Patent SG-11201901438V-A (SG)
Title: Solid forms of cenicriviroc mesylate and processes of making solid forms of cenicriviroc mesylate
Inventor: PHIASIVONGSA PASIT
IPC: A61K45/00
Filed: 2017-08-30
Abstract: INTERNATIONAL APPLICATION PUBLISHED UNDER THE PATENT COOPERATION TREATY (PCT) (19) World Intellectual Property Organization International Bureau (43) International Publication Date 08 March 2018 (08.03.2018) WIP0 I PCT ill~~~~~~~~ 011101010VIIIOH olo olommoonmll °nom oimIE (10) International Publication Number WO 2018/045043 Al (51) International Patent Classification: A61K 31/395 (2006.01) A61K 31/513 (2006.01) A61K 31/4164 (2006.01) A61K 31/55 (2006.01) A61K 31/4178 (2006.01) A61K 45/00 (2006.01) (21) International Application Number: PCT/US2017/049400 (22) International Filing Date: 30 August 2017 (30.08.2017) (25) Filing Language: English (26) Publication Language: English (30) Priority Data: 62/382,153 31 August 2016 (31.08.2016) US (71) Applicant: TOBIRA THERAPEUTICS, INC. [US/US]; 400 Interpace Parkway, Parsippany, New Jersey 07054 (US). (72) Inventors: PHIASIVONGSA, Pasit; 930 Mission Road, Unit 29, South San Francisco, California 94080 (US). COOPER, Martin Ian; c/o Johnson Matthey Plc., Phar- morphix, 250 Cambridge Science Park, Milton Road, Cam- bridge Cambridgeshire CB4 OWE (GB). SHARP, Em- ma Kay; c/o Johnson Matthey Plc., Pharmorphix, 250 Cambridge Science Park, Milton Road, Cambridge Cam- bridgeshire CB4 OWE (GB). (74) Agent: BLINKA, Thomas A. et al.; Cooley LLP, 1299 Pennsylvania Avenue, N.W., Suite 700, Washington, Dis- trict of Columbia 20004-2400 (US). (81) Designated States (unless otherwise indicated, for every kind of national protection available): AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DJ, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JO, JP, KE, KG, KH, KN, KP, KR, KW, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW. (84) Designated States (unless otherwise indicated, for every kind of regional protection available): ARIPO (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW), Eurasian (AM, AZ, BY, KG, KZ, RU, TJ, TM), European (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, (54) Title: SOLID FORMS OF CENICRIVIROC MESYLATE AND PROCESSES OF MAKING SOLID FORMS OF CENICRIVIROC MESYLATE 24 2-Theta Scale FIG. 1 (57) : The invention relates to solid forms of cenicriviroc mesylate, methods of their preparation, pharmaceutical compositions C thereof and methods of their use. [Continued on next page] WO 2018/045043 Al MIDEDIMOHNIIMEIHRIMENNIMIRMOVOIS TR), OAPI (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG). Published: with international search report (Art. 21(3)) before the expiration of the time limit for amending the claims and to be republished in the event of receipt of amendments (Rule 48.2(h))