baber/WOPTO huggingface dataset:
Patent CZ-286516-B6 (CZ)
Title: Recovery process of physical and mechanical properties of railway track bed  ballast and apparatus for making the same
Inventor: AMBROZ LUDVIK
IPC: E01B37/00
Filed: 1996-12-03
Abstract: The proposed recovery process of physical and mechanical properties of railway track bed  ballast is characterized in that ballast is subjected to working process by the action of mechanical forces under interaction of physical surface and capillary forces at a temperature in the range of -2 to 60 degC in order to remove undesired soft admixtures and fine grain fraction. The apparatus for making the process is formed by a machine (14) for preliminary treatment having a water feeding device (13), a kinetic crusher (10) with a rotor (3) with either horizontal or vertical axis of rotation and provided with a rebound strips (8) and a stator (2) with impact plates (6) that are arranged on supporting segments (5) with adjusting mechanisms (4) for adjusting the profiled impact plates (6), a sieve sorter (18) with cascades of flat vibrating screens being provided with motors, rubber conveyor belts (16a, 16b) of various lengths and vibrating feeding troughs (17a, 17b). The machine (14) has a gap (y) extending between the kinetic crusher (10) rotor (3) rebound strips (8) and the supporting segment (5) impact plates (6), which gap (y) is adjustable within the range of 10 to 300 mm through the mediation of an adjusting mechanism (4).
Patent SK-285979-B6 (SK)
Title: Process for the preparation of substituted thiazolidinedione
Inventor: GILES ROBERT GORDON
IPC: C07D417/12
Filed: 1998-02-13
Abstract: A process for preparing 5-{4-[2-(N-methyl-N-(2- pyridyl)amino)ethoxy]benzyl}-2,4-thiazolidinedione (a compound of formula (IA)) or a tautomeric form thereof or a pharmaceutically acceptable salt thereof or a pharmaceutically acceptable solvate thereof, which process comprises reducing 5-{4-[2-(N-methyl-N-(2- pyridyl)amino)ethoxy]benzyl}-2,4-thiazolidinedione (a compound of formula (IIB)) or a tautomeric form thereof or a salt thereof or a solvate thereof, with a complex hydride reducing agent; and thereafter, as required, preparing a pharmaceutically acceptable salt or a pharmaceutically acceptable solvate of the compound of formula (I) or a tautomeric form thereof.
Patent SK-278865-B6 (SK)
Title: Interphenylene-7-oxabicycloheptyl substituted heterocyclic amide prostaglandin analogs, method for their preparing, pharmaceutical composition and use
Inventor: MISRA RAJ NARAIN
IPC: C07D405/04
Filed: 1990-03-30
Abstract: This patent describes analogue compounds related to prostaglandin of hetero cyclic amines with a general formula (I), where the values of variables m, n, X, Y, R1, R2, R3 and R3a are described in a patent description, together with a procedure closed to the production of prostaglandin wit a general formula (I), where the individual symbols are of the described meaning, while a compound with a general formula (I), where R is of the described meaning, except carboxyl group, and its salts with alkaline metal and remaining general symbol are of the described meaning, is converted to halogenide of acid, and after that a reaction of this compound with amine having a general formula NHR1R2 is provided, and the symbols R1 and R2 are of the above mentioned meaning, and the resulting product can be divided to individual isomers and / or the product, where R means alkoxycarbonyl with 1 up to 12 carbon atoms in the alkoxyl part, is hydrolysed and a compound is created, where R means carboxyl group and this compound can be converted, so that the appropriate alkaline metal salt is created.
Patent SK-281799-B6 (SK)
Title: Method for production of human erythropoetin
Inventor: FRITSCH EDWARD
IPC: C12N15/85
Filed: 1985-12-03
Abstract: The invention refers to recombinant DNA plasmid vector containing cDNA encoding human EPO of clone lambda HEPOFL13 (ATCC 40153) and mammalian cell transformed with this vector or with a plasmid which contains the entire bovine papilloma virus DNA and the cDNA sequence of Table 3 coding for human EPO are which useful in the preparation of recombinant human erythropoietin which is characterized by the presence of O-linked glycosilation.
Patent SK-278010-B6 (SK)
Title: Generator of nonlinear functions with hysteresis
Inventor: CERNAK JOZEF
IPC: H03K3/02
Filed: 1990-10-11
Abstract: On first part (7) of information exit programable combining circuit (1) is connected the digital-analog converter (3), the second part (8) of information exit of programable combining circuit (1) is connected on inlet of register (2), exit (9) of register (2) and digital outlet (5) are connected on first input of programable combining circuit (1), on its second input is joined the system bus (10) of computer (4).
Patent CZ-297624-B6 (CZ)
Inventor: ROHLAND JOERG
IPC: B62D65/18
Filed: 2000-03-03
Abstract: Predlozené resení se týká prepravního zarízení pro svarovací prípravky trubkové konstrukce pro svarování cástí karoserií aut, zvláste podlahových cástí, s visutými tratemi (9, 10) pro prísun a odsun svarovaných cástí. Prícne k visutým dopravním tratím (9, 10) a mezi visutými dopravními tratemi (9, 10) jsou na obou stranách upínacího zarízení (1) pro svarované cásti usporádané vodicí nosníky (4) ana nich pojízdne ulozený výlozník (5). Na obou stranách výlozníku (5) smerem k dopravním tratím (9,10) jsou ulozené svisle pojízdne ulozené hlavní sane (14.1, 14.2), vzdy se dvema proti sobe umístenými vodicími listami (13, 15), na kazdé vodicí dráze (15) ve smeru dopravních tratí (9, 10) hlavníchsaní (14.1, 14.2) jsou ulozené svisle pojízdne ulozené drapákové sane (16), a mezi hlavními sanemi (14.1, 14.2) na výlozníku (5) jsou pripevnené pohánecí motory (19), vzdy pro jedny hlavní sane (14.1, 14.2) a jejich drapákové sane (16).
Patent CZ-299888-B6 (CZ)
Title: Smokable flat or tubular food package or film with low water-vapor permeability for packaging foodstuffs
Inventor: PAVLINEC JURAJ
IPC: A22C13/00
Filed: 2005-05-06
Abstract: The present invention relates to a smokable flat or tubular food package or film that is made of homogeneous plastic melt of plastic mixture containing polyamide, block polyether-ester copolymer and Na ionomer, whereby the mixture exhibits: a polyamide fraction in an amount of 45 to 94 percent by weight, a fraction of block polyether-ester copolymer in an amount of 5 to 45 percent by weight, and a fraction of Na ionomer in an amount of 1 to 10 percent by weight. The invention further relates to the use of such flat or tubular food package or film for the manufacture of smoked meat products smoked by natural or liquid smoke, whereby the package or film wall thickness of 25 microns, at the most, exhibits at a temperature of 25 degC a water-vapor permeability less than 120 g/me2 for a period of 24 hours.
Patent SK-288243-B6 (SK)
Title: Movable contact of electric apparatus, particularly breaker
Inventor: HRUZA RADEK
IPC: H01H73/04
Filed: 2005-12-15
Abstract: A movable contact (1) of an electrical apparatus, in particular circuit breaker, is composed of the mutually associated bearing part (2) and the arm contact (3), wherein the electric conductive arm contact (3) comprising at least one transverse U-section, longitudinally and symmetric arranged at the end of the nose piece (2) of the moving contact (1). Arm contact (3) in the part of deployment to the end of the nose piece (2) of the moving contact (1) entails a transverse spot weld (8) together with the end of the electroconductive wire (9) of any of the trigger (4, 5) of the electrical apparatus or connected thereto by riveting, bonding or press-fitting according to the choice, whether the arm contact (3) is formed in the U-section by bent conductive shoulder, moldings from electroconductive metal or the casting and the like.
Patent SK-287208-B6 (SK)
Title: Dispensing device and method for filling thereof
Inventor: MAAS WILHELMUS JOHANNES JOSEPH
IPC: B05B11/00
Filed: 2001-11-27
Abstract: Dispensing device (1), comprising a container (2) and a dispensing head (5) connected thereto, said container (2) and head (5) including a co-operating snap coupling means comprising a plurality of lugs (6, 7) arranged on one of the two parts to be connected and a plurality of recesses (8) arranged in the other part for receiving the lugs (6, 7), in which at least one of the lugs (6, 7) is resiliently deformable and at least one other lug is relatively stiff and non-deformable. Such a dispensing device may swiftly and easily be filled and assembled (1). At least the lugs are advantageously made of thermoplastic polyester, like e.g. PET. The invention further relates to a method for filling such a dispensing device with a medium to be dispensed.
Patent SK-286984-B6 (SK)
Title: Use of derivatives of 3(2H)-pyridazinone for preparation of medicament for treatment of erectile dysfunction
Inventor: TANIKAWA KEIZO
IPC: A61K31/00
Filed: 1999-11-30
Abstract: This invention relates to the use of derivatives of 3(2H)-pyridazinone of the general formula (I) for the preparation of a medicament for the treatment of erectile dysfunction. Specifically, the 4-bromo-6-[3-(4-chlorophenyl)propoxy)-5-(3- pyridylmethylamino)-3(2H)-pyridazinone or 4-bromo-6-[3-(4- chlorophenyl)-3-hydroxypropoxy)-5-(3-pyridylmethylamino)-3(2H)- pyridazinone or a pharmaceutically acceptable salt thereof.
Patent SK-286152-B6 (SK)
Title: Process for preparing acylphosphines, acylphosphine oxides and acylphosphine sulfides
Inventor: LEPPARD DAVID GEORGE
IPC: C07F9/50
Filed: 1999-11-20
Abstract: The invention relates to a process for the preparation of bisacylphosphines of formula (I), wherein n is 1 or 2, by reacting (a) organic phosphorus halides of formula (II), wherein n is 1 or 2 and Y is Br or Cl, with an alkali metal or with magnesium in combination with lithium, or with mixtures thereof, optionally in the presence of a catalyst, and (b) subsequent reaction with an acid halide of formula (III), which process is carried out without isolation of the intermediates. Also disclosed is a process for the preparation of bisacylphosphine oxides and bisacylphosphine sulfides of formula (IV), wherein n is 1 or 2 and Z is O or S, by oxidation or reaction with sulfur of bisacylphosphine of formula (I). Bisacylphosphine oxides or bisacylphosphine sulfides so obtained find application as initiators in the photopolymerisation of unsaturated compounds.
Patent CZ-302588-B6 (CZ)
Title: Use of N-substituted indole-3-gloxylamide for preparing a medicament
Inventor: NICKEL BERND
IPC: A61K31/404
Filed: 1999-03-22
Abstract: The present invention relates to the use of N-substituted indole-3-gloxylamides of the general formula 1 or a pharmaceutically acceptable acid addition salts or N-oxides thereof for the preparation of a medicament intended for treating oncologic diseases such as leukemia, prostate cancer, ovarial carcinoma and epidermal carcinoma.
Patent CZ-296963-B6 (CZ)
Title: Process for producing multi-layered molded synthetic part and molded synthetic part obtained in such a manner
Inventor: DE WINTER HUGO
IPC: B29C43/20
Filed: 1999-10-15
Abstract: The present invention relates to a process for producing a multi-layered molded synthetic part comprising at least a preformed polyurethane elastomeric skin (5) and a molded carrier (8). In this process, the polyurethane elastomeric skin (5) is molded in a first step and the thermoplastic material for the carrier (8) is subsequently molded in molten state to the back of said molded skin (5). According to the invention, the molded skin is made of a thermosetting synthetic material. Described is also a multi-layered molded synthetic part produced in the above-indicated manner.
Patent CZ-302315-B6 (CZ)
Title: Process and apparatus for protecting railway bed when working on adjacent track
Inventor: MALY VACLAV
IPC: E01B27/00
Filed: 2003-12-03
Abstract: This invention solves a problem of protecting a railway bed when working on adjacent track by using an arresting element (1), which is spread to a prepared plain of railway superstructure or first construction layer of railway bed gravel and new railway bed gravel is arranged on a part of this way spread arresting element (1). The arresting element (1) is bent and new railway bed gravel is packed with the arresting element (1), which is then fitted to a working rail. The arresting element (1) is made of a strip of bendable material, for example steel wire lattice or geogrid and it is provided with grips (2) at both its longitudinal edges. A bracing element (4) is provided to the grips (2) of the arresting element (1) parallel to the rail, whereas the arresting element (1) is fitted to this rail. There is also provided an adjusting element (3) for stretching and tightening the arresting element (1), which contains gravel of the gravel bed, whereas the adjusting element (3) has to be placed between the grips (2) of the arresting element (1) or between the bracing element (4) and the rail, in which rail the arresting element (1) is fitted.
Patent SK-283833-B6 (SK)
Title: Benzothiadiazoles and derivatives
Inventor: NEUMANN BERNHARD PETER
IPC: A61K31/437
Filed: 1999-02-01
Abstract: The invention provides a compound of formula (I) wherein X, R1, R2 and Het are as defined in the description, and a process for preparing them. The compounds of formula (I) are useful as pharmaceuticals.
Patent SK-285285-B6 (SK)
Title: Cream and deodorant dispenser
Inventor: HOLTHAUS ULRIKE
IPC: A45D40/00
Filed: 2000-04-14
Abstract: The invention relates to a dispenser-type packaging (1) for a cream or other substance that is applied by stroking a surface, comprising a chamber (5) with a discharge opening (10), for holding and storing the sub-stance, a spindle (15) that is arranged in the chamber (5) in a longitudinal axial direction, in such a way that it can rotate, a plunger (18) which can be moved along the spindle (15) in the chamber (5), a toothed wheel (16) which is located outside the chamber (5) and is rotationally fixed to the spindle (15), and at least one activating button (4) which is located on the dispenser packaging (1) and which has a moulded-on pusher element (23), the at least one activating button (4) with the pusher element (23) is arranged so that it can be moved from a rest position to an end position and back in relation to the toothed wheel (16), in such a way that when the activating button (4) is activated and caused to move from the rest position to the end position, the pusher element (23) engages with a tooth (26) of the toothed wheel (16) and turns the toothed wheel. The aim of the invention is to ensure that the plunger can move back in the opposite direction to the pusher-driven direction of rotation. To this end, the dispenser packaging (1) has at least one pusher deflector (32), on which the at least one pusher element (23) is stopped before reaching the end position and which deflects the pusher element from its engagement with the toothed wheel (16).
Patent SK-285320-B6 (SK)
Title: Process of preparation and purification of tramadol and tramadol hydrochloride
Inventor: GAZOVIC ANTON
IPC: C07C213/00
Filed: 2002-11-08
Abstract: Described is the process of preparation and purification of tramadol and tramadol hydrochloride, which can be used as an analgesic. Tramadol is prepared by reaction 3-methoxyphenylmagnesium halide with 2-dimethylaminomethylcyklohexanone in tetrahydrofurane,the developed complex is hydrolyzated and the blend of (RR,SS)-tramadol, (RS,SR)-tramadol, 6-olefin and/or 1-olefin is isolated, than is epimerizated at the present of organic acid and after that, the blend is alkalized and freed based are extracted in organic solvent and in such a way isolated tramadol is treated in a reaction with hydrogen chloride in the blend of ethanol and ether to (RR,SS)-tramadol hydrochloride.
Patent SK-288479-B6 (SK)
Title: Method for modification superconducting cable
Inventor: VOJENCIAK MICHAL
IPC: H02K3/42
Filed: 2010-11-08
Abstract: Solution relates to a method of modification of the superconducting cable, which consist in it, that above the spaces between superconducting strips (2) are positioned on the circumference of the ring of the molding member (3) in one layer placed ferromagnetic strips (4).
Patent BR-PI0317796-B8 (BR)
Title: análogos da 1-desamino-8-d-arginil vasopressina
Inventor: Daniel f alonso
IPC: A61K38/00
Filed: 2003-12-29
Abstract: análogos da 1-desamino-8-d-arginil vasopressina. mpa-tyr-phe-x-y-cys-pro-d-arg-gly-nh2 (i) 1. análogos da 1-desamino-8-d-arginil vasopressina com a seguinte fórmula geral mpa-tyr-phe-x-y-cys-pro-d-arg-glynh2 na qual, o x é um aminoácido de um grupo composto de alanina, asparagina, glutamina, isoleucina, leucina e valina; e y é um aminoácido de um grupo composto de asparagina, glutamina, isoleucina, leucina e valina. 2. análogos de 1-desamino-8-d-arginil vasopressina, de acordo com a reivindicação 1, com a seguinte fórmula geral (i): na qual x é um aminoácido de um grupo composto de alanina, asparagina, glutamina, isoleucina, leucina e valina; e é um aminoácido de um grupo composto de asparagina, glutamina, isoleucina, leucina e valina.
Patent EP-1603052-B8 (EP)
Inventor: SCHNURR JEFFREY R
IPC: G06F17/00
Filed: 2004-06-02
Granted: 2008-09-10
Abstract: A representation of a spreadsheet is displayed on a mobile communication device after receiving a description of a spreadsheet. The description relates to a plurality of map cells, where each map cell corresponds to a cell block, and the description includes location information and primary data type information for each map cell. Based on the location and content-type information in the description, a pictorial representation of the spreadsheet may be generated and displayed to a user of the mobile communication device. A mobile device server may not only generate the description, but also may interpret the user's selection of a region of interest and transmit enough information about the region of interest for the mobile communication device to present the region of interest to the user in a conventional viewer. <IMAGE>
Patent EP-1843507-B8 (EP)
Inventor: COOPERMAN MARC S
IPC: H04N21/8352
Filed: 1996-06-07
Granted: 2015-09-09
Abstract: An apparatus and method for encoding and decoding additional information into a steam of digitized samples in an integral manner. The information is encoded using special keys. The information is contained in the samples, not prepended or appended to the sample stream. The method makes it extremely difficult to find the information in the samples if the proper keys are not possessed by the decoder. The method does not cause a significant degradation to the sample stream. The method is used to establish ownership of copyrighted digital multimedia content and provide a disincentive to piracy of such material.
Patent BR-PI0107598-B8 (BR)
Inventor: ESBJÖRN ERIKSSON
IPC: H01G4/015
Filed: 2001-01-11
Abstract: A capacitor element (20) for a power capacitor with a dielectric film layer (3) and an electrode layer arranged on each flat side of the film layer, which electrode layers are divided into at least three metallized areas (4, 9, 10), separated from each other, in order to form an inner series connection arranged to conduct a load current, of which three areas at least one is divided into segments (5) separated by non-metallized sections (6), and at least one bridge (7) arranged to electrically connect two of the segments together. In accordance with the invention the bridge is so arranged that, in the area divided into segments, the load current appears substantially only in the segments. The invention also relates to a power capacitor with such a capacitor element and also a metallized tape for such a power capacitor.
Patent BR-PI0210085-B8 (BR)
Inventor: ALPA PARIKH
IPC: A61K47/36
Filed: 2002-05-24
Abstract: The present invention is related to compositions of modafinil, including compositions of modafinil and one or more diluents, disintegrants, binders and lubricants, and the processes for their preparation thereof.
Patent BR-PI0520406-B8 (BR)
Inventor: CRAIG A ZIFICSAK
IPC: C07D233/54
Filed: 2005-06-29
Abstract: The invention relates to methods of synthesizing 2-substituted azole compunds of formula (I). The invention is also relates to compounds of formula (I) and to intermediate compounds in the synthesis method.
Patent BR-PI0721393-B8 (BR)
Title: método para obter lipídeo a monofosforilado da bordetella pertussis como um subproduto da produção de vacina celular contra coqueluche
Inventor: ISAIAS RAW
IPC: C07H13/06
Filed: 2007-03-22
Abstract: MÉTODO PARA OBTER LIPÍDEO A MONOFOSFORILADO DA BORDETELLA PERTUSSIS COMO UM SUBPRODUTO DA PRODUÇÃO DE VACINA CELULAR CONTRA COQUELUCHE, mais especificamente, um método de purificação de BpMPLA a partir do processamento de um extrato alcoólico geralmente rejeitado ou filtrado da coleta inativada da vacina de Bordetella pertussis (subproduto da produção de vacina principal, método de purificação de BpMPLA este que compreende o processamento de um extrato alcoólico geralmente rejeitado da coleta inativada de Bordetella pertussis, a submissão deste extrato final a uma coluna de afinidade e o envio da fração eluída de detergente à hidrólise ácida seguida por neutralização, liofilização e ressuspensão com água para injeção acrescida de detergente suave; o novo BpMPLA é usado em aplicações imunoestimuladoras, mais especificamente, como um adjuvante de vacina e, ainda mais especificamente, como um adjuvante de vacina contra gripe, com resultados promissores.
Patent BR-PI1015568-B8 (BR)
Title: derivados de imidazolidin-2-ona 1,3-dissubstituídos como inibidores de cyp 17, seus usos, e composição farmacêutica
Inventor: CHRISTOPH GAUL
IPC: C07D407/14
Filed: 2010-06-24
Abstract: derivados de imidazolidin-2-ona 1,3-dis-substituídos, composição farmacêutica, seus usos, bem como combinação compreendendo os referidos derivados. a presente invenção se refere a compostos de fórmulas (i) e (i-i), ou um sal farmaceuticamente aceitável do mesmo, onde r53, r54, p, q e n são conforme aqui definido. os compostos da presente invenção foram constatados ser úteis como inibidores de 17(alfa)-hidroxilase/c17, 20-liase.
Patent AU-2018287971-B8 (AU)
Title: 7-site substituted pyrrole triazine compounds or pharmaceutically acceptable salts thereof, and preparation method therefor and uses thereof
Inventor: YANG CHUNHAO
IPC: A61K31/5377
Filed: 2018-06-22
Granted: 2021-02-04
Abstract: The present invention relates to 7-site substituted pyrrole [2,1-f][1,2,4] triazine compounds or pharmaceutically acceptable salts thereof, and a preparation method therefor and uses thereof. This kind of compound shows good PI3K inhibition activity, can effectively inhibit the activity of the PI3K kinase; and due to the introduction of 7-site groups, bioavailability and other pharmacokinetic properties have been greatly improved. In addition, the compounds in the present invention show an unpredictable high selectivity and strong inhibitory activity on PI3kδ, accordingly, the compounds can be used to treat diseases associated with PI3K pathways, especially for resisting against cancers or treatment of tumors, leukemia and autoimmune diseases. After further optimization and screening, the compounds are expected to develop into new antitumor drugs.
Patent BR-112014000665-B8 (BR)
Title: composto, composição farmacêutica, agente antimicrobiano, e, uso de um composto
Inventor: DAISUKE OKA
IPC: A61K31/47
Filed: 2012-08-30
Abstract: composto, composição farmacêutica, agente antimicrobiano, e, uso de um composto a presente invenção fornece um composto representado pela fórmula (i) em que x é um átomo de hidrogênio ou um átomo de flúor; r é um átomo de hidrogênio ou alquila; r1 é (1) ciclopropila opcionalmente substituído por 1 a 3 átomos de halogênio ou (2) fenila opcionalmente substituído por 1 a 3 átomos de halogênio; r2 é alquila, alcóxi, haloalcóxi, um átomo de halogênio, ciano, etc.; e r3 é 7-oxo-7,8-diidro-1,8-naftiridinila, 3- piridila, etc., ou um sal do mesmo. o composto da presente invenção tem atividade antimicrobiana excelente contra clostridium difficile e é útil para a prevenção ou tratamento da infecção intestinal tal como diarreia associada à clostridium difficile.