group with the N to which they are bonded, are a heteroaryl ring; X is halogen; and L 2 is a halogen or sulfonyloxy group. G is OR 1, NR 2 R 3, or CX 3; R 1 is alkyl, substituted alkyl, aryl, substituted aryl, arylalkyl, or substituted aryl alkyl; R 2 and R 3 are either (a) two independent groups or (b) together form a single ring group with the N to which they are bonded; R 2 and R 3, when independent groups, are independently selected from the group consisting of: H, alkyl, substituted alkyl, aryl, substituted aryl, arylalkyl and substituted arylalkyl, R 2 and R 3, when together form a single ring group with the N to which they are bonded, are a heteroaryl ring; X is halogen; and L 2 is a halogen or sulfonyloxy group.
An agricultural working machine comprising at least one optical sensor means (3, 24), an image processing system, as well as a regulation and control device, wherein the at least one optical sensor means (2, 24) is configured to measure in anticipation an environment in the forefield of the working machine, wherein the image processing system is configured to detect the appearance of one or more obstacles in at least one obstacle region located in the environment in the forefield of the working machine by means of image analysis, characterized in that - the regulation and control device is configured to control working illumination comprising a plurality of light sources, and - the regulation and control device is configured to produce control signals which control an orientation of at least one of the light sources associated with the working machine which produces at least one bundled light beam consisting of visible light in order to orientate the at least one light beam onto the identified obstacle region. - the regulation and control device is configured to control working illumination comprising a plurality of light sources, and - the regulation and control device is configured to produce control signals which control an orientation of at least one of the light sources associated with the working machine which produces at least one bundled light beam consisting of visible light in order to orientate the at least one light beam onto the identified obstacle region.
Counter bearing sleeve for a profiled tube (4, 5) having at least one undercut longitudinal groove, with a through opening extending in an axial direction for feeding through a connecting screw, with an external self-tapping or thread-forming securing region, which has at least two securing sections (10, 11, 12) distributed around the circumference and spaced apart from one another in circumferential direction, characterized in that each securing section (10, 11, 12) has at least two tapping ridges adjacent to one another in axial direction which are offset in the insertion direction, so that when the counter bearing sleeve is screwed into a longitudinal groove of the profiled tube (4, 5) the tapping ridges cut successively into a groove base and at least one groove flank of the longitudinal groove.
A method of a terminal in a communication system including a wireless local area network, WLAN, access point, AP, the method comprising: receiving, from a base station, a control message including control information, wherein the control information is related to move traffic to the WLAN AP while the terminal is in a connection state with the base station; receiving, from the WLAN AP, traffic based on the control information while the terminal is in the connection state with the base station; maintaining a configuration based on the control information, in case that the terminal transitions to an idle state with the base station; and releasing the configuration, in case that a connection with another base station is setup. receiving, from a base station, a control message including control information, wherein the control information is related to move traffic to the WLAN AP while the terminal is in a connection state with the base station; receiving, from the WLAN AP, traffic based on the control information while the terminal is in the connection state with the base station; maintaining a configuration based on the control information, in case that the terminal transitions to an idle state with the base station; and releasing the configuration, in case that a connection with another base station is setup.
An apparatus for pointing spatial coordinates by a pointing tip, comprising a movable hand-held probe, having said pointing tip, and a portable base unit provided with a rotatably supported elongated arm arranged to rotate in two degrees of freedom, wherein said hand-held probe connects to said portable base unit by means of a cord or a wire via said elongated arm and wherein said base unit is provided with sensors arranged for measuring length or a change in length of said cord or said wire and rotation of said arm in said two degrees of freedom, and a computer-controlled processing means arranged for processing measuring signals delivered by said sensors into position data of said hand-held probe, characterized in that said hand-held probe further comprises orientation means arranged for determining data relating to orientation of said hand-held probe, and interface means arranged for exchanging said orientation data with said computer-controlled processing means, and wherein said computer-controlled processing means is further arranged for processing said measuring signals and orientation data into said spatial coordinates of said pointing tip of said hand-held probe.
A lens for distribution of light from a light emitter having an emitter axis and defining an emitter plane, comprising: an emitter-adjacent base end forming an opening to an inner cavity configured for surrounding the emitter; and an inner-cavity surface including (a) a cross-sectionally concave axis-adjacent first inner region configured for refracting emitter light rays away from the axis, (b) a cross-sectionally convex second inner region spaced from the first inner region and configured for refracting emitter light rays toward the axis, characterized in that the inner-cavity surface further includes (c) a cross-sectionally linear middle inner region joining and cross-sectionally asymptotical to the first and second inner regions (21, 22), the middle inner region being positioned with respect to the emitter to refract light away from the axis by progressively lesser amounts at positions progressively closer to the second inner region; and in that the lens further comprises an outer surface configured for refracting the light from each of the inner (21, 22, 23) regions. an emitter-adjacent base end forming an opening to an inner cavity configured for surrounding the emitter; and an inner-cavity surface including (a) a cross-sectionally concave axis-adjacent first inner region configured for refracting emitter light rays away from the axis, (b) a cross-sectionally convex second inner region spaced from the first inner region and configured for refracting emitter light rays toward the axis,
An aluminum alloy, comprising: from 0.7 wt. % to 1.5 wt. % Mg; from 0.25 wt. % to 0.45 wt. % Si; from 0.01 wt. % to 1.0 wt. % Fe; from 0.01 wt. % to 0.5 wt. % Cu; from 0.01 wt. % to 0.5 wt. % Mn; from 0.005 wt. % to 0.3 wt. % Cr; from 0.01 wt. % to 0.25 wt. % Ti; up to 0.4 wt. % Zn; up to 0.20 wt. % impurities; and remainder Al, wherein the Mg and Si are present in a ratio of from 5:1 to 2:1 of Mg to Si by weight. from 0.7 wt. % to 1.5 wt. % Mg; from 0.25 wt. % to 0.45 wt. % Si; from 0.01 wt. % to 1.0 wt. % Fe; from 0.01 wt. % to 0.5 wt. % Cu; from 0.01 wt. % to 0.5 wt. % Mn; from 0.005 wt. % to 0.3 wt. % Cr; from 0.01 wt. % to 0.25 wt. % Ti; up to 0.4 wt. % Zn; up to 0.20 wt. % impurities; and remainder Al, wherein the Mg and Si are present in a ratio of from 5:1 to 2:1 of Mg to Si by weight.
A growth hormone secretagogue for use for treating cancer in a subject, wherein the growth hormone secretagogue is represented by the structural formula III or a pharmaceutically acceptable salt, solvate or hydrate thereof.
Method for preparing a vinylphenyl sulfonate of the formula: in which R 1 is C 1 -C 6 -alkyl, phenyl, 4-methylphenyl or benzyl, and R 2 is halogen or methyl, characterized in that (a) a compound of the formula is reacted with an activator in the presence of a base to give a compound of the formula wherein one or more compounds are used as activator selected from the group consisting of thionyl chloride, phosgene, diphosgene, triphosgene, thiophosgene and chloroformic esters, and (b) the compound of the formula is reacted in the presence of a base with a compound of the formula R 1 -SO 2 -R 3, where R 3 is F, Cl, Br or OSO 2 R 1 and R 1 is as defined in formula, to give the vinylphenyl sulfonate of the formula. (a) a compound of the formula is reacted with an activator in the presence of a base to give a compound of the formula wherein one or more compounds are used as activator selected from the group consisting of thionyl chloride, phosgene, diphosgene, triphosgene, thiophosgene and chloroformic esters, and (b) the compound of the formula is reacted in the presence of a base with a compound of the formula R 1 -SO 2 -R 3,
A method for wireless communication performed by an interfering base station, comprising: obtaining an indication of a terminal observing interference from the interfering base station and communicating with a serving base station; reserving frequency resources for a predetermined time period based on a predetermined order to facilitate communication between the serving base station and the terminal; and reducing interference on the reserved frequency resources by the interfering base station, wherein the reducing includes avoiding transmitting on the reserved frequency resources by the interfering base station or reducing transmit power of the interfering base station on the reserved frequency resources to obtain a target interference level for the terminal. obtaining an indication of a terminal observing interference from the interfering base station and communicating with a serving base station; reserving frequency resources for a predetermined time period based on a predetermined order to facilitate communication between the serving base station and the terminal; and reducing interference on the reserved frequency resources by the interfering base station, wherein the reducing includes avoiding transmitting on the reserved frequency resources by the interfering base station or reducing transmit power of the interfering base station on the reserved frequency resources to obtain a target interference level for the terminal.