baber/WOPTO huggingface dataset:
Patent AR-018652-A1 (AR)
Title: Inhibidor de catepsina k del tipo pirrolidinona, composicion farmaceuticamente eficaz, usos de dichos compuestos para preparar medicamentos, yprocedimiento para producir dichos inhibidores
IPC: C07D207/24
Filed: 1999-06-10
Abstract: Inhibidor de catepsina K del tipo pirrolidinona que tiene la formula (I), en la que: X se selecciona del grupo formado por oxígeno, azufre, SO y SO2;Y se selecciona del grupo formado por H2 y oxígeno; donde, si Y es H2, entonces el enlace - - - - representa dos enlaces sencillos y donde si Y es O,entones el enlace - - - - representa un enlace doble; R1 se selecciona del grupo formado por hidrogeno, alquilo C1-6, alquenilo C2-6, alquinilo C2-6,cicloalquilC3-6-alquilo C0-6, Ar-alquilo C0-6, Het-alquilo C0-6, (CH2)0-6CO2R, y (CH2)0-6Ar; R11 se selecciona del grupo formado por hidrogeno, alquilo C1-6,alquenilo C2-6, alquinilo C2-6, cicloalquil C3-6-alquilo C0-6, Ar-alquilo C0-6 y Het-alquilo C0-6; R2 se selecciona del grupo formado por H, alquilo C1-6,alquenilo C2-6, alquinilo C2-6, cicloalquil C3-6-alquilo C0-6, Ar-alquilo C0-6 y Het-alquilo C0-6; R3 se selecciona del grupo formado por H, alquilo C1-6,alquenilo C2-6, alquinilo C2-6, cicloalquil C3-6-alquilo C0-6, Ar-alquilo C0-6 y Het-alquilo C0-6; alquilo C1-6 se selecciona del grupo formado pormetilo, etilo, n-propilo, isopropilo, n-butilo, isobutilo, t-butilo, pentilo, n-pentilo, isopentilo, neopentilo y hexilo sustituidos o no sustituidos, ylos isomeros alifáticos de los mismos;cicloalquilo C3-6 se selecciona del grupo formado por ciclopropano, ciclobutano, ciclopentano, y ciclohexanosustituidos y no sustituidos; alquenilo C2-6 es un grupo alquilo C2-6, en el que se ha sustituido un enlace sencillo carbono-carbono por un dobleenlace carbono-carbono; alquinilo C2-6 es un grupo alquilo C2-6, en el que se ha sustituido un enlace sencillo carbono-carbono por un triple enlacecarbono-carbono; Ar se selecciona del grupo formado por fenilo o naftilo; o fenilo o naftilo sustituido con uno o más de Ph-alquilo C0-6, Het-alquiloC0-6, alcoxi C1-6, Ph-alcoxi C0-6, Het-alcoxi C0-6, OH, (CH2)0-6CO2R, donde R es como se ha definido anteriormente, (CH2)1-6NRR, O(CH2)1-6NRR; ofenilo o naftilo sustituido con 1-3 restos seleccionadosentre alquilo C1-4, OR, N(R)2, SR, CF3, NO2, CN, CO2R, CON(R), F, Cl, Br e I, o sustituido
Patent AR-023331-A1 (AR)
Title: Un procedimiento para preparar un derivado de 2-aminotiazol-carboxamida y compuestos utiles como intermediarios en dicho procedimiento
Inventor: SANG-WHO LEE
IPC: C07D333/24
Filed: 1999-09-28
Abstract: La presente se relaciona con un procedimiento para preparar un derivado de 2-aminotiazol-carboxamida que está representado por la formula (1) en la cual R1representa alquilo C1-5, haloalquilo C1-5 o cicloalquilo C3-6, de cadena recta o ramificada, yR2 representa alquilo C1-3 o haloalquilo C1-3, caracterizadoporque un compuesto representado por la formula (2) en la cual R1 y R2 se definen tal como se describiera previamente y R3 representa fenilo, el cual puedeestar opcionalmente mono- a penta-s ustituido, en forma independiente, por cloro, metoxi, etoxi, fenoxi o nitro, se hace reaccionar con un compuestorepresentado por la formula (3) en la cual Y representa un grupo de salida, en un solvente, y en presencia de una base. Además sedivulga un compuesto utilcomo intermediario en el procedimiento arriba citado el cual se encuentra representado por la formula (2) en la cual R1, R2 y R3 se definen de acuerdo a loarriba expuesto y un compuesto util como intermediario en elprocedimiento arr iba citado el cual está representado por la formula (3) en la cual Y también sedefine de acuerdo con lo arriba expuesto.
Patent AR-025814-A1 (AR)
Title: Compuestos derivados de eritromicina, su procedimiento de preparacion, composiciones farmaceuticas y medicamentos
IPC: C07H17/08
Filed: 1999-11-10
Abstract: Compuestos derivados de eritromicina que comprenden los compuestos de formula (1) en la que X representa un átomo de hidrogeno o un átomo de halogeno y Zrepresenta un átomo de hidrogeno o el resto de un ácido así como sus sales de adicion con ácidos.Los compuestos de formula (1) presentan propiedadesantibioticas, son particularmente activos sobre las cepas resistentes a eritromicina como, por ejemplo, Streptococcus pyogenes y Streptococcus pneumoniae y S.aureus. Además se describe el procedimiento para su preparacion y composiciones farmacéuticas y medicamentos que los comprenden.
Patent WO-2007118260-A1 (WO)
Inventor: FARNSWORTH BRUCE
IPC: A61F2/00
Filed: 2007-04-06
Abstract: L'invention concerne un réseau implantable destiné à une reconstruction chirurgicale dans la zone du plancher pelvien, comprenant une partie de réseau antérieure (2) destinée à être placée entre la vessie (4) et le vagin (5), une partie de réseau postérieure (3) destinée à être placée entre le vagin (5) et le rectum (10), une paire de bras supports de transobturateur distaux (6) partant de la partie de réseau antérieure (2), une paire de bras supports de transobturateur proximaux (7) partant de la partie de réseau antérieure (2) et une paire de bras supports dorsaux inférieurs (15) partant de la partie de réseau postérieure (3). Le réseau présente en outre une partie intermédiaire (13) située entre la partie de réseau antérieure (2) et la partie de réseau postérieure (3), la paire de bras supports dorsaux inférieurs (15) s'étendant dans la zone de la partie de réseau postérieure (3) adjacente à la partie intermédiaire (13) et une paire de bras supports dorsaux supérieurs (14) s'étendant en outre dans la zone de la partie de réseau antérieure (2) adjacente à la partie intermédiaire (13).
Patent WO-2008003108-A1 (WO)
Title: Verfahren zur herstellung eines extrudierten formkörpers
Inventor: JAECKEL MANFRED
IPC: B22F5/00
Filed: 2007-07-03
Abstract: Die Erfindung beschreibt ein Verfahren zur Herstellung eines Formkörpers mit den Verfahrensschritten Herstellung einer Formmasse, Plastifizieren der Formmasse in einem Extruder und Austragen über eine Schlitzdüse, Zuführen des Grünlings in ein Glättwalzwerk, Glätten des Grünlings durch ein oder mehrere Glättvorgänge, chemisches und/oder thermisches Entbindern und Sintern. Das kontinuierlich arbeitende Verfahren ermöglich eine kostengünstige Herstellung von bevorzugt Flachprodukten mit hoher Oberflächenqualität.
Patent WO-2009100469-A1 (WO)
Inventor: EBNER BERNHARD
IPC: E21C25/16
Filed: 2009-01-16
Abstract: In a drift heading work machine (1, 24), comprising at least one cutting unit having a rotatably supported tool carrier (10, 39) with disk tools (11, 12, 40, 41), said carrier being pivotally connected to the machine frame, the heading work machine (1, 24) has an undercarriage, particularly a track-laying gear (2), the tool carrier (10, 39) is rotatably supported on a boom arm (6, 26) pivotal in the vertical direction, and the rotation axis (9) of the tool carrier (10, 39) runs transversely to the longitudinal axis of the boom arm (6, 26).
Patent WO-2014040093-A1 (WO)
Title: Procédé de fabrication d'aciers bainitiques pour rail, partie de voie et dispositif permettant de mettre en œuvre le procédé
Inventor: POINTNER PETER
IPC: C21D1/63
Filed: 2013-06-27
Abstract: L'invention concerne une partie de voie, en particulier un rail pour des véhicules ferroviaires en acier faiblement allié. L'acier dans le champignon de rail de la partie de voie présente une fraction de ferrite de 5-15 % en volume et une structure bainitique multiphasique constituée de fractions supérieure et inférieure de bainite.
Patent WO-2019232559-A1 (WO)
Title: Trägerkörper für ein schleifwerkzeug und verfahren zur herstellung eines trägerkörpers
Inventor: MAYRHOFER KARL
IPC: B24D5/02
Filed: 2019-04-30
Abstract: Trägerkörper (1) für ein Schleifwerkzeug (2), welcher eine, vorzugsweise umfangsseitige, Trägerfläche (3) für einen Schleifmittel (4), insbesondere Superschleifmittel, aufweisenden Schleifbelag (5) umfasst, wobei der Trägerkörper (1) im Wesentlichen aus einem schleifmittelfreien Verbundwerkstoff (6) aus einer Vielzahl übereinander angeordneter Schichten (7) eines Naturfaser-Werkstoffs, welche durch Kunststoff (8), vorzugsweise Phenolharz, miteinander verbunden sind, besteht, vorzugsweise wobei es sich beim Naturfaser-Werkstoff um ein Baumwollgewebe oder Papier handelt, wobei der Trägerkörper (1) einen ersten, vorzugsweise zylindrischen oder hohlzylindrischen, Körper (29, 30, 31, 32, 33) und wenigstens einen weiteren, vorzugsweise zylindrischen oder hohlzylindrischen, Körper (29, 30, 31, 32, 33) umfasst, wobei die Körper (29, 30, 31, 32, 33) miteinander verbunden, vorzugsweise verklebt, sind.
Patent WO-2022204739-A1 (WO)
Inventor: WITTMANN MICHAEL PETER
IPC: B29C45/76
Filed: 2022-03-12
Abstract: The invention relates to a plastic-processing system and to a method for avoiding parallelism of load peaks (21) of a plastic-processing machine, more particularly an injection molding machine (4), and at least one production means (2), for example a temperature-control device (13a), hot runner system, cooling device (13b), flow controller (13), granular-material dryer (12), tool dryer, metering device (11), robot (5), automation system, etc., wherein the injection molding machine (4) is connected, by means of an electrical cable (27) or data cable (27), to the at least one production means (2) directly or indirectly via an external working cell controller (26), and wherein the injection molding machine (4) or the external working cell controller (26) sends one or more control signals (22) or internal operating states (22) with increased load demand to the one or more production means (2) so that the one or more production means (2) carries out a load shift, load reduction or load shedding at the times (24) of the increased load demand of the injection molding machine (4).
Patent WO-2023133606-A1 (WO)
Title: Rohrpresskupplung
Inventor: HOPPE MARVIN
IPC: F16L33/02
Filed: 2023-01-12
Abstract: Die Erfindung betrifft eine Rohrpresskupplung (1) umfassend: - eine Stützhülse (5) mit einer außenliegenden Aufnahmefläche (11) zur Aufnahme eines Rohres (2); - eine Außenhülse (6) mit einer Außenhülseninnenmantelfläche (23), welche zur Anlage an einer Rohraußenmantelfläche (14) des Rohres (2) ausgebildet ist, und mit einem an einer Außenhülsenaußenmantelfläche (27) ausgebildeten Spannklammersitz (22); - eine Spannklammer (21) zum radialen nach innen verformen der Außenhülse (6) und somit zum Andrücken der Rohrinnenmantelfläche (13) des Rohres (2) an die Stützhülse (5), wobei die Spannklammer (21) die Außenhülse (6) schellenförmig umgibt und am Spannklammersitz (22) aufgenommen ist, wobei die Spannklammer (21) eine Keilaufnahme (32) bildet; - einen Fixierkeil (38), welcher im gefügten Zustand in der Keilaufnahme (32) der Außenhülse (6) aufgenommen ist und zum umfänglichen verkürzen und somit zum Andrücken der Spannklammer (21) an die Außenhülsenaußenmantelfläche (27) dient.
Patent AU-2002242923-A1 (AU)
Title: Plasma surface treatment method and device for carrying out said method
Inventor: SAMSONOV MICKHAIL
IPC: H01L21/3065
Filed: 2002-03-26
Abstract: The invention relates to a plasma surface treatment method for the surface of an object or particles to be treated consisting in creating a plasma and applying said plasma against the surface to be treated.  The inventive method is characterised in that the surface to be treated is excited or the plasma is made to vibrate acoustically in order to create a relative wave motion between the plasma and the surface to be treated.
Patent AU-2002311765-A1 (AU)
Title: Methods of making and uses of compositions that modulate intronic region-encoded protein function
Inventor: RALPH DAVID
IPC: C12Q1/68
Filed: 2002-02-26
Abstract: This invention relates to compositions and methods for modulating cellular activity of non-human organisms, and in particular fungi, and methods of identifying and using antifungal agents with improved specificity. More particularly, the technology described herein relates to the identification and use of compounds that target intron-encoded proteins, such as maturases.
Patent AU-2002312737-A1 (AU)
Title: Projection screen with several spherical section segments
Inventor: HOFFMANN PETER
IPC: G03B21/56
Filed: 2002-05-03
Abstract: Projection wall systems having projection walls are used, for example, for cinema screens or planetariums. They are provided in the form of cupola-shaped, dome-like superstructures, which have an exterior supporting structure and, on the inside, have a primarily concave surface that is used as a projection wall for special cinema projectors. The inventive device is a projection wall system comprising a projection wall with a simplified design, whereby segment constructional units (13) are fastened to a supporting structure (199) by means of retaining elements (222) provided with adjusting devices.
Patent AU-2002320779-A1 (AU)
Title: Disc brake pad
Inventor: GOTTI ANTONIO
IPC: F16D65/847
Filed: 2002-07-15
Abstract: A disc brake pad is suitable for cooperating with a fixed-caliper disc brake comprising a caliper body provided with a seat suitable for housing the pad. The pad seat is defined by a side wall with which the abutment surface of the plate of the pad is brought into abutment during braking. The pad also has, on the surface for supporting the friction material, zones which are free of friction material and which advantageously obstruct the flow of heat from the friction material to the side walls of the pad seat.
Patent AU-2002322035-A1 (AU)
Title: Peptide deformylase inhibitors
Inventor: CHRISTENSEN IV SIEGFRIED B
IPC: A61K31/19
Filed: 2002-06-04
Abstract: Novel PDF inhibitors and novel methods for their use are provided.
Patent AU-2002325298-A1 (AU)
Title: Delivery system having a rapid pusher assembly for self-expanding stent, and stent exchange configuration
Inventor: DORN JURGEN
IPC: A61F2/95
Filed: 2002-07-04
Abstract: A pusher assembly for a delivery system for a self-expanding stent (6) which is delivered by proximal withdrawal of a sheath (4) radially surrounding the stent has a stent pusher element (8) which defines a lumen for a guidewire (2), a pusher strand (16) that extends to the proximal end of the delivery system and bears an end-wise compressive stress during release of the stent. A transfer shaft (12) links the distal end of the pusher strand (16) to the pusher element (8) and lies side-by-side with the guidewire (2). In a rapid exchange version, an adapter (20) provides two lumens side-by-side, one (22) carrying the pusher strand (16) and the other (14) defining a proximal guidewire part. To the adapter is mounted the proximal end of the stent sheath (4). The system allows modular (14) construction, a tapered tip (4A) on the sheath, and an uncluttered internal configuration which facilitates passage of pulses (F) of liquids from the proximal to the distal end of the system.
Patent AU-2002344668-A1 (AU)
Title: Shielded structure for radiation treatment equipment and method of assembly
Inventor: OQUIST CHERI ANN
IPC: E04H1/12
Filed: 2002-05-14
Abstract: A modularized approach for rapidly and cost effectively assembling a structure suitable for housing radiation emitting equipment is disclosed. The modules include reinforced walls to contain radiation shielding fill material. The modules are transported empty and then filled on site with the fill material to form a radiation shielding barrier around radiation emitting equipment.
Patent AU-2002350779-A1 (AU)
Title: Analyzer and analysing method and a fluid cartridge
Inventor: TOLONEN PERTTI
IPC: G01N35/00
Filed: 2002-12-13
Abstract: The invention relates to a method for analysing a sample, in which method the sample is brought to an analyzer, it is subjected to measures relating to determining the concentration of analyte to be examined, and the sample is measured. The analyzer (1) is equipped with a sample container (5), a fluid cartridge (3) and at least one analysis cartridge (4), and at least part of the sample to be analysed is transferred from the sample container (5) to a sample chamber (22) of the fluid cartridge (3). At least part of the sample is transferred from the sample chamber (22) of the fluid cartridge (3) to the analysis cartridge (4) that comprises at least some of the reagents used in the analysis, and the sample contained in the analysis cartridge (4) is measured. The invention also relates for example to an analyzer used in the method according to the invention as well as to a fluid cartridge used for example in the method or analyzer according to the invention.
Patent AU-2002358162-A1 (AU)
Title: Cosmetic compositions comprising a cyclodipeptide compound
Inventor: FRANKLIN KEVIN RONALD
IPC: A61K8/31
Filed: 2002-12-19
Abstract: Cosmetic formulations containing a cosmetic active and a continuous phase comprising a water-immiscible liquid carrier, such as, amongst other materials, silicone oils, branched aliphatic alcohols or liquid aromatic/aliphatic esters that is structured by a cyclodipeptide derivative having the general formula in which R<SUB>A </SUB>represents a carbocyclic or heterocyclic group containing not more than 2 rings, other than unsubstituted cyclohexyl.
Patent AU-2002364492-A1 (AU)
Title: Process for the production of alginate having a high mannuronic acid-content
Inventor: HJELLAND FINN
IPC: A23L29/256
Filed: 2002-11-21
Abstract: The present invention concerns a process for the production of alginate having a mannuronic acid-content of at least 80 mole %, wherein said alginate is produced by: a) adding algae or seaweed to water under stirring, in a ratio of 1:3 to 1:20 respectively, at a pH above about 2.3, while maintaining a temperature above 20° C. for at least 30 minutes, and b) separating said alginate from the solid material of the suspension in a) by a standard separation method such as filtration, and optionallyc) recovering said alginate from the solution.
Patent AU-2003204505-A1 (AU)
Title: Amino acid free stable aluminum/zirconium antiperspirant solution
Inventor: PAREKH JAWAHAR CHUNILAL
IPC: A61K8/34
Filed: 2003-05-30
Abstract: An amino acid free stable aluminum zirconium polyhydric alcohol aqueous solution having a high anhydrous antiperspirant solid concentration and a high percentage of low molecular weight aluminum species, i.e., containing 60% or more of band IV peak area based on high pressure liquid chromatography, is prepared by adding a zirconium salt to an aqueous polyhydric alcohol solution of a basic aluminum chloride.
Patent AU-2003206388-A1 (AU)
Title: Prosthesis implantable in enteral vessels
Inventor: STINSON JONATHAN S
IPC: A61F2/90
Filed: 2003-01-03
Abstract: A body insertable tubular stent includes discrete tubular segments in an alternating sequence of segments having high axial stiffness and segments having low axial stiffness. The lower axial stiffness segments are intended for placement along more severely curved regions of the body vessel, to provide a greater degree of stent conformity to the vessel. The more axially flexible segments can be provided by winding a metallic or polymeric strand at a higher pitch along such segments, thus to form a higher braid angle in a braided stent. In such cases the more axially flexible segments also exert a higher radial force when the stent is radially compressed. Alternatively, the stent can consist of multiple interbraided strands, with each strand incorporating a higher number of filaments (at least two) along axially stiff segments, and incorporating a lower number of filaments (at least one) along axially flexible segments. In another alternative version, the device is formed of one or more resilient strands, each strand including a biostable filament and a bioabsorbable filament, so that after implantation the radial force and axial stiffness gradually decrease in vivo.
Patent AU-2003227083-A1 (AU)
Title: Quick-fixing device
Inventor: TETIK ADOLF
IPC: H02B1/052
Filed: 2003-04-11
Abstract: A device for the detachable quick-fixing of housings (2) of electric serial fittings (1), such as circuit breakers or fuse-switches and the like, on a profiled assembly rail (5),comprising a housing (2) with a recess (4) for the assembly rail (5), a coupling element (2) being maintained on the housing and being connected via journals (12), said coupling element being provided with an engaging end (15) with a hook (9) which engages from the rear with the assembly rail (5) in the position of fixing and an actuating section (14) which can be engaged in the fixing position of the element (8) on the housing (2). The coupling element (8) is embodied as a two-armed lever which is mounted on at least one side wall (1) of the housing (2) of the serial fitting (1) and the actuating section (14) overlaps with the housing (2). In order to actuate the coupling element in a simple manner, the actuating section (14) overlaps with a front side of the housing (2) which faces away from the recess (4) for the assembly rail (5) and which can be actuated by the front side.
Patent AU-2003232733-A1 (AU)
Title: Device for ejecting a liquid from a wiping element
Inventor: RUST HENDRIK
IPC: A47L13/58
Filed: 2003-05-07
Abstract: Device (20) for extracting liquid from a wiper body (14) held on a wiper head of a surface cleaning device under formation of a wiper surface (15) comprises a container (21) containing a wiper body holder (45) receiving the wiper body and a drive device rotationally driving the wiper body holder about an axis of rotation (55). The wiper body holder has a recess (49) in which the wiper body in inserted with the surface normal (16) of the wiper surface at an angle to the axis of rotation.  Preferred Features: The recess receives the wiper body with the surface normal of the wiper surface perpendicular to the axis of rotation. The recess has a guide with two parallel U-shaped guide elements (46, 47) in which the wiper body is inserted. The drive device is a drive motor consisting of a rechargeable energy supply unit.
Patent AU-2003237757-A1 (AU)
Title: Binding device
Inventor: REXHAJ FAHREDIN
IPC: B65B27/12
Filed: 2003-07-01
Abstract: Binding apparatus for binding wire around pulp bales are disclosed including a wire magazine, a wire feeder for feeding and stretching the wire, a guide for guiding the wire from the feeder around the pulp bale, a wire cutter and twister for cutting the wire and twisting together the wire ends and a take-up unit for taking up a loop in the wire obtained upon stretching of the wire around the pulp bale, the take-up unit including a take-up space having a pair of walls separated by a distance adapted to accept the wire but insufficient to accept a double strand of the wire, and the short sides of the take-up space separated by a distance adapted to accept a loop of the wire without being folded and the take-up space at one of the short sides including a wire guide space wider than the wire and formed by grooves in at least one of the walls.
Patent AU-2003245202-A1 (AU)
Title: An apparatus and a method for cleaving thin rods
Inventor: BOTTCHER UWE
IPC: G02B6/25
Filed: 2003-06-10
Abstract: A method for cleaving thin rods of glass or quartz with a rod cleaving blade (27) and body (28) carrying the blade, is provided. The body (28) is of material varying in length through application of electric and/or magnetic fields. Driving force (31, 33) achieves relatively steady movement of the blade (27) towards a desired cleaving point and relatively steady small-amplitude vibratory component of movement towards and away from the cleaving point superimposed to the relatively steady movement, by influencing the body (28) electrically and/or magnetically. The blade is driven to vibrate with a frequency below 1 kHz during cleaving operation.
Patent AU-2003249344-A1 (AU)
Title: Process for preparing 5-(1,3-oxazol-2-yl) benzoic acid derivatives
Inventor: REEDER MICHAEL R
IPC: C07D263/32
Filed: 2003-06-20
Abstract: Disclosed are compounds of formula III and a process to prepare a compound of formula III wherein R<SUB>1</SUB>, R<SUB>2</SUB>, R<SUB>3 </SUB>and R<SUB>6 </SUB>are defined herein, using a zinc chloride/optionally substituted oxazole adduct and an compound of formula I. Further disclosed are methods of using compounds of formula III to prepare compounds useful in the treatment of Alzheimer's disease and related conditions.