baber/WOPTO huggingface dataset:
Patent IE-880293-L (IE)
Title: Adenosine 5'-carboxamides
IPC: A61K31/7042
Filed: 1988-02-03
Abstract: The compounds of the formula I <CHEM> wherein R represents hydrogen or lower alkyl; R<1> represents cycloalkyl, cycloalkyl-lower alkyl, 2-norbornanyl, 2-norbornanyl-lower alkyl, aryl, aryl-lower alkyl, aryl-cycloalkyl, 9-fluorenyl, diaryl-lower alkyl or 9-fluorenyl-lower alkyl; or R<1> represents a bicyclic benzo-fused 5- or 6-membered saturated carbocyclic radical or a benzo-fused 5- or 6-membered saturated heterocyclic radical containing a heteroatom selected from oxygen and sulfur which is directly attached to the fused benzene ring, any said bicyclic radical being unsubstituted or substituted on the benzo portion by lower alkyl, lower alkoxy, hydroxy, halogen or trifluoromethyl, or by a substituent -W-Z in which W represents a direct bond, lower alkylene, lower alkenylene, thio-lower alkylene or oxy-lowe alkylene and Z represents cyano, carboxy or carboxy derivatized in the form of a pharmaceutically acceptable ester or amide; R<2> represents hydrogen, lower alkyl or aryl-lower alkyl; R<3> represents hydrogen or hydroxy; R<4> represents hydrogen, lower alkyl, aryl-lower alkyl, cycloalkyl or hydroxy-lower alkyl; pharmaceutically acceptable ester derivatives thereof in which free hydroxy groups are esterified in form of a pharmaceutically acceptable ester; pharmaceutically acceptable salts thereof; their preparation, and their use as adenosine-2 receptor agonists are disclosed.
[EP0277917A2]
Patent IE-41220-L (IE)
Title: Expanding thermoplastic polymers
IPC: C08J9/08
Filed: 1975-03-12
Abstract: 1466427 Metal carbonate blowing agents FISONS Ltd 2 April 1975 [3 April 1974] 14763/74 Heading C3C Blowing agents, which are used to expand thermoplastic polymers, comprise as primary blowing agent (i.e. provides at least 50% by volume of the gas evolved on heating) a carbonate of zinc, lead, cadmium and/or lithium, with the proviso that where lead carbonate is used there is less than 2% by wt. of strong acid present in the composition and where lithium carbonate is used the polymer is not a polyamide, polymethyl methacrylate, polyvinyl chloride or an acrylonitrile/butadiene/styrene copolymer. Polymers are expanded by heating a composition containing the above blowing agent, e.g. to a temperature between 200 C. and the degradation temperature of the polymer and above the in situ decomposition temperature of the blowing agent and above the softening point of the polymer; the composition may be free from strong acid and contain a nucleating agent, e.g. a pigment, filler, magnesium or aluminium silicate, a clay, fumed oxide, silica or magnesium oxide. The polymer may be a polycarbonate, polyphenylene sulphide, polysulphone, polyamide, polyester or a styrene polymer. In the examples blowing agents consisting of basic zinc carbonate talc, and optionally palmitic, lauric, stearic or trimesic acids; zinc carbonate and optionally talc and lauric acid; basic cadmium carbonate (CdCO 3 .2CdO.3H 2 O) and talc; or zinc and potassium carbonate were used to expand a polycarbonate, acrylonitrile/butadiene/styrene copolymer, asbestos or glass fibre reinforced polypropylene, nylon 6, polystyrene, polypropylene, polyethylene, modified polyphenylene oxide or polyethersulphone, by feeding the mixtures into injection moulding machines. In an Example (11) the blowing agent was mixed with polyethylene and formed into pellets which were then used as the blowing agent.
[GB1466427A]
Patent IE-780669-L (IE)
Title: Antihypertensive compositions
IPC: A61K31/415
Filed: 1978-04-05
Abstract: Therapeutic antihypertensive compositions containing N-(2,6-dichlorophenyl)-4,5-dihydro-1H-imidazol-2-amine and N-(2-chloroethyl)-N-(1-methyl-2-phenoxyethyl)benzenemethanamine or their non-toxic, pharmaceutically acceptable salts are described as well as a method of reducing blood pressure in mammals.
[US4215130A]
Patent IE-800693-L (IE)
Title: Cancer diagnostic test
IPC: G01N33/574
Filed: 1980-04-03
Abstract: Inhibitor protein X in its substantially pure form having the following characterising properties: (i) it is a protein isolatable from human blood serum; (ii) it has a molecular weight of about 64,000 daltons and a Pl of 5.9; (iii) it inhibits bleomycin-induced degradation of PM-2 DNA by binding to the DNA; and (iv) it is found in lower concentrations in the serum of human beings having cancer than in the serum of cancer-free human beings. h
[GB2047712A]
Patent IE-780851-L (IE)
Title: 2-benzylperhydroazepines.
IPC: C07D223/12
Filed: 1978-04-28
Abstract: This invention relates to 2-benzyl-perhydroazepines of the general formula I (I), in which R1 is a hydrogen atom, an aliphatic or alicyclic hydrocarbon radical, a cycloalkylalkyl group or an aralkyl group, R2, R3, R4 and R5 are the same or different and signify a hydrogen atom, a halogen atom, an alkyl group, a hydroxy group, an alkoxy group, an acyloxy group, an optionally substituted amino group, a nitro group, an optionally substituted phenyl group, R1 not being methyl if R2, R3, R4 and R5 mean hydrogen, and their acid addition salts. This invention also relates to a process for the preparation of these compounds from known materials. The compounds of formula (I) and their pharmacologically compatible acid addition salts are useful in human and veterinary medicine because they produce central stimulation, an increase in vigilance, promote normal and pathologically inhibited drive of warm-blood animals. In addition some representatives display a strong analgesic action or an action which influences the blood pressure.
[CA1114374A]
Patent IE-36914-L (IE)
Title: Prostanoic acid derivatives.
IPC: C07D307/935
Filed: 1972-06-22
Abstract: 1372541 Prostaglandins IMPERIAL CHEMICAL INDUSTRIES Ltd 19 June 1972 [14 July 1971 16 Dec 1971] 33049/71 and 58399/71 Headings C2C and C2P [Also in Divisions C3 and A5] The invention comprises prostaglandins of the formula wherein R<SP>1</SP> is -CH 2 OH, -COOH or alkoxycarbonyl of up to 12 carbon atoms; either R<SP>2</SP> is OH or C 1-4 alkenoyloxy and R<SP>3</SP> is H, or R<SP>2</SP> and R<SP>3</SP> together form = O ; Y is ethylene or vinylene; A is ethylene or trans-vinylene; and R<SP>4</SP> is an aryl radical optionally substituted by halogen atoms, nitro, C 1-3 alkyl, C 1-3 haloalkyl, C 1-3 alkoxy or di(C 1-3 alkyl)amino radicals, and pharmaceutically acceptable salts of those compounds in which R<SP>1</SP> is COOH, and their preparation. They are prepared by hydrolysing compounds of the formula or mixed anhydrates thereof, wherein R<SP>5</SP> and R<SP>6</SP> each or betrahydropyran-2-yloxy or carboxylic acyloxy, followed by, if desired, esterification and reduction of the resulting esters. 16 - Methyl - 9 - oxo - 11α,15 - bis - (tetrahydro pyran - 2 - yloxy) - 17 - (4 - trifluoromethylphenyl) - 18,19,20 - trinor - 5 - cis,13 - transprostadienoic acid is prepared by oxidizing the corresponding 9α-hydroxy compound. Ethyl 2 - methyl - 3 - (3,4 - dichlorophenyl)- propionate is obtained by hydrogenating ethyl 3 - (3,4 - dichlorophenyl) - 2 - methylacrylate resulting from the reaction between ethyl 2-(diethylphosphono)propionate with 3,4-dichlorobenzaldehyde in the presence of butyllithium. Cyclopenta[b]furans of the Formula VI wherein Ac is p-phenylbenzoyl are prepared by reacting 5α - (4 - phenylbenzoylozy) - 4#- formyl - 3,3aα,4,5,6,6aα - hexahydro - 2H- cyclopenta[b]furan-2-one with phosphonates of the formula (MeO) 2 P(O) CH 2 -CO-CH(CH 3 )- OH 2 R<SP>4</SP> in the presence of butyllithium. 9α - Hydroxy - 16 - methyl - 17 - phenyl - 11α, 15 - bis - (tetrahydropyran - 2 - yloxy) - 18,19,20- trinor - 5 - cis, 13 - trans - prostadienoic acid is prepared by reacting (4-carboxybutyl)triphenyl phosphonium bromide with 2-hydroxy-3,3aα,- 4,5,6,6aα - hexahydro - 4# - (4 - methyl - 5 - phenyl- 3 - (tetrahydropyran - 2 - yloxy) - 1 - transpentenyl] - 5α - (tetrahydropyran - 2 - yloxy) - 2H- cyclopenta[b]furan, obtained by reducing the corresponding hexahydro - 2H - cyclopenta[b]- furan-2-one, resulting from the reaction hydropyran on the corresponding diol, which is prepared by hydrolyzing 3,3aα,4,5,5,6aα-hexahydro - 4# - (3 - hydroxy - 4 - methyl - 5 - phenyl- 1 - trans - pentenyl) - 5α - (4 - phenylbenzoyloxy) - 2H - cyclopenta[b]furen - 2 - one, resulting from the reduction of the corresponding cyclopenta- [b]furan of Formula VI above. Phosphonates of the formula are prepared by reacting dimethyl methylphonphosate with esters of the formula R<SP>4</SP>CH 2 CH(CH 3 )COO-alkyl.
[GB1372541A]
Patent FI-810431-L (FI)
Inventor: BRUYNES CORNELIS ADRIANUS
IPC: C07D501/24
Filed: 1981-02-12
Abstract: 3 min -Bromo-substituted deacetoxycephalosporanic acid sulphoxide derivatives are prepared by silylating the carboxy group (in order to protect same) of a 3 min -unsubstituted deacetoxycephalosporanic acid sulphoxide derivative in an inert anhydrous organic solvent, and then brominating the resulting silyl ester of the deacetoxycephalosporanic acid sulphoxide in situ.
Patent IE-781172-L (IE)
Title: Continuous business forms assemblies
IPC: B42D5/02
Filed: 1978-06-09
Abstract: The form arrangement consists of multi-layer sets of forms, connected one behind the other, which can be advanced through the printer of an office machine. Two outer, endless layers (11, 12) are separably connected to each other at the longitudinal edges and have tractor feed perforations (13) and, for separation, transverse lines (36) of weakness. In between the latter lie intermediate layers (21, 22, 23, 24, 28) which are connected to form individual sections. The sections are connected, only along one longitudinal side of the form arrangement, to each other and to only one of the outer layers, in a separable manner. The printed sets of forms are each completely separated at the transverse lines of weakness. With this arrangement, however, only the section and one outer layer (11) of the last printed set of forms can be separated easily, whereas the other outer layer (12) can be left as a drive web for initiating the advance of the subsequent sets of forms to be printed. As a result, the whole set of forms is not wasted for this purpose. <IMAGE>
[GB1600836A]
Patent IE-45360-L (IE)
Title: Herbicidally active carbamic acid esters
IPC: C07C239/00
Filed: 1977-07-15
Abstract: Carbamic acid ester of the formula <IMAGE> in which R and R1 are the same or different and are hydrogen, an aliphatic hydrocarbon residue which may also be substituted, a cycloaliphatic hydrocarbon residue which may also be substituted, an aromatic hydrocarbon residue which may also be substituted or a heterocyclic residue or wherein R and R1 together with the adjoining nitrogen atom form a heterocyclic residue. The compounds of the invention are herbicidal agents of particularly strong activity.
[US4257804A]
Patent IE-37516-L (IE)
Title: Radio position fixing
IPC: G01S5/10
Filed: 1972-12-14
Abstract: A radio position-fixing system using hyperbolic phase measurement, including two transmitting stations which radiate a specific, programmed, sequential and recurrent waveform and a movable receiver capable of synchronously receiving and detecting the transmitted waveforms and, by combining the signals in a predetermined manner, measuring certain phase differences in the signals which are representative of the hyperbolic position-line information for the receiver relative to the two transmitters.
[US3983559A]
Patent IE-821862-L (IE)
Title: Ganglioside derivatives
IPC: C07H19/00
Filed: 1982-08-03
Abstract: The invention relates to a method for preparing inner ester ganglioside derivates which comprises: (a) dissolving a ganglioside or a mixture of gangliosides obtained from a mammal in a non-aqueous organic solvent; (b) converting the carboxylate groups in the gangliosides to carboxyl groups or a salt thereof by means of ion exchange; and (c) reacting the resultant ganglioside or mixture of gangliosides with a lactonization reagent to form at least one lactonic bond in said inner ester ganglioside derivatives. 
[EP0072722A2]
Patent IE-871935-L (IE)
Title: Controlling the growth of weeds at a cereal crop locus.
IPC: A01N43/40
Filed: 1987-07-17
Abstract: The present invention relates to a method of controlling the growth of weeds at a cereal crop locus which comprises applying to the locus (a) diclofop, which is (R,S)-2-[4-(2,4-dichlorophenoxy)phenoxy]-propionic acid or an agriculturally acceptable salt or ester thereof and (b) diflufenican which is N-(2,4-difluorophenyl)-2-(3-trifluoromethylphenoxy)nicotinamide.
Patent IE-782006-L (IE)
Title: Non-refillable pourer fitment
IPC: B65D49/02
Filed: 1978-10-09
Abstract: There is described a non-refillable pourer fitment for the neck of a container comprising inner and outer parts captively attached to each other, a valve member located and movable in a longitudinal bore in the inner part and the outer part being formed with a longitudinal bore at its inner end and a dispensing aperture at its outer end, the longitudinal bore in the outer part varying in radius along its length from a portion of relatively large radius to a portion of relatively small radius, an obturator disc intermediate said portion of relatively small radius and said outer end having a radius greater than said relatively small radius. An inwardly extending peg on the obturator disc suitably controls the limit of movement of the valve member, and the obturator disc is preferably attached through spaced frangible stays to an annular ring adapted to fit tightly within the entrance of the bore of a container to which the fitment is fitted.
[US4217988A]
Patent IE-46096-L (IE)
Title: Coin testing device
IPC: H01L31/00
Filed: 1977-11-28
Abstract: A coin testing device for discriminating between an acceptable coin and an unacceptable coin of similar diameter but having a different edge characteristic. The device comprises a coin passageway defining a path along which coins pass through the device. A light source positioned to throw light on the edge of a coin as it passes along the coin passageway and a light sensor is positioned to receive light reflected from the edge of an acceptable coin as it moves along the coin passageway. Means are provided for examining a time-dependent quality of the reflected light received by the sensor such as the duration or the number of pulses and for comparing the value of the quality with the value for an acceptable coin.
[US4172222A]
Patent IE-822488-L (IE)
Title: Cloning vectors for use in streptomyces and related¹organisms
IPC: C12N15/76
Filed: 1982-10-14
Abstract: The present invention discloses selectable recombinant DNA cloning vectors for use in Streptomyces and related organisms.
[US4513086A]
Patent IE-882636-L (IE)
Title: Implants
IPC: A61K6/896
Filed: 1988-08-30
Abstract: Uniform adherent coatings of antimicrobial agents are applied to the surface of implants by applying a film of silicone oil to the surface of the implant and contacting the film-bearing surface with antimicrobial agents in a film-adherent form. A durable antimicrobial coating is formed. The coated implants can be packaged using mechanized implant handling equipment without significant loss of the antimicrobial coating.
[EP0306212A2]
Patent IE-842870-L (IE)
Title: Fungicidal triazoles
IPC: A01N43/653
Filed: 1984-11-08
Abstract: There are provided novel  alpha -(halo-substituted phenyl)- alpha -alkyl- beta -(1,2,4-triazol-1-yl)propanenitriles of Formula I below <CHEM> wherein X is fluoro, chloro or bromo and R is (C3-C8)alkyl with the proviso that when R is branched chain (C3-C6)alkyl the branching does not occur at the  alpha -carbon of the R substituent. There are also provided agronomically acceptable acid addition salts or agronomically acceptable metal salt complexes of a propanenitrile of Formula I. The above compounds are useful for combating phytopathogenic fungi.
Patent IE-893339-L (IE)
Title: Computer animation production system
IPC: G06T13/00
Filed: 1989-10-17
Abstract: A computer animation production system (2) for processing digital image data is disclosed. The computer animation production system (2) contains at least one information processing device (44-76) for enabling at least one user to develop, utilize and enhance digital image data. The information processing device (44-76) is associated with a first (4) and a second (6, 8, 10, 12 and 14) global area network (4). The first global area network (4) is for communicating digital control information to at least one information processing device. The digital control information includes image database information. The second global area network (6, 8, 10, 12 and 14) is for communicating the digital image data to the at least one information processing device (44-76). The digital image data includes pixel characteristic information for image reproduction on the information processing device. The second global area network (6, 8, 12 and 14) also includes a means for arbitrating (36, 38, 40, 42 or 43) access of the digital image data to the information processing device (44-76). Associated with the means for arbitrating is a temporary memory means (28, 30, 32, 34 or 35) for storing the digital image data likely to be accessed by the information processing device (44-76). A relational database management system (23) maintains the digital control information for production scheduling and tracking purposes.
Patent NO-750431-L (NO)
Inventor: JANSSEN E
IPC: E04D/
Filed: 1975-02-11
Abstract: Taksluk med elektrisk varmeelernent
Patent NO-791981-L (NO)
Title: Luftbaaren, terreng-gaaende medisinsk enhet.
Inventor: LEGUEU RENE
IPC: A61G/
Filed: 1979-06-14
Abstract: Luftbåren, terrenggående, medisinsk enhet
Patent NO-841613-L (NO)
Inventor: BARR PHILIP J
IPC: C12N15/16
Filed: 1984-04-24
Abstract: Prodn. of human insulin-like growth factor (IGF) comprises growing host cells contg. a structural gene which comprises a functional DNA construct of the gene encoding IGF joined in proper reading frame with secretory leader and processing signal sequences recognised by the host, and isolating secreted human IGF. The structural gene is downstream from and under transcriptional regulatory control of a transcriptional initiation region in a vector compatible with the host. The host is pref. a yeast. A DNA construct comprising a coding sequence for human IGF under transcriptional regulation of regulatory signals utilised by yeast is new. Also claimed is a construct contg. the IGF gene for expression in a cultured cellular host. Nucleotide sequences are defined with corresp. aminoacid sequence.
Patent NO-843555-L (NO)
Inventor: BLEEKER JAN JACOB
IPC: C08L101/00
Filed: 1984-09-07
Abstract: Biopolymer formulation, in particular a polysaccharide-containing water in oil emulsion, process for preparing such emulsions and process for concentrating these emulsions. Aqueous systems thickened by the incorporationof biopolymer emulsions.
Patent NO-850451-L (NO)
Title: Tannboerste
Inventor: AMOS WALTER
IPC: A46B9/04
Filed: 1985-02-06
Abstract: En tannbørste hvis børstehode (1) oppviser sekskantede hull (2) til opptak av børstebunter, hvorved børstefel-tet oppviser en sterkere tetthet av børster enn hos kjente tannbørster.
Patent NO-850926-L (NO)
Inventor: KARAGOZ BERCH YENOFK
IPC: H05B7/12
Filed: 1985-03-08
Abstract: A composite water-cooled electrode for electric arc steel furnaces comprises a tubular graphite body held in compression by means of tension stressed internal water supply pipe located between a metal header at one end and a hollow metal nipple at the other end of the electrode.
Patent NO-852088-L (NO)
Inventor: TOENSMANN ARMIN
IPC: E04B2/28
Filed: 1985-05-24
Abstract: The face or the roofing consists of a metal framework whose bays are filled with glass panes (27). On the building side, the metal framework consists of main profiles 16 and of crossmember profiles (28) extending transversely thereto, and on the outside, of cover profiles 24, 29 which cover the edges of the panes and are screwed to the main profiles or the crossmember profiles. The main profiles, the crossmember profiles and the cover profiles possess anchoring grooves for sealing strips supported on the edges of the panes. The main profiles and the crossmember profiles are equipped with receiving channels 20, 37 for condensation water and with receiving grooves 19, 32 for leakage water. The bottom of the receiving grooves 32 of the crossmember profiles for the leakage water extends up to the top edge of the associated receiving grooves 19 of the main profile and is supported on this top edge. The crossmember profiles 28 possess a main chamber 30 and a subsidiary chamber 31. The bottom of the subsidiary chamber is aligned with the bottoms of the receiving channels 37. Separate drainage systems are provided both for carrying off the leakage water and for carrying off the condensation water dripping off the inner edges of the panes. It is not necessary to make notches in the main profiles 16 in order to create a flow connection between the receiving grooves for the leakage water and between the receiving channels for the condensation water, which are provided in the cross- members and in the main profiles. <IMAGE>
Patent NO-852719-L (NO)
Inventor: VOELKER THEODOR
IPC: C08K5/04
Filed: 1985-07-05
Abstract: Stabilizer mixtures for vinyl chloride polymerizates for the improvement of the initial clarity and the heat constancy thereof. The stabilizer mixture contains nitrogen-free 3,5-substituted tetrahydropyrane-2,4,6-trione compounds of the formula:   <IMAGE> wherein R is a substituted or unsubstituted alkyl radical having 1 to 6 C atoms, and a metal salt of an organic acid and/or a metal phenolate.
Patent NO-855144-L (NO)
Inventor: LISIECKI ROBERT E
IPC: B31B50/64
Filed: 1985-12-18
Abstract: There is disclosed a container structure including a sealed side seam having a protected internal raw edge, and a method for accomplishing same. The method includes skiving or cutting a side seam flap along a taper to a feather edge, applying a sealant to the skived surface, and pressing the sealant-covered strip under heat and pressure into contact with the inside surface of the adjacent side wall panel to become sealed thereto without an exposed internal raw edge. Alternatively, the sealant may be applied to the side wall panel adjacent the skived tapered surface.
Patent NO-865251-L (NO)
Inventor: TOENSMANN ARMIN
IPC: E05B1/00
Filed: 1986-12-22
Abstract: An actuating handle arrangement for the actuation of fittings of a window casement or a door leaf includes an actuating handle which is mounted for turning about a turning axis on a housing which is secured to a window casement or door leaf frame. The actuating handle operates a pusher bar fitting which is coupled with an entraining member of a slide which is mounted in the housing for displacement in the longitudinal direction. The slide is provided with a guiding groove, in which there engages an entraining pin of an eccentric which is connected with the actuating handle. In the end positions of the actuating handle which correspond to the closing and the tilting position of the window casement, the line connecting the intersection point of the turning axis and the intersection point of a central axis of the entraining point with an imaginary plane along which the slide moves extends at right angles to the central longitudinal axis of the guiding groove.
Patent NO-880188-L (NO)
Inventor: SERGE LADRIERE
IPC: F42B5/18
Filed: 1988-01-18
Abstract: The disclosed weapon system comprises a gun barrel and a cooperating caseless ammunition. The ammunition is temporarily retained within the gun barrel by means of a conical force fit. The coupling comprises a female conical surface in the rear of the gun barrel and a male conical surface on the rear of the projectile wherein both surfaces have the same conicity.