baber/WOPTO huggingface dataset:
Patent AU-550607-B2 (AU)
Title: Allylamines as monoamine oxidase inhibitors; intermediate allyl alcohols
Inventor: BEY PHILIPPE
IPC: C07C43/23
Filed: 1982-05-27
Granted: 1986-03-27
Abstract: Compounds of the formula:wherein:R is 3,4-methylendioxyphenyl; phenyl; phenyl monosubstituted, disubstituted, or trisubstituted by (C<sub>1</sub>-C<sub>8</sub>)alkyl, (C<sub>l</sub>-C<sub>a</sub>)alkoxy, (C<sub>1</sub>-C<sub>6</sub>)alkylcarbonyloxy, hydroxy, chlorine, bromine, iodine, fluorine, trifluoromethyl, nitro, (C<sub>1</sub>-C<sub>6</sub>)alkylcarbonyl, benzoyl, or phenyl; 1- or 2-naphthyl; 1-, 2-, or 3-indenyl; 1-, 2-, or 9-fluorenyl; 2-pyridinyl; 1-, 2- or 3-piperidinyl; 2- or 3-pyrrolyl; 2- or 3-thienyl; 2- or 3-furanyl; 2- or 3-indolyl; 2- or 3-thianaphthenyl; or 2- or 3-benzofuranyl;R, is hydrogen, (C<sub>1</sub>-C<sub>8</sub>)alkyl, benzyl, or phenethyl; X and Y,independently, are hydrogen, fluorine, chlorine, or bromine; and A is a divalent radical of the formula:wherein R is hydrogen, methyl, or ethyl, and m and n, independently, are an integer from 0 to 4, provided that m + n cannot be greater than 4;-(CH<sub>2</sub>)<sub>p</sub>-D-(CH<sub>2</sub>)<sub>q</sub>-, wherein D is oxygen or sulfur, p is an integer from 2 to 4, and q is an integer from 0 to 2 provided that p + q cannot be greater than 4; or-(CH<sub>2</sub>),CH=CH(CH<sub>2</sub>)<sub>s</sub>-, wherein r is an integer from 1 to 3 and s is an integer from 0 to 2, provided that r + s cannot be greater than 3;or a non-toxic pharmaceutically acceptable acid addition salt thereof; provided that when each of X and Y in Formula I is hydrogen, R cannot be phenyl; are MAO inhibitors useful for treating depression. Processes and intermediates for preparing the compounds of Formula I or II are also described.
Patent AU-650048-B2 (AU)
Title: Treatment of obesity with an alpha-2-adrenergic agonist and a growth hormone releasing peptide
Inventor: MUGICA JESUS DEVESA
IPC: A61K45/00
Filed: 1991-09-06
Granted: 1994-06-09
Abstract: Obese patients may be effectively treated by cojointly administering an alpha-2-adrenergic agonist, such as clonidine, and a growth hormone releasing peptide, such as GHRH, to restore or substantially enhance growth hormone release in such patients.
Patent AU-548297-B2 (AU)
Title: Recoverable wrap around sleeve
Inventor: TIGHT DEXTER CORWIN
IPC: H02G15/18
Filed: 1982-06-15
Granted: 1985-12-05
Abstract: A recoverable wrap-around sleeve 4 secured by rails and channel 1,2 and which is used to seal a substrate can be re-entered and re-sealed in the following way. A central section of the sleeve is removed, after cutting away the rails and channel, leaving butts of the sleeve on the substrate. A new sleeve is then recovered across the butts of the old sleeve. If the new sleeve is to seal properly there should be no leak path between the old butts and the new sleeve. In order to avoid such a leak path, any gap between the remnants of the old rails must be filled with adhesive. This is achieved by providing means, such as deformations 7, at the base of one of the rails 1 or on a flap 3 adjacent one of the rails 1 which allows flow of adhesive 8 between the rails when the original sleeve 4 is installed.
Patent AU-637270-B2 (AU)
Title: Chemical intermediates
Inventor: HUTTON JONATHAN
IPC: C07D405/12
Filed: 1991-11-19
Granted: 1993-05-20
Abstract: The invention concerns quinolinium salt intermediates of the formula I <CHEM> and processes for their manufacture; and their use in the manufacture of aryloxymethyl-substituted 1-alkyl-2-quinolone derivatives which are 5-lipoxygenase inhibitors.
Patent AU-740691-B2 (AU)
Title: Cementitious panel with reinforced edges
Inventor: MATHIEU MARC-ANDRE
IPC: B28B23/02
Filed: 1998-09-09
Granted: 2001-11-08
Abstract: A cementitious panel comprising a cementitious core which is fabric-reinforced at the surface thereof and whose longitudinal edges are reinforced by a network of fibers. A panel may be obtained wherein the surface edge reinforcement layers are relatively strong and hard such that a nail or screw may be driven through the edge of panel without pre-drilling and without breaking, even when nailed or screwed almost at the very limit of the edge of the panel. Such a panel may provide a long lasting substrate for humid or wet areas such as shower rooms and bath rooms.
Patent DE-2004288-B2 (DE)
Title: Sealed installation chamber with tubular torque tool - enables valve part replacement without interrupting valve function
IPC: F16K27/00
Filed: 1970-01-30
Abstract: The operating knob of a thermostatically controlled regulating valve is replaced by a closed tubular chamber. An adaptor plate with a circular recess locates the base plate to which the offset chamber is attached. When the chamber is in line with the valve axis, a tubular screw tool operated from outside the sealed chamber, is used to unscrew seal ring and to retrieve the thermostat. By pulling the screw tube with the thermostat into the chamber, the base can be rotated through 180 deg. so that the valve is sealed off. This allows the replacement of the defective thermostat without removing the valve from its location and without interrupting its function.
Patent DE-2019122-B2 (DE)
Title: Vehicle hydraulic brake servo - has narrow end of spacer tube passed through fixed wall to increase effective area of diaphragms
IPC: B60T13/563
Filed: 1970-04-21
Abstract: The brake servo has a fixed wall (2) through the middle of the housing, separating two moving walls (3, 4) with the moving walls joined by a spacer tube (7). The tube is stepped and has its smaller diameter passing through the fixed wall. This increases the effective area of the moving walls by an amount equal to the difference in the tube diameters. The operating piston (9) is located in the wider section of tube. The servo provides an improved braking effect with a minimum of alteration. The moving walls are connected to the housing by rolling membranes (5, 6).
Patent DE-2043908-B2 (DE)
Title: Agricultural machine driven from a tractor engine - has a connection for the drive shaft, which can move in the direction of the connection's pivot axis
IPC: A01B71/00
Filed: 1970-09-04
Abstract: The connection part on the machine side in this case, a mitre gear, is driven by the drive shaft of a tractor. The mitre gear is situated with its base plate in a carriage guide of the machines chassis. A V-belt pulley is driven by another V-belt pulley and a V-belt, and rotate a conveyor screw inside a hopper. The mitre gear is joined to the carriage guide by means of tension springs so that the V-belt is always taut. As soon as the drive shaft exerts pressure on the connecting part, the mitre gear is able to move. At the same time, the V-belt is slackened and the drive stopped. Similarly the V-belt can slip through if the screw inside the hopper, for instance, is blocked.
Patent DE-2048376-B2 (DE)
Title: Prestressing ring advancing system for cylindrical concrete structure - involves wedges between them and sloping step faces, moved by rams
IPC: G21C13/093
Filed: 1970-10-01
Abstract: Serrated step sections with sloping faces are first produced on the periphery in prestressing a cylindrical concrete structure. Annular stress members are fitted and moved along the slopes to extend them and introduce ring stressing. Wedges (3) are built in, between sloping faces (2a) and stress members (5). These are displaced by rams (4), supported on adjacent step sections (2) end faces (2b) or on wedges built in on a counter-running sloping face at the top edge. End faces may be at right angles to sloping faces. This enables a number of ring stressing members to be simultaneously moved hydraulically.
Patent DE-2059125-B2 (DE)
Title: Soft solderability test rig - comprises controlled vertical travel dipping bar for dipping sample into solder bath
IPC: G01N19/00
Filed: 1970-12-01
Abstract: The soft solderability testing rig comprises a vertically displaceable holding bar to the bottom end of which is attached a sample. This bar which is held in a horizontal arm may be lowered at constant adjustable speeds derived from a geared constant speed electric motor into a soldering bath. The travel of the bar is pref. controlled by means of a cam disk at the end of the reduction gear of the motor, which disk engages a roller attached to the sample holder bar. The rig permits the constant controlled condition immersion of samples into soft solder baths thereby allowing the assessment of the solder wetability of untinned test pieces.
Patent DE-2109786-B2 (DE)
Title: Passenger transport continuously moving conveyor - has panels pivoted to conveyor band at front and rear edges to reduce wear at diverting points
IPC: B66B21/10
Filed: 1971-03-02
Abstract: The conveyor belt for transporting people, is of the platform type, with continuous sectioned conveyor length running forward and back at constant speed in the same plane, fitted with palettes in a row, attached to a traction medium. The palletes (4) are mounted to swivel on the traction medium in the area of their front and rear sides (8, 11), on the inside (7). Mountings are such that the interval between the front and rear attachment point (9, 12) for each palette is automatically variable as it swivels. Bolts (13) can be used at attachment points, with guideways for them on the palettes. This simple and wear-resistant and prevents sudden jerking of palettes.
Patent DE-2136854-B2 (DE)
Title: Shatter-proof junction box for HV machine - has burst-open wall made of four joined triangular plates
IPC: H02G3/08
Filed: 1971-07-23
Abstract: The shatterproof junction box, for HV machines, has one of its walls removed and replaced by four triangular plates (4-7). The plates are welded or bonded along their outer edges to the rim of the box and are joined together along their adjacent edges by copper rivets (17) or weld seams or nuts and bolts. A sudden increase in pressure inside the box causes this sectioned wall to burst outwards -- the plates separating along their joins with one another and not with the rim of the box.
Patent DE-2146770-B2 (DE)
Title: Time program controller - with stencilled mask for conductor tracks and revolving coded contour disc
IPC: H01H43/12
Filed: 1971-09-16
Abstract: A program controller with a timer for use in dryers, dish washers and washing machines includes a stencilled mask to clear selected conductor tracks, and a revolving cam disc with coded track contours. The switch elements form a sliding contact and are designed as one-piece finger contacts. The programmer is simple to produce, functionally reliable and can be adapted to a great variety of contact operations. The program can be easily changed.
Patent DE-2163328-B2 (DE)
Title: Terminal shoe for connecting conductors - has matched pair of shells which grip cable by means of clamp springs
IPC: H01R4/18
Filed: 1971-12-21
Abstract: Two semi-cylindrical shells are formed at the end of a cable shoe. They are disposed so that a hollow cylinder is produced with the split edges parallel to the cable axis. Parallel to the split edges are projections along the diametrically opposite outer walls. Two spring clamps grip these projections and thereby force the opposed shells together to grip a mating cable end offered between the shells. At least one of the shells is made of an electrically high conductive material.
Patent DE-2229592-B2 (DE)
Title: Hand-written character reconstruction and transmission device - has increment-absolute converter stage associated with pen positioning element
IPC: G06K11/02
Filed: 1972-06-16
Abstract: The device is used to transmit and reconstruct handwritten characters, as the latter are written by means of a special pen, movable in three perpendicular directions, across a recording field having a number of detectors to provide signals representing the pen movement. These signals are supplied to a threshold value circuit and a digital signal is supplied for each signal exceeding the threshold value which is then coverted into a frequency signal for subsequent transmission. For obtaining the absolute position of the pen, an increment/absolute converter stage is associated with the positioning element for the pen, driven by a stepping motor and coupled to an absolute value source.
Patent DE-2744798-B2 (DE)
IPC: G04C3/14
Filed: 1977-10-03
Abstract: A device for automatically correcting the date indicator of an electro-mechanical timepiece to the first date of the next month at the end of each month. A pulse driven motor advances the date indicator one date in response to a plurality of pulsed drive signals with the motor advancing one step for each drive signal pulse, and at a speed corresponding to the drive signal frequency. A fixed number of drive signal pulses are applied to the motor each month to advance the date indicator through the dates of each month to the first date of the next month. A predetermined number of the drive signal pulses, corresponding to the number of dates of each month, are applied to the motor at a normal advance frequency normally to advance the date indicator. The remaining number of the drive signal pulses, for each month having less than 31 days are applied to the motor at a rapid advance frequency which is greater than the normal advance frequency, rapidly to advance the date indicator and indicate the first date of the next month.
Patent DE-2914220-B2 (DE)
IPC: B63B41/00
Filed: 1979-04-09
Abstract: 1. Drop keel arrangement for a wind-surfing device with a drop keel base (4) and a drop keel (5) guided therein, wherein a bearing (24) for a spigot (7, 8) projecting at the drop keel (5) is provided in the side walls (11, 12) of the drop keel box (4) and the length (L) of the slot opening (17) of the drop keel box (4) is greater than the width (B) of the drop keel (5), characterised thereby, that the side walls (11, 12) of the drop keel box (4) have at least one further bearing (24) displaced relative to the first in longitudinal direction and the spigot (7, 8) is selectably insertable into one of the bearings (24).
Patent FR-2663638-B2 (FR)
IPC: C12N15/12
Filed: 1990-06-26
Granted: 1995-02-10
Abstract: The new polypeptides have a defined of 446 amino acids or comprise fragments of it; provided the fragments; (i) contain at least those sites necessary for, when the fragment is exposed at the surface of a cell, binding to its (ant)agonists, specifically and in a measurable way (e.g. by means of a radioative ligand); (ii) can be recognised by Abs which recognise the full sequence but not dopaminergic D1 or D2 receptors; or (iii) can generate Abs recognising the full sequence but not dopaminergic receptor D1 or D2. The polypeptides include variants having licalised mutations provided they have not lost their dopaminergic receptor properties. Preferrred polypeptides show agonist affinity, by competition with the ligand iodosulphide-1 125, in the order quinpirole greater than apomorphine = dopamine and antagonist activity in the order raclopiriae greater than UH232 = haloperidol. DNA encoding the polypeptides, recombinant vectors and transformed hosts are also claimed. Antibodies to the peptides and nucleotide probes are claimed. Also claimed are diagnostic methods and kits specifically for pathologic expression of dopaminergic D3 receptor and genetic abnormalities of D3 receptor (in vitro).
Patent IE-S66096-B2 (IE)
Title: Method and apparatus for transferring cheese curd
Inventor: KELLY GEORGE
IPC: A01J25/00
Filed: 1995-08-25
Abstract: An apparatus is described for the transfer of salted cheese curd from a salting conveyor which reduced the possibility of salted cheese curd blocking the pipelines used to transfer the curd to blockformers. The apparatus comprises:- a spiral feed auger which collects salted curd from the salting conveyor, a blow through rotary valve conected to the auger, a cyclone for collection of the curd particles, at least one pipeline for connecting the base of the rotary valve to the cyclone, and an air blowing pump, the pump being connected to the pipeline adjacent to the rotary valve. Also described is a method of manufacturing hard pressed cheeses in which the salted cheese curd is blown along a transfer pipeline from a spiral feed auger which collects salted curd from the salting conveyor, to a cyclone for collecting the curd particles.
Patent JP-H0229673-B2 (JP)
IPC: C07D271/10
Filed: 1981-02-10
Abstract: Novel phenylpiperazinylpropanols of 1,3,4-oxadiazolylphenols and their physiologically tolerated addition salts with acids, processes for their preparation, and pharmaceutical formulations which contain these compounds and are useful in the treatment of hypertonia.
Patent JP-S5828755-B2 (JP)
IPC: H01S5/00
Filed: 1978-03-22
Abstract: PURPOSE:To adhere a heat spreader composed of two kinds of metal to a heat sink hard enough in a region except the operating region of a semiconductor chip, without causing strain near the operating region. CONSTITUTION:On electrode 8 near luminous part 10 of semiconductor chip 1, metal layer 12 is formed approximate three times as wide as luminous part 10. This layer, plated with silver, copper, etc., is large in thermal conductivity and hard to be alloyed with In solder. On the remaining part on electrode 8, gold layer 13 is selectively formed which is easy to be alloyed with In. Heat spreaders 12 and 13 are mounted on heat sink 14 and then fixed by solder 15 and, in consequence, the solder remains as soft metal In is since layer 12 is never alloyed, so that no strain will appear in the active region of the chip. As a result, layer 13 is alloyed with In and comes in hard contact with the heat sink.
Patent JP-S6153813-B2 (JP)
IPC: H01H85/30
Filed: 1985-03-15
Abstract: An HRC-fuse as an insulating body surrounding a main fusible conductor and an auxiliary fusible conductor connected to a spring biased impact pin. A conductive cap serving as a terminal for the fusible conductors is arranged on the insulating body and is provided with an outlet opening opposite the impact pin. A tripping hollow pin or sleeve coaxially surrounds at least a part of the impact pin and passes through the outlet opening. A bimetal release pawl is arranged in the one cap parallel to the pin and being electrically connected to the fusible conductors. The pawl engages a rest on the tripping sleeve to counteract a biasing spring. The impact pin and the tripping sleeve are triggered independently one from the other either by a short-circuit current melting the auxiliary conductor, or by an overload which heats up the bimetal release and triggers the sleeve. Both the tripping sleeve and the impact pin act on a load interruptor arranged opposite the outlet opening.
Patent JP-H0154360-B2 (JP)
IPC: A61K35/12
Filed: 1981-04-10
Abstract: What are disclosed are a protein, PP9, useful for the diagnosis and monitoring of diseases involving tissue degradation, and a method for its isolation, said protein having: (a) a content of carbohydrates of 5.57+/-1.35%, of which are 4.9+/-1.0% hexoses, 0.1+/-0.1% hexoseamines, 0.07+/-0.05% fucose and 0.5+/-0.20% neuraminic acid; (b) a sedimentation coefficient S20,W of 3.2+/-0.2 S; (c) a molecular weight of 35,100+/-3,800 determined in the ultracentrifuge; (d) a molecular weight of 40,000+/-4,000 determined in sodium dodecylsulfate (SDS)-containing polyacrylamide gel; (e) an extinction coefficient E1 cm 1% (280 nm) of 14.6+/-1.0 ; (f) an electrophoretic mobility in the range of the  beta 1-globulins; and (g) an isoelectric point in a pH range of 5.0-6.8.
Patent JP-H0780122-B2 (JP)
IPC: B24B53/065
Filed: 1988-03-09
Abstract: To dress the grinding wheel (1), a revolver (20) rotatably mounted on a pivoting arm (12) and having at least two dressing tools (3, 21) is provided on a CNC grinding machine, the rotational axis (19) of the revolver running parallel to and at a distance from the CNC pivoting axis (6) of the pivoting arm. The stepping of the revolver is derived from the rotary movement of the pivoting arm about its pivoting axis by a recess (26) being formed in the revolver, into which recess (26) an indexing pin (31) axially displaceable in the bearing stand (11) of the pivoting arm can be moved in such a way that, when the pivoting arm rotates, the revolver held in place by the pin performs a relative rotary movement through which another dressing tool moves into working position. <IMAGE>
Patent JP-2518591-B2 (JP)
IPC: B26B13/00
Filed: 1993-03-16
Granted: 1996-07-24
Abstract: The invention relates to end cutters, in particular for cutting through cables, having two flat loose blades which are located one on top of the other, and rotatable about a common rotation shaft and can be driven by means of a drive device. Each loose blade is in this case acted on by a suitable cam disc which is located in the plane of the blade and is coupled to the drive device. A desired force response while cutting up material in the form of ropes can be achieved in a simple manner by selection of the radii of the cam discs.
Patent JP-H0576792-B2 (JP)
Inventor: OZAKI MASAHARU
IPC: G09G3/14
Filed: 1984-03-23
Abstract: PURPOSE:To prevent the titled circuit from being affected by the fluctuation of supply voltage and the change of an ambient temperature by a method wherein the circuit is provided with a detecting element connected in series with an LED, a reference voltage output circuit and a current limiting element driving circuit and the LED is driven in constant current. CONSTITUTION:The driving current of an LED3, which has been limited by an MOS transistor (TR)4, runs through a resistor 5 and detecting voltage V1 generates on both ends of the resistor 5. On the other hand, drain current ID to run on an MOSTR7 fluctuates according to a temperature change without being affected by the terminal voltage V0 of a DC power source 2. Voltage Vr, whose current generates on both ends of a resistor 8, is impressed on a voltage comparator 6. Accordingly, output voltage, which corresponds to the component of a difference between the voltage V1 and the voltage Vr, is outputted from the output of the comparator 6 and the conductivity of the TR4 is controlled by this output voltage. As a result, current, which corresponds to the level of the voltage Vr, runs on the LED3 through the TR4 and the LED3 is driven in constant current. Accordingly, the LED3 is driven in constant current despite the fluctuation of the voltage V0 and when the ambient temperature changes, the change of the luminous efficiency is corrected.
Patent JP-3483646-B2 (JP)
IPC: A61K31/16
Filed: 1995-03-22
Granted: 2004-01-06
Abstract: Use of deoxyspergualin (I), i.e. ( plus or minus )-1-amino-19-guanidino-11-hydroxy-4,9,12-triaza-nonadecane-10,13-dione .3HCl, to prepare a medicament for therapy and prophylaxis of inflammatory hyperreactive diseases is new.
Patent JP-2681212-B2 (JP)
IPC: C07C43/04
Filed: 1989-03-20
Granted: 1997-11-26
Abstract: Process for the preparation of methyl tert-butyl ether (MTBE) by reaction of methanol with a mixture of hydrocarbons containing isobutene. The invention is characterised in that: - the reactants are introduced into a reaction-distillation zone which contains at least two superposed and nonadjoining stationary beds (2a,2b) of catalyst of sulphonated resin type, in which beds passages are arranged for a vapour phase, at least one distillation tray (4a), at least one liquid redistribution tray (5), - the distillation conditions are maintained in the said zone so as to have a descending liquid phase and an ascending vapour phase, - a continuous liquid phase is maintained in the lower part of the said beds, - a vapour phase rich in unconverted hydrocarbons is discharged at the top (8) of the said zone, - a liquid phase rich in MTBE is drawn from the bottom (10) of the said zone. <IMAGE>
Patent JP-H0261466-B2 (JP)
IPC: C07D263/32
Filed: 1982-04-23
Abstract: The invention concerns a new anti-inflammatory agent calcium oxaprozin, its preparation and use in pharmaceutical formulations. Calcium oxaprozin is more palatable than oxaprozin itself.