baber/WOPTO huggingface dataset:
Patent LV-12569-A (LV)
Title: Epothilone derivatives
Inventor: VITE GREGORY D
IPC: C07D493/04
Filed: 2000-02-02
Abstract: The present invention relates to compounds of formula (I), Q is selected from the group consisting of (II), G is selected from the group consisting of alkyl, substituted alkyl, substituted or or unsubstituted aryl, heterocyclo, (III), W is O or NR15; X is O or H,H; Y is selected from the group consisting of O; H, OR16; OR17, OR17; NOR18; H, NOR19; H, NR20R21; H, H; or CHR22; OR17OR17 can be a cyclic ketal; Z1 and Z2 are selected from the group consisting of CH2, O, NR23, S or SO2, wherein only one of Z and Z2 is a heteroatom; B1 and B2 are selected from the group consisting of OR24, or OCOR25, or 2CNR26R27; when B1 is H and Y is OH, H they can form a six-membered ring ketal or acetal; D is selected from the group consisting of NR28R29, NR30COR31 or saturated heterocycle R1, R2, R3, R4, R5, R6, R7, R13, R14, R18, R19, R20, R21, R22, R26 and R27 are selected from the group H, alkyl, substituted alkyl, or aryl and when R1 and R2 are alkyl can be joined to form a cycloalkyl; R3 and R4 are alkyl can be joined to form a cycloalkyl; R9, R10, R16, R17, R24, R25, and R31 are selected from the group H, alkyl, or substituted alkyl; R8, R11, R12, R28, R30, R32, R33, and R30 are selected from the group consisting of H, alkyl, substituted alkyl, aryl, substituted aryl, cycloalkyl, or heterocyclo; R15, R23 and R29 are selected from the group consisting of H, alkyl, substituted alkyl, aryl, substituted aryl, cycloalkyl, heterocyclo, R32 C=O, R33 SO2, hydroxy, O-alkyl or O-substituted alkyl, the pharmaceutically acceptable salts thereof and any hydrates, solvates or geometric, optical and stereoisomers thereof, with the proviso that compounds wherein: W and X are both O; and R1, R2, R7 are H; and R3, R4, R6, are methyl; and R8, is H or methyl; and Z1, and Z2, are CH2; and G is 1-methyl-2-(substituted-4-thiazolyl)ethenyl; and Q is as defined above are excluded.
Patent LV-12559-A (LV)
Title: Derivatives of 1,3,4-oxadiazolone
Inventor: HEWAWASAM PIYASENA
IPC: A61P25/08
Filed: 2000-08-03
Abstract: The present invention provides novel oxadiazolone derivatives having general formula (I), wherein A, B, D and R are as defined herein, or a nontoxic pharmaceutically acceptable salt or solvate thereof and are useful in the treatment of disorders which are responsive to the opening of the large conductance calcium-activated potassium channels.
Patent LV-12591-A (LV)
Inventor: RASA ZIGURDS
IPC: C02F3/02
Filed: 1999-05-31
Abstract: The present invention concerns the field of biologically treatment of waste-water. It gives an opportunity to decrease the expenditure of electric energy used by power consumers in sewage treatment plant. Biologically sewage treatment plant contains several series-connected basins - aeration-basin, basin for water enriching with oxygen and basin for bio-filtration using higher aquatic plants. The above-mentioned effect in the sewage treatment plant is achieved by location of turbine, connected mechanically with generator, inside the air-supply pipe in aeration-basin. The generator is electrically connected with compressor or with other power consumers.
Patent ME-P28108-A (ME)
Title: Substituted beta-carbolines with ikb-kinase inhibiting activity
Inventor: RITZELER OLAF
IPC: A61P31/04
Filed: 2001-02-28
Abstract: The subject matter of the present invention is directed to novel substituted beta-carbolines, and specifically compounds of the formula I, which are suitable for the production of pharmaceuticals for the prophylaxis and therapy of disorders in whose course an increased activity of IkappaB kinase is involved.
Patent TR-25500-A (TR)
IPC: D06F39/02
Filed: 1991-11-26
Abstract: PCT No. PCT/US91/08824 Sec. 371 Date May 25, 1993 Sec. 102(e) Date May 25, 1993 PCT Filed Nov. 25, 1991 PCT Pub. No. WO92/09737 PCT Pub. Date Jun. 11, 1992.The equipment comprises a measuring and dispensing device of the reusable type for the machine washing of clothes, which comprises a hollow body (1) intended to receive the amount of liquid detergent prescribed for the wash, said body being provided with at least one filling opening (3) and outlets (7b) for the distribution of said product or products, as well as means (8) enabling the user to effect, once said device has been filled, the easy and controlled application of at least one product contained in it to selected areas of the clothing before the latter is subjected to washing in the machine, for the purpose of effecting the pretreatment of said areas before the washing cycle, said measuring and dispensing device, containing the amount of product remaining after the pretreatment, being introduced into the machine together with the clothes, said pretreatment means (8) being removable from the body of said device.
Patent YU-88903-A (YU)
Title: Hotwater boiler for open and closed heating systems for houses, appartments and offices
Inventor: JANIC RADOJKO
Filed: 2003-11-10
Abstract: Hotwater boiler for open and closed heating systems for houses, appartments and offices with burning the solid or gaseous fuelf from the bottom, according to the invention has a back side (1) and part of the ceiling (2) of a fire-box (3) achieved by bending the boiler sheet as a double wall body with a cavity through which water flows, while the lower wall of the ceiling (2) is achieved as a shallow transversal prismatic recess (2A), while the part of the ceiling (2) is achieved as a downward directed shallow boxlike converter (2B), while in the bottom part of the fire-boxt (3) is set a wirenetting grate (6) and that from the bottom side is set a fireproof walling (8) of thermostoring bricks, while behind the other boxlike converter (7) in the bottom part of the rear part of the fire-box (3) area is set the third boxlike converter (9). Between the upper part of the boxlike converter (9) and the top of the prsmatic recess (2A) is set a regulatory flap (10) for regulation of the blow, and beside a fume gas drain-pipe (11) on the back side of the boiler, on the lateral sides are intended for circular outlets (112) for connecting to the chimney either from one or the other lateral sides and in that from the circular outlets (112) from the bottom there are circular outlets (12) for cleaning and check. Hotwater boiler, according to the invention, has another emodiment solution with different arrangement of boxlike converters. This, so called flat boiler has a door of the fire box in the front side of the boiler.
Patent AU-1115699-A (AU)
Title: Real-time interactive directory
Inventor: PICKERING RICHARD B
IPC: H04W4/16
Filed: 1998-10-22
Abstract: An interactive directory provided for a workstation having a connected video monitor and adapted for network access has an interactive display for displaying status for individual entities, being persons and organizations. Entities are listed in the display along with status for each entity. There may be multiple fields for status, and some fields display telephone numbers and/or IP addresses for Internet telephones, while others may provide alphanumeric display. A remote access contact address is stored and associated with each directory entity, and when the directory is active, the workstation accesses status information from network sources associated with individual directory listings. Status for entities in the directory is therefore updated in real time as the directory is used. In some embodiments multiple graphic indicia, such as underlining, shading, font choice and the like are used to provide status indication in various fields of the interactive display. In some embodiments alpha-numeric status is provided as well. In other embodiments telephone calls, including Internet telephone calls, may be placed by interactive input to the directory.
Patent AU-1339499-A (AU)
Title: A method for modifying the channel impulse response in tdma systems
Inventor: HAPPONEN AKI
IPC: H04L27/01
Filed: 1998-11-18
Abstract: The present invention proposes a device for processing received signals (y) having been transmitted via a transmission channel (1), comprising: estimation means (2, 2a) adapted to obtain an estimated impulse response function (hk) of said channel (1) based on said received signals (y) which are received at a first time; derivation means (3; 3a-3f) adapted to derive history information (wink) based on at least one previously estimated impulse response function, calculation means (4; 4a, 4b) adapted to calculate modifying information (mwink) on the basis of said history information (wink), and modification means (5) adapted to modify said estimated impulse response function (hk) of said channel (1) obtained on the basis of said received signals (y), by applying said modifying information (mwink) to said estimated impulse response function (hk) of said channel obtained on the basis of said received signals (y), and adapted to output a modified impulse response function (hmk). The present invention also proposes a corresponding method.
Patent AU-1397101-A (AU)
Title: Intermediate coin storage with translational movement for public telephones
Inventor: GOMEZ DAMASO MARTIN
IPC: G07F1/04
Filed: 2000-11-07
Abstract: The deposit comprises a number of disc-shaped elements or partitions (2) arranged parallel to each other to form a fully open cylindrical body (1) with its longitudinal axis horizontal, so that the partitions or elements (2) define slots (3) for the coins (4) which arrive from the validator/selector (5), and with said coins (4) resting on a false floor (6) which envelopes a certain angle of the bottom perimeter of the deposit formed by the cylindrical body (1). This false floor (6) is provided with a groove (8) so that when said floor turns in one sense a coin (4) will fall towards the collection hopper, while when the floor (6) turns in the opposite sense all the remaining coins will fall towards the return hopper. <IMAGE>
Patent AU-1512888-A (AU)
Title: Non-contact determination of the position of a rectilinear feature of an article
Inventor: MORRISON BRUCE ROBERT
IPC: G01B11/24
Filed: 1987-04-22
Abstract: A high resolution CCD video camera (6) is positioned and aligned with respect to an illuminated article (7) so that a straight edge of the article, or a straight line junction between a bright zone and a dark zone of its surface, crosses the field of view of the camera in a direction substantially parallel to the rows of the camera's orthogonal array of rows and columns of light responsive elements,to divide that field of view into bright and dark zones. A frame store and digitiser (9) converts the individual signals generated by the elements into digital grey values. The grey values derived from the elements of each row are summed by a computer (10) to produce a linear array of summation values positionally related to the respective columns, and the computer then determines the position of the edge or junction to a sub-column spacing accuracy by determining the mean value of two of the summation values selected respectively from a row receiving energy from the bright zone and one receiving energy from the dark zone and establishing a position in the array for the mean value, and thus for the feature, by interpolating the mean value between the two summation values immediately above and below it in magnitude.
Patent AU-1548500-A (AU)
Title: Automatic height adjustment system for flails with toppers for root crop harvesters
Inventor: HOLMER ALFONS
IPC: A01D23/02
Filed: 1999-10-20
Abstract: The invention relates to an automatic height adjustment system for flails with toppers (11) for use in harvesters harvesting several rows of root crops. Said system is embodied in such a way that a scanning device (12) associated with the flail (1, 2, 3) impinges upon the shaft (2) or the housing (1) of the flail in such a way that the vertical movement carried out by the scanning device is transmitted proportionally to the housing or the shaft of the flail and a conventional support wheel arrangement is no longer needed. The scanned surface on the root crop is used to regulate both the cutting blade of the topper (13) and the flail.
Patent AU-1627988-A (AU)
Title: Process for recovering purified, oxidized, renatured recombinant interleukin-2 from microorganisms
Inventor: WOLFE SIDNEY N
IPC: C07K1/30
Filed: 1988-03-31
Abstract: A process for recovering highly pure, recombinant IL-2 from transformed microorganisms in which the cells are disrupted; impure recombinant IL-2 is isolated in the form of refractile bodies from the disruptate; the impure IL-2 is dissolved and denatured with at least 6 M guanidine hydrochloride containing a reducing agent; the reduced IL-2 is precipitated and resolubilized; the reduced solubilized IL-2 therein is oxidized by a controlled oxidation in which the concentration of guanidine hydrochloride is maintained at least at 6 M; the oxidized IL-2 is refolded by reducing the concentration of guanidine hydrochloride in the solution; and the oxidized, refolded IL-2 is further purified by ion exchange chromatography or hydrophobic interaction chromatography and ion exchange chromatography.
Patent AU-1686100-A (AU)
Title: Portable electronic device, method of controlling the device and recording medium for recording data used by the device
Inventor: KUTARAGI KEN
IPC: A63F13/28
Filed: 1999-12-15
Abstract: A portable electronic device that can be connected to a host machine and can be used alone as an ancillary machine to be used as a remote control unit, and allowing even visually impaired users to distinguish remote control operation information aurally is configured so that a remote control program and frequency division program are downloaded from a CD-ROM which is the recording medium to a program memory of the portable electronic device, and remote control voice data is also downloaded to a non-volatile memory of the device. Additionally, remote control voice data corresponding to operation items when the portable electronic device is used as a remote control unit undergoes frequency division, and sounds which allow the operation items to be distinguished, are generated from a speaker of the portable electronic device.
Patent AU-1878192-A (AU)
Title: Safety syringe with automatically retractable hollow needle
IPC: A61M5/50
Filed: 1992-05-29
Abstract: A syringe fitted with a clamping device for the needle and with means to enable the needle to be automatically retractable into the syringe body at the end of an injection comprises: outer and inner cylinders; openings at the ends of the outer cylinder; a third opening at an end of said inner cylinder; closing means for said third opening; a needle with a head; sealing means in said closing means; a first spring to push said needle against said closing means; a clamping device loaded by a second spring to maintain outward said syringe and to release said needle; a diaphragm in said closing means which bends before its breaking; a sharp element to break said diaphragm; closing means to prevent said needle from being reached and stopping means to prevent said second cylinder from being moved outward said syringe after its use.
Patent AU-1998583-A (AU)
Title: Pharmaceutical compositions of mopidamol
Inventor: SCHEPKY GOTTFRIED
IPC: A61K9/20
Filed: 1983-10-07
Abstract: This invention relates to vehicles for the administration of mopidamol. More specifically, this invention relates to a method of treating cardiovascular disorders, malignancy, or thrombosis in a host in need of such treatment which comprises administering to said host a cardiovascularly, antimetastic, or antithrombotic effective amount of a composition comprised of (i) mopidamol or an acid addition salt thereof and (ii) at least one pharmacologically acceptable acid or acid substance, the total amount of acid from acid addition salt present and acid or acid substance being in a ratio of at least about 1 acid equivalent to 1 mol of mopidamol or its acid addition salt.
Patent AU-2018188-A (AU)
Title: Spray head for the administration of a multi-component material by means of gas
Inventor: ZIMMERMANN JOSEF
IPC: A61M11/06
Filed: 1988-07-29
Abstract: In the spray head for the administration of a multi-component material by means of gas, a gas channel (2) with gas connection (3) is provided, which channel is divided by a separating web (4) into a plurality of channels (2a+B, 2b) running parallel to the separating web. Into these channels there open out boreholes (5, 5a) for receiving cannulas. The open ends of the boreholes (5, 5a) go into grooves (7, 7a) which serve for guiding the cannulas (6, 6a). The grooves are arranged parallel to the gas channel (2). The separating web (4) protrudes beyond the channel ends (9, 9a).
Patent AU-2163592-A (AU)
Title: A novel receptor-type tyrosine kinase and use thereof
IPC: A61K38/45
Filed: 1992-06-19
Abstract: The present invention relates to a method of screening for ligands to a receptor-type tyrosine kinase. The receptor-type tyrosine, in its naturally occurring form, is characterized by being reactive to monoclonal antibody III.A4, having an apparent molecular weight of approximately 120-150 kD in its glycosylated form, and having the N-terminal amino acid sequence E L I P Q P.
Patent AU-2246983-A (AU)
Title: Optically active araliphatic 2-(4(subst.ph/pyr)oxyphenoxy)proprionates
Inventor: MORIYA KOICHI
IPC: A01N43/40
Filed: 1983-12-16
Abstract: New dextrorotatory enantiomers of phenoxy propionic acid derivatives of the formula    <IMAGE>  (I)  in which R1 represents a radical of the formula   <IMAGE>  wherein X1 represents hydrogen or halogen, X2 represents halogen or trifluoromethyl, X3 represents halogen or trifluoromethyl, X4 represents hydrogen or halogen and X5 represents hydrogen or halogen, Y represents oxygen or the radical SOm, wherein m represents 0, 1 or 2, R2 represents hydrogen or methyl, n represents 1 or 2 and R3 and R4 independently of one another represent hydrogen, halogen, alkyl with 1 to 4 carbon atoms, alkoxy with 1 to 4 carbon atoms, alkylthio with 1 to 4 carbon atoms, nitro, cyano or alkoxycarbonyl with 1 to 4 carbon atoms in the alkoxy group, and their use as herbicides.
Patent AU-2262695-A (AU)
Title: Hybrid electricity and telecommunications distribution network
Inventor: BROWN PAUL ANTHONY
IPC: H04M3/00
Filed: 1995-04-20
Abstract: A telecommunications network is disclosed for linking a plurality of premises, comprising, typically, a fibre optic or coaxial cable (130), and a plurality of electrical power cables (134) each connected to a respective one of the premises for supplying mains electrical power thereto. Each of the power cables (134) is also connected to the fibre optic or coaxial cable (130) so that telecommunications signals are transmissible between the fibre optic or coaxial cable and each of the power cables. A telecommunications signal is transmissible to the plurality of premises by being transmitted along the fibre optic or coaxial cable and subsequently along the respective power cable of each of the premises.
Patent AU-2406102-A (AU)
Title: Relay device
Inventor: YABE TOSHIYASU
IPC: H04W40/34
Filed: 2001-11-21
Abstract: When a gateway server GWS receives an access demand to an IP server from a cellular phone MS via a mobile packet communication network MPN, the gateway server acquires information corresponding to a hostname included in the access demand from a primary conversion table T 1 . When the obtained information is a wide area IP address, gateway server GWS relays the access demand to a IP server on the Internet INET on the basis of the wide area IP address. When the obtained information is identification of a closed area network, gateway server GWS further acquires a closed area IP address corresponding to the hostname included in the access demand and relays the access demand to a IP server on the basis of the closed area IP address in the LAN corresponding to the identification of the closed area network.
Patent AU-2492500-A (AU)
Title: Aspartic protease inhibitors, compositions, and associated therapeutic methods
Inventor: RANDAD RAMNARAYAN S
IPC: C07D207/27
Filed: 2000-01-06
Abstract: The present invention provides an aspartic proteinase-inhibiting compound of the formula: wherein a, b, c, d, and e, can be the same or different and each are R<SUP>7</SUP>, OR<SUP>7</SUP>, SR<SUP>7</SUP>, NR<SUP>7</SUP>R<SUP>8</SUP>, NHCOR<SUP>7</SUP>, CO<SUB>2</SUB>R<SUP>7</SUP>, CN, NO<SUB>2</SUB>, NH<SUB>2</SUB>, N<SUB>3</SUB>, or a halogen, wherein R<SUP>7 </SUP>and R<SUP>8 </SUP>are independently H or an alkyl. Substituents R<SUP>1 </SUP>or R<SUP>2 </SUP>are each H or an alkyl. Substituent R<SUP>3 </SUP>is a straight chain or branched alkyl, alkenyl, or alkynyl substituent, or is a cycloalkyl. Substituent A is OH, NH<SUB>2</SUB>, or SH. Further provided are pharmaceutical compositions, which include a therapeutically effective amount of at least one of the foregoing compounds, and therapeutic methods of using the foregoing compounds.
Patent AU-2512488-A (AU)
Title: Public key/signature cryptosystem with enhanced digital signature certification
Inventor: FISCHER ADDISON M
IPC: G06Q20/38
Filed: 1988-11-15
Abstract: A public key cryptographic system is disclosed with enhanced digital signature certification which authenticates the identity of the public key holder. A hierarchy of nested certifications and signatures are employed which indicate the authority and responsibility levels of the individual whose signature is being certified. The present invention enhances the capabilities of public key cryptography so that it may be employed in a wider variety of business transactions, even those where two parties may be virtually unknown to each other. Counter-signature and joint-signature requirements are referenced in each digital certification to permit business transactions to take place electronically, which heretofore often only would take place after at least one party physically winds his way through a corporate bureaucracy. The certifier in constructing a certificate generates a special message that includes fields identifying the public key which is being certified, and the name of the certifiee. In addition, the certificate constructed by the certifier includes the authority which is being granted including information which reflects issues of concern to the certifier such as, for example, the monetary limit for the certifiee and the level of trust which is granted to the certifiee. The certificate may also specify cosignature requirements which are being imposed upon the certifiee.
Patent AU-2567995-A (AU)
Title: Medicament chamber in an inhalation apparatus
Inventor: LANKINEN TAPIO
IPC: A61J1/05
Filed: 1995-05-26
Abstract: PCT No. PCT/FI95/00291 Sec. 371 Date Nov. 25, 1997 Sec. 102(e) Date Nov. 25, 1997 PCT Filed May 26, 1995 PCT Pub. No. WO95/32752 PCT Pub. Date Dec. 7, 1995The invention relates to a medicament chamber (6) included in an inhalation apparatus and provided with a container (2) containing a desiccant. The chamber (6) is tightly sealed and has a moisture permeability as poor as possible, and the container (2) is permeable to moisture.
Patent AU-2595699-A (AU)
Title: Chelated 8-hydroxyquinoline for the treatment of epithelial lesions
Inventor: JORDAN RUSSEL T
IPC: A61K33/24
Filed: 1999-02-10
Abstract: A chelation complex including 8-hydroxyquinoline and zinc mixed with a carrier demonstrates therapeutic efficacy in treating lesions including cancerous lesions, precancerous lesions, cysts and warts.
Patent AU-2610588-A (AU)
Title: Dna encoding ige receptor alpha-subunit or fragment thereof
Inventor: SIRAGANIAN REUBEN
IPC: C12Q1/6876
Filed: 1988-11-29
Abstract: A cDNA sequence (I) encoding the alpha-subunit of human mast cell IgE surface receptor (II) or its IgE binding fragment is new. Also claimed is a vector contg. (I), a sol. fragment of the alpha -subunit of (II), the fragment being capable of binding to human IgE, and recombinant alpha-subunit of (II).