baber/WOPTO huggingface dataset:
Patent SK-285381-B6 (SK)
Title: Gonadotropin-releasing hormone (GnRH) antagonist peptide, pharmaceutical composition containing the same, the use thereof and an intermediate
Inventor: SEMPLE GRAEME
IPC: A61K38/00
Filed: 1998-04-13
Abstract: Peptides are provided which have improved duration of GnRH antagonistic properties. These antagonists may be used to regulate fertility and to treat steroid-dependent tumors and for other short-term and long-term treatment indications. These antagonists have a derivative of aminoPhe or its equivalent in the 5- or the 5- and 6- positions. This derivative is modified so as to contain a carbamoyl group or heterocycle, including a urea moiety in its side chain. Particularly effective decapeptides, which continue to exhibit very substantial suppression of LH secretion at 96 hours following injection, have the formulae Ac-D-2Nal-D-4Cpa-D-3Pal-Ser-4Aph(L-hydroorotyl)-D-4Aph(acetyl)- Leu-Lys(isopropyl)-Pro-D-Ala-NH2, and Ac-D-2Nal-D-4Cpa-D-3Pal- Ser-4Aph(L-hydroorotyl)-D-4Amf(Q2)-Leu-Lys(isopropyl)-Pro-Xaa10, wherein Q2 is Cbm or MeCbm and Xaa10 is D-Ala-NH2, D-Ala-ol or Ala-ol.
Patent SK-278276-B6 (SK)
Title: Device for sealing of room between two surfaces
Inventor: BOGSCH ALFRED
IPC: F16J15/44
Filed: 1988-07-28
Abstract: This invention mission statement is the solution of the equipment dealing with the tightening of the space between a moving and a stationary surface, which are in a motion to each other. The tightening plates (4) are fixed to the created fixing plate, in the such sufficient number, they to be able to cover all of the cross-section between the second sheeted surface (5). Each of the tightening plate (4), except the fixing part, consists of the swivelling element closed to motional part and these parts are connected together with the use of the hinge (7). The swivelling moving parts of the tightening plates (4) are equipped with a closing rope (3) having a constant or variable force, however they are covering each other and they are tightening the cross-section between both of the surfaces. The fixing and swivelling moving parts closed to the tightening plates are connected with the use of the tensile spring (2).
Patent CZ-300151-B6 (CZ)
Title: Particulate form of beta-carboline free medicament, process for its preparation and use as well as pharmaceutical composition in which the particulate form is comprised
Inventor: ANDERSON NEIL R
IPC: C07D471/04
Filed: 2000-08-01
Abstract: In the present invention, there is disclosed a free medicament particulate form of a compound having a general formula I and pharmaceutically acceptable salts and solvates thereof, comprising particles of the compound wherein at least 90 percent of the particles have a particle size of less than about 40 microns. There is also disclosed a process for preparing the free medicament particulate form comprising (a) providing a solid, free form of the compound, and (b) comminuting the solid free form of the compound to provide particles of the compound wherein at least 90 percent of the particles have a particle size of less than about 40 microns wherein the medicament is intended particularly for the treatment of male erectile dysfunction or female sexual arousal disorder, wherein the preparation process further comprises the step of admixing the particles of step (b) with one or more pharmaceutically acceptable carriers, diluents, or excipients.
Patent CZ-300134-B6 (CZ)
Title: Two-component geopolymeric binding agent and process for producing thereof
Inventor: BORTNOVSKY OLEG
IPC: C04B7/14
Filed: 2007-02-14
Abstract: In the present invention, there is disclosed a two-component geopolymeric binding agent comprised of a solid component and a liquid component. The solid component is formed by raw materials containing metakaolinite, i.e. slate-clay or kaolin calcined dust, and ground blast furnace slag. The liquid component consists of a liquid sodium-silica glass functioning as an activator. Dry matter of the invented two-component geopolymeric binding agent comprises 43 to 60 percent by weight of a raw material containing metakaolinite, 11 to 37 percent by weight of ground blast furnace slag and 11 to 32 percent by weight of activator. The raw materials containing metakaolinite comprise more than 35 percent by weight of Ali2Oi3 and the activator silicate module SiOi2 : Nai2O is equal to 1.6 to 2.1 : 1. There is also disclosed a process for producing the above-described two-component geopolymeric binding agent, which process is characterized in that, when producing a two-component geopolymeric binding agent consisting of a solid component and a liquid component, said solid component and said liquid component are produced separately. Production of the solid component is characterized by mixing a raw material containing metakaolinite and a ground blast furnace slag in weight ratio 54 to 83 : 17 to 46. The liquid component is then prepared by adding water to a sodium alkaline activator containing 40 to 50 percent by weight of dry matter expressed as a sum of Nai2O + SiOi2 concentrations, in weight ratio within the range of 0 to 0.9 : 1.
Patent CZ-304541-B6 (CZ)
Title: Heating pellet
Inventor: SOUČEK JIŘÍ
IPC: B09B3/32
Filed: 2012-07-20
Abstract: The present invention relates to a heating pellet being characterized in that it is manufactured from disintegrated non-separated flax stems, the total amount of water in the pressed raw material is at the most 22 percent by weight and that it comprises particles of maximum length of 1.2 multiple of the diameter of the pressing apertures in the die.
Patent CZ-307217-B6 (CZ)
Title: An improved manufacturing process and new intermediates for synthesis of ticagrelor
Inventor: ŘÍHA JAROSLAV
IPC: C07D237/10
Filed: 2013-03-14
Abstract: A method for the preparation of ticagrelor of formula I, wherein the key reaction of the entire synthesis is condensation of an amino cyclopentane diol with pyrimidine, providing the isolated intermediate of formula IV. The amino cyclopentane diol is used for the reaction with pyrimidine without any protecting group on the hydroxyls in positions 1 and 2. Using the compound without a protecting group eliminates the necessity of deprotection in the subsequent synthetic steps.
Patent CZ-305917-B6 (CZ)
Title: Passive combined adsorber for purification of water electrolysis hydrogen
Inventor: Tenkrát Daniel
IPC: C01B3/58
Filed: 2014-03-21
Abstract: In the present invention, there is disclosed a passive combined adsorber for removing water vapor and low concentrations of oxygen from hydrogen produced by water electrolysis, the adsorber comprising an adsorber body (1), a lower detachable cover (7) and an upper detachable cover (8), wherein an inlet of hydrogen to be purified is arranged in the lower detachable cover (7). A first active zone (2) is arranged in the lower portion of the adsorber body (1) wherein a desiccating agent of high sorptive capacity of the silicagel type for partial preliminary purification of hydrogen and increase of the efficiency of a second active zone (3) is placed therein. The second active zone (3), following up with the first active zone (2) and being fixedly coupled with the adsorber body (1), comprises a porous material charge of high content of copper for the removal of oxygen from the purified hydrogen. A third active zone (4) comprising a material of a molecular sieve type for the removal of residual moisture and water occurred in the second active zone (3) is arranged above said second active zone (3). In the upper detachable cover (8), there is arranged outlet of the purified hydrogen, whereby the external portion of the adsorber body (1) jacket is provided with a passive air cooler (10) in the form of lamellas or ribs.
Patent CZ-305701-B6 (CZ)
Title: Label precursor, label and use thereof
Inventor: RYBNÍČEK JAN
IPC: G09F3/04
Filed: 2014-10-17
Abstract: The present invention relates to a label precursor consisting only of one layer of plastic sheet, which is able of being stuck to a backing cloth by making simultaneous use of elevated temperature and pressure. The invention further relates to a label comprising a label precursor and data in the form of a printed text or a graphical symbol in the form of an electronic carrier.
Patent CZ-307386-B6 (CZ)
Title: An actuation and steering module of robotic wheeled vehicles
Inventor: MIKUNDA PAVEL
IPC: B60K17/344
Filed: 2015-03-06
Abstract: The module consists of a wheel with actuation and steering suspended on the vehicle body. Each wheel (2) with a hub (10) is connected, in its axis, to a pitman (5), to an epicyclic gear (7) coupled to an electric motor (6) provided, on its right front, with a speed sensor (21) of the electric motor through a cardan shaft (9) via a flange (8). On the pitman (5), an upper arm (3), which is fastened to the vehicle body (1) by means of an upper arm attachment pin (12), is attached oppositely by means of a ball joint (14), and a lower arm, which is fastened to the vehicle body (1) by means of a lower arm attachment pin (13), is attached oppositely by means of a ball joint (15). The ball joints (14) of the upper arm and (15) the lower arm and the ball pin (18) of the actuation located at the end of the steering rod (16) and attached to the pitman (5) are located in one plane formed by these three points perpendicular to the wheel (2) axis. A hydraulic shock absorber (19) and a spiral spring (20) are attached to the upper arm (3) and, with their opposite ends, they are attached to the body (1), to which electric actuators (11) connected by the steering rod (16), by the joint (17) and by the ball pin (18) of the steering with the pitman (5), are also attached.
Patent CZ-308573-B6 (CZ)
Title: Combined test equipment for motor vehicle technical inspection stations
Inventor: Hořejší Josef
IPC: G01M17/007
Filed: 2019-10-14
Abstract: The combined test equipment for motor vehicle technical inspection stations is particularly for measuring exhaust emissions, vehicle braking force and brake performance as part of mandatory periodic vehicle inspections. The combined test equipment is based on a low-profile modular system, where a module with a pair of rolling cylinders is used for each wheel of the vehicle coupled to an electric motor, which is used as a source of load for measuring the braking force of the vehicle wheels.
Patent SK-284637-B6 (SK)
Title: Method for racemate splitting of 2-hydroxypropionic acids
Inventor: BERNARD HARALD
IPC: C07C59/64
Filed: 1999-10-16
Abstract: Process for the racemate resolution of 2-hydroxypropionic acids by reacting the racemic acid with an optically active base and subsequently separating off a diastereomeric salt of acid and base wherein 1-(4-chlorophenyl)ethylamine is used as the optically active base. A preferred embodiment is the racemate resolution of 2-hydroxy-3-methoxy-3,3-diphenylpropionic acid or 2-hydroxy-3-methyl-3,3-diphenylpropionic acid.
Patent SK-284769-B6 (SK)
Title: Pharmaceutical preparations containing pentaerythritol tetranitrate or its metabolites and method for the preparation thereof
Inventor: GUNTHER ULRICH
IPC: A61K9/20
Filed: 1998-10-16
Abstract: Perorally administered pharmaceutical preparations contain as medicinal substance pentaerythritol tetranitrate (PETN) or its metabolites pentaerythritol trinitrate, pentaerythritol dinatrate as either pentaerythrito mononitrate in such amounts which guarantee the patient a sufficient dosage with one administering (per day).
Patent SK-286088-B6 (SK)
Title: Method of mechanical classification of boards or beams and apparatus for making the same
Inventor: BINDER HANS
IPC: B27M1/08
Filed: 2003-06-02
Abstract: It is described apparatus and method of mechanical classification of boards or beams as an intermediate product for the production of laminated wood boards or beams. The apparatus involves a planning device (102) in which they are planed and then a measuring device in which they are analysed and classified with regard to their strength and where applicable also optical criteria, where the classified boards or beams are then sorted mechanically by classification. In the production line at least two measuring devices (106, 108) are arranged in parallel and the boards or beams leaving the planning device (102) can be guided via a switch device (104) alternately to the at least two measuring devices (106, 108), where the transport speed with which the boards or beams pass through the measuring device (106, 108) is less than the transport speed with which they pass through the planning device (102).
Patent CZ-301733-B6 (CZ)
Title: Cubicle switchboard and frame arm for such cubicle switchboard
Inventor: SCHMITT OLIVER
IPC: H02B1/01
Filed: 2000-04-07
Abstract: In the present invention, there is disclosed a cubicle switchboard (10) comprising a framed cubicle (55) composed of individual vertical frame arms (11, ..., 14) and horizontal frame arms (15, ..., 18, 25, 30, ..., 32) of the same type and encompassing an interior (56) in the form of a rectangular. In said rectangular interior (56), there can be fastened between the vertical frame arms (11, ..., 14) pertaining to one longitudinal side or to one transversal side, rails, especially DIN-rails (20, 21, 22) for fastening electrical and/or electronic functional units (23). All the frame arms (11, ..., 14, 15, ..., 18, 25, 30, ..., 32) have rectangular cross section that us adapted to the depth of the rails, optionally DIN-rails (20, 21, 22). When installing the rails (20, 21, 22) onto the vertical frame arms (11, ..., 14), the rail (20, 21, 22) sides turned toward the cubicle switchboard (10) interior (56) lie in one plane with inwardly oriented surfaces of the vertical frame arms (11, ..., 14). There is also disclosed a frame arm (11, ..., 14, 15, ..., 18, 25, 30, ..., 32) used for the above-described cubicle switchboard (10).
Patent CZ-301355-B6 (CZ)
Title: I.S. machine
Inventor: FENTON FRANK ALAN
IPC: C03B/
Filed: 2000-10-27
Abstract: In the present invention, there is disclosed an I.S. machine, which has at least one section having a mold station wherein a glass forming operation is performed within a mold which includes an opposed pair of mold halves(56A, 56B, 56C). Each pair of mold halves (56A, 56B, 56C) has a different band diameter (D1, D2, D3) within a selected range, and a planar surface (71A, 71B, 71C), to be calmingly engaged with the planar surface (71A, 71B, 71C) of the other mold half (56A, 56B, 56C) at a mold centerline 90. The invented I.S. machine further comprises a pair of opposed mold holders for holding at least one opposed pair of mold halves (56A, 56B, 56C), the opposed mold holders being displaceable towards and away from the mold centerline (90), and drive assembly means for displacing said mold holders a predetermined distance from an open position to the mold closed position, the predetermined distance being a direct function of the dimension of the band diameter (D1, D2, D3) of the mold halves (56A, 56B, 56C) supported on the mold holders.
Patent CZ-297823-B6 (CZ)
Title: Stocking, sock or the like and process for producing thereof
Inventor: KALDE FRANZ-JOSEF
IPC: A41B11/04
Filed: 2000-08-11
Abstract: In the present invention, there is disclosed a stocking, a sock or a similar product, comprising a foot area (2), an upper (shin) part (3) connected to the foot area, a collar (4) that forms a single piece with the upper (shin) part (3) and is arranged opposite to the foot area (2), a retaining aid (5) performed on the inner side (6) of the collar (4), as well as several interspaced adhesive structures (7, 7a, 8, 12, 15, 19), which form said retaining aid (5). At least one adhesive structure (12) is formed by agglomeration of microstructures (14). There is also disclosed a process for producing such stocking or sock or the like article wherein the process is characterized by completely knitting the whole stocking, sock or the like article and subsequently forming adhesive structures (7, 7a, 8, 12, 15, 19).
Patent CZ-299065-B6 (CZ)
Title: Method for determining presence of antibody
Inventor: HAAHEIM LARS REINHARDT
IPC: G01N33/53
Filed: 2000-06-14
Abstract: The present invention relates to a method of determining the presence or amount of newly synthesized antibody in a sample of body liquid in response to an immunogen by detecting the released antibodies or parts thereof in a sample containing lymphocytes, which have been disrupted in order to release the synthesized antibodies or parts thereof associated with said lymphocytes in order to determine the presence or amount of newly synthesized antibody in said sample. The invented method may also be modified to allow detection of non-specific infection indicators.
Patent CZ-301982-B6 (CZ)
Title: Contraceptive composition containing estradiol or ester thereof and nomegestrol acetate
Inventor: PARIS JACQUES
IPC: A61K31/565
Filed: 2000-10-24
Abstract: In the present invention, there is described the use of a composition consisting of (i) 0.3 to 3 mg estradiol or ester thereof, (ii) 0.1 to 1.25 mg nomegestrol acetate and (iii) pharmaceutically acceptable excipients, for preparing a peroral contraceptive product in the form of daily dosage forms.
Patent CZ-303356-B6 (CZ)
Title: Substituted alkylamine derivative and pharmaceutical composition containing thereof
Inventor: CHEN GUOQING
IPC: A61K31/506
Filed: 2002-01-11
Abstract: In the present invention, there is disclosed a substituted alkylamine derivative of the general formula XI, in which R represents a unsubstituted pyridyl, Re1 denotes 2,3-dihydro-1H-indolyl substituted with one or two methyl groups, Re2 represents a hydrogen atom, Re4 denotes a straight bond and ReZ represents a methylenyl group, and pharmaceutically acceptable salts thereof. The derivative of the present invention can be used for treatment of cancer, neoplasia, cell proliferation and angiogenesis.
Patent CZ-295558-B6 (CZ)
Title: 5-Halogen-6-phenyl-7-fluoroalkylamino-triazolopyrimidines, process of their preparation and composition for controlling phytopathogenic fungi
Inventor: TORMO I BLASCO JORDI
IPC: A01N43/90
Filed: 2002-04-06
Abstract: In the present invention, there are disclosed 5-halogen-6-phenyl-7-fluoroalkylamino-triazolopyrimidines of the general formula I in which Re1 represents a hydrogen atom, a fluorine atom, an alkyl group, an alkenyl group, an alkynyl group, an alkadienyl group, where the carbon chains of these radicals may be unsubstituted or substituted; Re2 represents  a hydrogen atom, an alkyl group,  an alkenyl group, an alkynyl group, an alkadienyl group, where these radicals may be unsubstituted or substituted; Re3 denotes a fluoroalkyl group or  a fluoroalkenyl group; X represents a halogen atom; n is 0 or an integer from 1 to 4; L each independently represents a halogen atom, a nitro group, an alkyl group, a haloalkyl group, an alkoxy group or a haloalkoxy group. Disclosed are also processes for their preparation, compositions containing them and their use for controlling phytopathogenic fungi.
Patent SK-285528-B6 (SK)
Title: Method for producing base or salt of citalopram
Inventor: PETERSEN HANS
IPC: C07D307/00
Filed: 2001-02-28
Abstract: In method for production salts of citalopram is the base of citalopram isolated and precipitated in crystalline form, further can be re-crystallised one or more times and then is converted into its salt.
Patent SK-288915-B6 (SK)
Title: Biopreparation from Exiguobacterium undae, method of production and use thereof
Inventor: PANGALLO DOMENICO
IPC: C12N9/52
Filed: 2018-03-06
Abstract: The biopreparation from Exiguobacterium undae contains two major extracellular proteins: extracellular metalloendopeptidase – bacillolysin with a molecular weight of 33 kDa at a concentration of 0.01 to 0.05 mg/ml and peptide binding protein for ABC transporter with a molecular weight of 61 kDa at a concentration of 0.01 to 0,05 mg/ml and other proteolytic enzymes, peptidase M6 with a molecular weight of 86.7 kDa, 4-phytase with a molecular weight of 58.4 kDa, endonuclease with a molecular weight of 59.9 kDa, menaquinol-cytochrome C reductase with a molecular weight of 18,7 kDa, bifunctional metallophosphatase/5-nucleotidase with a molecular weight of 76.2 kDa, a peptidase with a molecular weight of 27.4 kDa as well as two other isoforms of the peptide binding protein for the ABC transporter with a molecular weight of 61 kDa. The biopreparation has good degrading effects on animal glue and animal glue adhesives and is suitable, for example, for use in the restoration work of wooden organ pipes.
Patent BR-PI0209362-B8 (BR)
Inventor: PRESTON JANINE ANDREA
IPC: C08L57/00
Filed: 2002-04-19
Abstract: Polymeric particles comprising a polymeric matrix and colourant distributed throughout the matrix, wherein the polymeric matrix that has been formed from a blend of monomers comprising a first monomer which is an ethylenically unsaturated ionic monomer and a second monomer which is an ethylenically unsaturated hydrophobic monomer which is capable of forming a homopolymer of glass transition temperature in excess of 50° C., and in which the first monomer is a salt of a volatile counterion component, characterized in that the polymeric matrix is impermeable to the colourant The particles obtainable by the process of the invention can be used in a variety of industrial processes, for instance in the manufacture of inks, paper and cosmetics.
Patent BR-PI0313082-B8 (BR)
Inventor: ALESSANDRO ANELLI
IPC: A61K31/715
Filed: 2003-06-30
Abstract: An Echinacea angustifolia extract and a process for the preparation thereof are herein described. The extract is characterized by an alkylamides content lower than 0.1%, an echinacoside content ranging from 1 to 10% and containing from 1 to 15% of a polysaccharide characteristic of Echinacea angustifolia. The extract can be used for the treatment of pathological conditions in which it is desirable to strengthen the immune defenses.
Patent EP-1867932-B8 (EP)
Inventor: BAGWELL RICK A
IPC: F24F1/0067
Filed: 2006-01-06
Granted: 2011-03-30
Abstract: Displacement ventilation systems are generally poor performers when it comes to heating. The instant patent application discusses devices and systems for improving heating performance while retaining the benefits of displacement ventilation without wholesale co-location of independent space conditioning systems.
Patent EP-2478893-B8 (EP)
Inventor: STINCHCOMB AUDRA LYNN
IPC: A61K9/00
Filed: 2008-12-01
Granted: 2013-10-09
Abstract: Described herein is a method of transdermally administering one or more pharmaceutically active agents to a mammal The method comprises administering one or more active pharmaceutical agents to the skm of the subject, in conjunction with microneedles and one or more COX inhibitors, whereby the COX inhibitors facilitate the absorption of the active pharmaceutical agents by prolonging the pore opening created by the application of the microneedle
Patent BR-PI0414254-B8 (BR)
Title: composição farmacêutica compreendendo hcl de cinacalceto
Inventor: FRANCISCO J ALVAREZ
IPC: A61K9/20
Filed: 2004-09-10
Abstract: composição farmacêutica, e, métodos para fabricar uma composição farmacêutica, para o tratamento de pelo menos uma doença e para controlar a taxa de dissolução de uma formulação a presente invenção diz respeito a uma composição farmacêutica que compreende uma quantidade terapeuticamente eficaz de um composto ativo receptor de cálcio e pelo menos um excipiente farmaceuticamente aceitável, em que a composição tem um perfil de dissolução controlado. a presente invenção ainda diz respeito a um método para fabricar a composição farmacêutica, bem como um método de tratar uma doença usando a composição farmacêutica.
Patent BR-PI0518269-B8 (BR)
Inventor: WALTER SARSTEDT
IPC: A61M5/34
Filed: 2005-10-21
Abstract: A specimen tube for receiving bodily fluids, particularly blood, has a sealing cap having a tip with a pierceable membrane, stopper or similar device, at its end. A guide sleeve can be placed on the tip and carries a single or double needle. The tube can also be provided with an emergency indicator that is configured as an emergency signal colored ring surrounding the tip but leaving free access from outside to the pierceable element at the end of the tip.