baber/WOPTO huggingface dataset:
Patent IL-179679-A0 (IL)
Title: Fluid permeable composite material and process for same
IPC: C08L33/10
Filed: 2006-11-28
Abstract: A fluid permeable material is disclosed. The fluid permeable material is suitable for use as a paver, brick, tile, stormwater entry grate and the like, without being limited thereto. The fluid permeable material described in this invention is light weight and has a height characteristic breaking strength, and flexural strength. The fluid permeable material described allows fluid to flow freely through the structure without impacting on the structural integrity of the composite material, and filters particulate contaminants from the fluid as it passes through the structure.
Patent IL-182744-A0 (IL)
Title: Epothilone derivatives and their synthesis and use
IPC: A61P43/00
Filed: 2007-04-23
Abstract: The invention relates to epothilone analog represented by the formula I   
wherein 
(i)  R 2   is absent or oxygen;  "a"  can be either a single or double bond;  "b"  can be either absent or a single bond; and  "c"  can be either absent or a single bond, with the proviso that if  R 2   is oxygen then  "b"  and  "c"  are both a single bond and  "a"  is a single bond; if  R 2   is absent then  "b"  and  "c"  are absent and  "a"  is a double bond; and if  "a"  is a double bond, then  R 2 , "b"  and  "c"  are absent;  R 3   is a radical selected from the group consisting of hydrogen; lower alkyl; -CH=CH 2 ; 
-C¡CH; -CH 2 F; -CH 2 CI; -CH 2 -OH; -CH 2 -O-(C 1 -C 6 -alkyl); and -CH 2 -S-(C 1 -C 6 -alkyl);  R 4   and  R 5   are independently selected from hydrogen, methyl or a protecting group; and  R 1   is as defined in the specification, or a salt of a compound of the formula I where a salt-forming group is present. A further aspect of the invention is related to the synthesis of epothilone E.  These compounds have inter alia microtubuli depolymerisation inhibiting activity and are e.g. useful against proliferative diseases.
Patent IL-185164-A0 (IL)
Title: New isothiazoloquinolones and related compounds as anti-infective agents
Filed: 2007-08-09
Abstract: The invention provides certain compounds and salts of Formula I and Formula II: which possess antimicrobial activity. The invention also provides novel synthetic intermediates useful in making compounds of Formula I and Formula II. The variables A1, R2, R3, R5, R6, R7, A8 and R9 are defined herein. Certain compounds of Formula I and Formula II disclosed herein are potent and selective inhibitors of bacterial DNA synthesis and bacterial replication. The invention also provides antimicrobial compositions, including pharmaceutical compositions, containing one or more compounds of Formula I or Formula II and one or more carriers, excipients, or diluents. Such compositions may contain a compound of Formula I or Formula II as the only active agent or may contain a combination of a compound of Formula I or Formula II and one or more other active agents. The invention also provides methods for treating microbial infections in animals.
Patent AP-2001002143-A0 (AP)
Title: Substituted benzopyran analogs for the treatment of inflamation
Inventor: CARTER JEFFREY S
IPC: C07D335/06
Filed: 1999-10-15
Abstract: A class of benzopyrans, benzothiopyrans, dihydroquinolines, dihydronaphthalenes, and analogs thereof, is described for use in treating cyclooxygenase-2 mediated disorders. Compounds of particular interest are defined by formula (i')wherein x, a1, a2, a3, a4, r, r
Patent IE-910885-A1 (IE)
Title: Metering device
IPC: G05D11/00
Filed: 1991-03-15
Abstract: A metering apparatus has a filling cylinder (69) which can be filled via a closable filling channel (88) and can be emptied via a metering channel (87) by means of a displaceable piston (72). A filling device (80) can be rotated about an approximately horizontal axis together with the reservoir container. It releases the filling channel (88) in a first rotational position in which the reservoir container is in an upper position and closes it in a second rotational position in which the reservoir container assumes a lower position. Such a metering apparatus is convenient to handle. Furthermore, it is ensured that when the filling channel (88) is closed, no metering agent passes into the filling cylinder (69). In particular, such a metering apparatus is suitable for a device for cleaning pipelines, such as lines for beverages. 
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Patent LU-84252-A1 (LU)
Title: IR-emitting, high luminous-transmitting glazing material - comprises transparent sheet coated with a conductive metal oxide layer and a dielectric layer
Inventor: ISRAEL JACQUES S
IPC: E06B5/12
Filed: 1982-07-02
Abstract: Glazing material comprises a light-transmitting sheet overcoated with a conductive metal oxide layer (I) and a dielectric layer (II) of thickness not above 160 nm. The sheet and (I) alone would have a luminous transmissivity of at least 70%.
Patent LU-87310-A1 (LU)
Inventor: MAIGNAN JEAN
IPC: C07C323/25
Filed: 1988-08-04
Abstract: An N-(mercaptoalkyl) omega -hydroxyalkylamide having the formula, <IMAGE>   wherein n is 2 or 3 and m is 2 to 5 inclusive is employed as a reducing agent in the first stage reducing operation of permanently deforming hair.
Patent MA-23658-A1 (MA)
Inventor: MICHAEL EUGENE BURNS
IPC: C11D7/54
Filed: 1995-08-30
Abstract: Bleaching compositions, laundry and automatic dishwashing detergent compositions comprising particular neutral or anionically charged substituted bleach activators are provided. More specifically, the invention relates to compositions which provide enhanced cleaning/bleaching benefits through the selection of perhydrolysis-selective bleach activators having specific leaving groups with a conjugate acid pKa above 13 and with specific ratios of the rate of perhydrolysis to the rate of hydrolysis and the rate of perhydrolysis to the rate of diacylperoxide production. Included are preferred activator compounds and methods for washing fabrics, hard surfaces, and tableware using the activators.
Patent MA-27055-A1 (MA)
Title: 2-(3,5-bis-trifluoromethyl-phenyl)-n-[6-(1,1-dioxy-1 6-thiomorpholine-4-yl)-4-(2-methyl ou 4-fluoro-2-methyl substitue) phenyl-pyridine-3-yl]-n-methyl-isobutyramide
Inventor: BALLARD THERESA MARIA
IPC: A61P37/08
Filed: 2004-01-30
Abstract: 2- (3, 5-BIS-TRIFLUOROMETHYL-PHENYL) -N- [6- (1, 1-DIOXO-1(lambda),6-THIOMORPHOLIN-4-YL)-4-PHENYL (SUBSTITUE EN 2-METHYL OU EN 4-FLUORO-2-METHYL)-PYRIDIN-3-YL]-N-METHYL-ISOBUTYRAMIDE L'invention concerne les composés de 2-(3,5-bis-trif luorométhyl-phényl ) -N- [6- ( 1, 1-dioxo-1(lambda)-6-thiomorpholin-4-yl)-4-o-tolyl-pyridin-3-yl]-N-méthyl-isobutyramide et de 2-(3,5-bis-trifluorométhyl-phényl)-N-[6-(1, 1-dioxo-(lambda)-thiomorpholin-4-yl) -4- (4-fluoro-2-méthyl-phényl)-pyridin-3-yl]-N-méthyl-isobutyramide qui peuvent être utilisés pour le traitement de la migraine, de la polyarthrite rhumatoïde, de l'asthme, de l'hyperréactivité bronchique, de la maladie inflammatoire du côlon ou pour le traitement de troubles comprenant la maladie de Parkinson, l'anxiété, la dépression, la douleur, les céphalées, la maladie d'Alzheimer, la sclérose en plaques, l'dème, la rhinite allergique, la maladie de Crohn, des lésions oculaires, des maladies oculaires inflammatoires, la psychose, le mal des transports, les vomissements provoqués, les vomissements, l'incontinence urinaire, des troubles psycho-immunologiques ou psychosomatiques, le cancer, les symptômes de sevrage de drogues engendrant une toxicomanie, des opiacés ou de la nicotine, des lésions cérébrales traumatiques ou l'hyperplasie bénigne de la prostate.
Patent MA-38078-A1 (MA)
Title: Dérivé de pyridine
Inventor: MARUYAMA AKINOBU
IPC: C07D409/14
Filed: 2013-11-13
Abstract: Dérivé de pyridine représenté par la formule (i), promédicament de celui-ci, sel pharmaceutiquement acceptable du dérivé de pyridine ou du promédicament, ou solvate du dérivé de pyridine, du promédicament ou du sel pharmaceutiquement acceptable, qui est utile pour traiter ou prévenir les maladies associées à urat1 telles que la goutte, l'hyperuricémie, l'hypertension, les maladies rénales telles que la néphrite interstitielle, le diabète, l'artériosclérose et le syndrome de lesch-nyhan.
Patent UY-25422-A1 (UY)
Title: Plataforma flotante para aparato recolector de energia radiante
Inventor: ALLAN JAMES YEOMANS
IPC: F24S90/00
Filed: 1999-03-10
Abstract: Método y los medios para sostener a flote el aparato recolector de energía solar en un fluido que será fiable y eficaz en uso. La invención en un aspecto preferido tiene como objetivo establecer una disposición que permita la flotación de las boyas para que sean mantenidas o incrementadas en caso de perdida de flotación. El aparato recolector de energía radiante comprende un montaje de plataforma que flota sobre una extensión de líquido, cuya parte superior sostiene reflectores de concentradores solares y cuya parte inferior consta de una serie de compartimientos abiertos en sus lados más inferiores que contienen aire para hacer subir la boya para mantener los reflectores sobre el nivel de líquido. El aire puede ser suministrado a los compartimientos por un conducto de aire debajo del montaje de la plataforma, el conducto consta de un número de aberturas por donde pasa el aire.
Patent UY-27123-A1 (UY)
Title: Utilización de cromanos
Inventor: GERLACH DR IRENE
IPC: A61P25/16
Filed: 2002-01-14
Abstract: La presente invención se refiere a la utilización del 1,1-dioxido de 2-(4-(2R)-8- isopropoxi-croman-2-il)metil amino)butil)-1,2-benzisotiazol-3(2H)-ona, de sus sales, hidratos y/o solvatos fisiológicamente aceptables, en especial de sus clorhidratos para la preparación de un medicamento para la profilaxis y/o tratamiento de la enfermedad de Parkinson.
Patent UY-31427-A1 (UY)
Title: Derivados 1,2,4-triazol amino como moduladores de mglur5
Inventor: ISAAC METHVIN
IPC: A61P25/00
Filed: 2008-10-24
Abstract: La presente invencion está dirigida a nuevos compuestos, a un proceso para su preparacion, su uso en terapia y composiciones farmacéuticas que comprenden los nuevos compuestos.
Patent ES-165523-A1 (ES)
Title: PERFECCIONAMIENTOS EN LA FABRICACIoN DE HILO FUSIBLE PARA CORTOCIRCUITOS FUSIBLES
Filed: 1944-04-10
Abstract: Perfeccionamientos en la fabricación de hilos o tiras fusibles para cortacircuitos fusibles caracterizado porque el hilo o la tira son de una pieza cuya sección transversal posee la misma superficie sobre toda la longitud del hilo. pero la superficie irradiadora de calor por unidad de longitud del hilo está localmente ensanchada por ejemplo por laminado en la parte no destinada a la fusión.
Patent ES-169681-A1 (ES)
Title: MECANISMO DE DIRECCIoN DE CREMALLERA PARA TRACTORES AGRiCOLAS O VEHiCULOS SIMILARES
Filed: 1951-02-23
Abstract: Perfeccionamientos en artículos textiles tales como crines pajas cintas y sus similares caracterizándose por el hecho de estar constituídos por lo menos en parte por fibras discontínuas artificiales o sintéticas y que por lo menos en parte las expresadas fibras están encoladas entre sí en parte o en su totalidad pudiéndo presentarse la ensambladura de la fibras primitivas en forma de cinta de mecha de hilado de retorcidos.
Patent ES-194833-A1 (ES)
Title: UN PROCEDIMIENTO PARAQ LA PREPARACIoN DE VITAMINA B12
IPC: A61K31/00
Filed: 1950-10-05
Abstract: Procedimiento que comprende hacer reaccionar con materias similares a la vitamina B12 una sustancia que suministra iones de cianuro para convertir así dichas materias en vitamina B12.
Patent ES-198877-A1 (ES)
Title: UNA NUEVA MáQUINA PARA FABRICACIoN DE CORDELERiA
Filed: 1951-07-21
Abstract: Nueva máquina para fabricación de cordelería, caracterizada por estar constituida por dos partes una para el hilado de fibra y la otra para el corchado de los hilos, estando de tal modo dispuestas las muletillas que solo embragan, por fricción, con la rueda conductora cuando trabajan, merced a la tensión de la fibra y cuando el movimiento con la fricción por la acción de unos muelles montados en el eje, cuando con el trabajo de la fibra, cesa la tensión de este.
Patent ES-239586-A1 (ES)
Title: Polyester-vinyl monomer compositions containing amidino compound and a sulfhydryl compound and process for copolymerizing same
IPC: C08F283/01
Filed: 1958-01-15
Abstract: An unsaturated polyester resin composition comprises (1) an unsaturated linear polyester (2) a monomer co-polymerizable therewith and containing a CH2=C< group (3) a sulphydryl compound and (4) a compound containing an <FORM:0874289/IV (a)/1> group and having a boiling point above 60 DEG C. Long lists of compounds are given in the Specification, of which the following are a general summary: (i) the polyester may be derived from di- or poly-hydric alcohols and unsaturated polycarboxylic acids (e.g. maleic, fumaric, citraconic, mesaconi, chloromaleic, carbic, itaconic and aconitic) with or without saturated polycarboxylic acids (ii) the co-polymerizable monomer may be allyl or methallyl alcohol, a vinyl, allyl or polyallyl ester, acrolein, methacrolein, a vinyl alkyl ketone, methyl isopropenyl ketone, a vinyl ether, isobutylene, styrene, an alkyl or halo styrene, isopropenyl toluene, vinyl naphthalene, acrylates (including allyl), chloracrylates, alkacrylates (including allyl), acrylonitrile, methacrylonitrile, acrylamide, methacrylamide, N-methylol acrylamide, diallyl citraconate, muconate or itaconate, triallyl aconitate, vinylidene chloride or chlorofluoride, N-vinyl pyrrole, carbazole, indole or succinimide, diallyl carbonate, triallyl cyanurate, tri-allyl or trimethallyl phosphate, allyl (chloro) silanes, tetra-allyl silicate and hexallyl disiloxane (iii) the sulphydryl compound may be H2S, an inorganic hydrosulphide or a mercaptan, including such compounds which contain a sulphydryl group in a tantmeric form, e.g. thioacetamide, thioacetanilide, and thiohydantoin (iv) the <FORM:0874289/IV (a)/2> compound may be a guanidine, an amidine, a guanyl guanidine, a guanyl urea, a pseudo urea, a pseudo thiourea, or a salt thereof. This system acts as a promoter for a normal polymerization catalyst, e.g. peroxides, hydroperoxides, peracids or salts, peroxyesters, ozonides, a , a -azodiisobutyronitrile or cobalt naphthenate. Other compounds which may be present include inhibitors (e.g. phenols, hydroquinones, amines), ultra-violet light absorbers (e.g. hydroxybenzophenones), solvents for the additives (e.g. diethylene glycol, styrene, dibutyl phthalate or ethylene glycol), ground asbestos and glass fibres. In examples the following mixtures of compounds (iii) and (iv) are used: (1-5 and 7-11) lauryl mercaptan and benzamidine-HCl (6 and 12) lauryl mercaptan and ethylene-1, 2-guanidine hydrochloride (13) thioglycollic acid and lauryl-amidine-HCl (14) thiourea, 2-naphthalenethio, and ethylene-1, 2-guanidine hydrochloride (15) 2-mercaptobenzoic acid and 1, 3-dicyclohexyl guanidine (16) n-nonyl mercaptan and 1-ethyl pseudothiourea hydrobromide. Reference has been directed by the Comptroller to Specification 758,618.
Patent ES-291803-A1 (ES)
Title: Disubstituted isobutyric acid esters
IPC: C07D307/00
Filed: 1963-09-19
Abstract: The invention comprises the compound of formula <FORM:1020158/C2/1> and its preparation from b -(1-naphthyl)-b 1-tetrahydrofurylisobutyric acid either by azeotropically esterifying with diethylaminoethanol or by reacting with b -chloroethyl-N-diethylamine. Pharmaceutical compositions comprise compound I with carriers. Oral (tablets), rectal (suppositories) and parenteral (solutions) administration is mentioned. The compound is antispasmodic.
Patent ES-295279-A1 (ES)
Title: Oscillating disc liquid meter
IPC: G01F3/12
Filed: 1964-01-14
Abstract: A rotary liquid meter of the nutating disc type, comprises a two-part spherical body 1, 2, Fig. 1, having integral and aligned inlet and outlet connections 1a, 2a respectively and clamped therebetween the flange 15b of a cupmember 15 which supports a measuring chamber 13 of definite volume formed as a pressing in stainless steel. The measuring chamber is closed at its upper end by a flat plate 2c formed integral with the body part 2 and formed at its lower end 13e with a surface co-operable with a substantially conical oscillating disc 12 having a spherical boss 12a seated in a depression 13d in the lower end 13e and a hole in the plate 2c. Liquid passes into the measuring chamber 13 through the inlet connection 1 a, a strainer 4 and aligned ports 15c, 13b, Fig. 2, in the cupmember 15 and measuring chamber 13 respectively. The liquid oscillates the disc 12 and then leaves the chamber through a port 13a in the chamber, a recess 15d in the cup and the outlet connection 2a, the ports 15c, 13b being separated from the port 13a and recess 15d by a barrier plate 14 engaging the boss 12a and slotted into the bottom and part-spherical surfaces of the measuring chamber 13 and the flat plate 2c. Oscillation of the disc 12 rotates a peg 12b which through a magnetic coupling 8, 9 and gears 18, 19, 20 rotates a counter 5. A glass cover 7 encloses the counting mechanism.
Patent ES-310136-A1 (ES)
Title: Protecting slipper for an edge roller in a glass sheet support bath
IPC: C03B18/06
Filed: 1965-03-04
Abstract: <PICT:1025065/C1/1> <PICT:1025065/C1/2> An apparatus, for use in the manufacture of flat glass during which glass in ribbon form is advanced along a bath of molten metal contained in a tank structure, comprises a trough-shaped slipper 2 mounted relative to the tank structure and held sloping downwardly and partially submerged in the molten metal 3, and an edge roll 24 projecting through the tank side wall into the trough in the slipper 2 so that the top surface of the edge roll lies above the top edge of the slipper and can engage under a margin 22 of a ribbon of glass 23 advanced along the bath, while the slipper preserves the edge roll from contact with the molten metal bath 3. The slipper 2 is preferably made of carbon, although it may be made of refractory material and have carbon inserts dove-tailed in its top edges (see 31, Fig. 5, not shown). The slipper 2 is supported by two cantilever beams 14, 15, bolted to a block 20 outside the tank structure. The block 20 also supports a bearing mounting 26 through which the shank 25 of the edge roll 24 passes, said shank also passing through a channel 13 in the outer end wall of the slipper. There is a clearance gap between the slipper and the edge roll 24. The edge roll is made of spheroidal graphite cast iron, mild steel or stainless steel, and both it and its shank 25 are hollow and water cooled. An upper edge roll 29 also mounted through the tank side wall, and block 20 may be located above the edge roll 24 to co-operate with edge roll 24 to grip the margin 22 of the glass ribbon 23 thus to advance it down the bath.
Patent ES-315201-A1 (ES)
Title: Radiant heating devices
IPC: F23D14/72
Filed: 1965-07-10
Abstract: A radiant gas burner having a perforated radiant plate 5, Fig. 1, (not shown), has a thermocouple 10 located in a chamber 9 separated from the outer surface of the radiant plate 5 by a perforated plate 7 which is more prone to backfiring than the radiant plate 5. If the flame back-fires into the chamber 9 the thermocouple 10 closes an electromagnetic fuel valve 1 supplying the burner. The perforated plate 7 may be made of material of greater heat conductivity than the radiant plate 5 or it may have passages of larger cross-section than the passages in the radiant plate 5. A further thermocouple 11 is disposed outside the radiant plate 5 and generates a current which holds the fuel valve 1 open. The two thermocouples oppose each other. The chamber 9 may be disposed within or below the radiant plate 5.
Patent ES-318601-A1 (ES)
Title: Apparatus for the mechanical extraction of coal and other materials occurring in seamformation by the long wall method of working
IPC: E21C35/12
Filed: 1965-10-16
Abstract: In a longwall mineral-mining installation in which an endless cutter chain is caused to circulate in a plane parallel to a mineral face to be worked to kerf the top and bottom of the face for the full length thereof articulated chain guides are so connected to the fronts of the face conveyor and to the alternately advanceable roof support frames of the installation that the guides can be angularly adjusted about axes parallel to the lengths of the troughing sections of the conveyor to permit of variation of the angle of attack of the chain to the face.
Patent ES-337859-A1 (ES)
Title: Improvements in electrical fittings
IPC: H01R13/453
Filed: 1967-03-10
Abstract: The housing of an electrical fitting, which may be a fuse base, has contacts (13), (Fig. 2, not shown), covered by shrouds 3, 4 of e.g. nylon, the shrouds having at least one resilient flap 11, 12, formed by slots 8, 9, 10 in alignment with contacts (13), the flaps being normally in a closed position to shield the contacts, but yieldable under pressure to permit passage therethrough of further contacts (14). The flaps may be made thinner than the other parts of the shrouds to be readily yieldable, and the contacts (13) may be as described in Specification 1,123,067.
Patent ES-338881-A1 (ES)
Title: Device for the continuous and automatic measurement of gamma-ray emission of a solution
IPC: G01T7/02
Filed: 1967-04-04
Abstract: The radioactivity of a liquid containing fission products is measured by a two-path photo-electric system in order to compensate for errors due to adsorption of fission products on the walls of the measurement cell. The liquid 2, which is y-ray emitting, is passed through a tank 4 having two parallel walls 5, 7, but of changing depth. Lead shielding is provided all round the tank and the shielding wall 6 is provided with collimator apertures 8, 10 so that scintillation counters 12-16 and 14-18 can respectively view volumes v 1 and v 2 of the liquid, and areas s 1 and s 2 of the top y-ray transparent wall 5 on which fission products are adsorbed. (Adsorption takes place on the bottom wall 7 but this is arranged to be distant engouh from the scintillators not to be detectable). Volumes v 1 and v 2 are in a fixed ratio p 1 and areas s 1 and s 2 in a fixed ratio p 2 different from # 1 . An equation is derived for the activity A u of the liquid as A u = 1/V 2 (N 1 - p 2 N 2 ) / p 1 - p 2 ) where N 1 and N 2 are the counts obtained in a certain time interval by counters 20, 22. For simplicity, the volumes viewed by the detectors are arranged to be equal (v) and the areas s 1 and S 2 in the ratio 1:2 so that the activity per unit volume is obtained as A u = 1/V(2N 1 - N 2 ). Thus by feeding the outputs of counters 20, 22 to a subtraction circuit 24, the value N 1 - N 2 is obtained. Addition of the output of counter 22 to this in adding circuit 26 gives an output which can be calibrated to equal the activity per unit volume.
Patent ES-339492-A1 (ES)
Title: Process for the manufacture of stable aqueous dispersions of vinyl esters of organic acids and ethylene
IPC: C08F10/00
Filed: 1967-04-19
Abstract: A stable aqueous dispersion of a copolymer of a vinyl ester of an organic acid and ethylene is prepared by forming a solution having a predetermined concentration of ethylene in a vinyl ester of a saturated mono-carboxylic acid, passing the solution to a polymerization zone and polymerizing the solution as an aqueous emulsion in the presence of a free radical catalyst, a surface active agent and/or a protective colloid whilst maintaining the zone full of emulsion at sufficient pressure to retain the ethylene in solution. In examples were used: ethylene and vinyl acetate sodium decyl benzene sulphonate, nonyl phenol-ethylene oxide condensate, polyvinyl alcohol, potassium bicarbonate, water, ammonium persulphate, formic acid and sodium metabisulphite.