baber/WOPTO huggingface dataset:
Patent YU-80202-A (YU)
Title: Novel phenyl-propargylether derivatives
Inventor: LAMBERTH CLEMENS
IPC: C07D213/02
Filed: 2001-05-15
Abstract: The invention relates to phenyl-propargylether derivatives of general formula (I) including the optical isomers thereof and mixtures of such isomers, wherein R1 is hydrogen, alkyl, cycloalkyl or optionally substituted aryl, R2 and R3 are each independently hydrogen or alkyl, R4 is alkyl, alkenyl or alkynyl, R5 R6, R7, and R8 are each independently hydrogen or alkyl, R9 is hydrogen, optionally substituted alkyl, optionally substituted alkenyl or optionally substituted alkynyl, R10 is optionally substituted aryl or optionally substituted heteroaryl, and Z is halogen, optionally substituted aryloxy, optionally substituted alkoxy, optionally substituted alkenyloxy, optionally substituted alkynyloxy, optionally substituted arylthio, optionally substituted alkylthio, optionally substituted alkenylthio, optionally substituted alkynylthio, optionally substituted alkylsulfinyl, optionally substituted alkenylsulfinyl, optionally substituted alkynylsulfinyl, optionally substituted alkylsulfonyl, optionally substituted alkenylsulfonyl or optionally substituted alkynylsulfonyl. These compounds possess useful plant protecting properties and may advantageously be employed in agricultural practice for controlling or preventing the infestation of plants by phytopathogenic microorganisms, especially fungi.
Patent AP-484-A (AP)
Title: Novel imidazole compounds, processes for the preparation thereof and their use in therapy.
Inventor: ADAMS JERRY LEROY
IPC: C07D213/53
Filed: 1994-07-13
Granted: 1996-04-23
Abstract: Novel 1, 4, 6-substituted imidazole compounds, processes for the preparation thereof,
Patent AP-767-A (AP)
Title: Quinoxalinediones
Inventor: CARR CHRISTOPHER LEE
IPC: A61P25/28
Filed: 1997-03-06
Granted: 1999-09-29
Abstract: The invention provides compounds of formula (I) and the pharmaceutically acceptable salts thereof, wherein R is a 5-membered ring heteroaryl group containing 3 or 4 nitrogen heteroatoms which is linked to the quinoxalinedione ring by a ring carbon or nitrogen atom, or is a 6-membered ring heteroaryl group containing from 1 to 3 nitrogen heteroatomt which is linked to the quinoxalinedione ring by a ring carbon atom, either of said groups being optionally benzo-fused and optionally substituted, including in the benzo-fused portion, by 1 or 2 substituents each independently selected from Ci-CU alkyl, Cj-C4 alkenyl, Cj-C? cycloalkyl, halo, hydroxy, Ci-CU alkoxy, Ci-Oi cycloalkyloxy, -COOH, Ci-C* alkoxycarbonyl, -CONR3R4. -NR'R4, -S(O)p(Ci-Ct alkyl), -SOiNR3R4, aryl, aryloxy, aryl(Ci-Cx)aIkoxy and net, said Ci-C< alkyl being optionally substituted by Cs-C? cycloalkyl, halo, hydroxy, Ci-O alkoxy, halo(Ci-C«)alkoxy, Cj-C? cycloalkyloxy, Cs-C7 cycloalkyl(Ci-O)alkoxy, -COOH, Ci-C< alkoxycarbonyl, -CONR3R4, -NR3R4, -S(O)p(Ci-C4 alkyl), -SOaCaryl), -SO2NR3R4,morpholino, aryl, aryloxy, aryl(C]-C4)alkoxy or bet, and said C2-C4 alkenyl being optionally substituted by aryl; R1 and R selected fromH Fluoro chloro bromo C1-C4 Arkyl and halo (C1-C4)alkyl R3 and R4 are cither each independently SO2NR3R4,morpholino, aryl, aryloxy, aryl SO2NR3R4,morpholino, aryl, aryloxy, aryl(C]-C4)alkoxy or bet, and said C2-C4 alkenyl being optionally substituted by aryl; R1 and R selected fromH Fluoro chloro bromo C1-C4 Arkyl and halo (C1-C4)alkyl R3 and R4 are either each independently selected from H AND c1-c4 alkyl or when, taken together, are C3-C7 alkylene; p is 0, 1 or 2; together with the preparation of compositions containing the uses of and intermediates used in the synthesis of, such compounds. The compounds are useful as NMDA receptor antagonists for treating acute neurodegenerative and chronic neurological disorders.
Patent AU-1023492-A (AU)
Title: Process for the preparation of n-mono- or n,n-disubstituted ureas
Inventor: ROSSLER MARKUS
IPC: C07C273/18
Filed: 1992-01-14
Abstract: Process for the preparation of N-mono- or N,N-disubstituted ureas by reacting ammonium isocyanate with a primary or secondary amine in a diluent.
Patent AU-1051001-A (AU)
Title: Synthetic human genes and polypeptides and their use in the treatment of autoimmune diseases
Inventor: BEN-NUN AVRAHAM
IPC: C12N15/12
Filed: 2000-10-26
Abstract: Synthetic human target autoantigen genes comprising sequences coding for at least two immunogenic epitopic clusters (hereinafter IEC) of autoantigen(s) related to a specific autoimmune disease, wherein said at least two IECs may be derived from a sole autoantigen or from at least two different autoantigens related to said autoimmune disease, and polypeptides encoded thereby, can be used for the treatment and the diagnosis of autoimmune diseases such as multiple sclerosis (MS), insulin-dependent diabetes mellitus (IDDM), rheumatoid arthritis (RA), myasthenia gravis (MG) and uveitis.
Patent AU-1114692-A (AU)
Title: Vector
Inventor: BARTH PETER THOMAS
IPC: C12N15/70
Filed: 1992-02-24
Abstract: The invention relates to vectors which include an inducible selection gene and a sequence which codes for a heterologous polypeptide. In a particular example the selection gene comprises the tetA and tetR genes. The vector may also include a sequence which is capable of conferring stability on the vector, such as the cer sequence, a transcription terminator, such as gene 32 from bacteriophage T4, a ribosome binding site, and a multi-cloning site. Hosts transformed with the vector, processes for preparing these hots, and processes for preparing polypeptides using these hosts.
Patent AU-1184288-A (AU)
Title: Improved hair treating resins
Inventor: CHUANG JUI-CHANG
IPC: A61K8/31
Filed: 1987-12-21
Abstract: An improved hair spray resin comprising microspheres of vinyl acetate/mono-n-C4-C5 alkyl maleate/ an isobornyl acrylate terpolymer in a molar ratio of about 1:0.35-1:0.05-0.25 and a one-step suspension polymerization process for the preparation of said resin in yields above 85%.
Patent AU-1189897-A (AU)
Title: A decanter centrifuge
Inventor: MADSEN BENT
IPC: B04B11/02
Filed: 1996-12-18
Abstract: PCT No. PCT/DK96/00544 Sec. 371 Date Jun. 9, 1998 Sec. 102(e) Date Jun. 9, 1998 PCT Filed Dec. 18, 1996 PCT Pub. No. WO97/22411 PCT Pub. Date Jun. 26, 1997The decanter centrifuge has a bowl with a screw conveyor having a body (4) and a screw (7). Material to be separated into a light phase is supplied through inlet ports (6) in the body, and the heavy phase is discharged through discharge ports in the bowl at one end of the conveyor. Between the inlet ports and the discharge ports for the heavy phase, the body of the screw conveyor carries a baffle (8c), generally shaped as a radial rib which forms a helical surface turning in the same direction as the screw (7). Owing to its shape the baffle actively contributes to the transport of the heavy phase, and with retention of the same gap between the baffle and the inner surface of the bowl, the gap area can be increased by increasing the axial length of the baffle.
Patent AU-1271392-A (AU)
Title: Synthesis of intermediates in the preparation of acat inhibitors
Inventor: KELLY SARAH E
IPC: C07D217/02
Filed: 1991-11-27
Abstract: PCT No. PCT/US91/08758 Sec. 371 Date Sep. 13, 1993 Sec. 102(e) Date Sep. 13, 1993 PCT Filed Nov. 27, 1991 PCT Pub. No. WO92/13843 PCT Pub. Date Aug. 20, 1992.This invention relates to novel processes for synthesizing intermediates in the preparation of N-aryl and N-heteroarylamide inhibitors of the enzyme acyl coenzyme A: cholesterol acyltransferase (ACAT), and to novel intermediates used in such processes.
Patent AU-1300983-A (AU)
Title: Ethylene copolymers for hot melt systems
Inventor: ALIANI GIORGIO
IPC: C08F210/02
Filed: 1983-03-30
Abstract: Ethylene-vinyl acetate copolymers having a melt index of 700 to 10000 and containing from 11 to 40% vinyl acetate are useful in hot melt systems and particularly in formulating low viscosity hot melt adhesives, preferably in binary compositions with natural or synthetic resin tackifiers. The adhesives show long open times with short setting times, and excellent adhesive properties. The EVAs are prepared by a high pressure polymerization, preferably by using chain transfer agent such as isobutylene to achieve high melt indices.
Patent AU-1353295-A (AU)
Title: Peptides derived from a retrovirus of the HIV group, and their use
Inventor: BRUST STEFAN DR
IPC: C07K16/10
Filed: 1995-02-21
Abstract: An immunologically active peptide comprising approximately 15 to 50 (pref. 20-30) consecutive amino acids (AA), selected from the sequence (I) is new:VWGIRQLRAR LQALETLIQN QQRLNLWGX KGKLIXYTSV KWNTSWSGR (I). In (I), X = C or S. Also claimed are: (a) the peptide produced either recombinantly or synthetically; (b) an isolated DNA fragment coding for a peptide as above; and (c) a test kit for the detection of viral antibodies causing immune deficiencies, pref. a Western Blot or an ELISA.
Patent AU-1390001-A (AU)
Title: Male-sterile brassica plants and methods for producing same
Inventor: WESTON BRIGITTE
IPC: A01H5/10
Filed: 2000-10-26
Abstract: This invention pertains to methods for determining the presence or absence in Brassica plant material of elite event MS-B2, which is a specific transformation event of a construct comprising a male-sterility gene, at a specific location in the Brassica genome, using PCR and primers specific to the construct, and kits for use in the methods.
Patent AU-1403400-A (AU)
Title: Polypropylene graft copolymers with improved scratch and mar resistance
Inventor: SMITH JEANINE A
IPC: C08F255/02
Filed: 1999-12-08
Abstract: A polymer composition with improved scratch and mar resistance contains (1) a graft copolymer comprising a backbone of a propylene polymer material having graft polymerized thereto at least one vinyl monomer capable of being polymerized by free radicals, and (2) an additive selected from the group consisting of (a) about 0.5% to about 10% of at least one low molecular weight ethylene polymer or a functionalized derivative thereof, and (b) a combination of (i) about 0.5% to about 10% of at least one of the low molecular weight ethylene polymers in (a) and (ii) about 0.5% to about 10% of inorganic microspheres, based on the total weight of the composition. Optionally the composition can also contain a compatibilizing agent such as an unsaturated carboxylic acid-functionalized propylene polymer material. The composition can optionally contain about 2% to about 30% of one or more rubber components, about 15% to about 50% of a broad molecular weight distribution propylene polymer material, or a combination of the two.
Patent AU-1466601-A (AU)
Title: Improved process for the preparation of trifluoropropanal and its oxime
Inventor: PUY MICHAEL VAN DER
IPC: C07C45/51
Filed: 2000-11-03
Abstract: A compound having the formula 3,3,3-trifluoropropanal oxime, and an improved process for forming the same. The oxime is prepared by reacting hydroxylamine with 3,3,3-trifluoropropanal under conditions sufficient to produce 3,3,3-trifluoropropanal oxime.
Patent AU-1683583-A (AU)
Title: Self locking collasible/expandable structure and clip there for
Inventor: ZIEGLER THEODORE R
IPC: E04B1/344
Filed: 1983-07-14
Abstract: This disclosure relates to a clip (80) for securing together adjacent collapsible, expandable, self-locking, self-supporting structures which include a plurality of pairs of crossed rod elements (27,28) pivotally joined in scissored fashion (29) to each other and to hubs (62, 66) having openings (0) therein, the structures having at least one hub (62, 66) of each section adjacent each other, and the clip (80) having at least two stems (83, 83') with each stem (83) being interlockingly received in an associated opening (0) of the adjacent hubs to thereby secure the structures to each other in any one of a plurality of different configurations.
Patent AU-1885301-A (AU)
Title: Method and apparatus for manufacturing three-dimensional knitwear and hosiery items and products obtained thereby
Inventor: SCIACCA FRANCO
IPC: A41B11/14
Filed: 2000-11-14
Abstract: The invention relates to a method and apparatus for manufacturing three-dimensional tubular knitwear items, preferably provided with shoulder straps, neck portion and/or various openings for feet, legs or arms, manufactured without the usual expensive fabric scraps deriving from the cutting/sewing operations. By means of a suitable selection of needles, or thanks to a particular yarn which melts completely during finishing, according to the jacquard design or to the work cycle of the textile machine, the present invention enables the separation and/or the automatic programmed resumption of knitted courses according to specific zones or areas, thus obtaining at least one opening (5,5A) or shoulder strap, provided with a singe or double welt. The hosiery items are automatically closed on their ends, corresponding to the foot heel or toe, and provided with at least one opening with single or double welt.
Patent AU-2109097-A (AU)
Title: Isoquinolines useful as analgesics
Inventor: DIMAIO JOHN
IPC: A61K38/00
Filed: 1997-02-25
Abstract: PCT No. PCT/SE97/00315 Sec. 371 Date Oct. 6, 1997 Sec. 102(e) Date Oct. 6, 1997 PCT Filed Feb. 25, 1997 PCT Pub. No. WO97/31940 PCT Pub. Date Sep. 4, 1997The present invention is directed to compounds that act as analgesics and that have the structure of formula (I): wherein; Z is wherein, n is 1 or 2, and R0 is C6-12 aryl or C7-8 aralkyl; or R1 is selected from the group consisting of hydrogen; -NH-C1-6 alkyl; C1-6 alkyl; C6-12 aryl; C7-18 aralkyl; arginyl; and R30NHC(=NH)-, wherein R30 is hydrogen, C6-12 aryl, C7-18 aralkyl, or C1-6 alkyl; R2 is hydrogen; C1-6 alkyl; or OH; R3 is C6-12 aryl; C7-18 aralkyl; -CH2-C6H2R8R9;or -CH2-OHC6HR8R9, wherein each of R8 and R9 is independently, or hydrogen; R4 C6-12 aryl; C7-18 aralkyl; C1-12 alkyl; or a substituted or unsubstituted cyclohexyl; R5 is C1-6 alkyl; hydrogen; OH; halogen; SH; NO2; NH2; -NH-C1-6 alkyl; NH2C (=NH-; NH2C (=NH)-NH-; COOR31, wherein, R31 is hydrogen, or C1-6 alkyl; X is CH2NHC(O)-; CH2NHC(O)O; -C(O)NH-; or CH2NH-; and L is a C1-12 alkylene chain which can be substituted with at least one substituent selected from the group consisting of; a C3-C12 cycloalkyl containing at least one heteroatom; C1-6 alkyl; OR31; -NHC(O)R33; -OC(O)R34 -NHR35 wherein; and NR6R7; with the proviso that when R5 is hydrogen, Z is and X is -C(O)NH-, or -CH2NH-, then L is a C1-12 alkyl chain substituted with at least one substituent selected from the group consisting of; a C3-C12 cycloalkyl containing at least one heteroatom; C1-6 alkyl; OR31; SR32; -NHC(O)R33; -OC(O)R34, -NHR35; and NR6R7.
Patent AU-2277500-A (AU)
Title: Method and device for transmitting short messages in telecommunications networks
Inventor: KEHR KLAUS
IPC: H04N1/00
Filed: 1999-12-15
Abstract: The invention relates to a method and a device for transmitting short messages in communications networks. The inventive method advantageously enables the individually structurable content of short messages (SMS) to be transmitted to subscriber lines with analogue terminals. The content of the SMS is converted into signals in such a way that transmission to the analogue terminal is possible. A transmission in the opposite direction is also possible. Two components are required to carry out the method: a gateway for converting the content of the SMS into a suitable format for transmission to the analogue terminal and a terminal (TIX: <u>T</u>extual <u>I</u>nformation E<u>X</u>change) for encoding or decoding the SMS content at the user end.
Patent AU-2407788-A (AU)
Title: Method and apparatus for receiving printed products from a revolvingly driven bucket wheel of a printing machine
Inventor: HANSCH EGON
IPC: B65H29/66
Filed: 1988-10-20
Abstract: An outfeed conveyor is arranged beneath a rotary bucket wheel driven to rotate in a predetermined rotational direction. A belt conveyor is arranged downstream of, and a product entrainment arrangement is arranged upstream of, the outfeed conveyor. An endless revolving belt is guided about belt rolls of the outfeed conveyor and upon which come to bear the printed products in inbricated formation. Entrainment elements of the product entrainment arrangement completely stuff the printed products into the pockets of the bucket wheel. Upon ejection of the printed products out of the bucket wheel they are fixedly clamped at their trailing edges between a support element and extensions or cantilever arms of the entrainment elements until the entrainment elements have passed the support element and thus an intersection location between the entrainment elements and the support element. The resiliently arranged extensions of the entrainment elements are pivoted by the support element in a predetermined direction, such as clockwise, so that the printed products are cyclically released. There is thus formed an inbricated formation of the printed products within which all prnited products are aligned and there can be maintained a substantially constant mutual spacing between the individual printed products.
Patent AU-2449395-A (AU)
Title: Inflatable lighting balloon
Inventor: CHABERT PIERRE GABRIEL
IPC: A63H27/10
Filed: 1995-04-27
Abstract: The balloon (1) has a flexible outer surface (1) which is connected an electric cable with an outer sheath (27). A sealed connection through the balloon wall is made by an outer plate (4) with inner ring and sealed connections (13). Nut connections (28) on the outer wall allow connection to an inner section. The cable connects a power source on the ground to a light in the centre of the balloon. An actuation device inside the balloon consists of a spring (7) which is tensioned by a flexible connector and connected to the loop (17) of a two-sided pin (19). Switches (25) are positioned between the power source and the light. A wire (5) links part of the surface and the actuator which is positioned at another location at the surface periphery. The pin has a sliding holder (24) and an inner spring (15). The pin base (21) is clear of the switch (26) when the balloon is inflated, but pushes the switch closed when the balloon is deflated, switching off the electricity. <IMAGE>
Patent AU-2599002-A (AU)
Title: Fusion cells and cytokine compositions for treatment of disease
Inventor: OHNO TSUNEYA
IPC: A61P35/02
Filed: 2001-10-22
Abstract: The present invention relates to methods and compositions for treating and preventing cancer and infectious disease by administering a therapeutically effective dose of fusion cells formed by fusion of autologous dendritic cells and autologous non-dendritic cells, in combination with a cytokine or other molecule which stimulates or induces a cytotoxic T cell response and/or a humoral immune response.
Patent AU-2632395-A (AU)
Title: A system for monitoring telephone networks and/or data communication networks, especially mobile telephone networks
Inventor: DAHL ERIK
IPC: H04M3/22
Filed: 1995-05-31
Abstract: PCT No. PCT/NO95/00086 Sec. 371 Date Apr. 8, 1997 Sec. 102(e) Date Apr. 8, 1997 PCT Filed May 31, 1995 PCT Pub. No. WO95/33352 PCT Pub. Date Dec. 7, 1995A system and method monitors telephone networks and/or data communication networks, especially cellular mobile telephone networks (CeN), and provides good evidence of performance and quality of the services to be delivered by the network. At the same time, the system and method is easy to handle and includes components that require only small spaces and that are effective in use. According to the invention, a method and system (CeNA) includes one or more fixed and/or mobile units (FTU, MTU), herein designated as field units or test units, that enable quality observations and communication with a network operator or operation center (CU).
Patent AU-2698592-A (AU)
Title: Cdw52 - specific antibody for treatment of t-cell mediated inflammation of the joints
IPC: A61K38/00
Filed: 1992-10-14
Abstract: The invention relates to the use of an antibody recognising the CDw52 antigen for the treatment of T-cell mediated inflammation of the joints, in particular for the treatment of rheumatoid arthritis. Preferably the antibody is the humanised antibody CAMPATH-1H which may be used together with another immunosuppressive antibody or an immunosuppressive agent such as a steroid.
Patent AU-2721402-A (AU)
Title: Anilinopyrimidine derivatives as jnk pathway inhibitors and compositions and methods related thereto
Inventor: KOIS ADAM
IPC: A61P31/04
Filed: 2001-12-05
Abstract: Compounds having activity as inhibitors of the JNK pathway are disclosed. The compounds of this invention are anilinopyrimidine derivatives having the following structure: wherein R<SUB>1 </SUB>through R<SUB>6 </SUB>are as defined herein. Such compounds have utility in the treatment of a wide range of conditions that are responsive to inhibition of the JNK pathway. Thus, methods of treating such conditions are also disclosed, as are pharmaceutical compositions containing one or more compounds of the above compounds.
Patent AU-2725000-A (AU)
Title: Omega-carboxy aryl substituted diphenyl ureas as p38 kinase inhibitors
Inventor: RIEDL BERND DR
IPC: A61K31/4453
Filed: 2000-01-13
Abstract: This invention relates to the use of a group of aryl ureas in treating p38 mediated diseases, and pharmaceutical compositions for use in such therapy.
Patent AU-2773795-A (AU)
Title: Dental composition and method
Inventor: HUANG CHIN-TEH
IPC: A61K6/083
Filed: 1995-06-13
Abstract: Use of a composition comprising a component which is a liquid reaction product obtained by reacting one mole of a 4,4'-oxydiphtalic anhydride (5,5'-oxybis-1,3-isobenzo furandione) with two moles of one or more compounds of the general formula ROH, wherein R is a polymerizable unsaturated moiety having from 2 to 13 carbon atoms in the presence of an acid, base or suitable catalyst for the preparation of a dental restorative composition for binding to hard tooth, metal and ceramic.
Patent AU-3021695-A (AU)
Title: Process for the preparation of the (-)-N-methyl-N-{4-(4- phenyl-4-acetylaminopiperidin-1-yl)-2-(3,4-dichlorophenyl) butyl}benzamide and its pharmaceutically acceptable salts
Inventor: DESCAMPS MARCEL
IPC: A61K31/445
Filed: 1995-08-23
Abstract: A process is described for the preparation of (+)-2-(3,4-dichlorophenyl)-4-hydroxybutylamine of formula (I) and for the preparation of the (-)-N-methyl-N-Ä4-(4-phenyl-4-acetylamino-piperidin-1-yl)-2-(3,4-dichl orophenyl)butylÜ benzamide and of its pharmaceutically acceptable salts using the compound of formula (I) as synthesis intermediate.
Patent AU-3093484-A (AU)
Title: Connector block slotted plate with polytropic air gap
Inventor: GERKE DIETER
IPC: H01R4/24
Filed: 1984-07-23
Abstract: The subject matter of the invention is a connector block (1) with solderless, non-screwed and stripping-free terminal elements (2, 3) having a polytropic air gap, for terminating dropwire cables (6) and cable wires (7). The terminal elements (2, 3), which comprise a terminal contact (2b, 3b) and a center contact (2a, 3a), have a semi-circular extension (2a') on the underside (2') of the center contact (2a, 3a), the spacing of said semi-circular extension relative to an earth bar (4) mounted in the housing lower half (12) being variable by tilting the earth bar (4) about 180 DEG ; said earth bar (4) is adapted to be mounted at either of two different levels. Thereby it is possible to select a high-voltage spark-gap function.
Patent AU-3111095-A (AU)
Title: Alginate fibres, method of preparation and use
Inventor: MAHONEY PETER M J
IPC: A61K9/70
Filed: 1995-07-14
Abstract: PCT No. PCT/EP95/02771 Sec. 371 Date May 30, 1997 Sec. 102(e) Date May 30, 1997 PCT Filed Jul. 14, 1995 PCT Pub. No. WO96/02283 PCT Pub. Date Feb. 1, 1996The present invention is concerned with alginate fibres, and in particular the use thereof as a wound dressing and a method of preparing the same. There is provided alginate fibres for use in the absorption of at least 10% by weight based on the weight of the alginate fibres of proteinaceous material from a wound environment into the structure of the fibres.