bluuebunny/crossref_metadata_2025_split huggingface dataset:
Porocytosis: A transient pore array secretes the neurotransmitter packet
Authors: Kriebel Mahlon E. , Keller Bruce , Silver Robert B. , Pappas George D. 
Published: January 2005

AbstractThe porocytosis hypothesis is based on the arrayed nature of synaptic vesicles which forms the anatomical functional unit of secretion. The presynaptic array and the postsynaptic array of receptors form a synaptomere which is the unit of transmission. A transient increase in calcium ions, triggered by an action potential, activates all pores of the array to pulse transmitter. The array insures transmission while permitting a frequency dependent amount of secretion. Therefore the amount of secretion is variable which permits plasticity. Secretion from the array has the property of immediate synaptic plasticity whereas a change in array size would change synaptic strength. The robust nature of the array insures fidelity of transmission, a frequency dependent dynamic signature of transmission giving the property of immediate plasticity; and, a change in array size yields a change in synaptic strength for long term reliability. Anat Rec (Part B: New Anat) 282B:38–41, 2005. © 2005 Wiley‐Liss, Inc.
Non‐Thiol Farnesyltransferase Inhibitors: Utilization of the Far Aryl Binding Site by Arylthienylacryloylaminobenzophenones
Authors: Mitsch Andreas , Altenkämper Mirko , Sattler Isabel , Schlitzer Martin 
Published: January 2005

AbstractWe recently described two novel aryl binding sites of farnesyltransferase. The 4‐ and 5‐arylsubstituted thienylacryloyl moieties turned out as appropriate substituents for our benzophenone‐based AAX—peptidomimetic capable for occupying the far aryl binding site.
Anti‐inflammatory and Gastro Sparing Activity of Some New Indomethacin Derivatives
Authors: Amir Mohd. , Kumar Shikha 
Published: January 2005

AbstractIndomethacin is a non‐steroidal anti‐inflammatory drug but its use is associated with high degree of gastric toxicity therefore it is prescribed only in severe conditions. In order to reduce the gastric toxicity of indomethacin, various oxadiazole, triazole, thiadiazole and triazine derivatives have been synthesized. Out of thirteen cyclized derivatives, eleven were screened for anti‐inflammatory activity by Winter et al. method. Four compounds showed highly significant activity and were further tested for analgesic, ulcerogenic and lipid peroxidation activities. The tested compounds showed anti‐inflammatory activities in the range from about 32% to 85% as compared to that of indomethacin of about 96%. The compounds showing high anti‐inflammatory activity also exhibited reduction in severity index. These compounds also produced less malondialdehyde content in gastric mucosa than the standard drug indomethacin. The study showed that the compounds inhibited the induction of gastric mucosal lesions and it can be suggested from our results that their protective effects may be related to inhibition of lipid peroxidation in the gastric mucosa.
2, 3‐Bis(5‐alkyl‐2‐thiono‐1, 3, 5‐thiadiazin‐3‐yl) Propionic Acid: One‐Pot Domino Synthesis and Antimicrobial Activity
Authors: El Bialy Serry A. A. , Abdelal Ali M. , El‐Shorbagi Abdel‐Nasser , Kheira Samy M. M. 
Published: January 2005

AbstractIn a search for promising antibacterial and antifungal compounds, two new series of 2, 3‐bis(5‐alkyl‐2‐thiono‐1, 3, 5‐thiadiazin‐3‐yl)propionic acid 1 and their corresponding N, N‐dimethylpropionamide 6 have been synthesized. The reaction of 2, 3‐diaminopropionate 3, carbon disulfide, formaldehyde, and the appropriate alkyl amines furnished the title compound 1. N, N‐dimethylpropionamides 6 were obtained by the reaction of 1 with dimethyl amine in the presence of POCl3. The newly prepared compounds were screened in vitro against certain strains of Gram‐positive and Gram‐negative bacteria and compared with nalidixic acid and ciprofloxacin. Moreover, the title compounds were tested for their antifungal activity in vitro against Candida albicans, phytopathogenic, Penicillum expansum and Trichoderma hazianum, and aflatoxin‐producing Aspergillus flavus. These compounds exhibit varied activity against the tested pathogenic bacteria and remarkable inhibitory effects on growth or sporulation of some of the tested fungal species.
Synthesis and Antiparasitic Properties of New 4‐N‐Benzylamino‐4‐Hetarylbut‐1‐enes
Authors: Kouznetsov Vladimir V. , Castro Juliette Rivero , Puentes Cristian Ochoa , Stashenko Elena E. , Martínez Jairo René , Ochoa Carmen , Pereira David Montero , Ruiz Juan J. Nogal , Portillo Carlos Fernández , Serrano Susana Muelas , Barrio Alicia Gómez , Bahsas Alí , Amaro‐Luis Juan 
Published: January 2005

AbstractNew derivatives of 4‐N‐benzylamino‐4‐hetarylbut‐1‐ene containing a pyridyl nucleus were synthesized from benzylamines and pyridine aldehydes. N‐oxide derivatives were obtained from these homoallylamines. Study of the antiparasitic properties of obtained pyridine derivatives as well as of four related benzazepines previously described, was carried out using cytotoxicity assays against Trichomonas vaginalis and epimastigote form of Trypanosoma cruzi protozoa. Compounds showing activity against epimastigote T. cruzi were tested against the amastigote form; unspecific cytotoxicity against macrophages was also studied.
Synthesis of New Lipophilic Ipomeanol Analogues and Their Cytotoxic Activities
Authors: Krauss Jürgen , Unterreitmeier Doris 
Published: January 2005

AbstractAnalogues of the cytotoxic natural product (±)‐4‐ipomeanol (1) have been synthesized starting from furan‐3‐carbaldehyde and furan‐2‐carbaldehyde, followed by Grignard reaction and Sharpless dihydroxylation. The resulting alcohols were esterified with octanoyl chloride. The cytotoxic activities of the resulting compounds were determined in the MTT assay against a human leukaemia cell line (HL‐60).
Synthesis and Biological Evaluation of Tacrine‐Thiadiazolidinone Hybrids as Dual Acetylcholinesterase Inhibitors
Authors: Dorronsoro Isabel , Alonso Diana , Castro Ana , del Monte Maria , García‐Palomero Esther , Martínez Ana 
Published: January 2005

AbstractThe synthesis of tacrine‐thiadiazolidinone hybrids is described. These compounds are designed as dual acetylcholinesterase inhibitors binding simultaneously to the peripheral and catalytic sites of the enzyme. All tested compounds exhibit significant AChE inhibitory activity. Competition assays using propidium as reference of selective ligand for the peripheral anionic site on acetylcholinesterase indicates the influence of the designed compounds over the peripheral site. They can be considered as new leads in the optimization of Alzheimer's disease modifying agents.
Biotransformation of Desoxypeganine by Microsomal Enzymes of the Rabbit Liver
Authors: Illgner Sascha , Matusch Rudolf 
Published: January 2005

AbstractThe biotransformation of the anticholinergic quinazoline alkaloid Desoxypeganine is studied by means of aerobic incubation with the non‐induced supernatant obtained at 9000g from rabbit liver homogenates as enzyme source followed by an admixture of NADPH. The metabolites were identified by highperformance liquid chromatography, chemical ionisation mass spectrometry (LC‐CI MS) and electron impact mass spectrometry (LC‐EI MS) in comparison with synthetic reference compounds and typical ion fragments taken from literature data. C‐oxidation of Desoxypeganine to the major metabolite Pegenone was observed as well as the hydroxylation of the alicyclic ring. The incubation mixture followed Michaelis‐Menten kinetics characterised by Km = 5.8 × 10—5 mol L—1 and Vmax = 4.32 nmol Pegenone/min per mg protein or 3.37 nmol Pegenone/min per nmol CYP 450, respectively. These in vitro results demonstrate that the bioactive substance Desoxypeganine is easily oxidised to its ineffective metabolite Pegenone. This provokes a problem for correct dosage finding in formulations for the treatment of Alzheimer' disease and in the therapy of alcoholism and nicotine dependence.
Pharmacokinetics of 5‐fluorouracil in rats with diabetes mellitus induced by streptozotocin
Authors: Choi Young H. , Lee Ae K. , Bae Soo K. , Kim Sun O. , Lee Myung G. 
Published: January 2005

AbstractThe pharmacokinetic parameters of 5‐fluorouracil were compared after intravenous administration at a dose of 30 mg/kg to control Sprague–Dawley rats and to rats with diabetes mellitus induced by streptozotocin (DMIS). In DMIS rats, the area under the plasma concentration–time curve from time zero to time infinity (AUC) was significantly smaller (603 versus 909 µg min/ml) due to the significantly faster total body clearance (Cl; 47.8 versus 33.0 ml/min/kg). The faster Cl was due to the significantly faster renal (8.54 versus 4.02 ml/min/kg) and nonrenal (38.5 versus 28.7 ml/min/kg) clearances. In DMIS rats, the total amount of unchanged 5‐fluorouracil excreted in 24 h urine was significantly greater (34.1% versus 13.0% of intravenous dose) due to the urine flow rate‐dependent renal clearance of 5‐fluorouracil in rats (the greater the urine flow rate, the greater the urinary excretion of 5‐fluorouracil). Greater urinary excretion and a significantly smaller AUC resulted in a significantly faster Clr in DMIS rats. The faster Clnr in DMIS rats could be due to an increase in the expression and mRNA level of CYP1A1/2 in the rats. Copyright © 2005 John Wiley & Sons, Ltd.
Novel approach to quantify immobilized‐enzyme distributions
Authors: van Roon J. L. , Groenendijk E. , Kieft H. , Schroën C. G. P. H. , Tramper J. , Beeftink H. H. 
Published: January 2005

AbstractThe quantitative intraparticle enzyme distribution of Assemblase, an industrially employed polydisperse immobilized penicillin‐G acylase, was measured. Because of strong autofluorescence of the carrier, the generally applied technique of confocal scanning microscopy could not be used; light microscopy was our method of choice. To do so, Assemblase particles of various sizes were sectioned, labeled with antibodies specifically against the enzyme, and analyzed light microscopically. Image analysis software was developed and used to determine the intraparticle enzyme distribution, which was found to be heterogeneous, with most enzyme located in the outer regions of the particles. Larger particles showed steeper gradients than smaller ones. A mathematical representation of the intraparticle profiles, based on in‐stationary enzyme diffusion into the particles, was validated successfully for a broad range of particle sizes using data for volume‐averaged particle size and enzyme loading. The enzyme gradients determined in this work will be used as input for a physical model that quantitatively describes the complex behavior of Assemblase. Such a physical model will lead to identification of the current bottlenecks in Assemblase and can serve as a starting point for the design of improved biocatalysts that also may be based on intelligent use of enzyme gradients. © 2005 Wiley Periodicals, Inc.
Harderoporphyrin: a misnomer
Authors: Gorchein A. , Danton M. , Lim C. K. 
Published: January 2005

AbstractMore than 30 years ago it was reported that rodent Harderian glands contained a tricarboxylic acid porphyrin, which the authors named Harderoporphyrin. The recent finding in rat Harderian glands of the porphyrin glycoconjugate, protoporphyrin‐1‐O‐acyl‐β‐xyloside as a major component led to scrutiny of earlier publications. It became apparent that the results were flawed and that the conclusions were unsustainable. The procedural artefacts which led to the errors are discussed and their bases are demonstrated experimentally. Harderoporphyrin as originally defined never existed. Copyright © 2005 John Wiley & Sons, Ltd.
Hypervalency Avoided: Simple Substituted BrF3 and BrF5 Molecules. Structures, Thermochemistry, and Electron Affinities of the Bromine Hydrogen Fluorides HBrF2 and HBrF4.
Authors: Li Qianshu , Gong Liangfa , Xie Yaoming , Schaefer Henry F. III 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Covalently Bonded ∞1[Pt]‐ Chains in BaPt: Extension of the Zintl—Klemm Concept to Anionic Transition Metals?
Authors: Karpov Andrey , Nuss Juergen , Wedig Ulrich , Jansen Martin 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Synthesis and Structural Characterization of K0.33Gd0.67F2.33 (KGd2F7) and K0.31Gd0.69F1.84O0.27.
Authors: Gredin Patrick , Labeguerie Jessica , Pierrard Angelique , Vaulay Marie‐Josee , de Kozak Ariel 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Cation and Anion Disorder in New Cubic Rare Earth Carbonates Na2LiLn(CO3)3 (Ln: Eu—Er, Yb, Lu, Y); Synthesis, Crystal Structures, IR, Raman and NMR Characterizations.
Authors: Ali A. Ben , Maisonneuve V. , Houlbert S. , Silly G. , Buzare J. Y. , Leblanc M. 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Anion Ordering and Defect Structure in Ruddlesden—Popper Strontium Niobium Oxynitrides.
Authors: Tobias Gerard , Beltran‐Porter Daniel , Lebedev Oleg I. , Van Tendeloo Gustaaf , Rodriguez‐Carvajal Juan , Fuertes Amparo 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Structure and Physical Properties of Ln2Ge2In (Ln: La, Ce, Pr, Nd).
Authors: Zaremba Vasyl' I. , Kaczorowski Dariusz , Nychyporuk Galyna P. , Rodewald Ute Ch. , Poettgen Rainer 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Structural, Vibrational and Dielectric Properties of the New Mixed Solution K0.84(NH4)1.16SO4×Te (OH)6.
Authors: Ktari L. , Dammak M. , Hadrich A. , Cousson A. , Nierlich M. , Romain F. , Mhiri T. 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Synthesis and Characterization of a Novel Tantalum Chalcogen‐Rich Molecular Cluster with Square Planar Metal Core.
Authors: Sokolov Maxim N. , Gushchin Artyom L. , Virovets Alexandr V. , Peresypkina Eugenia V. , Kozlova Svetlana G. , Fedin Vladimir P. 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Isolation and Molecular Structure of a Monomeric, Tris[peroxotitanium(IV)]‐Substituted α‐Dawson Polyoxometalate Derived from the Tetrameric Anhydride Form Composed of Four Tris[titanium(IV)]‐Substituted α‐Dawson Substructures and Four Bridging Titanium(IV) Octahedral Groups.
Authors: Sakai Yoshitaka , Kitakoga Yuh , Hayashi Kunihiko , Yoza Kenji , Nomiya Kenji 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Chiral Phosphinooxazolidine Ligands for Palladium‐ and Platinum‐Catalyzed Asymmetric Diels—Alder Reactions.
Authors: Nakano Hiroto , Takahashi Kouichi , Okuyama Yuko , Senoo Chieko , Tsugawa Natsumi , Suzuki Yuichiro , Fujita Reiko , Sasaki Kazuo , Kabuto Chizuko 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Synthesis of 1‐Iodo‐1,2,3,4,4a,9a‐hexahydrocarbazole, 2a,3,4,5,5a,10a‐Hexahydrooxazolocarbazolium Iodide and 4‐Bromo‐1,2,3,4,4a,11b‐hexahydrodibenzoxazepine from N‐Benzoyl‐2‐(cyclohex‐2‐en‐1‐yl)aniline.
Authors: Gataullin Rail R. , Ishberdina Razida R. , Shitikova Olga V. , Spirikhin Leonid V. , Kazhanova Tat'jana V. , Abdrakhmanov Ildus B. 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
2‐(1,3,5‐Dithiazinan‐5‐yl)ethanol Heterocycles, Structure and Reactivity.
Authors: Galvez‐Ruiz Juan Carlos , Jaen‐Gaspar Javier C. , Castellanos‐Arzola Indira G. , Contreras Rosalinda , Flores‐Parra Angelina 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Thiopropenoylstannanes: The First Access to the Class of Thioacylstannanes.
Authors: Degl'Innocenti Alessandro , Capperucci Antonella , Nocentini Tiziano , Biondi Simona , Fratini Valentina , Castagnoli Giulio , Malesci Irene 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Nitrous Oxide Oxidation Catalyzed by Ruthenium Porphyrin Complex.
Authors: Tanaka Hirotaka , Hashimoto Kentaro , Suzuki Kyosuke , Kitaichi Yasunori , Sato Mitsuo , Ikeno Taketo , Yamada Tohru 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Selective Oxidation of Acetylenic 1,4‐Diols with Dioxiranes in Comparison with the Methyltrioxorhenium—Hydrogen Peroxide Oxidant.
Authors: D'Accolti Lucia , Fiorentino Michele , Fusco Caterina , Crupi Pasquale , Curci Ruggero 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Sustainable Transesterification of β‐Ketoesters Catalyzed by Amine Grafted on Silica Gel.
Authors: Hagiwara Hisahiro , Koseki Aiko , Isobe Kohei , Shimizu Ken‐ichi , Hoshi Takashi , Suzuki Toshio 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Selective Conversion of Epoxides to vic‐Halo Alcohols and Symmetrical or Unsymmetrical Dihalides by Triphenylphosphine/2,3‐Dichloro‐5,6‐dicyano‐1,4‐benzoquinone (DDQ) in the Presence of Quaternary Ammonium Halides.
Authors: Iranpoor Nasser , Firouzabadi Habib , Aghapour Ghasem , Nahid Azarmidokht 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Synthetic Studies on the Seven‐ and Eight‐Membered Rings by the Intramolecular Nozaki—Hiyama Reaction of the Allylic Phosphates.
Authors: Iwamoto Mitsuhiro , Miyano Masayuki , Utsugi Masayuki , Kawada Hatsuo , Nakada Masahisa 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Asymmetric Transfer Hydrogenation of α‐Aminoalkyl α′‐Chloromethyl Ketones with Chiral Rh Complexes.
Authors: Hamada Takayuki , Torii Takayoshi , Onishi Tomoyuki , Izawa Kunisuke , Ikariya Takao 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
New Selective Metal‐Free Oxidations of Primary Alcohols by HNO3 or HNO3 and O2, Catalyzed by Br2.
Authors: Minisci Francesco , Porta Ombretta , Recupero Francesco , Punta Carlo , Gambarotti Cristian , Pierini Monica , Galimberti Laura 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
1,3‐Phenylene‐bis‐(1H)‐tetrazole Pincer Ligand for Palladium‐Catalyzed Suzuki Cross‐Coupling Reactions of Arylhalides with Arylboronic Acids.
Authors: Gupta Arun Kumar , Rim Chul Yun , Oh Chang Ho 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Cyclopropyl‐ and Allyl‐Substituted Arenes in Reaction with Dinitrogen Tetroxide. Effect of Substrate Oxidation Potential on Reaction Direction.
Authors: Mochalov S. S. , Gazzaeva R. A. , Fedotov A. N. , Trofimova E. V. , Trushkov I. V. , Zefirov N. S. 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Reformatsky Reaction of Methyl α‐Bromoisobutyrate with Schiff Bases Derived from Salicylaldehyde and 2‐Hydroxynaphthalene‐1‐carbaldehyde.
Authors: Shchepin V. V. , Fotin D. V. , Vakhrin M. I. 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Reaction Between tert‐Butyl Isocyanide and 1,1,1‐Trifluoro‐4‐aryl‐butane‐2,4‐diones Synthesis of New Trifluoromethylated Furan Derivatives.
Authors: Mosslemin Mohammad H. , Yavari Issa , Anary‐Abbasinejad Mohammad , Nateghi Mohammad R. 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Synthesis of Fluorinated Dialkyl 1‐Aryl‐4‐alkoxy‐5‐oxo‐2,5‐dihydro‐1H‐pyrrole‐2,3‐dicarboxylates.
Authors: Yavari I. , Nasiri F. , Djahaniani H. 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Synthesis, Spectroscopic Studies and Crystal Structure of 5,5′‐Dimethoxy‐3,3′‐methanediyl‐bis‐indole as the Inhibitor of Cell Proliferation of Human Tumors.
Authors: Maciejewska Dorota , Niemyjska Maria , Wolska Irena , Wlostowski Marek , Rasztawicka Magdalena 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
5‐Amidinoindoles as Dual Inhibitors of Coagulation Factors IXa and Xa.
Authors: Batt Douglas G. , Qiao Jennifer X. , Modi Dilip P. , Houghton Gregory C. , Pierson Deborah A. , Rossi Karen A. , Luettgen Joseph M. , Knabb Robert M. , Jadhav P. K. , Wexler Ruth R. 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Rapid and Efficient Synthesis of Optically Active Pyrazoles under Solvent‐Free Conditions.
Authors: Yadav J. S. , Reddy B. V. S. , Satheesh G. , Lakshmi P. Naga , Kumar S. Kiran , Kunwar A. C. 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Studies on the Catalytic Hydrogenation of Baylis—Hillman Derivatives of Substituted Isoxazolecarbaldehydes. Unusual Retention of Isoxazole Ring During Pd—C‐Promoted hydrogenation of Baylis—Hillman Adducts.
Authors: Saxena R. , Singh V. , Batra S. 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Preparation of New Derivatives of Thiazole, Thiazolidine, and Thiazol‐2‐ylpyrazolo[3,4‐D]pyrimidine Sulfonamido Conjugates.
Authors: Khafagy Moustafa M. , El‐Maghraby Ahmed A. , Hassan Saber M. , Bashandy Mahmoud S. 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Synthesis and Complexing Properties of Alkyl (3‐Oxo‐2,3‐dihydrothiophen‐2‐ylidene)‐ and (4‐Oxothiazolidin‐5‐ylidene)acetate Derivatives.
Authors: Kosterina M. F. , Morzherin Yu. Yu. , Kramarenko O. A. , Berseneva V. S. , Matern A. I. , Tkachev A. V. , Bakulev V. A. 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Ortho‐Selective Nucleophilic Aromatic Substitution Reactions of Polyhaloanilines with Potassium/Sodium O‐Ethyl Xanthate: A Convenient Access to Halogenated 2(3H)‐Benzothiazolethiones.
Authors: Zhu Lei , Zhang Mingbao 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Synthesis of Trifluoroalkyl‐ and Fluoroaryl‐Substituted 4,5‐Dihydro‐1H‐1,2,4‐triazole‐5‐thiones
Authors: Vasil'eva E. B. , Sevenard D. V. , Khomutov O. G. , Kuznetsova O. A. , Karpenko N. S. , Filyakova V. I. 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Synthesis of 1‐Substituted 3‐Alkyl‐1,2,3‐triazol‐3‐ium‐5‐olates.
Authors: Nein Yu. I. , Polyakova A. Yu. , Morzherin Yu. Yu. , Savel'eva E. A. , Rozin Yu. A. , Bakulev V. A. 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Reaction of 1‐(o‐Aminophenyl)‐1,2,3‐triazole‐5‐thiols with Cyclizing Reagents.
Authors: Tarasov E. V. , Volkova N. N. , Morzherin Yu. Yu. , Bakulev V. A. 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Allosteric Potentiators of the Metabotropic Glutamate Receptor 2 (mGlu2). Part 1. Identification and Synthesis of Phenyl‐tetrazolyl Acetophenones.
Authors: Pinkerton Anthony B. , Cube Rowena V. , Hutchinson John H. , Rowe Blake A. , Schaffhauser Herve , Zhao Xiumin , Daggett Lorrie P. , Vernier Jean‐Michel 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Synthesis of 3‐(3‐Alkyl‐5‐thioxo‐1H‐4,5‐dihydro‐1,2,4‐triazol‐4‐yl) aminocarbonylchromones.
Authors: Cao Linghua , Zhang Lin , Cui Pengyuan 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Azinyl Sulfides. Part 82. Synthesis of 1‐Methyl‐3‐methylthio‐ and 1‐Methyl‐3‐methylsulfinyl‐4‐substituted 2(1H)‐Quinolinones.
Authors: Chrobak Elwira , Maslankiewicz Andrzej 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Simple, Facile, and One‐Pot Conversion of the Baylis—Hillman Adducts into Functionalized 1,2,3,4‐Tetrahydroacridines and Cyclopenta[b]quinolines.
Authors: Basavaiah Deevi , Rao Jamjanam Srivardhana , Reddy Raju Jannapu 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Synthesis and Reactions of Some New Heterocyclic Compounds Containing the Thienylthieno[2,3‐b]pyridine Moiety.
Authors: Bakhite Etify A. , Abdel‐Rahman Abdu E. , Mohamed Omima S. , Thabet Eman A. 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.
Synthesis of New Heterocyclic Systems: 3,4‐Dihydro‐1‐isoquinolinyl‐ and Spiro[4,5]benzo[8,9]‐6‐azadec‐6‐en‐7‐ylthieno[2,3‐b]pyridine‐3‐amines.
Authors: Kaigorodova E. A. , Kostenko E. S. , Stashina G. A. , Krapivin G. D. 
Published: January 2005

AbstractFor Abstract see ChemInform Abstract in Full Text.