baber/WOPTO huggingface dataset:
Patent IE-791682-L (IE)
Title: Omega-aroyl (propionyl or butyryl)-l-prolines
IPC: C07D207/10
Filed: 1979-09-04
Abstract: The present invention provides novel substituted omega -aroyl(propionyl or butyryl) -L-prolines, pharmaceutical compositions containing them useful for reducing blood pressure by inhibiting the conversion of angiotensin I to angiotensin II, and processes for preparing the novel compounds. The novel compounds are those of the formulae: <CHEM> <CHEM> <CHEM> wherein n is zero or one; R1 is hydrogen or alkyl having up to 3 carbon atoms; R2 is hydrogen, phenyl or alkyl having up to 3 carbon atoms; R3 is mercapto, formylthio, benzoylthio, all anoylthio having from 2 to 4 carbon atoms or moieties of the formulae: <CHEM> -S-CO2R5 , -S-CH2CO2R5 -S-@-NHR5 , <CHEM> <CHEM> <CHEM> and <CHEM> and wherein R9 is phenyl or substituted phenyl; R4 is hydrogen, phenyl or alkyl having up to 4 carbon atoms; R5 is hydrogen or alkyl having up to 4 carbon atoms; and ARYL is selected from the group consisting of 1-naphthyl, 2-naphthyl, 4-chloro-1-naphthyl 5,6,7,8-tetrahydro -1-naphthyl, 5, 6, 7, 8-tetrahydro -2-naphthyl, 4-methoxy-1 -naphthyl, 5-acenaphthyl, 4-biphenylyl, 5-indanyl, 4-indanyl and moieties of the formula: <CHEM> wherein R6 is selected from the group consisting of hydrogen, fluoro, chloro, bromo, trifluoromethyl, cyano, amino, phenoxy, halophenoxy, phenylthio, halophenylthio, p-cyclohexylphenoxy, alkyl having up to 4 carbon atoms, alkoxy having up to 4 carbon atoms, alkylamino having up to 4 carbon atoms, alkanoylamino having from 2 to 4 carbon atoms and alkoxycarbonyl having from 2 to 4 carbon atoms, R7 is selected from the group consisting of chloro, fluoro, bromo, alkyl having up to 4 carbon atoms and alkoxy having up to 4 carbon atoms, and m is zero, one or two; and the pharmacologically acceptable cationic salts thereof when R5 is hydrogen.
[EP0010347A1]
Patent IE-841796-L (IE)
Title: Protein solutions
IPC: A61K39/395
Filed: 1984-07-12
Abstract: The invention relates to aqueous solutions of proteins with a molecular weight above 8,500 daltons, which contain a compound of the formula I R2O-Xn-R3 (I) in which Xn is a chain of n members of the formula II or III   <IMAGE>   in any desired sequence, n denotes 2 to 200 and R1 denotes hydrogen, methyl or ethyl, it being possible for the radicals R1 to be identical or different but R1 being hydrogen in at least half of the chain members, and R2 and R3 are identical or different and denote hydrogen or an organic radical, to processes for their preparation and to their use. The invention furthermore relates to the use of compounds of the formula I for the pretreatment of hydrophobic surfaces to avoid adsorption of denaturing of proteins.
Patent IE-832001-L (IE)
Title: IMIDAZO £1,2-a| PYRIMIDINES.
IPC: A61P25/18
Filed: 1983-08-26
Abstract: Novel imidazo[1,2-a]pyrimidines of the formula <IMAGE> I wherein R is selected from the group consisting of alkyl of 1 to 8 carbon atoms, alkenyl of 2 to 8 carbon atoms, cycloalkyl of 3 to 7 carbon atoms, cycloalkylalkyl of 4 to 12 carbon atoms, aryl of 6 to 12 carbon atoms, thienyl and pyridyl, each of said group being optionally substituted with at least one member of the group consisting of halogen, alkyl of 1 to 5 carbon atoms, alkoxy and alkylthio of 1 to 5 carbon atoms, trifluoromethyl, amino, alkylamino of 1 to 5 alkyl carbon atoms and dialkylamino with alkyl of 1 to 5 carbons atoms, R1 and R2 are individually selected from the group consisting of hydrogen, alkyl of 1 to 8 carbon atoms, alkenyl of 2 to 5 carbon atoms, cycloalkyl of 3 to 7 carbon atoms, cycloalkylalkyl of 4 to 12 carbon atoms, benzyl and phenethyl, or taken together form alkylene of 3 to 5 carbon atoms, each of said groups being optionally substituted with at least one member of the group consisting of halogen, alkyl of 1 to 5 carbon atoms, alkoxy and alkylthio of 1 to 5 carbon atoms, trifluoromethyl, amino, alkylamino of 1 to 5 alkyl carbon atoms and dialkylamino with alkyls of 1 to 5 carbon atoms, X is selected from the group consisting of oxygen and sulfur and R3 is alkyl of 1 to 5 carbon atoms and their non-toxic, pharmaceutically acceptable acid addition salts, having anxiolytic activity and novel intermediates.
[US4532243A]
Patent IE-782060-L (IE)
Title: Silver-bismuth double chromate
IPC: C01G37/14
Filed: 1978-10-17
Abstract: Novel double chromate compositions having the general formula: MM'(CrO4)2, wherein M and M' are silver and bismuth, respectively. Methods of making AgBi (CrO4)2 are characterized by reacting silver dichromate with a bismuth salt to provide equal numbers of silver and bismuth atoms. These double chromate compositions have particular utility in batteries as active positive material. Due to the steadiness of discharge voltage and duration of discharge of batteries employing these double chromate compositions, such batteries are especially adapted for use in clocks and in cardiostimulators or pacemakers. (From US4184016 A) [FR2406898A1]
Patent IE-43968-L (IE)
Title: Cap liner dispensing apparatus.
IPC: B29C33/36
Filed: 1976-10-26
Abstract: An apparatus for dispensing predetermined amounts of lining material into cap shells, particularly of the deeply recessed type, includes a conveyor including a passage for conveying cap shells at predetermined speeds, an extruder provided above and along the shell-conveying passage for extruding predetermined quantities of a lining material through a discharge passage, a blade fitted adjacent to the exit end of the discharge passage and rotatably across it for cutting the lining material, and a drive for rotating the blade in response to the conveying of the cap shells. The drive is adapted to rotate the blade at a non-uniform speed in response to the speed of shell conveyance so that its speed gradually decreases as the exterior end of the blade in its radial direction approaches the shell-conveying passage, and gradually increases as it departs from it, whereby collision between the tip of the blade and the cap shells can be completely avoided.
[US4060053A]
Patent IE-772665-L (IE)
Title: Plant extract
IPC: C07J17/00
Filed: 1977-12-30
Abstract: Active Extract of plants of the family of the hypoxidaceae. This extract is obtained by carrying out the extraction of the whole plant or immediately after having cut out it or to have reduced it in particles. One heats this plant at a temperature of at least 60 degrees c until the enzymes which it contains are decontaminated then one carries out the of the aforesaid extraction plants at a temperature from 0 to 30 degrees c with an aqueous containing alcohol solution from 30 to 75% in volume of ethanol, during 1 to 15 days. [FR2375866A1]
Patent IE-852672-L (IE)
Title: Immunogenic complex
IPC: A61K39/44
Filed: 1985-11-01
Abstract: The invention relates to a process for preparing an immunogenic complex comprising a carrier molecule prepared by mixing viruses, mycoplasmas, bacterias, animal cells or proteins or peptides having hydrophobic regions with one or more solubilizing agents, whereby a complex having been formed between proteins or peptides and solubilizing agents, whereafter the proteins or the peptides have been separated from the solubilizing agent in the presence of a glycoside solution which contains one or more glycosides having hydrophobic and hydrophilic regions in a concentration of at least the critical micellular concentration, or alternatively have been separated from the solubilizing agent and transferred directly to the aforementioned glycoside solution, and the carrier molecule being bound to one or more molecules selected from peptides, proteins, carbohydrates, lipoproteins, glycolipides or small molecules, such as biotine, by coupling with known methods between functional coupling groups in the bound molecules and functional groups in the peptides or the proteins in the carrier molecule. 
<??>The invention also relates to a method for preparing such immunogenic complexes, compositions, vaccines containing such complexes and to reagents.
Patent IE-883426-L (IE)
Title: Frothflotation of mineral fines
IPC: B03D1/016
Filed: 1988-11-16
Abstract: Particles of a desired mineral are recovered from particles of an unwanted mineral in an aqueous slurry by a froth flotation process in which, after treatment of the mineral particles with a collector, a predominantly hydrophobic polymeric flocculating agent, which will selectively flocculate the desired mineral particles, is added to the slurry. The predominantly hydrophobic polymeric flocculating agent may be for example a polyvinyl ether or a polybutadiene and may be predispersed in a carrier liquid, which may be the frother used to produce the froth.
[US4956077A]
Patent IE-873469-L (IE)
Title: Resolution of 1,4-dihydropyridine derivatives
IPC: A61K/
Filed: 1987-12-21
Abstract: Optically active compounds of the formula <CHEM> or a salt thereof wherein R1 is H or lower alkyl; R2 and R6 are each independently lower alkyl, aryl, or arylalkyl; R3 is CN, NO2, CO2R5, CONHR5, SO2R5, or P(O)(OR5)2, where R5 is lower alkyl, lower alkoxyalkyl, aryl, or arylalkyl; R4 is aryl, heterocyclyl, or fused-ring heterocyclyl, optionally substituted with one, two, or three halo, NO2, CN, lower alkyl, lower alkoxy, lower alkylamino, CF3, OCH2F, or OCF3; are formed from a salt mixture of the compound with a resolving agent in a hot solvent mixture of an organic solvent and water.
[EP0273349A2]
Patent NO-811209-L (NO)
Inventor: DESPLANCHES GERARD
IPC: B28B21/18
Filed: 1981-04-08
Abstract: An outer casing (1) and an inner mandrel (2), both of which are cylindrical and are substantially coaxial, with powder (3) for manufacturing the tubular parts (11) filling the space which lies between them, contain a stationary distance piece (5) disposed against a shoulder (4) formed in the upper portion of the mandrel (2) and around the upper portion. A cover (6) also is provided around the upper portion and bears firstly against the upper end of the stationary distance piece (5) and secondly against the end of the casing (1), the cover (6) being hollowed out so as to provide an annular space (7) around the stationary distance piece (5), a moving distance piece (8) being disposed in the space (7) and bearing against the surface of the powder (3) so that during isostatic compression, the upper end of the moulded part (11) can extend into the space (7) while driving the moving distance piece (8). The apparatus can be used to manufacture beta sodium alumina tubes suitable for use as solid electrolytes in sodium-sulphur electric cells.
Patent NO-811431-L (NO)
Title: Tube av plast.
Inventor: GOTTAUF GEORG
IPC: G01F11/08
Filed: 1981-04-28
Abstract: For en mer nøyaktig og porsjonsvis dosering av innholdet oppviser en tube av plast et membranlignende . område (5) som f.eks. avgrenses av en rundtgående fure, rille, skår, spor e.l. (6), eller har mindre veggtykkelse enn tube-legemet (3) for øvrig. Tmmingen kan videre lettes ved. at tuben har ovalt tverrsnitt.
Patent NO-814410-L (NO)
Inventor: TAYLOR JAMES LONG
IPC: A61K9/50
Filed: 1981-12-22
Abstract: A process for producing lipid membrane structures (vesicles or liposomes) is disclosed, wherein a solution of bilayer forming compounds in a narrowly-defined two component solvent system is dispersed in an aqueous solution and, subsequently, at least a portion of that solvent system is stripped off. This process permits the readily-reproducible production of lipid membrane structures under gentle processing conditions, ideal for use when they contain pharmaceutically-active materials.
Patent NO-840409-L (NO)
Inventor: FONTANA LUDOVICO
IPC: B64D1/02
Filed: 1984-02-03
Abstract: The invention relates to a box distributor for sequentially discharging objects from aircraft and landcraft, particularly for sowing mines from helicopters. The distributor comprises a box-shaped framework with a plurality of vertical compartments closed at the base by shutters (1) tilting under control, the box-shaped framework being formed of a rigid box-shaped base (B), in which are housed the tilting bottom shutters (1) and their respective controls. Two sidewalls (P) are hinged on the two opposed longitudinal edges of the base, and a top wall (T) is releasably fixed at the top of the sidewalls of the box. For transport, the top wall is housed under the box-shaped base (B), while the sidewalls (P) are turned one over the other above the upper face of the base.
Patent NO-851294-L (NO)
Inventor: LUNDBAECK STIG
IPC: A61M60/882
Filed: 1985-03-29
Abstract: A double pump adapted for use as an artificial heart includes two ventricle-simulating chambers that are provided with respective inlets and outlets having valves incorporated therein and that are separated by a common partitioning wall structure. The wall structure has sections that are driven away from each other to reduce the volumes of respective ventricle chambers and expel liquid from the chambers through the outlets. The wall structure can also move laterally in response to differences in pressure between the chambers and hence change the volumetric ratio between them. This ensures a balanced action between the two halves of the heart- simulating pump during a systole phase and a diastole phase. The link mechanism is actuated by a cord through a motor, although only in one direction in the pressure phase, and hence the aforementioned changed volumes are readjusted primarily through the pressure exerted by the inflowing fluid. The pump may also include a variable volume atrium-simulating chamber communicating with the inlet to each ventricle-simulating chamber and having volume that is controlled in part by an externally acting gas pressure that varies in accordance with changes in the volumes of the ventricle chambers.
Patent NO-864235-L (NO)
Inventor: ZARATE JACOBO
IPC: C08F8/14
Filed: 1986-10-23
Abstract: 1. A method of using an ester of a 1-alkene/acrylic or methacrylic acid copolymer with an alcohol of the general formula  see diagramm : EP0220611,P10,F3  where R1 is an alkyl of 10 to 24 carbon atoms, R2 and R3 , which may be identical or different, are each hydrogen or an alkyl of from 1 to 3 carbon atoms, and x is from 2 to 30, for improving the flow properties of crude oil.
Patent NO-885489-L (NO)
Inventor: JAEGGI KNUT A
IPC: C07F9/38
Filed: 1988-12-09
Abstract: Araliphatylaminoalkanediphosphonic acids of the formula <IMAGE> in which R1 represents an aromatically substituted aliphatic radical, R2 represents hydrogen or a monovalent aliphatic radical and alk denotes a divalent aliphatic radical, and their salts have a marked regulating action on calcium metabolism and can be used as medicaments for the treatment of diseases which can be traced back to disorders thereof. They are prepared, for example, by reacting a compound of the formula <IMAGE> in which X3 denotes carboxyl and R0 denotes a radical R2, with phosphorous acid and phosphorus trichloride and hydrolysing the primary product.
Patent NO-885736-L (NO)
Inventor: SCHOLTHOLT HANS
IPC: H05K7/18
Filed: 1988-12-23
Abstract: Connecting strips (1) with connecting elements for the incoming and outgoing lines are attached to a supporting part (2). The latter is constructed from thin material, in the manner of a duct. The distance between the side limbs (5) of the supporting part (2) is approximately equal to the length of the connecting strips (1) which are placed on the ends of the side limbs. The latter have cut-outs (7) for the attachment of connecting strips, into which latching elements (8) and attachment elements (9) of the connecting strips engage, as a result of which the supporting part (2) is mechanically stabilised. <IMAGE>
Patent NO-891191-L (NO)
Title: Fremgangsmaate for fremstilling av nye, terapeutisk virksomme catecholderivater.
Inventor: FUKAZAWA NOBUYUKI
IPC: C07C233/22
Filed: 1989-03-17
Abstract: Terapeutisk virksomme catecholderi-vater med den generelle formelt. hvor er et hydrogenatom eller en acetylgruppe, og Rer en gruppe. hvor R. og Ruavhengig av hverandre. betegner et hydrogenatom, en alkylgruppe, en cycloalkylgruppe, en aryl-. gruppe eller en substituert arylgruppe, Rer et hydrogenatom, en alkylgruppe, en arylgruppe, en substituert arylgruppe eller en alkoxycarbonylgruppe, og X. er en direkte binding, et oxygenatom,. et nitrogenatom eller en methylengruppe, og i farmasøytisk henseende aksepterbare salter derav. Disse catécholderivater er i stand til a produsere nervevekst-faktor i spesielle vev i hjernen og er egnet til å forebygge og behandle regressive forstyrrelser i sentralnerve-systemet, deriblant senil demens av Alzheimers type. Fremstillingen av catecholderivatene er beskrevet.
Patent NO-892359-L (NO)
Inventor: FRISCH MARTIN
IPC: A47J31/36
Filed: 1989-06-08
Abstract: This device is arranged between a pump body and an extraction system and comprises a horizontal heating body (17) and a water circulation circuit (3,5,7,9,11,13,15), the said circuit comprising water circulation ducts and pockets for the retention of air, situated above the normal water level. Air can thus be dissolved in the water in order to provide an espresso coffee having lasting froth. 
<IMAGE>
Patent NO-903378-L (NO)
Inventor: CIDARIA DANTE
IPC: A01N63/50
Filed: 1990-07-31
Abstract: Disclosed is a Bacillus thuringiensis var. donegani, pathotype C, NCIMB 40152 and a preparation or toxin obtained therefrom, endowed with insecticidal activity against Coleoptera.
Patent NO-910355-L (NO)
Inventor: UTSCH FRANCIS V
IPC: A24B15/42
Filed: 1991-01-30
Abstract: An article (10) is provided in which a flavor-generating medium (11) is electrically heated by heaters (110) to combustion to evolve inhalable flavors such as tobacco or other components in vapor and/or aerosol form. The article has a plurality of charges (111) or flavor-generating medium which are heated to combustion sequentially to provide individual puffs. The charges are located in a portion (11) of the article detachable from a second section (12) in which is located a power source (121). The heaters are connected to the power source by finger (114) on the first section which are received in recesses (120) on the second section. A mouthpiece may be provided on the first section through which vapor and for aerosol may be inhaled.   <IMAGE>
Patent NO-910832-L (NO)
Inventor: DOTZAUER BERNHARD
IPC: C08L33/02
Filed: 1991-03-01
Abstract: Mouldings containing, as principal constituents, finely divided natural or synthetic materials and products of the condensation of high-molecular-weight polycarboxylic acids and polyhydric alcohols, alkanolamines or polyamines, their production and their use as ceiling tiles.
Patent NO-912860-L (NO)
Inventor: MACOR JOHN EUGENE
IPC: A61P3/06
Filed: 1991-07-22
Abstract: 3-(1,2,5,6-Tetrahydropyridyl) pyrrolopyridine derivs. of formula (I) and pharmaceutically acceptable salts and intermediates of formula (IIA) are new: where one of A,B,D,E = N and the others are C; R1,R2 = H or 1-6C alkyl; R3-6 = H, halogen, OH, 1-6C alkyl, 1-8C alkoxy, phenyl-(1-6C)alkoxy, phenoxy, NR7R8, CN, COOR10 or CONR11R12; R7,R8 = H, 1-6C alkyl, 1-6C alkanoyl or COOR9; and R9-11 = H or 1-6C alkyl. - Pref. R1,R2,R5,R6 = H; A = N; and R3 is absent; and esp. R4 = H, OMe, OEt, OPr, OBu or OH.
Patent NO-914680-L (NO)
Title: Fremgangsmaate til montasje av en konstruksjon til havs i ly av en beskyttelsesinnretning, og en beskyttelsesinnretning til utfoerelse av fremgangsmaaten
Inventor: BROUGHTON PETER
IPC: E02B17/00
Filed: 1991-11-28
Abstract: Beskyttende sperreinnretning (1) som hviler på havbunnen (2) via en basis (6), er montert på et drifts- eller montasje- sted (3). En passasje (8) er tildannet i det evre parti av sperreinnretningen (1) for å tillate innforing av en flytende konstruksjon (9) til stedet (3) etter montasje av sperreinnretningen. Ben (12) blir deretter senket til havbunnen (2) for å heve dekket (13) over den frie vannoverflate (14). Passasjen (8) kan deretter fylles med et lukkeelement (15) for å fullføre sperreinnretningen (1) . Oppfinnelsen benyttes til montasje av en oljefeltundersøkelses- og produksjons- plattform til havs.
Patent NO-924909-L (NO)
Inventor: BARTON DEREK JOHN
IPC: C11D17/06
Filed: 1992-12-18
Abstract: This invention relates to a process for binding water-sensitive active materials by forming a dough from a formulation which has the active material and an organophilic clay binder in particulate form using a non-aqueous liquid medium, shaping the dough and drying the shapes so formed. The granules so formed are releasably bound in the clay and the active species is released when the granules come into contact with water. The process of this invention is particularly suited to granulation of water-sensitive bleaches and bleach activators used in powder detergent formulations.
Patent NO-930970-L (NO)
Title: Halvleder-kondensator og mikrofonanordninger
Inventor: LOEPPERT PETER V
IPC: H04R25/00
Filed: 1993-03-17
Abstract: Det er frembragt en kompakt miniatyrkondensator og kon- densatormikrofon med god sensitivitet. Den omfatter en fast perforert bakplate som utgjør en fast elektrode i en paral- lellkondensator, følsom for innfallende lydtrykkbølge, og som utgjcr en bevegbar plate i parallellplate-kondensatoren, inn- retning for å posisjonere membranen i forhold til bakplaten uten å påtrykke vesentlig spenning på membranen, og FET- kretser som tilveiebringer et utgangssignal som er proporsjo- nalt i kapasitet til kondensatoren når membranen beveger seg i forhold til bakplaten.
Patent NO-933397-L (NO)
Inventor: SELIGER HEINZ HARTMUT
IPC: C12N15/11
Filed: 1993-09-23
Abstract: The invention relates to oligoribonucleotide analogues with terminal 3'-3' or 5'-5' internucleotide linkages. This modification stabilises the molecules modified in this way, including ribozymes, without adversely changing their properties, including catalytic activities where appropriate.
Patent NO-940369-L (NO)
Title: Maskin for påsetting av merker/skilt på kjöttvarer o.l.
Inventor: MARCHESONI UMBERTO
IPC: B65C/
Filed: 1994-02-04
Abstract: Maskin for automatisk påføring av merker /skilt (8), generelt på kjøtt- varer o.l., omfattende en tilbøyer (9) som bøyer merkenes (8) endeparti (8B) etter å være ført inn i kjøttvaren.
Patent NO-940629-L (NO)
Title: System og fremgangsmåte for detektering i olje- eller gassbrönn
Inventor: DAVIS JAMES LLOYD
IPC: E21B47/09
Filed: 1994-02-24
Abstract: System for å avføle passeringen av et element forbi et forutbestemt sted langs et produksjonsrør (4) som er anbragt l en olje- eller gassbrønn omfatter: en magnet (16) koblet til elementet (6), Idet magneten har et mykt legeme slik at magneten kan bores ut av en borekrone som senkes Inn l brønnen etter at elementet har passert det forutbestemte stedet, og en føler (18) koblet til utsiden av produksjonsrøret (4) på det forutbestemte stedet, for å detektere et magnetfelt fra magneten (16) når elementet (6) med magneten (16) som er koblet til dette passerer føleren (18). En fremgangsmåte for å hjelpe til med den riktige plassering av en sementblandlng l en olje- og gassbrønn omfatter: å pumpe en sementblandlng (8) gjennom et produksjonsrør (4) Inn l en olje- eller gassbrønn, å frigjøre en sementeringsplugg (6) Inn l produksjons- røret l serie med sementblandlngen, Idet sementerlngs- pluggen har en magnet (16) som angitt ovenfor, og å avføle sementerlngspluggen (6) på et forutbestemt sted langs produksjonsrøret, Innbefattende: å generere et nullslgnal som reaksjon på tilveiebringelse av et forspennende magnetfelt l motsetning til et magnetfelt som naturlig opptrer l produksjonsrøret på det forutbestemte stedet, og å endre nullslgnalet til et Indikatorsignal som reaksjonn på at magneten (16) beveger seg i produksjonsrøret (4) til det forut- bestemte stedet.