baber/WOPTO huggingface dataset:
Patent AP-2002002698-A0 (AP)
Title: 3-Azabicyclo[3.1.0] hexane derivatives useful in therapy.
Inventor: BANKS BERNARD JOSEPH
IPC: A61P9/00
Filed: 2001-06-07
Abstract: Compounds of formula (1), where the substituents are as defined herein, and the pharmaceutically or veterinarily acceptable derivatives or prodrugs thereof, are pharmaceutically and veterinarily useful, in particular they bind to opiate receptors, (e.g. mu, kappa and delta opioid receptors). They are likely to be useful in the treatment of diseases or conditions modulated by opiate receptors, for example irritable bowel syndrome; constipation; nausea; vomiting; pruritic dermatoses, such as allergic dermatitis and atopy; eating disorders; opiate overdoses; depression; smoking and alcohol addiction; sexual dysfunction; shock; stroke; spinal damage; and head trauma.
Patent ZW-6691-A1 (ZW)
Title: Pyrroie insecticides
Inventor: PHILIP REID TIMMONS
IPC: A01N43/36
Filed: 1991-06-04
Abstract: Substituted 1-arylpyrrole compounds of formula (II) below, are useful as pesticides, in particular for the control of insects, arachnids, and nematodes. Processes to make the compounds and intermediates used for their preparation are described. Additionally, compositions containing the compounds and methods of use therefore are provided. The compounds are of a formula (II) <CHEM>  wherein typical substituents are: X is halogen or a group R<5>S(O)n, in which n is 0, 1 or 2 and R<5> is CF3, CCl3, CF2Cl, CFCl2, CF2Br, CHF2, CHCl2 or CHClF; R<1> is H, Br, SCH3, CH3 optionally substituted or alkoxyalkylideneimino;     R<2> is CN;     R<3> is H, Cl or CH3 optionally substituted;     Y is CF3 or Cl;     X<1> and X<4> are each Cl; and X<2> and X<3> are each H. e us
Patent IE-910260-A1 (IE)
Title: Indole derivatives, their preparation and use
Inventor: JEPPESEN LONE
IPC: C07D491/18
Filed: 1991-01-25
Abstract: Indole derivatives of formula (I)   <IMAGE> (I)  wherein R1, R2, R3 and R4 may be hydrogen or lower alkyl optionally substituted by halogen; A1 represents a straight or branched alkylene chain containing from 2 to 4 carbon atoms; R5 is hydrogen or a straight or branched alkyl group; A2 is a straight or branched, saturated or unsaturated hydrocarbon chain containing from 2 to 6 carbon atoms; and R6 is selected from a group consisting of various structures, have been found to exhibit central nervous system activities.
Patent LU-88270-A1 (LU)
Title: Transparent polyurethane film - is made by depositing a reaction mixt. of a polyether polyalcohol, di:isocyanate and chain extender on a support
Inventor: LIN L Y
IPC: C08G18/73
Filed: 1993-05-17
Abstract: The film is made by deposition on a support of a reaction mixt. contg. an isocyanate cpd. obtained by polycondensn. of (A) a polyether-polyalcohol with mol.wt. 3000-6000 with (B) a di-isocyanate and (C) a chain-extending agent based on a polyether-polyol with mol.wt. 400-700 and viscosity 600-1200 mPa.s. Ratio between the free NCO gps. in (A) and the free OH gps. in (A) is around 2.
Patent MA-22581-A1 (MA)
Inventor: A FASSLER
IPC: C07C269/06
Filed: 1992-07-01
Abstract: The invention relates to compounds of the formula <IMAGE> in which R1 and R9 are, independently of one another, hydrogen, acyl, unsubstituted or substituted alkyl, alkenyl or alkynyl; heterocyclyl; sulpho, or sulphonyl which is substituted by unsubstituted or substituted alkyl, aryl, heterocyclyl, alkoxy, which is unsubstituted or substituted, or by aryloxy; sulphamoyl which is unsubstituted or substituted on the nitrogen; or phosphoryl which is substituted by one or two radicals selected independently of one another from unsubstituted or substituted alkyl, from unsubstituted or substituted cycloalkyl, from aryl, from hydroxyl, from unsubstituted or substituted alkoxy, from cycloalkoxy and from aryloxy, with the proviso that not more than one of the radicals R1 and R9 is hydrogen; and R2 and R8 are each, independently of one another, hydrogen or one of the radicals mentioned above for R1 and R9; or the pairs of substituents R1 and R2 or R8 and R9 can each, independently of one another, form together with the nitrogen atom to which they are bonded certain heterocyclic rings; R3 and R4 are, independently of one another, hydrogen, unsubstituted or substituted alkyl or cycloalkyl; aryl; heterocyclyl; or unsubstituted or substituted alkenyl; or R3 and R4 together are unsubstituted or substituted alkylene, alkylidene or benzo-fused alkylene; R5 is hydroxyl; R6 is hydrogen; or R5 and R6 together are oxo; and R7 is unsubstituted or substituted alkyl or cycloalkyl; aryl; heterocyclyl; or unsubstituted or substituted alkenyl; as well as the salts of the said compounds where salt-forming groups are present, furthermore process for the preparation thereof, pharmaceutical products, the use as pharmaceutical composition or for the preparation of pharmaceutical products, as well as intermediates for the preparation of these compounds.
Patent MA-28254-A1 (MA)
Title: Appareil permettant de connaitre le feu allume dans un croisement routier a l'interieur de son vehicule
Inventor: AIT ALI BRAIM YOUSSEF
Filed: 2005-04-18
Abstract: « Appareil permettant de connaître le feu allumé dans un croisement routier à l'intérieur de son véhicule » La présente invention concerne un appareil pour informer les conducteurs sur l'état des feux de trafic . Tous les chauffeurs rencontrent quotidiennement des problèmes de circulation liés essentiellement aux croisements avec feu rouge. Ces feux, bien qu'ils veillent à l'organisation de la bonne circulation, ils peuvent être la source de certains embouteillages et de certaines mésententes entre les gens. L'appareil vient donc pour remédier aux effets in souhaitables crées par ces feux rouge, et notamment mettre le conducteur dans de bonnes conditions sur la route avec moins de d'accidents.
Patent MA-20150343-A1 (MA)
Title: Lave mains mobile
Inventor: ER-RACHEDY MASSAOUD
IPC: A47K1/02
Filed: 2013-12-02
Abstract: -	l’invention concerne un dispositif lave-mains mobile comprenant un bassin pour évacuation d’eau, un réservoir d’eau, des robinets et un distributeur de savon liquide.
Patent MA-37379-A1 (MA)
Title: Formes polymorphes de l'acide -2-(1-(9h-purine-6-ylamino)propyl)-5-fluoro-3-phénylquinazolin-4(3h)-one
Inventor: CARRA ERNEST
IPC: C07D473/34
Filed: 2014-09-26
Abstract: Cette invention concerne des polymorphes de l'acide -2-(1-(9h-purine-6-ylamino)propyl)-5-fluoro-3-phénylquinazolin-4(3h)-one, des compositions de ceux-ci, des procédés pour leur préparation et pour leur utilisation.
Patent MA-37409-A1 (MA)
Inventor: GRIGUER HAFID
Filed: 2014-10-09
Abstract: L'invention concerne un dispositif autonome de conversion de l'énergie électromagnétique en énergie électrique composé d'une sonde absorbante électromagnétique (31). La dite sonde comprend des absorbants électromagnétiques (3) et (8) permettant de concentrer et amplifier l'énergie électromagnétique provenant de sources internes et externes sur une antenne intégrée (5). La dite antenne (5) est reliée à un convertisseur radiofréquence (15) pour transformer le signal rf alternatif fournis par celle-ci en un courant électrique continu (oc). L'énergie produite est gérée par un circuit (30) à plusieurs étages.
Patent MA-49350-A1 (MA)
Title: Procédés d'émission et de réception de sous-trames sib1-nb supplémentaires dans un réseau nb-iot
Inventor: SUI YUTAO
IPC: H04W72/04
Filed: 2018-11-16
Abstract: Selon certains modes de réalisation, un procédé mis en œuvre par un nœud de réseau consiste à diffuser une émission d'informations système. L'émission comprend des bits codés obtenus par lecture d'un tampon circulaire. L'émission est diffusée dans un premier ensemble de sous-trames correspondant à des sous-trames n°4 d'une pluralité de trames radio. Le procédé comprend en outre la diffusion d'une émission supplémentaire d'informations système. L'émission supplémentaire comprend des bits codés supplémentaires obtenus par poursuite de la lecture à partir du tampon circulaire. L'émission supplémentaire est diffusée dans un second ensemble de sous-trames correspondant à des sous-trames de la pluralité de trames radio autres que les sous-trames n°4.
Patent MA-51964-A1 (MA)
Title: Système de détection, d’identification et de traitement des adventices par télédétection
Inventor: ZENNAYI Yahya
IPC: B64D47/08
Filed: 2020-12-30
Abstract: La présente invention concerne un dispositif et méthode à base d’au moins d’un capteur optique embarqué sur drone permettant la détection et l’identification des adventices dans une parcelle cultivé en ligne, afin de faire un traitement phytosanitaire localisé et sur mesure. Ce système permet le suivi d’une culture en ligne durant la période de croissance. Un drone équipé d’au moins d’un capteur optique et d’un module de géolocalisation permet de filmer une parcelle, une méthode à base de traitement vidéo et l’intelligence artificielle permettant la détection et l’identification des adventices, cette information sera utilisée par le système pour déclencher un traitement de produit phytosanitaire sur mesure, à l’aide d’au moins une buse et d’un réservoir multi chambre.
Patent MA-53069-A1 (MA)
Title: Anticorps igf-1r et son utilisation comme véhicule d'adressage pour le traitement du cancer
Inventor: BEAU-LARVOR CHARLOTTE
IPC: C07K16/28
Filed: 2015-04-27
Abstract: La présente invention concerne un anticorps, en particulier un anticorps monoclonal, pouvant se lier spécifiquement à igf-1r, ainsi que des séquences d'acides aminés et d'acides nucléiques codant pour cet anticorps. Dans un aspect, l'invention concerne un anticorps, ou un fragment de liaison d'antigène de celui-ci, pouvant se lier à l'igf-1r et, par l'induction d'une internalisation d'igf-1r, étant internalisé dans la cellule. L'invention concerne également l'utilisation de cet anticorps en tant que véhicule d'adressage conjugué à d'autres composés anticancéreux, tels que des toxines, des radioéléments ou des médicaments, et l'utilisation de ceux-ci pour le traitement de certains cancers.
Patent MA-53532-A1 (MA)
Title: Modèle du système respiratoire en mode pression contrôlée à base du transistor mos
Inventor: EL MANSOURI KHALIFA
IPC: A61B5/08
Filed: 2021-06-15
Abstract: La présente invention concerne de manière générale un modèle et un circuit d'analyse des caractéristiques du système respiratoire humain en utilisant des composants électriques et électroniques. La présente invention offre une alternative améliorée du modèle respiratoire à base du circuit résistance-capacité, la compliance pulmonaire variable qu'est présentée par un transistor mos et la résistance des voies respiratoires sont calculés à partir d'un certain nombre de mesures physiologiques à savoir la pression, le débit, l'écoulement laminaire et une exponentielle invariante déterminée empiriquement. Ce circuit électronique est validé dans le contexte de la ventilation mécanique en utilisant le mode de pression contrôlée, le courant qui représente le débit a été mesuré et démontre la validité du modèle proposé. Ce circuit électronique est un moyen paramétrique de diagnostic et d'analyse de diverses pathologies du système respiratoire humain.
Patent UY-23458-A1 (UY)
Title: Recipiente de mezclado inclinable
Inventor: HEIBERG JAKOB
IPC: B65D8/04
Filed: 1992-08-10
Abstract: Un recipiente de mezclado (10) con configuración generalmente arqueada y que incluye costillas (32) estabilizantes espaciadas lateralmente, que se extienden sobre su superficie exterior entre la base y un borde que define una boca (18). Las costillas al inclinar el recipiente, definen continuamente un plano de soporte que se extiende lateralmente. El interior del recipiente es de material suave y rígido, mientras que su exterior es de un material que mejora la fricción no deslizante. La boca del recipiente está circundada por un borde abocinante (20) con una superficie interior que mejora la sujeción. La figura 1 ilustra la presente invención.
Patent UY-24665-A1 (UY)
Title: Procedimiento para cubrir con tapas encuadernaciones cosidas con espirales
IPC: B42B5/12
Filed: 1997-08-12
Abstract: La presente invención se refiere a un procedimiento para cubrir con tapas las encuadernaciones cosidas con espirales, caracterizado por: a) se colocan las hojas con falsa guarda y se perforan juntas; b) se coloca el espiral que coserá las hojas con la falsa guarda; c) se coloca la faja que unirá las falsa guardas; d) se pegarán las falsa guardas sobre la tapa. Para realizar encuadernaciones con lengüeta, se caracteriza por: a) la falsa guarda se dobla al medio hacia su revés y se perfora en el doblez. b) se pega la falsa guarda en la tapa, dejando que los ojales de las perforaciones sobresalgan (lengüeta) en el centro del lomo. Para realizar encuadernaciones con hilo cosido flojo, se caracteriza por: a) se pega la tira de cartón en el reverso de la falsa guarda en su centro; b) se hacen cinco perforaciones en el centro del cartón (y falsa guarda adherida); c) se hace una costura floja por las perforaciones que se inicia en la del centro y recorriendo las otras (por delante y por el reverso) y se remata en donde se inició. d) se pega la falsa guarda (con cartón y costura) en la tapa, debiendo quedar la costura en el centro del lomo. En la figura 1 se muestra un libro terminado.
Patent UY-24881-A1 (UY)
Title: 2-amino-6-(4-fenoxi-2-sustituido)-piridinas sustituidas
Inventor: NOWAKOWSKI J
IPC: C07D401/12
Filed: 1998-02-06
Abstract: Compuestos derivados de (2-amino-6-(4-fenoxi-2-sustituido)-piridina, composiciones que los contienen para tratamiento y prevención de trastornos del sistema nervioso central así como otras afecciones. Los compuestos de fnrmula(I) donde R1 y R2 se seleccionan entre H, halo, OH, alcoxi, alquilo, alquenilo; G es H, alquilo, aminocarbonil; R3 y R4 se seleccionan entre H, alquilo, donde el radical arilo es fenilo o naftilo, etc. La presente invención se refiere a un procedimiento para tratar o prevenir una afección seleccionada entre el grupo de compuesto por migrana, enfermedades inflamatorias como asma, psoriasis o artritis, demencia asociada con el SIDA, dependencia de drogas, alcoholismo y nicotina
Patent UY-26332-A1 (UY)
Title: Nuevos derivados del ácido aminodicarboxílico con propiedades farmacéuticas.
Inventor: ALONSO-ALIJA DR
IPC: C07C229/38
Filed: 2000-09-11
Abstract: La presente invención se refiere al uso de compuestos de fórmula (i) así como sus sales y estereoismeros para la producción de medicamentos para el tratamiento de enfermedades cardíacas y del sistema circulatorio.
Patent UY-30443-A1 (UY)
Title: Derivados de peririna 5-halo o ciano, composiciones y aplicaciones.
Inventor: ZETTERBERG FREDRIK
IPC: C07D205/04
Filed: 2007-06-27
Abstract: La presente invencion se refiere a ciertos nuevos análogos de piridina Formula (I) a procesos para preparar dichos compuestos, a su utilidad en medicina en general y especialmente como inhibidores de P2Y12 y como agentes antitromboticos, etc. , a su uso como medicamentos en enfermedades cardiovasculares así como también a composiciones farmacéuticas que los contienen.
Patent AT-526030-A1 (AT)
Title: Energiewandler zur Erzeugung elektrischer Energie für eine Schließeinrichtung
Inventor: REINHARD ENNE
IPC: E05B47/00
Filed: 2022-03-28
Abstract: Ein Energiewandler zur Erzeugung elektrischer Energie für eine Schließeinrichtung umfasst eine Handhabe (4) zur Betätigung der Schließeinrichtung und einen von der Handhabe (4) angetriebenen elektrischen Generator (9), wobei der elektrische Generator (9) als Axialfluss-Permanentmagnet- Generator mit wenigstens einem Stator (10) und einem relativ dazu drehbar gelagerten Rotor (13a, 13b) ausgebildet ist und der Rotor (13a, 13b) als Schwungrad ausgebildet ist oder mit einem Schwungrad zusammenwirkt.
Patent CS-189484-A1 (CS)
Title: Plynovy chromatograf
Inventor: AJRAPETJAN ARAM S
IPC: G01N30/02
Filed: 1984-03-16
Abstract: The gas chromatograph has programmed variation of column temp. by means of a thermostat. High accuracy of analysis is obtd. by stabilisation of the volumetric flow of gas-carrier through the chromatographic column during programming of its temp. This is achieved by using five-membrane comparator and a sealed vessel volume filled with gas. The input of the five membrane element is connected to the source of the gas carrier. - The inputs of press. regulator (2) and the five membrane comparator (3) receive gas carrier from source (1). In the initial state, the adjustment of regulator (2) sets the reqd. press. The comparator (3) operates in the repeater mode and ensures the necessary flow of gas passing via column (5) and detector (8). After this unit (4) receives a sample of the analysed prod. and in relation with a given programme the temp. of thermostatic vessel (7) increases. Since the press. of the constant vessel (6) is increased proportional to the increase of temp. of the thermostat (7) in accordance with the given programme, the element (3) operating as a summator realises algebraic equality of the output press. with the set press. plus the press. in vessel (6) and tends to increase, compensating the redn. of flow of gas from column (5) by increase of the gas-carrier at the output of element (3). Thus in the entire process during heating and cooling a constant volume flow of gas is ensured through the detector.
Patent ES-177773-A1 (ES)
Title: Un vehiculo-automovil con carroceria insonorizada
Filed: 1947-04-12
Abstract: Un vehículo con carrocería insonorizable caracterizado por la interposición de un tapiz de materia flexible amortiguadora o un dispositivo flexible equivalente entre un cuadro central portador de las suspensiones delantera y trasera el motor y el radiador y por otra parte la carrocería comprendido el capó y las alas el piso y además de manera que ningún órgano rígido pueda transmitir vibraciones del cuadro a la corrocería.
Patent ES-260694-A1 (ES)
Title: Synergistic nematocide
IPC: A01N29/02
Filed: 1960-08-30
Abstract: A nematocidal composition comprises 1 : 3 dichloropropene and an alkyl (other than methyl) or alkenyl isothiocyanate, preferably having 2 to 6 carbon atoms in the alkyl or alkenyl group or a cycloalkyl isothiocyanate, preferably containing up to 8 carbon atoms in the cycloalkyl group. Specified isothiocyanates are allyl, cyclohexyl, and n-butyl isothiocyanate. The compositions may contain inert carriers e.g. solvents such as deodorised kerosene, ketones, esters, alcohols, chlorinated hydrocarbons, various low boiling petroleum fractions or N.N.dimethyl formamide, or may be in the form of a dispersion or emulsion. The composition may contain 5-50 and preferably 10-30% isothiocyanate by weight. Specification 866,970 is referred to.
Patent ES-272760-A1 (ES)
Title: Process for the preparation of esters from dibasic acid anhydrides and organic sulphites
IPC: C07C69/60
Filed: 1961-12-07
Abstract: Diesters of dibasic acids and tetraesters of tetrabasic acids, capable of forming internal anhydrides, are prepared by reaction of said anhydrides with sulphites derived from aliphatic primary alcohols having not more than 16 carbon atoms or phenols in the presence of, as catalyst, alkali metal salts of organic carboxylic acids or inorganic acids, at a temperature in the range of from 100 to 200 DEG C. Examples of anhydrides which may be used and the anhydrides of phthalicacid and its substitution and hydrogenation products, pyromellitic, naphthalic, prehnitic, diphenic, maleic and succinic acids and their substitution products. Suitable sulphites are dialkyl sulphites in which the alkyl groups may be the same or different and may contain substituents and/or may be interrupted by oxygen atoms, for example, dimethyl, diethyl, bismethoxyethyl, di-n-butyl, di-(2-ethylhexyl), diphenyl and ethylbutyl sulphite. From 0.1 to 5% by weight of catalyst may be used, examples of catalysts being lithium bromide and chloride potassium fluoride, bromide, diphthalate, bicarbonate and sulphate. In carrying out the reaction, it is generally preferable to use a quantity of sulphite greater than that stoichiometrically required.
Patent ES-303011-A1 (ES)
Title: Process for obtaining sulfuric acid
IPC: C01B17/775
Filed: 1964-08-11
Abstract: A process for obtaining sulphuric acid comprises bringing a gaseous current containing SO3 at a temperature corresponding to the dew point of the gases into contact with a supply of an aqueous sulphuric acid solution containing 75 to 90% by weight of H2SO4, the volume and concentration of the solution being kept substantially constant by continuously extracting a quantity of this solution (corresponding to the acid formed by the absorption of the SO3) which is concentrated by being caused to flow in countercurrent and intimate contact with the gaseous current at a temperature of about 30 DEG C. above that corresponding to the dew point of <PICT:1074434/C1/1> the gases, before the current has come into contact with the sulphuric acid solution. The gaseous stream containing SO3 at, e.g. 250 DEG C. passes through heat exchanger 12 (Fig. 2) where it is cooled to a temperature of 30 DEG C. above that corresponding to the dew point of the gases the gaseous stream then passes through the concentrator 14 in intimate contact with H2SO4 from the absorber 20 via 19 concentrated H2SO4, e.g. 94% by weight is withdrawn at 16 the gases now at the temperature corresponding to their dew point leave 14 at 18 and pass to absorber 20 where they are contacted with H2SO4 of, e.g. 80% by weight which is circulated via 23 and is cooled at heat exchanger 24 excess acid formed due to the absorption of SO3 passes to concentrator 14 via 19. The gaseous current may contain 0.8-9% by volume SO3 and originate from the burning of a residual gas containing vesicular S and/or S compounds with natural gas, the oxidation of SO2 to SO3 then being effected catalytically.
Patent ES-322051-A1 (ES)
Title: Electric cell having electrode contact cap covered with protective seal
IPC: H01M2/34
Filed: 1966-01-21
Abstract: A primary cell has a protective seal 8 of polyethylene having a planar portion 9 covering the terminal cap 4 of electrode 3 and a flange portion 10 tightly fitted in opening 6 of the cap 4. The seal 8 is provided by injection moulding (Fig. 2, not shown). Access to electrode 3 is provided by removing seal 8 with the finger nail. Carbon rod 3 is centrally positioned in a zinc cup 1 surrounded by a plastics envelope 2.
Patent ES-337317-A1 (ES)
Title: Pneumatic tire compositions comprising ethylene / propylene / dicyclopentadiene terpolymer rubber
IPC: B60C1/00
Filed: 1967-02-27
Abstract: A composition suitable for forming the sidewall portion of a tyre comprises a blend of one or more elastomers with a terpolymer of two different alpha-monoolefins and dicyclopentadiene, there being 10 to 35 parts of terpolymer in 100 parts of total elastomer. The other elastomer may be natural rubber, polyisoprene, a mixture of neoprene rubber and natural rubber, a mixture of SBR and natural rubber, a mixture of polyisoprene and neoprene rubber, and a mixture of chlorosulphonated polyethylene, natural rubber and neoprene rubber. Fillers and vulcanizing agents may be present. The composition does not require any additional antiozonant. The EPDM elastomer may be oilextended.