baber/WOPTO huggingface dataset:
Patent IL-154743-A0 (IL)
Title: Boundary representation per feature methods and systems
IPC: G06F9/455
Filed: 2001-08-30
Abstract: Computer implemented methods and systems for CAD data exchange, and in particular for creating boundary representations ("breps") on a feature-by-feature basis are disclosed. According to an embodiment of the techniques described herein, a parameterized feature from a parametric based design system is exported from a source CAD system ( 404 ). Iterative steps and complimentary extraction techniques are employed by one or more processors ( 452, 456 ) to create an importable design model of the parameterized feature ( 433 ), which is imported into a target CAD system ( 408 ). While the techniques can include API ( 436 ), pattern matching ( 440 ), and user emulation ( 444 ) techniques, they include a brep per feature ( 450 ) technique. By exporting the brep on a per feature ( 453 ) basis from the source CAD system ( 404 ), the design intent of a CAD designer can be preserved on importation into the target CAD system ( 408 ). In particular, where a parametric representation ( 433 ) of the feature fails to import into the target system ( 408 ), an unparameterized representation ( 453 ) of the feature can be substituted.
Patent IL-156203-A0 (IL)
Title: Use of 2,2,3,3, tetramethylcyclopropane carboxylic acid derivatives for treating psychiatric disorders
IPC: A61P25/18
Filed: 2003-05-29
Abstract: The invention relates to the use of 2,2,3,3 tetramethylcyclopropane carboxylic acid derivative compounds for the preparation of a medicament for treating a psychiatric disorder preferably a bipolar disorder. The invention additionally relates to the use of the compounds for the preparation of an inhibitor of MIP synthase and to a pharmaceutical composition comprising the compounds for treating a psychiatric disorder. A method for treating a psychiatric disorder preferably a bipolar disorder and a method for inhibiting an enzyme having MIP synthase activity is provided.
Patent IL-163836-A0 (IL)
Title: Isostructural pseudopolymorphs of 9-deoxo-9A-aza-9-a-methyl-9A-homoerythromycin a
IPC: A61P33/02
Filed: 2003-03-18
Abstract: A substantially pure isostructural pseudopolymorph of 9-deoxo-9a-aza-9a-methyl-9a-homoerythromycin A having the Formula I:    
wherein S is an organic solvent which is at least partially miscible with water, x is 1, y is 0, 0.5, or 1, the pseudopolymorph being characterized by the monoclinic space group  P 2 1  and average unit cell parameters comprising: crystal axis lengths of a = 15.5 - 17.0 Å, b = 15.5 - 17.0 Å and c = 17.5 - 19.5 Å, and angles between the crystal axes of ± = ³ = 90° and ² = 106° - 112°.
Patent IL-172448-A0 (IL)
Title: Cartesian loop transmitter and method of adjusting an output level of such transmitter
IPC: H03F1/32
Filed: 2005-12-07
Abstract: A Cartesian loop transmitter having isolator eliminator circuitry is presented. The isolator eliminator circuitry includes a set of low pass and wide band pass as well as narrow band pass filters for each of I- and Q-channels, root mean square detectors and dividers connected to a means for comparing. Signals from the means for comparing are received by a microprocessor which controls attenuation setting. The output level of the transmitter is adjusted by generating a small signal measuring an on-channel signal level and a small signal level and then calculating a ratio of the small signal to the on-channel signal. The attenuation setting is increased if the ratio exceeds a defined threshold.
Patent IL-174826-A0 (IL)
Title: Antibodies to nik their preparation and use
IPC: C12N9/12
Filed: 2006-04-06
Abstract: An antibody or antibody fragment preparation being capable of specifically binding the amino acid sequence 60-76, 86-98, 135-149, 215-227, 363-377, 385-397, 405-419, 427-440, 509-522, 605-619, 635-649, 666-680, 696-711, 752-766, 836-851, 871-884, and/or 904-916 of NIK, or being capable of specifically binding a specific portion of the amino acid sequence is provided.
Patent IL-176547-A0 (IL)
Title: 1,3,5-trisubstituted 4,5-dihydro-1h-pyrazole derivatives having cb1-antagonistic activity
IPC: C07D231/06
Filed: 2006-06-26
Abstract: The present invention relates to 1,3,5-trisubstituted 4,5-dihydro-1 H-pyrazole derivatives as CB1 antagonists, to methods for the preparation of these compounds and to novel intermediates useful for the synthesis of said pyrazole derivatives. The invention also relates to the use of a compound disclosed herein for the manufacture of a medicament giving a beneficial effect. The compounds have the general formula (I) wherein the symbols have the meanings given in the specification.
Patent IL-181247-A0 (IL)
Title: Composition and method for improved bioavailability and enhanced brain delivery of 5,5-diphenyl barbituric acid
IPC: A61K31/515
Filed: 2007-02-08
Abstract: The present invention relates to a composition and a method of delivering a barbituric acid derivative to the central nervous system of a mammal in need of treatment for neurological conditions. In particular, the present invention relates to a method of administering an oral dosage form of a sodium salt of 5,5-diphenyl barburtic acid to enhance the bioavailability of 5,5-diphenyl barbituric acid and brain delivery of same.
Patent IL-183449-A0 (IL)
Title: Process for the preparation of carvedilol and its enantiomers
Filed: 2007-05-28
Abstract: The present invention relates to a process for the preparation of carvedilol as well as of the optically active R and S enantiomers thereof and of mixtures of these enantiomers and, more particularly, relates to an improved process for the preparation of carvedilol and its enantiomers characterized by the use of ethyl acetate as reaction solvent.
Patent IL-239024-A0 (IL)
Title: Method and apparatus for providing timing alignment
IPC: H04W74/08
Filed: 2015-05-27
Abstract: An approach includes generating a control message having a format designated for resource allocation, wherein the control message includes a plurality of control fields. One of the control fields is reserved to specify information other than information for resource allocation, the value indicating timing alignment information or information for starting a random access procedure. The control message is transmitted over a control channel according to a lower layer protocol.
Patent RO-126103-A0 (RO)
Title: Metal form sealing system
Inventor: SECĂREANU ION
IPC: B28B7/02
Filed: 2010-10-29
Abstract: The invention relates to a system for sealing metal forms used for manufacturing various elements of gas formed concrete. According to the invention, the system comprises a base plate (1), side walls (2) and covers (3), on the outline of the base plate (1) there is welded a convex metal profile (4), having the cross-section in the shape of an equilateral trapezium, on which the side walls (2) are placed perpendicularly, said walls having welded at their lower part another concave trapezium shaped metal profile (5), inside the concave profile (5) a recess (b) is worked, wherein a rubberized seal (6) is mounted for sealing and wherein the side walls (2) of the form (F) are compressed on the base plate (1) by means of some clamping screws (7) also ensuring the guiding of the concave profile (5) onto the convex profile (4).
Patent RO-135099-A0 (RO)
Title: Anti-fogging device
Inventor: LUPU SEBASTIAN
IPC: A62B23/02
Filed: 2020-10-14
Abstract: The invention relates to an anti-fogging device for glasses, mounted on a protective mask meant to protect the user's face from contamination, over which the pair of glasses is put. According to the invention, the device is made of a biodegradable plastic, such as polylactic acid, and it consists of a nose support (1) of round or oval shape, having a variable radius (R) depending on the user's face and body size, which has in the upper part a reinforcement (2), the nose support (1) being symmetrically continued in the lateral sides with some arms (3 and 4), namely a vertical arm (3) on each lateral side, continued with a horizontal arm (4), the arms (3 and 4) having a U-shaped profile and meeting in an angle (β) which varies from 90° to 120°, the U-profile of the arms (3 and 4) having a thickness (g) of 1...1.5 mm and being provided with two spurs (5) at the top of the U profile, for attaching the protective mask, the two lateral sides of the U-shaped profile being arranged under an angle (α) which varies between 0° and 30°.
Patent RO-135877-A0 (RO)
Title: Device for tracing centroids of non-circular spiral toothed wheels with digital angle measurement
Inventor: BOGDAN-ROTH MIHAIL
IPC: B23F17/00
Filed: 2022-01-21
Abstract: The invention relates to a device for tracing the centroids of non-circular spiral toothed wheels, namely the head, indexing and flank centroids, with digital angle measurement. According to the invention, the device consists of a disc (1) on which a paper disc of the same diameter is fixed, on which the concerned spiral will be traced, the value of the angle α is fixed on a digital screen (12) by locking the protractor arm (6) with a screw (8), the slide (11) is fixed with the zero mark in the apex of the angle formed by the two arms of the protractor, the tip of a pencil is inserted in the channel of the slide (11) and the disc (1) is moved laterally over an interval Φ=0...2, together with the pencil tip, up to the start circle which sets the spiral set (S), the shape of the corresponding spiral being automatically obtained on the disc, after which the disc (1) is removed from the shaft (4) and the so-obtained spiral is used together with the data.
Patent AP-2003002901-A0 (AP)
Title: Use of HIV-protease inhibitors to block cell migration and/or invasion, tissue infiltration and oedema formation
Inventor: ENSOLI BARBARA
IPC: A61K31/341
Filed: 2002-04-18
Abstract: The present invention relates to a method to block the invasion of normal, neoplasticor immune cells, tissue infiltration, and/or oedema formation through inhibition or modulation of molecules and proteolytic enzymes such as -but not exclusively-MMPS, for the therapy of all diseases whose pathogenesis is related to the above processes, including tumours, non-neoplastic angioproliferative diseases, inflamatory diseases, or autoimmune diseases, the method being based on the use of inhibitors of the protease of the protease of the HIV virus(HIV-PI)
Patent CU-21829-A1 (CU)
Title: Composicion de grasas de conservacion temporal
Inventor: ECHEVERRIA LAGE CARLOS A
IPC: C08L91/00
Filed: 1985-03-21
Abstract: Los compuestos de conservación temporal, se emplean en la protección anticorrosiva de piezas, equipos, accesorios, materiales metálicos, etc. en las etapas de elaboración, transportación y almacenamiento. La invención persigue la obtención, a partir de materia prima de bajo costo, de compuesto constituidos por cebo de res, grasa de calcio, hidrato de calcio tipo A, cemento Portland-250, cera cruda de abejas y cera cruda de cana de azúcar en forma de pasta o en forma líquida con un solvente adecuado, los cuales garantizan una fácil aplicación y desconservación, resisten la acción de la atmósfera con influencia salina, la lluvia y mejoran sus propiedades protectoras bajo el efecto de la radiación solar, proporcionando un compuesto duro y resistente, que permiten la protección a la intemperie en períodos de seis meses a un ano. Encuentran amplia aplicación en diferentes ramas de la economía, en almacenes, equipos, maquinarias, piezas, etc.
Patent IE-910171-A1 (IE)
Title: New thiazole derivatives
IPC: A61K31/425
Filed: 1991-01-18
Abstract: New thiazole derivatives which are a substituted 4- or 5-( omega -aminoalkyl)thiazole with formula (1), wherein X represents a nitrogen atom and Y represents a sulphur atom or alternatively X represents a sulphur atom and Y represents a nitrogen atom, n is 1-6, R1 represents a straight or branched alkyl group containing 1-4 carbon atoms and R2 represents an amino group, a process for the preparation of said compounds by ring closure of a 3-bromo- omega -phthalimidoalkan-2-one with thiourea under mild conditions, followed by hydrazinolysis or hydrolysis with diluted hydrochloric acid of the resulting phthalimido derivatives and medicaments containing said derivates with formula (1) for the treatment of congestive heart diseases or for the treatment of allergic disorders.
Patent IE-910267-A1 (IE)
Title: Transdermal therapeutic system comprising tulobuterol as active substance
Inventor: HOFFMANN DR HANS-RAINER
IPC: A61L15/44
Filed: 1991-01-25
Abstract: The invention relates to a transdermal therapeutic system containing tulobuterol or one of its pharmaceutically compatible salts as active ingredient, comprising a backing layer which is essentially impermeable to active ingredient, and at least one matrix layer which contains the active ingredient and contains at least one styrene/1,3-diene/styrene block copolymer, and to a process for the production thereof.
Patent MA-22520-A1 (MA)
Inventor: PS JUNEJA
IPC: A61K8/86
Filed: 1992-05-06
Abstract: Antiperspirant compositions in the form of gel sticks, which provide the user with excellent antiperspirant efficacy while exhibiting good stability, are disclosed. Specifically, the compositions have an acidic pH and include an antiperspirant active, a gelling agent which comprises dibenzylidene alditols, a solvent for the gelling agent, and a gelling agent stabilizer which is a basic metallic salt of an acid having a pKa of from about 3.8 to about 6.5 at 25 DEG  C, said salts being at least partially soluble in the composition, and said stabilizer being a salt selected from the group consisting of C4-C6 alkyl dicarboxylates, C6-C8 alkyl monocarboxylates, and substituted and unsubstituted benzoates, and mixtures thereof, wherein said gelling agent stabilizer does not contain amino or amido functionalities. Methods of preventing and controlling perspiration wetness using these compositions and of making the compositions are also disclosed.
Patent MA-37510-A1 (MA)
Title: Surfactant derive du quinolinium pour la modification d'argile
Inventor: BOUHFID RACHID
IPC: C07D215/00
Filed: 2014-11-11
Abstract: Un nanocomposite fi base d’un polymère thermoplastique et d’argile modifiée par un surfactant de la famille de d’alkyl styryl quinolinium ayant une bonne stabilité thermique et des priopriétés mécaniques améliorées.
Patent MA-40654-A1 (MA)
Title: Capteur solaire
Inventor: SCHILDER JOHANNES JACOBUS MARIA
IPC: F24S23/30
Filed: 2014-12-19
Abstract: L'invention concerne un capteur solaire 1 pour le stockage temporaire de chaleur provenant d'un rayonnement solaire, comprenant un conducteur de rayonnement 8, 9 pour conduire le rayonnement solaire, et un moyen de lentille 7 pour concentrer le rayonnement solaire sur une première extrémité du conducteur de rayonnement. Une âme thermiquement isolée 2 est ménagée sur une seconde extrémité opposée du conducteur de rayonnement 8, 9 afin d'être chauffée par le rayonnement solaire libéré du conducteur de rayon
Patent MA-42169-A1 (MA)
Title: Machine de rainurage à came
Inventor: DOLE DOUGLAS
IPC: B21H1/22
Filed: 2016-11-22
Abstract: La présente invention concerne un dispositif de formage à froid d'éléments de tuyau doté de deux cames ou plus, chacune des cames ayant un engrenage qui s'engrène avec un pignon qui fait lui-même tourner l'ensemble des cames. Chacune des cames présente une surface de came incluant une région de rayon croissant et peut comporter une zone de rayon constant s'étendant autour d'un corps de came. Chacune des cames présente également une surface de traction s'étendant autour d'un corps de came. Une discontinuit
Patent UY-24347-A1 (UY)
Title: Procedimiento y aparato para tejer genero de punto con hilo no elastico e hilo elastomerico sin recubrir y construccion de genero de punto para sweaters
Inventor: BRACH ERNESTO
IPC: D04B1/00
Filed: 1996-10-11
Abstract: Género de punto para sweaters que contiene hilado duro entretejido junto con hilado elastomérico sin recubrimiento. El mismo se realiza mediante un proceso en el cual el hilado elastomérico sin recubrimiento se suministra bajo una tensión que varía menos del 17%, a una máquina de tejer en la cual la demanda de hilo fluctúa a medida que se teje el género. Es un género que se teje en una máquina de tejer en tiras o bandas circular o en una maquina de tejr en tiras o bandas rectilineas. Estas máquinas de tejer, insertan un hilo separador entre las bandas o tiras tejidas y/o tejen un borde terminado, por ejemplo pretina o un puño, al comienzo de la tira o banda de sweter. Cuando la tension del hilo se mantiene constante durante el tejido, el règimen de alimenacion de hilado es igual a la momentaria de manda de hilado elastomérico de la máquina de tejer.
Patent UY-28483-A1 (UY)
Title: Derivados de naftiridina sustituidos como inhibidores del factor inhibidor de la migración de macrófagos y su uso en el tratamiento de enfermedades en el hombre
Inventor: SIRCAR JAGADISH
IPC: A61P37/06
Filed: 2004-08-20
Abstract: Se proveen inhibidores del factor inhibidor de la migración de macrófagos (MIF) con una estructura principal de naftiridina que son de utilidad en el tratamiento de una variedad de trastornos, incluyendo el tratamiento de afecciones patológicas asociadas con la actividad del MIF. Los inhibidores del MIF tienen las siguientes estructuras: que incluyen estereoisómeros, prodrogas y sales aceptables para uso farmacéutico de los mismos, donde n, R,R1, R2, X, Y y Z tienen los valores que se definen en la memoria descriptiva. También se proveen composiciones que contienen un inhibidor de MIF en combinación con un vehículo aceptable para uso farmacéutico, así como métodos para utilizarlos.
Patent UY-29240-A1 (UY)
Title: Nuevos derivados de piridotienopirimidina
Inventor: FERRER JORDI GRACIA
IPC: C07D311/00
Filed: 2005-11-29
Abstract: Nuevos derivados de piridotienopirimidina terapéuticamente útiles, procedimientos de preparación de los mismos y composiciones farmacéuticas que los contienen. Estos compuestos son inhibidores potentes y selectivos de las fosfodiesterasas 4(PDE4) y, por tanto, son útiles en el tratamiento, prevención o supresión de estados patológicos, enfermedades y trastornos que se sabe son susceptibles de mejorar por la inhibición de la PDE4.
Patent UY-29809-A1 (UY)
Title: Detector de fase para equipos rotativos
Inventor: CHENG CHENG GI
IPC: F15B11/22
Filed: 2006-09-26
Abstract: Se describe un sistema muy preciso para detectar la fase de rotación que está conformado por dos discos primero y segundo codificados con una secuencia pseudorrandómica de 31 dígitos, donde los discos primero y segundo están unidos a los miembros que están acoplados en su rotación. La codificación se logra dividiendo los discos en 31 secciones a lo largo del contorno de la periferia de los discos, de forma tal que las secciones correspondientes a 1 tienen un radio más largo y las secciones correspondientes a 0 tienen un radio menor.
Patent UY-31135-A1 (UY)
Title: Derivados de piperidina/piperazina (ii)
Inventor: DAVIDENKO PETR VLADIMIRIVICH
IPC: A61K31/495
Filed: 2008-06-09
Abstract: La invención se refiere a un inhibidor de DGAT de fórmula incluyendo sus isómeros estereoquímicos, donde A representa CH o N; la línea punteada representa un enlace opcional en caso que A sea un átomo de carbono; salvo que si X representa -O.C(=O)-, entonces r2 representa R3, excluyendo un N-óxido o una sal farmacéuticamente aceptable o un solvato de los mismos. También se refiere a métodos para preparar tales compuestos, a composiciones farmacéuticas y al uso como medicamentos de dichos compuestos.
Patent ES-150883-A1 (ES)
Title: UN PROCEDIMIENTO PARA LA OBTENCIoN DE N-SULFONILUREAS
Filed: 1940-11-15
Abstract: Propiedad y explotación exclusivas de un procedimiento para la obtención de N-sulfonilureas aromáticas de la fórmula siguiente: Aril-SO2-NR1-CO-NH-R2 caracterizado por hacerse actuar sobre sulfonilamidas aromáticas primarias o secundarias de la fórmula general Aril-SO2-NH-R1 derivados del ácido ciánico o isociánico de la fórmula (CON)-R2 o sus salesy respectivamente aquellos compuestos o sus sales de los cuales pueden producirse durante la reacción como productos intermedios los mencionados derivados del ácido ciánico o isociánicoteniendo los símbolos el significado siguiente: Aril= núcleo aromático sustituido o no sustituido o un sistema cíclico aromático. R1 y R2= hidrógenoalquiloaralquilo o arilo.
Patent ES-179746-A1 (ES)
Title: Mejoras introducidas en sistemas de moduladores
IPC: H03K7/08
Filed: 1947-09-16
Abstract: Mejoras en sistemas demoduladores caracterizados por un método para demodular un tren de impulsos cuyos impulsos están modulados en ancho de acuerdo con una señal de tipo audio determinada caracterizado a su vez por las etapas de convertir los impulsos modulados en ancho en ondulaciones cuyo ancho sea sustancialmente constante y cuya amplitud varíe como modulación respectiva en ancho de los referidos impulsos y producir una envolvente de tipo audio de las referidas ondulaciones moduladas en amplitud.
Patent ES-180753-A1 (ES)
Title: UN SISTEMA DE CONDENSADOR ELÉCTRICO PERMANENTE IMPERFORABLE, SoLIDO, ANTIELECTROLiTICO
Filed: 1947-12-03
Abstract: Sistema de condensador eléctrico permanente imperforable sólido antielectrolítico, caracterizado fundamentalmente por descarga interna amortiguada del condensador contra la perforación, por la sustitución de la hoja de estaño o aluminio laminada, usada corrientemente, por una finísima película semiconductora de elevada resistencia eléctrica, transmisora del potencial eléctrico, adherida al dieléctrico para imposibilitar la perforación del condensador eléctrico, (según figura 1, 2, 3, 4 y descripción correspondiente).
Patent ES-191862-A1 (ES)
Title: MEJORAS INTRODUCIDAS EN LAS MáQUINAS PARA ASERRAR BLOQUES DE PIEDRA, MáRMOL Y SIMILARES, IMPRIMIENDO A LOS ELEMENTOS CORTANTES UN MOVIMIENTO RECTILiNEO DE VAIVÉN.
Filed: 1950-02-27
Abstract: Mejoras introducidas en las máquinas para aserrar bloques de piedramármoles y similaresimprimiendo a los elementos cortantes un movimiento rectilíneo de vaivéncaracterizadas por el hecho de que como hojas cortantes se emplean unas tiras metálicasguarnecidas por una por sucesión de pastilla de material abrasivodirectamente moldeado sobre unos salientes determinados por el dentado de una de las aristas de dichas tiraslas cuales se disponen paralelamente dentro de un marco o bastidorque está dotado de un movimiento rectilíneo de vaivénen sentido horizontalcombinado con otro movimiento de descenso paulatino del conjunto del marcoa fin de que las pastillas de material abrasivoque constituyen el medio directo para producir el corteno pierdan contacto con el bloque en nigún momento de su trayectoria horizontallo que permite el máximo aprovechamiento del trabajo desarrollado y por lo tanto un rápido aserrado del bloque.
Patent ES-192784-A1 (ES)
Title: Un procedimiento de fabricacion de flores y ramilletes artificiales
Filed: 1950-05-03
Abstract: Procedimiento de fabricación de flores y ramilletes artificiales caracterizado por que las corolas se obtienen por cocción en hornos de reverbero o eléctricos de una pasta formada por barro de kaolin a la que se ha dotado a mano de la forma de una corola floral constituida por pétalos.
Patent ES-292681-A1 (ES)
Title: Menadione bisulfite adducts of dicyanodiamidine-2, 4, 6-triamino-1, 3, 5-triazine and pyrimidines substituted at the two positions and feeds
IPC: C07D251/70
Filed: 1963-10-19
Abstract: The invention comprises a menadione-bisulphite derivative having Vitamin K activity, low solubility in water, containing no water of crystallization, and giving rise to a saturated aqueous solution with a pH value below 4.5. The derivative may be obtained by reacting an aqueous solution of an addition compound of menadione and a bisulphite, e.g. sodium bisulphite, with a solution of a base containing the group <FORM:1002503/C2/1> where R1 is OH, NH2 or SH, or by reacting menadione with an aqueous solution of the bisulphite salt of the base. In examples compounds are prepared by reacting menadionesodium bisulphite with dicyanodiamidinium sulphate, 2,3,6-triamino-1,3,5-triazine, 2,4-diamino-6-hydroxy-pyrimidine, 2-hydroxy-4,6-dimethyl-pyrimidinium sulphate and 2-amino-4,6-dimethyl-pyrimidine.