baber/WOPTO huggingface dataset:
Patent EA-011033-B1 (EA)
Title: 3-substituted-2-(arylalkyl)-1-azabicycloalkanes and methods of use thereof
Inventor: MAZUROV ANATOLY A
IPC: C07D487/08
Filed: 2004-02-20
Abstract: The present invention relates to 3-substituted-2-(arylalkyl)-1-azabicycloalkanes of formula:pharmaceutically acceptable salts thereof, wherein: m is 2 and n is 1 and p is 1; X is oxygen or NR', Y is oxygen or sulfur, Z is NR', a covalent bond or a linker species A, A is -CR'= CR'-, wherein when Z is a covalent bond or A, X must be NR' nitrogen, Ar is an unsubstituted or substituted, comprising: phenyl, pyridinyl, thienyl, pyrrolyl, indolyl, benzimidazolyl, benzothiephenyl, benzofuranyl, naphthofuranyl, naphthalenyl; Cy is pyridinyl. The invention also relates to said compounds, radiolabelled, pharmaceutical compositions comprising said compounds, pharmaceutical and diagnostic compositions, comprising radiolabelled compounds, use of such compositions for diagnosis of CNS disorders or for monitoring in patients subtypes of selective nicotinic receptors and to methods of treatment using said compounds.The compounds exhibit activity at nicotinic acetylcholine receptors (nAChRs), particularly the a7 nAChR subtype, and are useful towards modulating neurotransmission and the release of ligands involved in neurotransmission. Methods for preventing or treating conditions and disorders, including central nervous system (CNS) disorders, which are characterized by an alteration in normal neurotransmission, are also disclosed. Also disclosed are methods for treating inflammation, autoimmune disorders, pain and excess neovascularization, such as that associated with tumor growth.
Patent EA-012601-B1 (EA)
Title: Plant growth regulation
Inventor: BASTIAANS HENRICUS M M
IPC: A01N43/82
Filed: 2005-04-30
Abstract: The present invention relates to the use of a compound which is a 3,4-disubstituted maleimide derivative of formula (I) or an agriculturally acceptable salt thereof,wherein radicals have values as defined in the invention claims for plant growth regulation, to a composition for plant growth regulation comprising one or more compounds of formula (I) or an agriculturally acceptable salt thereof, carriers and/or surfactants useful for plant protection formulations, to the use of said composition for plant growth regulation, in which the plant is a monocotyledoneous or dicotyledoneous crop plant and to a method for growth regulation in crop plants, which comprises applying an effective amount of a compound of formula (I) to the site where the action is desired said method comprising applying to plants, to seeds from which they grow or to the locus in which they grow, a non-phytotoxic, effective plant growth regulating amount of one or more compounds of formula (1).
Patent EA-012453-B1 (EA)
Title: Reverse micelles based on phytosterols and acylglycerols and therapeutic uses thereof
Inventor: MAUREL EAN
IPC: A61K9/00
Filed: 2005-11-02
Abstract: The present invention relates generally to reverse-m ice liar system comprising a hydrosoluble therapeutically active agent. Reverse micelles according to the invention are particularly useful to deliver drugs. The present invention also relates to pharmaceutical composition comprising said reverse micelles and methods for preparing the same.
Patent EA-013680-B1 (EA)
Title: Microspherical vascular embolus of sodium alginate containing a gynecological pharmaceutics and preparation thereof
Inventor: XU CONGJIAN
IPC: A61K9/02
Filed: 2005-04-15
Abstract: The present invention relates to a form of the microspherical vascular embolus of sodium alginate containing the gynecological pharmaceutics and to the preparation thereof. The preparation consists of the following stages: preparing a solution of the gynecological pharmaceutics, sodium alginate and divalent metals cations, for example BaCl
Patent EA-014007-B1 (EA)
Title: Method of damp proof bulkhead erection in underground working
Inventor: SMYCHNIK ANATOLIJ DANILOVICH
IPC: E21F15/00
Filed: 2008-10-24
Abstract: The invention concerns mining engineering and may be used for isolation of underground working watered ground from a mining zone. The proposed method of drilling-and-blasting damp-proof bulkhead erection in an underground working allows improving of damp-proof properties of drilling-and-blasting rock bulkhead and thereby improving of underground work safety in difficult hydrogeological conditions. The assigned objective is accomplished in the following manner. The method of drilling-and-blasting rock bulkhead reaction by roof collapse, including two-stages formation of embankment by blasting of two sections of roof with reservation between them of rock mass in the shape of inverse trapezia, provides for forming from the inflow side an embankment which fully blocks the working. From the side opposite to the inflow a waterproof rubber-fabric membrane, whose edges are hermetically and nohermetically fixed on the bottom, walls and roof of the working, is put on the embankment material; the rubber-fabric membrane is covered with a layer of retaining lump rock by a pinpoint blast of the second section of the roof. The waterproof rubber-fabric membrane area and solidity, width of zone of its contact to the bottom, roof and walls of the working, height, volume and size of embankment lumps and retaining lump rock layer covering the rubber-fabric membrane are calculated depending on the roof rock properties, expected shifts of embankment wall covered with the rubber-fabric membrane and possible hydrostatic head.
Patent EA-013392-B1 (EA)
Title: Process for preparing a catalyst component for propylene polymerization
Inventor: RAMJOIE YVES JOHANN ELIZABETH
IPC: C08F4/654
Filed: 2007-05-23
Abstract: The invention relates to a process for preparing a polymerization catalyst component wherein a solid compound with formula Mg(OR)Clwherein x is larger than O and smaller than 2, and each R, independently, represents an alkyl group, said compound being obtained by reacting a Grignard compound with an alkoxy- or aryloxy-containing silane compound, is contacted with at least one activating compound selected from the group formed by internal electron donors and compounds of formula M(OR)(R), wherein M can be Ti, Zr, Hf, Al or Si, each Rand R, independently, represent an alkyl, alkenyl or aryl group, v is the valency of M and w is smaller than v, in the presence of an inert dispersant to give an intermediate reaction product, and wherein the intermediate reaction product is contacted with a halogen-containing Ti-compound. A catalyst system comprising said component shows improved performance in olefin polymerization. The invention also relates to a polymerization catalyst system comprising the catalyst component and to a process of making a polyolefin by contacting at least one olefin with a polymerization catalyst system comprising the catalyst component.
Patent EA-014630-B1 (EA)
Title: Diagonal brace apparatus
Inventor: BEAUJOT NORBERT
IPC: A01B61/00
Filed: 2007-02-06
Abstract: A diagonal brace apparatus for an implement frame includes a bias element connected to a front location on a front portion of the implement frame and connected to a rear location on a rear portion of the implement frame laterally offset from the front location. The bias element is operative to exert a bias force resisting rearward movement of an outer end of the implement frame with respect to an inner end of the implement frame. Conveniently the bias element is provided by a hydraulic cylinder which exerts a bias force and can extend to allow the frame to flex to reduce shock loading on the implement when excessive forces are exerted on the frame.
Patent EA-022797-B1 (EA)
Title: THIAZOLE DERIVATIVES AS STEAROYL-CoA- DESATURASE INHIBITORS, PHARMACEUTICAL COMPOSITION COMPRISING THEM, AND USE THEREOF
Inventor: CHOWDHURY SULTAN
IPC: A61P3/00
Filed: 2009-02-18
Abstract: The present application provides thiazole derivatives that modulate the activity of stearoyl-CoA desaturase. Methods of using such derivatives to modulate the activity of stearoyl-CoA desaturase and pharmaceutical compositions which inhibit the activity of human stearoyl-CoA desaturase (hSCD) comprising thiazole derivatives are also encompassed. The compounds of the present invention are provided for treating in a subject a disorder or disease mediated by inhibition of stearoyl-CoA desaturase, in particular skin disease, wherein the disease is eczema, acne, psoriasis, or keloid scar formation.
Patent EA-019556-B1 (EA)
Title: Molding process for simultaneously making an upper mold and a lower mold and a flaskless molding machine
Inventor: HADANO YUTAKA
IPC: B22C15/02
Filed: 2009-12-25
Abstract: A molding process and a flaskless molding machine for simultaneously making an upper flaskless mold and a lower flaskless mold are provided such that the bottom surfaces of the molds can be in a stable and horizontal position, the stripping of the flasks can be reliably carried out, and the configuration of the molding machine can be simplified. The process comprises the steps of defining a lower molding space by a drag flask that is arranged to enter or leave a molding space in which molds are made, a match plate having patterns on the upper and lower surfaces and mounted on the upper surface of the drag flask, a lower filling frame provided with molding-sand introducing ports on the surfaces of the sidewalls and being connectable to the lower end of the drag flask to allow the lower filling frame to ascend and descend, and an ascendable and descendable lower squeeze board, the step also defining an upper molding space by a cope flask provided with molding-sand introducing ports on the surfaces of the sidewalls and being mountable on the match plate to allow the cope flask to ascend and descend, and an upper squeeze board that is opposed to and fixedly provided above the match plate; simultaneously introducing molding sand into the upper molding space and the lower molding space; squeezing the molding sand by raising the lower squeeze board to simultaneously make an upper mold and a lower mold; drawing the upper mold from the pattern on the upper surface of the match plate, while drawing the lower mold from the pattern on the lower surface of the match plate.
Patent EA-022792-B1 (EA)
Title: Method of producing electric-grade wire from aluminium alloy
Inventor: ANIKEEV YURY GEORGIEVICH
IPC: B21C1/00
Filed: 2010-10-04
Abstract: The technical solution relates to metal forming process, in particular to producing wire by continuous drawing. The technical result is increased microcontinuity of wire surface, its strength, electric conductivity, and reduced cost of wire manufacturing. The technical result is attained by a method of wire manufacturing characterised by cold drawing of wire blanks through a grooved roll, annealing and natural cooling of blanks in a cold furnace at an ambient temperature, then heating in a furnace to 350-450°C and holding in heated state. Then the blanks are cooled and their ends are welded forming a long string, which is subjected to drawing, said cycle of wire blank string treatment being performed repeatedly.
Patent EA-025202-B1 (EA)
Title: Molecule for treating an inflammatory disorder
Inventor: ALONSO BEDATE CARLOS
IPC: C07K14/44
Filed: 2012-05-08
Abstract: The invention provides a L19 source as a medicament, preferably for preventing or treating an inflammatory disorder in an individual.
Patent EA-029768-B1 (EA)
Title: Heterocyclyl compounds
Inventor: DAVE BHAVESH
IPC: C07D471/04
Filed: 2013-03-11
Abstract: The present invention relates to heteroaryl compounds such as MEK inhibitors. The present invention includes heteroaryl compounds of formula I, pharmaceutically acceptable salts thereof, pharmaceutical compositions thereof. The present invention also relates to methods of treating various cancers.
Patent EA-025050-B1 (EA)
Title: Cyclic bridgehead ethers as dgat1 inhibitors
Inventor: CHEN XIN
IPC: C07D417/12
Filed: 2013-04-25
Abstract: The invention relates to compounds of formula (I), useful for treating disorders mediated by acyl coA-diacylglycerol acyl transferase 1 (DGAT1), e.g. metabolic disorders. The invention also provides methods of treating such disorders, and compounds and compositions etc. for their treatment.
Patent EA-027982-B1 (EA)
Title: Use of vegfr-3 inhibitors for treating hepatocellular carcinoma
Inventor: ALAM ANTOINE
IPC: A61K31/4375
Filed: 2013-07-16
Abstract: The present invention is related to the use of inhibitors of vascular endothelial growth factor receptor 3 for treating hepatocellular carcinoma.
Patent EA-036018-B1 (EA)
Title: Use of ultra lightweight particulates in multi-path gravel packing operations
Inventor: MALBREL CHRISTOPHE A
IPC: E21B43/08
Filed: 2015-05-04
Abstract: A well penetrating a subterranean formation may be subjected to a multi-path gravel packing operation by using a fluid containing ultra lightweight particulates having an apparent specific gravity less than or equal to 2.45 which are substantially neutrally buoyant in a carrier fluid. The fluid is flowed through one or more transport tubes which, with a gravel packing screen, constitute a screen assembly. A gravel pack is formed onto the screen of the screen assembly in-situ.
Patent EA-035072-B1 (EA)
Title: NOVEL PHOSPHINANE AND AZAPHOSPHINANE DERIVATIVES THAT ARE TAFIa INHIBITORS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME
Inventor: GLOANEC PHILIPPE
IPC: A61P9/00
Filed: 2017-01-13
Abstract: The present invention relates to compounds of formula (I)as described and defined herein, pharmaceutical compositions comprising said compounds and the use of said compounds that are TAFIa inhibitors in treating, preventing or secondary preventing diseases.
Patent EA-036640-B1 (EA)
Title: Deck hoist tractor for an unmanned offshore platform
Inventor: ENGENE KNUT
IPC: B66C19/00
Filed: 2017-04-18
Abstract: A deck hoist tractor (DHT) for an unmanned platform (1) comprising an elongated base frame structure (12) carrying respective caterpillar drives (18) on each side enabling the tractor (2) to move forward and rearward, characterised in that the tractor (2) further comprising a tower frame structure (10) extending in substantially vertical direction from one end section of the base frame structure (12), which tower frame structure (10) is carrying a cantilevered top frame structure (11) carrying a lifting apparatus (22, 21), said caterpillar drives (18) are located at the same end section as said top frame structure (11), that said base frame structure (12) is extended by respective cantilevered beams (12a) space apart with an opening between them, each cantilevered beam (12) having an adjustable support structure (19) adjacent to their distal end (12b) from the caterpillar drive (18), said cantilevered top frame structure (11) is extended to vertically correspond with said respective cantilevered beams (12a), and said lifting apparatus (20, 21) is arranged to be shifted both forward and rearward, in addition to laterally in said top frame structure in order to position a load supported in the lifting apparatus. The invention also relates to a temporarily installed escape chute (54) and a method for installing a tote tank (70) on the platform (1) and removing the tank from the platform.
Patent EA-038064-B1 (EA)
Title: Method for separating biomass from solid fermentation product
Inventor: BOKHOVE JEROEN
IPC: C12P7/56
Filed: 2017-05-29
Abstract: The invention pertains to a method for separating biomass from solid fermentation product, wherein a slurry comprising biomass and solid fermentation product is provided to the top of a biomass separator unit and an aqueous medium is provided to the bottom of a biomass separator unit, while a product stream comprising solid fermentation product is withdrawn from the bottom of the biomass separator unit and a waste stream comprising biomass is withdrawn from the top of the biomass separator unit. It has been found that the method according to the invention makes it possible to provide a solid fermentation product which comprises very low amounts of remaining biomass, while product loss can be limited.
Patent EA-039274-B1 (EA)
Title: Friction shock absorber
Inventor: GOLOVACh Oleg Nikolaevich
IPC: B61G11/14
Filed: 2019-09-06
Abstract: The invention relates to the field of transport engineering, in particular, to vehicle shock absorbers. The objective is to improve efficiency and reliability of the absorbing device. The shock absorbing device (Fig. 1) comprises a housing (1) formed by wide walls (2), narrow walls (2') and a bottom (3), accommodating a friction unit (4) consisting of a cavity (P) with a bottom (5') and protruding with its outer end (T) from the body (1) of the pressure wedge (5), spacer wedges (6), fixed plates (7) equipped with lateral supports (8') of movable plates (8) and a base plate (9). Between the base plate (9) and the bottom (3), along the longitudinal axis (01) of the housing (1), a back-and-forth device (10) is located that is braced through a centering rod connection (13, 16), resting at one end in a bush (14) of the bottom (3) of the housing (1), and on the other end on the bottom (5') of the cavity (P) of the pressure wedge (5). The pressing wedge (5) is provided with projections (11), the ends (V) of which face the bottom (3) of the housing (1); on the projections (11) of the pressure wedge (5), curved surfaces (f) are formed, between which and the wide walls (2) of the housing (1) said gaps (z) are formed to provide the possibility of free rotation of the pressure wedge (5) relative to the longitudinal axis (O1). Other distinctive features of this invention and links between them are also described.
Patent ES-2166305-B1 (ES)
Title: Mecanismo extractor para maquinas de venta automatica.
Inventor: LOPEZ RUIZ JOSE MARIA
IPC: G07F11/24
Filed: 2000-02-07
Granted: 2003-05-01
Abstract: Mejoras en la patente n° 9900290, relativa a un mecanismo extractor para máquinas de venta automática, especialmente para venta de productos estuchados de recipientes cilíndricos apilados, dispuestos al tresbolillo formando dos columnas verticales que quedan limitadas entre tabiques paralelos. El mecanismo está compuesto por un elemento de retención sobre el que apoya el envase que ocupa la posición inferior, siendo este elemento giratorio en ambos sentidos, girando alternativamente, a partir de una posición intermedia de reposo, con una amplitud angular máxima igual, suficiente para permitir cada vez la salida de un envase perteneciente a una columna diferente.
Patent ES-2192940-B1 (ES)
Title: Telefono movil transformable en consola.
Inventor: CODINA TORRES JUAN BAUTISTA
IPC: G06F1/16
Filed: 2001-06-11
Granted: 2005-02-16
Abstract: El objeto de esta Patente es un teléfono móvil transformable en consola, cuyo uso aparece explícito en el propio enunciado de la invención. Su estructura comprende elementos fijos (caja (1) y la mitad del teclado (2)) y móviles giratorios (pantalla (3) y la otra mitad del teclado (4)), sobre un soporte común (5), susceptible de girar 180°. Durante el giro del soporte (5) alrededor de su centro (6), la pantalla (3) gira sobre sí misma 270° mediante un sector circular dentado (8) unido a ella, que engrana con otro dentado (10) dispuesto en el centro (6) de la plataforma común (5''). Cuando se requiere la transformación, la plataforma (5'') es expulsada de la caja (1) por un resorte (13) desenclavado por un pulsador (11) que la retenía, pudiendo girar libremente el soporte (5) del teclado móvil (4).
Patent ES-2199068-B1 (ES)
Title: Metodo de control antiexplosiones en combustibles gaseosos.
Inventor: LIN TING-AN
IPC: F23N1/00
Filed: 2002-07-17
Granted: 2005-05-01
Abstract: Método de control antiexplosiones en combustibles gaseosos. Método de control antiexplosión de un gas combustible que comprende las siguientes etapas: (a) montaje de un dispositivo detector de realimentación en una base de válvula de control; (b) hacer que el conducto de entrada de gas combustible sea capaz de apertura o cierre inmediatos; y (c) producir la ignición en el quemador con un flujo de gas combustible adecuado. Con intermedio de la apertura y cierre inmediatos se consigue un control estable del flujo de gas combustible mejorando la seguridad del usuario.
Patent ES-2253052-B1 (ES)
Title: Sistema luminoso y fonico de señalizacion y balizamiento.
Inventor: SUAREZ LENCINA NICOLAS
IPC: G09F27/00
Filed: 2004-02-03
Granted: 2007-07-16
Abstract: Sistema luminoso y fónico de señalización y balizamiento. El sistema incluye una estructura base (1) fijable por cualquier medio o sistema apropiado a una superficie que puede ser un techo (2), un paramento o cualquier tipo de superficie en funciones de soporte, estructura base (1) a la que está relacionada una pantalla (4) portadora de las señalizaciones o mensajes que se pretenden visualizar, pudiendo realizarse esa visión mediante un medio de iluminación primario (5), a expensas de la red general, o bien por un medio de iluminación secundario (6), que entra en funcionamiento cuando falla el medio de iluminación primario (5) e incluso por un medio de iluminación terciario (7) basado en componentes luminiscentes que se aplican sobre la pantalla (7) o sobre los mensajes, indicaciones o señalizaciones previstas en ella. Esos tres medios de iluminación se complementan con un sistema fónico (8) que permita transmitir mensajes sonoros en combinación o independientemente a los mensajes iluminables.
Patent ES-2284344-B1 (ES)
Title: Uso de aminoacido tipo micosporina (shimorine) en productos para prevencion y tratamiento de parkinson y alzheimer.
Inventor: DE LA COBA LUQUE FRANCISCA
IPC: A61P25/16
Filed: 2005-08-31
Granted: 2008-11-01
Abstract: Uso de aminoácido tipo micosporina (shinorine) en productos para prevención y tratamiento de Parkinson y Alzheimer. La presente invención se encuadra en el sector biotecnológico y se refiere al uso de un aminoácido tipo micosporina (MAA), concretamente de shinorine aislado del alga roja Gymnogongrus devoniensis, en la preparación de productos de parafarmacia, productos farmacéuticos, preparados nutraceúticos, o en alimentos funcionales, para la prevención y tratamiento terapéutico de Parkinson y Alzheimer.
Patent ES-2272184-B1 (ES)
Title: Pastilla de doble capa para tratamiento y desinfeccion de aguas.
Inventor: HERNANDEZ NUNO JOSE LUIS
IPC: C02F1/76
Filed: 2005-10-05
Granted: 2008-03-01
Abstract: Pastilla de doble capa para tratamiento y desinfección de aguas. Una pastilla de doble capa, una capa de mantenimiento y otra capa de tratamiento de choque, en la que la capa de tratamiento de choque comprende una mezcla reactiva y sustancias adyuvantes, mientras que la capa de mantenimiento comprende una mezcla de sustancias que permiten el mantenimiento prolongado de la calidad del agua, en medios acuáticos tales como, piscinas y parques acuáticos.
Patent ES-2291096-B1 (ES)
Inventor: ALBANDOZ RUIZ DE OCENDA CARMEL
IPC: D06F79/02
Filed: 2005-11-14
Granted: 2008-11-01
Abstract: The invention relates to a cleaning device (1) for a steam iron (2) comprising a base plate (22) with at least two steam outlets (23a to 23g), the steam outlets leading to a steam compartment (21) of the steam iron. The cleaning device is designed as a separate system, having a first cleaning element (13c, 13d, 13e) and at least a second cleaning element for cleaning at least the steam compartment. The first cleaning element can be introduced into a first steam outlet and the second cleaning element can be introduced into a second steam outlet.