bluuebunny/crossref_metadata_2025_split huggingface dataset:
ChemInform Abstract: Co(III)(salen)‐Catalyzed HKR of Two Stereocentered Alkoxy‐ and Azido Epoxides: A Concise Enantioselective Synthesis of (S,S)‐Reboxetine and (+)‐epi‐Cytoxazone.
Authors: Reddy R. Santhosh , Chouthaiwale Pandurang V. , Suryavanshi Gurunath , Chavan Vilas B. , Sudalai Arumugam 
Published: October 2010

AbstractChiral cobalt complexes are efficient catalysts for the hydrolytic kinetic resolution of a variety of syn‐ and anti‐epoxides.
ChemInform Abstract: Chiral Induction by Cinchona Alkaloids in the Rhodium(II) Catalyzed O—H Insertion Reaction.
Authors: Saito Hiroaki , Iwai Ryo , Uchiyama Taketo , Miyake Muneharu , Miyairi Shinichi 
Published: October 2010

AbstractA highly efficient method for the catalytic enantioselective O‐H insertion reaction of α‐phenyldiazoacetate is presented.
ChemInform Abstract: An Alkynylboronate Cycloaddition Strategy to Functionalized Benzyne Derivatives.
Authors: Kirkham James D. , Delaney Parick M. , Ellames George J. , Row Eleanor C. , Harrity Joseph P. A. 
Published: October 2010

AbstractThe cycloaddition of 2‐pyrones with alkynylboronate (II) followed by C‐B bond oxidation and a subsequent triflation gives rise to mixtures of regioisomers (VI) and (VII), which are shown to be useful benzyne precursors.
ChemInform Abstract: Highly Efficient Solvent‐Free Catalytic Hydrogenation of Solid Alkenes and Nitro‐Aromatics Using Pd Nanoparticles Entrapped in Aluminum Oxy‐Hydroxide.
Authors: Chang Fei , Kim Hakwon , Lee Byeongno , Park Sungho , Park Jaiwook 
Published: October 2010

AbstractThe substrates are hydrogenated without further reduction of other functional groups.
ChemInform Abstract: A Simple and Efficient Thiocyanation of Indoles, Anilines and Keto Compounds Catalyzed by a Polystyrene Resin Amberlyst‐15.
Authors: Lenin Racha , Raju Rallabandi M. 
Published: October 2010

AbstractAdvantages of the title procedure are the mild reaction conditions, the ease of product isolation, and the cheap and commercially available catalyst.
ChemInform Abstract: Autoxidative Carbon—Carbon Bond Formation from Carbon—Hydrogen Bonds.
Authors: Pinter Aron , Sud Abhishek , Sureshkumar Devarajulu , Klussmann Martin 
Published: October 2010

AbstractActivated benzylic CH2‐groups in xanthene (I) or dihydroacridines (IV) undergo acid‐catalyzed oxidative coupling towards carbonyl compounds.
ChemInform Abstract: Stereoselective Synthesis of 1,2,3,4‐Tetrasubstituted Dienes from Allenoates and Aldehydes: An Observation of Phosphine‐Induced Chemoselectivity.
Authors: Xu Silong , Zou Wen , Wu Guiping , Song Haibin , He Zhengjie 
Published: October 2010

AbstractThe choice of phosphine is important for the course of the title reaction.
ChemInform Abstract: Acid Catalyzed Reaction of Indanones, Tetralones and Benzosuberone with Neopentyl Glycol and Other Alkanediols under Forced Conditions.
Authors: Imai Masao , Ribeiro Morais Goreti , al‐Hindawi Bassam , al‐Sulaibi Mazen A. M. , Meetani Mohammad , Thiemann Thies 
Published: October 2010

Abstractα‐Benzocycloalkenones in general form benzocycloalkadienes when they are subjected to reactions with neopentyl glycol or other alkanediols under forced conditions.
ChemInform Abstract: Rasta Resin‐PPh3 and Its Use in Chromatography‐Free Wittig Reactions.
Authors: Leung Peter Shu‐Wai , Teng Yan , Toy Patrick H. 
Published: October 2010

AbstractA novel heterogeneous polystyrene‐based phosphine is used for in situ generation of phosphorane reactant for the Wittig reaction with aldehydes.
ChemInform Abstract: Catalytic Asymmetric Roskamp Reaction of α‐Alkyl‐α‐diazoesters with Aromatic Aldehydes: Highly Enantioselective Synthesis of α‐Alkyl‐β‐keto Esters.
Authors: Li Wei , Wang Jun , Hu Xiaolei , Shen Ke , Wang Wentao , Chu Yangyang , Lin Lili , Liu Xiaohua , Feng Xiaoming 
Published: October 2010

AbstractThe e.e.‐values shown are determined after silica gel chromatography.
ChemInform Abstract: Decarboxylative Benzylations of Alkynes and Ketones.
Authors: Torregrosa Robert R. P. , Ariyarathna Yamuna , Chattopadhyay Kalicharan , Tunge Jon A. 
Published: October 2010

AbstractA new catalytic decarboxylative benzylation of alkynes and ketones without the use of strong bases and/or organometallics is developed.
ChemInform Abstract: The Use of Polyhedral Oligomeric Silsesquioxane (POSS) as a Soluble Support for Organic Synthesis: A Case Study with a POSS‐Bound Isocyanate Scavenger Reagent.
Authors: York Mark , Evans Richard A. 
Published: October 2010

AbstractThe use of POSS for the scavenging of hydrogen chloride allows the high‐yielding preparation of amides and a sulfonamide with high purity.
ChemInform Abstract: A Convenient Procedure for the Preparation of Bis(dialkylamino)malononitriles.
Authors: Tiritiris Ioannis , Kantlehner Willi 
Published: October 2010

AbstractExothermic reaction of chloroformamidinium chlorides (I) with trimethylsilyl cyanide under neat reaction conditions gives the chemically interesting title compounds in good yields.
ChemInform Abstract: TCCA‐Promoted Solvent‐Free Chemoselective Synthesis of Thiosulfonates on Grinding.
Authors: Xu Yali , Peng Yong , Sun Junhui , Chen Jiuxi , Ding Jinchang , Wu Huayue 
Published: October 2010

AbstractSymmetric, aromatic disulfides (I) containing electron‐donating and electron‐withdrawing groups are oxidized equally well by trichloroisocyanuric acid upon grinding with a pestle in a mortar.
ChemInform Abstract: Alkyl 2‐Alkoxy(aryloxy)‐2‐isocyanato‐3,3,3‐trifluoropropionates
Authors: Sokolov V. B. , Goreva T. V. , Epishina T. A. , Aksinenko A. Yu. 
Published: October 2010

Abstractsynthesis of the previously unknown title compounds (IV) and transformation into urea derivatives (VI) (11 examples)
ChemInform Abstract: The Conversion of Alkynes into Substituted Cyclopropanes Effected by CH2I2—R3Al (R: Me, Et, i‐Bu).
Authors: Ramazanov Ilfir R. , Dil'mukhametova Leisan K. , Dzhemilev Usein M. , Nefedov Oleg M. 
Published: October 2010

AbstractThe cyclopropanation reaction of internal and terminal alkynes with diiodomethane in the presence of trimethylaluminum (III) provides access towards β‐iodoethyl‐substituted cyclopropanes, e.g. (IV), (VIII), (XI).
ChemInform Abstract: Gold(I)‐Catalyzed Intermolecular [2 + 2] Cycloaddition of Alkynes with Alkenes.
Authors: Lopez‐Carrillo Veronica , Echavarren Antonio M. 
Published: October 2010

AbstractA sterically hindered cationic Au(I) complex is used as catalyst in the intramolecular reaction of terminal alkynes with alkenes that results in a [2 + 2] cycloaddition.
ChemInform Abstract: Selective Synthesis of α‐Methylenyl Zirconacyclopentene via Cross‐Coupling of Alkyne and Allene.
Authors: Zheng Weixin , Wu Yangfeng , Zheng Fenfen , Hu Linfeng , Hong Ya 
Published: October 2010

AbstractReductive intermolecular cross‐coupling of alkynes with allenes, promoted by ZrEt2Cp2, gives the title zirconacycle.
ChemInform Abstract: Amination of Aryl Iodides Using a Fluorous‐Tagged Ammonia Equivalent.
Authors: Nielsen Simon Dalsgaard , Smith Garrick , Begtrup Mikael , Kristensen Jesper Langgard 
Published: October 2010

AbstractThe Cu‐catalyzed amination of aryl iodides using a fluorous‐tagged ammonia equivalent is described.
ChemInform Abstract: Highly Enantioselective Rh‐Catalyzed Transfer Hydrogenation of N‐Sulfonyl Ketimines.
Authors: Kwak Se Hun , Lee Sun Ah , Lee Kee‐In 
Published: October 2010

AbstractA wide range of aromatic N‐sulfonylimines successfully undergoes Rh‐catalyzed transfer hydrogenation to give the corresponding benzylic amines (II) in excellent yields and enantioselectivity.
ChemInform Abstract: An Effective Aza‐Michael Addition of Aromatic Amines to Electron‐Deficient Alkenes in Alkaline Al2O3.
Authors: Ai Xin , Wang Xin , Liu Jin‐ming , Ge Ze‐mei , Cheng Tie‐ming , Li Run‐tao 
Published: October 2010

AbstractA wide range of aromatic and aliphatic primary and secondary amines smoothly undergoes aza‐Michael reaction with electron‐deficient olefins in the presence of alkaline alumina.
ChemInform Abstract: Silver Oxide as a Novel Catalyst for Carbon—Carbon Bond‐Forming Reactions in Aqueous Media.
Authors: Ueno Masaharu , Tanoue Arata , Kobayashi Shu 
Published: October 2010

AbstractSilver oxide is found to be an excellent catalyst for allylation reactions of allyltributyltins (II) and (IV) with aldehydes (I) in aqueous media.
ChemInform Abstract: Microwave‐Assisted Synthesis of Aromatic Bis‐Esters in Liquid Phase.
Authors: Zbancioc Gheorghita N. , Zbancioc Ana Maria V. , Mangalagiu Ionel I. 
Published: October 2010

AbstractThe synthesis of bis‐esters of type (III), (VI), or (IX) proceeds in higher yields and with considerably shorter reaction times when conducted under microwave irradiation compared to conventional heating.
ChemInform Abstract: Highly Enantioselective Michael Addition of Aldehydes to Nitroolefins Catalyzed by Primary Amine Thiourea Organocatalysts.
Authors: Chen Jia‐Rong , Zou You‐Quan , Fu Liang , Ren Fan , Tan Fen , Xiao Wen‐Jing 
Published: October 2010

AbstractBifunctional cinchonidine‐derived thiourea catalysts (I), (II) are prepared for the highly enantioselective Michael addition of α‐branched aldehydes towards aromatic nitroolefins.
ChemInform Abstract: Camphor‐10‐sulfonamide‐Based Prolinamide Organocatalyst for the Direct Intermolecular Aldol Reaction Between Ketones and Aromatic Aldehydes.
Authors: Rani Rashmi , Peddinti Rama Krishna 
Published: October 2010

AbstractAsymmetric aldol reaction of six‐membered cyclic ketones (I) and (IV) with aromatic aldehydes (II) in the presence of a CSA‐derived prolinamide organocatalyst provides access to the aldol adducts (III) and (V), resp., in good yields and stereoselectivities (up to 98% d.e., and <99% e.e.).
ChemInform Abstract: VB1—Al2O3‐Catalyzed One‐Pot Condensation of Aromatic Ketone, Aromatic Aldehyde, and Amide.
Authors: Lei Min , Ma Lei , Hu Lihong 
Published: October 2010

AbstractVitamin B1 immobilized on Al2O3, is described as an efficient catalyst for the three‐component condensation.
ChemInform Abstract: Domino [3 + 3] Annulation/Ring‐Cleavage Reactions of 1,3‐Bis(trimethylsilyloxy)‐1,3‐butadienes with 5‐Aryl‐ and 5‐Vinyl‐3‐acyl‐4,5‐dihydrofurans: Efficient Synthesis of 5‐(4‐Chlorobut‐2‐en‐1‐yl)‐ and 5‐(2‐Aryl‐2‐chloroethyl)salicylates.
Authors: Lau Matthias , Sher Muhammad , Villinger Alexander , Fischer Christine , Langer Peter 
Published: October 2010

AbstractThe title reactions afford highly functionalized arenes, that are not readily available by other methods.
ChemInform Abstract: A New Method of Reducing 2‐Mercapto‐Substituted 1,3,4‐Oxadiazoles: Synthesis of Acylhydrazine Derivatives.
Authors: Zareef Muhammad , Iqbal Rashid , Zaidi Javid Hussain , Arfan Muhammad , Ali Muhammad , Khan Khalid M. 
Published: October 2010

AbstractThe synthesis of acylhydrazines (III) is achieved for the first time by reduction of unsymmetrical oxadiazoles (I) by using sodium borohydride /AcOH combination, followed by conversion to the corresponding sulfonamide derivatives (III).
ChemInform Abstract: Facile Synthesis of Palladium Nanoparticles with High Chemical Activity Using Cucurbit[6]uril as Protecting Agent.
Authors: Cao Minna , Lin Jingxiang , Yang Hongxun , Cao Rong 
Published: October 2010

AbstractUsing curcubit[6]uril as protecting agent, well‐defined Pd nanoparticles are prepared.
ChemInform Abstract: Chiral Chalcogen Peptides as Ligands for the Catalytic Enantioselective Aryl Transfer Reaction to Aldehydes.
Authors: Schwab Ricardo S. , Soares Letiere C. , Dornelles Luciano , Rodrigues Oscar E. D. , Paixao Marcio W. , Godoi Marcelo , Braga Antonio L. 
Published: October 2010

AbstractA new class of chiral chalcogen peptide based ligands is prepared and applied in the zinc‐catalyzed addition of arylboronic acids to aldehydes.
ChemInform Abstract: Ionic Liquids in Barbier—Zaitsev Reaction. Synthesis of 1‐(Perfluorophenyl)‐2‐phenylethanol in the Presence of Iron Pentacarbonyl.
Authors: Vasil'eva T. T. , Ambartsumyan A. A. , Chakhovskaya O. V. , Kochetkov K. A. 
Published: October 2010

AbstractThis is the first example for a Barbier—Zaitsev reaction of pentafluorobenzaldehyde promoted by iron pentacarbonyl in the presence of an equimolar amount of ionic liquid.
ChemInform Abstract: 4‐Thio Derivatives of Dibenzosuberone: Potential Antidepressant Compounds.
Authors: Martins Paulo R. C. , Romeiro Gilberto A. , Ribeiro Carlos M. R. 
Published: October 2010

AbstractTitle compounds are prepared by regioselective iodination with Tl(tfa)3/KI followed by a modified Ullmann reaction.
ChemInform Abstract: Thiol‐Mediated Tandem Michael—Aldol Reaction: A Convenient Method for the Synthesis of Fused Cyclopentenones.
Authors: Samanta Shubhankar , Yasmin Nasima , Kundu Debasish , Ray Jayanta K. 
Published: October 2010

AbstractEsters of type (I) bearing a formyl group are treated with methyl thioglycolate in order to get thiopyrans of type (IV).
ChemInform Abstract: Asymmetric Organocatalytic Michael Addition of Anthrone to Enone.
Authors: Wu Chunlin , Li Wenjun , Yang Juanjuan , Liang Xinmiao , Ye Jinxing 
Published: October 2010

AbstractThe Michael addition of anthrones (I) towards enones (II) and (IV) is achieved in high yields and enantioselectivities (up to 93% e.e.) in the presence of a novel quinine‐derived thiourea catalyst.
ChemInform Abstract: Gold‐Catalyzed One‐Step Practical Synthesis of Oxetan‐3‐ones from Readily Available Propargylic Alcohols.
Authors: Ye Longwu , He Weimin , Zhang Liming 
Published: October 2010

AbstractThis strategy uses alkynes as synthetic equivalents to α—diazoketones for accessing intermediary α—oxo metal carbenes.
ChemInform Abstract: N‐Heterocyclic Carbene Catalyzed [2 + 2] Cycloaddition of Aryl Isothiocyanates and Nitroolefines: An Efficient Synthesis of β‐Thiolactams.
Authors: Awasthi Chhama , Yadav Lal Dhar S. 
Published: October 2010

AbstractThe reaction proceeds with high diastereoselectivity in favor of the cis‐substituted products.
ChemInform Abstract: Tetrahydrofurans from Substituted Hex‐5‐yne‐1,4‐diols.
Authors: Schwehm Carolin , Wohland Max , Maier Martin E. 
Published: October 2010

AbstractIt is discovered that hex‐5‐yne‐1,4‐diols of type (I) undergo metal‐catalyzed Meyer—Schuster rearrangement followed by an intramolecular Michael addition to yield 2,5‐disubstituted tetrahydrofurans.
ChemInform Abstract: Quaternary Ammonium (Hypo)iodite Catalysis for Enantioselective Oxidative Cycloetherification.
Authors: Uyanik Muhammet , Okamoto Hiroaki , Yasui Takeshi , Ishihara Kazuaki 
Published: October 2010

AbstractAsymmetric oxidative cyclization of ketophenols (I) proceeds smoothly in the presence of an in situ generated chiral quaternary ammonium hypoiodite to afford 2‐acyldihydrobenzofuran derivatives (II) in up to 92% optical purity.
ChemInform Abstract: 1‐Bromo‐2‐trifluoroacetylcyclobutenes as Novel Building Blocks for the Construction of Trifluoromethyl Substituted Heterocycles. Part 2. Synthesis of Trifluoromethyl Substituted Thiophenes, Condensed with Cyclobutene Moieties.
Authors: Koldobskii Andrey B. , Tsvetkov Nikolay P. , Solodova Ekaterina V. , Kalinin Valery N. 
Published: October 2010

AbstractA novel general method for the construction of cyclobutarenes containing trifluoromethylated thiophenes fused with the strained cyclobutene ring is elaborated.
ChemInform Abstract: Domino Allylic Amination/Sonogashira/Heterocyclization Reactions: Palladium‐Catalyzed Three‐Component Synthesis of Pyrroles.
Authors: Lamande‐Langle Sandrine , Abarbri Mohamed , Thibonnet Jerome , Duchene Alain , Parrain Jean‐Luc 
Published: October 2010

AbstractOptimal reaction conditions are found for the three‐component synthesis of pyrroles (IV), (VI), and (IX).
ChemInform Abstract: Synthesis, Antibacterial Activity Evaluation and QSAR Studies of Novel Dispiropyrrolidines.
Authors: Karthikeyan K. , Sivakumar P. M. , Doble M. , Perumal P. T. 
Published: October 2010

AbstractCycloaddition of an azomethine ylide, generated in situ from isatins (IV) and sarcosine (V), with the dipolarophile (III) yields the dispiropyrrolidines (VI) in good yields.
ChemInform Abstract: Synthesis, Analgesic and Antiinflammatory Activities of Some Novel Pyrazolines Derivatives.
Authors: Joshi Ratnadeep S. , Mandhane Priyanka G. , Diwakar Santosh D. , Dabhade Sanjay K. , Gill Charansingh H. 
Published: October 2010

AbstractThe title compounds (IIa), (IIb), (IId), (IVa), (IVc), and (IVd) exhibit good analgesic and antiinflammatory inhibition and are almost equipotent to the standard compound.
ChemInform Abstract: Isoprene‐Mediated Lithiation of 1‐Alkylimidazoles: Chiral Induction of the Alkyl Substituent.
Authors: Pastor Isidro M. , Torregrosa Rosario , Yus Miguel 
Published: October 2010

AbstractThe isoprene‐mediated lithiation of imidazoles (IV) bearing a secondary alkyl substituent at the nitrogen and subsequent nucleophilic addition to aldehydes and ketones (V) allows the preparation of the corresponding 2‐functionalized imidazoles (VI).
ChemInform Abstract: Amino Acid Derivatives. Part 4. Synthesis and anti‐HIV Activity of New Naphthalene Derivatives.
Authors: Hamad Nawar S. , Al‐Haidery Nahed H. , Al‐Maosudi Iman A. , Sabri Mey , Sabri Luma , Al‐Masoudi Najim A. 
Published: October 2010

AbstractAmong the compounds synthesized, derivative (VI) is found to be a potent inhibitor in vitro for the replication of HIV‐1.
ChemInform Abstract: Synthesis and Antiproliferative Evaluation of 5‐oxo and 5‐thio Derivatives of 1,4‐Diaryl Tetrazoles.
Authors: Gundugola Aditya S. , Chandra Kusum Lata , Perchellet Elisabeth M. , Waters Andrew M. , Perchellet Jean‐Pierre H. , Rayat Sundeep 
Published: October 2010

AbstractA series of title compounds are tested for their antiproliferative activities.
ChemInform Abstract: Synthesis and Theoretical Studies of Gallium Complexes Back‐Shielded by a Cage‐Shaped Framework of Tris(m‐oxybenzyl)arene.
Authors: Nakajima Hideto , Yasuda Makoto , Chiba Kouji , Baba Akio 
Published: October 2010

AbstractFour novel cage‐shaped gallium complexes (I) are prepared and evaluated for their catalytic activity in a hetero Diels—Alder reaction of Danishefsky′s diene (II) with benzaldehyde.
ChemInform Abstract: Regioselective Vinylation of Kojic Acid Using Acetylenic Esters in the Presence of Triphenylphosphine or tert‐Butyl Isocyanide.
Authors: Asghari Sakineh , Faraji‐Najjarkolaee Maryam , Ahmadipour Mohammad 
Published: October 2010

AbstractPPh3‐mediated reaction of Kojic acid (I) with acetylenedicarboxylates (II) gives the C‐vinylated products (III), whereas the tBuNC‐mediated reaction of (I) with acetylenecarboxylates (IV) under similar conditions provides the O‐vinylated products (V).
ChemInform Abstract: Synthesis and in vitro Cytotoxicity of Poly‐Functionalized 4‐(2‐Arylthiazol‐4‐yl)‐4H‐chromenes.
Authors: Foroumadi Alireza , et al. et al. 
Published: October 2010

AbstractA new series of thiazolylchromene derivatives (IV) is synthesized via one‐pot, three‐component condensation of thiazolecarbaldehyde (III) with m‐aminophenol (I) and malononitrile.
ChemInform Abstract: Synthetic and Biological Studies on Some Fused Pyrazoles (VI) and Their Ethoxyphthalimide Derivatives (VIII).
Authors: Joshi Ajit , Sain Devendra K. , Thadhaney Bhawana , Ojha Swati , Hussain Nasir , Talesara Ganpat L. 
Published: October 2010

AbstractDerivatives (VIIIc) and (VIIId) show moderate to good antimicrobial activities.
ChemInform Abstract: Synthesis of 2‐Halogenated Quinolines by Halide‐Mediated Intramolecular Cyclization of o‐Alkynylaryl Isocyanides.
Authors: Mitamura Takenori , Nomoto Akihiro , Sonoda Motohiro , Ogawa Akiya 
Published: October 2010

AbstractDifferent types of halide sources are used for the preparation of the title quinolines.
ChemInform Abstract: Metal‐Free Reductions of N‐Heterocycles via Lewis Acid Catalyzed Hydrogenation.
Authors: Geier Stephen J. , Chase Preston A. , Stephan Douglas W. 
Published: October 2010

AbstractThe B(C6F5)3‐catalyzed hydrogenation of quinolines (I) proceeds readily to afford 1,2,3,4‐tetrahydroquinolines (II) in good yields.
ChemInform Abstract: Novel Pyridobenzimidazole Derivatives Exhibiting Antifungal Activity by the Inhibition of β‐1,6‐Glucan Synthesis.
Authors: Takeshita Hiroshi , Watanabe Jun , Kimura Yoichi , Kawakami Katsuhiro , Takahashi Hisashi , Takemura Makoto , Kitamura Akihiro , Someya Kazuhiko , Nakajima Ryohei 
Published: October 2010

AbstractSeveral title compounds of type (VI), (VIII), or (IX) are evaluated for their antifungal activities.
ChemInform Abstract: Novel Thiophenes, Thienopyrimidines, and Triazolothienopyrimidines for the Evaluation of Anticancer and Augmentation Effects of γ‐Radiation.
Authors: Shaaban Mohamed A. , Ghorab Mostafa M. , Heiba Helmy I. , Kamel Mona M. , Zaher Nashwa H. , Mostafa Mohamed I. 
Published: October 2010

AbstractCompounds (III), (IV), (VIII) and (X) show significant in vitro cytotoxic activity against hepatocellular carcinoma compared to the reference drug doxorubicin.
ChemInform Abstract: Synthesis of 2‐(4‐Substitutedsulfonyl piperazin‐1‐yl‐methyl)‐3‐aryl‐quinazolin‐4(3H)‐one.
Authors: Acharyulu Palle V. R. , Dubey P. K. , Reddy P. V. V. Prasada , Suresh Thatipally 
Published: October 2010

AbstractSimple, efficient and novel routes for the synthesis of the title compounds (VI) (9 examples) are given.
ChemInform Abstract: Synthesis, Characterization and in vitro Antimicrobial Studies of New 2,3‐Disubstituted Quinazolin‐4(3H)‐ones of 2‐[2‐(2,6‐Dichlorophenyl)amino]phenyl Acetic Acid.
Authors: Patel Navin B. , Shaikh Asif R. 
Published: October 2010

AbstractMost of the synthesized compounds (VII) (15 examples) show comparable antibacterial activity like ampicillin and strong activity against C.
ChemInform Abstract: Nickel‐Catalyzed Regio‐ and Enantioselective Annulation Reactions of 1,2,3,4‐Benzothiatriazine‐1,1(2H)‐dioxides with Allenes.
Authors: Miura Tomoya , Yamauchi Motoshi , Kosaka Akira , Murakami Masahiro 
Published: October 2010

AbstractA wide range of benzothiazine dioxides is smoothly prepared by Ni‐catalyzed asymmetric recyclization of title benzothiatriazine dioxides (I), (VII) with allenes.
ChemInform Abstract: Intramolecular N‐Arylation in Heterocyclization: Synthesis of New Pyrido‐Fused Pyrrolo[1,2‐a][1,4]diazepinones.
Authors: Legeren Loreto , Dominguez Domingo 
Published: October 2010

AbstractOptimized reaction conditions are developed for the cyclization of pyridine‐substituted L‐proline amides to give the title compounds via intramolecular N‐arylation.
ChemInform Abstract: A Tailored Hybrid BODIPY—Oligothiophene Donor for Molecular Bulk Heterojunction Solar Cells with Improved Performances.
Authors: Rosseau Theodulf , Cravino Antonio , Ripaud Emilie , Leriche Philippe , Rihn Sandra , De Nicola Antoinette , Ziessel Raymond , Roncali Jean 
Published: October 2010

AbstractFixation of a hexyl‐2,2′‐bithienyl unit on a conjugated BODIPY donor increases the conversion efficiency of the resulting molecular bulk heterojunction solar cell significantly.
ChemInform Abstract: Full Chirality Transfer in the Conversion of Secondary Alcohols into Tertiary Boronic Esters and Alcohols Using Lithiation—Borylation Reactions.
Authors: Bagutski Viktor , French Rosalind M. , Aggarwal Varinder K. 
Published: October 2010

AbstractNew reaction conditions for the synthesis of enantioenriched tertiary boronic esters or alcohols are developed.
ChemInform Abstract: Dichotomous Reactivity in the Reaction of Triethyl‐ and Triphenylphosphane HBr Salts with Dimethyl Acetals: A Novel Entry to α‐Alkoxy‐Functionalized Ylides and General Synthesis of Vinyl Ethers and Alkoxy Dienes.
Authors: Das Priyabrata , McNulty James 
Published: October 2010

AbstractThe reaction of triethylphosphane hydrobromide with dimethyl acetals gives the corresponding α‐methoxy phosphonium salts under mild conditions.
ChemInform Abstract: Nonenzymatic Kinetic Resolution of Racemic β‐Hydroxyalkanephosphonates with a Chiral Copper Catalyst.
Authors: Moriyama Atsushi , Matsumura Shintaro , Kuriyama Masami , Onomura Osamu 
Published: October 2010

AbstractA wide range of aromatic and aliphatic β‐hydroxyphosphonates (I) and (IV) is kinetically resolved via o‐fluorobenzoylation in the presence of a Cu—box catalyst.