baber/WOPTO huggingface dataset:
Patent HU-T67959-A (HU)
Title: Corticosteroid-17-alkyl-carbonate-21-[o]-carboxylic-and carbonate esters, process for producing them and pharmaceutical compositions containing them
Inventor: DUERCKHEIMER WALTER
IPC: A61P29/00
Filed: 1994-08-25
Abstract: There are described 17-alkyl carbonate-21-carbonic/carboxylic acid esters of corticosteroids of the formula I <IMAGE> where A is CHOH or CHCl, CH2, C = O, a 9(11) double bond; Y is H, F, Cl; Z is H, F, CH3; R(1) is aryl, hetaryl; n and m are zero or 1; R(2) is alkyl, -(CH2)2-OCH3; R(3) is H, methyl. They are obtained by reacting a compound of the formula II <IMAGE> in which R(5) is OH, with an activated carboxylic acid of the formula III  R(6)-CO-(O)n-[(C1-C4)-alkyl]m-R(1)      III The compounds I have very potent local and topical anti-inflammatory activity and show a very good ratio of local to systemic anti-inflammatory action, which is often clearly superior compared with analogous corticoid 17-alkyl carbonate 21-esters which do not carry an aryl or hetaryl group in the 21 ester radical.
Patent HU-T77133-A (HU)
Title: Aminoguanidine carboxylates for the treatment of non-insulin-dependent diabetes mellitus
Inventor: LARSEN SCOTT D
IPC: A61K31/198
Filed: 1995-11-13
Abstract: The present invention provides novel compounds of the formula I and II for the treatment of non-insulin dependent diabetes mellitius (NIDDM) and a new use of known compounds for this purpose.
Patent IL-71617-A (IL)
Title: 3-(amino-1-carboxylalkyl)amino-4-oxo-2,3,4,5-tetrahydro-1,5-benzothiazepine-5-acetic acid derivatives,method for producing them and pharmaceutical compositions containing them
IPC: C07C69/738
Filed: 1984-04-22
Abstract: Novel condensed, seven-membered ring compounds of formula:wherein R' and R<sup>2</sup> each represent hydrogen, halogen, trif- fluoromethyl, lower alkyl or alkoxy, or both jointly form tri-or imethylene; R' is hydrogen, lower alkyl or aralkyl; R<sup>4</sup> is alogen or alkyl, aralkyl or cyclo-alkytalkyl which may be stituted; X is a group represented by the formula S(O)n ere n is an integer of 0 to 2); Y is a carboxyl group which be esterified or amidated; m is 1 or 2) and salts thereof. These compounds exhibit inhibitory activity on angioten- converting enzyme and so forth, and are of value as an it for diagnosis, prevention and treatment of hypertension.
Patent IL-76915-A (IL)
Title: Prefabricated modules,and the use thereof in the building industry
IPC: E04C2/06
Filed: 1985-11-01
Abstract: There is described a prefabricated module comprising a three-dimensional armature formed by welded wires, and flat elements from light and/or heat-insulating material, retained on either side of the armature to form at least one continuous panel. One and the same module may be used either for bearing structures extending vertically, or for bearing structures extending horizontally, and having retaining means for the armatures.
Patent IL-87573-A (IL)
Title: Methyl-3-methoxy-2- phenylpropenoate derivatives, their preparation and fungicidal compositions comprising them
IPC: C07C69/734
Filed: 1988-08-26
Abstract: Fungicidal compounds of the formula (I) : <CHEM> and stereoisomers thereof, wherein K is oxygen or sulphur; Z is optionally substituted aryl or optionally substituted heteroaryl; X is O, S(O)n, NR<4>, CR<1>R<2>, CHR<5>, CO, CR<1>(OR<2>), C=CR<1>R<2>, CHR<1>CHR<2>, CR<1>=CR<2>, CHR<1>CR<2>=CH, C IDENTICAL C, OCHR<1>, CHR<1>O, OCHR<1>O, S(O)nCHR<1>, S(O)nCHR<1>O, CHR<1>S(O)n, CHR<1>OSO2, NR<4>CHR<1>, CHR<1>NR<4>, CO2, O2C, SO2O, OSO2, CO.CO, COCHR<1>, COCHR<1>O, CHR<1>CO, CHOH.CHR<1>, CHR<1>.CHOH, <CHEM> CONR<4>, OCONR<4>, NR<4>CO, CSNR<4>, OCS.NR<4>, SCO.NR<4>, NR<4>CO2, NR<4>CS, NR<4>CSO, NR<4>COS, NR<4>CONR<4>, S(O)nNR<4>, NR<4>S(O)n, CS2, S2C, CO.S, SCO, N=N, N=CR<1>, CR<1>=N, CHR<1>CHR<2>CH(OH), CHR<1>OCO, CHR<1>SCO, CHR<1>NR<4>CO, CHR<1>NR<4>COR<4>, CHR<1>CHR<2>CO, O.N=CR<1>, CHR<1>O.N=CR<2>, CO.OCR<1>R<2>, CHR<1>CHR<2>CHR<3>, OCHR<1>CHR<2>, (CH2)mO, CHR<1>OCHR<2>, CHR<1>CHR<2>O, OCHR<1>CHR<2>O, S(O)nCHR<1>CHR<2>, CHR<1>S(O)nCHR<2>, CHR<1>CHR<2>S(O)n, CR<1>=NNR<4>, NR<4>N=CR<1>, CHR<1>CONR<2>, CHR<1>OCO.NR<2>, CH=CHCH2O, COCHR<1>CHR<2>O or (R<5>)2P<+>CHR<2>Q<->; A, B and E, which may be the same or different, are H, hydroxy, halo, C1-4 alkyl, C1-4 alkoxy, C1-4 haloalkyl, C1-4 haloalkoxy, C1-4 alkylcarbonyl, C1-4 alkoxycarbonyl, phenoxy, nitro or cyano; R<1>, R<2> and R<3>, which may be the same or different, are H, C1-4 alkyl or phenyl; R<4> is H, C1-4 alkyl or COR<1>; R<5> is optionally substituted phenyl; Q<-> is a halide anion; n is 0, 1 or 2 and m is a 3, 4 or 5; except that when Z is unsubstituted phenyl and X and K are oxygen, A, B and E are not all hydrogen.
Patent IL-89865-A (IL)
Title: Use of variable region sequences of the t-cell receptor for detection and inhibition of autoimmune disease
IPC: C12Q1/68
Filed: 1989-04-06
Abstract: Polymorphic regions of the variable region gene of T-cell receptors can be identified as being associated with particular autoimmune diseases. By detecting the presence of the particular sequence in the host genome, particularly rearranged, or the T-cell receptor expression product, the propensity for the autoimmune disease may be diagnosed. In addition, antibodies or peptides related to the specific sequence may be prepared for use in prophylaxis and therapy.
Patent JP-S60156649-A (JP)
Title: Method for extracting aromatic amine
Inventor: ANDOU NAOKI
IPC: C07C209/86
Filed: 1984-01-25
Abstract: PURPOSE:To make it possible to extract an aromatic amine with improved phase separation and a high distribution ratio for the aromatic amine, by extracting the aromatic amine from an aqueous solution, etc. containing the aromatic amine with an extractant consisting essentially of tetrahydrofuran. CONSTITUTION:An extractant consisting essentially of tetrahydrofuran is added to an aqueous solution or aqueous suspension (extraction feed) containing an aromatic amine and preferably 5-50pts.wt. based on 100pts.wt. water in the extraction feed, NH3 and/or electrolyte present therein at 0.5-5 wtight ratio between the extractant and extraction feed to extract the aromatic amine at 10-100 deg.C, and the resultant aromatic amine is washed with an aqueous solution of an alkali metal hydroxide, etc. to reduce remarkably an ammonium halide in the extract, etc. The resultant extract can be distilled, etc. to separate the aimed aromatic amine, e.g. phenylenediamine, scarcely causing coloration, e.g. blackening, even on storing in air. EFFECT:The extractant can be easily recovered by distillation, scarcely forming heavy materials.
Patent JP-H11213830-A (JP)
Title: Electronic switch
Inventor: KITAMURA TSUNEHIRO
IPC: H01H47/32
Filed: 1998-01-22
Abstract: PROBLEM TO BE SOLVED: To eliminate the need for changing current-resistance capacity of a double-way thyristor to a large capacity, and to avoid the generation of rush current to the double-way thyristor in the case of a large load capacity. SOLUTION: An electronic switch for controlling power value to be applied to a load L using a two-way thyristor is prepared with a pair of relay contacts 16 which are connected in parallel with the two-way thyristor and a relay coil 15 for controlling opening and closing of the relay contacts 16. In cases where a current value of the two-way thyristor detected by a transformer 13 does not reach a predetermined value, the relay coil 15 controls the paired relay contacts 16 for opening, and in cases where the current value of the two- way thyristor detected by the transformer exceeds the predetermined current value, the relay coil 15 controls the relay contacts 16 for closing.
Patent JP-S58127923-A (JP)
Title: Photosensitive composition
Inventor: NAMIZONO JIYUNJI
IPC: G03F7/021
Filed: 1982-01-26
Abstract: PURPOSE:To obtain a photosensitive composition for a lithographic plate with high sensitivity, superior wear resistance and printing resistance by using a (co) polymer having specified repeating uits each having a diazonium salt group. CONSTITUTION:A (co)polymer having a photosensitive diazonium salt as repeating units represented by the formula[where R is (substituted) aldyl, (substituted) alkenyl, (substituted) aryl or (substituted) aralkyl, each of Z1 and Z2 is a univalent substituent, each of p and q is O or 1-4, and when it is >=2, the univalent substituents may be identical with or different from each other]is copolymerized with other copolymerizable monomer, and the resulting copolymer is applied to a support such as an Al plate to form a photosensitive material. The material is exposed, and by removing the unexposed part with an aqueous developer, a lithographic plate with high sensitivity, wear resistance and printing resistance is obtd.
Patent JP-S5395514-A (JP)
Title: Test system for subscriber line
Inventor: AKIYAMA NOBUYOSHI
IPC: H04M3/26
Filed: 1977-02-01
Abstract: PURPOSE:To enable the subscriber line test in spatial split type electronic communicating path and time sharing communicating path, by using the subscriber line test equipment the same as the case of electromagnetic communicating path, through the use of detour switch.
Patent JP-H07215922-A (JP)
Title: Optical resolution of 1-amino-2-indanols
Inventor: MATSUMOTO HIROO
IPC: C07C213/10
Filed: 1994-02-01
Abstract: PURPOSE:To carry out optical resolution of a 1-amino-2-indanol by separating an optically active 1-amino-2-indanole in the form of a new diastereomer salt using an optically active carboxylic acid which is abundantly and ecomomically available as a reagent for optical resolution. CONSTITUTION:Optical resolution of a 1-amino-2-indanol of formula (+ or -)-I or formula (+ or -)-II (R<1> to R<4> are H, an alkyl, an alkoxy, a halogen, cyano, nitro) is carried out by reacting the 1-amino-2-indanol with an optically active carboxylic acid of formula (+)-III or formula (-)-III as a reagent for optical resolution and separating the produced new diastereomer salt. For example, a compound of formula (-)-I can be obtained through a new diastereomer salt by optically resolving a compound of formula (+ or -)-I using a carboxylic acid of formula (+)-III. As the compound of formula (+ or -)-I, trans-1- amino-2-indanol or cis-1-amino-2-indanol is especially preferably used. This optically active 1-amino-2-indanol is useful as an intermediate for synthesis of agricultural and medical drugs.
Patent JP-2000215637-A (JP)
Title: Tape cartridge
Inventor: HASHIZUME KENJI
IPC: G11B23/087
Filed: 1999-01-19
Abstract: PROBLEM TO BE SOLVED: To avoid contact between coupling plates and a tape by providing the coupling plates toward the lower side from the right and left end portions of the main surface plate and forming a recess to the part facing the tape at the rear internal surface of both coupling plates. SOLUTION: A hub brake 8 consists of a main surface plate, a couple of brake pawls extending to the rear hub side from such main surface plate, coupling plates extending to the lower side from the right and left ends of the main surface plate, an arm extending to the front side from such coupling plates and a projection 85 provided at the end part of the arm. At the position facing the tape at the rear internal surface of the coupling plates, a chamfering part 87 is formed through tapering toward the rear external side and this part is formed as the recess, for example, as the stepped portion. When the tape 4 is guided to the front side with a pair of pins P, if the wound tape diameter is large, the tape 4 is located closer to the coupling part of the hub brake 8 but if the tape is in contact with the coupling plate, it never receives any damage owing to such recess.
Patent JP-S58127306-A (JP)
Title: Transporting apparatus for oil-filled electrical device
Inventor: HARADA AKIHIRO
IPC: H01F27/14
Filed: 1982-01-26
Abstract: PURPOSE:To lighten the restrictions on the transport path and improve the reliability against the breakage or other accidents of a nonpermeable bag member during transport, by disposing the nonpermeable bag member outside an outer casing. CONSTITUTION:A vent pipe 9 provides a communication between an opening 601 of a nonpermeable bag member 6 and an outer casing 1. A protecting container 10, which is mounted on a truck 2 to house the nonpermeable bag member 6, is constituted by a protecting cover which covers the nonpermeable bag member 6 from the upper side and  is allowed to communicate with the outside air through a hygroscopic respirator 8. According to such a constitution, since the nonpermeable bag member 6 is disposed outside the outer casing 1, the height of the outer casing 1 can be reduced, so that the restrictions on transport can be lightened. In addition, it becomes possible to design and manufacture an oil- filled electrical device body 4 effectively utilizing the transport  limitations to the maximum. Moreover, it becomes unnecessary to clean the nonpermeable bag member 6 as well as protect the oil-filled electrical device 4 and the nonpermeable bag member 6. Furthermore, there is no need of any operation for taking out the nonpermeable bag member 6 from the outer casing 1, so that the operation is facilitated.
Patent JP-H02190039-A (JP)
Title: Line connection method for decentralized radio system
Inventor: FURUYA YUKITSUNA
IPC: H04M1/72511
Filed: 1989-01-18
Abstract: PURPOSE:To evade the interference at the time of introducing a system and to secure a channel at the time of congesting the system by increasing a threshold level when no idle channel is found out by a carrier sense and decreasing the threshold level when the idle channel is found out. CONSTITUTION:A signal received from an antenna 100 is inputted to a mixer 11 via a hybrid 20, multiplied with a carrier signal from a synthesizer 16 and the result is converted into an IF signal. After the IF signal is converted into a signal level of a power detector 12, the result is compared with a threshold level stored in a threshold level memory 14 at a comparator circuit 13. Based on the result, a microprocessor 15 changes the frequency of the synthesizer 16 or revises the threshold level of the threshold level memory. When the system is out congested, a low threshold level is selected and when the system is congested, a high threshold level is selected. Thus, the interference at system introduction is avoided and the call loss at line congestion is evaded.
Patent JP-S55101883-A (JP)
Title: Timer mechanism
Inventor: NAKANISHI RIYUUSUKE
IPC: F16H37/06
Filed: 1979-01-31
Abstract: PURPOSE: To provide a timer mechanism with good operating property that enables to cut power transmission by either positive or negative setting of timer operation time and having clutch that can be reset to the state of power transmission after completion of setting.  
     CONSTITUTION: Elastic clutch wheel 1 having outer tooth 8 is mounted into engaging portion 21 of spindle 12. Plate spring 30 is mounted to clutch wheel so that it contact the above engaged portion. Internal wall 9 of arm and protrusion 10 of spindle are faced so as to prevent inward bending of a pair of arms 6 protruded from the base 5. The outer tooth 8 is engaged with inner tooth of transmission gear 22 that idly engaged with the spindle 12. Thus, the spindle rotation causes transmission gear 22 to elastically deform arm 6 in inward direction so that engagement of inner tooth 29 and outer tooth 8 is released. As a result, when clutch is in connection state, both teeth are engaged to transmit power and clutch is cut. That is, when operation time is set, engagement is released, and when setting is completed, clutch automatically resets to connecting condition. 
     COPYRIGHT: (C)1980,JPO&Japio
Patent JP-2000204558-A (JP)
Title: Greening base material and greening method for face of slope or the like
Inventor: KANEYOSHI HIROYUKI
IPC: A01G1/00
Filed: 1999-01-19
Abstract: PROBLEM TO BE SOLVED: To permit to eliminate germination and growth inhibitor for plants, odor and high cost by mixing together the base materials comprising organic wood chips and soil dressing, and growth promotion agent, greening materials and base stabilizing agent. SOLUTION: 10 to 60% of organic wood chips and 90 to 40% of surface soil or the like are mixed together. This base material is graded to less than 15 mm in mean maximum diameter, and further mixed by adding a growth promotion agent, greening materials and a base stabilizing agent thereby creating a basic greening material. As a growth promotion agent, photosynthetic bacteria and nitrogen fertilizer are used. Next, greening material comprising seeds and other fertilizers is blended. Moreover, a base stabilizer either an inorganic stabilizer such as cement or an organic stabilizer is blended. Loss of greening base material due to rain water is prevented. In this way, greening can be performed easily and definitely and this is effective for maintaining for many years a greening base layer not easily affected by rain water or meteorology.
Patent JP-H01187436-A (JP)
Title: Plasma monitor
Inventor: KOMIYAMA YUZURU
IPC: G01N21/64
Filed: 1988-01-22
Abstract: PURPOSE:To calculate the concentration of produced chemical species quantitatively by irradiating the chemical species in plasma with pulse light while varying and adjusting the quantity of light of a light source, and diffracting spectrally light emitted by the chemical species and measuring its intensity in synchronism with the pulse frequency. CONSTITUTION:A light source part 1 emits exciting light 2, which is varied in quantity by sliding a light quantity variable adjustment part 3 consisting of filters to generate pulse light 2. The light 2 passed through a beam splitter 4 passes in the plasma 6 to excite the chemical species. The light emitted by the excitation is converged 8 and the light emission spectrum is separated and detected by a spectral light measurement part 9 and amplified by a synchronous amplification part 10. The light 2 reflected by the splitter 4, on the other hand, is converted 7 photoelectrically and sent to the amplification part 10. While the light emission intensity of the light emission spectrum of the output of the amplification part 10 and the light 2 are made to correspond to each other, a data processing arithmetic part 11 substitutes the light emission intensity ratio of the chemical species in the plasma when the light 2 is not projected in a calculation expression of correlation of variation in the light emission intensity to variation in the quantity of the light 2 to calculate the atomic number of the chemical species, i.e. concentration.
Patent JP-H03221325-A (JP)
Title: Heating device for shrinkage fit
Inventor: YANO SHIGEO
IPC: B23P11/02
Filed: 1990-01-22
Abstract: PURPOSE:To shorten the heating time of a work, to contract the equipment space, to reduce a running cost and to facilitate the temperature control of a work, by controlling a hot plate driving means according to the output signal of a temperature sensor, and equipping a control means which separates the hot plate from a work. CONSTITUTION:Two works W are set at a heating position, when a stopper 18 is opened and a slide carrier 15 is advanced. The work W is then heated with hot plates 3 -5 being driven by air cylinders 6 - 8 and each hot plate main bodies 3a - 5a being press-fitted to the work W and also a temperature sensor 14 is brought into contact with the specific part of the work W with the descent of a probe 13. When the rise of the temperature of the work W up to about 180 - 185 deg.C is detected by the temperature sensor 14, the hot plates 6 - 8 are retreated from the work W with the air cylinders 6 - 8 being actuated. The probe 13 is also ascended, the work W is carried out by a carry-out conveyor 16 and the following work cycle is started.
Patent JP-S63179177-A (JP)
Title: Ignition timing controlling device for internal combustion engine
Inventor: KOMURASAKI SATORU
IPC: F02P5/155
Filed: 1987-01-20
Abstract: PURPOSE:To prevent drop of engine output, worsening of fuel consumption and so forth, in the captioned device which delayed angle controls ignition timing based on the output of a knock sensor, by controlling the ignition timing corresponding to the voltage that a detected part by noise is subtracted from the knock detecting voltage. CONSTITUTION:An output signal of an acceleration sensor 1 which detects vibration acceleration of an engine is put in through a frequency filter 2 and an analogue gate 3 and compared at a comparator 6 with the output of a noise level detector 5 which detects the level of vibration noise other than knocking of the engine. The output pulse of this comparator 6 is integrated at an integrator 7, and the integration voltage according to the knocking strength is generated. And in this case, an output signal of the integrator 7 is received by a subtracter 35 through an AD converter 25, and the voltage corresponding to the noise signal of the engine to the knock detecting voltage which is digitally signalized is subtracted, and the signal after subtraction processing is put out to a distributing circuit 26 and the desired ignition timing control is carried out.
Patent JP-2000209645-A (JP)
Title: Mobile communication unit and incoming call control method
Inventor: TANABE HISASHI
IPC: H04W88/02
Filed: 1999-01-19
Abstract: PROBLEM TO BE SOLVED: To select a call reception mode in response to a carrying environment without troublesome operations by informing the arrival of an incoming call with a plurality of notice modes, detecting environmental vibration so as to send a reply signal for the arrival of the incoming call and to store the incoming call information and storing and controlling the notice or call reception mode corresponding to each of a plurality of environmental vibration patterns. SOLUTION: A notice circuit 30 informs a user of the arrival of an incoming call when a radio communication section receives an incoming signal. A control section 10 controls the notice mode when the notice circuit 13 informs of the arrival of the incoming call and has a reply section 10a that outputs a reply message to a caller when the incoming call is received and stores the arrived voice signal or the like. A pattern discrimination section 12 selects the notice circuit 13 to a call reception state operating mode related to each of various patterns via the control section 10 on the basis of a pattern such as vibration registered in a pattern registration table 2 in a portable communication unit 1 when receiving a detection signal from a vibration sensor 11.
Patent JP-S60153607-A (JP)
Title: Electromagnetic wave reflecting body
Inventor: AOKI MASAMI
IPC: B32B7/02
Filed: 1984-01-24
Abstract: PURPOSE:To attain light weight, ease of processing, excellent durability and improvement of the reflection characteristic by providing a conductive synthetic resin layer formed with a conductive film on the surface of a resin film surface to a surface layer or an inner layer of a synthetic resin mold. CONSTITUTION:A synthetic resin is coated with a metal or a metallic compound while using electroless plating or chalcocite processing. When chalcocite is used as a means for the provision of conductivity, univalent copper ions are adsorbed scatteringly to an urethane foam by applying heat treatment to the urethane foam containing a nitrile radical at a temperature of 50-120 deg.C in a bath containing bivalent copper ions, a reduction agent and an acid. On the other hand, a resin molding body is formed by using a thermoplastic or a thermosetting resin. Then a conductive synthetic resin is provided to either the surface layer or the innerlayer of the resin molding body.
Patent JP-S59144692-A (JP)
Inventor: ROBAATO JIEI SUTAUITSUKI
IPC: D21C9/147
Filed: 1984-01-24
Abstract: (57)【要約】本公報は電子出願前の出願データであるた め要約のデータは記録されません。