baber/WOPTO huggingface dataset:
Patent CH-535769-A (CH)
Title: Cpds. of general formulae I and II, and intermediates of general formula III where A = H or one or more of the following:- halogen, lower alkyl, -CF
Inventor: FRANK J VILLANI
IPC: A61K31/00
Filed: 1964-04-20
Abstract: Cpds. of general formulae I and II, and intermediates of general formula III - where - A = H or one or more of the following:- halogen, lower alkyl, -CF3, OH, Oalkyl, O-lower acyl, in any positions but pref. 7 and 8. - B = a pyridine nucleus residue - U = a monovalent residue contng. an amino group at least 2C atoms distant from the tricyclic nucleus e.g. 3- or 4-piperidyl, or -X-NR'R2 - V = a divalent residue contng. an amino group at least 2C atoms distant from the tricyclic nucleus, e.g. 3- or 4-piperidylidene, or =Y-NR'R2 - W = H or OH - R' and R2 independently = H or lower alkyl, or together with the N atom, C atoms and not more than one other N or O, form a 5 or 6 membered hetero cyclic ring. - X and Y = (2-9C) hydrocarbon residues - Antihistamines, antiseratonins, antianaphylactics.  Dose 0.1-15 mg./kg./day. - I and II-4 aza cpds. and II (V=piperidylidene) are partic. active antihistamines. - II (V= =CH.CH2CH2NMe2) are C.N.S. active cpds.  I and II-3 aza cpds. are antihypertensives.
Patent CY-1758-A (CY)
Title: Substituted 1-(1H-imidazol-4-yl) alkyl-benzamides
IPC: C07D233/64
Filed: 1994-07-15
Abstract: New substituted 1-(1H-imidazol-4-yl)alkyl-benzamides and their salts, processes for the preparation thereof and pharmaceutical compositions. These compounds have the formula  <IMAGE>  wherein R1, R2=hydrogen or C1-C4-alkyl, R3=hydrogen, amino, hydroxyl, C1-C4-alkyl or C1-C4-hydroxyalkyl, R4=hydrogen or C1-C4-alkyl, or R3R4N=pyrrolidino, piperidino or morpholino, R5 and R6=hydrogen, hydroxyl, C1-C4-alkyl or C1-C4-alkoxy, at least one of R5 and R6 being other than hydrogen. These compounds are prepared either by reacting a nitrogen compound with an alkyl 1-(1H-imidazol-4-yl)alkyl-benzoate or with a 1-(1H-imidazol-4-yl)alkyl-benzoic acid, or by hydrolyzing in an acid medium a 2-hydroxy-3-[1-(1H-imidazol-4-yl)alkyl]-benzonitrile. The compounds have anti-ischemic and  alpha 2-adrenoceptor agonist activities.
Patent DK-166981-A (DK)
Inventor: TRUMMLITZ G
IPC: C07D275/06
Filed: 1981-04-13
Abstract: Compounds of the formula   <IMAGE>   wherein R1 is hydrogen or hydroxyl, and non-toxic, pharmacologically acceptable salts thereof formed with inorganic or organic bases. The compounds as well as their salts are useful as sweetening agents.
Patent DK-203285-A (DK)
Inventor: OPSVIK PETER
IPC: A47C7/24
Filed: 1985-05-07
Abstract: A chair provided with a seat (1) and possibly a back rest (4) said seat (1) having a longitudinal saddle shaped part, the upper surface cross-section of which having approximately the shape of an inverted U, and saddle-like members (2, 3) projecting transversely out from a mid-portion of each longitudinal side of said seat part to support the rear, upper thigh portion of the chair user, said seat as viewed from above being substantially shaped like a groin-vault or a Welsh - or underpitch vault.
Patent DK-310687-A (DK)
Inventor: FRANSSON GUNNAR SVANTE
IPC: H01R/
Filed: 1987-06-18
Abstract: A connection element for insertion in a terminal strip is designed with a hole 5 at one end, which hole is threaded for a screw, and with a soldering eye 3 at its other end. The connection element 1 is constructed in a plate material with two different thicknesses, as the soldering eye 3 is constructed of a material which is considerably thinner than the material around the threaded hole 5. In addition the connection element 1 is constructed with two legs 7 with considerably less width than the width of the connection element around the threaded hole 5, which legs connect the material around the threaded hole 5 to the soldering eye 3 and are bent at an angle. <IMAGE>
Patent DK-367884-A (DK)
Inventor: TIETJEN MARLENE
IPC: A61K8/34
Filed: 1984-07-27
Abstract: Cosmetic products which do not suffer phase separation comprise a mixture of a cosmetically acceptable wax with dimethylpolysiloxane and either an organosilane or an organically substituted polysiloxane.
Patent DK-369182-A (DK)
Inventor: LINDHARDTSEN PAUL VOERSAA
IPC: E04B/
Filed: 1982-08-18
Abstract: A construction element comprising a timber frame, in which the timber frame can be built one section at a time and the centuries-old process of initially fitting a corner post and then continuing the construction of the timber frame by fitting the posts individually one after the other is therefore made redundant. This is made possible by the use of a fixture 1, comprising a series of four hooks 3 fitted about 50 cm apart on a moulding. These hooks 3 can engage in holes 4 placed the same distance apart on another moulding on an adjoining element. As the backboard, glass wool matting is used, covered by a damp course and a plasterboard. On top of this can be mounted any cladding which might be desired. <IMAGE>
Patent DK-430586-A (DK)
Inventor: CLARK MICHAEL THOMAS
IPC: A01N43/12
Filed: 1986-09-09
Abstract: Phenoxy phthalide derivatives having the general formula <CHEM> wherein R1 represents a hydrogen or halogen atom or an alkyl or haloalkyl group; R2 and R3, which may be the same or different, each independently represents a hydrogen or halogen atom or an alkyl, haloalkyl, nitro or cyano group; and R4 and R5, which may be the same or different, each independently represents an alkyl group. Processes for the preparation of such compounds, herbicidal compositions containing them, and their herbicidal use.
Patent DK-504789-A (DK)
Inventor: ALEXANDER STEPHEN EDWARD
IPC: A61P1/02
Filed: 1989-10-11
Abstract: The problem of formulating a dentifrice which is compatible with a bis-biguanide anti-bacterial agent, for instance chlorhexidine or alexidine, is solved by using a nonionic thickening agent; a nonionic surfactant; and an abrasive which is either a sparingly soluble salt, for instance calcium carbonate, (used in combination with an agent to suppress anion formation), or an essentially insoluble compound, for instance, a silica of low anion content, or a mixture thereof. Preferably, the composition has a flavour which is mainly aniseed, balanced by mints. Preferably during the preparation of a silica containing dentifrice, chlorhexidine and saccharin are added together at an early stage, prior to the addition of silica, to avoid the formation of lumps. Such dentifrices are useful in the prophylaxis and/or treatment of periodontal disease and caries.
Patent DK-511385-A (DK)
Inventor: BRECHOT CHRISTIAN
IPC: C12Q1/70
Filed: 1985-11-06
Abstract: A reagent for quantitatively determining a viral DNA or RNA, for example derived from hepatitis B virus, consists of a previously ascertained concentration of a phage which contains a DNA sample, together with proteins, which can be hybridized with the viral DNA. The process is carried out by the reagent being brought into contact with the sample, which contains the viral DNA to be analysed, under conditions which permit hybridization and by the quantity of hybrid formed being compared with a predetermined nomogram for the purpose of finally determining the content of viral DNA in the sample.
Patent DK-515186-A (DK)
Inventor: BEACHY ROGER NEIL
IPC: A01N65/38
Filed: 1986-10-28
Abstract: A process for producing genetically transformed plants which are resistant to infection by a plant virus, comprises the steps of:   (a) inserting into the genome of a plant cell a recombinant, double-stranded DNA molecule comprising (i) a promoter which functions in plant cells to cause the production of RNA sequences of said plant virus; (ii) a DNA sequence that corresponds to an RNA sequence of said plant virus. (iii) a 3' non-translated region which functions in plant cells to cause the addition of polyadenylated nucleotides to the 3' end of said RNA sequence;   (b) obtaining transformed plant cells; and (c) regenerating from the transformed plant cells genetically transformed plants which have increased resistance to infection by said plant virus. o
Patent DK-594688-A (DK)
Inventor: SUVANTO ERKKI
IPC: B60C/
Filed: 1988-10-26
Abstract: PCT No. PCT/FI88/00017 Sec. 371 Date Oct. 25, 1988 Sec. 102(e) Date Oct. 25, 1988 PCT Filed Feb. 8, 1988 PCT Pub. No. WO88/06538 PCT Pub. Date Sep. 7, 1988.The invention concerns a sleeve-mounted spike (10) fitted on a vehicle tire, comprising a rivet (11), a head (12), a tip (13) and a sleeve (14). The part (11a) of the rivet towards the tip and the part (11b) towards the head subtend an angle ( alpha ) having a magnitude in the range from 150 to 179 degrees, whereby no rectilinear contact is established between the rivet (11) and the sleeve (14), as a result of which when the rivet (11) is urged against the sleeve (14) in vehicle acceleration, braking or sideslipping situations a greater force is required to push the rivet (11) into the tire rubber, however without arresting the movement of the rivet (11) within the sleeve (14).
Patent FI-862244-A (FI)
Inventor: ATABEKOV IOSIF GRIGORIEVICH
IPC: G01N33/543
Filed: 1986-05-27
Abstract: The procedure for determining an antigen comprises the production of a conjugate through cross-bonding of an anti-body with an inorganic pyrophosphate, transformation of the conjugate so obtained with the antigen - to be determined - bonded to the surface of a solid phase, separation of the solid phase from the liquid phase and transformation of one of the said phases with a substrate consisting of a salt of pyrophosphoric acid. After the reaction has been effected, a colour reagent is added to the resulting reaction mixture, which reagent contains a salt of molybdenic acid, a surfactant, malachite green and a strong inorganic acid. The antigen content is then determined on the basis of the optical density.
Patent FI-863269-A (FI)
Inventor: BRAENDLI MAX
IPC: B60B33/04
Filed: 1986-08-12
Abstract: This device prevents individual components of a load from being thrown off during halting of a conveying vehicle at a high rate of deceleration. A blocking device for the suspension of the caster which instantly assumes a front position as viewed in the direction of travel, prevents the vehicle from forwardly and downwardly dipping about the axle of the center-mounted drive wheels. The blocking device automatically adjusts itself corresponding to the direction of motion. A sliding stop vertically displaceably mounted on a pivotable part of a caster arrangement and a stop component fixedly mounted on the vehicle body cooperate to block the suspension of this front caster when the front caster experiences a predetermined degree of suspension displacement. At the caster instantly assuming the rear position, the stop component and the sliding stop are positioned at 180 DEG  to one another, thus precluding inadvertent engagement and permitting full suspension displacement. When changing direction of travel, both casters pivot automatically about a vertical axis, blocking the suspension of the front caster in the new direction of travel and permitting the rear caster to exploit its full suspension displacement range.
Patent FI-872284-A (FI)
Inventor: SCHNELL KARL
IPC: A22C11/02
Filed: 1987-05-22
Abstract: A machine for filling pasteous media, particularly sausage stuffing, into a hose-shaped sleeve, comprises a filling pump having a pressure side, a filling pipe for receiving a sausage sleeve and connected with the pressure side of the filling pump and having a free end, a braking ring arranged so that a medium is pulled through the sleeve between the braking ring and the free end of the filling pipe, an electrically controlled motor which intermittently drives at least the pump, and a microcomputer which controls the motor.
Patent FI-872753-A (FI)
Inventor: RUDOLPH RAINER
IPC: C12P21/00
Filed: 1987-06-22
Abstract: Method for activating non-glycosylated tissue plasminogen activator (t-PA) after its expression in prokaryotic cells comprises cell lysis; solubilisation under denaturing and reducing conditions, and reactivation under oxidising conditions in presence of reduced and oxidised glutathione (G5H, G55G). The new feature is that in the last stage is at pH 9-12 (pref. 9.5-11) with G5H and G55G concns. 0.1-20, pref. 0.2-10, mM and 0.01-3, pref. 0.5-1, mM, respectively, and with a non-denaturing concn. of the denaturing agent. Esp. the method is applied to t-PA expressed in E.coli and P. putida. The denaturing agent is pref. arginine, guanidine hydrochloride (both at 0.1-1, esp. 0.25-0.75, mM) or urea, at 0.5-4 (esp. 1-3.5) M in the last stage.
Patent FI-873021-A (FI)
Inventor: BUZAS ANDRE
IPC: C07D209/46
Filed: 1987-07-08
Abstract: Derivatives, of formula: 
<IMAGE>
 in which:
 R1, R2, R3 and R4 independently of each other denote a hydrogen atom, a halogen atom, a lower alkyl group, a lower alkoxy group or the trifluoromethyl group;
 n is an integer in between 1 and 6 inclusive;
 R5 and R6 denote, one a hydrogen atom and the other a substituted or unsubstituted benzoyl group; or
 R5 and R6 form, with the nitrogen atom to which they are bonded, a substituted or unsubstituted 5- or 6-membered heterocyclic group chosen from the following groups: succinimidyl, 4-phenylsuccinimidyl, phthalimidyl, naphthalimidyl, phthalimidinyl, 3-hydroxyphthalimidinyl, 2-oxobenzimidazolinyl, 3-benzyl-2-oxobenzimidazolinyl, 1,2,3,4-tetrahydro-2,4-dioxoquinazolinyl, 3,4-dihydro-4-oxoquinazolinyl, 3,4-dihydro-4-oxo-2-methylquinazolinyl, 3,7-dihydro-1,3-dimethyl-2,6-dioxo-1H-purinyl, 3,7-dihydro-3,7-dimethyl-2,6-dioxo-1H-purinyl. The invention also relates to processes for obtaining the said derivatives and to pharmaceutical compositions containing them. The said derivatives exhibit an antihistaminic activity without any sedative component.
Patent FI-873347-A (FI)
Inventor: MUTIKAINEN RISTO
IPC: H01G4/06
Filed: 1987-08-03
Abstract: This invention describes a method for manufacture of thin film capacitors, according to which method a bottom electrode film 2 is constructed on a substrate 1, a resist mask 3 is constructed on the bottom electrode film 3, which resist mask has openings 7 by which the capacitor area a is delimited, the layer of insulation 5 of the capacitor is constructed for each capacitor area either electrolytically or in gas phase, the counter electrode area b is delimited and the counter electrode 8 is constructed on each layer of insulation 5 by vacuum evaporation. According to the invention the capacitors are delimited by means of a lift-off lithographic resist mask 3 whereby the area of the cross-sectional surface of the lower part of each opening 7 which delimits the insulation layer 5 of the capacitor area is larger than the cross-sectional area b of the upper part which delimits the counter electrode area 8 and the perpendicular projection at the lower part of the opening of the cross-section of the opening's upper part falls within the lower part of the opening. By means of the method according to the invention the inspection of the counter electrode is carried out during self alignment. <IMAGE>
Patent FI-893725-A (FI)
Inventor: ZINNEN HERMANN A
IPC: C07C15/08
Filed: 1989-08-07
Abstract: Para-xylene is separated from other C8 isomers and/or C9 aromates by causing a mixture containing para-xylene to come into contact with an X or Y zeolite adsorbent whose exchangeable cation layer has been replaced with cations from Groups IA or IIA, e.g. barium and/or potassium. Para- xylene is adsorbed selectively by the adsorbent. The mixture is precipitated from the adsorbent and para- xylene is recovered from the resultant enriched adsorbent by desorption with diethyltoluene. The C8 components and other xylene isomers are typically recovered from the refined product containing desorbent and can be separated from this desorbent by fractionation of the raffinate, with the desorbent being returned to the process.
Patent FI-921179-A (FI)
Inventor: FEIGELSON GREGG BRIAN
IPC: C07F7/18
Filed: 1992-03-19
Abstract: New 4-substituted azetidinones having the formulae I and II: <CHEM> with R<1>, R<2>, R<3>, R<4>, R<5> and X defined hereafter, which are intermediates for the preparation of carbapenem and carbacephem antibacterials and processes for producing such antibacterials through the utilization of an acid mediated ring closure reaction.
Patent FI-923268-A (FI)
Inventor: PETERSEN UWE
IPC: A61K31/4709
Filed: 1992-07-16
Abstract: The invention relates to novel 8-vinyl- and 8-ethynyl- quinolonecarboxylic acids, a process for their preparation and antibacterial agents and feed additives containing them.
Patent FI-931172-A (FI)
Inventor: HEERTEN GEORG
IPC: E02B3/16
Filed: 1993-03-16
Abstract: Described is a process for the continuous production of a water- and/or oil-impermeable (impervious) liner (sealing matt) wherein expansive (swellable) clay is needled into between a carrier layer and a nonwoven top (cover) layer while at the same time an expansive clay additionally sprinkled onto the upper surface of the top layer is incorporated into the top layer. Subsequently the expansive clay present in the top layer is incipiently moistened and re-dried. A modified embodiment uses only a carrier layer made of a nonwoven, woven fabric or knitted fabric and/or a foil, the foil being a plastic film, a fabric-reinforced plastic film or paper, and a coarsely porous nonwoven or a non-consolidated crosslaid (fibre-crossed) card web or a random-laid fibre web, to which the pulverulent expansive clay is applied and needled in, moistened and dried. Instead of the needling technique it is also possible to use the knitting and/or sew-knitting technique.
Patent FI-932442-A (FI)
Inventor: CECCHIN GIULIANO
IPC: C08J5/18
Filed: 1993-05-28
Abstract: Crystalline polymers and copolymers of propylene having total MIL values > 2 g/10 minutes, total [ eta ] values in tetrahydronaphthalene at 135<o>C </= 2.8 dl/g, Mw/Mn values > 20, a fraction insoluble in xylene at 25<o>C >/= 94, and comprising from 10 to 60% by weight of a fraction (A) having [ eta ] >/= 2.6, are prepared by way of sequential polymerization in at least two stages, in the presence of particular Ziegler-Natta catalysts supported on magnesium halides. Said polymers have high melt strength, high mechanical properties, and are particularly adequate for the manufacture of articles by using various conversion technologies, such as for example extrusion in thin sheets to be subjected to thermoforming, as well as for injection molding, and blow molding.
Patent FI-934228-A (FI)
Inventor: KLAVENESS JO
IPC: A61K49/22
Filed: 1993-09-27
Abstract: Cross-linking agents containing or adapted to generate methylene diester or diamide groups of formula -(Z)m.Y.X.C(R<1>R<2>).X.Y.(Z)n- (where each X and Z is selected from -O-, -S- and -NR- (where R is hydrogen or an organic group); each Y is carbonyl, thiocarbonyl, sulphonyl, phosphoryl or a similar acid-forming group; m and n are each zero or 1; and R<1> and R<2> are each hydrogen, an organic group or a group -X.Y(Z)m-, or together form a divalent organic group) are useful in the preparation of substrates containing biodegradable cross-linking groups.
Patent FI-934301-A (FI)
Inventor: SCHOEPS MICHAEL
IPC: D06N5/00
Filed: 1993-09-30
Abstract: There is described a bituminised (bituminous) roofing underfelt (under-roofing felt, sarking, underslating felt) comprising a spunbonded (nonwoven) of polyester, in particular polyethylene terephthalate, filaments having a filament linear density (individual titre) of 1-8 dtex embedded in a bitumen matrix, characterised in that the weight of the bitumen accounts for 40 to 90%, and that of the spunbonded for 10 to 60%, of the basis weight of the roofing underfelt, and in that the spunbonded is consolidated by a meltable binder whose melting point is below the processing temperature of the bitumen used in making the bituminised roofing underfelt and which is present in the spunbonded in a weight proportion from 5 to 20% of the total weight. The spunbonded preferably bears an embossed pattern, for example a plain-weave embossment. There is also described a process for manufacturing the roofing underfelt and the spunbonded present therein.
Patent FI-940210-A (FI)
Inventor: FERRARO FRANK A
IPC: B26B21/14
Filed: 1994-01-14
Abstract: Segmented guard bar wherein segments of adjacent guard bars are tapered such that the skin flow through spaces between the segments is reduced. According to one preferred, illustrated embodiment, the distance between the rearward portion of adjacent segments is less than the space between the forward portions of those segments. Though not limited to any specific type of razor, the present invention is particularly suited for use with a flexible razor head having a cap member, at least one and preferably two blades separated by a spacer, a blade seat having a plurality of blade support portions separated by corrugations, and a segmented guard bar with each segment independently connected to the blade support portions.
Patent FI-941455-A (FI)
Inventor: DE SOETE GERARD
IPC: B01D53/56
Filed: 1994-03-29
Abstract: PCT No. PCT/EP92/02173 Sec. 371 Date Jun. 22, 1994 Sec. 102(e) Date Jun. 22, 1994 PCT Filed Sep. 18, 1992 PCT Pub. No. WO93/06916 PCT Pub. Date Apr. 15, 1993.A process for purifying a gas containing nitrogen monoxide to remove nitrogen monoxide therefrom, includes adjusting oxygen content of the gas to provide a quantity of oxygen which is at least equal to a stoichiometric quantity which is necessary in order to oxidize the nitrogen monoxide contained in the gas to nitrogen dioxide; contacting the gas, substantially in the absence of any liquid, with an alkali metal pyrosulphite which is a solid and which is employed in a quantity which is sufficient to convert the nitrogen monoxide contained in the gas to alkali metal nitrite and alkali metal nitrate; and removing the alkali metal nitrite and the alkali metal nitrate from the gas.
Patent FI-943545-A (FI)
Inventor: STADLER MONIKA
IPC: A61K35/16
Filed: 1994-07-28
Abstract: PCT No. PCT/EP93/00114 Sec. 371 Date Aug. 29, 1994 Sec. 102(e) Date Aug. 29, 1994 PCT Filed Jan. 20, 1993 PCT Pub. No. WO93/15105 PCT Pub. Date Aug. 5, 1993Described is an economical process for the recovery of factor VIII from blood plasma or cryoprecipitate. In the process, anion exchanger chromatography is conducted using a separating material based on carriers containing hydroxyl groups, the surfaces of which carriers have been coated with covalently boded polymers. The polymers contain repeating units represented by formula (I).    <IMAGE>
Patent FI-945412-A (FI)
Inventor: RUSSELL KEITH
IPC: A61K31/44
Filed: 1994-11-17
Abstract: Compounds of formula I    <IMAGE>  I  wherein X, A, B, R1 and R2 have the meanings given in the specification, and pharmaceutically acceptable salts and pharmaceutically acceptable in vivo hydrolysable ester thereof, processes for preparing the compounds and pharmaceutical compositions comprising them. The compounds are useful as potassium channel openers and as therapeutic agents in the treatment of urinary incontinence.
Patent FI-954539-A (FI)
Inventor: SAITO YUTAKA
IPC: A24B3/12
Filed: 1995-09-25
Abstract: A smoking article (10) contains a flavor component retainer obtained by heating and gelling a mixture of a flavor component and a non-gelled glucan and containing heat-irreversibly gelled glucan, and a flavor generation material containing the flavor component retained by this retainer as a combustion smoking raw material (12). Since the flavor component is firmly fixed and retained inside a three-dimensional network structure of gelled glucan, preservability and emission durability of the flavor component can be improved. <MATH>