Patent DE-102008041214-A1 (DE)
Title: New N-substituted azinylalkyl-azincarboxamide compounds useful e.g. in plant protection, for combating animal pests, arthropods, nematodes and plant diseases, and for protecting industrial materials against attack and destruction by insect
Inventor: FRACKENPOHL JENS
IPC: A01N43/40
Filed: 2008-08-13
Abstract: N-Substituted azinylalkyl-azincarboxamide compounds (I), and their analogs, salts and N-oxides are new. N-Substituted azinylalkyl-azincarboxamide compounds of formula (I), and their analogs, salts and N-oxides are new. X : O or S; A 1>-A 4>N or C-Y 1>, provided that more than two N atoms are not in adjacent position; A 5>CH or N; either Y 1>1-8C alkyl, 1-8C haloalkyl, 1-8C alkoxy, 1-8C alkylthio, 1-8C alkylsulfinyl, 1-8C alkylsulfonyl, 1-8C alkylamino, di(1-8C)-alkylamino, (hetero)aryl or heterocyclyl (all optionally substituted), H, nitro, amino, CN or halo; or two adjacent Y 1>5- to 6-membered ring system; R 2>H or 1-8C alkyl, 1-8C alkyl 3-7C cycloalkyl, 4-9C spirocycloalkyl or 1-8C alkoxycarbonyl (all optionally substituted); and R 1>1-8C alkyl, 3-7C cycloalkyl, 1-8C alkyl(3-7C)-cycloalkyl, 3-10C alkylalkenyl, 2-9C alkenyl, 2-9C alkylcarbonyl, 4-8C cycloalkylcarbonyl, arylcarbonyl, 1-8C alkoxycarbonyl, 1-8C alkylsulfonyl, arylsulfonyl, 1-6C-alkoxy-carbonylcarbonyl, aryloxycarbonyl-carbonyl, 1-8C alkylamino-thiocarbonyl, 3-7C cycloalkylaminothiocarbonyl, -C(=O)-cyclobutane, -C(=O)-(CH 2) 2-CH 3, -C(=O)-CH(CH 3) 2, -C(=O)-(CH 2) 4-CH 3, -C(=O)-(CH 2) 5-CH 3, -C(=O)- cyclohexane, -C(=O)-CH 2-CH 3, -C(=O)-cyclopentane, -C(=O)-(CH 2) 3-CH 3, chloro-phenyl groups of formula (Q-10) or (Q-11), -C(=O)-O-CH 2-CH(CH 3) 2, -C(=O)-O-CH 2-CH 3, -C(=O)-O-(CH 2) 2-O-CH 3, -C(=O)-CH 2-CH(CH 3) 2, -C(=O)-O-CH 2-Ctriple boundCH, -C(=CH-CH(CH 3) 2)(O-C(=O)-CH 2-CH(CH 3) 2), -C(=O)-cyclopropane, -C(=O)-O-CH 2-phenyl, -C(=O)-O-(CH 2) 2-CH 3, -C(=O)-O-CH 2-Ctriple boundC-CH 3, phenyl group of formula (Q-22), -C(=O)-O-CH 2-CH(Cl) 3, cyclopropane group of formula (Q-24), -C(=O)-O-CH(CH 3) 2, -C(=S)-O-phenyl, -C(=O)-C(CH 3) 3, -C(=O)-O-CH 3, adamantane group of formula (Q-29), dimethyl-cyclopropane group of formula (Q-30), 2,4-dichlorobenzene group of formula (Q-31), trifluoromethyl-benzene group of formula (Q-32), methyl-benzene group of formula (Q-33), methoxy-benzene group of formula (Q-34), 3,4-dichlorobenzene group of formula (Q-35), fluorobenzene group of formula (Q-36), biphenyl group of formula (Q-37), cyclopropane groups of formula (Q-38)-(Q-44), -C(=O)-CH 3, -CH 2-CH=CH 2, -(CH 2) 2-CH 3, -CH 2-CH 3, cyclopropane group of formula (Q-49), phenyl groups of formula (Q-50) or (Q-51), cyclopropane groups of formula (Q-52)-(Q-55), -(CH 2) 5-CH 3, phenyl groups of formula (Q-57) or (Q-58), -S(=O) 2-CH 3, phenyl groups of formula (Q-60)-(Q-66), -C(=O)-C(=O)-O-CH 2-CH 3, -(CH 2) 3-CH 3, -(C=O)-O-(CH 2) 2-CH(CH 3) 2, -C(=O)-O-CH 2-C(=CH 2)-CH 3, -C(=O)-O-CH 2-CH=CH 2, phenyl groups of formula (Q-72)-(Q-74), -C(=O)-O-C(CH 3) 3, phenyl groups of formula (Q-76)-(Q-80), -C(=S)-NH-cyclopropane, -C(=S)-NH-CH 2-cyclopropane, -C(=S)-NH-CH 2-CH 3, -CH 2-CH(CH 3) 2, -CH 2-cyclopropane, -(CH 2) 2-CH=CH 2, CH 3or phenyl group of formula (Q-84). [Image] [Image] [Image] [Image] [Image] [Image] [Image] [Image] [Image] [Image] ACTIVITY : Plant Protectant; Arthropodicide; Nematocide; Insecticide; Antifouling; Arachnicide; Acaricide; Antiparasitic; Antihelmintic; Protozoacide. MECHANISM OF ACTION : None given.