bluuebunny/crossref_metadata_2025_split huggingface dataset:
ChemInform Abstract: Simple Chiral Sulfonamide Primary Amine Catalyzed Highly Enantioselective Michael Addition of Malonates to Enones.
Authors: Luo Chunhua , Jin Yu , Du Da‐Ming 
Published: September 2012

AbstractThe sulfonamide catalyst, which is readily available from chiral 1,2‐diamine, is successfully applied to the cheap and facile title reaction.
ChemInform Abstract: Reaction Discovery by Using a Sandwich Immunoassay.
Authors: Quinton Julia , Kolodych Sergii , Chaumonet Manon , Bevilacqua Valentina , Nevers Marie‐Claire , Volland Herve , Gabillet Sandra , Thuery Pierre , Creminon Christophe , Taran Frederic 
Published: September 2012

AbstractTwo novel reactions, a copper‐catalyzed desulfuration of thioureas leading to isoureas and a copper‐promoted cyclization reaction leading to thiazoles from alkynes and N‐hydroxy thioureas are discovered using a sandwich immunoassay screening technique which allows to measure at least 1000 reaction yields per day by a single operator.
ChemInform Abstract: Metal‐Free Synthesis of Allylic Amines by Cross‐Dehydrogenative‐Coupling of 1,3‐Diarylpropenes with Anilines and Amides under Mild Conditions.
Authors: Wang Zhiming , Mo Hanjie , Cheng Dongping , Bao Weiliang 
Published: September 2012

AbstractA highly facile, efficient, mild, and new method for the synthesis of the title amines is presented.
ChemInform Abstract: Palladium Nanoparticles Supported on a Poly(N‐vinyl‐2‐pyrrolidone)‐Modified Mesoporous Carbon Nanocage as a Novel Heterogeneous Catalyst for the Heck Reaction in Water.
Authors: Kalbasi Roozbeh Javad , Mosaddegh Neda , Abbaspourrad Alireza 
Published: September 2012

AbstractThe title Pd‐catalyst is successfully applied to the Heck reaction of aromatic aryl halides and styrene to give E‐stilbenes.
ChemInform Abstract: Pd‐Catalyzed Cross‐Coupling of Aryl Carboxylic Acids with Propiophenones Through a Combination of Decarboxylation and Dehydrogenation.
Authors: Zhou Jun , Wu Ge , Zhang Min , Jie Xiaoming , Su Weiping 
Published: September 2012

AbstractThe reaction (II) to propiophenones proceeds under adjusted conditions to give chalcones (III) and (V) tolerating a variety of functional groups.
ChemInform Abstract: One‐Pot Solvent‐Free Sonochemical Synthesis of 1‐Amidoalkyl‐2‐naphthols.
Authors: Puri Saurabh , Kaur Balbir , Parmar Anupama , Kumar Harish 
Published: September 2012

AbstractA general, efficient and eco‐friendly procedure for the synthesis of 1‐amidoalkylnaphthols (IV) (12 examples) via a ultrasound‐mediated three‐component reaction is given.
ChemInform Abstract: Microwave Assisted Synthesis of Spirocyclic Pyrrolidines — σ1 Receptor Ligands with Modified Benzene‐N‐distance.
Authors: Jasper Annemarie , Schepmann Dirk , Lehmkuhl Kirstin , Vela Jose Miguel , Buschmann Helmut , Holent Joerg , Wuensch Bernhard 
Published: September 2012

AbstractSpirocyclic benzofurans (IV), (V) and (VII) as well as the corresponding benzopyrans are produced and tested as 1:1 mixtures of cis and trans diastereomers.
ChemInform Abstract: Copper Bis(oxazolines) as Catalysts for Stereoselective Aziridination of Styrenes with N‐Tosyloxycarbamates.
Authors: Lebel Helene , Parmentier Michael , Leogane Olivier , Ross Karen , Spitz Cedric 
Published: September 2012

AbstractThe aziridination of styrenes (I) carrying electron.withdrawing groups with chiral N‐tosyloxycarbamate (II) gives the aziridines (III) with good to excellent diastereoselectivity.
ChemInform Abstract: Zinc or Indium‐Mediated Barbier‐Type Allylation of Aldehydes with 3‐Bromomethyl‐5H‐furan‐2‐one in Aqueous Media: An Efficient Synthesis Method for α‐Methylene‐γ‐butyrolactone.
Authors: Gao Yu‐Zhe , Wang Xue , Sun Li‐Dong , Xie Long‐Guan , Xu Xiao‐Hua 
Published: September 2012

AbstractMild and convenient methods for the diastereoselective synthesis of the compounds (III) and (V) are developed.
ChemInform Abstract: Intramolecular Etherification of Five‐Membered Cyclic Carbonates Bearing Hydroxyalkyl Groups.
Authors: Tomczyk Karolina M. , Gunka Piotr A. , Parzuchowski Pawel G. , Zachara Janusz , Rokicki Gabriel 
Published: September 2012

AbstractDiols with vicinal hydroxyl groups easily form five‐membered cyclic carbonates (III) in high yields with dimethyl carbonate (II) in the presence of a alkaline catalyst.
ChemInform Abstract: Simple, Convenient Method for the Synthesis of Substituted Furan‐2(5H)‐one Derivatives Using Tin(II) Chloride.
Authors: Nagarapu Lingaiah , Kumar U. Nikhil , Upendra P. , Bantu Rajashaker 
Published: September 2012

AbstractA simple and efficient tin‐catalyzed three‐component reaction of DMAD (I) with aromatic aldehydes and amines is presented.
ChemInform Abstract: A Highly Efficient One‐Pot Reaction of 2‐(gem‐Dibromovinyl)phenols(thiophenols) with K4Fe(CN)6 to 2‐Cyanobenzofurans(thiophenes).
Authors: Zhou Wei , Chen Wei , Wang Lei 
Published: September 2012

AbstractThe novel title reaction is reported under mild and low‐toxic reactions conditions.
ChemInform Abstract: Gold(I)‐Catalyzed Cyclization of 2‐(1‐Alkynyl)‐alk‐2‐en‐1‐one Oximes: A Facile Access to Highly Substituted N‐Alkoxypyrroles.
Authors: Zhang Mei , Zhang Junliang 
Published: September 2012

AbstractAn efficient, mild, and atom‐economic route to substituted N‐alkoxypyrroles uses various nucleophiles in the title reaction.
ChemInform Abstract: An Insight into Solvent‐Free Diimide Porphyrin Reduction: A Versatile Approach for meso‐Aryl Hydroporphyrin Synthesis.
Authors: Pereira Mariette M. , Abreu Artur R. , Goncalves Nuno P. F. , Calvete Mario J. F. , Simoes Ana V. C. , Monteiro Carlos J. P. , Arnaut Luis G. , Eusebio Maria Ermelinda , Canotilho Joao 
Published: September 2012

AbstractThe preparation of meso‐aryl hydroporphyrins, namely chlorins (II) and bacteriochlorins (IV), proceeds via reduction of porphyrins (I) and (III) with diimide in the absence of solvents and bases.
ChemInform Abstract: PEG‐SO3H as a Catalyst for the Preparation of Bisindolyl and Trisindolyl Methanes in Aqueous Media.
Authors: Rani V. Jhansi , Vani K. Veena , Rao C. Venkata 
Published: September 2012

AbstractAdvantages of the presented method are operational simplicity and remarkably short reaction times.
ChemInform Abstract: Synthesis and Photoluminescent Properties of New Cationic Carbazole‐Containing Luminophores.
Authors: Baran A. , Plotniece A. , Sobolev A. , Vigante B. , Gosteva M. , Olkhovik V. 
Published: September 2012

Abstract8 Title compounds of type (I) or (II) are prepared and their photoluminescent properties are measured.
ChemInform Abstract: Electron‐Poor N‐Substituted Imide‐Fused Corannulenes.
Authors: Schmidt Bernd M. , Topolinski Berit , Roesch Philipp , Lentz Dieter 
Published: September 2012

AbstractNovel corannulenes (V) are obtained by Wohl—Ziegler bromination of tetramethylfluoranthenes (IV) followed by a nickel‐mediated intramolecular coupling reaction.
ChemInform Abstract: Tandem Knoevenagel—Michael Reaction of 1‐Phenyl‐3‐methyl‐5‐pyrazolone with Aldehydes Using 3‐Aminopropylated Silica Gel as an Efficient and Reusable Heterogeneous Catalyst.
Authors: Sobhani Sara , Hasaninejad Ali‐Reza , Maleki Mahdi Faal , Parizi Zahra Pakdin 
Published: September 2012

AbstractAminopropylated silica gel is shown to be an efficient heterogeneous catalyst for the tandem Knoevenagel—Michael reaction of pyrazolone (I) with various aldehydes.
ChemInform Abstract: Efficient Catalytic Cyclizations of Three and Two Imine Assemblies: Direct Access to Tetrahydroimidazo[1,5‐c]imidazol‐7‐ones and Imidazoles.
Authors: Saima Yasmin , Khamarui Saikat , Gayen Krishnanka S. , Pandit Palash , Maiti Dilip K. 
Published: September 2012

AbstractTreatment of in situ prepared aldimines with proline leads diastereoselectively to tetrahydroimidazo[1,5‐c]imidazol‐7‐ones (III).
ChemInform Abstract: Synthesis and Synthetic Applications of 1‐Aryl‐2‐alkyl‐4,5‐dihydro‐1H‐imidazoles.
Authors: Reverdito Ana M. , Perillo Isabel A. , Salerno Alejandra 
Published: September 2012

AbstractThe microwave‐assisted cyclocondensation of N‐aryl‐N′‐acyldiamines (I) gives easy access to title dihydroimidazoles (II).
ChemInform Abstract: Functionalized Orthoesters as Powerful Building Blocks for the Efficient Preparation of Heteroaromatic Bicycles.
Authors: Bastug Gulluzar , Eviolitte Christophe , Marko Istvan E. 
Published: September 2012

AbstractTreatment of 2‐aminothiophenols, 2‐aminophenols, and benzene‐1,2‐diamines with functionalized orthoesters allows an efficient access to the title scaffolds.
ChemInform Abstract: Palladium‐Catalyzed Selective C—H Benzylation Towards Functionalized Azoles with a Quaternary Carbon Center.
Authors: Xie Pan , Huang Hanmin , Xie Yinjun , Guo Shengmei , Xia Chungu 
Published: September 2012

AbstractThe method efficiently generates a wide range of tribenzylated azoles (III) with a quaternary carbon center.
ChemInform Abstract: Isoxazolo(aza)naphthoquinones: A New Class of Cytotoxic Hsp90 Inhibitors.
Authors: Dallavalle Sabrina , et al. et al. 
Published: September 2012

AbstractCycloaddition of in situ prepared benzonitriloxides to quinones is exploited for the synthesis of substituted isoxazolo‐fused naphthoquinones.
ChemInform Abstract: Discovery, Design and Synthesis of Y‐Shaped Peroxisome Proliferator‐Activated Receptor δ Agonists as Potent anti‐Obesity Agents in vivo.
Authors: Chin Jungwook , et al. et al. 
Published: September 2012

AbstractNovel Y‐shaped PPARδ ligands are synthesized by combination of a known ligand and a marine natural product using automatic docking experiments.
ChemInform Abstract: Easy Access to 2‐Alkyl and 2‐Arylthiazolines Using a Modified Heteropolyacid Catalysis: Application to the Synthesis of Bacillamide A.
Authors: Fache F. , Cros F. , Piva O. , Lefebvre F. 
Published: September 2012

AbstractA straightforward access to 2‐alkyl and 2‐arylthiazoles (III) by condensation of β‐aminothiols and nitriles, catalyzed by tungstophosphoric acid under microwave irradiation, is described.
ChemInform Abstract: Iron‐Catalyzed Arylation of Benzoazoles with Aromatic Aldehydes Using Oxygen as Oxidant.
Authors: Liu Saiwen , Chen Ru , Guo Xiangyu , Yang Huiqiong , Deng Guojun , Li Chao‐Jun 
Published: September 2012

AbstractOne aliphatic aldehyde, e.g. (IIb), is also included which gives the corresponding product (IIIb) in moderate yield.
ChemInform Abstract: Reactions of 4‐Phenyl‐1,2,4‐triazoline‐3,5‐dione with 2‐Pyrazolines.
Authors: Novikov R. A. , Korolev V. A. , Tomilov Yu. V. 
Published: September 2012

AbstractThe mechanisms behind the reactions of 4‐phenyl‐1,2,4‐triazoline‐3,5‐dione (PTAD) with both 1‐unsubstituted and 1‐substituted 2‐pyrazolines are discussed.
ChemInform Abstract: Synthesis of 3‐Nitramino‐4‐(1H‐1,2,3‐triazol‐1‐yl)‐1,2,5‐oxadiazoles and Their Salts.
Authors: Rozhkov V. Yu. , Batog L. V. , Struchkova M. I. 
Published: September 2012

AbstractTriazolylfurazans bearing a primary nitramino group attached to the furazan ring, e.g. (II), are prepared for the first time.
ChemInform Abstract: ZnO as an Effective and Reusable Heterogeneous Catalyst for the Synthesis of Arylaminotetrazoles.
Authors: Habibi Davood , Nasrollahzadeh Mahmoud 
Published: September 2012

AbstractThe formation of either 1‐aryl‐5‐amino‐1H‐tetrazoles (II) or 5‐arylamino‐1H‐tetrazoles (IV) from the ZnO‐catalyzed reaction of arylcyanamides and sodium azide is strongly influenced by the electronic nature of aryl substituents.
ChemInform Abstract: A Novel Organocatalytic Multi‐Component Reaction: An Efficient Synthesis of Polysubstituted Pyrano‐Fused Spirooxindoles.
Authors: Tisseh Zeinab Noroozi , Ahmadi Fereshteh , Dabiri Minoo , Khavasi Hamid Reza , Bazgir Ayoob 
Published: September 2012

AbstractA simple protocol is presented for the three‐component reaction of isatins, malononitrile and acetylene derivatives to give the title compounds (IV).
ChemInform Abstract: Diastereoselective 1,3‐Dipolar Cycloaddition of Pyrylium Ylides with Chiral Enamides.
Authors: Tchabanenko Kirill , Sloan Colleen , Bunetel Yves‐Mael , Mullen Philip 
Published: September 2012

AbstractThe first example of the use of amides as alkene in the title reaction is demonstrated.
ChemInform Abstract: A Tandem Olefin Migration and Prins Cyclization Using Cu(OTf)2—Bisphosphine Complexes: An Improved Synthesis of Functionalized Tetrahydropyrans.
Authors: Ghosh Arun K. , Nicponski Daniel R. , Kass Jorden 
Published: September 2012

AbstractThe scope of the Cu(OTf)2—bisphoshine catalyzed tandem olefin migration and Prins cyclization of the hexenol (I) with aldehydes is investigated using a quite stable bisphoshine ligand with low air‐sensitivity.
ChemInform Abstract: Me3SiI‐Promoted Reaction of Salicylic Aldehydes with Ketones: A Facile Way to Construct Benzopyranic [2,3‐b]Ketals and Spiroketals.
Authors: Wang Feijun , Qu Mingliang , Lu Xi , Chen Feng , Chen Feng , Shi Min 
Published: September 2012

AbstractA highly versatile one‐pot methodology for the synthesis of heteroannular ketals and spiroketals is described.
ChemInform Abstract: Borderline Metal‐Catalyzed Carboarylation of Alkynylarenes Using N,O‐Acetals.
Authors: Komeyama Kimihiro , Yamada Takahiro , Igawa Ryoichi , Takaki Ken 
Published: September 2012

AbstractThe carboarylation of alkynylarenes with N‐acyliminium ions, generated from N,O‐acetals, is catalyzed by Bi(O‐Tf)3 or Fe(O‐Tf)3.
ChemInform Abstract: Facile Syntheses of 2‐Substituted 3‐Cyanochromones.
Authors: Levchenko K. S. , Semenova I. S. , Yarovenko V. N. , Shmelin P. S. , Krayushkin M. M. 
Published: September 2012

AbstractBased on the condensation of carboxylic acid chlorides or anhydrides with 3‐(2‐hydroxyphenyl)‐3‐oxopropionitrile (I), a general synthesis of the title compounds (III) is described.
ChemInform Abstract: Effective Synthesis of tert‐Butyl‐Substituted 3‐Carboxy Coumarins in Water Using TEBAC as Catalyst.
Authors: Li Yang , Gao Wentao 
Published: September 2012

AbstractHitherto unreported hydrophobically substituted 3‐carboxycoumarin derivatives (III) are synthesized by modifying a known method through use of benzyltriethylammonium chloride as catalyst.
ChemInform Abstract: Efficient Synthesis of 12‐Aryl‐8,9,10,12‐tetrahydrobenzo[a]xanthen‐11‐one Derivatives Catalyzed by p‐Dodecylbenzenesulfonic Acid in Aqueous Media under Ultrasound Irradiation.
Authors: Li Ji‐Tai , Li Yan‐Wei , Song Ya‐Li 
Published: September 2012

AbstractDodecylbenzenesulfonic acid acts as both Broensted acid and phase‐transfer catalyst.
ChemInform Abstract: Synthesis of 3‐Aroyl‐4‐hydroxy‐4‐arylpiperidine Derivatives by DBU‐Catalyzed Reactions of Amines with Vinyl Ketones.
Authors: Liu Xiaodong , chen Qiao , Li Wenyi , Wang Rui 
Published: September 2012

AbstractA highly efficient cascade reaction of primary amines, generally sulfonamides, with aryl vinyl ketones results in the diastereoselective formation of functionalized piperidines, key structures of natural products and drugs.
ChemInform Abstract: Solvent‐ and Catalyst‐Free Synthesis of New Hydroxylated Trisubstituted Pyridines under Microwave Irradiation.
Authors: Yin Guodong , Liu Qiong , Ma Junrui , She Nengfang 
Published: September 2012

AbstractThe expected products are obtained through a simplified purification procedure without protection of the hydroxyl group.
ChemInform Abstract: K2CO3‐Mediated, One‐Pot, Multicomponent Synthesis of Medicinally Potent Pyridine and Chromeno[2,3‐b]pyridine Scaffolds.
Authors: Mishra Sarita , Ghosh Rina 
Published: September 2012

AbstractAn efficient potassium carbonate‐catalyzed three‐component reaction of malononitrile (I) with a wide variety of aldehydes (II), (V), (VII) and thiols (III), (VIII) is presented to afford dihydropyrimidine intermediates which are aromatized with potassium permanganate.
ChemInform Abstract: Asymmetric Synthesis of 2‐Alkyl‐substituted Tetrahydroquinolines by an Enantioselective Aza‐Michael Reaction.
Authors: Taylor Laura L. , Goldberg Frederick W. , Hii King Kuok 
Published: September 2012

AbstractAn enantioselective Pd‐catalyzed aza‐Michael reaction is used as the key step in the preparation of Galipea alkaloids angustureine, galipeine and cuspareine (V).
ChemInform Abstract: Efficient Synthesis of Substituted Quinolines Through Intramolecular Addition of Aryl Anion to Carbonyl Carbon.
Authors: Kobayashi Yuichi , Igarashi Junji , Feng Chao , Tojo Toshifumi 
Published: September 2012

AbstractThe convenient three‐step synthesis of quinolines is based on intramolecular cyclization of N‐Michael addition products (III) followed by an acetyl chloride mediated dehydration‐deprotection‐dehydrogenation sequence.
ChemInform Abstract: Synthesis and Biological Studies of Some New Acrylic Acid Ethyl Esters of Quinolinone.
Authors: Kalkhambkar Rajesh G. , Aridoss G. , Kulkarni Geeta M. , Bapset R. M. , Kadakol J. C. , Premkumar N. , Jeong Yeon Tae 
Published: September 2012

AbstractMost of the compounds with chloro‐substitution at the C‐6 or C‐7 position show potent antibacterial and antifungal as well as analgesic and antiinflammatory activities.
ChemInform Abstract: Gold(I)‐Catalyzed Cycloisomerization of Nitrogen‐ and Oxygen‐Tethered Alkylidenecyclopropanes to Tricyclic Compounds.
Authors: Zhang Di‐Han , Wei Yin , Shi Min 
Published: September 2012

AbstractThe new, very mild, air‐ and moisture‐tolerant title reaction is presented.
ChemInform Abstract: A Solvent‐Free, Four‐Component Synthesis and 1,3‐Dipolar Cycloaddition of 4(H)‐Pyrans with Nitrile Oxides: Synthesis and Discovery of Antimycobacterial Activity of Enantiomerically Pure 1,2,4‐Oxadiazoles.
Authors: Almansour Abdulrahman I. , Kumar Raju Suresh , Arumugam Natarajan , Sriram Dharmarajan 
Published: September 2012

AbstractFour‐component reaction between tetrahydropyridinone derivative (I), an aromatic aldehyde (II) and malononitrile (III) under solvent‐free conditions affords an inseparable mixture of two diastereomeric pyrans (IV) in near quantitative yield.
ChemInform Abstract: Synthesis of a Novel Series of 1,6‐Disubstituted‐3‐(cyclohexylmethoxy)‐β‐carboline Derivatives via Minisci Reaction.
Authors: Lin Guowu , Wang Yue , Zhou Qingfa , Wang Jian , Yang Taotao , Wang Zhanwei , Lu Tao 
Published: September 2012

AbstractA simple and efficient synthetic route fallows the formation of title compounds (VII) (22 examples) via Minisci reaction as the key step [→ (VI)].
ChemInform Abstract: Acetic Anhydride Mediated Condensation of Aromatic o‐Diacid Dichlorides with Benzimidazoles to Provide Electroreducible p‐Dione Adducts.
Authors: Joyce Eamonn , Kavanagh Paul , Leech Donal , Karpinska Jolanta , McArdle Patrick , Aldabbagh Fawaz 
Published: September 2012

AbstractIt is demonstrated that acetic anhydride allows a very rapid condensation of o‐diacid dichlorides with imidazole and benzimidazoles.
ChemInform Abstract: NH2SO3H and H6P2W18O62·18H2 O‐Catalyzed, Three‐Component, One‐Pot Synthesis of Benzo[c]acridine Derivatives.
Authors: Heravi Majid M. , Alinejhad Hamideh , Derikvand Fatemeh , Oskooie Hossein A. , Baghernejad Bita , Bamoharram Fatemeh F. 
Published: September 2012

AbstractAn efficient and practical three‐component, one‐pot preparation of polyhydroacridine derivatives proceeds under neat conditions in the presence of sulfamic acid or Wells—Dawson acid as catalyst.
ChemInform Abstract: Quinazolino—Benzothiazoles: Fused Pharmacophores as Anticonvulsant Agents.
Authors: Ugale Vinod G. , Patel Harun M. , Wadodkar Sudhir G. , Bari Sanjay B. , Shirkhedkar Atul A. , Surana Sanjay J. 
Published: September 2012

AbstractA benzothiazole moiety is incorporated in the quinazoline nucleus by recyclization of benzoxazinone (I) with substituted aminobenzothiazoles (II).
ChemInform Abstract: Acid Catalysis in the Oxidative Nucleophilic Alkoxylation of 1,3,7‐Triazapyrenes.
Authors: Borovlev I. V. , Demidov O. P. , Saigakova N. A. 
Published: September 2012

AbstractThe method leads to dialkoxylated products irrespective of the substrate ratio.
ChemInform Abstract: A Novel Intramolecular Ugi 3CC for the Synthesis of N‐Alkyl‐3‐oxo‐2‐aryl‐1,2,3,4‐tetrahydropyrazino [1,2‐a]indole‐1‐carboxamides.
Authors: Reddy B. V. Subba , Dey Sujit Kumar , Yadav J. S. , Sridhar B. 
Published: September 2012

AbstractA novel intramolecular Ugi three‐component reaction of substrate (I) with amines and isonitriles is reported to provide the title compounds (IV).
ChemInform Abstract: Synthesis, Antitumor Activity and SAR Study of Novel [1,2,4]Triazino[4,5‐a]benzimidazole Derivatives.
Authors: El‐Nassan Hala Bakr 
Published: September 2012

AbstractTitle derivatives (III) are obtained upon cyclocondensation of benzimidazole derivative (I) with aryl and heteroaryl aldehydes (II).
ChemInform Abstract: Mannich‐Type Reaction for Synthesis of 3‐Methyl‐4‐nitroimino‐tetrahydro‐1,3,5‐oxadiazine.
Authors: Qu Wen‐Yan , She Dong‐Mei , Zhao Jian , Lin De‐Jie , Huang Qi‐Liang , Li Feng‐Min 
Published: September 2012

AbstractMannich reaction of N‐methyl‐N′‐nitroguanidine (I) in the presence of alkaline catalysts provides access to the title oxadiazine (III) and triazine derivative (IV).
ChemInform Abstract: Synthesis of a 1,3,5‐Benzotriazepine‐2,4‐dione Based Library.
Authors: Chuckowree Irina , Syed Murtaza Ali , Getti Giulia , Patel Asha Parbhu , Garner Hannah , Tizzard Graham J. , Coles Simon J. , Spencer John 
Published: September 2012

AbstractIn order to develop selective pyrathyroid hormone‐1‐receptor antagonists the cyclocondensation of functionalized o‐phenylenediamines (I) with phenyl isocyanatoformate is described to synthesize 1,3,5‐benzotriazepinediones.
ChemInform Abstract: A Concise Route to Indoloazocines via a Sequential Ugi—Gold‐Catalyzed Intramolecular Hydroarylation.
Authors: Modha Sachin G. , Vachhani Dipak D. , Jacobs Jeroen , Van Meervelt Luc , Van der Eycken Erik V. 
Published: September 2012

AbstractThe sequence affords the desired indoloazocines (VI).
ChemInform Abstract: A New Polycyclic System Containing the 1,4‐Benzodiazepine and Isoindolinone Fragments: Synthesis and Structure.
Authors: Ukhin L. Yu. , Suponitskii K. Yu. , Shepelenko E. N. , Belousova L. V. , Orlova Zh. I. , Borodkin G. S. 
Published: September 2012

AbstractThe formation of fused benzodiazepines (III) proceeds smoothly without any acid catalyst.
ChemInform Abstract: Synthesis of Functionalized Diarylborinic 8‐Oxyquinolates via Bimetallic Boron—Lithium Intermediates.
Authors: Wesela‐Bauman Grzegorz , Jastrzebski Lech , Kurach Pawel , Lulinski Sergiusz , Serwatowski Janusz , Wozniak Krzysztof 
Published: September 2012

AbstractFor the synthesis of the novel title compounds a simple one‐pot protocol, which uses readily available starting materials, is presented.
ChemInform Abstract: Alkylboronic Esters from Palladium‐ and Nickel‐Catalyzed Borylation of Primary and Secondary Alkyl Bromides.
Authors: Yi Jun , Liu Jin‐Hui , Liang Jun , Dai Jian‐Jun , Yang Chu‐Ting , Fu Yao , Liu Lei 
Published: September 2012

AbstractCross‐coupling reactions of primary alkyl bromides (I) with diboron reagent (II) give the desired organo‐boron compounds (III) in the presence of a palladium catalyst.
ChemInform Abstract: Synthesis of Functionalized 2,3,4,5‐Tetraphenylsilole Derivatives Through Hydrosilylation and Their Crystal Structures.
Authors: Zhang Yunsheng , Li Shuhong , Wang Rui , Chen Limin , Xu Caihong 
Published: September 2012

AbstractTitle compounds (III), prepared by hydrosilylation of p‐ethynylarenes (II), show aggregation‐induced emission effects.
ChemInform Abstract: Dialkyl (1‐Ethoxycarbonyl‐2,2,2‐trifluoro‐1‐phenylsulfonylaminoethyl) phosphonates.
Authors: Aksinenko A. Yu. , Sokolov V. B. , Goreva T. V. , Makhaeva G. F. 
Published: September 2012

AbstractNovel fluorinated α‐amino phosphonates (III) are synthesized.
ChemInform Abstract: Mild and Efficient Esterification of Alkylphosphonic Acids Using Polymer‐Bound Triphenylphosphine.
Authors: Purohit Ajay Kumar , Pardasani Deepak , Tak Vijay , Kumar Ajeet , Jain Rajeev , Dubey Devendra Kumar 
Published: September 2012

AbstractA convenient procedure is developed for the synthesis of dialkyl phosphonates from alkylphosphonic acids and primary alcohols under mild conditions.