bluuebunny/crossref_metadata_2025_split huggingface dataset:
Small Molecule Restores Itaconate Sensitivity in Salmonella enterica: A Potential New Approach to Treating Bacterial Infections
Authors: Hammerer Fabien , Chang Justin H. , Duncan Dustin , Castañeda Ruiz Angel , Auclair Karine 
Published: June 2016

AbstractIn the context of increasing global antibiotic resistance, the need for alternative therapeutic targets is great. Although new antibiotics and resistance inhibitors provide temporary solutions, they are bound to become obsolete. In this work, we propose a new approach, coined “bacterio‐modulation” that aims to restore macrophage potency towards bacterial strains that are able to survive in phagolysosomes. One key defense in the macrophage's arsenal is itaconate, an endogenous molecule with antimicrobial activity. Some intracellular pathogens have evolved to produce itaconate‐degrading enzymes, which are required for intracellular proliferation and to promote pathogenicity. We herein present the first molecule able to resensitize Salmonella enterica to itaconate.
Highly Sensitive Measurement of Inositol 1,4,5‐Trisphosphate by Using a New Fluorescent Ligand and Ligand Binding Domain Combination
Authors: Oura Tai , Murata Kaori , Morita Takao , Nezu Akihiro , Arisawa Mitsuhiro , Shuto Satoshi , Tanimura Akihiko 
Published: June 2016

AbstractBased on the results of our previous adenophostin A structure–activity relationship studies, two fluorescent inositol 1,4,5‐trisphosphate (IP3) receptor ligands, fluorescent adenophostin A (FADA) and fluorescent low‐affinity ligand (FLL), were designed. Binding of the fluorescent ligands to the fluorescent IP3 sensor in protein‐expressing cells caused FRET. This principle was extended to a cell‐free assay system by using the fluorescent IP3 sensor bound to agarose beads. The effect of FLL on the FRET signal was reduced by subsequent addition of IP3. The IC50 values of IP3 on the FRET signals were 139.7 and 352.1 nm for 30 and 100 nm FLL, respectively. This method allowed quantitative measurement of IP3 concentrations below 10 nm and was applied to measure cytosolic IP3 concentrations in COS‐7 cells and to examine the potency of synthesized adenophostin A analogues.
Ac‐LPFFD‐Th: A Trehalose‐Conjugated Peptidomimetic as a Strong Suppressor of Amyloid‐β Oligomer Formation and Cytotoxicity
Authors: Sinopoli Alessandro , Giuffrida Alessandro , Tomasello Marianna Flora , Giuffrida Maria Laura , Leone Marilisa , Attanasio Francesco , Caraci Filippo , De Bona Paolo , Naletova Irina , Saviano Michele , Copani Agata , Pappalardo Giuseppe , Rizzarelli Enrico 
Published: June 2016

AbstractThe inhibition of amyloid formation is a promising therapeutic approach for the treatment of neurodegenerative diseases. Peptide‐based inhibitors, which have been widely investigated, are generally derived from original amyloid sequences. Most interestingly, trehalose, a nonreducing disaccharide of α‐glucose, is effective in preventing the aggregation of numerous proteins. We have determined that the development of hybrid compounds could provide new molecules with improved properties that might synergically increase the potency of their single moieties. In this work, the ability of Ac‐LPFFD‐Th, a C‐terminally trehalose‐conjugated derivative, to slow down the Aβ aggregation process was investigated by means of different biophysical techniques, including thioflavin T fluorescence, dynamic light scattering, ESI‐MS, and NMR spectroscopy. Moreover, we demonstrate that Ac‐LPFFD‐Th modifies the aggregation features of Aβ and protects neurons from Aβ oligomers' toxic insult.
Site‐Selective Aliphatic C−H Silylation of 2‐Alkyloxazolines Catalyzed by Ruthenium Complexes
Authors: Kon Kazumasa , Suzuki Hiroyuki , Takada Kosuke , Kohari Yoshihito , Namikoshi Takeshi , Watanabe Shinji , Murata Miki 
Published: June 2016

AbstractThe Ru‐catalyzed dehydrogenative silylation of 2‐alkyloxazolines with 1,1,1,3,5,5,5‐heptamethyltrisiloxane took place site‐selectively at methyl C(sp3)−H bonds located γ to the nitrogen atom of the oxazolyl groups. Pyridine and pyrazole rings could also be used as a directing group. A catalytic mechanism based upon successive σ‐bond metathesis is proposed.
LiTi2(PO4)3/C Anode Material with a Spindle‐Like Morphology for Batteries with High Rate Capability and Improved Cycle Life
Authors: Yu Shicheng , Tempel Hermann , Schierholz Roland , Aslanbas Özgür , Gao Xin , Mertens Josef , de Haart Lambertus G. J. , Kungl Hans , Eichel Rüdiger‐A. 
Published: June 2016

AbstractNanocrystalline LiTi2(PO4)3/C has been synthesized by employing a solvothermal process in which oxalic acid was used as a solubilizer for the titanium source, a surfactant, and a carbon source. Additionally, Pechini's sol–gel‐based method was also used as the synthesis method for comparison. LiTi2(PO4)3/C prepared by using a solvothermal route showed a homogenous particle size with spindle‐like microstructures formed from self‐assembled nanosized‐platelets, whereas preparation by the sol–gel process resulted in agglomerated powders with irregular morphology and particle size. The different morphologies of LiTi2(PO4)3/C prepared in the two synthesis methods tend to form different electrode layer structures, which results in remarkable differences in their electrochemical properties. In particular, the solvothermally synthesized LiTi2(PO4)3/C composite exhibits superior high‐rate‐discharge capability and cycling stability. A capacity of approximately 97.7 % of the initial capacity was maintained for the solvothermal sample after 500 cycles at 5 C.
Solar Thermal Energy Storage in a Photochromic Macrocycle
Authors: Vlasceanu Alexandru , Broman Søren L. , Hansen Anne S. , Skov Anders B. , Cacciarini Martina , Kadziola Anders , Kjaergaard Henrik G. , Mikkelsen Kurt V. , Nielsen Mogens Brøndsted 
Published: June 2016

AbstractThe conversion and efficient storage of solar energy is recognized to hold significant potential with regard to future energy solutions. Molecular solar thermal batteries based on photochromic systems exemplify one possible technology able to harness and apply this potential. Herein is described the synthesis of a macrocycle based on a dimer of the dihydroazulene/vinylheptafulvene (DHA/VHF) photo/thermal couple. By taking advantage of conformational strain, this DHA–DHA macrocycle presents an improved ability to absorb and store incident light energy in chemical bonds (VHF–VHF). A stepwise energy release over two sequential ring‐closing reactions (VHF→DHA) combines the advantages of an initially fast discharge, hypothetically addressing immediate energy consumption needs, followed by a slow process for consistent, long‐term use. This exemplifies another step forward in the molecular engineering and design of functional organic materials towards solar thermal energy storage and release.
ChemInform Abstract: Crystal Structure Redetermination of ε‐Ni3Si2 from a Single Nanowire by Dynamical Refinement of Precession Electron Diffraction Data.
Authors: Correa Cinthia Antunes , Klementova Mariana , Drinek Vladislav , Kopecek Jaromir , Palatinus Lukas 
Published: June 2016

AbstractPrecession electron diffraction tomography (PEDT) is used to re‐determine the crystal structure of ε‐Ni3Si2 from a nanowire with a diameter of 35 nm.
ChemInform Abstract: Enhanced Thermoelectric Properties of Earth‐Abundant Cu2SnS3 via in Doping Effect.
Authors: Tan Qing , Sun Wei , Li Zhiliang , Li Jing‐Feng 
Published: June 2016

AbstractBulk samples of Cu2Sn1‐xInxS3 (x = 0—0.2) are prepared by mechanical alloying (450 rpm, 24 h) followed by spark plasma sintering in vacuum (873 K, 5 min).
ChemInform Abstract: Ce11Ge3.73(2)In6.27: Solid‐State Synthesis, Crystal Structure and Site‐Preference.
Authors: Jeon Beom‐Yong , Nam Gnu , Lee Dong Woo , Ok Kang Min , You Tae‐Soo 
Published: June 2016

AbstractBar‐shaped single‐crystals of Ce11Ge3.73In6.27 are prepared by solid state reaction of a 11:3:7 molar mixture of Ce, Ge, and In (sealed Nb ampoule in silica jacket, 950 °C, 2 d).
ChemInform Abstract: Symbiotic Transition‐Metal and Organocatalysis for Catalytic Ambient Amine Oxidation and Alkene Reduction Reactions.
Authors: Murray Alexander T. , King Rose , Donnelly Joseph V. G. , Dowley Myles J. H. , Tuna Floriana , Sells Daniel , John Matthew P. , Carbery David R. 
Published: June 2016

AbstractA catalytic system of CuCl and alloxane is applied for the aerobic oxidative dimerization of benzylic amines (III) and cross‐coupling of amines (III) with anilines (V).
ChemInform Abstract: Iridium‐Catalyzed C—C Coupling of a Simple Propargyl Ether with Primary Alcohols: Enantioselective Homoaldol Addition via Redox‐Triggered (Z)‐Siloxyallylation.
Authors: Liang Tao , Zhang Wandi , Krische Michael J. 
Published: June 2016

AbstractIr‐catalyzed enantioselective C—C coupling of silylated propargyl ether (I) with alcohols (II) gives rise to γ‐hydroxy (Z)‐enol silanes (III), which can be readily converted into γ‐lactones (IV) and trisubstituted furans (V).
ChemInform Abstract: Palladium‐Catalyzed Enantioselective Domino Heck/Intermolecular C—H Bond Functionalization: Development and Application to the Synthesis of (+)‐Esermethole.
Authors: Kong Wangqing , Wang Qian , Zhu Jieping 
Published: June 2016

AbstractA series of oxindoles (III) is obtained by a Pd‐catalyzed reaction of triflates (I) with oxadiazoles (II).
ChemInform Abstract: Enantioselective Synthesis of 3,5,6‐Substituted Dihydropyranones and Dihydropyridinones Using Isothiourea‐Mediated Catalysis.
Authors: Stark Daniel G. , Morrill Louis C. , Cordes David B. , Slawin Alexandra M. Z. , O'Riordan Timothy J. C. , Smith Andrew D. 
Published: June 2016

AbstractThe title compounds are synthesized from N‐tosyliminoacrylates and aroylacrylates by a Michael addition‐lactamization/lactonization cascade reaction.
ChemInform Abstract: Chain Walking as a Strategy for Carbon—Carbon Bond Formation at Unreactive Sites in Organic Synthesis: Catalytic Cycloisomerization of Various 1,n‐Dienes
Authors: Hamasaki Taro , Aoyama Yuka , Kawasaki Junichi , Kakiuchi Fumitoshi , Kochi Takuya 
Published: June 2016

Abstract20 examples
ChemInform Abstract: Nucleophilic Substitution of the Hydroxyl Group in Stereogenic Alcohols with Chirality Transfer.
Authors: Bunrit Anon , Dahlstrand Christian , Srifa Pemikar , Olsson Sandra K. , Huang Genping , Biswas Srijit , Himo Fahmi , Samec Joseph S. M. 
Published: June 2016

AbstractAn intramolecular substitution of the OH group in enantioenriched alcohols is achieved by acid/base bifunctional catalysis.
ChemInform Abstract: An Eco‐Friendly, Hantzsch‐Based, Solvent‐Free Approach to 2‐Aminothiazoles and 2‐Aminoselenazoles.
Authors: Facchinetti Victor , Avellar Marcela M. , Nery Ana C. S. , Gomes Claudia R. B. , Vasconcelos Thatyana R. A. , de Souza Marcus V. N. 
Published: June 2016

AbstractA very fast method for the synthesis of the title thiazoles and selenazoles through Hantzsch cyclization starting from thiourea and selenurea, resp., is developed.
ChemInform Abstract: Divergent Reactivity via Cobalt Catalysis: An Epoxide Olefination.
Authors: Jamieson Megan L. , Hume Paul A. , Furkert Daniel P. , Brimble Margaret A. 
Published: June 2016

AbstractCobalt‐catalyzed reaction of epoxides with dimethylsulfoxonium methylide provides a two‐carbon epoxide homologation/ring‐opening tandem process.
ChemInform Abstract: Towards a General Ruthenium‐Catalyzed Hydrogenation of Secondary and Tertiary Amides to Amines.
Authors: Cabrero‐Antonino Jose R. , Alberico Elisabetta , Junge Kathrin , Junge Henrik , Beller Matthias 
Published: June 2016

AbstractA broad range of secondary and tertiary amides is hydrogenated to the corresponding amines under mild conditions using an in situ catalyst generated by combining [Ru(acac)3], 1,1,1‐tris(diphenylphosphinomethyl)ethane (Triphos) and Yb(OTf)3.
ChemInform Abstract: Silver(I)‐Catalyzed Iodination of Arenes: Tuning the Lewis Acidity of N‐Iodosuccinimide Activation.
Authors: Racys Daugirdas T. , Sharif Salaheddin A. I. , Pimlott Sally L. , Sutherland Andrew 
Published: June 2016

AbstractA general method for the iodination of a wide range of arenes is developed.
ChemInform Abstract: Synthesis of Novel Imidazo[1,2‐a]pyridine‐4‐hydroxy‐2H‐coumarins by Groebke—Blackburn—Bienayme Multicomponent Reaction as Potential NS5B Inhibitors.
Authors: Manvar Parth , Shaikh Faraz , Kakadiya Rajesh , Mehariya Krunal , Khunt Ranjan , Pandey Bipin , Shah Anamik 
Published: June 2016

AbstractA Groebke—Blackburn—Bienayme three component reaction of 4‐hydroxy‐3‐formylcoumarin, alkyl isocyanides, and 2‐aminoazines is demonstrated to give various imidazo[1,2‐a] fused heterocycles containing the coumarin scaffold.
ChemInform Abstract: Diastereoselective Synthesis of Tetrasubstituted Propargylamines via Hydroamination and Metalation of 1‐Alkynes and Their Enantioselective Conversion to Trisubstituted Chiral Allenes.
Authors: Periasamy Mariappan , Reddy Polimera Obula , Satyanarayana Iddum , Mohan Lakavathu , Edukondalu Athukuri 
Published: June 2016

AbstractThe reactions involve the diastereoselective addition of in situ formed alkynylcopper complexes to in situ formed iminium ions regioselectively affording the corresponding propargylamines.
ChemInform Abstract: Oxydifluoromethylation of Alkenes by Photoredox Catalysis: Simple Synthesis of CF2H‐Containing Alcohols.
Authors: Arai Yusuke , Tomita Ren , Ando Gaku , Koike Takashi , Akita Munetaka 
Published: June 2016

AbstractThe title reaction allows a single‐step and regioselective formation of C(sp3)—CF2H and C(sp3)—O bonds from C=C double bonds in terminal and internal alkenes, e.g. (I), (IV), (VI), and (VIII).
ChemInform Abstract: A General Method for the Synthesis of Enantiopure 1,5‐Amino Alcohols.
Authors: Guignard Guillaume , Llor Nuria , Urbina Aina , Bosch Joan , Amat Mercedes 
Published: June 2016

AbstractOxazolopiperidone lactams undergo an unprecedented reductive ring opening upon treatment with LiNH2BH3.
ChemInform Abstract: Visible Light‐Induced Iodine‐Catalyzed Transformation of Terminal Alkynes to Primary Amides via CC Bond Cleavage under Aqueous Conditions.
Authors: Dighe Shashikant U. , Batra Sanjay 
Published: June 2016

AbstractThis metal‐free protocol, which ensues via initial hydroamination of the acetylene bond, followed by release of CH2I2, is suitable for aromatic, heteroaromatic, and aliphatic alkynes.
ChemInform Abstract: Catalytic Suzuki Couplings by an Amido Pincer Complex of Palladium.
Authors: Liang Lan‐Chang , Chien Pin‐Shu , Song Liang‐Hua 
Published: June 2016

AbstractNoteworthy, the catalysis succeeds in the high yield production of sterically encumbered tri‐ortho‐substituted biaryls (VI).
ChemInform Abstract: Microwave Directed Metal‐Free Regiodivergent Synthesis of 1,2‐Teraryls and Study of Supramolecular Interactions.
Authors: Singh Surjeet , Shally Shally , Shaw Ranjay , Yadav Reena , Kumar Abhinav , Pratap Ramendra 
Published: June 2016

AbstractThe title compounds are prepared by ring transformation of pyrancarbonitriles by benzyl cyanides under basic conditions with moderate yields.
ChemInform Abstract: Concise Asymmetric Construction of C2‐Symmetric 1,9‐Diarylnonanoids Using a Hypervalent Silicon Complex: Total Synthesis of (‐)‐Ericanone.
Authors: Kotani Shunsuke , Kai Kosuke , Shimoda Yasushi , Hu Hao , Gao Shen , Sugiura Masaharu , Ogasawara Masamichi , Nakajima Makoto 
Published: June 2016

AbstractDiarylnonanoids are concisely synthesized by phosphine oxide‐catalyzed enantioselective double aldol reaction in one step.
ChemInform Abstract: DDQ‐Mediated Oxidative Radical Cycloisomerization of 1,5‐Diynols: Regioselective Synthesis of Benzo[b]fluorenones under Metal‐Free Conditions.
Authors: Zhu Hui , Chen Zhiyuan 
Published: June 2016

AbstractA synthesis of benzo[b]fluorenones via DDQ‐mediated oxidative cycloisomerization reaction of acyclic 1,5‐diynols is developed.
ChemInform Abstract: Cascade Pd(II)‐Catalyzed Wacker Lactonization—Heck Reaction: Rapid Assembly of Spiranoid Lactones.
Authors: Albarghouti Ghassan , Kotikalapudi Ramesh , Lankri David , Valerio Viviana , Tsvelikhovsky Dmitry 
Published: June 2016

AbstractThe new unprecedented Wacker—Heck lactonization‐cyclization reaction provides bi‐ and tricyclic spiranoid lactones in good yields.
ChemInform Abstract: 1,3‐Dipolar Cycloaddition Enabled Isoxazole‐Fused Spiropyrrolidine Oxindoles Syntheses from 3‐Methyl‐4‐nitro‐5‐alkenyl‐isoxazoles and Azomethine Ylides.
Authors: Liu Xiong‐Wei , Yao Zhen , Yang Jun , Chen Zhi‐Yong , Liu Xiong‐Li , Zhao Zhi , Lu Yi , Zhou Ying , Cao Yu 
Published: June 2016

Abstract1,3‐Dipolar cycloaddition of in situ thermally generated azomethine ylides with alkenyl substituted isoxazoles offers a convenient synthesis of fused spiropyrrolidine oxindoles in good diastereoselectivity.
ChemInform Abstract: The Deep Eutectic Melt of Sorbitol and Metformin Hydrochloride: Synthesis of 3‐Substituted 2‐Aminonaphtho[2,3‐b]furan‐4,9‐diones and Their Photophysical Properties.
Authors: Rad‐Moghadam Kurosh , Mousazadeh Hassani Seyyed Ali Reza , Toorchi Roudsari Saeedeh 
Published: June 2016

AbstractThe title compounds are obtained in one‐pot by reaction of naphthoquinone, various β‐nitrostyrenes, and ammonium acetate using the deep eutectic melt as readily available, biocompatible, and easily recyclable catalytic system.
ChemInform Abstract: Iodine Mediated Intramolecular C2‐Amidative Cyclization of Indoles: A Facile Access to Indole Fused Tetracycles.
Authors: Badigenchala Sindhura , Rajeshkumar Venkatachalam , Sekar Govindasamy 
Published: June 2016

AbstractA novel, metal‐free and efficient iodine mediated intramolecular sulfonamidation of indoles is reported which gives general access to different indole fused heterocycles.
ChemInform Abstract: Synthesis of Tetra‐Substituted 5‐Trifluoromethylpyrazoles via Sequential Halogenation/Palladium‐Catalyzed C—C and C—N Cross‐Coupling.
Authors: Wiethan Carson , Rosa Wilian C. , Bonacorso Helio G. , Stradiotto Mark 
Published: June 2016

AbstractThe new synthetically useful methodology to construct tetrasubstituted trifluoromethylpyrazoles involves halogenation of starting trifluoromethylpyrazoles, and subsequent palladium‐catalyzed Negishi coupling or Buchwald‐Hartwig amination with (hetero)arylzinc chlorides and primary alkylamines.
ChemInform Abstract: Conversion of Carbon Dioxide into 2‐Oxazolidinones and 2(3H)‐Oxazolones Catalyzed by 2,2′,2′′‐Terpyridine.
Authors: Liu Huixin , Hua Ruimao 
Published: June 2016

Abstract2,2′,2′′‐Terpyridine is described as efficient catalyst for the three component reaction of propargyl alcohols, primary amines and CO2 to give oxazolidinone derivatives (IV) and (VI).
ChemInform Abstract: An Efficient and Tunable Route to Bis(1,2,3‐triazol‐1‐yl)methane‐Based Nitrogen Compounds.
Authors: Castro‐Osma Jose A. , Lara‐Sanchez Agustin , Otero Antonio , Rodriguez Ana M. , de la Torre Maria C. , Sierra Miguel A. 
Published: June 2016

Abstract1,3‐Dipolar cycloaddition of geminal diazides with alkynes provides the title species (III) and (V).
ChemInform Abstract: A General Metal‐Free Route Towards the Synthesis of 1,2,3‐Triazoles from Readily Available Primary Amines and Ketones.
Authors: Thomas Joice , Jana Sampad , John Jubi , Liekens Sandra , Dehaen Wim 
Published: June 2016

AbstractAn unprecedented selective preparation of 1,5‐disubstituted 1,2,3‐triazoles from readily available primary amines, enolizable ketones and 4‐nitrophenyl azide as a renewable source of dinitrogen is developed.
ChemInform Abstract: A Binuclear Cu(I) Complex as a Novel Catalyst Towards the Direct Synthesis of N‐2‐Aryl‐substituted‐1,2,3‐triazoles from Chalcones.
Authors: Singh Divya Pratap , Allam Bharat Kumar , Singh Rahul , Singh Krishna Nand , Singh Vinod Prasad 
Published: June 2016

AbstractThe title triazoles are prepared by click reaction of chalcones and sodium azide followed by N‐arylation with (di)nitrohalobenzenes.
ChemInform Abstract: Bovine Serum Albumin Catalyzed One‐Pot, Three‐Component Synthesis of Dihydropyrano[2,3‐c]pyrazole Derivatives in Aqueous Ethanol.
Authors: Dalal Kiran S. , Tayade Yogesh A. , Wagh Yogesh B. , Trivedi Darshak R. , Dalal Dipak S. , Chaudhari Bhushan L. 
Published: June 2016

AbstractAn environmentally benign method for preparation of the title compounds by reaction of ketones/isatins/aldehydes with malononitrile and pyrazolone is developed.
ChemInform Abstract: Inherently Chiral Heterocyclic Resorcinarenes Using a Diels—Alder Reaction.
Authors: Iwanek W. , Stefanska K. , Szumna A. , Wierzbicki M. 
Published: June 2016

AbstractThe title compounds are prepared with unusually high diastereoselectivity in one‐pot via thermal generation of o‐quinomethide resorcinarene derivatives and subsequent Diels—Alder reaction with dienophiles, such as α‐methylstyrene.
ChemInform Abstract: Palladium‐Catalyzed Thioetherification of Quinolone Derivatives via Decarboxylative C—S Cross‐Couplings
Authors: Xia Chengcai , Wei Zhenjiang , Yang Yong , Yu Wenbo , Liao Hanxiao , Shen Chao , Zhang Pengfei 
Published: June 2016

Abstractusing diaryl disulfides
ChemInform Abstract: Copper‐Mediated Cross‐Dehydrogenative Coupling of 2‐Methylpyridine and 8‐Methylquinoline with Methyl Ketones and Benzamides.
Authors: Kumar Gadde Sathish , Boyle Joshua William , Tejo Ciputra , Chan Philip Wai Hong 
Published: June 2016

AbstractMethyl ketones as coupling partners seem to react via an aldehyde intermediate, whereas benzamides and an aniline derivatives seem to react via a radical mediated process.
ChemInform Abstract: A Simple, Efficient and Solvent‐Free Reaction for the Synthesis of Quinolines Using Caesium Iodide.
Authors: Mokhtarpour Nazanin , Eshghi Hossein , Bakavoli Mehdi , Eshkil Fatemeh 
Published: June 2016

AbstractThe new method has the advantages of good yields, a clean reaction, simple methodology, short reaction times, easy work‐up and green conditions.
ChemInform Abstract: Nano‐NiFe2O4 Catalyzed Microwave Assisted One‐Pot Regioselective Synthesis of Novel 2‐Alkoxyimidazo[1,2‐a]pyridines under Aerobic Conditions
Authors: Payra Soumen , Saha Arijit , Banerjee Subhash 
Published: June 2016

Abstractstarting from 2‐aminopyridine, β‐nitrostyrenes, and various alcohols
ChemInform Abstract: Multicomponent Cascade Reaction: Dual Role of Copper in the Synthesis of 1,2,3‐Triazole Tethered Benzimidazo[1,2‐a]quinoline and Their Photophysical Studies.
Authors: Nagesh Hunsur Nagendra , Suresh Amaroju , Reddy Muthyala Nagarjuna , Suresh Narva , Subbalakshmi Jayanty , Chandra Sekhar Kondapalli Venkata G. 
Published: June 2016

AbstractThe title compounds are prepared from (azidomethyl)benzimidazoles, acetylenes, and benzaldehydes by domino/cascade reaction including click reaction, N—C bond formation, and Knoevenagel condensation.
ChemInform Abstract: Gold‐Catalyzed Chemo‐ and Diastereoselective C(sp2)—H Functionalization of Enaminones for the Synthesis of Pyrrolo[3,4‐c]‐quinolin‐1‐one Derivatives.
Authors: Zhao Yulei , Duan Qizhao , Zhou Yuanyuan , Yao Qiyi , Li Yanzhong 
Published: June 2016

AbstractNovel one‐pot procedure for the synthesis of pyrrolo[3,4‐c]‐quinolinones starting from enaminones and diazo compounds by sequential addition of the Au(I) catalyst and TosOH under mild reaction conditions is developed.
ChemInform Abstract: Mechanistic Insights into a Catalyst‐Free Method to Construct Quinazolinones Through Multiple Oxidative Cyclization.
Authors: Wang Zhen‐zhen , Tang Yu 
Published: June 2016

AbstractAn oxidative cyclization of 2‐aminobenzamides with benzylic alcohols is developed to give varying yields of 2‐acylated quinazolinones in the presence of elemental oxygen as terminal oxidant.
ChemInform Abstract: First Catalytic Asymmetric Hydrogenation of Quinoxaline‐2‐carboxylates.
Authors: Maj Anna M. , Heyte Svetlana , Araque Marcia , Dumeignil Franck , Paul Sebastien , Suisse Isabelle , Agbossou‐Niedercorn Francine 
Published: June 2016

AbstractThe catalytic hydrogenation of alkyl quinoxaline‐2‐carboxylates is studied under continuous flow conditions in the presence of in situ generated Ir‐catalyst but the resulting ee′s are rather low.