baber/WOPTO huggingface dataset:
Patent FI-885839-A0 (FI)
Inventor: COOK DAVID CHARLES
IPC: A61K31/16
Filed: 1988-12-16
Abstract: Therapeutically useful thioformamide derivatives of the formula: <CHEM> wherein R represents alkyl, Ar represents optionally substituted phenyl group, Y represents ethylene, methylene or a valency bond, and X represents carbonyl, hydroxymethylene, >C=NOR<1>, >C=NN(R<1>)2 or >C=NN(R<1>)CON(R<1>)2 in which R<1> represents hydrogen or optionally substituted alkyl, benzyl, phenethyl, 1-naphthylmethyl, 2-naphthylmethyl or pyrid-3-ylmethyl or two R<1> substituents on the same nitrogen atom may together form optionally substituted alkylene, and salts thereof, processes for their preparation and compositions containing them are described.
Patent FI-891962-A0 (FI)
Inventor: LARSSON KENNETH LARS
IPC: E21B17/00
Filed: 1989-04-25
Abstract: The present invention relates to a drill string element adapted to be coupled to other similar drill string elements by thread connections (19) thus forming a drill string for top hammer drilling. Each drill string element includes at least one rod (15;15 min ;15 sec ) for transferring impact energy to a drill bit (11) provided at the lower end of the drill string (10) and a tube assembly (21;21 min ;21 sec ) for transferring rotation to the drill bit (11), said tube assembly surrounding the rod. When handling drill string elements of the above-mentioned type it is extremely important that this handling can take place in a safe way without any risk for accidents during operation working site. Previously known drill string elements of the type in question have the disadvantage that the rod can fall out of the tube assembly in one direction. Also the accessibility to the interior of the drill string element in connection with repairs/service must be considered and the drill string elements must stay intact during operation, especially when they are unscrewed from each other. The invention is characterized by that the tube assembly (21;21 min ;21 sec ) in the area of the two ends of the rod (15;15 min ;15 sec ) is provided with an internal diameter reducing (27;27 min ,27 sec ;27'''), and that the rod (15;15 min ;15 sec ) is provided with cooperating radial projections (28;28 min ) or shoulder means (28 sec ). Also the tube assembly (21;21 min ;21 sec ) includes at least two tubular members (18;18 min ;18 sec ) that are coupled to each other by a thread connection that is harder to unscrew than the thread connection (19) for coupling together the drill string elements.
Patent FI-913801-A0 (FI)
Inventor: EFFLAND RICHARD CHARLES
IPC: C07D209/42
Filed: 1991-08-09
Abstract: This invention relates to compounds of the formula <CHEM>  where   R1   is hydrogen, loweralkyl, arylloweralkyl, loweralkenyl or loweralkynyl; R2   is hydrogen, loweralkyl, loweralkenyl, formyl or cyano; R3   is hydrogen or loweralkyl; R4   is loweralkyl, arylloweralkyl, cycloalkyl, aryl, heteroaryl, heteroarylloweralkyl, <CHEM>  or NR3R4 taken together constitute <CHEM>   R5   is hydrogen, loweralkyl or aryl; R6   is hydrogen, loweralkyl, aryl, arylloweralkyl, formyl, loweralkanoyl or arylloweralkanoyl, X and Y   are independently hydrogen, nitro, amino, halogen, loweralkyl, loweralkoxy or hydroxy; or the pharmaceutically acceptable acid addition salts thereof, and where applicable, the geometric and optical isomers and racemic mixtures thereof.   The compounds of this invention are useful for the treatment of various memory dysfunctions characterized by a decreased cholinergic function, such as Alzheimer's disease.
Patent FI-935726-A0 (FI)
Inventor: O'NEILL BRIAN THOMAS
IPC: A61K31/4025
Filed: 1993-12-20
Abstract: PCT No. PCT/US92/04697 Sec. 371 Date Dec. 14, 1993 Sec. 102(e) Date Dec. 14, 1993 PCT Filed Jun. 11, 1992 PCT Pub. No. WO93/00330 PCT Pub. Date Jan. 7, 1993The present invention relates to novel azanorbornane derivatives having the formula    <IMAGE>, and to novel intermediates used in their synthesis. The compounds having formula I are useful in the treatment of inflammatory and central nervous system disorders, as well as other disorders.
Patent FI-945081-A0 (FI)
Inventor: JOHNSON DONALD A
IPC: A61K31/545
Filed: 1994-10-28
Abstract: PCT No. PCT/US93/03856 Sec. 371 Date Oct. 27, 1994 Sec. 102(e) Date Oct. 27, 1994 PCT Filed Apr. 30, 1993 PCT Pub. No. WO93/21923 PCT Pub. Date Nov. 11, 1993A dry hydrated cephalosporin, e.g. ceftibuten having about 7 to 14% by weight of water, powder formulation, pharmaceutical compositions in the form of an oral suspension dosage form and a method of making the dry powder formulations are disclosed.
Patent FI-952045-A0 (FI)
Inventor: HOWIE JOHN KEENEY
IPC: A23L1/308
Filed: 1995-04-28
Abstract: Nondigestible fat compositions useful as a replacement for triglyceride fats or oils in foods are disclosed. The compositions have relatively flat Solid Fat Content (SFC) profile slopes between typical room and body temperatures. The nondigestible fat compositions comprise a liquid nondigestible oil and nondigestible solid polyglycerol ester particles dispersed in the oil in an amount sufficient to control passive oil loss. The ester groups of the solid polyglycerol ester particles comprise long chain (C16-C24) fatty acid radicals, with at least about 40% of the long chain fatty acid radicals being saturated and having at least 18 carbon atoms. The Iodine Value of these polyglycerol ester is less about 1. Edible fat-containing products containing these nondigestible fat compositions can be less waxy tasting due to the lower level of solids required for passive oil loss control.
Patent FI-960887-A0 (FI)
Inventor: MESENS JEAN LOUIS
IPC: A61P25/04
Filed: 1996-02-26
Abstract: PCT No. PCT/EP94/02764 Sec. 371 Date Jan. 26, 1996 Sec. 102(e) Date Jan. 26, 1996 PCT Filed Aug. 19, 1994 PCT Pub. No. WO95/05815 PCT Pub. Date Mar. 2, 1995The present invention relates to the iontophoretic delivery to a patient, more in particular to a migraine patient, of a compound of formula (I) as shown hereinunder. The invention also relates to a device for the iontophoretic delivery of a compound of formula (I), as well as to a composition containing a compound of formula (I), which can be applied in a device for iontophoretic delivery. Said compounds are benzopyranalkylaminoalkyl substituted guanidines having the formula    <IMAGE>  (I)  the pharmaceutically acceptable acid addition salts thereof, and the stereochemically isomeric forms thereof, wherein R1 is hydrogen or C1-6alkyl; R2 is hydrogen, C1-6alkyl, C3-6alkenyl or C3-6alkynyl; R3 is hydrogen or C1-6alkyl; or R2 and R3 taken together form a bivalent radical of formula -(CH2)m- wherein m is 4 or 5; or R1 and R2 taken together form a bivalent radical of formula -CH=CH- or of formula -(CH2)n-, wherein n is 2, 3 or 4; or R3 may represent a bond when R1 and R2 taken together form a bivalent radical of formula -CH=CH-CH=; R4 and R5 each independently are hydrogen or C1-6alkyl; Alk1 is a bivalent C1-3alkanediyl radical; Alk2 is a bivalent C2-15alkanediyl radical; and R6 and R7 each independently are hydrogen, halo, C1-6alkyl, C3-6alkenyl, C3-6alkynyl, hydroxy, C1-6alkyloxy or cyano.
Patent FI-960895-A0 (FI)
Inventor: LEHTONEN ARTO H
IPC: H04W4/00
Filed: 1996-02-26
Abstract: The present invention relates to a terminal (1) for a communication network having means (2 - 5) for wireless communication, and menus including menu items for performing certain commands. The terminal comprises a memory (14) for storing data, and a menu application. The menu application is capable of creating menu items in the terminal memory (14) according to predetermined commands. The terminal has means (3 - 5) for wirelessly receiving commands relating to said menu application via the communication network, and the menu application has been arranged to create menu items in the terminal in response to receiving said commands. <IMAGE>
Patent FI-963997-A0 (FI)
Inventor: KENNEALLY COREY JAMES
IPC: C07C69/587
Filed: 1996-10-04
Abstract: A process for preparing polyol fatty acid polyesters having levels of triglyceride below 0.5% is described. Methyl esters having a level of monoglycerides below 500 ppm, a nondetectable level of di- and triglyceride and a glycerine level of less than about 200 ppm are prepared and then used in a two-stage, solvent-free transesterification reaction to prepare the polyol fatty acid polyesters.
Patent IL-58064-A0 (IL)
Title: Fluorinated polyene compounds their preparation and pharmaceutical compositions containing them
IPC: C07C45/00
Filed: 1979-08-17
Abstract: {PG,1 9-Substituted, 4- or 6-fluorine substituted retinoic acid derivatives useful as antitumor agents and in the treatment of acne as well as a method for their manufacture are disclosed. Substituents at the 9-position include substituted phenyl, thienyl and furyl groups.
Patent IL-58971-A0 (IL)
Title: 2-phenylimino-imidazolidine derivatives their preparation and pharmaceutical compositions containing them
IPC: A61P9/00
Filed: 1979-12-17
Abstract: 1. Claims for the contracting states : BE, CH, DE, FR, GB, IT, LU, NL, SE 3,4-Disubstituted 2-phenylimino-imidazolidines of general formula (I)  see diagramm : EP0012822,P5,F1  wherein Z represents a radical selected from the group comprising 3-fluoro-4-methylphenyl, 4-fluoro-3-methylphenyl, 4-fluoro-3-nitrophenyl, 4-fluoro-3-chlorophenyl and 4-fluoro-3-aminophenyl, and the acid addition salts thereof. 1. Claims for the contracting state : AT Process for the preparation of 3,4-disubstituted 2-phenylimino-imidazolidines of general formula (I)  see diagramm : EP0012822,P6,F1  wherein Z represents a radical selected from the group comprising 3-fluoro-4-methylphenyl, 4-fluoro-3-methylphenyl, 4-fluoro-3-nitrophenyl, 4-fluoro-3-chlorophenyl and 4-fluoro-3-aminophenyl, and the acid additions salts thereof, characterised in that a) a compound of the formula (II)  see diagramm : EP0012822,P6,F3  wherein Z is as hereinbefore defined and X and Y, which may be the same or different, represent a chlorine atom, an alkylthio group with 1 to 4 carbon atoms or an amino or ammonium group, is reacted with ethylenediamine or an acid addition salt thereof ; or b) the aliphatic acyl group is hydrolytically split off from a 1-acyl-2-phenylamino-imidazoline of general formula (III)  see diagramm : EP0012822,P6,F5  wherein Z is as hereinbefore defined and R represents an aliphatic acyl group ; or c) in order to prepare 2-(4-fluoro-3-aminophenylimino)-imidazolidine, 2-(4-fluoro-3-nitrophenylimino)-imidazoline is hydrogenated and, if desired, the compound thus obtained is converted into a physiologically acceptable acid addition salt.
Patent IL-69682-A0 (IL)
Title: Benzamido-derivatives
IPC: C07C65/05
Filed: 1983-09-07
Abstract: Novel therapeutically active compounds of the formulawherein R is a straight or branched alkyl group with 6-18 carbon atoms, R<sup>1</sup> is hydrogen, chlorine, bromine or an alkyl group with 1-3 carbon atoms and R<sup>2</sup> is chlorine, bromine or an alkyl group with 1-3 carbon atoms; or a physiologically acceptable salt or an optical isomer thereof, methods and intermediates for their preparation, pharmaceutical preparations containing them and methods for their therapeutical use.
Patent IL-75328-A0 (IL)
Title: Production of alpha-chloroacetoacetic acid monomethylamide
IPC: C07B61/00
Filed: 1985-05-28
Abstract: 1. A process for producing alpha-chloroacetoacetic acid monomethylamide by reaction of chlorine with acetoacetic acid monomethylamide in an aqueous medium, at temperatures of -20 to +10 degrees C, in the presence of urea and alkali metal salts, neutralisation of the reaction mixture, separation of solid alpha-chloroacetoacetic acid monomethylamide, and feeding back of the mother liquor into the chlorination reaction, wherein the mother liquor obtained each time after the separation of alpha-chloroacetoacetic acid monomethylamide is extracted, before being recycled, with 2-10% by weight, relative to the total amount of the mother liquor, of an inert solvent immiscible with water.
Patent IL-82793-A0 (IL)
Title: Decorative plastics laminate and method for its manufacture
IPC: D21H11/02
Filed: 1987-06-08
Abstract: The decorative plastics laminate comprises a plurality of superposed translucent sheets constituted by 60 to 100% of alpha-cellulose and 0 to 40% of rayon fibres, impregnated with a thermosetting amino resin and bonded together by pressure and heat. Together with the characteristics of resistance to abrasion, water, impacts and chemical reagents, the laminate has a particular decorative effect obtained by virtue of the transparency of the cellulose sheets used.
Patent IL-92740-A0 (IL)
Title: Recombinant dna expression vectors and dna compounds that encode isopenicillin n epimerase(racemase)activity
IPC: C12N15/80
Filed: 1989-12-15
Abstract: The present invention provides DNA compounds that encode isopenicillin N epimerase (racemase) activity. The compounds can be used to construct recombinant DNA expression vectors for a wide variety of host cells, including E. coli, Penicillium, Streptomyces, Aspergillus, and Cephalosporium.
Patent AU-PS212502-A0 (AU)
Title: Method and device for local treatment of substrates with fluids
IPC: C23C4/123
Filed: 2002-05-07
Abstract: This invention relates to a process for fabricating a working electrode for use in a Dye Solar Cell (DSC). The method including the steps of: providing a transparent substrate with a Transparent Electronic Conductor (TEC) layer; coating an area of the TEC layer with a layer of semiconducting material; applying a layer of dye over both the Transparent Electronic Conductor (TEC) layer an the layer of semiconducting material; locally treating the substrate with a fluid, the fluid being selected to dissolve the dye; said process comprising creating and directing at least one jet of fluid towards local areas of the substrate; the local areas being coated by dye, but not coated by the semiconducting material and applying a vacuum suction force to the said local areas.
Patent FI-20001374-A0 (FI)
Inventor: WIIO ANTTI
IPC: G01C21/34
Filed: 2000-06-09
Abstract: The invention relates to a method for implementing a route guidance service in a telecommunications system. In order for it to be possible to utilize both the data transmission capacity of the telecommunications system and the memory and processing capacity of the user workstation efficiently in the execution of a route animation based on a three-dimensional model, the description of the 3D model sent to the terminal is restricted by first defining a route between desired route points and thereafter selecting from the 3D model comprising surface elements at least some of the surface elements that are visible to said route. A partial model comprising only these selected surface elements is transmitted to the user workstation, and in addition the requisite description of how the route animation is constructed on the basis of the partial model.
Patent FI-20020619-A0 (FI)
Inventor: YLITALO JARI
IPC: B60L50/10
Filed: 2002-03-28
Abstract: The present invention relates to a propeller drive arrangement for vessels used in water-borne traffic, and specifically to a propeller drive arrangement containing a propulsion unit, and to such an arrangement, which contains a propulsion unit, which is turnable relative the hull of the vessel. Particularly the present invention relates to a system and a method for braking a motor of a propulsion unit. The solution for braking the propulsion unit according to the present invention is based on short-circuiting a permanently magnetized motor.
Patent FI-20040230-A0 (FI)
Inventor: HELOSVUORI JUHANI
IPC: H01F27/10
Filed: 2004-02-13
Abstract: The invention relates to a liquid-cooled choke comprising a choke core (1), a choke coil (2) and a path (3) for a cooling liquid to cool the choke. The choke core (1) is divided into at least two parts (1a, 1b) arranged in a cooling profile (4) to which the path (3) for the cooling liquid is arranged and which at the same time provides the choke with a frame and an assembly jig.
Patent IL-117812-A0 (IL)
Title: N-substituted heterocyclic compounds their preparation and pharmaceutical compositions containing them
IPC: A61P25/04
Filed: 1996-04-03
Abstract: The present invention relates to novel N-substituted amino acids and esters thereof in which a substituted alkyl chain forms part of the N-substituent or salts thereof, to methods for their preparation, to compositions containing them, and to their use for the clinical treatment of painful, hyperalgesic and/or inflammatory conditions in which C-fibers play a pathophysiological role by eliciting neurogenic pain or inflammation.
Patent IL-124669-A0 (IL)
Title: Flush-mounted electrical installation unit having a swing-out cover
IPC: H02G3/18
Filed: 1998-05-27
Abstract: A below-ground protective enclosure for electrical equipment has a cover (3) which tilts about a horizontal axis (14) in a frame (2) so that in the closed position it is flush with the ground surface and seals against the packing ring (15). A spring-biased sliding bolt mechanism opposite the axis (14) provides secure fixing via a gate profile in the closed and one or more open positions of the cover (3) to facilitate cabling or other work. Release from a bolted condition is achieved using a tool entered through the slot (3c) to engage the sliding plates (4,13) which when moved against the spring pressure free the latch (6).
Patent IL-124686-A0 (IL)
Title: Process for the manufacture of a colour-marked object
IPC: B41M5/46
Filed: 1996-11-28
Abstract: Process for the manufacture of a colour-marked object by irradiating the surface of the object with laser light, characterized in that the object, at least at the location where the marking is applied, consists of a plastic composition which contains at least three light-absorbing components which exhibit a maximum in their light absorption spectra at different wavelengths and lose their light-absorbing capacity under the influence of laser light, with the marking being applied in the form of matrix dots by irradiating the object's surface at the location of the matrix dots with laser light of such wavelength and intensity and for such duration that at least one of the light-absorbing components has wholly or partially lost its light-absorbing capacity.
Patent IL-129781-A0 (IL)
Title: Mathematical teaching apparatus and method
IPC: G09B1/30
Filed: 1997-11-19
Abstract: A mathematical teaching apparatus comprising block elements that fit inside a block element container. The block element container will not close until the proper number of block elements are inserted. For teaching counting and addition concepts for a number base, such as base ten, a user will quickly grasp the concepts of grouping an arbitrary number of block elements into units, such as ones, tens and hundreds. A container for holding block element containers is also provided. The block elements and containers have the same shape, and maintain a proportional ratio with each other. All block elements and containers are counted and grouped using counting devices which provide an indication of the number of units of each type present. The counting devices also signal when ten block elements or ten block element containers are inserted, signaling to a user that the block elements or containers should be inserted into a next-larger size container. A method of teaching using the mathematical apparatus is also presented. The mathematical teaching apparatus allows children to learn the concepts of number magnitude, addition and subtraction, including carrying and borrowing. A computer program implementing these ideas can also be used to present the mathematical concepts.
Patent IL-130470-A0 (IL)
Title: Process for the preparation of heteroaryl-zinc halides
IPC: C07D277/30
Filed: 1998-01-12
Abstract: A process for the preparation of heteroaryl-zinc halides of the formula (II): Het-Zn-X, wherein Het is an optionally substituted 5 or 6 membered aromatic heterocyclic group with one or two heteroatoms selected among nitrogen, oxygen or sulphur; X is a chlorine, bromine or iodine atom; comprising metallation reaction of heteroarylhalide with metallic zinc optionally activated by washing with acids, is described. Compounds of the formula (II) are intermediates useful in the synthesis for the preparation of compounds endowed with pharmacological activity.
Patent IL-133217-A0 (IL)
Title: Broad band antennas
IPC: H01Q1/36
Filed: 1999-11-30
Abstract: The outer turns (3) of a spiral antenna are radially modulated to extend the low-frequency response. The modulation amplitude increases progressively with spiral angle. The unmodulated region may consist of equally-spaced inner turns (1), and outer turns (2) whose spacing increases with angle. The track width of the outer turns may progressively decrease. Alternatively the track width of the outer unmodulated region may increase, the width of the modulated turns then progressively decreasing. Similar modulation may be applied to the outer ends of the arms of sinuous antennas. <IMAGE>
Patent IL-146367-A0 (IL)
Title: High capacitance niobium powders and electrolytic capacitor anodes
IPC: C22C27/02
Filed: 2000-05-05
Abstract: A niobium powder is described which when formed into an electrolytic capacitor anode, the anode has the capacitance of at least 62,000 CV/g. Methods of making flaked niobium powder which have high capacitance capability when formed into electrolytic capacitor anodes is also described. Besides niobium, the present invention is also applicable to other metals, including valve metals.
Patent IL-146382-A0 (IL)
Title: Adjuvant combination formulations
IPC: A61P31/16
Filed: 2000-05-12
Abstract: The use of 3-O-deacylated monophosphoryl lipid A or monophosphoryl lipid A and derivatives and analogs thereof, in combination with a cytokine or lymphokine such as granulocyte macrophage colony stimulating factor or interleukin-12 is useful as an adjuvant combination in an antigenic composition to enhance the immune response in a vertebrate host to a selected antigen.
Patent IL-162283-A0 (IL)
Title: Medicament cartridge having identification means
IPC: A61M5/24
Filed: 2002-12-05
Abstract: Many of those having diabetes take a combination of slow and fast acting types of insulin. It is important that the different forms of medicament do not become confused and that the patient does not receive the incorrect medicament. In combination a medicament delivery apparatus and a medicament cartridge are provided, the medicament delivery apparatus including at least one switch and the medicament cartridge comprising a cartridge housing 4 within which a medicament is provided, a displaceable piston 14 located internally at one en of the housing 4 and a raised ring 10 of material about an external periphery of the medicament cartridge, the ring 10 of material being of sufficient dimensions, in use, to trip the at least one switch of the medicament delivery apparatus.
Patent IL-164366-A0 (IL)
Title: Biological substance-immobilized gel and microarray using the same
IPC: C40B50/06
Filed: 2003-04-03
Abstract: A gel has a bio substance fixed to it wherein the bio substance is fixed to such gel that contains 2-7 weight% N,N-dimethylacrylamide. Independent claims are also included for: (1) a similar gel containing a composition (weight%) of N,N-dimethylacrylamide (2-7) and crosslinking agent (0.1-1.5); (2) a method for producing the gel having a bio substance by fixing the bio substance to such N,N-dimethylacrylamide-containing gel; (3) hollow tube bodies filled with the gel; (4) a process for producing micro arrays with the gel by bundling a number of the filled hollow tube bodies and cutting in the crossing direction along the lengthwise direction of such bundle; (5) micro arrays produced by placing the gel at a number of regions on them for imaging purposes, or by using the bundles of filled tube bodies; and (6) a method for detecting an assay object by reacting such analyte in a sample with the micro array before detection.