bluuebunny/crossref_metadata_2025_split huggingface dataset:
ChemInform Abstract: A Photoirradiative Phase‐Vanishing Method: Efficient Generation of HBr from Alkanes and Molecular Bromine and Its Use for Subsequent Radical Addition to Terminal Alkenes.
Authors: Matsubara Hiroshi , Tsukida Masaaki , Ishihara Daisuke , Kuniyoshi Kenji , Ryu Ilhyong 
Published: October 2010

AbstractA direct method for the photocatalytic in situ generation of HBr from bromine and isooctane and subsequent photocatalyzed regioselective addition is presented.
ChemInform Abstract: Ni(I) and Ni(II) Ring‐Expanded N‐Heterocyclic Carbene Complexes: C—H Activation, Indole Elimination and Catalytic Hydrodehalogenation.
Authors: Davies Caroline J. E. , Page Michael J. , Ellul Charles E. , Mahon Mary F. , Whittlesey Michael K. 
Published: October 2010

AbstractA nickel N‐heterocyclic carbene complex is synthesized via an indole elimination process and successfully applied for the catalytic hydrodechlorination of 1‐chloro‐4‐fluorobenzene (Ia) and hydrodebromination of 1‐bromo‐4‐fluorobenzene (Ia) under mild reaction conditions.
ChemInform Abstract: Convenient Direct Reductive Amination of Carbonyl Compounds in a Completely Aqueous Media.
Authors: Simion Cristian , Simion Alina M. , Arimura Takashi , Miyazawa Akira , Tashiro Masashi 
Published: October 2010

AbstractThe synthesis of secondary and tertiary amines through a direct reductive amination process carried out for the first time in completely aqueous media is reported.
ChemInform Abstract: A Rhodium IBiox[(‐)‐menthyl] Complex as a Highly Selective Catalyst for the Asymmetric Hydroarylation of Azabicycles: An Alternative Route to Epibatidine.
Authors: Bexrud Jason , Lautens Mark 
Published: October 2010

AbstractThe newly synthesized chiral rhodium N‐heterocyclic carbene complex ROXI is together with its dimer used as an efficient catalyst mixture for the asymmetric hydroarylation of azabicycles.
ChemInform Abstract: Synthesis of α‐Trifluoromethyl‐α‐hydroxycarboxylate Derivatives and Their Phosphorus‐Containing Analogues with the Use of Fluorinated Diazo Compounds.
Authors: Titanyuk I. D. , Vorob'eva D. V. , Osipov S. N. , Beletskaya I. P. 
Published: October 2010

AbstractA novel access to derivates of α‐trifluoromethyl‐substituted hydroxycarboxylates (III) or (V) and hydroxyphosphonates (XII) is described.
ChemInform Abstract: Introducing Catalytic Activity in Helical Nanostructures: Microwave Assisted Oxathioacetalisation Catalyzed by Al‐Containing Helical Mesoporous Silicas.
Authors: Carrillo Adela I. , Sarrano Elena , Luque Rafael , Garcia Matinez Javier 
Published: October 2010

AbstractAluminum‐containing helical mesoporous silica is prepared and successfully applied as a reusable catalyst for the oxathioacetalization of carbonyl compounds (I) under microwave irradiation.
ChemInform Abstract: Highly Effective and Enantioselective α‐Amination of Aldehydes Promoted by Chiral Proline Amide—Thiourea Bifunctional Catalysts.
Authors: Fu Ji‐Ya , Huang Qing‐Chun , Wang Qiao‐Wei , Wang Li‐Xin , Xu Xiao‐Ying 
Published: October 2010

AbstractOptimized ATC is successfully applied to the direct asymmetric α‐amination of aldehydes with azodicarboxylates in enantioselectivities up to 99% ee.
ChemInform Abstract: Fluoroalcohols: Versatile Solvents in Hypervalent Iodine Chemistry and Syntheses of Diaryliodonium(III) Salts.
Authors: Dohi Toshifumi , Yamaoka Nobutaka , Kita Yasuyuki 
Published: October 2010

AbstractThe present work reveals that fluoroalcohols can positively affect the dehydrative condensation of hypervalent iodine reagents toward aromatic and heteroaromatic compounds.
ChemInform Abstract: Novel Periodic Mesoporous Silica Chlorides (PMSCl) with 2D P6mm Hexagonal Structures: Efficient Catalysts for the Beckmann Rearrangement.
Authors: Karimi Babak , Behzadnia Hesam 
Published: October 2010

AbstractTreatment of mesoporous silica SBA‐15 in refluxing thionyl chloride generates novel surface‐chlorinated mesoporous silica materials which are found to be useful recyclable catalysts for the selective Beckmann rearrangement.
ChemInform Abstract: A New Chiral N‐Heterocyclic Carbene Silver(I) Cylinder: Synthesis, Crystal Structure and Catalytic Properties.
Authors: Wang Dehui , Zhang Bingguang , He Cheng , Wu Pengyan , Duan Chunying 
Published: October 2010

AbstractA novel N‐heterocyclic carbene silver complex is synthesized and its catalytic activity in the enantioselective cyanosilylation of Schiff bases (I) is evaluated.
ChemInform Abstract: Competing Regiodirecting Effects of Ester and Aryl Groups in [3 + 3] Cyclocondensations of 1,3‐Bis(trimethylsilyloxy)‐1,3‐butadienes: Regioselective Synthesis of 3‐Hydroxyphthalates and 2‐Hydroxyterephthalates.
Authors: Shkoor Mohanad , Fatunsin Olumide , Riahi Abdolmajid , Lubbe Mathias , Reim Stefanie , Sher Muhammad , Villinger Alexander , Fischer Christine , Langer Peter 
Published: October 2010

Abstract[3+3] Cyclocondensations of 1,3‐bis(trimethylsilyloxy)‐1,3‐butadienes with ester‐substituted 3‐ethoxy‐ and 3‐silyloxy‐2‐en‐1‐ones provide a regioselective approach to 3‐hydroxyphthalates and 2‐hydroxyterephthalates.
ChemInform Abstract: Highly Stereoselective Preparation of Chiral α‐Substituted Sulfides from α‐Chloro Sulfides via 1,2‐Asymmetric Induction.
Authors: Raghavan Sadagopan , Kumar V. Vinoth , Chowhan L. Raju 
Published: October 2010

AbstractThe reaction of racemic and chiral α‐chlorosulfides with organozinc bromides affords the syn‐products.
ChemInform Abstract: Chiral Triphenylprolinol Ligands for the Efficient Catalytic Asymmetric Arylation of Aldehydes.
Authors: Moro Angelica Venturini , Tiekink Edward R. T. , Zukerman‐Schpector Julio , Luedtke Diogo S. , Correia Carlos Roque D. 
Published: October 2010

AbstractNew and recyclable chiral amino alcohols are prepared and used as chiral ligands in catalytic asymmetric aryl transfer reactions.
ChemInform Abstract: A Radical‐Based Approach to Hydroxytetralones from Unprotected Phenols.
Authors: Petit Laurent , Zard Samir Z. 
Published: October 2010

AbstractXanthates derived from unprotected 2‐hydroxyacetophenones undergo intermolecular addition to unactivated alkenes such as (II) and subsequent intramolecular ring closure to give hydroxytetralones (IV), (VI) and (VIII).
ChemInform Abstract: Palladium‐Catalyzed Direct Heteroarylation of Bromobenzylacetamide Derivatives: A Simple Access to Heteroarylated Benzylamine Derivatives.
Authors: Laidaoui Nouria , Miloudi Abdellah , El Abed Douniazad , Doucet Henri 
Published: October 2010

AbstractThe method renders possible the access to a broad spectrum of target compounds for pharmaceutical research.
ChemInform Abstract: Synthesis of Novel Spiro Pyrrolidine and Pyrrolizine Derivatives by 1,3‐Dipolar Cycloaddition.
Authors: Li Xiaofang , Zheng Aiting , Liu Bin , Yu Xianyong , Yi Pinggui 
Published: October 2010

AbstractAzomethine ylides, derived from isatin and sarcosine or proline, react with substrates of type (I)/(V) to give the novel dispiroheterocycles regio‐ and stereoselectively.
ChemInform Abstract: Diastereoselective Synthesis of 2‐Fluoroaziridine‐2‐carboxylates by Reformatsky‐Type Aza‐Darzens Reaction.
Authors: Tarui Atsushi , Kawashima Naoto , Sato Kazuyuki , Omote Masaaki , Ando Akira 
Published: October 2010

AbstractOptimized conditions A) are highly suitable for the exclusive preparation of the desired aziridines (substructures of bioactive molecules) with the syn isomer predominating.
ChemInform Abstract: Synthesis of Alkylpyrroles by Use of a Vinamidinium Salt.
Authors: Wright Mathew T. , Carroll David G. , Smith Timothy M. , Smith Stanton Q. 
Published: October 2010

AbstractA new route is presented to synthesize pyrrole 2‐carboxylates, pharmaceutically important substructures, via cyclocondensation of salts (I) with glycine esters.
ChemInform Abstract: Synthesis of Hydrogenated 2,7‐Dimethylpyrrolo[3,4‐b]indoles — Analogues of Dimebon.
Authors: Ivachtchenko A. V. , Frolov E. B. , Mitkin O. D. , Tkachenko S. E. , Khvat A. V. 
Published: October 2010

AbstractA variety of novel 2,7‐dimethyldihydro‐ and previously unknown cis‐hexahydropyrrolo[3,4‐b]indoles are synthesized and evaluated for their ability to block calcium currents induced by the H1 histamine receptor and to interact with serotonin 5‐HT6 receptors.
ChemInform Abstract: Diversity‐Oriented Pyrazol‐3‐one Synthesis Based on Hydrazinodipeptide‐Like Units Prepared via the Ugi Reaction.
Authors: Lakontseva Ekaterina , Krasavin Mikhail 
Published: October 2010

AbstractA remarkable switch of reactivity for the Ugi‐type products (V) is observed under basic and acidic reaction conditions resulting in formation of different types of pyrazoles as single products.
ChemInform Abstract: Synthesis and Structure—Activity Relationship Studies of Pyrazole‐Based Heterocycles as Antitumor Agents.
Authors: Farag Ahmad M. , Mayhoub Abdelrahman S. , Eldebss Taha M. A. , Amr Abdel‐Galil E. , Ali Korany A. K. , Abdel‐Hafez Naglaa A. , Abdulla Mohamed M. 
Published: October 2010

AbstractA variety of new 1,5‐diphenylpyrazole derivatives substituted by different triazole or triazole bioisosteres at position 3 is synthesized and evaluated for their anti‐estrogenic effects and their cytotoxic properties against estrogen‐dependent tumor cell lines.
ChemInform Abstract: Microwave Assisted Transformation of Benzimidazolyl Chalcones into N1‐Substituted Pyrazolines and Evaluation of Their Antimicrobial Activities.
Authors: Rajora Jayanti , Yadav Janardan , Kumar Ravindra , Srivastava Yogendra K. 
Published: October 2010

AbstractAll the pyrazoline derivatives synthesized are found to possess moderate to good antibacterial activity.
ChemInform Abstract: A Solvent‐Free Protocol for the Green Synthesis of Arylalkylidene Rhodanines in a Task‐Specific Ionic Liquid.
Authors: Alizadeh Abdolhamid , Khodaei Mohammad M. , Eshghi Ali 
Published: October 2010

AbstractKnoevenagel condensation of rhodanine (I) with carbonyl compounds (II), (IV) or (VI) proceeds efficiently in the presence of a minimum amount of a novel ionic liquid.
ChemInform Abstract: o‐Aminothiophenol in Reactions with Carbonyl Compounds and Isocyanides: A Word of Caution.
Authors: Tsirulnikov Sergey , Dmitriev Dmitry , Krasavin Mikhail 
Published: October 2010

AbstractThe sequential reaction of o‐aminothiophenol with carbonyl compounds and tert‐butyl isocyanide is reinvestigated.
ChemInform Abstract: Efficient Synthesis of Allylic Azides and One‐Pot Regioselective Synthesis of 1,4‐Disubstituted 1,2,3‐Triazoles from Homoallyl Alcohols.
Authors: Reddy P. Surendra , Ravi V. , Sreedhar B. 
Published: October 2010

AbstractA Pd‐catalyzed hydroazidation of homoallyl alcohols is developed to give good yields of allylic azides.
ChemInform Abstract: Synthesis, Antimicrobial and Insecticidal Activity of Some 4H‐1,2,4‐Triazole Derivatives.
Authors: Gautam Nidhi , Chourasia O. P. 
Published: October 2010

AbstractThe majority of the synthesized triazole derivatives (IV) (12 examples) exhibit excellent antibacterial, promising antifungal and marked insecticidal activities.
ChemInform Abstract: Synthesis and Structural Characterization of 2,4‐Bis(5‐aryl‐1,3,4‐oxadiazol‐2‐yl)pyridine Derivatives
Authors: Wang XiaoQing , Zhao ZhiGang , Liu XingLi , Li WeiJie 
Published: October 2010

Abstractas biologically interesting substances; 10 examples
ChemInform Abstract: A Novel Synthesis of 3‐Aryl Coumarins and Evaluation of Their Antioxidant and Lipoxygenase Inhibitory Activity.
Authors: Roussaki Marina , Kontogiorgis Christos A. , Hadjipavlou‐Litina Dimitra , Hamilakis Stylianos , Detsi Anastasia 
Published: October 2010

Abstract15 Title compounds of type (III) are prepared and tested for their antioxidant and lipoxygenase inhibitory activities.
ChemInform Abstract: One‐Pot Four Component Synthesis of 4,6‐Disubstituted 3‐Cyano‐2‐pyridones in Polyethylene Glycol.
Authors: Nalage Santosh V. , Nikum Ajay P. , Kalyankar Mohan B. , Patil Vijay S. , Patil Umesh D. , Desale Kamlesh R. , Patil Shamkant L. , Bhosale Sidhanath V. 
Published: October 2010

AbstractThe reaction in polyethylene glycol in the absence of any catalyst is a novel and eco‐friendly method for the synthesis of pyridones.
ChemInform Abstract: Facile and Efficient Aromatization of 1,4‐Dihydropyridines with M(NO3)2·XH2O, TNCB, TBAP and HMTAI and Preparation of Deuterium Labeled Dehydronifedipine from Nifedipine‐d3.
Authors: Shaikh Ajam C. , Chen Chinpiao 
Published: October 2010

AbstractMetal nitrates, tetrabutyl ammonium periodate (TBAP), and hexamethylenetetramine‐iodine (HMTAI) are valuable oxidants for the oxidation of Hantzsch′s 1,4‐dihydropyridines (I) without the need of external activation such as microwave or ultrasound.
ChemInform Abstract: New Quinoline Derivatives: Synthesis and Investigation of Antibacterial and Antituberculosis Properties.
Authors: Eswaran Sumesh , Adhikari Airody Vasudeva , Chowdhury Imran H. , Pal Nishith K. , Thomas K. D. 
Published: October 2010

AbstractThe new quinoline derivatives, wherein active pharmacophores, viz.
ChemInform Abstract: Three‐Component Synthesis of 1‐Substituted 6′,7′‐Dimethoxy‐4′H‐spiro[adamantane‐2,3′‐isoquinolines].
Authors: Rozhkova Yu. S. , Gorbunov A. A. , Shklyaev Yu. V. 
Published: October 2010

AbstractTitle compounds (IV) and (VI) are formed by Ritter‐type reaction between 2‐epoxymethyleneadamantane (I), 1,2‐dimethoxybenzene as activated arene, and nitriles (III) or (V).
ChemInform Abstract: Reaction of 3,4‐Dihydro‐β‐carbolines with 4‐Fluorophenyl‐nitrile Oxide.
Authors: Milen Matyas , Abranyi‐Balogh Peter , Dancso Andras , Simig Gyula , Keglevich Gyoergy 
Published: October 2010

AbstractThe reaction of carbolines (I) with the nitrile oxide generated from (II) affords novel adducts (III) in high yields.
ChemInform Abstract: Advancing the Morita—Baylis—Hillman Chemistry of 1‐Formyl‐β‐carbolines for the Synthesis of Indolizino‐indole Derivatives.
Authors: Singh Virender , Hutait Samiran , Batra Sanjay 
Published: October 2010

AbstractThe utility of the Morita—Baylis—Hillman reaction of N‐substituted 1‐formyl‐β‐carbolines for the synthesis of indolizino‐indole derivatives mimicking harmicine and homofascaplysin frameworks is described.
ChemInform Abstract: Synthesis and Antimicrobial Activity of Tetrazolo[1,5‐a]quinoline‐4‐carbonitrile Derivatives.
Authors: Kategaonkar Amol H. , Labade Vilas B. , Shinde Pravin V. , Kategaonkar Atul H. , Shingate Bapurao B. , Shingare Murlidhar S. 
Published: October 2010

AbstractAll compounds (III) demonstrate potent inhibition against all the strains tested.
ChemInform Abstract: Synthesis of 2‐(Pyrimidin‐2‐yl)‐1‐phenyl‐2,3,4,9‐tetrahydro‐1H‐β‐carbolines as Antileishmanial Agents.
Authors: Kumar Ravi , Khan Shahnawaz , Verma Aditya , Srivastava Saumya , Viswakarma Preeti , Gupta Suman , Meena Sanjeev , Singh Neetu , Sarkar Jayanta , Chauhan Prem M. S. 
Published: October 2010

AbstractThe synthetic pathway to β‐carbolines (V) and (VII) involves oxidation of educt (I) to its sulfone followed by nucleophilic substitution of the formed mesyl group with tryptamine (II).
ChemInform Abstract: Synthesis and in vitro Antitumor Activity of Selected 7‐Fluoro‐6‐(4‐methyl‐1‐piperazinyl)‐2‐(thiosubstituted)‐4 (3H)‐quinazolinones.
Authors: Abdel‐Jalil Raid J. , Al‐Momani Ehab , Tahtamooni Lubna , Machulla H.‐Juergen , Voelter Wolfgang 
Published: October 2010

AbstractThe title compound (Va) is tested against 60 different human tumor cell lines.
ChemInform Abstract: New Pyrazolo[1,5a]pyridimines as Orally Active Inhibitors of Lck.
Authors: Gommermann Nina , Buehlmayer Peter , von Matt Anette , Breitenstein Werner , Masuya Keiichi , Pirard Bernard , Furet Pascal , Cowan‐Jacob Sandra W. , Weckbecker Gisbert 
Published: October 2010

AbstractReaction of acid chlorides (VI) or chloroformates (VIII) with key intermediate (V) affords a new series of pyrazolopyrimidines.
ChemInform Abstract: Novel 6,8‐Dibromo‐4(3H)quinazolinone Derivatives of Antibacterial and Antifungal Activities.
Authors: Mohamed Mosaad S. , Kamel Mohsen M. , Kassem Emad M. M. , Abotaleb Nageh , El‐moez Sherein I. Abd , Ahmed Marwa F. 
Published: October 2010

AbstractStarting from the hydrazole (I) a new series of Schiff bases (III) and their cyclized products, thiazolidinones (V), pyrazoles, e.g. (X), oxadiazole, pyrroles, and other related products are synthesized.
ChemInform Abstract: N‐Iodosaccharin (NISac): A New Reusable Catalyst for Formal [2 + 4] Cycloaddition of Imines and Enones.
Authors: Rai Ankita , Yadav Lal Dhar S. 
Published: October 2010

AbstractNSA acts as an efficient promotor to give the pharmaceutically important oxazine derivatives (16 examples) with complete diastereoselectively.
ChemInform Abstract: anti‐Neuroinflammatory Activity of 1,5‐Benzodiazepine Derivatives.
Authors: Ha Sang Keun , Shobha Donthabhaktuni , Moon Eunjung , Chari Murugulla A. , Mukkanti Kagga , Kim Sung‐Hoon , Ahn Kwang‐Hyun , Kim Sun Yeou 
Published: October 2010

AbstractA series of 10 title compounds of type (III) is prepared.
ChemInform Abstract: Rhodium‐Catalyzed Dehydroborylation of Styrenes with Naphthalene‐1,8‐diaminatoborane [(dan)BH]: New Synthesis of Masked β‐Borylstyrenes as New Phenylene—Vinylene Cross‐Coupling Modules.
Authors: Iwadate Noriyuki , Suginome Michinori 
Published: October 2010

AbstractStyrenes (I) undergo dehydroborylation with title compound (II) in the presence of a Rh‐complex, to give β‐borylstyrenes (III) in good yields.
ChemInform Abstract: Direct Functionalization of BODIPY Dyes by Oxidative Nucleophilic Hydrogen Substitution at the 3‐ or 3,5‐Positions.
Authors: Leen Volker , Zaragozi Gonzalvo Veronica , Deborggraeve Wim M. , Boens Noel , Dehaen Wim 
Published: October 2010

AbstractThe reaction of boron dipyrromethene (I) with amines (II) in the presence of oxygen leads to 3‐substituted BODIPY derivatives.
ChemInform Abstract: 8‐PropargylaminoBODIPY: Unprecedented Blue‐Emitting Pyrromethene Dye. Synthesis, Photophysics and Laser Properties.
Authors: Gomez‐Duran C. F. Azael , Garcia‐Moreno Immaculada , Costela Angel , Martin Virginia , Sastre Roberto , Banuelos Jorge , Lopez Arbeloa Fernando , Lopez Arbeloa Inigo , Pena‐Cabrera Eduardo 
Published: October 2010

AbstractThe title compound (III) is the first highly efficient BODIPY laser dye with emission in the blue spectral region of the visible spectrum.
ChemInform Abstract: Metal‐Free Catalytic Boration at the β‐Position of α,β‐Unsaturated Compounds: A Challenging Asymmetric Induction.
Authors: Bonet Amadeu , Gulyas Henrik , Fernandez Elena 
Published: October 2010

AbstractA metal free method for the synthesis of β‐borated carbonyl compounds by reacting B2pin2 with either α,β‐unsaturated esters or ketones in the presence of chiral phosphine catalysts is reported.
ChemInform Abstract: Testing the Functional Tolerance of the Piers—Rubinsztajn Reaction: A New Strategy for Functional Silicones.
Authors: Grande John B. , Thompson David B. , Gonzaga Ferdinand , Brook Michael A. 
Published: October 2010

AbstractTris(pentafluorophenyl)borane is a good catalyst for the preparation of functionalized siloxanes such as (III) and (VI) by Piers—Rubinsztajn reaction of alkoxysilanes with hydrosilanes.
ChemInform Abstract: Synthesis of Cytotoxic Ferrocenyl Flavones via a Ferricenium‐Mediated 1,6‐Oxidative Cyclization.
Authors: Monserrat Jean‐Philippe , Chabot Guy G. , Hamon Louis , Quentin Lionel , Scherman Daniel , Jaouen Gerard , Hillard Elizabeth A. 
Published: October 2010

AbstractThe oxidation of the ferrocenyl group of 2′‐hydroxyferrocenyl chalcones (II) activates the β‐position of the unsaturated ketone to nucleophilic attack to yield the first examples of ferrocenyl flavones (III).
ChemInform Abstract: Total Synthesis of Furanether B. Construction of a Hydroazulene Skeleton via a Novel [5 + 2] Cycloaddition Reaction of Silyloxyallene.
Authors: Mitachi Katsuhiko , Yamamoto Takashi , Kondo Fumikatsu , Shimizu Tadashi , Miyashita Masaaki , Tanino Keiji 
Published: October 2010

AbstractA new synthetic method for cycloheptanone derivatives is developed on the basis of a novel [5 + 2] cycloaddition reaction using a dicobalt hexacarbonyl propargyl cation species and a silyloxyallene (II).
ChemInform Abstract: Syntheses and Antibacterial Activities of Diterpene Catechol Derivatives with Abietane, Totarane and Podocarpane Skeletons Against Methicillin‐Resistant Staphylococcus aureus and Propionibacterium acnes.
Authors: Tada Masahiro , Kurabe Jun , Yoshida Takashi , Ohkanda Tomoyuki , Matsumoto Yusuke 
Published: October 2010

AbstractAbietaquinone methide (I) and totaratrienediol (II) show potent activities against MRSA and P.
ChemInform Abstract: Cytosporolides A—C, Antimicrobial Meroterpenoids with a Unique Peroxylactone Skeleton from Cytospora sp.
Authors: Li Yan , Niu Subin , Sun Bingda , Liu Shuchun , Liu Xingzhong , Che Yongsheng 
Published: October 2010

AbstractFor all three components, significant antimicrobial activity is observed against the Gram‐positive bacteria Staphylococcus aureus and Streptococcus pneumoniae.
ChemInform Abstract: Synthesis of the Azetidinyl‐Thiazoline Fragment of Vioprolides A and C.
Authors: Chopin Nathalie , Couty Francois , Evano Gwilherm 
Published: October 2010

AbstractKey steps of the synthetic approach include formation of the four‐membered ring by intramolecular alkylation of suitable protected precursor(III) followed by ring closure with L‐cysteine (V) affording the title thiazoline fragment (VI).
ChemInform Abstract: A Reasonably Stereospecific Multistep Conversion of Boc‐Protected α‐Amino Acids to Phth‐Protected β3‐Amino Acids.
Authors: Temperini Andrea , Capperucci Antonella , Degl'Innocenti Alessandro , Terlizzi Raffaella , Tiecco Marcello 
Published: October 2010

AbstractA five‐step one‐pot procedure is presented to convert N‐Boc protected amino acids to N‐phthaloyl propargylic amines.
ChemInform Abstract: Synthesis of Sugar‐Fused Isoxazoline N‐Oxides from 2‐Nitroglycals.
Authors: Zhang Qingju , Sun Jiansong , Zhang Fuyi , Yu Biao 
Published: October 2010

AbstractA new type of sugar‐fused isoxazoline N‐oxides (III) is synthesized from 2‐nitroglycals by [4+2] condensation.
ChemInform Abstract: N‐Bromosuccinimide‐Mediated Conversion of Allyl Glycosides to Glycosyl Hemiacetals.
Authors: Panchadhayee Rajib , Misra Anup Kumar 
Published: October 2010

AbstractThe hydrolysis of differentially functionalized allyl glycosides to their corresponding glycosyl hemiacetal derivatives under mild and metal‐free conditions proceeds exceptionally fast and is compatible with most of the functional groups used in oligosaccharide synthesis.
ChemInform Abstract: Efficient Asymmetric Organocatalytic Formation of Erythrose and Threose under Aqueous Conditions.
Authors: Burroughs Laurence , Vale Matthew E. , Gilks James A. R. , Forintos Henrietta , Hayes Christopher J. , Clarke Paul A. 
Published: October 2010

AbstractEthyl ester of N‐methyl‐L‐leucine is applied as a chiral catalyst for the aldol dimerization of aldehyde (I).
ChemInform Abstract: Syntheses and Biological Evaluation of Ring‐C Modified Colchicine Analogues.
Authors: Yang Baiyuan , Zhu Zhiqing C. , Goodson Holly V. , Miller Marvin J. 
Published: October 2010

AbstractDiels—Alder reactions of colchicine (I) with iminonitroso agents (II) afford the ring‐C modified alkaloids (III) and (IV) as regioisomeric adducts.
ChemInform Abstract: A 1,3‐Strain Enabled Retention of Chirality During Bis‐Cyclization of β‐Ketoamides: Total Synthesis of (‐)‐Salinosporamide A and (‐)‐Homosalinosporamide A.
Authors: Nguyen Henry , Ma Gil , Romo Daniel 
Published: October 2010

Abstract(‐)‐Salinosporamide A (IVa) and (‐)‐homosalinosporamide A (IVb) are prepared via a diastereoselective bis‐cyclization of β‐keto tertiary amide of type (II) as key step.
ChemInform Abstract: Three New Oligostilbenes from the Seeds of Paeonia suffruticosa.
Authors: He Chun‐Nian , Peng Yong , Xu Li‐Jia , Liu Zheng‐An , Gu Jing , Zhong Ai‐Guo , Xiao Pei‐Gen 
Published: October 2010

Abstractisolation and extensive structural elucidation of trans‐suffruticosol D (II), cis‐suffruticosol D (Ia), and cis‐gnetin H (Ib)