mhurhangee/ep-ind-claims huggingface dataset:
A compound represented by: wherein R 25 is C 7-10 alkylene substituted on the terminal end by -COOH, -C -O-Me, or -C -Et; and pharmaceutically acceptable salts or stereoisomers thereof. R 25 is C 7-10 alkylene substituted on the terminal end by -COOH, -C -O-Me, or -C -Et; and pharmaceutically acceptable salts or stereoisomers thereof.
A compound having Formula: or pharmaceutically acceptable salts thereof; wherein Wis A 1 and A 4 are independently C; each A 2 and A 3 is C; R 1 and R 2 together form an optionally substituted 5-6 membered aryl, or heteroaryl or heterocyclic ring comprising 1-3 nitrogen atoms; R 3 is SO 2 R 12, SO 2 NH 2, SO 2 NRR 12, CONRR 12, CO 1-2 R 12, or cyano; R 5, R 5, R 7 and R 10 are independently H; R is H or C 1-6 alkyl; R 6 is OR 12; R 8 and R 9 are independently C 1-6 alkyl, C 2-6 alkenyl, C 2-6 alkynyl, halo or X, or one of R 8 and R 9 is H; and provided one of R 8 and R 9 is X; X is (CR 2) q Y, cyano, C O 0-1 R 12, CONR(R 12), CONR(CR 2)pNR(R 12), CONR(CR 2) p OR 12, CONR(CR 2) p SR 12, CONR(CR 2) p S 1-2 R 12 or (CR 2) 1-6 NR(CR 2) p OR 12; Y is an optionally substituted 3-12 membered carbocyclic ring, a 5-12 membered aryl, or a 5-12 membered heteroaryl or heterocyclic ring comprising N, O and/or S and attached to A 2 or A 3 or both via a carbon atom of said heteroaryl or heterocyclic ring when q in (CR 2) q Y is 0; R 12 is C 1-6 alkyl; and n is 0; and p and q are independently 0-4 wherein the optional substituent(s) in each optionally substituted group are selected from C 1-6 alkyl, C 2-6 alkenyl or C 3-6 alkynyl, each of which may be optionally halogenated or optionally having a carbon that may be replaced or substituted with N, S, O, or a combination thereof; halo, amino, amidino, C 1-6 alkoxy, hydroxyl, methylenedioxy, carboxy; C 1-8 alkylcarbonyl, C 1-8 alkoxycarbonyl, carbamoyl, C 1-8 alkylcarbamoyl, sulfamoyl, cyano, oxo, nitro, or a carbocyclic ring, heterocyclic ring, aryl or heteroaryl. Wis A 1 and A 4 are independently C; each A 2 and A 3 is C; R 1 and R 2 together form an optionally substituted 5-6 membered aryl, or heteroaryl or heterocyclic ring comprising 1-3 nitrogen atoms; R 3 is SO 2 R 12, SO 2 NH 2, SO 2 NRR 12, CONRR 12, CO 1-2 R 12, or cyano; R 5, R 5, R 7 and R 10 are independently H; R is H or C 1-6 alkyl; R 6 is OR 12; R 8 and R 9 are independently C 1-6 alkyl, C 2-6 alkenyl, C 2-6 alkynyl, halo or X, or one of R 8 and R 9 is H; and provided one of R 8 and R 9 is X; X is (CR 2) q Y, cyano, C O 0-1 R 12, CONR(R 12), CONR(CR 2)pNR(R 12), CONR(CR 2) p OR 12, CONR(CR 2) p SR 12, CONR(CR 2) p S 1-2 R 12 or (CR 2) 1-6 NR(CR 2) p OR 12; Y is an optionally substituted 3-12 membered carbocyclic ring, a 5-12 membered aryl, or a 5-12 membered heteroaryl or heterocyclic ring comprising N, O and/or S and attached to A 2 or A 3 or both via a carbon atom of said heteroaryl or heterocyclic ring when q in (CR 2) q Y is 0; R 12 is C 1-6 alkyl; and n is 0; and p and q are independently 0-4 wherein the optional substituent(s) in each optionally substituted group are selected from C 1-6 alkyl, C 2-6 alkenyl or C 3-6 alkynyl, each of which may be optionally halogenated or optionally having a carbon that may be replaced or substituted with N, S, O, or a combination thereof; halo, amino, amidino, C 1-6 alkoxy, hydroxyl, methylenedioxy, carboxy; C 1-8 alkylcarbonyl, C 1-8 alkoxycarbonyl, carbamoyl, C 1-8 alkylcarbamoyl, sulfamoyl, cyano, oxo, nitro, or a carbocyclic ring, heterocyclic ring, aryl or heteroaryl.
Method for detecting and characterising defects in a heterogeneous material by ultrasound, comprising the following steps: - emission of ultrasounds from an ultrasonic emitting transducer (14, 24) placed against the material, - acquisition by an ultrasonic receiving transducer (15, 25) at different positions with respect to said material of a plurality of temporal signals representing the amplitude of the ultrasounds propagated in the material as a function of time for a position of the ultrasonic receiving transducer, characterised in that the method comprises the steps of: - determination of a temporal function representing a spatially-average power of the temporal signals corresponding to different positions of the ultrasonic receiving transducer (15, 25), the temporal function representing the spatially-average power of the temporal signals being of the general formula: f t = β ∑ z | x z, t − m t | α γ with α, β and γ non-zero, x(z,t) the temporal signal representing the amplitude of the sound propagated in the material as a function of time for a position z of the ultrasonic receiving transducer, and m(t) a function of time, - normalisation of the temporal signals by means of said temporal function to obtain normalised temporal signatures, - detection and characterisation of the defects of the material based on said normalised temporal signals. - emission of ultrasounds from an ultrasonic emitting transducer (14, 24) placed against the material, - acquisition by an ultrasonic receiving transducer (15, 25) at different positions with respect to said material of a plurality of temporal signals representing the amplitude of the ultrasounds propagated in the material as a function of time for a position of the ultrasonic receiving transducer, - determination of a temporal function representing a spatially-average power of the temporal signals corresponding to different positions of the ultrasonic receiving transducer (15, 25), the temporal function representing the spatially-average power of the temporal signals being of the general formula: f t = β ∑ z | x z, t − m t | α γ with α, β and γ non-zero, x(z,t) the temporal signal representing the amplitude of the sound propagated in the material as a function of time for a position z of the ultrasonic receiving transducer, and m(t) a function of time, - normalisation of the temporal signals by means of said temporal function to obtain normalised temporal signatures, - detection and characterisation of the defects of the material based on said normalised temporal signals.
A printed circuit board soldered using a solder jet flow, comprising: a piezoelectric element including a primary side electrode pair and a secondary side electrode for outputting a voltage, characterized in that the primary side electrode pair is coupled by a electrically conductive resistor; and a slit ( 610A; 610B; 610C) is formed in the printed circuit board at a position shifted from arrangement positions of the primary side electrode pair of said piezoelectric elementwherein the slit ( 610A; 610B; 610C) is arranged at a position different from a position facing the conductive resistor between a position facing said primary side electrode pair and a position facing the secondary side electrode. a piezoelectric element including a primary side electrode pair and a secondary side electrode for outputting a voltage, characterized in that the primary side electrode pair is coupled by a electrically conductive resistor; and a slit ( 610A; 610B; 610C) is formed in the printed circuit board at a position shifted from arrangement positions of the primary side electrode pair of said piezoelectric elementwherein the slit ( 610A; 610B; 610C) is arranged at a position different from a position facing the conductive resistor between a position facing said primary side electrode pair and a position facing the secondary side electrode.
Money item dispensing apparatus for a money item-operated machine, the apparatus comprising: a money item store; a money item receptacle; means for feeding a money item from the money item store into the receptacle (32, 28); an outlet motor means for moving the money item in the receptacle to a position associated with the outlet; and means (34,101) for ejecting the money item from the receptacle through the outlet; characterised by a gate arrangement (103, 108) operable to direct the money item after passing the outlet along either a first path to a money item return opening for a user to collect or a second path to an opening for a cashbox, the second path comprising a purge chute (104, 105) for purging money items in the money item dispensing apparatus. a money item store; a money item receptacle; means for feeding a money item from the money item store into the receptacle (32, 28); an outlet motor means for moving the money item in the receptacle to a position associated with the outlet; and means (34,101) for ejecting the money item from the receptacle through the outlet;
A method for enhancing a proximity warning sound characterized by the steps of: determining an indicator of a distance between a first object and a second object; and generating a proximity warning sound including a reverberation mimicking component that includes a reverberation tail components having a tail length indicative of the proximity of the first object to the second object responsive to a determined distance indicator; where the reverberation mimicking component included in the proximity warning sound is indicative of the determined distance indicator. determining an indicator of a distance between a first object and a second object; and generating a proximity warning sound including a reverberation mimicking component that includes a reverberation tail components having a tail length indicative of the proximity of the first object to the second object responsive to a determined distance indicator; where the reverberation mimicking component included in the proximity warning sound is indicative of the determined distance indicator.
A method of performing channel access at a specific station in a wireless communication system, the method comprising: receiving, at the specific station from an access point, a beacon frame including information on channel access interval assigned to each group of stations (220, 230), wherein the specific station is allowed to access a channel within a channel access interval assigned to a specific station group including the specific station; transmitting (S221a; S3510), at the specific station, a poll frame to the access point; and receiving (S231; S3540), at the specific station from the access point, a response frame in response to the poll frame, the response frame including a channel access start offset value for the specific station, and determining, at the specific station, a channel access interval for the specific station based on the channel access start offset included in the response frame. receiving, at the specific station from an access point, a beacon frame including information on channel access interval assigned to each group of stations (220, 230), wherein the specific station is allowed to access a channel within a channel access interval assigned to a specific station group including the specific station; transmitting (S221a; S3510), at the specific station, a poll frame to the access point; and receiving (S231; S3540), at the specific station from the access point, a response frame in response to the poll frame, the response frame including a channel access start offset value for the specific station, and determining, at the specific station, a channel access interval for the specific station based on the channel access start offset included in the response frame.
A display device for a vehicle, comprising: a first frame; a second frame configured to be movable in a first direction with respect to the first frame; a first roller configured to be spaced apart from the first frame; a second roller configured to be rotatably coupled to the second frame and move in the first direction in accordance with movement of the second frame; a flexible display configured to be partially wound around the second roller and bent by the second roller and have one end portion fixed to the first frame; a moving part configured to move the second roller in the first direction; and a guider configured to guide the movement of the moving part, wherein the flexible display is provided such that an externally exposed area on a front surface is increased as a distance between the first roller and the second roller is increased, characterized in that the moving part comprises: a moving plate configured to have one end portion which is coupled to the second frame and move in the first direction as the second roller moves in the first direction; and a chain configured to have one end portion coupled to the moving plate, be bent by the first roller, and support at least a part of a rear surface of the flexible display. a first frame; a second frame configured to be movable in a first direction with respect to the first frame; a first roller configured to be spaced apart from the first frame; a second roller configured to be rotatably coupled to the second frame and move in the first direction in accordance with movement of the second frame; a flexible display configured to be partially wound around the second roller and bent by the second roller and have one end portion fixed to the first frame; a moving part configured to move the second roller in the first direction; and a guider configured to guide the movement of the moving part, wherein the flexible display is provided such that an externally exposed area on a front surface is increased as a distance between the first roller and the second roller is increased, characterized in that the moving part comprises: a moving plate configured to have one end portion which is coupled to the second frame and move in the first direction as the second roller moves in the first direction; and a chain configured to have one end portion coupled to the moving plate, be bent by the first roller, and support at least a part of a rear surface of the flexible display. a moving plate configured to have one end portion which is coupled to the second frame and move in the first direction as the second roller moves in the first direction; and a chain configured to have one end portion coupled to the moving plate, be bent by the first roller, and support at least a part of a rear surface of the flexible display.
An image processing apparatus comprising: a controller configured to transfer image data having a plurality of color components; a first processing module configured to receive the image data transferred from the controller, and execute image processing; and a second processing module configured to receive the image data transferred from the controller via the first processing module, and execute image processing on the image data, characterized in that the image processing apparatus is further configured such that processed data obtained by the first processing module by performing the image processing on the received image data is transferred to the controller, processed data obtained by the second processing module by performing the image processing on the image data received via the first processing module is transferred to the controller via the first processing module, and the number of color components as targets of the image processing to be executed by the first processing module is smaller than the number of color components as targets of the image processing to be executed by the second processing module. a controller configured to transfer image data having a plurality of color components; a first processing module configured to receive the image data transferred from the controller, and execute image processing; and a second processing module configured to receive the image data transferred from the controller via the first processing module, and execute image processing on the image data, characterized in that the image processing apparatus is further configured such that processed data obtained by the first processing module by performing the image processing on the received image data is transferred to the controller, processed data obtained by the second processing module by performing the image processing on the image data received via the first processing module is transferred to the controller via the first processing module, and the number of color components as targets of the image processing to be executed by the first processing module is smaller than the number of color components as targets of the image processing to be executed by the second processing module.
An adenovirus expressing an E1B55kD protein and an E4orf6 protein prior to an E1A12S protein, wherein the adenovirus comprises at least one nucleic acid coding for a E1A12S protein, wherein the expression of the E1A12S protein is under the control of a promoter and is controlled by said promoter, wherein the promoter is different from the promoter controlling the expression of the protein in a wild type adenovirus, wherein the promoter is selected from the group consisting of tumor-specific promoters, organ-specific promoters, tissue-specific promoters, heterologous promoters and adenoviral promoters, wherein the adenoviral promoter is different from the E1A promoter, wherein the adenovirus is replication-deficient, but replicates in cells comprising YB-1 in the cell nulceus or comprising deregulated YB-1 in the cytoplasma, wherein deregulated YB-1 is one which is present in a form which is quantitatively different from the one in a non-tumor cell.
A method, implemented by a receiving device, the method comprising: receiving, from a proxy server, a promise frame indicating that the proxy server will deliver a packet to the receiving device from a sending device later; sending an acknowledgement of the packet to the sending device via the proxy server; receiving the packet from the proxy server after having sent the acknowledgement of the packet to the sending device via the proxy server. receiving, from a proxy server, a promise frame indicating that the proxy server will deliver a packet to the receiving device from a sending device later; sending an acknowledgement of the packet to the sending device via the proxy server; receiving the packet from the proxy server after having sent the acknowledgement of the packet to the sending device via the proxy server.
A method of injection molding comprising: continuously feeding a supply of a first molten polymeric material to a first nozzle in selective communication with a plurality of mold cavities (220a, 220b, 220c) via first feed channels; continuously feeding a supply of a second molten polymeric material to a second nozzle in selective communication with the plurality of mold cavities via second feed channels, characterized by providing the first and second feed channels with valves; detecting pressure of molten polymeric material in each of the mold cavities; and based on the detected pressure, adjusting the pressure in an individual mold by means of the valve in the respective feed channel. continuously feeding a supply of a first molten polymeric material to a first nozzle in selective communication with a plurality of mold cavities (220a, 220b, 220c) via first feed channels; continuously feeding a supply of a second molten polymeric material to a second nozzle in selective communication with the plurality of mold cavities via second feed channels, characterized by providing the first and second feed channels with valves; detecting pressure of molten polymeric material in each of the mold cavities; and based on the detected pressure, adjusting the pressure in an individual mold by means of the valve in the respective feed channel.
A portable terminal comprising: a first conductor (641,741) patterned on a board (636,736); a second conductor (642,742) patterned on an outer periphery of the first conductor; a metal dome (643,743) electrically connected to the second conductor and transformed responsive to a key being pressed so as to contact the first conductor; and an elastic supporting member (660,760) configured to support a supported point of the metal dome in a state of being supported by the second conductor, and elastically move the support point of the metal dome when the key is pressed, characterized in that the first and second conductors (641, 642) are disposed at a recess portion recessed into the board by a predetermined depth. a first conductor (641,741) patterned on a board (636,736); a second conductor (642,742) patterned on an outer periphery of the first conductor; a metal dome (643,743) electrically connected to the second conductor and transformed responsive to a key being pressed so as to contact the first conductor; and an elastic supporting member (660,760) configured to support a supported point of the metal dome in a state of being supported by the second conductor, and elastically move the support point of the metal dome when the key is pressed, characterized in that the first and second conductors (641, 642) are disposed at a recess portion recessed into the board by a predetermined depth.
A feed air wall bushing, having a duct with an outside end and an inside end, for installation in a wall through which the bushing is to pass and which has an outside and an inside, the duct being formed at least partially by an inside end section, a central section and an outside end section of the feed air wall bushing, characterised in that at least one flap (31, 32) or slat is provided in the outside end section, by means of which flap or slat the duct for the feed air can be closed, and an actuation device that actuates the at least one flap or slat is arranged in and/or on the inside end section, wherein the actuation device is mechanically coupled to the flap(s) (31, 32) or slat(s) inside the duct, wherein the central section effects thermal decoupling of the outside end section from the inside end section.