baber/WOPTO huggingface dataset:
Patent AU-756175-B2 (AU)
Title: Catalytic domain of the human effector cell cycle checkpoint protein kinase, Chk1, materials and methods for identification of inhibitors thereof
Inventor: CHEN PING
IPC: C07K19/00
Filed: 2000-10-26
Granted: 2003-01-09
Abstract: The present invention relates to the identification, isolation and purification of the catalytic domain of the human effector checkpoint protein kinase (hChk1). A 1.7 &cir&  crystal structure of the hChk1 kinase domain in the active conformation is reported herein. The kinase domain of hChk1 and its associated crystal structure is described for use in the discovery, identification and characterization of inhibitors of hChk1. This structure provides a three-dimensional description of the binding site of the hChk1 for structure-based design of small molecule inhibitors thereof as therapeutic agents. Inhibitors of hChk1 find utility in the treatment of hyperproliferative disorders such as HIV and cancer.
Patent AU-584286-B2 (AU)
Title: Synthesis of 2-aminopyrimido``4,5-g`` quinolines
Inventor: WEIGEL LELAND OTTO
IPC: C07D215/20
Filed: 1987-03-30
Granted: 1989-05-18
Abstract: This invention provides a process for preparing trans 2-aminopyrimido[4,5-g]quinolines of formula <CHEM> wherein R is hydrogen, cyano, C1-C3 alklyl or allyl; R<1> is amino, -NHR<3> or -NR<4>R<5>; R<2> is hydrogen or methyl; R<3> is methyl, ethyl, n-propyl, C1-C3 alkyl-CO, phenyl-CO or substituted phenyl-CO, wherein said substituents are 1 or 2 members selected from the group consisting of chloro, fluoro, bromo, methyl, ethyl, methoxy, ethoxy and trifluoromethyl; and R<4> and R<5> are individually methyl, ethyl or n-propyl, which comprises reacting a compound of the formula <CHEM> wherein R<6> is C1-C3 alkyl, phenyl, 4-chlorophenyl, 4-bromophenyl or 4-methylphenyl, with a guanidine salt. The compounds are dopamine agonists.
Patent AU-712012-B2 (AU)
Title: Indole derivatives and medical application thereof
Inventor: NAGASE HIROSHI
IPC: C07D491/22
Filed: 1996-09-26
Granted: 1999-10-28
Abstract: The present invention relates to indole derivatives represented by the following compound 1 and the pharmacologically acceptable acid addition salt thereof. <CHEM> The compounds of the present invention were found to exhibit strong antitussive and analgesic actions as a result of pharmacological evaluation, and can be used in the pharmaceutical field as effective antitussives and analgesics.
Patent AU-545454-B2 (AU)
Title: Measuring the thickness of a strip
Inventor: ENGELHARDT WERNER
IPC: G01B15/02
Filed: 1981-07-31
Granted: 1985-07-18
Abstract: An arrangement for measuring the thickness of a strip emerging from a rolling mill is provided with a thickness measuring device and at least one linear inductor. The linear inductor exerts a pulling force on the strip which flatens the strip in the vicinity of the measuring device. This permits a measuring beam from the measuring device to pass through the strip in a direction orthogonal to the surface of the strip. In some embodiments, a plurality of linear inductors may be provided on either side of the strip, and on either side of the measuring device. The frequency of operation of the linear inductors may be controlled by a converter, in response to the speed of the emerging strip.
Patent AU-600517-B2 (AU)
Title: A riding saddle and method of manufacture
Inventor: PATRICK DUMOULIN
IPC: B68C1/02
Filed: 1987-09-08
Granted: 1990-08-16
Abstract: The invention relates to a riding saddle comprising a molded tree of composite material placed between two molded parts of cellular plastic material which constitute the seat and the underside of the saddle respectively. The tree (20) is formed as a single part comprising a thin strip of composite material and including a rigid arch (22) which is terminated at its front side ends by flexible flat tabs or "points" (30), together with a rear portion (32) in the form of a curved U-shape which includes zones (B, C) of flexibility for adapting to the shape of a horse's back.
Patent AU-674262-B2 (AU)
Title: Polymerizable Yellow Dyes and Their Use in Ophthalmic Lenses
Inventor: JINKERSON DAVID L
IPC: C08F220/60
Filed: 1994-10-11
Granted: 1996-12-12
Abstract: Novel polymerizable yellow dyes are disclosed. Additionally, novel and known dyes are used to block or lower the intensity of blue light transmitted through ocular lenses and other windows.
Patent AU-612604-B2 (AU)
Title: A frame for the box-shaped body of a commercial vehicle
Inventor: ROLLIN ULRICH
IPC: B61D17/08
Filed: 1987-11-02
Granted: 1991-07-18
Abstract: A set of profiles consisting of a U-shaped basic profile (20) and a covering profile (30) which can be attached to its legs (22, 23) is used for the framework of a utility vehicle body, particularly as posts (6). The basic profile (20) is incorporated into the framework with outwardly open channel (24) and connected to the cross bands (2, 3) through its solid wall base (21) by means of connecting elements (25, 26) and bolts (27). In order to increase the angular rigidity, reinforcing elements (28) are inserted in the basic profile channel (24) at the corner joints as required. Since the covering profile (30) is fitted subsequently all the fastening and reinforcing elements are concealed. <IMAGE>
Patent AU-605203-B2 (AU)
Title: Novel substituted aminomethanediphosphonic acids
Inventor: WIDLER LEO
IPC: C07F9/547
Filed: 1987-11-20
Granted: 1991-01-10
Abstract: Heteroarylaminomethanediphosphonic acids of the formula <IMAGE> in which R1 represents an optionally benzo- or cyclohexeno-fused 5-membered heteroaryl radical having 2 to 4 N atoms or 1 or 2 N atoms and 1 O or S atom as hetero atom(s) and which is unsubstituted or substituted by lower alkyl, phenyl which is unsubstituted or substituted by lower alkyl, lower alkoxy and/or halogen, lower alkoxy, hydroxyl, di-lower alkylamino, lower alkylthio and/or halogen and R2 denotes hydrogen or lower alkyl, and their salts have an action regulating the metabolism of calcium and can be used as pharmaceutical active compounds for the treatment of diseases which can be traced back to disorders thereof. They are prepared, for example, by converting the group(s) X into free phosphono in a compound of the formula <IMAGE> in which X1 denotes a functionally modified phosphono group X and X2 denotes phosphono or likewise a functionally modified phosphono group X.
Patent AU-632704-B2 (AU)
Title: Information processing apparatus with replaceable security element
IPC: H04N7/167
Filed: 1991-08-13
Granted: 1993-01-07
Abstract: A field upgradeable security system deciphers signals received from a communication network. An information processor (10) includes a receptacle for receiving a replaceable security element (12). The replaceable security element generates a working key (WK) necessary to the operation of the information processor. The working key is communicated to the information processor encrypted under a secret key (A(M)). The information processor decrypts the encrypted working key for use in deciphering a received communication signal. Additional layers of encryption (A(C), U(M), U(C)) can be added to the communications between the information processor and security element to increase the level of security. <IMAGE>
Patent AU-599735-B2 (AU)
Title: Switch-mode power supply protective circuit arrangement
Inventor: PREIS JOSEF
IPC: H02H9/00
Filed: 1987-12-22
Granted: 1990-07-26
Abstract: Circuit arrangement for limiting the switch-on current and for overvoltage protection of switched power supply apparatuses having an input-side storage capacitor (12), which forms a low-impedance voltage source for a power supply arrangement connected thereto. Such a power supply apparatus is intended to be provided with a circuit which not only limits the switch-on current but also ensures protection against overvoltages on the storage capacitor (12). This is achieved with the aid of a field-effect transistor (11) arranged between the supply voltage source (1) and the storage capacitor (12), which is not only controlled by an amplifier in the sense of current limiting but is also controlled by a delay member in the sense of delayed switching on. The power supply apparatus is particularly suitable for plug-in assemblies with voltage converters for supplying electrical telecommunications devices. 
<IMAGE>
Patent AU-646369-B2 (AU)
Title: Apparatus and method for a needle tip cover
Inventor: PURDY EDMUND R
IPC: A61M5/32
Filed: 1991-09-05
Granted: 1994-02-17
Abstract: A needle (10) cooperates with a tip cover (11) that coaxially fits about the needle (10) and slides axially relative thereto. A thin walled tube (15) of the needle (10) has a shank portion (12) extending from the proximal end (17) toward the distal end (16) and a tip portion (14) extending from the distal end (16) toward the proximal end (17). The tip portion (14) has a diameter ("A") that is larger than the diameter ("B") of the shank portion (12). The needle (10) includes a transition zone (13) between the shank and tip portions wherein the axial distance ("C") of the transition zone (13) is about an order of magnitude greater than the difference in the diameters of the tip and shank portions. The tip portion (14) includes a bevel (18) extending from the distal end (16) toward the transition zone (13) as a sharpened edge (19) to ease insertion. The cover (11) includes a bearing (21) and a tip protecting part (22). The bearing (21) is sized to coaxially fit about the shank portion (12) and slide axially relative thereto. The difference in the diameters of the tip and shank portions is such that the bearing (21) can not slide distally over the transition zone (13). The cover (11) is positioned on the needle (10) to locate the tip protecting part (22) over the sharpened edge (19) when the bearing (21) is at the transition zone (13). The transition zone (13) is shaped frusto conically and is located between the shank and tip portions. The frusto conical shape (20) is at angle relative to the axis ("E") of the needle (10) due to a difference in the first and second diameters thus providing a diametrical imperceptible change. <IMAGE>
Patent AU-533741-B2 (AU)
Title: On-line dehydrogenation or fibre preforms
Inventor: MODONE EROS
IPC: C03C13/00
Filed: 1982-06-09
Granted: 1983-12-08
Abstract: Vapor deposition of doped silica in a reaction chamber on a rotating supporting surface, in the manufacture of a preform for the drawing of an optical fiber, is accompanied by the continuous admixture of deuterium with a flow of carrier gas, specifically oxygen, by which the reactants are transported to the reaction chamber. An isotopic substitution of deuterium for the hydrogen of hydroxyl groups in the reaction products shifts the major absorption peaks to wavelengths outside the minimum-attenuation range of 0.7 to 1.6 mu  used for fiber-optical signaling. The proper ratio of deuterium to carrier gas is maintained with the aid of a mixer having two compartments separated by a perforated diaphragm or a thin metallic foil, one compartment being connected to a deuterium tank while the other communicates with a conduit through which the vapors entrained by the carrier gas pass to the reaction chamber.
Patent AU-729116-B2 (AU)
Title: Composite prosthesis for preventing postsurgical adhesions and method for obtaining same
Inventor: ORY FRANCOIS REGIS
IPC: A61L31/12
Filed: 1998-07-22
Granted: 2001-01-25
Abstract: The composite prosthesis comprises a prosthetic fabric having a three-dimensional structure separating two surfaces, one of which is open to post-surgical cell colonization. The composite prosthesis further comprises at least one film of a collagenous material linked to the other surface of the prosthetic fabric. The composite prosthesis may be used to prevent post-surgical adhesion.
Patent AU-567864-B2 (AU)
Title: Skin barrier for ostomates
Inventor: CILENTO RUDOLFO D
IPC: A61F5/44
Filed: 1982-11-04
Granted: 1987-12-10
Abstract: A composite skin barrier including a first adhesive component which fits around a stoma, a coupling element, and a second adhesive component which is flexible, light and has a degree of porosity. The second adhesive component contacts the skin at a distance from the stoma.
Patent AU-733597-B2 (AU)
Title: Apparatus and method for reclaiming useful oil products from waste oil including hydrogen injection
Inventor: SHURTLEFF EDWARD CALTON
IPC: C10M175/00
Filed: 1998-10-23
Granted: 2001-05-17
Abstract: An apparatus and method for reclaiming a useful oil product, from waste oil provides an evaporation chamber in which waste oil is heated and vaporized, preferably at a temperature which causes some cracking of the oil. Hydrogen is injected into the vaporized oil, so to cause saturation of at least some of the olefins in the vaporized oil. The vaporized oil is then condensed and recovered as a useful oil product. The apparatus operates at substantially atmospheric pressure, or a pressure only slightly above atmospheric pressure. Hydrogenation of the vaporized oil stabilizes the recovered oil, and prevents formation of tars and other heavier hydrocarbons, which can cause difficulties in use of the recovered oil.
Patent DE-1926787-B2 (DE)
Title: Hollow material roll extraction tool - has single-hand grip with toggle link to serrated expanding jaws
IPC: B65G7/12
Filed: 1969-05-24
Abstract: The tool is for use with materials wound onto hollow bodies and of different diameters, lying on top of each other in a shelf system, being particularly for handling textiles. It is equipped with a grip (6) for one hand, extended at one end to form a recess (8) for a toggle coupling (5) to one shank of two (2, 3), to which gripping jaws (1) are welded. These shanks intersect at axis pins (4, 7), and the jaws have annular teeth milled in them with a depth of 2mm and a pitch of 5mm. the design avoids any distortion of or damage to the material handled, even in the case of rolls of cardboard.
Patent DE-2038161-B2 (DE)
Title: Automatic railway wagon marshalling layout - has single carrier wagon for shunt conveyor and distance recorder with block travel indicator
IPC: B61J3/04
Filed: 1970-07-31
Abstract: The shunting zone for a railway marshalling yard has wagons automatically collected in classification tracks. This is divided into monitoring sections, with a common shunter, drive position, reverse position, traction drives and carrier wagons and a monitoring circuit for block movement. The shunt conveyor (4-7) has only a single carrier wagon (7). The monitoring circuit has an impulse transmitter (16), linked to the shunt conveyor drive (14), with a carrier wagon distance recorder (17). After block travel the drive is monitored by a block travel indicator (22) connected to the distance recorder.
Patent DE-2048096-B2 (DE)
Title: Pulse duration checking cct. for telecoms - checks pulse duration within stipulated limits checks amplitude and rejects noise
IPC: G01R29/027
Filed: 1970-09-30
Abstract: If the pulse duration lies within stipulated limits, the circuit itself produces a pulse which may be used to set a bistable and a display. If the received pulse is outside these limits, the circuit produces no output. The device consists essentially of two parts, one of which records the fact that a pulse has arrived. This it does by switching the magnetization in a transformer core of square-loop hysteresis material. The arrival of such a pulse initiates action in the second part of the device which then checks the amplitude duration and edge characteristics of the pulse. If these are satisfactory, an 'and' gate is satisfied and a clock pulse suitably delayed is produced via an amplifier in the first unit.
Patent DE-2059060-B2 (DE)
Title: Automatic camera with manual exposure correction - has photocell over variable transmission edge of thin filter
IPC: G03B7/0993
Filed: 1970-12-01
Abstract: The automatic camera has a photocell mounted behind a separate objective fitted alongside the main objective of the camera. A large filter plate is mounted to cover both objectives. In order to cater for some manual correction in the exposure the filter is swivelled in its mounting with the edge regions of the filter having variable transmission factors. This enables the user to over expose or under expose the film by a calculated amount. The filter mounting ring is provided with calibrated markings with over exposure in one direction and under exposure in the other direction.
Patent DE-2109374-B2 (DE)
Title: HV rotary isolating switch - has each switch arm made from two flat metal strips with one arm forcing strips of other apart in closed state
IPC: H01H31/28
Filed: 1971-02-27
Abstract: Insulating rotary supports (3, 4) for the h.v. isolator carry switch arms (5, 6) made from parallel flat strips (5a, 5b and 6a, 6b) of e.g. copper or aluminium. the ends of the strips of one arm(5) are brought together and then out-turned to provide contact elements (8) which in the engaged condition of the switch force the strips (6a, 6b) of the other arm apart against the action of a spring (9). In the engaged condition of the switch a pin (10) carried by one arm (5) engages in a slot in the strip (6b) of the other arm (6). Stops (12) for the pin (10) are provided on this other arm (6). In a modification, instead of the strips of one arm being out-turned they carry a contact element which cooperates with contact elements by the other arm.
Patent DE-2230822-B2 (DE)
Title: Loose leaf book binding machine - uses plastics strip with parallel fingers fed singly from hopper via channel with spreader at lower end
IPC: B42B5/10
Filed: 1972-06-23
Abstract: A machine for binding loose leaf books with plastic binders feeds the binders one at a time to the device (44) which uncoils the binder to fit it into the holes in the stack of pages. The plastic binders (10) are formed from strips parallel fingers to correspond to the holes in the pages (50). The binder (10) is then coiled about an axis perpendicular to the finger to form a long cylinder. The coiled binders (10) are fed from a hopper (18) into a slot (26). An oscillating U shaped member (56) cooperates with a second oscillating member (62) so that their combined motion controls the rate at which individual binders (10) drop to the uncoiling device (44). The coiled binders drop vertically down a channel which at the upper end has an opening corresponding to the dia. of a released binder. A guide strip from this opening has a spreader device (36) with grippers passing through spaces between the binder fingers.
Patent DE-2257306-B2 (DE)
Title: Switch with two fixed contact pairs - has pivoted deflector carrying moving contact and knife engaging slot in second pivoted sliding deflector
IPC: H01H5/06
Filed: 1972-11-22
Abstract: The switch has deflectors pivoting about parallel axes. One deflector (6) can slide perpendicular to its axis of rotation (5) in its longitudinal direction against the action of an elastic device (7). This deflector has a V-shaped support face (6b) at its free end parallel to its axis of rotation. The knife-like end (9b) of the second deflector (9) rests in this V-shaped face. The second deflector is pivoted at its other end by a bracket (8) and is moved from one end position to the other by a sliding piston (11). The piston is moved in one direction by a helical spring (12).
Patent IE-S80733-B2 (IE)
Title: A vehicle with hydraulically steerable wheels
Inventor: MCVICAR MARTIN
IPC: B62D5/20
Filed: 1998-07-22
Abstract: A vehicle such as a forklift truck has a pair of wheels (12L, 12R), each steerable by a respective hydraulic cylinder (24L, 24R) such that each wheel is turned to an angle determined by the position of the piston head in the respective cylinder. Each cylinder (24L, 24R) has a full bore side (36L, 36R) and a rod side (38L, 38R) and the full bore side (36L) of the cylinder (24L) is hydraulically connected to the rod side (38R) of the cylinder (24R). The vehicle further includes means (46) for supplying hydraulic fluid under pressure selectively to the rod side (38L) of the cylinder (24L) or to the full bore side (36R) of the cylinder (24R). In other embodiments the full bore sides of the two cylinders may be hydraulically connected together and the hydraulic fluid under pressure supplied selectively to one or other of the rod sides, or the rod sides of the two cylinders may be hydraulically connected together and the hydraulic fluid under pressure supplied selectively to one or other of the full bore sides.
Patent JP-H0472523-B2 (JP)
IPC: A43C11/14
Filed: 1987-01-22
Abstract: This ski boot fastener comprises a stretching lever having pivotally mounted therein at least two nipples each fulcrumed on a crosspin, and boot closing cables having each one end passing through the corresponding nipple and anchored to a cable head or socket movable along the cable and reacting against the corresponding nipple. The head or socket consists of an internally screw-threaded tube engaged by an externally screw-threaded core soldered to the cable end. The adjustment is obtained by rotating the socket.
Patent JP-H0739548-B2 (JP)
IPC: C08K5/06
Filed: 1993-02-12
Abstract: Organopolysiloxane compositions containing   (A) a salt of a water-soluble, organic or inorganic acid and organopolysiloxane having at least one SiC-bound organic radical with basic nitrogen, and   (B) alkoxylated alcohol and, if appropriate, (C) a salt of a water-insoluble organic acid and organopolysiloxane having at least one SiC-bound organic radical with basic nitrogen.
Patent JP-S6358452-B2 (JP)
IPC: B60Q1/05
Filed: 1984-02-23
Abstract: PURPOSE:To stabilize a light-up angle adjusting drive irrespective of and variation in supply voltage as well as to make it performable with a simple electrical element. CONSTITUTION:A connection line, which connects an output line of a switch gear 40 for tilt angle indication to an emitter of a transistor TR2, is broken off and then a duty control unit is interposingly inset in the broken wires. And, when up signals a=L appear in an output line of the switch gear 40, an output transistor 54b of a relay driver 54 between these signals a=L repeats on-off operations in pulse form at a constant period. Time width in time of ON is short at a time when supply voltage is high but long when it is low. And, when the transistor TR2 of a motor driver is in a state of being energized with current, a relay RY1 is energized or intercepted by on-off operation of the transistor 54b whereby the relay RY1 gives an energizing current to a motor 10. With this constitution, a constant current is given to the motor 10 irrespective of supply voltage. Therefore, a light-up adjuster becomes stable and accurate enough.
Patent JP-H0441245-B2 (JP)
IPC: C03B5/16
Filed: 1987-02-19
Abstract: A multi-outlet burner (32) for heating material comprises nozzles (42) which are positioned along a longitudinally extending portion (44) of the burner (32) that generally parallels the material surface. Combustion gas and fuel are combined at each nozzle (42) to produce a plurality of flames that are directed in a sweeping direction over the surface. The burner (32) has a first longitudinally conduit (56) for passing fuel, a second longitudinally conduit (54) for passing combustion gas and openings (72,74) to mix fuel and gas at the nozzles (42).
Patent JP-2847238-B2 (JP)
IPC: C07C319/20
Filed: 1996-02-28
Granted: 1999-01-13
Abstract: A process for the synthesis of fluorinated derivs. comprises a step in which a substrate is reacted with a cpd. comprising the association of a Bronsted base with a defined number (n) of HF species (n=3-20, pref. 15, and esp. 10). The substrate comprises at least one halo-carrying C of sp<3> hybridisation, attached to at least two halogens, of which at least one is a halogen of atomic number greater than F, bonded to at least one chalcogen.