baber/WOPTO huggingface dataset:
Patent UY-27952-A1 (UY)
Title: Nuevos derivados de benzoimidazol útiles como agentes antiproliferativos
Inventor: KATH JOHN CHARLES
IPC: C07D405/14
Filed: 2003-08-26
Abstract: La invención se refiere a compuestos de fórmula 1 y a sales, profármacos, y solvatos farmacéuticamente aceptables de los mismos, donde R1, R2, R3 y R4 son como se han definido anteriormente. La invención también se refiere a procedimientos para tratar el crecimiento celular anormal, tal como cáncer, en mamíferos administrando los compuestos de fórmula 1 y a composiciones farmacéuticas para tratar tales trastornos que contienen los compuestos de fórmula 1. La invención también se refiere a procedimientos para preparar los compuestos de fórmula 1
Patent UY-28698-A1 (UY)
Title: Compuestos de 1-(azolin-2-il)amino-1,2-difeniletano para combatir insectos, arácnidos y nematodos.
Inventor: BAUMANN DR ERNST
IPC: C07D263/28
Filed: 2004-12-23
Abstract: La presente invención se refiere a compuestos de 1-(azolin-2-il)amino-1,2-difeniletano de la fórmula general I en donde A es un radical de las fórmula A1 o A2: y en donde m es 0,1,2,3,4 o 5,n es 0,1,2,3,4 o 5, X es azufre u oxígeno, y en donde las variables R1, R2, R3, R4, R5a, R5b, R5c, R5d son tal como se definieron en las reivindicaciones, y a sus sales aceptables en agricultura. La invención también se refiere a un método para combatir plagas animales, seleccionadas de insectos, arácnidos y nematodos y a un método para proteger los cultivos del ataque o la infestación de insectos, arácnidos o nematodos, que comprende poner en contacto un cultivo con una cantidad de eficacia plaguicida de un compuesto de 1-(azolin-2-il)amino-1,2-difeniletano de la fórmula general I y/o al menos una de sus sales.
Patent UY-28887-A1 (UY)
Title: Procedimiento de preparación de derivados del ácido 1,5-difenilpirazol carboxílico
Inventor: PHILIPPE VAYRON
IPC: C07D231/14
Filed: 2005-05-06
Abstract: La presente invención se refiere a un procedimiento para la preparación de un compuesto de fórmula : en la cual: - W representa un grupo -COOR o un radical -CN; - R1 representa un átomo de hidrógeno o de halógeno, o un grupo alquilo (C1-C4); - R2 R3, R4, R5, R6, R7 representan cada uno, independientemente entre sí, un átomo de hidrógeno o de halógeno, o un grupo alquilo (C1-C4), alcoxi (C1-C4) o trifluorometilo; - R representa un grupo alquilo (C1-C4) o bencilo.
Patent UY-30036-A1 (UY)
Title: Uso de derivados heterociclicos benzo-fusionados de sulfamida para reducir los lipidos y los niveles de glucosa en la sangre
Inventor: REITZ ALLEN B
IPC: A61P3/00
Filed: 2006-12-19
Abstract: La presente invención es un método para los trastornos relacionados con la glucosa y trstornos relacionados con los lípidos que comprende administrar a un sujeto que lo necesita una cantidad terapéuticamente efectiva de uno o más derivados heterocíclicos benzo-fusionados de sulfonamida de fórmula (I) o fórmula (II) como se describe aquí. La presente invención se refiere, además a métodos de tratamiento que comprenden tratamiento concomitante con un agente antidiabético y agente anti-lipídico y/o un agente anti-obesidad.
Patent UY-30372-A1 (UY)
Title: Sistema inteligente de información controlada en semáforos
Inventor: ALBERTO AMORIN PALOMEQUE
IPC: G08G1/09
Filed: 2007-05-28
Abstract: El SIICS, como Tecnología de la Información y las Comunicaciones asociada a la Electrónica, se desarrolla y aplica en el campo de la Comunicación en vía pública, particularmente la comunicación semafórica. En este campo se inscriben, los carteles de información publicitaria, los de información turística e información vial y los carteles de senalización para ordenamiento del tránsito, incluidos los semáforos.
Patent UY-31527-A1 (UY)
Title: Derivados ciclopropilamina
Inventor: BRACKEMEYER PAUL J
IPC: A61K31/40
Filed: 2008-12-12
Abstract: Compuesto con formula (I) donde R1, R2, R3, R3a, R3b, R4, y R5 tienen los valores que se definen en la memoria descriptiva, que son utiles para tratar condiciones o trastornos que se pueden prevenir o mejorar mediante los ligandos del receptor de histamina-3. También se divulgan composiciones farmacéuticas que comprenden los ligandos del receptor de histamina-3, métodos para usar dichos compuestos y composiciones, y un proceso para preparar compuestos dentro del alcance de la formula (I).
Patent ES-165905-A1 (ES)
Title: UN DISPOSITIVO QUE CONTIENE UNA CAMPANA DE VACiO EN LA CUAL ES ENGENDRADO UN HAZ ELECTRoNICO
Filed: 1944-05-05
Abstract: Un dispositivo que contiene una campana de vacío en la cual se engendra un haz de electrones cuya velocidad es modulada por mediación de un sistema de electrodos por una oscilación de control de alta frecuencia y en el cual esta variación de velocidad se transforma en variación de intensidad caracterizado por el hecho de que el haz electrónico que penetra en el sistema modulador consiste en una mezcla con preferencia homogénea de grupo de electrones que provienen de por lo menos dos fuentes distintas pudiendo presentar además este dispositivo las particularidades siguientes tomadas por separado en las diversas combinaciones posibles: a) los grupos de electrones procedentes de por lo menos dos fuentes diferentes penetran en el sistema modulador a diferentes velocidades. b) La diferencia de velocidades de los electrones de los diversos grupos es regulable c) Los grupos de electrones que penetran en el sistema modulador proceden respectivamente de un cátodo y de por lo menos un electrodo colocado entre el cátodo y el sistema modulador que emite electrones secundarios y que permite el paso de los electrones. d) Los electrodos que emiten electrones secundarios se ponen en tensión positiva con relación al cátodo. e) Los grupos de electrones que penetran en el sistema modulador provienen de por lo menos dos superficies
Patent ES-182164-A1 (ES)
Title: UN SISTEMA DE RADIODETENCIoN POR TIEMPOS
IPC: G01S19/46
Filed: 1948-02-07
Abstract: Sistema de Radiodetección por tiempos para producir un tren de ondas constituido por una serie de oscilaciones de amplitud practicamente constante comprendiendo la generación de un tren de ondas atenuadas y compensación por el descenso del tren de ondas atenuadas por una pluralidad de oscilaciones del mismo.
Patent ES-188718-A1 (ES)
Title: Procedimiento para el aumento de resistencias de los hormigones
Filed: 1949-06-18
Abstract: Procedimiento para el aumento de resistencia de los hormigones que se caracteriza por someter las piezas de hormigón durante el fraguado a presión en moldes de acero mediante una prensa hidráulica que actúa durante un tiempo variable determinado con arreglo a las características de la pieza las cuales transcurrido el tiempo debido se extraen del molde y por haberse reducido con la presión la distancia intermolecular resultarán de una resistencia 200% superior a las ordinarias de mayor capacidad y aumento de peso específico impermeables y de mayor homogeneidad que las ordinarias.
Patent ES-190871-A1 (ES)
Title: MEJORAS EN LOS DISPOSITIVOS PARA QUITAR LOS DEPoSITOS DE LAS PAREDES DE TUBOS Y SIMILARES
Filed: 1949-12-19
Abstract: :Mejoras en los dispositivos para quitar los depósitos de las paredes de tubos y similares el cual comprende un árbol rotatorio provisto de mayales dispuestos a intervalos a lo largo del mismo y que desde él se extienden hacia afuera en diferentes direcciones llevando cada mayal un elemento cortante en su extremo exterior y estando el dispositivo adaptado para girar y atravesar axilmente en el tubo gracias a lo cual al funcionar los elementos cortantes de los mayales se hace que produzcan impactos sobre las paredes del tubo y desprendan de ellas los depósitos.
Patent ES-193329-A1 (ES)
Title: Nuevo amplificador
Filed: 1950-06-09
Abstract: El nuevo amplificador lleva un armazón en el que van montados los elementos que lo integran. Este armazón está formado por una palanca horizontal que le sirve de base por dos soportes perpendiculares a dicha plancha y por dos barras horizontales que unen entre si a aquellos soportes. Cada uno de estos lleva en la parte superior dos cojinetes y en la parte inferior cerca de la base otros dos cojinetes que sirven a otros tantos ejes. Además de esto cada uo de dichos soportes lleva solidario un cilindro hueco que servirá a la vez de eje al centrifugador correspondiente y de cojinete al eje central del nuevo amplificador.
Patent ES-196038-A1 (ES)
Title: UNA INSTALACIoN DE TURBINA DE GAS.
Filed: 1951-01-05
Abstract: Instalación de turbina de gas en la cual le es aportado calor al agente del ciclo en una cámara de combustión o un permutador térmico caracterizada porque el agente del ciclo en la aportación de calor está a la presión del ambiente por apertura del ciclo delante de la turbina.
Patent ES-267086-A1 (ES)
Title: Process for producing l-glutamic acid
IPC: C12P13/18
Filed: 1961-04-22
Abstract: L-Glutamic acid is prepared by aerobic culture of a micro-organism of the genus Brevibacterium in a culture medium including one or more carbohydrates, one or more amino acids, a nitrogen source other than an amino acid, one or more inorganic salts and one or more of the nutrients desthiobiotin, biotin-d-sulphoxide and biocytin. Suitable micro-organisms are B. roseum, B. flavum, B. immariophirium, B. Saccharolyticum, and B. lactofermentum. Suitable nitrogen sources are inorganic and organic ammonium salts, urea, nitrates, nitrites, aqueous ammonia and ammonia gas. Specifications 873,448, 876,943 and 889,187 are referred to.
Patent ES-273492-A1 (ES)
Title: Method for the preparation of codeinone from thebaine
IPC: C07D489/02
Filed: 1962-01-09
Abstract: Codeinone is prepared by reacting thebaine or a salt thereof with a hydrohalic acid in an anhydrous organic medium and adjusting the pH of the reaction mixture to 8-12 by treatment (preferably in an aqueous medium) with a basic agent selected from alkali and alkaline-earth metal hydroxides, carbonates and bicarbonates, ammonia, salts having an alkaline action, an organic bases.
Patent ES-337068-A1 (ES)
Title: Two-for-one twisting machine
IPC: D02J3/16
Filed: 1967-02-20
Abstract: A two-for-one twisting machine has provision to singe the yarn. Yarn 1 from a spool 2 is drawn off upwardly and passed downwardly through a spindle 3, leaves the spindle radially between a cage 4 and a balloon limiting device 5, passes through a guide ring 13, around a stripper 12, over a guide 6 and is wound by a traversing mechanism 7 onto a package 8 driven by a friction roller 9. Between the ring 13 and a guide eye 19 the balloon of yarn passes through the gas flames of a singeing device 11. The device 11 may be of arcuate shape (Fig. 2, not shown), circular shape (Fig. 5, not shown) or may be an electrically heated ring (Fig. 6, not shown) with a polygonal shaped inner surface whose flats contact the yarn. In Fig. 10 (not shown) the yarn is singed above the guide 19 where it is caused to revolve in a inverted cone orientation by a guide (24) on a plate that is driven by a friction wheel. In Fig. 11 (not shown) the rotation is cylindrical and is caused by two guides driven by the friction wheel. In Fig. 12 (not shown) the singeing device is a roller with gas jets driven in the opposite direction to the passage of the yarn. In Fig. 13 (not shown) the roller is electrically heated and in Fig. 14 (not shown) the electrical heating is radiant so that only the portion of the roller over which the yarn passes is heated. In Fig. 15 yarn 44 from a stationary package is drawn upwardly through a rotating spindle 45, radially outwardly and then downwardly through a tube 49 to be wound by a traversing mechanism 51 onto a package 52 that does not rotate with the spindle 45. In Figure 17 yarn from a stationary package 2 is drawn upwardly through a rotating spindle 61 from which it passes radially to a rotating guide 66. The package 2 is maintained stationary magnetically. Fig. 18 (not shown) shows a similar arrangement in which the package rotates. The guide ring 13 (Fig. 3, not shown) is in three pieces with a ceramic facing 14. The stripper 12 is a roller with slot of zig-zag formation around which the yarn passes.
Patent ES-338758-A1 (ES)
Title: Apparatus for the continuous casting of metal
IPC: B22D11/06
Filed: 1967-03-31
Abstract: A continuous casting mould 1 is formed by four flexible endless sheet-metal belts 5 movable on rollers 6, 7 and 8, the face of the belts forming the mould walls being inclined inwards towards the bottom of the mould to compensate for shrinkage of the solidifying strand 14, and the axis 12 of each mould wall being also inclined laterally relative to the mould axis, so that the four walls of the mould form a section of an inverted rectangular based right pyramid. One edge of each of the belts 5 is forced against the surface of an adjacent belt to seal the mould corners. Each belt 5 moves on rollers 6, 7 and 8 and spring-biased pressure rollers 21-24 that are mounted on a frame 16 that is movable with two degrees of freedom, i.e. rotationally about two horizontal axes formed through a pivot (36) (Figs. 3 and 4, not shown), by an hydraulic jack (39) to ensure that the mould walls conform with the tapered form of the solidifying strand 14. The belts 5 are cooled by water jets 30 and the rollers 6, 7 and 8 may have projections thereon to enable cooling water to pass between the rollers and belt. The strand 14 is lowered by extraction rolls 15, 15a
Patent ES-339076-A1 (ES)
Title: Cooling tower.
IPC: F28F25/04
Filed: 1967-04-08
Abstract: In a cooling tower wherein water to be cooled is conveyed above irrigation plates 14 by channels 1, said channels are provided with base apertures 2 and with overflows 3 and 4, water emerging from the apertures 2 being evenly distributed over the plates 14 via distributer devices 16, while surplus water flowing through overflows 3 and 4 reaches the distributer devices 16 via guide means 17. In other embodiments, each individual channel 1 can either have a further outer channel (Figs. 4-6) around it, the latter channel being provided with a discharge which concentrically surrounds the outlet socket of the internal channel, or have said outer channel replaced by a guiding device consisting of a box (Figs. 7-9) enclosing said inner channel. Further embodiments include subdividing the channel 1, by a partition wall (11, Fig. 10) situated longitudinally in the channel, into two parts, the surplus from the water conveyed into the first part flowing into the second part via overflows situated in said intermediate wall, or as in another case, providing in the outlet of the channels, concentric pipes (12, Fig. 13) of small diameter, said pipes terminating at various heights.
Patent ES-341855-A1 (ES)
Title: Compass card autopilot with 360 degree directional control
IPC: G05D1/02
Filed: 1967-06-15
Abstract: In an automatic pilot (see Division G3) the card 30 of a liquid-filled magnetic compass is mounted eccentrically within a housing 40 so that, when a ship carrying the compass deviates from a desired heading, photo-conductive cells 57, 58 become unequally illuminated in a corresponding sense from lamps 55, 56. The desired heading is selected by setting a dial 70 which rotates housing 40 by means of a card 76. Cells 57, 58 are connected to a printed circuit associated with transistors on a board 50 which is connected by a cable to a power transistor circuit controlling a rudder servomotor.
Patent ES-343304-A1 (ES)
Title: Pyrroline derivatives
IPC: C07D207/26
Filed: 1967-07-21
Abstract: Novel compounds of formula and acid addition salts thereof, wherein R and R1 are each H or alkyl and the phenyl nucleus may be unsubstituted or substituted by one or more of alkyl, alkoxy, OH, halogen, NO 2 or amino substituents, are prepared in the case of amino substituted phenyl by reduction of the corresponding nitro substituted phenyl compound and in all other cases either by reaction of the amine HNRR1 with an ether or thioether of Formula (III) wherein Y is O or S and R 1 is C 1-3 alkyl, or by reaction of HNRR1 with a complex of formula wherein T is -OPOCl 2 , -OCOCl or -OSOCl, which is prepared in situ from the pyrrolidone of Formula (V) Ethers of Formula (III) above (Y=O) are prepared by reaction of trialkoxonium boron fluoride and a pyrrolidone of Formula (V), which is itself prepared by decarboxylation of the 3-carboxy derivative obtained by hydrolysis of the 3-methoxycarbonyl derivative formed by reductive cyclization of methyl 2-methoxycarbonyl - 3 - (optionally substituted phenyl)- 4-nitrobutyrate obtained by condensation of dimethyl malonate and the appropriate 1-nitro- 2-phenylethylene compound. 4 - (4 - Chlorophenyl) - pyrrolidone - 2 is prepared by action of Cu 2 Cl 2 on the diazotized amino compound. 1 - Nitro - 2 - (2,6 - dichlorophenyl) - ethylene is prepared by condensing 2,6-dichlorobenzaldehyde and nitromethane. Thioethers of Formula (III) above (Y=S) are prepared from thioketones of formula which are obtained by action of P 2 S 5 on the corresponding pyrrolidones. Pharmaceutical compositions having antidepressant and hypertensive effects and in conventional forms for oral, rectal, topical or parenteral administration comprise an above novel compound and a diluent or carrier therefor.
Patent ES-351750-A1 (ES)
Title: Method and apparatus for winding beams
IPC: B65H54/00
Filed: 1968-03-18
Abstract: Tape yarns are passed over a roller 21 immediately adjacent the location at which the yarns begin to wind on to a beam in order to ensure that the yarns lie with their longer dimension parallel to the beam axis. The roller 21 is carried by a pantograph link system 12, 13, 18, 19, attached to a ram 15 for lifting the roller, the pantograph ensuring that the roller maintains the same relative position in relation to the winding point regardless of the condition of winding. The yarn passes through a comb 38, fluted roller 37, draw roller 35, and yarn tension control roller 29 to the roller 21. The roller 29 is mounted on levers 31 carried by a strain gauge 32 and maintains the tension constant for different angles of winding.
Patent ES-353015-A1 (ES)
Title: Carbamate leveling agents in emulsion floor polish
IPC: C08K5/205
Filed: 1968-04-22
Abstract: An aqueous emulsion floor polish composition comprise., in its solids content, a major proportion by weight of a water-insoluble thermoplastic polymer, other than a waxy material, and a waxy material which is a wax or emulsifiable polyethylene, a minor proportion by weight of an ammonia-soluble thermoplastic levelling resin, and from to 2% by weight of a levelling agent, which is at least one carbamate having the general formula in which R 1 is an unsubstituted C 6-10 alkyl radical or mixtures thereof and R 2 and R 3 are hydrogen, unsubstituted C 1-4 alkyl radicals or monohydroxy substituted C 1-2 alkyl radicals. The levelling agent may be 2-ethylhexyl carbamate, 2 - ethylhexyl N - methylcarbamate, 2 - ethylhexyl N,N - dimethylcarbamate, nhexyl carbamate, or mixed hexyl-decyl carbamates, iso-octyl carbamates, iso-octyl N- methylcarbamates, octyl - decyl carbamates, octyl-decyl N-methylcarbamates or decyl carbamates. The water-insoluble polymer may be polystyrene blended with shellac, a polyacrylate, or copolymers of an acrylate or acrylic acid with acrylonitrile or styrene respectively. The ammonic-soluble resin may be partially esterified modified rosin and styrene/maleic anhydride copolymers. The polishes may also contain diethylene glycol (mono-ethyl or -methyl) ether, ester and microcrystalline waxes, oleic acid, potassium hydroxide and morpholine.
Patent ES-363681-A1 (ES)
Title: Extrusion head for continuously extruding a compound strand of plastic materials
IPC: B29C48/05
Filed: 1969-02-14
Abstract: Apparatus for manufacturing a strongly integrated compound strand formed by pressing together at least two different plastic materials. A first extruded plastic strand is pressed through a hollow cylindrical die and a second extruded plastic strand is pressed through a generally radial passageway into an annular portion. A rotary part rotated about the axis of the cylindrical die includes a portion of the passageway for helically winding the second plastic strand into the first plastic strand.
Patent ES-367144-A1 (ES)
Title: Magnetically biased tank vent
IPC: F16K31/08
Filed: 1969-05-12
Abstract: The disclosure is similar to that of Specification 1,222,745 but the claims differ in scope.
Patent ES-367484-A1 (ES)
Title: Thermal neutron source
IPC: G21C1/30
Filed: 1969-05-21
Abstract: A beam of thermal neutrons, derived from a nuclear reactor core is passed to an external experimental facility and the neutron energy is controllable from the reactor exterior. Neutrons from the reactor core pass through the neutron moderating graphite block, 7, and the channels, 14 and 17 to the exterior. The temperature of 7 is adjusted by radiation energy derived from source, 10, and directed on to 7 along the channels 12, 14. Changes in the temperature of block, 7, cause corresponding variations of neutron energy. The source, 10, may be a magnetron, a laser or an arc furnace.
Patent ES-375722-A1 (ES)
Title: Short term peak shaving of natural gas
IPC: F17C9/02
Filed: 1970-01-21
Abstract: Apparatus and method for "peak shaving" storage of gas in a gas distribution system wherein the pressure varies from a maximum when demand is low to a minimum when demand is high, the method comprising cooling gas, in a gas storage chamber in open fluid communication with the system with a frozen cooling medium having a freezing point approximately midway between the minimum and maximum boiling points of the gas in the system. When the pressure in the system is high, gas in the chamber liquifies and is stored when the pressure in the system is low gas in the chamber vaporizes and is available for use.
Patent ES-375926-A1 (ES)
Title: 1-0,0-diethylthiophosphonyl-indazoles
IPC: A01N57/32
Filed: 1970-01-27
Abstract: Novel compounds of the general formula wherein R 1 is a halogen atom, a C 1 -C 4 alkyl radical, or a phenyl, cyano, carbamoyl or thiocarbamoyl group and R 2 is H, halogen, or NO 2 , are obtained by reacting (C 2 H 5 O) 2 P(S)Cl with an indazole derivative of the formula wherein M is H or an alkali metal. The reaction is preferably carried out in an aprotic polar solvent e.g. 2-N-methyl pyrrolidone, dimethylformamide, hexamethylphosphotriamide or dimethylsulphoxide at 0-30 C. When M is an alkali metal the alkali metal derivative can be prepared in situ e.g. by treating the indazole in which M is H with an alkali metal alkoxide in an alcohol. The products have insecticidal and fungicidal properties and may be admixed with one or more solid or liquid diluents or adjuvants to form conventional compositions which may also contain wetting, dispersing or emulsifying agents. 3 - Carbamoyl - 5 - nitroindazole is obtained by the action of nitric acid on 3-cyanoindazole in solution in sulphuric acid. 3 - Thiocarbamoylindazole is obtained by the action of HCl and O,O-diethyldithiophosphorie acid on 3-cyanoindazole in benzene solution. 3 - Carbamoyl - 5 - chloroindazole is obtained by the action of sulphuric acid on 3-cyano-5- chloroindazole which is itself obtained by reacting sodium chlorate with 3-cyanoindazole in solution in acetic acid.