baber/WOPTO huggingface dataset:
Patent IE-41525-B1 (IE)
Title: Meyhods and compositions for improving subsituded phenylglycephalosporins
IPC: C07D501/36
Filed: 1974-07-24
Abstract: 1449071 Substituted 7 - α - amino - α - phenylacetamidocephalosporins SMITHKLINE CORP 31 July 1974 [1 Aug 1973] 33764/74 Heading C2C The invention comprises compounds (I) where Y is -O-, -NH- or -S-; n is an integer of 1-5 ; R is -NH 2 , -OH or -O(C 1-4 - alkyl); M is hydrogen, ammonium or an alkali metal cation; and A is hydrogen, acetoxy, pyridinium, -SHet, -SH, -S(C 1-4 alkyl), -OH or -O(C 1-4 alkyl), Hot being a 5- or 6- membered heterocyclic ring containing carbon atoms and 1-4 N, O or S atoms, the ring being optionally substituted by 1 or 2 C 1-4 alkyl, C 1-4 alkoxy (C 1-4 alkyl), OH, CF 3 , SH or S(C 1-4 alkyl) groups. The compounds may be prepared by acylating a 7-aminocephalosporanic-acid with the appropriate phenylglycine; any necessary protective groups then being removed, and salts being converted to the zwitternonic form by known methods. 7 - Amino - 3 - (1 - methyl - 1,2,3,4 - tetrazol - 5- yl - thiomethyl) - 3 - cephem - 4 - carboxylic acid is made by reacting 7-aminocephalosporanic acid with 1-methyl-5-mercapto-1,2,3,4 - tetrazole. The 3 - (5 - methyl - 1,3,4 - thiadiazol - 2- ylthiomethyl) - and 3 - (1,2,3 - triazol - 4 - ylthiomethyl)-compounds are formed similarly.
Patent IE-49972-B1 (IE)
Title: Sanitary towels and other absorbent elements
IPC: A61F13/15
Filed: 1980-08-08
Abstract: A sanitary towel, baby nappy, bandage or other absorbent element comprises an absorbent material (9, 10) enclosed within an envelope including a layer of non-woven material (6) to contact the skin of the user. A layer (11) of a flexible material which has been expanded in a manner analogous to "expanded metal" by slitting and stretching perpendicular to the direction of the parallel lines of slits is included in the envelope with the absorbent material either as a flexible reinforcement or to facilitate passage of body liquids from the non-woven material (6) to the absorbent material (9, 10).
Patent IE-47160-B1 (IE)
Title: Apparatus for hide stretching
IPC: C14B1/26
Filed: 1978-08-28
Abstract: A hide stretching apparatus, in particular one for the tentering of hides for drying. The apparatus comprises a stretching frame with a number of mutually spaced radial sliding guides. The stretching clamps gripping the edges of the hide have been arranged to be reciprocatingly movable along the sliding guides. The stretching frame is placed upon a special hide changing table carrying under each sliding guide a clamp displacement member. The clamps carry jaws which attach to the edge of the hide to be stretched. The jaws are opened and closed by means of a lever turnably carried on the clamp. The clamp displacement member has two gripping members, which can be made to engage the clamp on both sides according to commands given, for the displacing of the clamps reciprocatingly along the sliding guides. The clamp comprises a brake engaging with the sliding guide and which with the jaws in closed position prevents the displacement of the clamp towards the center of the stretching frame. The lever turning the jaws into their opened and closed position pushes, when the jaws are opened, the brake against the force of a spring into a position such that the clamp is free to move in either direction, whereby the clamps can be moved into clamping position and into detachment position.
Patent IE-81120-B1 (IE)
Title: Esters of hyaluronic acid and their salts
Inventor: VALLE FRANCESCO DELLA
IPC: D01F/
Filed: 1986-07-04
Abstract: The invention concerns the esters of hyaluronic acid in which all or only a portion of the carboxylic groups of the acid are esterified, and the salts of the partial esters with metals or with pharmacologically acceptable organic bases. The compounds possess interesting and precious bio- plastic and pharmaceutical properties and may be used in innumerable fields, including cosmetics, surgery and medicine. The invention also includes pharmaceutical preparations containing, as an active ingredient, one or more hyaluronic acid esters, or a salt thereof as described above, as well as medicaments containing: 1) a pharmacologically active substance or an association of pharmacologically active substances and 2) a carrying vehicle containing a total or partial ester of hyaluronic acid. The invention includes also various uses of the hyaluronic esters or of the above mentioned medicaments, such as in medicine, surgery or cosmetics. The invention also relates to a new procedure for the preparation of polysaccharide esters containing carboxylic groups, such as in particular the above mentioned hayluronic acid esters.
Patent IE-47450-B1 (IE)
Title: Pharamaceutical compositions
IPC: A61K31/42
Filed: 1978-10-10
Abstract: A dry unit-dose pharmaceutical composition suitable for oral administration comprises 20 mg to 1500 mg of amoxycillin trihydrate, 20 mg to 500 mg of potassium clavulanate and a pharmaceutically acceptable carrier with the proviso that the weight ratio of amoxycillin trihydrate to potassium clavulanate is from 6:1 to 1:1.
Patent IE-57931-B1 (IE)
Title: Hyaluronic acid fractions having pharmaceutical activity,methods for preparation thereof,and pharmaceutical compositions containing the same
IPC: A61K47/36
Filed: 1984-10-10
Abstract: Two pharmaceutically useful fractions of hyaluronic acid are obtained comprising a first fraction with a molecular weight between 50,000 and 100,000 which is useful for wound healing, and a second fraction having a molecular weight between 500,000 and 730,000 which is useful for intraocular and intraarticular injections. The fractions of hyaluronic acid are further useful as vehicles for opthalmic drugs, provided formulations compatible with the corneal epithelium and enhancing in vivo activity of such drugs.
Patent IE-56307-B1 (IE)
Title: Hydroxyalkyl-azolyl derivatives substituted by heterocyclic substituents
IPC: A01N43/653
Filed: 1983-11-14
Abstract: Heterocyclyl-hydroxyalkyl-azolyl derivatives of the formula <IMAGE>  (I)  in which Az represents 1,2,4-triazol-1-yl, 1,2,4-triazol-4-yl or imidazol-1-yl, Het represents optionally substituted dioxolanyl or 1,3-dioxanyl, R represents alkyl, optionally substituted phenyl, optionally substituted phenylalkyl, optionally substituted phenoxyalky, optionally substituted phenylthioalkyl, optionally substituted cycloalkyl, optionally substituted cycloalkylalkyl, alkenyl, optionally substituted phenylalkenyl, optionally substituted cyclohexylalkenyl, furyl, naphthyloxymethyl or azolylalkyl, R' represents hydrogen, optionally substituted alkyl or alkenyl and n represents the number 0 or 1, or addition products thereof with acids or metal salts, which possess fungicidal activity.
Patent IE-66823-B1 (IE)
Title: Derivatives of 1,2,3,4-tetrahydro-9-acridinamine
Inventor: GRANGER COLIN
IPC: A61K31/00
Filed: 1990-07-30
Abstract: Novel prodrugs or depot derivatives of 1,2,3,4-tetrahydro-9-acridinamine of formula I <CHEM> are described, as well as methods for the preparation and pharmaceutical compositions of same, which are useful as analgesic agents for the treatment of pain, as sleep aids and as agents for treating the symptoms of senile dementia, Alzheimer's disease, Huntington's chorea, tardive dyskinesia, hyperkinesia, mania, or similar conditions of cerebral insufficiency characterized by decreased cerebral acetylcholine production or release.
Patent IE-52172-B1 (IE)
Title: (+)-4-substituted-2-indanols and insecticidal ester derivatives
IPC: C07C53/23
Filed: 1981-12-21
Abstract: Novel compounds of the formula (FORMULA) in which Rs is a phenyl, phenoxy, phenylthio, benzyl or heterocyclic radical which may be substituted, Rs is hydrogen, a substituted-vinylcyclopropane carbonyl group, a tetramethylcyclopropanecarbonyl group, or a 1-(substituted-phenyl)-2-methylpropylcarbonyl group, and the isomer of S configuration at C-2 of the indanyl ring is present in an enantiomeric excess over the isomer of R configuration. Also disclosed is a method for preparing the optically active alcohols. The compounds wherein R is other than hydrogen are insecticides.
Patent IE-62738-B1 (IE)
Title: Araliphatylaminoalkanediphosphonic acids
Inventor: JAEGGI KNUT A
IPC: C07F9/58
Filed: 1988-12-09
Abstract: Araliphatylaminoalkanediphosphonic acids of the formula <IMAGE> in which R1 represents an aromatically substituted aliphatic radical, R2 represents hydrogen or a monovalent aliphatic radical and alk denotes a divalent aliphatic radical, and their salts have a marked regulating action on calcium metabolism and can be used as medicaments for the treatment of diseases which can be traced back to disorders thereof. They are prepared, for example, by reacting a compound of the formula <IMAGE> in which X3 denotes carboxyl and R0 denotes a radical R2, with phosphorous acid and phosphorus trichloride and hydrolysing the primary product.
Patent IE-64696-B1 (IE)
Title: Medico-surgical and sanitary articles and materials
Inventor: WHITESIDE NEIL ADRIAN
IPC: A61F5/445
Filed: 1992-07-01
Abstract: A w.c. disposable ostomy bag (1) has its walls (2,4) made from a material comprising an outwardly presented layer (12) of alkali-soluble carboxylated acrylic polymer and a thinner, inwardly presented layer (18) of alkali-resistant polyvinylidene chloride. The inner layer (18) is applied as an aqueous coating to the outer layer (12) and is 2-3 micron thick which is sufficient to reduce odour transmission to an acceptable level. The bag is disposed of by adding an alkali to water in the w.c. so that the outer layer is broken up or dispersed whereas the inner layer is thin enough not to impede flushing.
Patent LU-100160-B1 (LU)
Title: Verwendung einer supraleitenden Leiteranordnung und Transportsystem mit einer supraleitenden Leiteranordnung
Inventor: REISER WOLFGANG
IPC: H02G15/34
Filed: 2017-04-04
Granted: 2018-10-15
Abstract: Die Erfindung betrifft eine Verwendung einer supraleitenden Leiteranordnung und ein Transportsystem mit einer supraleitenden Leiteranordnung. Die erfindungsgemäße Besonderheit liegt nun darin, dass das eigentlich störende Magnetfeld einer stromdurchflossenen supraleitenden Leiteranordnung zur Versorgung eines Verbrauchers gleichzeitig als elektromagnetisches Schwebesystem für ein Transportmittel genutzt wird. Die Leiteranordnung bildet daher „nebenbei" eine Träger- und/oder Führungsschiene für eine entlang der supraleitenden Leiteranordnung über die Länge körperkontaktfrei mittels des Magnetfeldes in Schwebe haltbaren und bewegbaren Transportkapsel. Der hohe Infrastrukturaufwand für eine sich über die Länge einer supraleitenden Stromleitung erstreckende Kühlung, deren Betrieb zudem hohe Kosten und Energie erfordert, fällt somit nur einmal an. Die dringend benötigten Stromtrassen werden somit zugleich auch ein modernes Transportsystem bzw. umgekehrt
Patent LU-101876-B1 (LU)
Title: Bridge pier testing device
Inventor: ZHANG JUN
IPC: E01D19/10
Filed: 2019-02-14
Granted: 2020-10-26
Abstract: The present invention provides a bridge pier testing device based on an electromagnetic spring technique, including an upper clamping mechanism, a lower clamping mechanism and a traction mechanism. The structure of the upper clamping mechanism is identical to the structure of the lower clamping mechanism. The upper clamping mechanism includes a housing, an upper clamping body and a lower clamping body. A ring top plate of the upper clamping body is fixedly mounted on a top fixed ring plate. The lower clamping body can axially move up and down inside the housing. The clamping electromagnet magnetically attracts the clamping iron block, so that the lower clamping body moves axially upward, and the wedge-shaped push head pushes the clamping support body to move radially inwards, so as to clamp the bridge pier. The traction electromagnet is energized to attract the traction iron block. The traction iron block pulls the traction rope so that the lower clamping mechanism moves axially relative to the upper clamping mechanism. The device of the present invention uses a powerful mechanical clamping mechanism to clamp the bridge pier, and the clamping mechanism can bear a large dead load without slipping during the testing process, which has good stability.
Patent LU-102865-B1 (LU)
Title: Microfluidic mixer
Inventor: HORNER DANIEL
IPC: B01L3/00
Filed: 2021-10-14
Granted: 2023-04-21
Abstract: The invention relates to and provides a microfluidic mixer, formed by two parts, a first part being a substrate having formations defining fluid channels on an outer surface that is directed towards a second part, which is a flexible layer, wherein the flexile layer has formations defining fluid channel which, when the flexible layer is positioned over the substrate so as to cover the fluid channels of the substrate to provide a fluid communication path, wherein a section of said communication path comprises at least a first and a second fluid channel for providing a first and a second fluid, wherein first and second fluid channel merge before an inlet of a mixing chamber into a merged fluid channel, wherein the mixing chamber comprises perturbation formations, and an outlet of the mixing chamber is connected to an outlet fluid channel, wherein the flexible layer comprises points for compression at the inlet and outlet of the mixing chamber for closing the merged fluid channel and the outlet fluid channel connected to inlet and outlet of the mixing chamber.
Patent LU-500324-B1 (LU)
Title: Photoelectric intelligent coal sorting device and sorting method therefor
Inventor: LIU LINGYUN
IPC: B07C5/36
Filed: 2021-06-24
Granted: 2022-01-07
Abstract: The present disclosure belongs to the field of coal sorting and specifically discloses a photoelectric intelligent coal sorting device and a sorting method therefor. The photoelectric intelligent coal sorting device includes: a conveyor belt; a guide assembly configured to guide a mixture of coal and gangue on the conveyor belt, so that units of the mixture of coal and gangue are arranged and conveyed in sequence in the middle of the conveyor belt; an identification assembly configured to identify the units of the mixture of coal and gangue on the conveyor belt that are arranged and conveyed in sequence in the middle of the conveyor belt and distinguish between the coal and the gangue; a sorting assembly configured to classify, by using the coal and the gangue as classification objects, the units of the mixture of coal and gangue that has been identified by the identification assembly; and a collection bin including a coal bin and a gangue bin separated by a separator. In this way, the coal and the gangue can be quickly sorted into the corresponding coal and gangue bins.
Patent NO-306332-B1 (NO)
Inventor: KAULE WITTICH
IPC: B32B7/00
Filed: 1995-08-18
Abstract: A transfer foil for use in a safety document includes a multilayer structure having a carrier layer and a plastic layer in which diffraction structures, for example holographic structures, are embossed in the form of a relief structure and which is combined with a reflective layer. The plastic layer includes a reaction lacquer layer selected from the group consisting of cationical curing lacquers, blue light-curing lacquers and chemical curing multicomponent lacquers.
Patent NO-304517-B1 (NO)
Inventor: YANAGISAWA HIROAKI
IPC: C07D401/04
Filed: 1995-11-09
Abstract: N-Phenylbenzyl imidazole derivs. of formula (I) and their pharmaceutically acceptable salts and esters are new. In (I), R1 = 1-6C alkyl or 3-6C alkenyl; R2 and R3 = H, 1-6C alkyl, 3-6C alkenyl, 3-10C cycloalkyl (opt. polycyclic), aryl(1-6C)alkyl, aryl or aryl fused to 3-10C cycloalkyl; R4 = H, 1-6C alkyl, 1-6C alkanoyl (opt. substd. by one or more halo or 1-6C alkoxy if other than formyl), 3-6C alkenoyl, arylcarbonyl, 1-6C alkoxycarbonyl, tetrahydropyranyl, tetrahydrothiopyranyl, tetrahydrothienyl or tetrahydrofuryl (these 4 opt. substd. by one or more halo or 1-6C alkoxy), SiRaRbRc, 1-6C alkoxymethyl, 1-6C alkoxy(1-6C)alkoxymethyl, halo(1-6C)alkoxymethyl, 1-6C alkyl substd. by at least one aryl, or 1-6C alkanoyl-oxymethoxycarbonyl; Ra, Rb and Rc = 1-6C alkyl or aryl, but not all aryl; R5 = COOH or CONR8R9; R8 and R9 = H, 1-6C alkyl (opt. substd. by at least one (a)) or together are 2-6C alkylene opt. substd. by at least one COOH or alkoxycarbonyl; R6 = H, 1-6C alkyl or alkoxy, or halo; R7 = COOH or tetrazol-5-yl; (a) = aryl, 5-6 membered heterocyclic with 1-4 N, O and/or S, halo, OH, 1-6C alkoxy, COOH, 1-6C alkoxycarbonyl, NH2 or acylamino (acyl = 1-6C alkanoyl or arylcarbonyl); aryl = 6-14C aromatic carbocyclic gp. opt. substd. by at least one of NO2, CN, halo, 6-10C carbocyclic aryl (unsubstd.), 1-6C alkyl or alkoxy, COOH, 1-6C alkoxy-carbonyl, or 1-3C alkylenedioxy or alkylidenedioxy. 23 Cpds. e.g. pivaloyloxymethyl (or (5-methyl-2-oxo -1,3-dioxolen-4-yl)methyl) 4-(1-hydroxy-1-methylethyl) -2-(ethyl, propyl or butyl)-1-(4-(2-tetrazol -5-yl)phenyl)phenyl)methylimidazole -5-carboxylate.
Patent NO-312055-B1 (NO)
Inventor: MARKWELL ROGER EDWARD
IPC: A61P25/28
Filed: 1997-04-24
Abstract: PCT No. PCT/EP95/04082 Sec. 371 Date Apr. 25, 1997 Sec. 102(e) Date Apr. 25, 1997 PCT Filed Oct. 17, 1995 PCT Pub. No. WO96/12486 PCT Pub. Date May 2, 1996A method of enhancing amyloid precursor protein processing along a non-amyloidogenic pathway in patients suffering from, or at risk of developing, Alzheimer's disease and a method of treatment or prophylaxis of Alzheimer's disease by reducing  beta A4 production in patients suffering from, or at risk of developing, Alzheimer's disease comprising administering to the patient an effective, non-toxic amount of an acetonitrile compound, use of the compound in preparation of a medicament for use in the method and a composition for use in the method.
Patent NO-323853-B1 (NO)
Inventor: ALLISON DANIELL S
IPC: A01K67/027
Filed: 1999-01-04
Abstract: The present invention relates to regulatory DNA sequences derived from the hamster EF-1± gene. The invention further encompasses expression constructs comprising regulatory DNA of the invention, host cells transformed or transfected with the regulatory DNA and methods of increasing gene transcription utilizing the regulatory DNA. Expression constructs comprising regulatory DNA of the invention operably linked to specific gene sequences are also comprehended.
Patent NO-325272-B1 (NO)
Inventor: HOPKINS TERENCE
IPC: A61P33/10
Filed: 1999-01-14
Abstract: The present invention relates to the preparation of orally administrable granules of hexahydropyrazine derivatives by mixing the active compound in the presence of suitable solvents with hydrophobic carriers, if appropriate in the presence of auxiliaries, and converting the resulting mixture, if appropriate, into other ready-to-use forms.
Patent AT-505124-B1 (AT)
IPC: B24D7/16
Filed: 2007-04-20
Granted: 2010-02-15
Abstract: The grinding wheel (1) has an opening in a region of a rotary axis (A), and fastening regions surrounding the opening in both sides of the grinding wheel. The fastening regions extend in a radial direction such that the grinding wheel is placed between wheel flanges of a grinding machine. A region (7) comprising projections (8) is attached to the fastening regions in the radial direction, where the fastening regions and the projections are composed of plastic. Thee projections are arranged around the rotary axis in a radially symmetric manner. An independent claim is also included for a method for manufacturing a grinding wheel.
Patent BG-62044-B1 (BG)
Title: Device for the stabilization of a wheel transport vehicle
Inventor: MARINOV VESELIN T
IPC: B62D39/00
Filed: 1994-03-23
Abstract: The device is used in the transport industry. It can beincluded in transport vehicles having at least two symmetricalwheels, and it improves their stability, especially when runningat high speeds in a curve. The device consists of a frame (1) anda supporting beam (2) pivotly connected to it included as a lowerpart in the make of a pivot four-section part connected to wheels(6). The device also includes a driving mechanism which is fittedto frame (1) and contains a supporting rod (10) and a mobilecasing (11) sliding on it. To the casing a connection rod (12) ispivotly connected, the other end of which is pivotly connected tothe supporting beam in a point ouside the symmetry axis of thetransport vehicle. The mobile casing (11) is controlled by anactuation system which includes a distributor controlled by aninertia sensor.5 claims, 4 figures
Patent BR-0014919-B1 (BR)
Inventor: AEBLI BEAT MICHAEL
IPC: C08L101/00
Filed: 2000-10-12
Abstract: Aqueous storage-stable, non-sedimenting photoinitiator suspensions comprising (a) a mono- or bis-acylphosphine oxide of formula (I), wherein R1 is C1-C20alkyl; C2-C20alkyl interrupted by one or more O atoms; C1-C12alkoxy; phenyl-C1-C4alkyl; or phenyl that is unsubstituted or substituted by C1C20alkyl, C1-C12alkoxy, halogen, cyclopentyl, cyclohexyl, C2-C12alkenyl, C2-C18alkyl interrupted by one or more O atoms, and/or by phenyl-C1-C4alkyl; or R1 is biphenylyl; R2 is an aromatic radical or has one of the meanings give for R1; R3 and R4 are each independently of the other C1-C12alkyl, C1-C12alkoxy or halogen; and R5 is hydrogen, C1-C12alkyl, C1-C12alkoxy or halogen; (b) a dispersant; and (c) water are suitable especially in the photopolymerisation of aqueous formulations comprising ethylenically unsaturated monomers.
Patent BR-0112853-B1 (BR)
Inventor: DE WINTER HUGO
IPC: B29C45/14
Filed: 2001-07-31
Abstract: A method for manufacturing at least a skin (2) for forming a visible front surface (3) of an interior trim part which comprises at least one premanufactured insert (6) showing a back face (7) situated at a distance behind said visible surface. The skin is made by applying at least one flowable skin material for producing an elastomeric, non-cellular or micro-cellular plastic skin (2) against at least one surface of a mould and by allowing this flowable skin material to harden. The insert (6) is maintained with its front face (12) at a distance from the mould surface against which the skin (2) is moulded by applying, before positioning the insert (6) into the mould, a first layer (33) of the flowable skin material against said mould surface and by positioning the insert (6) onto this first layer (33). A second layer (34) of a further flowable skin material is subsequently applied against a back side of said first layer (33) and against at least one side of the insert (6) so that the insert is adhesively fixed to said plastic material.
Patent BR-0210948-B1 (BR)
Inventor: ASRAR JAWED
IPC: A01N55/00
Filed: 2002-07-10
Abstract: A method of producing lignin-based matrix microparticles for the controlled release of an agricultural active includes forming an emulsion of an organic solution in an aqueous solution, wherein the organic solution contains a lignin derivative and an agricultural active in a volatile organic solvent and the aqueous solution contains an emulsifier; and removing the organic solvent, thereby producing microparticles having a matrix comprising the lignin derivative within which the agricultural active is distributed. Small, spherical lignin-based matrix microparticles that release an agricultural active at a controlled rate are described, as are plants and plant propagation materials that are treated with such microparticles.