baber/WOPTO huggingface dataset:
Patent FI-960902-A0 (FI)
Inventor: JANIN ROBERT
IPC: C07D317/46
Filed: 1996-02-27
Abstract: A process for the synthesis of fluorinated derivs. comprises a step in which a substrate is reacted with a cpd. comprising the association of a Bronsted base with a defined number (n) of HF species (n=3-20, pref. 15, and esp. 10). The substrate comprises at least one halo-carrying C of sp<3> hybridisation, attached to at least two halogens, of which at least one is a halogen of atomic number greater than F, bonded to at least one chalcogen.
Patent FI-980604-A0 (FI)
Inventor: KOIVUNEN ERKKI
IPC: A61P19/00
Filed: 1998-03-18
Abstract: The present invention relates to novel matrix metalloproteinase (MMP) inhibitors and down-regulators, to a process for the preparation of these inhibitors, to pharmaceutical compositions comprising these inhibitors/down-regulators, to the use of the novel MMP inhibitors for the manufacture of pharmaceutical and research preparations, to a method for inhibiting and down-regulating MMP-dependent conditions either in vivo or in vitro, to a method for inhibiting formation, synthesis, expression activations, and/or functions as well as actions of matrix metalloproteinases, and to the use of the novel MMP inhibitors and down-regulators in biochemical isolation and purification procedures of matrix metalloproteinases.
Patent AP-9801217-A0 (AP)
Title: Optical digital media recording and reproduction system.
Inventor: EDELKIND JAMIE
IPC: G11B7/0025
Filed: 1996-09-27
Abstract: The present invention provides a new method and system for producing a digiatl optical recording. The process can be divided into two separate operations: mastering of the optical recording on the surface of an elongated member, such as a cylinder, etc, and fast replication of the master record onto the surface of flexible film which is essentially parallel to the surface of the cylinder, etc.
Patent IL-58490-A0 (IL)
Title: Derivatives of polyene macrolide antibiotics process for the preparation thereof and pharmaceutical compositions containing them
IPC: A61K31/70
Filed: 1979-10-18
Abstract: Disclosed are novel derivatives of polyene macrolide antibiotics of the general formula <CHEM> wherein M is a polyene macrolide antibiotic moiety containing an amino sugar moiety, the amino group of which is substituted by X, wherein X is <CHEM>     -@-@-NH-@-@-NR3R4 (III),  -R5 or hydrogen, wherein A and B independently of each other are hydrogen or NR3R4 or one of A and B is hydrogen and the other is   -NH-@-R-NR3R4; R5 is an  alpha -amino acyl group; n is 1 to 3, t is zero or 1, and when t is zero p is zero to 4 and when t is I p is zero;  z is zero or I, and Y is hydrogen, alkyl, allyl, propargyl, benzyl or phenylpropargyl, with the proviso that, when X is hydrogen, z must be I and Y allyl, propargyl, benzyl or phenylpropargyl;  and the pharmaceutically acceptable acid addition salts thereof. The novel compounds may be prepared by methods known per se. Preferably the compounds are prepared by reaction of respective polyene macrolide antibiotic with a reactive derivative of a compound HOX wherein the amino group(s) is (are) protected. The compounds wherein X is hydrogen and Y is allyl, propargyl, benzyl or phenylpropargyl can be prepared by reaction of the respective N-protected polyene macrolide antibiotic with a reactive derivative of propene, propyne, phenylpropyne or toluene. The compounds show antifungal activity and are useful in the treatment of fungal infections.
Patent IL-87835-A0 (IL)
Title: Ceramic cutting tool inserts and production thereof
IPC: B24D3/34
Filed: 1988-09-23
Abstract: This invention is concerned with a hard, tough, thermally conductive ceramic cutting tool insert consisting essentially of a zirconia alloy in a hard refractory ceramic insert and the product thereof. The ceramic cutting tool insert exhibits performance conducive to use in turning operations and/or milling operations. In particular the invention provides a ceramic cutting tool insert exhibiting a hardness greater than 15 GPa, a toughness greater than 6 MPa 2ROOT m, and a thermal conductivity greater than 14 Wm<-><1><0>K<-><1> consisting essentially, expressed in terms of percent by weight, of 20-45% zirconia alloy and 55-80% hard refractory ceramic matrix, said alloy consisting essentially, expressed in terms of mole percent on the oxide basis, of 1-4% of a toughening agent selected from the group consisting of YNbO4, YTaO4, MNbO4, MTaO4, and mixtures thereof, wherein M consists of a cation which replaces a Y cation on a mole basis selected from the group consisting of Mg<+><2>, Ca<+><2>, Sc<+><3>, and a rare earth metal ion selected from the group consisting of La<+><3>, Ce<+><4>, Ce<+><3>, Pr<+><3>, Nd<+><3>, Sm<+><3>, Eu<+><3>, Gd<+><3>, Tb<+><3>, Dy<+><3>, Ho<+><3>, Er<+><3>, Tm<+><3>, Yb<+><3>, Lu<+><3>, and mixtures thereof, and the remainder zirconia.
Patent IL-97624-A0 (IL)
Title: Selective separation of gases by means of high pressure facilitated membranes
IPC: B01D53/22
Filed: 1991-03-21
Abstract: A process for the selective separation of at least one component eg propylene of a gaseous feedstream comprises passing the feedstream containing the component through a separation unit (50), the separation unit (50) containing a porous membrane (53), eg in the form of a hollow fiber, the membrane (53) having a feed side and a permeate side, and a pore size of from about 10 Angstroms to about 200 Angstroms. Disposed in the pores of the porous membrane (53) is a facilitator liquid comprising a carrier eg silver nitrate dissolved in a suitable solvent. The process includes the steps of   (a) dissolving the component in the facilitator liquid on the feed side of the porous membrane (53) at the feed gas/membrane interface;   (b) forming a component-carrier complex; (c) diffusing the complex to the permeate side of the porous membrane (53): and   (d) releasing the component from the carrier.   <IMAGE>
Patent AU-PQ821500-A0 (AU)
Title: Mask
IPC: A61M16/06
Filed: 2000-06-19
Abstract: A mask ( 10 ) for supplying gas under pressure to the nasal airway of a human includes a manifold ( 30 ) including means ( 36 ) for connection to a gas supply means, a gas supply element or elements ( 26 ) for providing said gas to the nasal airway without pressurising the exterior of the nose and a flexible strap ( 12 ) formed from an elastomeric material for securing the manifold ( 30 ) in position. The strap ( 12 ) extends either side of the manifold ( 30 ) and is shaped to generally conform with the shape of the upper lip and adjacent cheek area to act as a distributed anchor means for the mask ( 10 ).
Patent FI-20010267-A0 (FI)
Inventor: SYVAENNE TUOMO
IPC: G06F11/20
Filed: 2001-02-13
Abstract: A method (400, 500, 600, 700) for synchronizing state information in a security gateway cluster comprising at least two nodes comprises the following steps. Synchronizing (403) state information by sending state information from a first node of said at least two nodes, detecting (401) in said security gateway cluster a predetermined irregularly occurring action, and initiating (402) synchronization of state information as a response to said action. The state information is sent to at least a second node of said at least two nodes. Corresponding computer program, computer program product, software entities (910, 920), a node (900) of a security gateway cluster (950) and a security gateway cluster are also presented. <IMAGE>
Patent FI-20040434-A0 (FI)
Inventor: MAEKINEN ANTTI
IPC: D03D15/567
Filed: 2004-03-22
Abstract: The invention relates to a method of making a solid-liquid filtration cloth, a solid-liquid filtration cloth, and a filter in which the solid-liquid filtration cloth is arranged. The filter cloth (7) is provided with yarns (13b) having a highly changing length and a long free run in the weave. When the length of the yarns (13b) is allowed to shorten significantly, a filtration portion (15) on the side of a surface (14) of the cloth obtains a corrugated shape, providing the cloth with a large filtering area.
Patent IL-101055-A0 (IL)
Title: Protective garment containing polybenzazole
IPC: D03D15/00
Filed: 1992-02-24
Abstract: Fabrics containing polybenzazole fibers have high cut-resistance, and can be used to make cut-resistant and flame-resistant garments.
Patent IL-107811-A0 (IL)
Title: Process for forming borated lubricating oil additive
IPC: C10M159/16
Filed: 1993-11-30
Abstract: A low sediment process for forming a borated, oil soluble, polymer-substituted, nitrogen- or ester-containing lubricating oil additive. A polymer-substituted, nitrogen- or ester-containing additive in the presence of a solvent therefor, is contacted under boronating reaction conditions in a reaction zone with particulate boric acid. The boric acid has a particle size distribution in lubricating oil characterized by a  phi  value of not greater than about 450. The  phi  value is the ratio of said particles' total spherical volume divided by said particles' total spherical external surface area; i.e.,   <IMAGE>   wherein, for each of a plurality of distribution segments defining a particle size range; di is the average particle diameter for the ith distribution segment; Ni is the particle volume percent of the ith distribution segment; and the sum is taken over all the distribution segments.
Patent IL-110457-A0 (IL)
Title: Method and apparatus for tying articles
IPC: E04G21/12
Filed: 1994-07-26
Abstract: A method and an apparatus for automatically binding together rod-shaped articles such as reinforcing bars or tubular-shaped and other various articles with a wire-shaped binding material in an easy and portable manner. The apparatus comprises binding material feeding means (6), binding material bending means (8), encircling guide means (9), binding material cutting means (7) and twisting means (11). A portion of a continuous wire-shaped binding material (w) fed from the binding material feeding means is engaged with the binding material bending means to produce a starting point for bending into a U-shape. In this state, the binding material is fed from one side whereby it is guided around articles being bound together by the encircling guide means (9) while being bent into a substantially U-shape. The binding material is cut into a predetermined length and both ends of the cut binding material is twisted by a hook (25) of twisting means (11). The binding material is automatically bent into two lines so as to bind the articles in a roll, so that the binding material is increased in strength to bind strongly the articles with an extraordinarily strong binding force. Furthermore, as twisting progresses from a hook side toward the articles being bound together, it can progress until looseness of a bound portion of the articles being bound together is eliminated whereby tight binding will result.   <IMAGE>
Patent IL-111685-A0 (IL)
Title: Intradermal drug delivery device
IPC: A61N1/30
Filed: 1994-11-17
Abstract: An intradermal drug delivery device for delivering a liquid drug to a subject via the subject's skin includes a housing having a lower surface provided with an adhesive coating for adhering the housing to the subject's skin. An expansible-contractible chamber within the housing defines a reservoir which is expanded upon being filled with the drug and contracted to dispense the drug. A hollow needle extends through the lower surface of the housing and has an inner end which communicates with the reservoir and an outer end which projects outwardly of the housing a short distance to penetrate through the epidermis and into the dermis of the subject's skin when the housing is adhered thereto. The device permits delivery of drugs of relatively large molecular size and at slow rates which can be precisely controlled. A method of delivering a liquid drug intradermally includes adhering the intradermal delivery device to the skin of the subject and activating the means for actively discharging the at least one drug from the reservoir to the subject's skin via the needle.
Patent IL-135810-A0 (IL)
Title: Method for the generation if isa simulators and assemblers from a machine description
IPC: G06F11/28
Filed: 1998-10-30
Abstract: A method for generating software development tools to be used in hardware and software development. The invention is utilized by processing a hardware description and a syntax description of programmable electronics, such as a microprocessor, and generating a set of development tools useful to a hardware and/or software developer. Some of these tools include, for example, simulators, assemblers, decoders, disassemblers, behavior semantics, and attribute grammars.
Patent IL-136306-A0 (IL)
Title: Anticonvulsant and chemical nervous system-active bis(fluorophenyl) alkylamides
IPC: A61K31/16
Filed: 1998-12-09
Abstract: Bis(Fluorophenyl)alkylamides have been chemically synthesized which possess beneficial pharmacological properties (e.g., anticonvulsant activity) useful for the treatment of neurological diseases or disorders, such as, for example, epilepsy, convulsions, and seizure disorders. The preferred compounds of the invention also cause little sedation and have high therapeutic and protective indices in animal models of epilepsy. These compounds further possess long pharmacologic half-lives, which, in practical clinical therapeutic application, should translate into once-a-day dosing, of great benefit to patients suffering from these diseases and/or disorders. These compounds may also be of further clinical utility in the treatment of other diseases and disorders of the central and peripheral nervous systems, or diseases or disorders affected by them, including, but not limited to, spasticity, skeletal muscle spasms and pain, restless leg syndrome, anxiety and stress, and bipolar disorder.
Patent IL-154951-A0 (IL)
Title: A device and a method for filtering a fluid
IPC: B01D39/04
Filed: 2001-09-17
Abstract: A device for filtering a fluid includes a fiber housing having an inlet end with at least one inlet and an outlet end with at least one outlet. The fiber housing surrounds and defines an outer bound for a plurality of fibers extending longitudinally in the fiber housing between the inlet end and the outlet end, whereby longitudinally extending interspaces is provided between the fibers, with the interspaces defining a plurality of flow passages for the fluid. At least part of the fiber housing is formed of a flexible membrane surrounding the fibers, and a compression tool is provided for creating a pressure on an outer surface of the flexible membrane thereby compressing the fibers in a radial direction at least one location along the length of the fibers.
Patent IL-156584-A0 (IL)
Title: Substituted triazole diamine derivatives as kinase inhibitors
IPC: A61K31/4178
Filed: 2001-12-21
Abstract: The present invention provides substituted triazole diamine derivatives as selective kinase or dual-kinase inhibitors and a method for treating or ameliorating a selective kinase or dual-kinase mediated disorder.
Patent IL-162069-A0 (IL)
Title: Gabusectin derivatives, processes for preparing them and their use
IPC: C07D207/44
Filed: 2002-11-07
Abstract: 3-(Octahydronaphth-1-yl-methylene)-pyrrolidine derivatives (I) and its derivatives, are new.  Gabusectin compounds of formula (I) and their stereoisomers and tautomers (including mixtures in all ratios) and salts are new.  R1-R3 = H; or 1-6C alkyl, 2-6C alkenyl or 2-6C alkynyl (all optionally substituted by 1-2 of OH, =O, halo or NH2; or 1-6C alkoxy, 2-6C alkenyloxy, aryl, 1-6C alkylamino or 2-6C alkenylamino (all optionally substituted by CN, amide or oxime functions));  R4 = 1-6C alkyl or 2-6C alkenyl (both optionally substituted as in R1-R3); R5 = H or Me; X1-X5 = O, NH, N-(1-6C alkyl), N-(2-6C alkenyl), N-(2-6C alkynyl), N-acyl, N-aryl, N-O-R1 or S. Independent claims are also included for:  (1) the preparation of (I); and  (2) the new microorganism ST003236 (DSM 14476).
Patent IL-174545-A0 (IL)
Title: Hair growth inhibition
IPC: A61K8/66
Filed: 2006-03-23
Abstract: The invention relates to the use of a composition for the preparation of a hair growth inhibitor and furthermore to the use of a system for the preparation of a hair growth inhibitor. The invention also relates to a composition comprising at least one enzyme, a solvent, and a water activity reducing agent. Moreover, the invention concerns a system for hair growth inhibition comprising a first component and a second component, wherein the first composition of the first component comprises at least one enzyme, a solvent and a water activity reducing agent, and wherein the second composition of the second component comprises an enzyme-activating agent and/or a anti-inflammatory, penetration-promoting agent and/or a preservative agent. The invention in addition relates to a method for inhibiting hair growth and a method for the preparation of a hair growth inhibitor.
Patent IL-175346-A0 (IL)
Title: Floorboard, system and method for forming a flooring, and a flooring formed thereof
IPC: E04F15/04
Filed: 2006-05-01
Abstract: A method of producing floor panels is disclosed. The method comprises the steps of separating a sheet- or roll formed surface material (51) into surface strips (53) and gluing said surface strips to a core (50) with a space (54) between the surface strips (53).
Patent IL-175970-A0 (IL)
Title: Conduit for conveying media
Filed: 2006-05-28
Abstract: A conduit pipe for conveying media, having a core pipe made of a copper alloy and a jacketing made of a plastic material from the group of the polyolefins having functional groups. The ratio between the thickness of the jacketing wall and the thickness of the core pipe wall ranges between 2:1 and 14:1, while the ratio between the thickness (D) of the core pipe wall and its inside diameter (ID) ranges between 0.01 and 0.05.
Patent IL-181737-A0 (IL)
Title: Method for the low-deformation diffusion-welding of sintered unoxidised ceramic components, and structure consisting of unoxidised ceramic with a seamless join
Filed: 2007-03-06
Abstract: To bond two components of a sintered and non-oxide ceramic material, they are joined together by diffusion welding in a hot press in a protective gas atmosphere. They are heated to a temperature of at least 1600 [deg] C, preferably >= 1800 [deg] C and especially >= 2000 [deg] C. They are pressed together with a low distortion into a monolith, with a plastic distortion towards the application of force of = 5% and preferably = 1%.
Patent RO-133355-A0 (RO)
Title: Counter-rotating wind motor system with differential speed amplifier and counter-rotating electric generator
Inventor: NEAGOE MIRCEA
IPC: F16H37/08
Filed: 2019-01-04
Abstract: The invention relates to a wind motor system meant to convert the wind energy into electric energy. According to the invention, the system consists of two coaxial counter-rotating wind rotors (A and B), a main one and a secondary one, respectively, and a counter-rotating electric generator having a mobile rotor (E) and a mobile stator (F), interconnected with a differential planetary speed amplifier with two counter-rotating inputs and two counter-rotating outputs, formed by coupling a conical differential planetary unit (C) with a cylindrical differential planetary unit (D) with simple satellites, where the conical differential planetary unit (C) comprises a sun bevel gear (1), made integral with the main wind rotor (A), a double satellite comprising two coaxial satellite bevel gears (2 and 3) and articulated by a rotation coupling on a mobile axes-support element (4), which is made integral with the secondary wind rotor (B) and articulated through a rotation coupling on the sun gear shaft (1), the second satellite bevel gear (3) engaging with the sun gear (1), and the first satellite gear (2) with a sun bevel gear (5), the cylindrical differential planetary unit (D) comprises a cylindrical gear wheel (6) with interior toothing made integral with the sun bevel gear (5), another axes-support element (7) made integral with the sun gear (1) and articulated through a rotation coupling to a cylindrical satellite gear (8), which simultaneously engages with the cylindrical gear wheel (6) and a cylindrical sun gear (9) with exterior toothing, where the mobile rotor (E) is made integral with the cylindrical sun gear (9), and the mobile stator (F) is made integral with an element (10) fixed coaxially with the cylindrical gear wheel (6) .
Patent RO-137526-A0 (RO)
Title: Mobile rotating horizontal gasifier
Inventor: DINCĂ CRISTIAN- FLORIAN
IPC: F23G5/027
Filed: 2023-02-27
Abstract: The invention refers to a mobile rotating horizontal gasifier intended for energy recovery from biomass/waste. According to the invention, the gasifier comprises a chassis (A) to which a vertical body (B), a horizontal rotating body (C), a feed system supporting body (D), a feed system (E) of dual screw-piston type and an ash discharge system (F) are attached, where, in order to have a precise sequential biomass/waste feed, the feed system (E), which is mounted in the body (D) supporting the feed system, has a dual piston-screw drive mode, consisting of a support body (6) rigidly attached to a plate (7) which is rigidly mounted in the body (D) supporting the feed system by means of a body (15), in the support body (6) there being located a main body (8) which has mounted at one end a motor (9) which drives a short screw (10) and which, being operated by a linear actuator (12) and being attached to a linear guide (11), slides inside the support body (6), the main body (8) working in tandem with a hatch (13) which slides within the support body (6) and which is operated by the linear actuator (14), a useful loading space (16) being formed between the hatch (13) and the end of the short screw (10).
Patent AP-2000001950-A0 (AP)
Title: Paroxetine maleate.
Inventor: JACEWICZ VICTOR WITOLD
IPC: C07D405/12
Filed: 1999-04-09
Abstract: Paroxetine maleate and its preparation and use in the treatment and prevention of inter alia depression
Patent IE-910703-A1 (IE)
Title: Continuously operating massage drum, and method for massaging meat
Inventor: LOGTENBERG HARRY
IPC: A23L13/70
Filed: 1991-03-04
Abstract: A continuously operating massage drum suitable for mechanically massaging salted or unsalted meat products is disclosed. Said drum is provided with drive means for rotating the drum, and end plates with a feed and discharge aperture respectively. The internal surface of the drum is provided with projecting massage elements consisting of an inside wall (4) which is continuously ribbed in the peripheral direction. Preferably the inside wall (4) of the drum has an essentially star-shaped cross-section. The drum is further provided with residence time spread reducing means, advantageously consisting of an internal thread, preferably of 0,1 to 0,8 m, and adapted to the internal shape of the drum. <IMAGE>
Patent MA-19106-A1 (MA)
IPC: A61K31/395
Filed: 1981-03-21
Abstract: Thioformamide derivatives of the formula:   <IMAGE>   wherein R represents hydrogen or alkyl of 1 through 4 carbon atoms, and (i) Het represents a heterocyclic radical selected from pyrid-3-yl, pyrid-4-yl, pyridazinyl, pyrazinyl, pyrimidinyl, quinolyl, imidazolyl, naphthyridinyl, quinoxalinyl and quinazolinyl, X represents sulphur or oxygen and Y represents sulphur or oxygen, a valency bond or methylene, or (ii) Het represents pyrid-2-yl, X represents sulphur or oxygen and Y represents sulphur or oxygen or methylene, or (iii) Het represents pyrid-2-yl, X represents oxygen and Y represents a valency bond, are new compounds possessing useful pharmacological properties. They are particularly useful in the treatment of gastrointestinal ulcers and in the treatment of hypertension, depending on the definition of the symbol Het.