baber/WOPTO huggingface dataset:
Patent AU-709219-B2 (AU)
Title: Thiolation of peptides for radionuclide-based radiodetection and radiotherapy
Inventor: GOVINDAN SERENGULAM V
IPC: A61K38/31
Filed: 1996-06-07
Granted: 1999-08-26
Abstract: A method of radiolabeling a peptide, e.g., somatostatin or an analogue thereof or vasoactive intestinal peptide, with a radioisotope of technetium or rhenium, comprises the steps of: (a) reacting the peptide with an acetyl-protected <u>t</u>-thiol-containing, amine-reactive bifunctional chelating agent; (b) deprotecting the acetyl-<u>t</u>-thiol group to generate a free <u>t</u>-thiol group; and either (c) admixing the peptide-<u>t</u>-thiol-containing conjugate with a stannous salt; and (d) reacting the mixture of step (c) with pertechnetate or perrhenate, or (c') adding reduced pertechnetate or perrhenate to said peptide-<u>t</u>-thiol-containing conjugate, thereby forming a radiolabeled peptide. Kits for effecting the radiolabeling method, and methods of tumor detection/imaging or therapy are provided.
Patent AU-580892-B2 (AU)
Title: Powder particles for fine-grained hard material alloys and a process for the preparation of such particles
Inventor: OSKARSSON ROLF GREGER
IPC: C23C8/24
Filed: 1986-09-04
Granted: 1989-02-02
Abstract: The present invention relates to powder particles consisting of hard principles and binder metal for the manufacture of superior, uniquely fine-grained hard material alloys and to a procedure for the preparation of said particles.The preparation is performed in an economical way because the procedure starts from conventional melt metallurgical raw materials. A pre-alloy consisting of hard principle forming and binder phase forming elements is subjected to a heat treatment such as nitriding and carburizing after being crushed. The final product is particles composed by hard principle phases and binder metal phases formed "in situ" in an effective binding.
Patent AU-548917-B2 (AU)
Title: Catalyst for polymerising ethylene
Inventor: BUJADOUX KAREL
IPC: C08F4/62
Filed: 1980-12-23
Granted: 1986-01-09
Abstract: A process for polymerizing ethylene in the presence of a catalyst system comprising at least two halogen compounds of transition metals, one of which has the formula (TiCl3,Y3 AlCl3)(MY3)x(MgYZ)y, where M is a transition metal of Group VB or V1B, X is a halogen and 0.3</=x</=3, 0</=y</=20, and a Group I to III hydryde or organometallic activator and the mean residence time of the catalyst system in the polymerization reactor is between 2 and 100 seconds.
Patent AU-544644-B2 (AU)
Title: A method and a device for recording and handling of information regarding time and activities
Inventor: BILLE D
IPC: G07C3/00
Filed: 1981-01-21
Granted: 1985-06-06
Abstract: The present invention refers to a method and a device for recording, handling and documentation oftime/activity data. The duration of different categories of work occasions and/or activities, as for example down time, can be measured by activation of a press button correspondantto each category of work. Hereby a pulse train (11), generated in a pulse generator (10), is provided to at least one of a plurality of possible storage cells (12). As the time between two pulses (11a), following after each other, is constant and known, e.g. one hundredth of an hour, the total number of pulses (11a), the storage cells (12) are fed with, will correspond to a time value required for the respective output of work and/or activity. When desired the information content of all storage cells (12) is read. This information is converted and/or handled at which the result by a printer (7) is written in a manually readable form on an information carrier (6). The information content of the storage cells (12) can also be transferred to and handled by a central reading unit.
Patent AU-587101-B2 (AU)
Title: Sound-producing amusement devices
Inventor: WEINER AVISH JACOB
IPC: A63F9/00
Filed: 1987-01-20
Granted: 1989-08-03
Abstract: A sound-producing amusement device, comprises: a read-only memory having recorded therein digital data representing sounds characteristic of the amusement device, and a sound-producing unit for producing the sounds represented by the digital data recorded in the read-only memory. The read-only memory is in a separate unit including connectors for connection to the sound-producing unit. The sound-producing unit includes mating connectors for removably attaching and electrically connecting the sound-producing unit to the read-only memory unit, a battery for supplying power to both the sound-producing unit and the read-only memory unit, and a speaker for producing the sounds represented by the data stored in the read-only memory unit.
Patent AU-735007-B2 (AU)
Title: Protective roll guard for clearing obstacles from caster wheels
Inventor: TUPPER BRADLEY J
IPC: B60B33/00
Filed: 1998-04-15
Granted: 2001-06-28
Abstract: A one-piece roll guard (10) having two half segments (12, 14) connected by an integral hinge (16) for protecting a caster (100) wheel by clearing obstacles away from its rolling path. The two segments of the roll guard (10) are closed and secured together around the caster wheel with a locking tab (18a) and matching locking slot (18b) integrally formed in the two segments. The roll guard is formed with a weighted lower lip (26) to improve stability by lowering the center of gravity of the roll guard (10).
Patent AU-685137-B2 (AU)
Title: Ortho-substituted benzoylguanidines, process for their preparation, their use as pharmaceutical or diagnostic, and pharmaceutical containing them
Inventor: WEICHERT ANDREAS
IPC: A61P9/10
Filed: 1994-08-26
Granted: 1998-01-15
Abstract: There are described ortho-substituted benzoylguanidines of the formula I <IMAGE>  in which:   R(1) is H, Hal, CN, NO2, (cyclo)alkyl, (O)(S)[NR(5)](CH2)b-(CF2)c-CF3,   R(5) is H, (C1-C4)-alkyl, -CdH2dR(6),   R(6) is cycloalkyl, (bi)phenyl(yl), naphthyl,  or   R(1) is -SR(10), -OR(10), -CR(10)R(11)R(12),   R(10) is -CfH2f-(C3-C8)-cycloalkyl, -(C1-C9)-heteroaryl or phenyl, R(11) and R(12) are defined as R(10) or are hydrogen, (C1-C4)-alkyl,  or   R(1) is naphthyl, (bi)phenyl(yl), (C1-C9)-heteroaryl,  or R(1) is -SR(13), -OR(13), -NHR(13), -NR(13)R(14), -CHR(13)R(15), -C[R(15)R(16)]OH, -C IDENTICAL CR(18), -C[R(19)]=CR(18), -[CR(20)R(21)]k-(CO)-[CR(22)R(23)R(24)]l,   R(13) and R(14) are -(CH2)g-(CHOH)h-(CH2)l-(CHOH)j-R(17),   R(17) is hydrogen, methyl, -(CH2)g-O-(CH2-CH2O)h-R(24), R(15) and R(16) are hydrogen, alkyl or, together with the carbon atom carrying them, cycloalkyl,   R(18) is phenyl, heteroaryl, (cyclo)alkyl,   R(19), R(20), R(21), R(22) and R(23) are hydrogen, methyl,   R(24) is H, (cyclo)alkyl, -CmH2m-R(18),   R(2) and R(3) are defined as R(1),   R(4) is alkyl, Hal, CN, -(CH2)n-(CF2)o-CF3,  and their pharmaceutically tolerable salts. Compounds I have no unwanted salidiuretic properties, but very good antiarrhythmic properties. They are outstandingly suitable as antiarrhythmic medicaments having a cardioprotective component for infarct prophylaxis and infarct treatment and for the treatment of angina pectoris, where they also preventively inhibit or greatly decrease the pathophysiological processes in the formation of ischaemically induced damage. Because of their protective actions against pathological hypoxic and ischaemic situations, the compounds of the formula I according to the invention, as a result of inhibition of the cellular Na<+>/H<+> exchange mechanism, can be used as medicaments for the treatment of all acute or chronic damage caused by ischaemia or illnesses primarily or secondarily induced thereby.
Patent AU-634041-B2 (AU)
Title: A load indicating device comprising a control nut containing a threaded joint assigned to anchors, particularly injection anchors for the mining industry or the like
IPC: E21D21/02
Filed: 1991-03-25
Granted: 1993-02-11
Abstract: A indicating-nut threaded coupling with load-indicating device (1) adapted to be arranged in particular on grouted anchors for mining or the like and in order to obtain a simple solution which is advantageous in use a free space is formed by at least one groove (4) equipped with a fold bottom (5), the groove being arranged in the outer wall (3) of a bushing (2) which extends spaced from the outer surface of the anchor.
Patent AU-607920-B2 (AU)
Title: Preparation of hydrolysed zirconium salt precursors and high purity zirconia
Inventor: HOUCHIN MARTIN RICHARD
IPC: C01G25/02
Filed: 1987-06-05
Granted: 1991-03-21
Abstract: In the economic production of hydrolysed zirconiferous precipitate, hydrolysis is carried out by the addition of base to aqueous acidic zirconium sulphate solution, to lower the H<+> to and maintain within a pH range of 3 to 7, preferably within 4 to 6. The base may be selected from ammonia, basic ammonium salts, e.g., ammonia-buffered ammonium salts, an alkali metal hydroxide, carbonate or bicarbonate. Specific bases include ammonia and ammonium/sodium/potassium hydroxide, carbonate or bicarbonate, with particular preference for ammonia and ammonium/sodium hydroxide. The starting materials may be incorporated in batchwise or continuous fashion, batchwise by combining them in a body of water, suitable electrolyte or solvent with thorough continuous mixing or continuously by mixing them together in a flowing stream. An additive in the form of an inorganic stabiliser or an organic surfactant may also be included. Inorganic stabilisers may be selected from one or more of Y2O3, Ce2O3, Al2O3, MgO and CaO or precursors thereof. In the finishing stage, either further base may be added to lower residual sulphate content or acid added to remove acid-soluble impurities. The precipitated product is then separated, (e.g., by filtration), washed and calcined to give pure zirconia. High purity zirconia has particular application in the electronics industry and for the production of partially stabilised zirconia ceramics.
Patent AU-743581-B2 (AU)
Title: Synthetic resin composition having resistance to thermal deterioration and molded articles
Inventor: NOSU TSUTOMU
IPC: C08K3/10
Filed: 1998-07-02
Granted: 2002-01-31
Abstract: A synthetic resin composition having heat deterioration resistance comprising:     (A) 100 parts by weight of a synthetic resin; and (B) 0.001 to 10 parts by weight of hydrotalcite particles defined by the following (i) to (iv):   (i) the hydrotalcite particles are represented by the following chemical structure formula (1): ä(Mg)y(Zn)zü1-x(Al)x(OH)2(A<n->)x/n.mH2O (ii) the hydrotalcite particles have an average secondary particle diameter of 2  mu m or less; (iii) the hydrotalcite particles have a specific surface area (measured by a BET method) of 1 to 30 m<2>/g; and (iv) the hydrotalcite particles contain an iron compound and a manganese compound in a total amount of 0.02 wt% or less in terms of metals (Fe + Mn).     A molded article formed from the above resin composition of the present invention is excellent in heat deterioration resistance and impact resistance and satisfactory in the dispersibility of hydrotalcite particles.
Patent AU-546929-B2 (AU)
Title: Control arrangement
Inventor: AXMANN ARNOLD
IPC: B66C13/46
Filed: 1982-03-12
Granted: 1985-09-26
Abstract: An arrangement for controlling movement of the grab bucket of a grabbing crane used for loading and unloading bulk material into and from ships is disclosed. Collisions of the grab bucket with the ship's superstructure and the hatch edges are avoided according to the invention by approaching the hatch edges with the grab bucket open and displaying the actual values so obtained as bars representing the horizontal position and width of the hatch on a display. To avoid collisions, the grab bucket drives are switched off if any desired value, set manually or by a marking line computer, exceeds an actual value.
Patent AU-608788-B2 (AU)
Title: Medicaments for the treatment of addiction
Inventor: TYERS MICHAEL BRIAN
IPC: A61K31/46
Filed: 1987-11-20
Granted: 1991-04-18
Abstract: The invention relates to the use of 1,2,3,9-tetrahydro-9-methyl-3-[(2-methyl-1H-imidazol-1-yl)methyl]-4H</ U>-carbazol-4-one and physiologically acceptable salts and solvates thereof in the relief or prevention of a withdrawal syndrome resulting from addiction to a drug or substance of abuse and/or for the suppression of dependence on drugs or susbtances of abuse.
Patent AU-597749-B2 (AU)
Title: Peptides
Inventor: NYEKI OLGA
IPC: C07K5/00
Filed: 1987-11-20
Granted: 1990-06-07
Abstract: The new peptides of the Formulae     (1) Glp-Lys-NH2   (2) Glp-Glu-Lys-NH2   (3) Arg-Lys-Glu-NH2   (4) Arg-Lys-Asp-NH2   (5) Arg-Lys-Glu-OH   (6) Arg-Lys-Gln-OH   (7) Leu-Val-Ala-OH   (8) Arg-Orn-Asp-Val-NH2   (9) Arg-Orn-Asp-Val-OH   (10) Lys-Glu-Lys-Lys-OH   (11) Lys-Leu-Lys-Lys-OH   (12) Lys-Asp-Leu-Lys-OH   (13) Glu-Leu-Val-Ala-OH and   (14) Leu-Pro-Ala-Gly-OH and acid addition salts thereof inhibit the proliferation of leukaemic cells and exhibit immunostimulant effect.
Patent AU-602744-B2 (AU)
Title: Device for the control of an ammonia converter etc.
Inventor: HERBORT HANS-JOACHIM
IPC: C01C1/04
Filed: 1987-12-17
Granted: 1990-10-25
Abstract: In the converter having a process gas inlet and outlet, at least one heat exchanger and at least one catalyst bed as well as a further gas feed and having a central pipe and a process gas feed to the heat exchanger and/or catalyst bed, the heat exchanger and the first catalyst bed around the latter being arranged rotationally symmetrically to the central pipe, control gas, quench gas, a part of the process gas at a different temperature and/or under other conditions at a point of a reactor is to be added to the particular gas streams in such a way that the mixing-in and/or the by-pass line are designed for complete isolation, partial loading and/or complete opening. For this purpose, the central pipe (14) for temperature control as a control gas feedpipe completely penetrates the heat exchanger (4 and/or 5 and/or 6) and is provided at its lower end with controllable outlets (18) for at least partial mixing of the control gas with the process gas stream, before the latter flows through the catalyst bed (4), and/or for mixing the control gas stream with the process gas stream after the latter has passed through the catalyst bed (4) and the heat exchanger (7). <IMAGE>
Patent AU-637937-B2 (AU)
Title: Flexible intumescent coating composition
IPC: C09K21/04
Filed: 1991-09-25
Granted: 1993-06-10
Abstract: Disclosed is an intumescent curable composition which contains as a resinous binder a flexible polyepoxide resin. The polyepoxide is cured with an appropriate curing agent adapted for the particular resin. An additive component is present which contains a mixture of materials which provide a source of     (i) zinc,   (ii) boron,   (iii) phosphorus, and (iv) an expansion gas upon thermal decomposition. The composition is capable of forming a carbonaceous char upon exposure to heat or flame, with the proviso that the cured, unburned composition has sufficient flexibility that it passes at least 10 continuous cycles of a cold cycle test without cracking. The cold cycle test involves the following steps: the composition is applied at a thickness of 0.5 inch (12.7 millimeters) to a 10 inch (0.254 meter) section of a 4W13 I-beam having two thermocouples attached to the surface, allowed to cure at ambient temperature for 16 hours, force cured for 5 days at about 60 DEG C and subjected to the cold cycle test. For one cycle, the beam is placed in a freezer operating at a temperature between about 0 DEG F (-18 DEG C) and about -10 DEG F (-23 DEG C) for sufficient time for the steel to reach a temperature between about 0 DEG F (-18 DEG C) and about (-10 DEG F) -23 DEG C as determined by the two thermocouples attached to the surface of the beam beneath the coating, removed from the freezer and a 50 square inch area (0.0323 square meter) of the surface warmed as shown in FIGS 1 and 2 by passing a heat gun (Model No. HG 50146, Alpha Division of Loral Corp, 14 amp: minimum temperature at tip 500 DEG F (260 DEG C)) a distance of 0.5 inch (12.7 millimeter) from the surface, uniformly over the surface until the surface temperature reaches 110 DEG F (43 DEG C) within a 3 minute period, as determined by a thermocouple moved about the surface and allowed to stand for at least 2 hours at ambient temperature.   <IMAGE>
Patent AU-655201-B2 (AU)
Title: Bag and the like for children, produced by molding
Inventor: GOTO FUMIO
IPC: A45C5/02
Filed: 1991-09-27
Granted: 1994-12-08
Abstract: A bag and the like for children, produced by molding, having a main body consisting of a front side portion (1) and a rear side portion (2), which are made by molding, respectively, said front side portion (1) suitably and precisely representing a complicated tridimensional shape such as a face of an animal, e.g. a panda, said rear side portion (2) being connected at a half portion thereof, which is closer to the bottom, to said front side portion (1) for forming a vacant space to receive articles, and an upper half of said rear side portion (2) constituting a lid (10) largely openable and closable on a hinge portion (4) integrally formed on said rear side portion (2). The lid (10), when closed with respect to the front side portion (1), can allow the main body of the bag to form a box construction having a satisfactory strength, so that the articles contained in the interior thereof can be protected safely. <IMAGE>
Patent AU-639154-B2 (AU)
Title: New imidazole compounds, a process for the preparation thereof, and pharmaceutical compositions containing them
IPC: C07D233/64
Filed: 1991-11-13
Granted: 1993-07-15
Abstract: The invention relates to the compounds of general formula (I): 
<IMAGE>
 in which 
 
  R represents a linear or branched (C1-C6) lower alkyl group, a (C3-C8) cycloalkyl group, an optionally substituted phenyl group, a pyridyl group or a naphthyl group, 
  R1 and R2, which may be identical or different, represent a hydrogen atom, a linear or branched (C1-C6) alkyl group or a linear or branched (C1-C6) acyl group, 
 to their enantiomers, diastereoisomers and epimers as well as to their addition salts with a pharmaceutically acceptable acid. 
<??>Medicaments.
Patent AU-746497-B2 (AU)
Title: A high quality, continuous throughput, tissue fixation-dehydration-fat removal-impregnation method
Inventor: ESSENFELD ERVIN
IPC: G01N33/48
Filed: 1998-08-19
Granted: 2002-05-02
Abstract: Described is an apparatus for rapid processing of tissue specimens for histology with continuous throughput, the apparatus comprising: 
(a) a microwave unit which (1) fixes, dehydrates, and defats the tissue specimens with a non-aqueous solution In a first vessel; (II) agitates the tissue specimens and the non-aqueous solution In the first vessel; and (III) exposes the tissue specimens and the non-aqueous solution in the first vessel to microwave energy to produce fixed, dehydrated, and defatted tissue specimens; and a source for the nen-aqueous solution which is fluidly coupled to the first vessel; 
(b) an Impregnator unit which (I) Impregnates the fixed, dehydrated, and defatted tissue specimens with a wax solution In cut second vessel; (ii) agitates the fixed, dehydrated, and defatted tissue specimens and the wax solution In the second vessel; and (iii) exposes the fixed, dehydrated, and defatted tissue specimens and the wax solution to elevated temperature under a vacuum to produce fixed, dehydrated, defatted, and impregnated tissue specimens; and a source for the wax solution which Is fluidly coupled to the second vessel; and  
wherein tissue specimens are sequentially transferred into the first vessel and then into the second vessel.
Patent DE-1917675-B2 (DE)
Title: Broadband microwave omnidirectional aerial - has dielectric dish mounted above circular hollow waveguide and inclinable relative to horizontal plane
IPC: H01Q13/04
Filed: 1969-04-05
Abstract: The broad-band microwave omnidirectional aerial has a vertical circular hollow waveguide and a metallic conical reflector. It is designed to provide, by simple means, amt with full retention of the broad-band feed, increased vertical focusing or beaming of the microwave radiation. A dielectric disc whose thickness decreases towards its periphery, is provided above the circular hollow waveguide. It is excited or energised by the latter such that, with horizontal radiation, the beam conicity angle ( k) is specif. 90 deg. More specif. with the radiation directed downwards by an angle alpha relative to the horizontal (plane), the cone angle k = 90 deg. + alpha amt. the dish or disc is inclined downwards by the angle alpha outwards to its rim.
Patent DE-1943939-B2 (DE)
Title: Fast concrete setting - in pressurised steam chamber
IPC: C04B40/02
Filed: 1969-08-29
Abstract: The process comprises the placing of the mouldings into a water filled pressure chamber in which it is subjected to an elevated pressure heating cycle consisting of a first heating step for 25-35 mins to 110-120 degrees C followed by a 140 min sec linear heating stage to 180 degrees C. Following this it is cooled slowly over 30 mins. which period is subdivided into three equal length steam bleeding, straight cooling down and final water draining stages. The initial compressed air pressure in the chamber is pref. 5 atm which rises to 14 atms as a result of heating. The whole process is pref. carried out in a fully automatic cycle pressure chamber.
Patent DE-1956351-B2 (DE)
Title: Vortex inlet chamber for IC engines - has spiral profiled inlet duct which induces rotational and axial flow into combustion chamber
IPC: F02F1/42
Filed: 1969-11-08
Abstract: A profiled inlet chamber for internal combustion engines is designed to induce vortex motion as an aid to charging and uniformity of combustion propagation. The engine has a fuel injection nozzle (1) that is offset to the centre line of cylinder axis (5). A circular inlet valve is located (3) in a position offset from the cylinder axis. Air flow is induced into the combustion chamber by a spiral chamber (12) that imparts both a rotational and axial flow component. The cross-section area of the inlet duct reduces progressively to the valve port.
Patent DE-2016481-B2 (DE)
Title: Fruit machine with totally independent drum motion - uses balls falling into holes to complete circuit to ensure random stopping process
IPC: G07F17/34
Filed: 1970-04-07
Abstract: A fruit machine based on rotating drums with symbols on the periphery, is designed to ensure that the spinning motion is independent of external and internal influences. A single drum (53) rotates within a stationary housing (52). One section of the drum has a number of holes (53) to provide location for a number of balls; one of which (30) is electrically conducting. The balls are initially located within the centre region and fall through an aperture (28) in an internal sleeve (27) into the holes. The conducting ball complete a circuit between the sleeve and a contact (24) to switch in a solenoid to sto p the drum.
Patent DE-2215258-B2 (DE)
Title: Current collector in electric motor vehicle - has pantograph link mechanism with support arm on axle of lever system fixed by bolts in slotted holes
IPC: B60L5/14
Filed: 1972-03-29
Abstract: The current collector is for an electrically-driven motor vehicle with a pantograph lever system. It consists of a base frame with link mechanism and spring loading. There is a lifting cylinder which can be adjusted between two end positions. The support arm (4) of the pantograph lever system (4-9) is rigidly attached to the axle of the rotating lever with shearing bolts (21). Two limiting cams (18) on the lever axle will be up against the stop (19) on the base frame in the two end positions of the cylinder.