baber/WOPTO huggingface dataset:
Patent DO-P2002000544-A (DO)
Title: Formas de sal e-2-metoxi-n-(3-{4-[3-metil-4-(6-metilpiridin-3-iloxi)fenilamino] quinazolin-6-il} alil) acetamida y procedimiento de producción
Inventor: RICHTER DANIEL TYLER
IPC: A61K31/573
Filed: 2002-12-10
Abstract: La invencion se refiere a las sales succinato y malonato de E-2-metoxi-N-(3-{4-[3-metil-4-(6-metil 5 piridin-3-iloxi)fenilamino]quinazolin-6-il}alil)acetamida de la siguiente formula I: Mas particularmente, la presente invencion se refiere a las sales sesquisuccinato y dimalonato de formula I. La invencion se refiere tambien a composiciones farmaceuticas que contienen las sales succinato y malonato de formula I. La invencion se refiere ademas a procedimientos de tratamiento de enfermedades hiperproliferativas tales como los cánceres en mamiferos, especialmente en seres humanos, mediante la administracionde las sales anteriores y procedimientos de preparacion de las sales anteriores.
Patent DO-P2011000245-A (DO)
Title: Derivados de tiadiazoles y oxadiazoles, su preparacion y su aplicacion en terapeutica
Inventor: NAMANE CLAUDIE
Filed: 2011-07-28
Abstract: La invención se refiere a compuestos que responden a la fórmula (l): en forma (i) de base o de sal de adición a un ácido o en forma (ii) de ácido o de sal de adición a una base, así como su procedimiento de preparación y sus aplicaciones en terapia.
Patent EC-SP11011008-A (EC)
Title: Proceso para la preparación de derivados de l-alanina protegidos
Inventor: VILLANI FRANK
IPC: C07C227/16
Filed: 2011-04-27
Abstract: La presente invención se refiere a un proceso novedoso para la preparación de derivados de L-alanina protegidos, útiles como intermediarios de la síntesis de los compuestos usados como moduladores opioides mu/delta.
Patent EC-SP13012664-A (EC)
Title: Formas cristalinas de la sal clorhidrato de (4a-r,9a-s)-1-(1h-benzoimidazol-5-carbonil-2,3,4,4a,9,9a-hexahidro-1h-inden[2,1-b]piridin-6-carbonitrilo y su uso como inhibidores de hsd 1
Inventor: ECKHARDT MATTHIAS
IPC: C07D401/06
Filed: 2013-06-05
Abstract: La presente invención se refiere a compuestos definidos por la fórmula I en la que las variables R1, R2, R3, R4 y m se definen como en la reivindicación 1, que tienen actividad farmacológica importante. En particular, los compuestos son inhibidores de 11 -hidroxiesteroide deshidrogenasa (HSD) 1 y, por lo tanto, son adecuados para el tratamiento y prevención de enfermedades que pueden verse influidas por la inhibición de esta enzima, tal como enfermedades metabólicas, en particular diabetes tipo 2, obesidad y dislipidemia.
Patent EC-SP14013250-A (EC)
Title: Suspension concentrada acuosa que comprende una sal ácida de dodecilguanidina
Inventor: PIROTTE ALAN
IPC: A01P3/00
Filed: 2014-03-17
Abstract: La invención se relaciona con un concentrado en suspensión que comprende, expresado en peso con base en el peso total de la composición:a) 40 a 80% de partículas de dodecilguanidina o una sal ácida de dodecilguanidina de la estructura (1),en donde X representa un residuo ácido de un ácido monocarboxílico, dicarboxílico o mineral,b) 0 a 10% de un compuesto anticongelante, c) 1 a 10% de un agente humectante y/o d) un agente dispersante, e) 0 a 5% de un agente antiespumante,f) agua restante caracterizado porque, el diámetro medio de las partículas (d50) es al menos 7 µm y bajo 40 µm; y su uso para el tratamiento de una enfermedad fungicida en cultivos o plantas ornamentales.
Patent EE-200100193-A (EE)
Inventor: HAAPALINNA ANTTI
IPC: A61K31/416
Filed: 1999-09-27
Abstract: The present invention relates to a method for obtaining analgesia by administering 3-(1H-imidazol-4-ylmethyl)-indan-5-ol, its enetiomer or pharmaceutically acceptable ester or salt thereof to a mammal intraspinally, 3-(1H-imidazol-4-ylmethyl)-indan-5-ol, its enantiomer or a pharmaceutically acceptable ester or salt thereof can be administered intraspinally to a mammal obtaining analgesia without side-effects, such as sedation. The present invention also relates to a method for using the drug as an adjunct to anaesthesia by administering it intraspinally.
Patent GB-189705218-A (GB)
Title: Improvements in Water Tube Steam Generators.
Inventor: NAEYER LOUIS DE
Filed: 1897-02-26
Granted: 1898-01-01
Abstract: 5218. Naeyer, L. de. Feb. 26. Water-tube boilers.-Each element is preferably made up of two superposed water-tubes fixed at their ends into sectional junction boxes. Each box has three openings on its inner face, two of which serve to receive the ends of the water-tubes, and the third to receive the coupler between the boxes. The lower boxes open to the transverse water chambers C, C<1>, which carry the lowermost series of tubes, and which directly communicate with the overhead steam and water drum A by external passages of large dimensions. The uppermost front headers also open to a transverse chamber L connected to the drum. The arrangement of the superposed end boxes is such that they take a step-like form at each end of the boiler.
Patent GB-189708510-A (GB)
Title: Paint or Composition to be used as a Coating, more especially in the Manufacture of Artificial Slates, and for Coating Tiles, Plates, and other articles.
Inventor: HAAKANSON CLAES ALGOT
Filed: 1897-04-02
Granted: 1898-05-02
Abstract: 8510. HÕkanson, C. A., HÕkanson, J. H., and HÕkanson, A. R. April 2. Furniture, materials for; tables.-A composition consisting of finely-powdered sandstone or the like mixed with a suitable pigment and with boiled linseed oil, a solution of common glue, cerotine or other suitable drier, and turpentine in suitable proportions to form a jelly, is used for making artificial slates or for coating pieces of cardboard or fabric for use in making parquet floors or other inlaid work, or in making imitation marble-top tables, or in other ways.
Patent GB-189711868-A (GB)
Title: Improvements in Shuttle Guards for Looms.
Inventor: SUTCLIFFE HERBERT
Filed: 1897-05-13
Granted: 1897-09-04
Abstract: 11,868. Sutcliffe, H., and Kellett, R. May 13. Loom shuttle guards.-The guard consists of a bar E attached to brackets C, which have pivot pins c' passing through holes in castings B fixed to the hand-rail. The brackets C have projections c<2>, which are maintained in engagement with recesses in the castings by springs D. The guard is moved out of the way by pressing it back beneath the hand-rail, the projections c<3> being forced out of the recesses. When the loom is re-started the guard automatically resumes the operative position.
Patent GB-189712028-A (GB)
Title: Improvements in Carbon Plates for Galvanic Batteries.
Inventor: ATKINSON ROBERT WILLIAM
Filed: 1897-05-15
Granted: 1898-01-22
Abstract: 12,028. Atkinson, R. W., and Walker, S. F. May 15. Primary batteries. - Carbon plates for use in batteries are saturated with sulphur. This is effected by first saturating them in vacuo or otherwise with a liquid volatile at the temperature of molten sulphur, such as chloride of carbon, water, or preferably chloride of sulphur, and then immersing the plates in molten sulphur, which volatilizes and replaces the liquid. The adherent sulphur is removed after the plates have cooled. When copper or other metal is to be deposited locally on the carbon, the desired portion is first immersed as an anode in an electrolyte such as copper sulphate to remove the sulphur, the copper &c. being then deposited in the usual manner.
Patent GB-189712038-A (GB)
Title: Improvements in Lubricators.
Inventor: BRISBIN GEORGE LEWIS
Filed: 1897-05-15
Granted: 1897-07-31
Abstract: 12,038. Brisbin, G. L. May 15. Lubricators, sight-feed, for steam-engine cylinders. The lubricator is attached to the steam pipe 22. The oil reservoir 1 is surrounded by a steam jacket 5 supplied from the steam pipe 22 by pipes 8 and 6 with stop valve 7. The pipe 8 is continued to below the oil reservoir, and after passing a stop valve 9 enters a condensing- reservoir 13, which also serves to take the overflow from the oil reservoir when the latter is heated by the steam jacket. The gauge-glass 10 shows the level of the water in the reservoir. The feed overflows through a passage 14 and rises through a sight-tube 17 to the steam-pipe connection 20. The latter has a stop valve 21, and the sight-tube has stop valves 19 and 27 at top and bottom ; a bye-pass 25 with valve 26 is provided for use when necessary.
Patent GB-189712089-A (GB)
Title: Apparatus for Controlling Electric Motor Generators at a Distance.
Filed: 1897-05-15
Granted: 1898-04-09
Abstract: 12,089. Siemens Bros. & Co. and Estler, P. T. J. May 15. Transformers; distributing; switches; cut-outs. -Relates to means for controlling, say from the generating-station, motor generators, situated at a distance. The primary from the generating-station is connected to the armature and also to a few coils on the field magnets of the motor, so that, on switching on the current, the motor can start. The generated current in the conductor G is at first cut off from the distributing-circuit L by the switch f, but flows from s through a solenoid h, the core of which is attached to a lever p pivoted at m and loosely connected at n to a rod reciprocated by an eccentric on the armature shaft a. This rod carries ratchet teeth b engaging, when the rod is thrown over by the action of the solenoid with a wheel c and thus moving the arm d and connecting G with L, contact at s being broken at the same time. When the field magnets are fully excited, the coils supplied by the generating current are short-circuited by the switch w the arm y being attracted by the magnets. The arm d is held in position by the electromagnetic catch e, which releases it, so acting as a cut-out when the current fails.
Patent GB-189712288-A (GB)
Title: Improvements in Rock and Ore Crushers.
Inventor: BURNS CLARENCE ALONZO
Filed: 1897-05-18
Granted: 1897-07-10
Abstract: 12,288. Burns, C. A. May 18. Mills and apparatus. -The shafts of rock and ore crushers with gyrating heads are provided at their upper ends with removable sleeves C, which serve to hold down the crusher heads B and are retained in place by caps D and bolts. The sleeves may be divided at c<3>. The heads are fixed on the coned part of the shaft by keys of soft metal.
Patent GB-189716567-A (GB)
Title: Combining Prism Pavements and Reflectors in the Forward Part of the Vault to Light Basements.
Inventor: EWEN JOHN MEIGGS
Filed: 1897-07-13
Granted: 1897-09-18
Abstract: 16,567. Ewen, J. M. July 13. Pavement-Lights.-The rays of light are reflected and refracted by the pavement prisms H on to an adjustable pivoted daylight reflector E, and are thrown back into the basement A in approximatelyhorizontal lines. The reflector may be constructed of reflecting louvres or strips, as shown in Fig. 3, or it may consist of a silvered prism plate, as shown in Fig. 4.
Patent GB-189722028-A (GB)
Title: Improvements in and relating to Combined Dividers and Computing Scales.
Inventor: OSWALD RUDOLF FRITZ
Filed: 1897-09-25
Granted: 1898-09-24
Abstract: 22,028. Oswald, R. F. Sept. 25 Dividers.-The legs b, k are semi-cylindrical and the surface is marked with a series of parallel scales showing lengths, squares, cubes, areas of circles, &c. A link a is pivoted to one leg at c and to a sliding index d on the other leg. When the legs are opened to measure any length, such length, its square, cube, &c. can be read on the scales opposite the index. When closed, the instrument may be used as a receptacle for pen, pencil, pricker, &c., a cap being fitted over the points.
Patent GB-189800976-A (GB)
Title: Improvements in Plates for Collecting or Separating Gold.
Inventor: GREENE CHARLES EDWARD
Filed: 1898-01-13
Granted: 1898-03-12
Abstract: 976. Greene, C. E. Jan. 13. Drawings to Specification. Amalgamating; alloys.-Plates for collecting gold are formed of an amalgam of zinc and mercury together with sodium or similar reagent. The amalgam is cast on to a suitable strengthening- plate. A sodium amalgam is first formed which is stirred into molten zinc, the mixture then being poured into a mould in which is placed a plate of galvanized iron of the desired size and shape. The finished plate may have a flat, grooved, or other suitable working surface.
Patent GB-189808987-A (GB)
Title: Improvements in Portable Spirit Stoves and Accessories adapted for Cyclists', Travellers', and Picnic use.
Inventor: APPLEBY WILLIAM
Filed: 1898-04-18
Granted: 1898-07-16
Abstract: 8987. Appleby, W. April 18. Spirit lamps or stoves.- Relates to combined apparatus for the use of cyclists, tourists, and others. It comprises a spirit lamp, stand, and boiler, with or without a drinking-vessel, cover, pepper and salt box, spoon, &c. Fig. 1 shows the apparatus detached. The vessels are made to taper, so that they may nest together and be packed in a small bag or case for transport.
Patent GB-189812584-A (GB)
Title: Manufacture of Paper or Card having Designs Printed or Embossed on Iridescent Grounds.
Inventor: IMRAY JOHN
Filed: 1898-06-04
Granted: 1898-10-29
Abstract: 12,584. Imray, J., [Soc. Anon. A. Roudillon et Cie.]. June 4. Ornamenting.-An iridescent surface is formed by the process described in Specification No. 10,901, A.D. 1897, on woven fabric or other material. The material is then further ornamented by printing, or by printing and embossing. The design may be printed and the iridescent surface form the ground, or vice versÔ.
Patent GB-189813682-A (GB)
Title: Improvements in Electric Incandescent Lamps.
Inventor: SAGLIER VICTOR
Filed: 1898-06-20
Granted: 1898-07-23
Abstract: 13,682. Saglier, V., and Marþay, E. de. June 20. Incandescent lamps are provided with central tinned glass or other reflectors, wh:ch may be coloured, or with central blocks A, of any material containing a rare earth, which may be enclosed in a transparent tube. The filament B may be twisted about the block A, or a cylindrical reflector, as shown, witbout contact with it. Or two straight loop filaments may enclose opposite plates of a block of +-section.
Patent GB-189815125-A (GB)
Title: Improvements in Sight Feed Lubricators for Steam Engines.
Inventor: GREATOREX WILLIAM HENRY
Filed: 1898-07-09
Granted: 1899-06-02
Abstract: 15,125. Greatorex, W. H. July 9. Lubricators, sight-feed. Steam passing through the pipe g enters an oblong chamber divided into two parts h, h<1> and condenses therein. The part h of the chamber is continued down into the oil chamber S terminating in an inverted cone the mouth of which is closed by the valve u. The oil reservoir is drained by the cock T, and is filled through the aperture d closed by the valve a. When this valve is closed, the bell-shaped cover B is pressed down by the spring c, to prevent dirt from lodging in the filling-aperture. The oil displaced by condensed water passes through the passage R, controlled by the regulating-valve R<1>, and thence through the sight-tube W to the chamber h<1>, where it mixes with the steam and enters the delivery passage. The lower end of the sight-tube W is packed in the ordinary manner. The upper end is made tight by a ring of rubber or other packing-material compressed by a thimble-shaped gland sliding within the nut b. This gland is forced down by the screw m, a leaden washer being inserted between the gland and screw to prevent escape of steam.
Patent GB-189817637-A (GB)
Title: An Improved Heel Protector for Boots and Shoes.
Inventor: MARTLAND WILLIAM
Filed: 1898-08-16
Granted: 1899-07-15
Abstract: 17,637. Martland, W., and Piggott, W. Aug. 16. Heel protectors are cast in three parts A, B, C, each of which has spikes or holes for nails.
Patent GB-189818348-A (GB)
Title: Improvements in and connected with Smoke-consuming Furnaces.
Inventor: LANGENBACH GUSTAV
Filed: 1898-08-26
Granted: 1899-08-12
Abstract: 18,348. Langenbach, G. Aug. 26. Smoke-consuming.-An arch-shaped firebridge b<1>, b<2> spans the rear portion a' of the grate. The space below the grate is divided off by partitions s and s<1>, and the admission of air thereto is restricted, small apertures a<3>, Fig. 1, being provided, or an adjustable slide being fitted as shown in Fig. 6. In Fig. 6 also the partition s is shown adjustable horizontally. Behind the bridge is a constricting-baffle either erect as shown at c, Fig. 1, or depending as shown at c<1>, Fig. 3, in the case of a marine boiler. The two parts b<1> of the bridge may be prolonged to meet in the centre, the part b<2> being dispensed with. The burning fuel on the grate is pushed back as shown in dotted lines in Fig. 1, before fresh fuel is added.
Patent GB-189818971-A (GB)
Title: Improvements in Spring Actuated Weighing Machines.
Inventor: STEINKE PAUL JOHANN
Filed: 1898-09-06
Granted: 1899-05-13
Abstract: 18,971. Steinke, P. J. Sept. 6. Spring apparatus ; indicating-mechanism.-Relates to means for determining fractional weights with precision. The inner end of the spiral spring o is connected to a casing surrounding the spindle g, and its outer end to the arm p connected to this spindle, which carries a pointer r adapted to move over the primary scale u, while the spindle s', which is connected to the casing of the spindle g by gear-wheels k, s, has a loose pointer v which, however, remains in any position in which it is placed by virtue of friction. When the article, the weight of which is, say, 5À45 grammes, is placed in the scale q, the pointer r lies between 5 and 6 on the scale u. The pointer v is now placed at 5 on the scale w, and the button t on the spindle s<1> is turned until the pointer r indicates 5. The pointer v will now stand at 5À45 on the scale w.
Patent GB-189819432-A (GB)
Title: Safety Attachment for Elevators.
Inventor: COOKE GEORGE EDWARD
Filed: 1898-09-13
Granted: 1898-10-29
Abstract: 19,432. Cooke, G. E., and Cooke, C. L. Sept. 13. Safety suspending or retaining apparatus.-Fig. 2 shows a section of Fig. 1. The sides of a lift cage are fitted with rollers 10 to engage with the fixed guides 6. At the bottom of each side cams 12 are also mounted, with eccentric pins 13 for the attachment of rods 14 and 16, connected respectively to levers 19 and cross-pieces 17. The latter support the free ends of a normally-compressed spring 18. The inner ends of the levers 19, pivoted at 21, engage with levers 23, pivoted at 22, the inner ends of which bear on the upper side of a flange 24 on the draw-bolt 25, which is allowed a certain amount of vertical play in the cross beam 8. During normal working, the spring 18 is compressed by the pull of the lifting-rope, and the cams 12 kept out of contact with the guides. Should the rope break, the spring 18 rotates the cams 12, and causes them to grip the guides and arrest the cage. In a modification, the spring 18 is replaced by spiral springs attached to the rods 14.
Patent GB-189820418-A (GB)
Title: Improvements relating to Motors for Electric Railways.
Inventor: SHORT SIDNEY HOWE
Filed: 1898-09-27
Granted: 1898-11-05
Abstract: 20,418. Short, S. H. Sept. 27. Electric locomotives and motor vehicles.-The motor is mounted on the vehicle so that the shaft of the former is brought nearer to that of the latter, to permit of larger motors being used. With this view, the shaft or axle B of the vehicle is received in bearings P in, or within, the motor ring or frame G, which may be in sections, as shown in Fig. 4, or otherwise. By this arrangement, the motor may be moved from a horizontal to a vertical position on the axle B. The seat or bearing of the axle B, on the motor frame, may be enlarged or cored out to receive the lubricating- drippings.
Patent GB-189820595-A (GB)
Title: Improvements in Multiple Cylinder Air Compressing Engines.
Inventor: SZIMAY GEORG
Filed: 1898-09-29
Granted: 1898-12-03
Abstract: 20,595. Szimay, G. Sept. 29. Compressing. - Four cylinders are employed, arranged in pairs; each pair c, c<1> has a common piston-rod c<2>, and the.two piston-rods are joined by a crosshead pin c<3> which is driven by a single connecting-rod g. Each pair has a common inlet valve u<1> for the left-hand end, and u for the right-hand end of the cylinders ; these valves are closed by springs. and opened by an eccentric through a rod p and levers q<1>. The left and right hand ends respectively of the cylinders are in communication through pipes band h, which are fitted with non- return valves o<1> o. From these pipes, delivery pipes d<2> with non-return valves i, i<1> branch and lead to the reservoir w.
Patent GB-189820721-A (GB)
Title: Medicinal Preparation for the Cure of Rheumatic Affections.
Inventor: GILLIES DAVID
Filed: 1898-10-01
Granted: 1898-11-19
Abstract: 20,721. Gillies, D. Oct. 1. Pills.-A medicinal preparation for the cure of rheumatic affections is composed of powdered digitalis, sulphate of cinchonidine, powdered salicin, sulphate of quinine, powdered opium, citrate of lithia, and powdered myrrh, mixed in specified proportions. The mixture is made up into the form of pills.
Patent GB-189823070-A (GB)
Title: New or Improved Automatic Means for Securing Opera-glasses or Lorgnettes and for Recording and Registering their Use on Hire.
Inventor: BALINT DESIDERIUS
Filed: 1898-11-02
Granted: 1900-01-02
Abstract: 23,070. Bßlint, D., Monostor, A. B. de, Laszky, A., and Laszky, S. Nov. 2. Hiring opera-glasses.-A pair of glasses attached by a cord s rests on a spring shelf f in a fixed box B, the door of which is fastened till after prepayment. Coin action; coin-discharging mechanism.-The coin drops from the shoot q into a loop o upon a lever g, so that, when the lever is pulled by a handle t, the coin is drawn off a shelf s<3> and makes a bell crank j lift the latch of the door. Signals; registers.-The shelf springs up afte removal of the glasses, and completes an electric circuit L containing a signal. Fraud, preventing; signals.-If the attachment cord is severed, an electric circuit is broken to release a key which completes the circuit of an alarm bell.
Patent GB-189823523-A (GB)
Title: Improvements in the Production of Plates or Blocks for Printing.
Inventor: HILDYARD GEORGE RICHARD
Filed: 1898-11-08
Granted: 1899-03-04
Abstract: 23,523. Hildyard, G. R. Nov. 8. Negatives for photo-mechanical printing, producing. -Ptates or blocks for printing designs showing any required variation in tone, tint, or grain are obtained by etching a sensitized plate which has been exposed to light beneath a succession of screens of varying degrees of fineness of grain or texture, and beneath the negative, which is placed upon the sensitized plate after every exposure beneath a screen. The sensitized plate, preferably of zinc, is then washed with water and etched in the usual way ; before etching, the plate may be dried, and heated until the resist becomes light brown. Between the exposures to successive screens, additional tints or tones may be produced by rubbing, splashing, drawing, or transferring, or all the tones or tints may be prepared by similar means. The screens mounted on glass preferably consist of sheets of gelatine, upon which impressions in black ink have been produced. The negative may be an ordinary photographic negative, or one prepared by drawing the design in black ink upon a sheet of sensitized gelatine, which is then exposed, washed, and mounted upon a sheet of ground glass. The zinc plate is preferably prepared by immersing in a bath of nitric acid and alum, and coating with a sensitizing solution containing fish glue, ammonium bichromate, chromic acid, albumen, and water.
Patent GB-189826562-A (GB)
Title: Improvements in Wire Ropeways.
Inventor: JENSEN PETER
Filed: 1898-12-15
Granted: 1899-11-18
Abstract: 26,562. Jensen, P., [Kemlo, W.]. Dec. 15. Rope railways and tramways; rope grips.-In connection with wire ropeways, shunt rails F at terminal stations take the load by means of the pulley D on the hanger A and deliver it on to the rope R, which is the n gripped by a pair of jaws E, E<1> pivoted at G, G and caused to work together by a pin-andslot connection E<x>. The jaws grip the rope all round, and can ride over the rope pulleys.