bluuebunny/crossref_metadata_2025_split huggingface dataset:
ChemInform Abstract: Cyclocondensation of N‐(Prop‐2‐yn‐1‐yl)‐ and N‐(Penta‐2,4‐diyn‐1‐yl)‐o‐phenylenediamines with Phenyl Isothiocyanate and Carbon Disulfide.
Authors: Novikov R. V. , Danilkina N. A. , Balova I. A. 
Published: March 2012

AbstractThe cyclocondensation of di‐ and monoacetylenic derivatives of o‐phenylenediamine with different substituents at the triple bond with Ph‐NCS or CS2 for studying the scope and limitations of the preparation of 2,3‐dihydro[1,3]thiazolo and [1,3]thiazolo[3,2‐a]benzimidazole derivatives is investigated.
ChemInform Abstract: Synthesis and Antimicrobial Activity of Novel Spiro‐isoxazolyl Oxazolidin‐4‐one‐[5,51]‐1,2,4‐oxadiazolines and Thiazolidin‐4‐one‐[5,51]‐1,2,4‐oxadiazolines.
Authors: Rajanarendar E. , Reddy A. Siva Rami , Reddy K. Govardhan , Raju S. 
Published: March 2012

AbstractA variety of novel title spiro‐compounds (VII) and (X) are synthesized via 1,3‐dipolar cycloaddition reactions of 2‐aryliminooxazoles (V) or ‐thiazoles, resp., with benzonitrile oxides.
ChemInform Abstract: An Efficient Synthesis of Flavans from Salicylaldehyde and Acetophenone Derivatives.
Authors: Mazimba Ofentse , Maseane Ishmael B. , Majinda Runner R. 
Published: March 2012

AbstractThe general route involves aldol condensation of salicylaldehydes with acetophenones and reduction of both the ketone and the double bond of the resulting chalcones with NaBH4.
ChemInform Abstract: Synthesis of 4,N‐Diaryl‐2,7,7‐trimethyl‐5‐oxo‐1,4,5,6,7,8‐hexahydro‐3‐quinolinecarbox amides.
Authors: Gein V. L. , Kazantseva M. I. , Kurbatova A. A. 
Published: March 2012

AbstractThe title compounds (IV) (11 examples) are obtained in an four‐component one‐pot reaction of dimedone, N‐aryl‐substituted acetoacetic acid amides, aryl aldehydes, and ammonium acetate.
ChemInform Abstract: Synthesis of Libraries of Quinoxalines Through Eco‐Friendly Tandem Oxidation—Condensation or Condensation Reactions.
Authors: Paul Susmita , Basu Basudeb 
Published: March 2012

AbstractCondensation of α‐dicarbonyl compounds, α‐hydroxy ketones, and α‐bromo ketones with 1,2‐diamines is efficiently promoted by KF on basic alumina to give quinoxalines and pyrazines in good yields.
ChemInform Abstract: BOP‐Mediated One‐Pot Synthesis of C5‐Symmetric Macrocyclic Pyridone Pentamers.
Authors: Du Zhiyun , Ren Changliang , Ye Ruijuan , Shen Jie , Maurizot Victor , Lu Yujin , Wang Jian , Zeng Huaqiang 
Published: March 2012

AbstractA greener, more cost‐effective and time‐saving method for the synthesis of the title compounds (II) is developed.
ChemInform Abstract: Palladium‐Catalyzed Enantioselective Desymmetrization of Silacyclobutanes: Construction of Silacycles Possessing a Tetraorganosilicon Stereocenter.
Authors: Shintani Ryo , Moriya Kohei , Hayashi Tamio 
Published: March 2012

AbstractA new method to prepare chiral organosilanes is reported.
ChemInform Abstract: Solvent‐Induced Selectivity Switching: Intermolecular Allylsilylation, Arylsilylation, and Silylation of Alkynes over Montmorillonite Catalyst.
Authors: Motokura Ken , Matsunaga Shigekazu , Miyaji Akimitsu , Yashima Tatsuaki , Baba Toshihide 
Published: March 2012

AbstractReactions of alkynes (I) with allylsilane (II), catalyzed by H+‐montmorillonite, are studied in various solvents.
ChemInform Abstract: Palladium‐Catalyzed Cross‐Coupling of PhSeSnBu3 with Aryl and Alkyl Halides in Ionic Liquids: A Practical Synthetic Method of Diorganyl Selenides.
Authors: Zhao Hong , Hao Wenyan , Xi Zhiwen , Cai Mingzhong 
Published: March 2012

AbstractThe Pd‐catalyzed reaction of phenylselenylstannane (II) with a wide variety of aromatic and aliphatic iodides and bromides proceeds smoothly in a room temperature ionic liquid to give the corresponding phenyl organyl selenides in good yields.
ChemInform Abstract: New Polyene Macrolide Family Produced by Submerged Culture of Streptomyces durmitorensis.
Authors: Flieger Miroslav , et al. et al. 
Published: March 2012

AbstractA new polyene macrolide, closely related to the pentaene macrolide antibiotic roflamycoin, is isolated from both fermentation broth and biomass of Streptomyces durmitorensis wild‐type strain MS405.
ChemInform Abstract: Mannuronic Acids: Reactivity and Selectivity
Authors: Codee Jeroen D. C. , Walvoort Marthe T. C. , de Jong Ana‐Rae , Lodder Gerrit , Overkleeft Herman S. , van der Marel Gijsbert A. 
Published: March 2012

AbstractReview: 41 refs.
ChemInform Abstract: Dynamic Recovery in Silicate‐Apatite Structures under Irradiation and Implications for Long‐Term Immobilization of Actinides.
Authors: Weber William J. , Zhang Yanwen , Xiao Haiyan , Wang Lumin 
Published: March 2012

AbstractIrradiation‐induced amorphization and recrystallization of Ca2La8(SiO4)6O2 and Sr2Nd8(SiO4)6O2 with the apatite structure are investigated to predict their long‐term behavior as host phases for immobilization of actinide elements from the nuclear fuel cycle.
ChemInform Abstract: UV Nonlinear Optical Crystal Ba2[B6O9(OH)4] Featuring Unique Chiral Layers with a New B18O42 Circle Based on BO3 and BO4 Units.
Authors: Wang Li , Pan Shilie , Chang Lixian , Hu Jianyang , Yu Hongwei 
Published: March 2012

AbstractThe new title compound is hydrothermally synthesized from a mixture of Ba(NO3)2, H3BO3, and LiOH in H2O (autoclave, 200 °C, 3 d, 85% yield).
ChemInform Abstract: Spectroscopic Studies of Sulfite‐Based Polyoxometalates at High Temperature and High Pressure.
Authors: Quesada Cabrera Raul , Firth Steven , Blackman Christopher S. , Long De‐Liang , Cronin Leroy , McMillan Paul F. 
Published: March 2012

AbstractThe eclipsed (α) and staggered (β) forms of (Pen4N)4 [Mo18O54(SO3)2]·MeCN (Pen: ‐(CH2)4‐Me) are characterized by a combination of IR, Raman, and visible spectroscopy at high temperature and high pressure.
ChemInform Abstract: The Structure and Luminescence Properties of Green Ca3Al2O6:Bi3+ Phosphors.
Authors: Ju Haidong , Deng Weiping , Wang Baoling , Liu Jie , Tao Xutang , Xu Shiqing 
Published: March 2012

AbstractThe title phosphors are prepared by solid state reaction of CaCO3, Al2O3, and Bi2O3 (air, 1300 °C, 6 h, alumina crucibles).
ChemInform Abstract: Crystal and Magnetic Structures and Magnetic Properties of Selenate Containing Natrochalcite, AIM2II(H3O2) (SeO4)2 Where A: Na or K and M: Mn, Co, or Ni.
Authors: Maalej Wassim , Vilminot Serge , Andre Gilles , Elaoud Zakaria , Mhiri Tahar , Kurmoo Mohamedally 
Published: March 2012

AbstractCompounds (IIIb,c) and (Vb) crystallize with the natrochalcite‐type structure in the monoclinic space group C2/m with Z = 2 (single crystal XRD for the Ni‐ and powder XRD for the Mn‐compound).
ChemInform Abstract: Phase Stability and Oxygen Nonstoichiometry of Highly Oxygen‐Deficient Perovskite‐Type Oxides: A Case Study of (Ba,Sr)(Co,Fe)O3‐δ.
Authors: Mueller David N. , De Souza Roger A. , Yoo Han‐Ill , Martin Manfred 
Published: March 2012

AbstractThe phase stability and oxygen nonstoichiometry of Ba0.5Sr0.5Co0.8Fe0.2 O3‐δ (BSCF5582) is investigated using thermogravimetry (TG) and coulometric titration (CT).
ChemInform Abstract: Studies on the Chemistry of [Cd(NH3)4](MnO4)2. A Low Temperature Synthesis Route of the CdMn2O4+x Type NOx and CH3SH Sensor Precursors.
Authors: Kotai Laszlo , et al. et al. 
Published: March 2012

Abstract[Cd(NH3)4](MnO4)2 (I) is synthesized from an aqueous solution of CdSO4, NH3, and NaMnO4 at 0 °C (86% yield).
ChemInform Abstract: Diastereoselective Synthesis of Enantiopure Homopropargylic N‐tert‐Butylsulfinylamines.
Authors: Cyklinsky Mathieu , Botuha Candice , Chemla Fabrice , Ferreira Franck , Perez‐Luna Alejandro 
Published: March 2012

AbstractThe propargylation of N‐tert‐butylsulfonylimines (I) and (IV) with allenylzinc reagent (II), generated in situ, proceeds with excellent regio‐ and diastereoselectivity to give alkynes (III) and (V), resp., as highly preferred products.
ChemInform Abstract: Cu(I)‐Catalyzed Tandem Benzyldiazoester Coupling with Terminal Alkyne—Allene Formation—Michael Reaction: Application to the Syntheses of Oxa and Azacycles.
Authors: Kumaraswamy Gullapalli , Jayaprakash Neerasa , Balakishan Guniganti 
Published: March 2012

AbstractA diastereoselective, simple, and practical procedure for the title synthesis is presented.
ChemInform Abstract: Radical‐Mediated Intramolecular C—C Bond Formation and the Deoxygenation of Alcohols under Solvent‐Free Conditions with Tributyl Methyl Ammonium Hypophosphite.
Authors: Lee Eun Hwa , Cho Dae Hyan , Satyender Apuri , Jang Doo Ok 
Published: March 2012

AbstractThe use of AHP as hydrogen donor under radical conditions allows the cyclization of iodoacetals (I).
ChemInform Abstract: Facile Synthesis of Hierarchical Core—Shell Fe3O4@MgAl—LDH@Au as Magnetically Recyclable Catalysts for Catalytic Oxidation of Alcohols.
Authors: Mi Fei , Chen Xitao , Ma Yuewen , Yin Shuangtao , Yuan Fanglong , Zhang Hui 
Published: March 2012

AbstractThe title catalyst exhibits excellent activity for the oxidation of 1‐phenylethanol.
ChemInform Abstract: Graphene Oxide: An Efficient and Reusable Carbocatalyst for Aza‐Michael Addition of Amines to Activated Alkenes.
Authors: Verma Sanny , Mungse Harshal P. , Kumar Neeraj , Choudhary Shivani , Jain Suman L. , Sain Bir , Khatri Om P. 
Published: March 2012

AbstractGraphene oxide is found to be a highly efficient organocatalyst for the aza‐Michael addition of amines (I) to activated alkenes (II) and (IV).
ChemInform Abstract: A Manganese/Copper Bimetallic Catalyst for C—N Coupling Reactions under Mild Conditions in Water.
Authors: Teo Yong‐Chua , Yong Fui‐Fong , Lim Gina Shiyun 
Published: March 2012

AbstractA low cost catalytic combination of MnF2, CuI and trans‐1,2‐diaminocyclohexane is developed to allow the regioselective N‐arylation of different N‐heterocycles.
ChemInform Abstract: Kumada Coupling of Aryl, Heteroaryl, and Vinyl Chlorides Catalyzed by Amido Pincer Nickel Complexes.
Authors: Liu Ning , Wang Zhong‐Xia 
Published: March 2012

AbstractBoth NPO and PON promote the cross‐coupling of aryl, heteroaryl, and vinyl chlorides with aromatic Grignard reagents.
ChemInform Abstract: InI3/Me3SiI‐Catalyzed Direct Alkylation of Enol Acetates Using Alkyl Acetates or Alkyl Ethers.
Authors: Onishi Yoshiharu , Nishimoto Yoshihiro , Yasuda Makoto , Baba Akio 
Published: March 2012

AbstractAn environmentally friendly catalytic system for the title alkylation is presented.
ChemInform Abstract: Cobalt Oxide Supported Gold Nanoparticles as a Stable and Readily‐Prepared Precursor for the in situ Generation of Cobalt Carbonyl Like Species.
Authors: Hamasaki Akiyuki , Muto Akiko , Haraguchi Shingo , Liu Xiaohao , Sakakibara Takanori , Yokoyama Takushi , Tokunaga Makoto 
Published: March 2012

AbstractThe Co species is an efficient catalyst for the alkoxycarbonylation of epoxides and alcohols and the intra‐ and intermolecular Pauson—Khand reaction.
ChemInform Abstract: Stereoselective γ‐Olefination of Substituted Cyclobutenediones by Organocatalysis.
Authors: Beesu Mallesh , Periasamy Mariappan 
Published: March 2012

AbstractAlkyl‐substituted cyclobutenediones react with aromatic aldehydes in the presence of catalytic amounts of pyrrolidine to afford alkenyl‐substituted derivatives (III) and (V) stereoselectively.
ChemInform Abstract: Reactivity of Mixed Organozinc and Mixed Organocopper Reagents. Part 6. Nickel‐Catalyzed Coupling of Methylarylzincs with Primary Alkyl Halides: An Atom‐Economic Aryl—Alkyl Coupling.
Authors: Pekel Oezgen Oemuer , Erdik Ender 
Published: March 2012

AbstractUnder optimized conditions, the method gives the products (III) in moderate yields.
ChemInform Abstract: Homogeneous Silver(I) Salts and Heterogeneous Ag3PW12O40‐Catalyzed Intermolecular Allylation of Arenes with Allylic Alcohols.
Authors: Chen Guo‐Qiang , Xu Zhen‐Jiang , Chan Sharon Lai‐Fung , Zhou Cong‐Ying , Che Chi‐Ming 
Published: March 2012

AbstractAgOTf is reported to be effective for the allylation of electron‐rich arenes with allylic alcohols.
ChemInform Abstract: Copper‐Mediated Chelation‐Assisted ortho‐Nitration of (Hetero)arenes.
Authors: Zhang Lin , Liu Zhenhua , Li Huiqin , Fang Guichun , Barry Badru‐Deen , Belay Tuemay Abadi , Bi Xihe , Liu Qun 
Published: March 2012

AbstractOptimized conditions A) allow the preparation of various products bearing electron‐donating or electron‐withdrawing groups at the 2‐, 3‐ or 4‐positions of the phenyl ring, where 2‐pyridyl is the most effective directing group.
ChemInform Abstract: A Catalytic Asymmetric Borono Variant of Hosomi—Sakurai Reactions with N,O‐Aminals.
Authors: Huang Yi‐Yong , Chakrabarti Ananya , Morita Naohide , Schneider Uwe , Kobayashi Shu 
Published: March 2012

AbstractUnder mild Lewis acidic conditions, boronates are more reactive and selective than silicon‐based reagents.
ChemInform Abstract: TiCl4‐Promoted Mukaiyama Aldol Reaction of Fluorinated Silyl Enolates for the Construction of a Quaternary Carbon Center.
Authors: Wang Wengui , Chen Qing‐Yun , Guo Yong 
Published: March 2012

AbstractThe Mukaiyama aldol reaction of fluorinated silyl enolate (I) with various aldehydes affords α‐fluoro‐β‐hydroxyphenones with up to 86% d.e.
ChemInform Abstract: Isocyanide‐Based Multicomponent Reactions: Synthesis of Alkyl‐2‐(1‐(alkylcarbamoyl)‐2,2‐dicyanoethyl)benzoate and Isochromeno[3,4‐b]pyrrole Derivatives.
Authors: Soleimani Ebrahim , Zainali Mohsen 
Published: March 2012

AbstractBase‐catalyzed treatment of 2‐formylbenzoic acids with malononitrile and isocyanides provides a new and efficient approach to isochromenopyrroles like (IV).
ChemInform Abstract: Synthesis of Azines in Solid State: Reactivity of Solid Hydrazine with Aldehydes and Ketones.
Authors: Lee Byeongno , Lee Kyu Hyung , Cho Jaeheung , Nam Wonwoo , Hur Nam Hwi 
Published: March 2012

AbstractThe reaction proceeds by solid state grinding of a hydrazine and aldehydes or ketones to afford the conjugated azines with < 97% yield.
ChemInform Abstract: Synthesis of 2‐Naphthols via Carbonylative Stille Coupling Reaction of 2‐Bromobenzyl Bromides with Tributylallylstannane Followed by the Heck Reaction.
Authors: Dai Yao , Feng Xiujuan , Liu Hesong , Jiang Hua , Bao Ming 
Published: March 2012

AbstractThe reaction with vinylstannane also yields 2‐naphthols.
ChemInform Abstract: A New Synthesis of trans‐2,3‐Diaryloxiranes and 2‐(1H‐Benzo[d][1,2,3]triazol‐1‐yl)‐1‐arylethanols via the Reactions of 1‐Benzyl‐3‐methylbenzotriazolium Ylide with Aryl Aldehydes.
Authors: Xiao Xiaohui , Lin Daqin , Tong Shuitian , Mo Hailan 
Published: March 2012

AbstractUnder optimized conditions the reaction of aryl chlorides with benzotriazolium ylide (I) allows the highly selective formation of trans‐2,3‐diaryloxiranes.
ChemInform Abstract: Organocatalytic Asymmetric Neber Reaction for the Synthesis of 2H‐Azirine Carboxylic Esters.
Authors: Sakamoto Shota , Inokuma Tsubasa , Takemoto Yoshiji 
Published: March 2012

AbstractThe reaction of β‐ketoxime sulfonates is catalyzed by a bifunctional thiourea catalyst to afford the enantioenriched target products with good yields and high enantioselectivities.
ChemInform Abstract: Catalytic, Enantioselective Intramolecular Hydroamination of Primary Amines Tethered to Di‐ and Trisubstituted Alkenes.
Authors: Chapurina Yulia , Ibrahim Houssein , Guillot Regis , Kolodziej Emilie , Collin Jacqueline , Trifonov Alexander , Schulz Emmanuelle , Hannedouche Jerome 
Published: March 2012

AbstractThe new complexes generated form Li(thf)4[Y(CH2SiMe3)4] and the diamines (I) effectively promote the asymmetric cyclization of amine substrates.
ChemInform Abstract: Diastereoselective Synthesis of 1,3,5‐Trisubstituted 4‐Nitropyrrolidin‐2‐ones via a Nitro‐Mannich/Lactamization Cascade.
Authors: Pelletier Sophie M.‐C. , Ray Peter C. , Dixon Darren J. 
Published: March 2012

AbstractA one‐pot reaction of amines, aldehydes and nitropropanoate esters leads to the target compounds with moderate to high diastereoselectivities.
ChemInform Abstract: Synthesis and Biological Evaluation of 2‐Indolinone Derivatives as Potential Antitumor Agents.
Authors: Zou Hongbin , Zhang Liang , Ouyang Jingfeng , Giulianotti Marc A. , Yu Yongping 
Published: March 2012

AbstractA variety of 3‐substituted indolinones and azaindolinones is synthesized and evaluated for antiproliferative effects.
ChemInform Abstract: InCl3‐Catalyzed Four‐Component Reaction: A Novel Synthesis of N‐Carbazolyl Dihydropyridines.
Authors: Yamuna Ezhumalai , Zeller Matthias , Prasad Karnam Jayarampillai Rajendra 
Published: March 2012

AbstractThe efficient domino process renders possible the synthesis of various pharmaceutically important products in high yields within a short time.
ChemInform Abstract: Application of Silica Gel‐Supported Polyphosphoric Acid (PPA/SiO2) as a Reusable Solid Acid Catalyst to the Synthesis of 3‐Benzoylisoxazoles and Isoxazolines.
Authors: Itoh Ken‐ichi , Aoyama Tadashi , Satoh Hiroaki , Fujii Yuki , Sakamaki Hiroshi , Takido Toshio , Kodomari Mitsuo 
Published: March 2012

Abstract1,3‐Dipolar cycloaddition of alkynes or alkenes with nitrile oxides results in regioselective formation of the title compounds.
ChemInform Abstract: Formation of Isoxazolidines by Enantioselective Copper‐Catalyzed Annulation of 2‐Nitrosopyridine with Allylstannanes.
Authors: Chatterjee Indranil , Froehlich Roland , Studer Armido 
Published: March 2012

AbstractA Walphos‐type ligand is found to be highly efficient for the formal [3 + 2] cycloaddition to give isoazolidines (III), in most cases with excellent stereoselectivity.
ChemInform Abstract: Regioselective Synthesis and Slow‐Release Suzuki—Miyaura Cross‐Coupling of MIDA Boronate‐Functionalized Isoxazoles and Triazoles.
Authors: Grob Jonathan E. , Nunez Jill , Dechantsreiter Michael A. , Hamann Lawrence G. 
Published: March 2012

AbstractEfficient methods to prepare various 5‐arylated isoxazoles and 4‐arylated triazoles are reported.
ChemInform Abstract: One‐Pot Synthesis and Biological Evaluation of 2‐Pyrrolidinyl‐4‐amino‐5‐(3′,4′,5′‐trimethoxybenzoyl)thiazole: A Unique, Highly Active Antimicrotubule Agent.
Authors: Romagnoli Romeo , et al. et al. 
Published: March 2012

AbstractNovel thiazole derivatives (IV) and (VI) are synthesized in a facile one‐pot procedure.
ChemInform Abstract: Polycyclic N‐Heterocyclic Compounds. Part 67. Reaction of 6,7‐Substituted N‐(Quinazolin‐4‐yl)amidine Derivatives with Hydroxylamine Hydrochloride. Formation of in vitro Inhibitors of Pentosidine.
Authors: Okuda Kensuke , Muroyama Hideki , Hirota Takashi 
Published: March 2012

AbstractThe synthesis of a variety of oxadiazolylphenyl formamide oxime derivatives (V), (VI), (IX) proceeds via reaction of N‐(quinazolin‐4‐yl)amidine derivatives with hydroxylamine hydrochloride.
ChemInform Abstract: Organocatalyzed Enantioselective Synthesis of 2‐Amino‐5‐oxo‐5,6,7,8‐tetrahydro‐4H‐chromene‐3‐carboxylates.
Authors: Ramireddy Naresh , Abbaraju Santhi , Zhao Cong‐Gui 
Published: March 2012

AbstractCondensation of cyclic 1,3‐diones with alkylidene cyanoacetates in the presence of the quinine‐based thiourea renders possible the preparation of various biologically interesting benzopyran structures.
ChemInform Abstract: Rhodium(III)‐Catalyzed Synthesis of Pyridines from α,β‐Unsaturated Ketoximes and Internal Alkynes.
Authors: Too Pei Chui , Noji Toshiharu , Lim Ying Jie , Li Xingwei , Chiba Shunsuke 
Published: March 2012

AbstractUnder optimized conditions, the reaction allows the synthesis of highly substituted products.
ChemInform Abstract: The Synthesis of 2‐Nitroaryl‐1,2,3,4‐tetrahydroisoquinolines, Nitro‐Substituted 5,6‐Dihydrobenzimidazo[2,1‐a]isoquinoline N‐Oxides and Related Heterocycles as Potential Bioreducible Substrates for the Enzymes NAD(P)H: Quinone Oxidoreductase 1 and E. coli Nitroreductase.
Authors: Burke Philip J. , Wong Lai Chun , Jenkins Terence C. , Knox Richard J. , Stanforth Stephen P. 
Published: March 2012

AbstractA series of title compounds is prepared and evaluated as potential bioreducible substrates for the enzymes NAD(P)H: quinone oxireductase 1 (NQO1) and Escherichia coli nitroreductase (NR).
ChemInform Abstract: Tandem One‐Pot Synthesis of Polysubstituted Pyridines Using the Blaise Reaction Intermediate and 1,3‐Enynes.
Authors: Chun Yu Sung , Lee Jun Hee , Kim Ju Hyun , Ko Young Ok , Lee Sang‐gi 
Published: March 2012

AbstractSequential reaction of nitriles, Reformatsky reagents and 1,3‐enynes proceeds with complete regio‐ and chemoselectivity to provide the polysubstituted pyridines.
ChemInform Abstract: Solvent‐Free Sonochemical One‐Pot Three‐Component Synthesis of 2H‐Indazolo[2,1‐b]phthalazine‐1,6,11‐triones and 1H‐Pyrazolo[1,2‐b]phthalazine‐5,10‐diones.
Authors: Shukla Gaurav , Verma Rajiv K. , Verma Girijesh K. , Singh Maya Shankar 
Published: March 2012

AbstractThe reaction under conventional heating or ultrasound gives the title compounds in comparable yields and reaction times.
ChemInform Abstract: New Imidazo[2,1‐b]thiazole Derivatives: Synthesis, in vitro Anticancer Evaluation, and in silico Studies.
Authors: Park Jin‐Hun , El‐Gamal Mohammed I. , Lee Yong Sup , Oh Chang‐Hyun 
Published: March 2012

AbstractCompounds (IIIb), (IIIf), (IVb), and (IVd)—(IVg) exhibit higher activity against A375P human melanoma cell line than the reference compound sorafenib.
ChemInform Abstract: Design, Synthesis and Biological Study of Novel Pyrido[2,3‐d]pyrimidine as Antiproliferative CDK2 Inhibitors.
Authors: Ibrahim Diaa A. , Ismail Nasser S. M. 
Published: March 2012

AbstractDesign and synthesis of a small library of 4‐aminopyrido[2,3‐d]pyrimidine derivatives are reported.
ChemInform Abstract: Synthesis and in vitro EGFR (ErbB1) Tyrosine Kinase Inhibitory Activity of 4‐N‐Substituted 6‐Aryl‐7H‐pyrrolo[2,3‐d]pyrimidine‐4‐amines.
Authors: Kaspersen Svein Jacob , Soerum Christopher , Willassen Veronica , Fuglseth Erik , Kjoebli Eli , Bjoerkoey Geir , Sundby Eirik , Hoff Baard Helge 
Published: March 2012

AbstractTitle compounds like (VIII) are synthesized and tested for their in vitro EGFR (ErbB1) tyrosine kinase inhibitory activity.
ChemInform Abstract: Facile Syntheses of 7,9‐Dimethoxypyrrolo[3,2,1‐ij]quinolin‐6‐ones.
Authors: Rajput Santosh , Leu Chao‐wei , Wood Kasey , Black David StC , Kumar Naresh 
Published: March 2012

AbstractTwo approaches starting from indoles (I) or quinolinone (VIII) are presented for the synthesis of title compounds (V) and (XI), respectively.
ChemInform Abstract: Phosphorus Pentachloride‐Induced Transformation of (1,2,3‐Thiadiazol‐5‐yl)hydrazones of Acetophenone.
Authors: Kalinina T. A. , Prokhorova P. E. , Glukhareva T. V. , Morzherin Yu. Yu. 
Published: March 2012

AbstractThe transformation of the 1,2,3‐thiadiazole moiety of title compounds (I), induced by phosphorus pentachloride, involves 4 atoms of the side chain and leads to triazolothiadiazine‐3‐carbonyl chlorides (II).
ChemInform Abstract: Polyethylene Glycol (PEG‐400) as an Efficient and Recyclable Reaction Medium for the One‐Pot Synthesis of N‐Substituted Azepines under Catalyst‐Free Conditions.
Authors: Mallepalli Raghu , Yeramanchi Lingappa , Bantu Rajashaker , Nagarapu Lingaiah 
Published: March 2012

AbstractA facile synthesis of N‐substituted azepine 2,3‐diesters is achieved through three‐component condensation in PEG 400 without the need for any catalyst.
ChemInform Abstract: The N‐Aryl Aminocarbonyl ortho‐Substituent Effect in Cu‐Catalyzed Aryl Amination and Its Application in the Synthesis of 5‐Substituted 11‐Oxo‐dibenzodiazepines.
Authors: Diao Xiaoqiong , Xu Lanting , Zhu Wei , Jiang Yongwen , Wang Haoyang , Guo Yinlong , Ma Dawei 
Published: March 2012

AbstractA variety of biologically important 11‐oxodibenzodiazepines is prepared tolerating a wide range of functional groups in the amine partner and substitution at both aromatic rings.
ChemInform Abstract: Synthesis and in vitro Anticancer Activity of 6,7‐Methylenedioxy (or 5‐Hydroxy‐6‐methoxy)‐2‐(substituted selenophenyl)quinolin‐4‐one Analogues.
Authors: Kuo Sheng‐Chu , et al. et al. 
Published: March 2012

AbstractA modified Camps approach is used for the synthesis of quinoline derivatives (IV).