baber/WOPTO huggingface dataset:
Patent ZA-957548-B (ZA)
Title: Benzoylguanidines substituted by heterocyclic n-oxide process for their preparation their use as a medicament or diagnostic agent medicament containing them and intermediate products for their preparation
Inventor: KLEEMANN HEINZ-WERNER
IPC: C07D213/89
Filed: 1995-09-08
Abstract: Benzoyl guanidine derivs. of formula (I) and their salts are new: one of R1-R3 = Het (linked by C or N), SR10, OR10, NR10R11 or CR10R11R12; and the other two of R1-R3 = H, halo, CN, X(CH2)p(CqF2q+1), SOuR22, CONR23R24, COR25, SO2NR26R27, 1-8C alkyl, 2-8C alkenyl, CmH2mR14, OR35 or NR35R36; R4, R5 = H, 1-4C alkyl, Fl, Cl, OR32, NR33R34 or CrF2r+1; R10 = CnH2n-Het; Het = 1-9C heteroaryl-N-oxide (opt. substd. by 1-3 F, Cl, CF3, OMe, OH, NH2, NHMe or NMe2); R11, R12 = as R10, H or 1-4C alkyl; R14 = 3-9C cycloalkyl or phenyl (opt. by 1-3 F, Cl, CF3, Me, OMe, NH2, NHMe or NMe2); R11, R12 = as R10, H or 1-4C alkyl; R14 = 3-8C cycloalkyl or phenyl (opt. substd. by 1-3 F, Cl, CF3, Me, OMe, NH2, NHMe or NMe2); X = a bond, O, S or NR28; R22 = 1-8C alkyl, 2-6C alkenyl, CmH2mR29 or CF3; R23, R25, R26 = H or as R22; R24, R27 = H or 1-4C alkyl; or R23 + R24, R26 + R27 = (CH2)4 or (CH2)5 (both opt. with a CH2 replaced by O, S, NH, NMe or N-benzyl); R28 = H or 1-3C alkyl; R29 = 3-7C cycloalkyl or phenyl (opt. mono- or tri-substd. by F, Cl, CF3, Me, OMe or NR30R31; R30, R31 = H or 1-4C alkyl; R35, R36 = H or 1-6C alkyl; or R35 + R36 = (CH2)y (opt with a CH2 replaced by O, S, NH, NMe or N-benzyl); R32-R34 = H or 1-3C alkyl; n, p, u = 0-2; m = 0-4; r = 1-4; q = 0-6; y = 4-7. Also claimed are cpds. of formula (IIIA); A = Cl, OR45, OH, OM or imidazol-1-yl; M = alkali or alkaline earth metal ion; and R45 = 1-8C alkyl or 1-4C alkylphenyl.
Patent ZA-966726-B (ZA)
Title: Extracts of shark cartilage having anti-collagenolytic, anti-inflammatory, anti-angiogenic and anti-tumoral activities; process of making, methods of using and compositions thereof.
Inventor: DUPONT ERIC
IPC: A61K33/14
Filed: 1996-08-07
Abstract: The present invention relates to cartilage extracts and to a method of producing the same. Shark cartilage extracts having anti-angiogenic, direct anti-tumor proliferating, anti-inflammatory and anti-collagenolytic activities have been obtained by an improved process. The process comprises the steps of obtaining a homogenate of cartilage in an aqueous solution, this homogenate being centrifuged and further fractionated to obtain a total extract having molecules of a molecular weight comprised between 0 to 500 KDa. The composition of the liquid extract has then been investigated by different ways. Further fractionation of this extract led to the preliminary characterization of some of its active components. Due to the multiplicity of biological activities of the total liquid extract, it can be used for treating numerous diseases or conditions such as those having components selected from the group consisting of tumor proliferation, angiogenesis, inflammation and collagenolysis. This extract has no offensive effect on normal body functions. Therefore, this shark cartilage extract has a very promising therapeutic value. The process for the obtention of cartilage extracts is simple and efficient. The unexpectedly valuable products obtained by this process are therefore an indication of a new and non-obvious process.
Patent ZA-977783-B (ZA)
Title: Method of inhibiting fibrosis with a somatostatin agonist
Inventor: CULLER MICHAEL D
IPC: A61K38/08
Filed: 1997-08-29
Abstract: The present invention relates to a method of inhibiting fibrosis in a patient. The method comprises administering a therapeutically effective amount of a somatostatin, a somatostatin agonist or a pharmaceutically acceptable salt thereof to said patient.
Patent ZA-987573-B (ZA)
Title: A cermet having a binder with improved plasticity a method for the manufacturing and use thereof
Inventor: HEINRICH HANS-WILM
IPC: C22C19/07
Filed: 1998-08-21
Abstract: Cermets having a Co-Ni-Fe-binder are described. The Co-Ni-Fe-binder is unique in that even when subjected to plastic deformation, the binder substantially maintains its face centered cubic crystal structure and avoids stress and/or strain induced phase transformations. Stated differently, the Co-Ni-Fe-binder exhibits reduced work hardening.
Patent AT-413341-B (AT)
IPC: B21F23/00
Filed: 2004-03-25
Granted: 2006-02-15
Abstract: A drivable device (5) is used to move the material (D) sideways out of the firing line (X-X) in a direction at right angles to the material length direction. The drivable device contains a guide channel acting as a firing channel (13) and at least one additional guide channel for receiving the material. The additional channel has at least one controllable braking device (18) for engaging with at least one length side of the material and a braking device for coaxial engagement with the material. A device is provided for ejecting individual pieces of braked material in the sideways direction. The drivable device is a round revolver with grooves evenly distributed around its periphery for acting as guide channels. Material is supplied continuously to the firing line.
Patent CH-631046-B (CH)
Inventor: IKENO HITOSHI
IPC: G04G3/00
Filed: 1976-08-25
Abstract: In order to manufacture a time-base signal generator, a quartz crystal having dimensions included within predetermined tolerances is formed, this quartz crystal is connected to an oscillating circuit and to a frequency divider, these circuits being constructed such that the division ratio is adjustable. According to the invention, the crystal is of the GT-cut type and the polishing is carried out in such a way that the ratio between the width (w) and the length (l) has precisely the value which corresponds to a zero frequency/temperature coefficient. The width and the length may have values which depart from the nominal values provided that they remain within the tolerances ( DELTA w) and ( DELTA l). Under these conditions, the generator of the time-base signal entirely forgoes any temperature-compensation element. <IMAGE>
Patent CH-617561-B (CH)
Inventor: MUERRLE KURT
IPC: G04B11/00
Filed: 1976-10-22
Abstract: A stepping gear is rotatably mounted with freedom of axial movement and formed with an axially facing shoulder and with teeth and tooth spaces defined by said teeth. A rotatably mounted pawl roller has first and second peripheral rings. A spring urges said pawl roller against said stepping gear. The first peripheral ring is adapted to enter one of said tooth spaces to oppose a rotation of said stepping gear. The second peripheral ring radially overlaps said shoulder to limit the freedom of axial movement of said stepping gear.
Patent CH-619580-B (CH)
Inventor: KOLCKMANN CLAUS
IPC: D04H11/00
Filed: 1976-11-10
Abstract: Water-permeable mat comprises textile fibres protruding upwards from a flexible wide-mesh base comprises solid plastic base portions connected to each other by webs so as to leave run-off channels beneath the webs. The solid portions pref. have a height of 3-15 mm and the webs have a height which is less by >=2 mm: the upper surfaces of solid portions and webs lie flush with each other. The solid portions are pref. made of PVC or polyurethane closed-cell foam, and consist of parallel beams with the webs extending transversely to them, or blocks separated from each other on all sides, with a star-like arrangement of webs. At least the webs are reinforced with a highly solidified fleece or with woven or knitted textile threads. The mat can be used on balconies and in swimming baths, and outdoors e.g. as an artificial lawn.
Patent GB-2365603-B (GB)
Title: Print job capture subsystem with pass-through support
Inventor: SIMPSON SHELL S
IPC: G06F3/12
Filed: 2001-03-09
Granted: 2004-11-10
Abstract: In response to print job communications from an application submitting a print job, a driver arrangement provides a driver type response appropriate for any pass-through data contained in the print job. Driver receives the data making up the print job and creates an intermediate representation of the print job comprising translated nonpass-through data and untranslated data comprising buffers of pass-through data. A data handler is associated with the pass-through data, and is responsible for directing the printing of the pass-through data at the designated printer.
Patent GB-2379854-B (GB)
Title: Dairy cow feed and the use thereof
Inventor: CHI FRANCIS
IPC: A23K1/18
Filed: 2001-09-19
Granted: 2006-04-19
Abstract: The use of cysteamine, a salt thereof or a composition containing cysteamine or a salt thereof for improving lactation of lactating animals.
Patent GB-2425274-B (GB)
Title: Paint roller support
Inventor: MARTIN BERJ A
IPC: B05C17/02
Filed: 2004-01-07
Granted: 2007-03-14
Abstract: Embodiments of a paint roller support for rotatably supporting a conventional paint roller cover are disclosed. In one embodiment, a paint roller support comprises a frame having an elongated shaft and at least one hub rotatably coupled to the shaft for supporting a conventional roller cover. A locking spring exerts a retaining force against an inner surface of the roller cover for frictionally retaining the roller cover on the hub while the paint roller support is used to deliver paint to a surface. Embodiments of a method for manufacturing a paint roller support also are disclosed.
Patent GB-2064561-B (GB)
Title: Sterically stabilised non-aqueous dispersions and their production via aqueous polymerization
IPC: C08F2/20
Filed: 1980-12-01
Granted: 1983-05-11
Abstract: A process is described for making sterically stabilised non-aqueous dispersions of polymer microparticles, in which (1) monomers including at least one crosslinking monomer are polymensed in an aqueous medium at a temperature at least 10 higher than the glass transition temperature of the polymer to be formed, in the presence of a block or graft copolymer stabilising agent containing in the molecule, as the component solvated by the aqueous medium, a polymer chain derived from a polyethylene glycol of molecular weight at least 1000, under conditions such that there is at no time present a separate monomer phase and (2) the microparticles thus obtained are transferred into a non-aqueous medium which is capable of dissolving the polyethylene glycol in question, when the latter is in the non-hydrated state, to the extent of at least 10% by weight at room temperature. The microparticles are of value for incorporation into coating compositions the main film-forming constituent of which is compatible with the polyethylene glycol-derived stabilising chains of the particles
Patent GB-2088397-B (GB)
Title: Cross-linked polyamides
IPC: B29C71/04
Filed: 1981-12-03
Granted: 1984-09-05
Abstract: Polyamides comprising substantial amounts of Nylon-11 and/or Nylon-12 units are cross-linked by irradiation in the presence of an unsaturated cross-linking agent, preferably triallyl isocyanurate. The cross-linked products are particularly useful in the form of heat-recoverable shaped articles, eg. heat-shrinkable tubing.
Patent GB-2115284-B (GB)
Title: Herbicidal mixtures
Inventor: ABILDT UWE
IPC: A01N43/70
Filed: 1983-02-21
Granted: 1985-06-05
Abstract: Flowable herbicidal compositions which contain an active component combination of at least one chlorotriazine and a chloroacetanilide form stable aqueous dispersions if the surfactant component of the composition consists of an anionic surfactant from the series of the mono- or diphosphoric acid esters of phenol polyglycol ethers and a mixture of two non-ionic surfactants from the series of the alkoxy, alkanoyloxy or phenol polyglycol ethers which differ by at least one glycol unit.
Patent GB-2192889-B (GB)
Title: Pyrimidine ribonucleoside 3'-phosphodiesters and their use in enzyme linked assays
Inventor: RABIN BRIAN ROBERT
IPC: C12Q1/6816
Filed: 1987-08-06
Granted: 1988-06-08
Abstract: A shall enzymically inactive peptide fragment of an enzyme (e.g. ribonuclease S-peptide) is used as the label and conjugated with the complementary fragment (S-protein) to form an enzyme which catalyses a primary reaction whose product is, or leads to, an essential coenzyme or prosthetic group for a second enzyme which catalyses a secondary reaction leading to a detectable result indicating the presence of analyte. Also disclosed are novel synthetic substrates for the primary reaction. Substrates for ribonuclease S conjugate enzyme are of the formula R-X where R is a pyrimidine 3 min -phosphate moiety and X is a leaving group linked to R through the 3 min -phosphate group and leads to said coenzyme or prosthetic group, e.g. via riboflavin, thiamine, pyridoxal, pyridoxine or pyridoxine phosphate.
Patent GB-2253546-B (GB)
Title: Radio communication apparatus with stored coding/decoding procedures
Inventor: NONAMI TAKAYUKI
IPC: H04W88/02
Filed: 1991-10-14
Granted: 1995-04-19
Abstract: A radio communication apparatus for transmitting and receiving a digital signal using a radio line which includes a memory means for storing a plurality of signal procedures in which each procedure has different ratio of the information code bits and error correction code bits. A signal processing circuit executes one of the procedures stored in the memory means according to line quality. Accordingly, the radio communication apparatus of the present invention selects the optimum procedure according to the line quality, and then reduces the consumed power.
Patent GB-2298250-B (GB)
Title: Plain bearing with overlay
Inventor: MCMEEKIN KENNETH MACLEOD
IPC: B23K20/04
Filed: 1996-02-21
Granted: 1999-02-17
Abstract: A method of making a multi-layer plain bearing (21) comprises roll-bonding a relatively soft aluminium-tin alloy overlay (12) to a harder aluminium-based bearing substrate (10) and then roll-bonding the composite to a steel backing (18). Following heat treatment conventional for reticulation of the aluminium-tin alloy, the surface is machined to give a precise overall bearing thickness of which the aluminium-tin overlay is in the range 0.01-0.10 mm, typical of an overlay but having greater fatigue strength and wear resistance than conventional electro-deposited materials. Aluminium interlayers may be included. The overlay, substrate and backing strips may be roll-bonded simultaneously (Figure 2) or the aluminium-tin alloy may be roll-bonded onto an intermediate bearing of copper-based alloy cast or sintered onto a steel or bronze backing (Figure 3).
Patent GB-2337521-B (GB)
Title: Improved film-forming compositions for protecting animal skin
Inventor: HEMLING THOMAS C
IPC: C09D175/08
Filed: 1998-06-08
Granted: 2001-11-07
Abstract: Improved film-forming skin protectant compositions are provided which are capable of forming a long-lasting elastic barrier film when applied to skin; the compositions have particular utility as barrier teat dips, for protecting cows against mastitis, especially during their susceptible non-lactating periods. The compositions include a film-forming component (preferably a mixture of polyether polyurethane and benzoin gum) dispersed in a compatible carrier and further having a minor amount of nitrocellulose incorporated therein in order to increase the time of adherence of the composition to skin, as compared with an otherwise identical composition without nitrocellulose. The compositions may also include a germicide (e.g., chlorhexidine diacetate), and a coloring dye. The most preferred compositions include polyether polyurethane, benzoin gum, a solvent system made up of tetrahydrafuran and a lower alcohol, and chlorhexidine diacetate.
Patent GB-2336365-B (GB)
Title: Woolgrease
Inventor: CAWTHORNE RICHARD NEIL
IPC: A61K8/00
Filed: 1998-01-14
Granted: 2000-09-06
Abstract: A process for recovering 18-methyl eicosanoic acid (18-MEA) and/or alpha hydroxy acids (AHAs) from woolwax acids or derivatives thereof comprises the steps of heating the woolwax acids or derivatives thereof to 100 to 230° C. to form estolides and polymeric species; distilling to obtain a distillate (D1) and a residue (R1); and recovering 18-MEA from the distillate and/or recovering AHAs from the residue.
Patent HU-214068-B (HU)
Inventor: ERICSON ROBERT B
IPC: H01R4/02
Filed: 1993-01-04
Abstract: (57) KIVONAT Vezető anyagú csőszerű elemet (10) tartalmazó vezetékcsatlakőzó (9)a csőszerű elembe (10) helyezett főrraszanyagtömböket ( 12) tartalmazés a csőszerű elemen ( 10) vezető (28) kicsúszását gátló elem ket,füleket (20) alakítűnk ki, amelyek a vezetők (28) lecsűpaszítőttvezető ereit (30) a főrraszanyagtömbök (12) melegítése ésmegőlvasztása sőrán elfőglalt helyzetükben tartják. A csőszerű elem(10 köré húzőtt, zsűgőrítható anyagból készült hüvely (14) csőszerűelemen (10) túlnyúló végei a vezetők (28) bevezetését megkönnyítőmódőn harang alakúak, míg a hüvely (14) középső része a csőszerű elere (10) van rázsűgőrítva a létrehőzőtt villamős kapcsőlatleszigetelése céljából. ŕ
Patent HU-219114-B (HU)
Title: Process for renovating pipes
Inventor: REIMELT ANDREAS
IPC: F16L58/10
Filed: 1995-08-29
Abstract: PCT No. PCT/DE95/01152 Sec. 371 Date May 28, 1997 Sec. 102(e) Date May 28, 1997 PCT Filed Aug. 29, 1995 PCT Pub. No. WO96/06710 PCT Pub. Date Mar. 7, 1996A process for renovating pipes wherein a particulate abrasive material is passed through the pipe to loosen the internal deposits, and after the abrasive material and internal deposits are removed from the pipe, a coating of a curable resinous or plastic material is applied to the interior of the pipe. An alternately produced pressure drop between the two ends of the pipe is employed to cause the particulate abrasive material to reciprocate within the interior of the pipe and thereby effectively loosen the internal deposits and avoid cloggages resulting from the loosened and detached internal deposits.
Patent IT-1186904-B (IT)
Title: Prefabricated self-supporting open-bottom ships cabin unit
Inventor: VIRTA HANNU
IPC: B63B/
Filed: 1985-07-03
Granted: 1987-12-16
Abstract: The arrangement provides a ship with self-supporting cabin units. A ships deck or similar flat surface is prepared to receive the units which each comprise side walls (2,3), a roof and an open bottom. The bottom is arranged to have temporarily fixed transport elements to enable moving the units along the deck surface. Each cabin unit may be pre-equipped with furniture etc. fixed to the walls so as to contribute to its rigidity (e.g. bathroom unit 11). Transport along deck may use wheels (20) or air cushion units releasably fixed (via 19) at the lower ends of the walls, pref. within the perimeter of the cabin.FL
Patent IT-1232509-B (IT)
Title: Floor sander (or similar surfaces)
Inventor: MARCO PREVIDI
IPC: B24B/
Filed: 1989-09-07
Granted: 1992-02-17
Abstract: Floor sander (or similar surfaces), with a frame; a sanding group (L); a motor (M) and a sanding load (L). In order to work also in angles and to change the load on the sanding group (l), the invention has two or more abrasives plates (30) working through planetary motion; the chassis has a front part (1A) on which the motor is mounted (M) and the sanding group (l) and a rear part (1B) on which the sanding (1) load (S) is mounted; the two parts (1A, 1B) of the chassis slide telescopically.
Patent IT-1215381-B (IT)
Inventor: GANDOLFI CARMELO A
IPC: C07D401/12
Filed: 1987-03-12
Granted: 1990-02-08
Abstract: Compounds of formula I <CHEM> wherein R1 is an acetyl, benzoyl, cyano, nitro, aminocarbonyl or alkoxycarbonyl group; - R2 is an optionally substituted aromatic group or a heterocyclic group;  - R3 is an alkoxycarbonyl group; - R4 is hydrogen, alkyl, cycloalkyl, optionally substituted phenyl, a heterocyclic group;  - R5 is hydrogen, alkyl, cycloalkyl, phenyl or benzyl;  - R6 is a <CHEM>  group wherein X is oxygen or sulphur, P is alkoxy, benzyloxy, alkylthio, benzylthio, a linear or cyclic amino group and Q is C1-C5-alkyl, aryl or alkylaryl. Compounds I are useful in human therapy.
Patent IT-1237442-B (IT)
Title: Shaft with dynamic fluid expansion parts to fix part B, made from materials such as paper, plastic, material and so on.
Inventor: STEFANO GATTRUGERI
IPC: F16C/
Filed: 1987-04-30
Granted: 1993-06-05
Abstract: This invention refers to dynamic fluid expansion parts, equipped or not with reserve valves that can be used to build expandable shafts to stop paper spools or generically made from material wrapped in rolls or for stopping circular knifes etc, to regulate the length of the flexible, material strips that need to be cut.
Patent IT-981039-B (IT)
IPC: F24H9/14
Filed: 1973-03-01
Granted: 1974-10-10
Abstract: A plurality of water conducting hollow members are assembled side by side and are interconnected by water ducts to enable water to circulate therethrough. Tie bars pass through the water ducts and have ends projecting through the end walls of the assembled hollow members, the tie bar ends being received in, and affixed to, sockets whereby the assembled members are anchored by the tie bars between the sockets to form a hot water radiator unit. Tie members clasp the side walls of the unit, the tie members being U-shaped elements having free ends with notches and the hollow members having ribs engaged by the notches.
Patent IT-1207465-B (IT)
Title: L-carnitine-methyl-glutarate
Inventor: SCHIENA MICHELE DI
IPC: C07C/
Filed: 1983-06-22
Granted: 1989-05-25
Abstract: The speed of mobile (10) in communication with a base (14) is determined by monitoring Rayleigh fading of the signal strength received from base in order to adjust a threshold level so that the threshold increases with decrease in mobile speed. If the median of the signal strength received at mobile (10) from another base (16) or (18) exceeds that received from base by more than the threshold level, a handoff request is issued. Rayleigh fading is monitored by detecting the rate at which the instantaneous signal strength received at mobile (10) from base (14) crosses the short-term median level of that signal, that rate being dependent on the maximum doppler frequency which increases with mobile speed. The median measuring time period may increase with decrease in the maximum doppler frequency.
Patent IT-1175859-B (IT)
Title: Hydroxy-ethoxy-methyl guanidine derivs. having pharmaceutical activity
Inventor: PURICELLI LAURA
IPC: A61K/
Filed: 1984-08-31
Granted: 1987-07-15
Abstract: Continuous prodn. of snacks from ceral flour comprises: (a) continuously feeding the flour into an enclosure having feed and delivery ends (b) transporting the flour inside the enclosure under friction from the feed to the delivery end with conditions preventing its swelling; (c) subjecting the flour inside the enclosure to a gradually increasing temp. to plasticize and rpessurize it; (d) extruding the plastizcized flour through a die so that it swells up and solidifies to produce a continuous body; and (e) comminuting the continuous body
Patent IT-1232935-B (IT)
Title: Moulding Polyolefin mixture
Inventor: BALLABIO ADRIANO
IPC: C08F/
Filed: 1987-11-06
Granted: 1992-03-10
Abstract: The present invention concerns a moulding mixture containing a propylene polymer, a high-density ethylene polymer and a very low-density ethylene copolymer. Said mixture enhances both physical and chemical properties of products obtained through injection moulding. In particular, said mixture improves colour resilience against sunrays and weathering.
Patent IT-1098385-B (IT)
Title: Dry pigment composition for aqueous make-up foundation - contains talc, pigment, and hydrophobic and hydrophilic silicas
IPC: A61K/
Filed: 1978-08-28
Granted: 1985-09-07
Abstract: A dry pigment composition for incorporation into aqueous makeup foundations consists essentially of 50-90% talc, 5-49% cosmetically acceptable pigment, 0.5-3% hydrophilic fumed silica and 0.5-5% hydrophobic fumed silica. Preferably the dry pigment composition contains 88% talc,10% titanium dioxide, 1% hydrophilic fumed silica and 1% hydrophobic fumed silica. The dry pigment composition can also contain 52% talc, 40% ferric oxide, 3% hydrophilic fumed silica and 5% hydrophobic fumed silica.