baber/WOPTO huggingface dataset:
Patent BG-106018-A (BG)
Title: Data processing system using a dual monitor and controlling method of such system connected in a network
Inventor: LEE EUN SEOG
IPC: H04N/
Filed: 2001-10-16
Abstract: The invention relates to a data processing system using a dual monitor as a display device, displaying different contents. It improves the effectiveness in using the computer and the advertising effect. The system includes, memory for data processing using programs (32, 34), an input device for inputting data (40, 42), a first graphic video generating adapter (VGA) (46) for generating screen data for a result processed by programs, a second graphic video generating adapter (VGA) for the generation of video signal for displaying the results of the work of the programs, the results being different from those displayed by the first VGA processor (30) processing the input data produced by the input device using the memory and outputting the processed result through the first and second VGAs (46, 48), a first monitor (12) for displaying screen data from the first VGA, and a second monitor (14) for displaying screen data from the second VGA. A digital camera (20), a speaker (22), microphone (24), TV and radio receiving attachment (50) and a sound attachment (52) can also be included in the system. 22 claims, 2 figures
Patent BG-107216-A (BG)
Title: 2-aminocarbonyl-9h-purine derivatives
Inventor: MANTELL SIMON J
IPC: A61K31/7076
Filed: 2002-10-23
Abstract: The present invention relates to compounds of formula and pharmaceutically acceptable salts and solvates thereof, and to processes for the preparation of intermediates used in the preparation of, compositions containing and the uses of such compounds. 73 claims
Patent BG-110448-A (BG)
Title: An ecological collector oval-shaped multifunctional infrastructural tunnel
Inventor: TSOKOV TSANKO
IPC: E03F3/02
Filed: 2009-08-19
Abstract: This tunnel is intended for gathering together all kinds of engineering infrastructure: water supply, drain system, telephone installations, Internet, electrification, street illumination, and others. It is installed under the pavement in close proximity to the curb stone of the traffic way. The bottom of the tunnel (1) is formed in such a way that rain water in different quantities can be gathered and transported to the nearest sewer. In the wall of the tunnel (1) a parabolic open channel (2) is installed which disposes everyday waste water in the treatment station. The wall radius of the open channel (2) is the same as that of the oval tunnel (2) so that it sticks firmly to the wall of the tunnel (1) at various heights. Also a water supply tube (4) with a stop valve (6) is installed for the work of a water supply unit positioned closely to the tunnel (1). Various electric supply nets (5) for low and high voltage are also installed. The tunnel serves simultaneously for installation,repair, maintenance and testing of the condition of infrastructure as well as for a universal rain pouring without the usual inspection pits. The access to the devices placed in it by the respective authorized persons is easy and does not impose the necessity of digging up the traffic way and the footpath pavement.
Patent CN-1317746-A (CN)
Title: 电脑保安和家电智能控制系统
Inventor: GUOYING CHEN
IPC: G06F13/10
Filed: 2000-04-12
Abstract: 一种电脑保安和家电智能控制系统，用于家庭，办公室，工厂，酒店，学校等，它包括电脑主机以及与电脑主机电连接的分电脑装置，包括电子门钥匙分电脑装置，红外线灯光遥控分电脑装置，家电控制器分电脑装置，紧急求救遥控器分电脑装置，还包括移动感应器分电脑装置，电话转换器分电脑装置，电脑主机通过预定程序对各分电脑进行控制，各分电脑按各自预定程序独立运作，还包括远距离遥控，远距离监听，电话未挂断提示等功能。
Patent CN-1309882-A (CN)
Title: 玉米种子丸粒化加工工艺
Inventor: HUANG GUIQIN
IPC: A01C1/06
Filed: 2000-02-22
Abstract: 一种玉米种子丸粒化加工工艺,属于农业播种前种子的处理方法,特别是涉及玉米种子包衣丸粒的加工方法。为了解决现有玉米播种时对种子的浪费,以及为了降低现有播种机的复杂化,本发明提供一种通过在丸化机中旋转,使玉米种子外粘有各种玉米生长所需物质,并且种子形状、尺寸基本相同的玉米种子丸粒化加工工艺。
Patent CN-1354962-A (CN)
Title: 在无线通信系统中分配资源的方法
Inventor: SOMMER V
IPC: H04J13/18
Filed: 2000-03-06
Abstract: 根据本发明,由基站提供的一部分信道脱离了所属基站控制器的专门控制。通过第二基站控制器的协作可以改变该部分信道的数量。通过为所述第二基站控制器预留信道可以降低信令耗费。脱离所属基站控制器专门控制的那部分信道不是逐帧地、而是在很大的间隔内实现改变的。该资源分配可以以FDD模式和TDD模式应用于具有CDMA用户分离的无线通信系统中。
Patent CN-1309337-A (CN)
Title: 机体内装有sim卡的电话手表
Inventor: MARTIN J C
IPC: H04B1/3827
Filed: 2001-02-16
Abstract: 电话手表(1)具有一个内部装有用于接纳SIM(用户识别模件)卡(4)的机体(3)的后盖(2)。带有铰链(6)的盖子(5)封闭上述的后盖(2)。设置了保证盖子(5)的密封性的密封机构(8)和锁紧机构(7)。上述的铰链(6)安装成被完全封闭在后盖(2)之内。
Patent CN-1408590-A (CN)
Title: 阻燃、防爆安全加油站
Inventor: HUANG XIAODONG
IPC: A62C3/06
Filed: 2001-09-25
Abstract: 一种阻燃、防爆安全加油站，它是一种从根本上杜绝贮油罐爆炸的新型加油站。它包括有贮油罐和加油机，在贮油罐的左、右两端连接有加油室，加油室内设有加油机及防火卷帘门。贮油罐通过输油管道和防爆阀门与加油机相连接。在贮油罐和输油管道的外部有防火保温材料，在贮油罐内充满有抑爆网或者是抑爆球。该加油站将贮油罐外防火和贮油罐内防爆、阻燃合理的结合在一起，可从根本上杜绝贮油罐的爆炸。对加油站的安全管理和对周边环境限制可以放宽，而且加油站的占地面积少又便于整体安装，大大降低建设成本和日常管理费用。
Patent CN-1361576-A (CN)
Title: 旋转电机
Inventor: TOSHINORI TANAKA
IPC: H02K23/30
Filed: 2001-12-21
Abstract: 一种旋转电机,具有:轭铁;整流子片(112)间并列连接有n个(n为磁极(102)的极数与槽数(101)的数的公约数,但在2以上)绕组部(4B),并且,该绕组部(4B)相对机械角360度相互对称配置,从整流子片(112)看,在圆周方向最近的绕组部(4B)的其他绕组部(4B)的各导线部(5B)向同一圆周方向导出。配置于机械上平衡的位置的绕组部导线部不会交叉、可提高绕线的作业性、并可抑制绝缘不良。
Patent CN-1463750-A (CN)
Title: 用于生产乳白鱼肝油的乳化剂
Inventor: JI MINGHOU
IPC: A61P3/02
Filed: 2002-06-19
Abstract: 本发明公开了一种用于生产乳白鱼肝油的乳化剂，以重量百分比计，由65－85％田菁胶、10－20％瓜尔胶和5－15％黄原胶组成。本发明以田菁胶为主要成份，该产品为国内生产，可大大降低该乳化剂的成本。本发明所提供的乳化剂用于乳白鱼肝油的生产，其鱼肝油的乳化性能好，且所含的维生素保存效果好，乳化体的保存期(室温)在2年以上。
Patent CN-1479340-A (CN)
Inventor: JIAN YUTING
IPC: H01J17/49
Filed: 2002-08-29
Abstract: 本发明提供一种等离子体显示器的电极对结构。该电极对结构包含有一第一金属电极设置于一前基板表面，以及一第二金属电极与该第一金属电极平行地设置于该前基板表面，其中该第一金属电极与该第二金属电极分别由多个六边形且中空的金属结构串联而成。
Patent CN-1424042-A (CN)
Title: 山楂叶总黄酮滴丸制剂及其制备方法
Inventor: SU JUAN
IPC: A61K31/7048
Filed: 2002-12-19
Abstract: 本发明是一种山楂叶总黄酮滴丸制剂及其制备方法。该滴丸制备以山楂叶总黄酮为主要成分，与聚乙二醇、泊洛沙姆按一定工艺组配制成。本发明的滴丸制剂与其它剂型相比，药物起效快、生物利用度高，制备工艺适合于工业化生产。
Patent CN-1452114-A (CN)
Title: 半导体存储装置
Inventor: TATSUYA KUNIKIYO
IPC: H01L21/8246
Filed: 2002-12-16
Abstract: 在包括滤波器和放大器等的模拟电路中，提供一种能修正制造工序中的加工离散引起的各元件的值的离散的模拟电路。滤波器FT1是将磁隧道电阻MR和电容器C连接成L型的低通滤波器。另外，在滤波器FT1中，端子T1及T2是输入端子，端子T3及T4是输出端子。另外，通过电流源IP供给改变磁隧道电阻MR的磁化方向的电流。
Patent CN-1489837-A (CN)
Inventor: ALBERTH WILLIAM P
IPC: H04B7/185
Filed: 2002-01-18
Abstract: 本发明公开了一种卫星定位系统使能的移动终端(12)及其定位方法，其具有一个卫星定位系统信号接收接口(例如一个GPS接收器(14))一个与该卫星定位系统信号接收接口相连接的信息处理器(22)，该信息处理器控制卫星定位系统信号接收接口，用以接收卫星定位系统信号，基于卫星定位系统信号、基于卫星定位系统的位置方位产生速率指令，可以确定移动终端的定位。
Patent CN-1500317-A (CN)
Inventor: BEOM-SIK BAE
IPC: H04W28/00
Filed: 2002-03-25
Abstract: 一种在移动通信系统中的反向传输控制方法，在接收到命令提高或降低从基站在前向控制信道上接收的反向数据率的前向信息之后，如果前向信息命令反向数据率提高，则移动台确定是否在接收前向信息之前在反向控制信道上被发送到基站的前一个速率提高可行信息指示提高反向数据率可行。如果所述速率提高可行信息指示反向数据率提高可行，则移动台将当前反向数据率提高到等于或小于最大反向数据率的数据率，并且移动台以所提高的反向数据率发送反向数据。
Patent CN-1571917-A (CN)
Title: 粉粒料计量装置
Inventor: SHOZO KAWANISHI
IPC: G01G19/393
Filed: 2002-10-22
Abstract: 本发明提供一种粉粒料计量装置，所述粉粒料计量装置在构成组合秤的多个单元秤(10)上，分别设有安装于粉粒料斗(12)下部的截止门(11)、将供给自截止门(11)的粉粒料作暂时保持的供给料斗(13)、对供给自供给料斗(13)的粉粒料进行计量的闸门式计量料斗(14)、将自供给计量料斗(14)排出的粉粒料集聚、供给至包装机的聚料滑槽(16)。计量料斗(14)上安装有负载传感器(15)。该负载传感器(15)为进行计量料斗(14)内的组合运算而对粉粒料重量进行计测。在截止门(11)、供给料斗(13)、计量料斗(14)及聚料滑槽(16)的各构成要素之间设有防尘皱纹软管(18)。由此，可对粉粒料进行高速计量。
Patent CN-1517320-A (CN)
Inventor: YANG SONG
IPC: B09B3/00
Filed: 2003-01-14
Abstract: 本发明公开了一种利用流化床煤矸石沸腾炉渣(灰)来代替传统工程细集料，包括天然砂和人工砂，在现浇混凝土及混凝土预制构件中的应用，代替传统工程细集料的比例为20％－100％，与水泥、石灰膏、粗骨料的重量配比为：1.5－4∶1∶0－0.1∶2－6，本发明解决了长期以来流化床煤矸石沸腾炉渣(灰)给环境带来的污染问题，能广泛应用于预制空心楼板、花块(格)、隔热板、地砖、轨枕、盖板等混凝土预制构件以及现浇混凝土，为工业废渣的综合利用开辟了一条新路。
Patent CN-1496988-A (CN)
Inventor: DING MINGWU
IPC: A01N43/50
Filed: 2002-01-04
Abstract: 一类具有杀菌活性的2－(4－甲硫苯氧基)－5－呋喃亚甲基咪唑啉酮衍生物。通式为下式的具有杀菌活性的咪唑啉酮衍生物，式中Ar表示(取代)苯基，取代基为3－氯、4－氯、4－甲基。上述化合物对稻瘟菌、水稻纹枯菌、芦笋褐斑菌、苹果轮纹菌、小麦赤霉菌及棉花枯萎菌具有良好的抑制活性，可用作杀菌剂。
Patent CN-1672287-A (CN)
Inventor: SEXTON ROBERT J
IPC: H01P3/02
Filed: 2003-05-28
Abstract: 一种非均匀传输线包括至少一个构图传导层(102、104)、与(多个)构图传导层(102、104)相邻的电介质层(103)和包围该(多个)构图传导层和电介质层的绝缘层(101、105)。
Patent CN-1682138-A (CN)
Inventor: WAYNE BALCH ERNEST
IPC: G02B6/13
Filed: 2003-07-24
Abstract: 适于制造波导(30)的方法，该方法包括：测量光子器件(31，32，34)相对于衬底(20)的位置偏差；生成计算机可读的指令，用于使用多个图形元素(16)以形成波导；以及按照计算机可读的指令在衬底上为波导进行照相排版。中间掩模(14)包括多个图形元素，该多个图形元素中至少一个包括锥形端部。波导(30)包括多个波导分段(22)，该多个波导分段中的每一个包括锥形端部且与该多个波导分段中其他的至少一个相邻接。
Patent CN-1788501-A (CN)
Title: 在通用移动通信系统无线接入网中实现区分服务的方法
Inventor: LIU CHENG ZHAO
IPC: H04L47/31
Filed: 2003-06-18
Abstract: 本发明提供一种在基于IP传输的通用移动通信系统(UMTS)无线接入网中应用区分服务(DiffServ)实现服务质量(QoS)保证时IP分组分类与区分服务码点(DSCP)标记的方法。本发明对于在节点B侧Iub接口外出方向的数据流、在无线网络控制器侧Iub接口外出方向的数据流以及在无线网络控制器侧Iur接口外出方向的数据流，按照各个数据的流向和处理方式进行分类，并且按照优化QoS与无线资源的原则分配和调整所分类的各个数据流的优先级。当网络出现拥塞时，级别高的数据流在排队和占用资源时比级别低的数据流有更高的优先权，同一队列中丢弃优先级越低的分组。区分服务只包含有限数量的业务级别，状态信息的数量少，因此实现简单，扩展性较好。
Patent CN-85107808-A (CN)
IPC: H05K3/30
Filed: 1985-09-10
Abstract: 本发明公开了一种在印刷电路板上安装芯片型电路元件的方法及其作用设备，它不需要配置一个X-Y工作台从而简化了这种装置的结构，并且缩短了把一个电路元件安装到印刷电路板上所需的时间。由装在各安装头中的许多抽吸头来吸起芯片型电路元件，它们被传送到一个对中和翻转部件，然后被逐步地安装到一块印刷电路板上。安装头的特点在于当它在Y方往复运动一次时，在X向可作往复运动多次。
Patent CN-87104817-A (CN)
Title: 用于防污涂层的热喷粉
IPC: C09D5/14
Filed: 1987-07-11
Abstract: 本发明说明了一种复合热喷粉含有由热软化树脂和一种对海洋生物有毒性的如铜或氧化铜那样的粉状矿物组成的颗粒，粉状矿物可以具有一个大于0.25平方米/克的比表面积，最好是薄片形的。
Patent CN-87106177-A (CN)
Title: 唾液酸糖基胆甾醇，它们的制备方法及含有它们的治疗神经病的药物
IPC: C07J17/00
Filed: 1987-09-03
Abstract: 本发明是关于唾液酸糖基胆甾醇的钠盐。本发明的化合物具有很好的水溶解性，因此该化合物作为治疗由于周围神经和中枢神经损伤所致的各种疾病的药物是十分有用的。
Patent CN-1039544-A (CN)
Title: 十字轴毛坯成型工艺及模具
Inventor: HUIYU WANG
IPC: B21C25/02
Filed: 1989-04-08
Abstract: 一种十字轴温、热挤压成型工艺及模具，它是首先将棒料加热至一定的温度，然后放入挤压模中挤压成型，改变了原来的胎模锻打加工十字轴毛坯的方法，大大提高了原材料的利用率，减少加工量，并且采用本发明的方法，加工十字轴毛坯的尺寸稳定，降低了废品率。
Patent CN-1047124-A (CN)
Inventor: QIHUA ZHANG
IPC: D06M13/395
Filed: 1989-05-10
Abstract: 一种无纺布类织物用防水整理剂，主要由脂肪酸、表面活性剂、有机胺类交联剂、有机酸酯、有机酸盐、分子结构内有异氰酸基、活泼羟基的化合物及水组成，有防水效果好、价格低廉、处理效率高、生产工艺简便的优点，主要可应用于无纺布类的防水整理工艺中。
Patent CN-1049361-A (CN)
Title: 聚碳酸亚烃酯离散粒子的制备方法
Inventor: HOSTETLER DONALK E
IPC: C08J3/09
Filed: 1989-08-09
Abstract: 选用能够在高温下使聚碳酸亚烃酯完全溶解而
在低温下却又完全不溶解该聚合物的适宜的溶剂体
系制备适用于许多运输、加工与应用场合的聚合物离
散粒子，其粒径被控制在大约30-300微米。
Patent CN-1085561-A (CN)
Inventor: DENINNO MICHAEL PAUL
IPC: C07J71/00
Filed: 1993-06-25
Abstract: 本发明公开了一些可用作为降低血胆甾醇药物
和治疗动脉粥样硬化药物的甾族苷。
Patent CN-1131310-A (CN)
Title: 使用cd并具有双用途cd-rom驱动器的视象歌曲伴奏装置
Inventor: CHOI KWANG-SIK
IPC: G10K15/04
Filed: 1995-10-20
Abstract: 本发明的视象歌曲伴奏装置包括一个CD重放装置，指令输入装置，用于输入指令信号，显示装置，CD-ROM解码器，CD-OK重放装置，CD-ROM接口装置，音频选择器，视频选择器，主控制装置，通过识别盘的种类控制音频选择器和视频选择器的信号选择，有选择地控制CD-OK重放装置和CD-ROM接口装置的CD-ROM数据输入使能状态。
Patent CN-1131454-A (CN)
Inventor: GANCHEV NIKOLAI IVANOV
IPC: F16D11/10
Filed: 1995-07-21
Abstract: 一种端面销离合器，用于转换机械的齿轮传动装置的速度。端面销离合器包括一主体，在主体中装有一个或多个可自由移动的销(4)，以及拉伸弹簧(6)，弹簧(6)钩在夹住主体的板(8)上。这方案使设计简单，消除了转换速度时存害的游隙及噪音，在操作中可方便地转换速度。
Patent CN-1190744-A (CN)
Inventor: ZENG WENZUO
IPC: G02B7/28
Filed: 1997-02-14
Abstract: 一种用于多镜头光学系统的自动调焦系统,对多镜头光学系统自动进行锐度与放大倍率的校准,它包含多个归位传感器、多个微传感器、多个镜头、一取像装置、一取像装置控制电动机、一基座操控电动机与一镜头切换电动机。利用取像装置控制电动机与基座操控电动机分别控制取像装置与镜头的移动,来进行锐度与放大倍率的校准,直到锐度与放大倍率皆符合系统要求为止。
Patent CN-1284041-A (CN)
Title: 半导体晶片放入/取出处理系统
Inventor: DAVIS JEFFRY A
IPC: H01L21/00
Filed: 1998-12-15
Abstract: 用于处理如半导体晶片类物品的处理器,包括限定封闭的洁净处理腔室的机箱和至少一个设在该腔室内的处理工位;邻接部分有连接开口,装有待处理物品的容器经开口被装入或从中卸载。邻接部分以卫生的方式与处理腔室分开。适于与所述容器密封的物品提取机构能够把被装于容器内的物品送入处理腔室内,而不使这些物品在所述邻接部分中暴露于周围的空气条件下。本物品处理器还包括物品插入机构,适于与放在邻接部分内的容器密封。
Patent CN-1324525-A (CN)
Title: 第三代移动无线系统中的搜索接收机
Inventor: FALKENBERG A
IPC: H04W24/04
Filed: 1999-10-27
Abstract: 为了与已知的搜索接收机相比如此改善适合于具有在移动的和/或静止的发送/接收设备之间,特别是在第三代移动无线系统中的无线通信的通信系统的搜索接收机,即关于功能块和逻辑门电路的应用数目的节省是可能的,预先规定一个流水线体系结构,在该体系结构中象在流水作业线上一样完成各个计算步骤。
Patent CR-20110167-A (CR)
Title: Composición para mejorar la eficacia de herbicidas
Inventor: KRAPP MICHAEL
IPC: A01N25/02
Filed: 2011-03-24
Abstract: Una novedosa composición para mejorar la eficacia de herbicidas, el uso de esa composición para mejorar la eficacia de herbicidas, un agente herbicida que contiene esa composición y por lo menos un herbicida, y el uso de ese agente herbicida para combatir el crecimiento indeseado de plantas.
Patent CR-20120155-A (CR)
Title: Combinacion
Inventor: DUMBLE MELISSA
IPC: A01N43/90
Filed: 2012-03-27
Abstract: Una combinación novedosa que comprende el inhibidor de MEK de N-{3-[3-ciclopropil-5-(2-fluoro-4-yodo-fenil-amino)-6,8-dimetil-2,4,7-trioxo-3,4,6,7-tetrahidro-2H-pirido-[4,3-d]-pirimidin-1-il]-fenil}-acetamida, o una sal farmacéuticamente aceptable o un solvato de la misma, con un inhibidor de B-Raf, en particular N-{3-[5-(2-amino-4-pirimidinil)-2-(1,1-dimetil-etil)-1,3-tiazol-4-il]-2-fluoro-fenil}-2,6-difluoro-bencen-sulfonamida o una sal farmacéuticamente aceptable de la misma, composiciones farmacéuticas que la comprenden, y métodos para utilizar estas combinaciones y composiciones en el tratamiento de las condiciones en donde sea benéfica la inhibición de MEK y/o B-Raf, por ejemplo, cáncer.
Patent CR-20150196-A (CR)
Title: Moléculas de unión il-17a novedosas y usos médicos de las mismas
Inventor: SILACCI MELKKO MICHELA
IPC: C07K14/00
Filed: 2015-04-16
Abstract: La presente invención se relaciona a un polipéptido que inhibe la actividad de IL-17A glicosilada, en donde el polipéptido comprende o consiste de una secuencia de aminoácido seleccionada del grupo que consiste de: (a) GVTLFVALYDY(X1)(X2)(X3)(X4)(X5)(X6)DLSFHKGEKFQILSTHEYEDWWEARSLTTGETGYIPSNYVAPVDSIQ (SEC ID NO: 1), en donde las posiciones de aminoácidos (X1) a (X6) puede ser cualquier secuencia de aminoácido; y (b) una secuencia de aminoácido la cual es al menos 85% idéntica a la secuencia de aminoácido de (a), en donde la determinación de identidad excluye posiciones de aminoácido (X1) a (X6) y siempre que se conserve la secuencia de aminoácido STHEYE (SEC ID NO: 2) en posiciones de aminoácido 31 a 36 de la SEC ID NO: 1.
Patent CR-20170070-A (CR)
Title: Composición, método y preparación del ácido biliar sintético
Inventor: PRASAD ACHAMPETA RATHAN
IPC: C07J75/00
Filed: 2008-06-18
Abstract: Ácidos biliares y composiciones relacionadas y métodos de síntesis y uso. Más específicamente, el ácido desoxicólico y las composiciones relacionadas, dichas composiciones están libres de todas las porciones de orígen animal y libres de porciones pirogénicas.
Patent CR-20170250-A (CR)
Title: TETRAHIDRO-PIRIDO[3,4-b]INDOLES MODULADORES DE RECEPTORES DE ESTRÓGENOS Y USOS DE LOS MISMOS
Inventor: LABADIE SHARADA
IPC: C07D471/04
Filed: 2015-12-17
Abstract: Se describen compuestos tetrahidro-pirido[3,4-b]indol-1-ilo con actividad o función de modulación de los receptores de estrógenos modulación, que tienen la estructura de la fórmula I: y los estereoisómeros, tautómeros o sales farmacéuticamente aceptables de los mismos, con los sustituyentes y características estructurales aquí descritos. Se describen también composiciones farmacéuticas y medicamentos que incluyen los compuestos de la fórmula I, así como métodos de uso de tales moduladores de receptores de estrógenos, solos o en combinación con otros agentes terapéuticos, para tratar enfermedades o estados patológicos que están mediados o dependen de receptores de estrógenos.
Patent CR-20210041-A (CR)
Title: Amino acid compounds with unbranched linkers and methods of use
Inventor: CHA JACOB
IPC: C07C53/00
Filed: 2019-06-27
Abstract: <p>The invention relates to compounds of formula (A): or a salt thereof, wherein R<sup>1</sup>, R<sup>2</sup>, R<sup>5a</sup>, R<sup>5b</sup>, R<sup>6a</sup>, R<sup>6b</sup>, R<sup>7a</sup>, R<sup>7b</sup>, R<sup>8a</sup>, R<sup>8b</sup>, R<sup>9a</sup>, R<sup>9b</sup>, R<sup>10a</sup>, R<sup>10b</sup>, R<sup>11a</sup>, R<sup>11b</sup>, R<sup>21</sup>, n, and G are as described herein. Compounds of formula (I) and pharmaceutical compositions thereof are ανβ6 integrin inhibitors that are useful for treating fibrosis such, as idiopathic pulmonary fibrosis (IPF) and nonspecific interstitial pneumonia (NSIP).</p>
Patent CR-20210139-A (CR)
Title: Novel sulfonamideurea compounds
Inventor: CARRILLO ARREGUI JOKIN
IPC: C07D487/10
Filed: 2019-08-12
Abstract: The present invention relates to compounds of formula (I): wherein Q is selected from O or S; R<sup>1</sup> and R<sup>3</sup> are each independently hydrogen or an optionally substituted hydrocarbyl group, or R<sup>1</sup> and R<sup>3</sup> together with the nitrogen atom to which they are attached may form a 3- to 12-membered optionally substituted cyclic group; and R<sup>2</sup> is a cyclic group substituted at the oposition, wherein R<sup>2</sup> may optionally be further substituted. The present invention further relates to salts, solvates and prodrugs of such compounds, to pharmaceutical compositions comprising such compounds, and to the use of such compounds in the treatment and prevention of medical disorders and diseases, most especially by the inhibition of NLRP3.
Patent CR-20220001-A (CR)
Title: A pharmaceutical composition for diabetes mellitus
Inventor: VERMA RAJAN
IPC: A61K31/40
Filed: 2020-05-29
Abstract: The present invention relates to a pharmaceutical composition of Dipeptidyl peptidase-IV (DPP-IV) inhibitors for use in treatment of Diabetes Mellitus (DM). More particularly, the present invention relates to a modified or extended release dosage form comprising a composition of Vildagliptin or a pharmaceutically acceptable salt thereof with desired physical and chemical parameters for improved patient compliance.
Patent EC-SP067115-A (EC)
Title: Uso medicinal de lingados de receptor
Inventor: ULVEN TROND
IPC: A61K31/415
Filed: 2006-12-26
Abstract: Los compuestos de la fórmula (I) son útiles para el tratamiento de enfermedad senciblea la modulación de actividad de receptor CRTH2, tales como es asma, rinitis, síndrome alérgico de vías aéreas y ridobronquitis alérgica.
Patent EC-SP077397-A (EC)
Title: Preparación y uso de derivados de ácido bifenil-4-il-carbonilamino para el tratamiento de obesidad
Inventor: LOWE DEREK B
IPC: A61K31/454
Filed: 2007-04-13
Abstract: Esta invención se refiere a ciertos compuestos de ácido bifenil-4-il carbonilamino, composiciones y métodos para tratar o prevenir obesidad y enfermedades relacionadas.
Patent EC-SP088312-A (EC)
Title: Derivados plaguicidas de bifenilamidina
Inventor: DUNKEL RALF
IPC: C07C257/12
Filed: 2008-03-26
Abstract: La presente invención se refiere a derivados de bifenilamidina de fórmula (I) en los que los sustituyentes son tal como en la descripción, a procedimientos para su preparación, su uso como agentes activos fungicidas o insecticidas, particularmente en la forma de composiciones fungicidas o insecticidas, y a métodos para el control de hongos fitopatógenos o insectos dañinos, especialmente de plantas, que usan estos compuestos o composiciones:
Patent EC-SP088681-A (EC)
Title: Dispositivo de distribución de fármaco
Inventor: MODI PANKAJ
IPC: A61J1/10
Filed: 2008-08-15
Abstract: Se proporciona un nuevo dispositivo y el método para la distribución intradérmica de un agente activo. El dispositivo comprende un alojamiento que contiene una cámara de reservorio. Un reservorio flexible que contiene el agente activo está situado en la cámara. Tras la presión a un accionador el agente activo es distribuido a través de una aguja hueca a la piel.
Patent EC-SP992910-A (EC)
Title: Procedimiento para alquilar sulfonamidas impedidas estericamente
Inventor: HAWKINS JOEL MICHAEL
IPC: A61K31/18
Filed: 1999-04-09
Abstract: La presente invención se refiere a un procedimiento para alquilar sulfonamidas impedidas estéricamente, mediante una reacción de adicción de Michael, a propiolatos y a nuevos intermedios preparados en el citado.
Patent FI-20020756-A (FI)
Inventor: SUNDHOLM GOERAN
IPC: F02M25/028
Filed: 2002-04-19
Abstract: A water spraying system, especially for the humidification of the intake air of a piston engine to reduce nitrogen oxide emissions, said system comprising at least one nozzle ( 9, 10, 11, 12, 13 ) for spraying an aqueous liquid mist into the air intake duct ( 2 ) and means for conveying the liquid to be sprayed to the nozzle. The system comprises means for accomplishing the injection of a spray of aqueous liquid mist to at least one point in the air intake duct ( 2 ) depending on the load and/or speed of rotation and/or temperature of the engine.
Patent FR-1603186-A (FR)
Title: Production of a polyester resin from diepoxy resin and
IPC: C08L63/02
Filed: 1968-08-01
Granted: 1971-03-22
Abstract: A high-molecular linear polyester with hydroxy and epoxy functions is prepared by reacting a resinous diepoxy component and a dicarboxylic acid component. The dicarboxylic acid is mainly aromatic and is of the type which forms linear polyesters with ethylene glycol. The reaction between the diepoxy resin and the acid is carried out in the presence of a basic catalyst, and in an organic solvent, at a concentration of solid resin of not 50 weight.%. The acid number of the resin is  20 and the ratio of diepoxy component : dibasic acid is 3 : 2 - 6 : 5. The preparation is a simple 1 - or 2 - step process. The resins have improved heat stability. They give coatings with outstanding gloss, good resistance to solvents and good flow properties.
Patent FR-1604705-A (FR)
IPC: D06P1/52
Filed: 1968-06-10
Granted: 1972-01-24
Abstract: 1,247,589. Treating keratinic fibres. L'OREAL. 9 June, 1969 [10 June, 1968], No. 29158/ 69. Heading D1B. [Also in Divisions A5, A6, C3, C4 and C5] Keratinic fibres, e.g. wool, are treated with polymers containing a -CO-NRM group where R is hydrogen, lower (C 1-6 ) alkyl or lower hydroxyalkyl and M is a group containing a thiol residue. The fibres may then be dyed. Exemplified polymers are the reaction product of #-mercaptoethylamine and N,N-diethylpropylene diamine with a maleic anhydride-itaconic anhydride copolymer and the reaction product of #-mercaptoethylamine with a methyl acrylate-acrylic anhydride copolymer.
Patent GB-1010556-A (GB)
IPC: B65D5/36
Abstract: 1,010,556. Boxes. METAL BOX CO. Ltd. Aug. 2, 1963 [Oct. 30, 1962], No. 41054/62. Heading B8P. A six-sided box having one end thereof 5 wedge-shaped has a window in the wedgeshaped portion 7 in order that the contents of the box may be inspected. The side-panels 9 of the box are hinged to the bottom and a retaining panel 13, 14 which is hinged to the top is also provided on each side. Each retaining panel is foldable lengthwise along a creaseline 12 and the bottom part 14 is glued to the side, thus enabling the box in its open condition to be collapsed. In a second embodiment, the box is made from the blank shown in Fig. 4, the wedge-shaped portion being formed by folding triangular portions 23, 24 to overlie each other. The blank also includes a handle forming element 28, and is closed by selfinterlocking flaps 17a, the flaps 15a being connected to them as by adhesive.
Patent GB-1054555-A (GB)
IPC: C08G59/40
Abstract: 1,054,555. Carbamates. TILE COUNCIL OF AMERICA Inc. July 22,1963 [Sept. 25, 1962]. No. 28931/63. Heading C2C, [Also in Divisions C3 and E1] Carbaminates (the ammonium carbonatecarbamate forms) of polyamines are prepared by reacting the polyamine with carbon dioxide under anhydrous conditions. Polyamines specified are the alkylenepolyamines, N-alkyltrimethylenediamines and N-tallow bis (aminopropyl)-amine. Examples describe the preparation of the carbaminates of diethylenetriamine and of N-tallow bis (aminopropyl) amine.
Patent GB-1054692-A (GB)
IPC: C07C233/00
Abstract: 1,054,692. Hydroxyphenylacetamides. HASSLE, APOTEKARE PAUL NORDSTROMS FABRIKER A.B. May 20, 1964, No. 20890/64. Heading C2C. The invention comprises compounds of formula wherein R is a C 1-4  alkyl or alkoxy group, and their preparation by reaction with ammonia of formula wherein R<SP>1</SP> and R<SP>2</SP> are hydrogen atoms or protecting groups, or a reactive derivative formed therefrom, for example an acid halide, anhydride, mixed anhydride, ester or internal lactone, the protective groups, when present. being removed after the reaction. α - Ethyl - 2,3 - dihydroxyphenyl - acetic acid lactone is prepared by reaction of 2,3-dimethoxybenzyl cyanide with ethyl iodide and sodium ethoxide to form α - ethyl - 2,3 - dimethoxybenzyl cyanide, hydrolysing this to α-ethyl-2,3- dimethoxy - phenylacetic acid, and treating this with red phosphorus and iodine. α - Methoxy - 2,3 - dibenzyloxyphenyl - acetic acid is prepared by reaction of 2,3-dibenzyloxybenzaldehyde with bromoform, methanol and potassium hydroxide. The compounds of the invention block enzymatic body hydroxylation of aromatic aminoacids, and may be used in pharmaceutical compositions in combination with a carrier, for example in forms suitable for oral or parenteral administration.