baber/WOPTO huggingface dataset:
Patent MA-24349-A1 (MA)
IPC: C07D401/14
Filed: 1997-07-07
Abstract: A compound of formula (I): or a salt thereof, or a solvate thereof, wherein Ra represents a group R<SUB>5 </SUB>which is hydrogen, alkyl or optionally substituted aryl and Rb represents a moiety of formula (a): wherein X represents a hydroxy or an alkoxy group wherein the alkyl group may be substitued or unsubstituted or X represents a group NR<SUB>s</SUB>R<SUB>t </SUB>wherein R<SUB>s </SUB>and R<SUB>t </SUB>each independently represent hydrogen, alkyl, substituted alkyl, optionally substituted alkenyl, optionally substituted aryl, optionally substituted arylalkyl, an optionally substituted heterocyclic group or an optionally substituted heterocyclylalkyl group, or R<SUB>s </SUB>and R<SUB>t </SUB>together with the nitrogen to which they are attached form a heterocyclic group; R<SUB>1 </SUB>represents an alkyl or a substituted or unsubstituted aryl group; and R<SUB>2</SUB>, R<SUB>3 </SUB>and R<SUB>4 </SUB>each independently represent hydrogen, alkyl, aryl or substituted aryl; R<SUB>6 </SUB>and R<SUB>7 </SUB>each independently represent hydrogen, hydroxy, amino, alkoxy, optionally substituted aryloxy, optionally substituted benzyloxy, alkylamino, dialkylamino, halo, trifluoromethyl, trifluoromethoxy, nitro, alkyl, carboxy, carbalkoxy, carbamoyl, alkylcarbamoyl, or R<SUB>6 </SUB>and R<SUB>7 </SUB>together represent methylenedioxy, carbonyldioxy or carbonyldiamino; and R<SUB>8 </SUB>represents hydrogen, hydroxy, alkynoyl, alkyl, aminoalkyl, hydroxyalkyl, carboxyalky, carbalkoxyalkyl, carbamoyl or aminosulphonyl; a process for preparing such a compound, a pharmaceutical composition containing such a compound and the use of such a compound in medicine.
Patent MA-27662-A1 (MA)
Inventor: BESSE JEROME
IPC: A61K45/06
Filed: 2005-08-26
Abstract: A method for the manufacture of a pharmaceutical composition containing the active ingredient fenofibrate or one of its derivatives, optionally in combination with a second active ingredient, in the form of tablets, characterized in that it comprises a compression step of the active ingredient and excipients by means of a dry method of granulation
Patent MA-54776-A1 (MA)
Title: Méthode de déploiement d’une nouvelle politique de sécurité de pare-feu dans un réseau informatique.
Inventor: KARTIT ALI
IPC: G06F17/00
Filed: 2021-10-29
Abstract: La présente invention concerne une méthode de déploiement de nouvelle politique de sécurité de pare-feu pour des réseaux informatique et afin palier aux différents risques d’une politique courante. Il s’agit d’une démarche de mise à jour d’une politique de sécurité initiale (i) basée sur un algorithme qui automatise cette démarche et minimise les risques de sécurité inhérents au moment de déploiement d’une nouvelle politique de sécurité (t). Ceci par la création d’une politique intermédiaire (r) qui reçoit progressivement les nouvelles règles de (t) à implémenter et selon un ordre bien précis. La démarche de déploiement selon l’invention s’achève lorsque la politique (r) est égale la politique cible (t).
Patent UY-26308-A1 (UY)
Title: Nuevas indolinonas sustituidas, su preparación y su empleo como medicamentos
Inventor: WALTER DR GERALD JURGEN ROTH D
IPC: C07D401/12
Filed: 2000-08-23
Abstract: La presente invención se refiere a indolinonas sustituidas de la fórmula general (i), en la que r1 a r6 y x están definidos como en la reivindicación 1, a sus isómeros y sus sales, en particular sus sales fisiológicamente compatibles, que presentan valiosas propiedades farmacológicas, en particular un efecto inhibidor sobre diferentes tirosinquinasas de receptor y complejos de ciclina/cdk, así como sobre la proliferación de células endoteliales y diferentes células tumorales, a medicamentos que contienen estos compuestos, a su empleo y a procedimientos para su preparación.
Patent UY-29949-A1 (UY)
Title: Composición farmacéutica con edulcorante de alta intensidad
Inventor: DUBOIS GRANT E
IPC: A23L27/30
Filed: 2006-11-21
Abstract: Composiciones farmacéuticas que comprenden edulcorantes no calóricos o hipocalóricos de alta potencia y los métodos para hacerlos y usarlos. En particular, la invención refiere a diferentes composiciones farmacéuticas que comprenden al menos un edulcorante natural y/o sintético no calórico o hipocalórico de alta potencia, al menos una composición para mejorar el sabor dulce y al menos una sustancia activa farmacéuticamente.
Patent UY-30716-A1 (UY)
Title: Combinaciones de herbicidas con sulfonilureas especiales.
Inventor: MARCELES VICTOR
IPC: A01N43/40
Filed: 2007-11-13
Abstract: Se divulgan combinaciones de herbicidas que contienen uno o varios herbicidas tomados del conjunto formado por las sulfonilureas de la formula (I) y sus sales con uno o varios herbicidas tomados del conjunto formado por los compuestos de la formula (II) y sus sales ésteres, en la que los sustituyentes quedan descriptos en la Memoria y en las Reivindicaciones.
Patent ES-162888-A1 (ES)
Title: PROCEDIMIENTO PARA PRODUCIR UNA CINTA SIN FIN CON INSCRIPCIoN SONORA EXPLORABLE MECANICAMENTE
Filed: 1943-08-27
Abstract: Procedimiento de producir cintas sin fin con varias huellas sonoras explorables mecánicamente y de curso paralelo o casi paralelo al canto de la cinta por moldeado de una matriz limitada producida de una cinta sonora original sin fin (cinta encerada etc); caracterizado porque la cinta sonora original o la cinta de matriz se proveen a ambos lados de la línea de separación que se ha de trazar transversalmente a la cinta de marcas por medio de una plantilla siendo estas marcas moldeadas también al hacer la multiplicación de las cintas y poniéndose las marcas moldeadas de la cinta multiplicada mediante la plantilla de nuevo en la posición recíproca que asegura el ajuste reglamentario de las huellas sonoras del haz de las mismas en los dos extremos de la cinta.
Patent ES-170776-A1 (ES)
Title: Un aparato manual para producir hielo
Filed: 1945-08-20
Abstract: Aparato manual para la producción de hielo mediante la caida de temperatura determinada por la ebullición del agua sin aportación de calor por el enrarecimiento del aire en el recipiente que la contiene caracterizado porque se disponen conectados en serie una bomba aspirante un recipiente con una sustancia ávida de agua ácido sulfúrico de 66º Bé por ejemplo y un recipiente parcialmente lleno de agua con lo que al ser accionada la bomba se produce en el recipiente de agua un enrarecimiento que determina la ebullición del líquido con el consiguiente descenso de la temperatura colaborando la absorción del vapor de agua por el ácido sulfúrico a la rápida vaporización del agua que determina a voluntad su simple enfriamiento o su congelación.
Patent ES-181914-A1 (ES)
Title: Mejoras en juntas herméticas y forma de efectuarlas
Filed: 1948-01-29
Abstract: Mejoras en juntas herméticas y forma de efectuarlas mediante un método de cerrar o sellar una junta que consta de un plaste humedecido que tiene por lo menos sus superficies formadas por un material soluble con un disolvente par dicho material y aun cuando el material de tales superficies está todavía húmedo, con el disolvente empleado, se llevan las superficies de las partes de la junta a hacer contacto.
Patent ES-183350-A1 (ES)
Title: Un motor eléctrico
IPC: H02P25/12
Filed: 1948-04-20
Abstract: Un motor eléctrico que comprende un armazón, devanados de campo estacionarios, un inducido montado en el armazón y que tiene un colector, escobillas que cooperan con el colector, y un interruptor de inversión para cambiar las conexiones eléctricas a alas escobillas, caracterizado porque el funcionamiento del interruptor cambia la posición de las escobillas con respecto a los devanados de campo.
Patent ES-186985-A1 (ES)
Title: Un dispositivo electromagn''etico
Filed: 1949-02-10
Abstract: Un dispositivo electromagnético por ejemplo una bobina de auto-inducción en el cual un campo magnético alterno es desarrollado en un medio ferro-magnético-alterno caracterizado por medios debido a los cuales el medio ferro-magnético que con preferencia está hecho de ferrita muy permeable esencialmente no conductora es influído por un campo magnético polarizador permanente o semipermanente en una dirección en ángulo recto con un componente del campo magnético alterno siendo tal la intensidad del campo magnético de polarización que la frecuencia de precisión correspondiente de los electrones a los cuales son debidas las propiedades magnéticas y que rodean el vector del campo de polarización coincide virtualmente con la frecuencia del campo magnético alterno.
Patent ES-187818-A1 (ES)
Title: PERFECCIONAMIENTOS EN LAS INSTALACIONES MOTRICES PARA NAViOS, QUE COMPRENDEN GRUPOS DE TURBINAS ALIMENTADAS CON VAPOR RECALENTADO
Filed: 1949-04-16
Abstract: Perfeccionamiento en las instalaciones motriIces para navíos que comprenden grupos de turbinas alimentadas con vapor recalentado caracterizado por la.disposición en el circuito de alimentación de las turbinas de un recalentador en que se hace pasar todo o una parte del vapor recalentado.que vá a las turbinas.
Patent ES-191174-A1 (ES)
Title: PROCEDIMIENTO Y DISPOSITIVOS PARA LA FABRICACIoN DE PIEZAS DE HORMIGoN ARMADO CON ACABADO ESPECIAL
Filed: 1950-01-11
Abstract: Procedimiento y dispositivos para la fabricación de piezas de hormigón armado con acabado especial caracterizado porque en una primera fase se obtienen las piezas moldeadas y vibradas mediante moldes constituidos por laterales que se unen entre sí por tornillos de apriete y fijación que pasan por taladros dispuestos al efecto en aquellos interponiendo entre esos laterales topes que limitan el tamaño de las piezas aumentando la posible altura de estas si procede por regletas o listones colocados sobre tales laterales de modo que por la combinación de tales elementos se consigan piezas de las dimensiones y perfiles que se deseen armadas de modo conveniente.
Patent ES-195152-A1 (ES)
Title: UN DISPOSITIVO PARA SUBIR Y BAJAR EL BANCO DE HUSOS O ANILLOS DE MáQUINAS HILADORAS O RETORCEDORAS DE ANILLOS
Filed: 1950-10-28
Abstract: Dispositivo para subir y bajar el banco de husos o de anillos de las máquinas hiladoras o retorcedoras de anillos compuesto de un par de roscas caracterizado porque la marca roscada (2) va montada en una corredera elevadora. (5) y las dos partes van guiadas en al árbol roscado (1) con independencia una. de otra.
Patent ES-275516-A1 (ES)
Title: Meat tendering compositions
IPC: A23L13/70
Filed: 1962-03-15
Abstract: A bacteria-free enzyme composition suitable for use in the ante-mortem treatment of meat-bearing animals comprises a proteolytic enzyme in aqueous solution, the solution having an activity of 250-14,000 tyrosyl units per milliliter, a ratio of tyrosyl units to milk-clotting units of 55-100 and a ratio of tyrosyl units to available milk-clotting units of more than 200. Preferred enzymes are plant-derived enzymes such as papain, ficin and bromelin. The Specification describes methods of determining milk clotting and tyrosyl values. Specifications 913,202 and 913,203 are referred to.ALSO:In the procedure of Specification 913,202, which relates to tenderizing meat by treating living animals with proteolytic enzymes prior to slaughter, there is utilised a bacteria-free composition comprising a proteolytic enzyme in aqueous solution, the solution having an activity of 250-14,000 tyrosyl units per millilitre, a ratio of tyrosyl units to milk-clotting units of 55-100 and a ratio of tyrosyl units to available milk-clotting units of more than 200. Preferred enzymes are plant-derived enzymes such as papain, ficin and bromelin. The Specification describes methods of determining milk-clotting and tyrosyl values. Specification 913,203 also is referred to.
Patent ES-296966-A1 (ES)
Title: Improvements in welding jaws for heat sealing sheets of plastics material
IPC: B29C65/18
Filed: 1964-02-27
Abstract: Apparatus for welding synthetic plastic sheets 14 comprises a pair of jaws 1, 2 of which the surface 3 of the jaw 1 is bare and the surface 4 of the jaw 2 is covered with a sheet 5 of elastomer freely positioned and held on the jaw 2 so as not to be subjected to lateral or longitudinal strain when compressed by the closing of the jaws, and a projection of small thickness with respect to that of the weld to be produced formed on the face 4 and extending along a line which will be the longitudinal axis of the weld, the faces of the jaws 1, 2 to be applied to the sheets 14 being, other than at the position of the projection, strictly flat so as to be applied exactly one against the other. The entire periphery of the sheet 5 has reduced thickness edges 6 located with both horizontal and vertical play in a frame formed by angle irons 7 secured to the jaw 2. In one embodiment, Fig. 1, a longitudinal groove 8 is formed in the face 4 and receives a replaceable bar 9 providing the projection. In a second embodiment, Fig. 2, the jaw 2 is provided with a slot 8a opening into a wider slot 10 closed at the lower end by a liner 11. The projection is formed by an extension 9a of a bar 12 sliding vertically in the slot 10. The amount of projection of the extension 9a above the face 4 may be adjusted by two screws 13 engaging threads in the liner 11.
Patent ES-341600-A1 (ES)
Title: Improvements relating to Refrigerating Systems
IPC: F25B31/00
Filed: 1967-06-09
Abstract: Refrigerant from the compressor 8 of a hermetically encapsulated motor-compressor unit passes sequentially through a heat exchanger 16 and a jacket 12 surrounding the compressor cylinder to cool the latter before being condensed in the condenser 19.
Patent ES-345601-A1 (ES)
Title: Methods of Coating Semiconductive Materials with Conductive Metals.
IPC: H01L21/306
Filed: 1967-09-19
Abstract: A method of forming metallic contacts on semi-conductor bodies by electroless plating may be applied to silicon double diffused diodes. Doped silicon slices are provided on their opposite faces with organic solutions of boron trioxide and phosphorus pentoxide and heated to form diffused regions. Hydrofluoric acid etching is effected through when sufficient to remove the borosilicate glass formed by the diffusion process (the less resistant phosphosilicate glass is also removed) it deactivates the silicon surface for electroless plating. The slices are therefore next dipped in hot aqueous ammonia to activate their surfaces and (after an optional hydrofluoric acid etch to remove any thin oxide formed in this process) are dipped in any standard electroless coating solution, such as a bath containing nickelous chloride and sodium hypochlorite. The slices are diced and are provided with leads and housings or mountings.
Patent ES-348819-A1 (ES)
Title: Aqueous waste disposal in process for preparation of isoprene from isobutylene
IPC: C07C1/247
Filed: 1967-12-30
Abstract: In the production of isoprene by (1) reacting isobutene with aqueous formaldehyde in the presence of a catalyst to form 4,4-dimethyl-mdioxane, and (2) decomposing the thus-formed 4,4 - dimethyl - m - dioxane, the by-products less volatile than water which are produced in step (1) and are dissolved in the aqueous phase are concentrated, e.g. by evaporation, and are then catalytically decomposed to yield further isoprene. Readily volatile or extractable substances may be removed from the aqueous phase before concentration, e.g. by distillation or extraction with the isobutene feed to step (1). The preferred decomposition catalyst is phosphoric acid on silicic acid particles used as a fluidized bed.
Patent ES-351074-A1 (ES)
Title: Carboxylic acid ester substituted polyhydantions
IPC: C08G18/38
Filed: 1968-02-29
Abstract: Amino succinic acid derivatives are prepared by reacting a diester of an ethylene-1,2-dicarboxylic acid with a primary polyamine containing 2 to 4 amino groups. In specific examples, such derivatives are prepared from (1) dimethyl maleate and 4,41-diaminodiphenylmethane, (2) hexamethylene diamine and dimethyl maleate, (4 and 7) hexahydro-pphenylene diamine and dimethyl maleate, (8) aniline, m-phenylene diamine and dimethyl maleate. The amino succinic acid derivatives may be reacted with polyisocyanates to form a polyurea which may be subsequently or simultaneously subjected to a ring closure reaction to form polymeric polycarboxylic acid esters containing hydantoin rings.
Patent ES-355580-A1 (ES)
Title: Manufacture of lubricating oil with the use of new catalysts
IPC: B01J23/85
Filed: 1968-06-28
Abstract: Cracking catalysts are made by incorporating as active ingredient into a carrier, a free metal or an oxide or sulphide of the metal selected from Groups VIA and VIII of the MendelÚef Periodic Table, or mixtures of these metals and metal compounds, the carrier being prepared by suspending a silica or alumina gel in an aqueous phase at a pH value of between 7.5 and 11 so as to obtain particles in the range of from 0.1 to 10Á, introducing an aluminium or silicon compound into the suspension to precipitate an alumina or silica gel onto the already present particles of SiO 2 , or Al 2 O 3 gel thereby coating the latter so as to produce particles of a mixed gel. Preferably the SiO 2 -Al 2 O 3 supports 2-10% of Co or Ni and 10-30% of Mo or W, expressed as oxides. The catalysts may be presulphided before use.
Patent ES-355697-A1 (ES)
Title: Continuous production of articles from a roll of thermoplastic material
IPC: B29C51/44
Filed: 1968-06-25
Abstract: In a sheet forming apparatus of the type in which a continuous sheet is intermittently fed by pairs of edge engaging belts through heating and forming stations, the formed articles are separated from the rest of the sheet at a blanking station located beyond the belts. The distance between the forming and blanking stations is such that the sheet cools to a sufficient extent to avoid warping during the blanking and successive articles are separated by transverse channels which channels provide narrow zones in which deformation can occur during the movement of the sheet from the forming to the blanking station. In the described embodiment, a sheet 32 drawn from a roll supported upon a moving belt 40 is first heated at station 33 and then formed into pairs of side-by-side egg cartons between cooled matched moulds at station 34. The heater side of each mould is provided with a cooled heat shield, the edges of the shields co-operating during each mould closure to form a transverse distortable channel which separates successive pairs of cartons. The cartons are then forwarded under a printer 36 and move from chains 45 and 46 along guides to clamping and blanking stations 37, 38. At these stations one pair of articles is clamped and perforated whilst the preceding pair perforated in the preceding operation is stripped from the sheet by suitable shaped co-operable cutting dies. The perforation is effected by the apparatus shown in Fig. 15. The cover portion of each pair of containers is gripped between members 155 and 162 and is perforated by an hydraulically actuated punch 167 passing through cooperating sleeved holes 164 located in the members.
Patent ES-355971-A1 (ES)
Title: Amino alkyl esters of 5beta-pregn-20-ene-21-carboxylic acids and the 3-glycosides thereof
IPC: A61K31/573
Filed: 1968-07-10
Abstract: Pharmaceutical compositions comprise one or more steroids of formula wherein R1 and R2 are each alkyl or are joined together with the intervening nitrogen atom to form a heterocyclic ring, A is alkylene, R3 is hydrogen and R4 is hydroxy, acyloxy, glycosyloxy or acylated glycosyloxy, or R3 and R4 together with the intervening carbon atom form the carbonyl group, and wherein the steroid nucleus from carbon atoms 1-19 optionally bears one or more additional substituents selected from oxo, hydroxy, acyloxy and alkylenedioxy radicals, and wherein said nucleus optionally contains one or more olefinic double bonds, or a salt thereof with an organic or inorganic acid. These compounds possess digitalis-like activity, and the compositions may be administered orally or parenterally. The compositions may additionally include #- adrenergic blocking agents (e.g. propanolol), other cardiotonic agents (e.g. digoxin, digitalis preparations, digitoxin, laratoside C), diuretics (e.g. frusemide, ethacrymic acid), thiazide diuretics (e.g. hydrochlorothiazide, bendrofluazide), aldosterone antagonists (e.g. spironolactone), coronary vasodilators (e.g. glyceryl trinitrate, pentaerythritol tetranitrate, sorbide nitrate), .xanthine derivatives (e.g. theophylline, theobromine, aminophylline), dipyridamole, and potassium salts (e.g. potassium chloride, potassium gluconate).
Patent ES-363119-A1 (ES)
Title: Figure toy having apparatus for moving eyes in simulated reading motion
IPC: A63H3/40
Filed: 1969-01-30
Abstract: A figure toy has movable eyes with eye moving means for moving the eyes at a first rate in one direction and at a second slower rate in the reverse direction so that the eyes move through simulated reading patterns. Additionally, the toy is provided with movable arms and a sound producing device, the two being attached, so that when the arms are moved to a first position the sound producing device produces a first character of sound corresponding to non-reading sounds, and when the arms are moved to a second position the sound producing device produces a second character of sound corresponding to reading sounds. The eye drive structure is shown in Fig. 9 wherein the eyeballs 20 and 22 are mounted in transparent bubbles 24 and 26 which in turn are mounted in eye sockets 28 and 30 within head 12 of the toy. Cross link 36 is a unitary structure with pins 38 and 40 which engage on the back of the eyeballs. Thin sections 42 and 44 act as hinges to permit relative bending movement of the link with respect to the eyeball. Guide bar 46 is positioned under link 36 and a similar guide bar can be placed over it and so the eyeballs will rotate upon their own vertical axis. The eye moving mechanism is operated by means of a pulley 54 carried on a worm shaft 48 (not shown) which also carries worm 58 which is in gear tooth engagement with gear 60 (Fig. 9). Gear 60 is pivoted on pin 62, which is secured inside the head 12, and engages gear 64, which carries crank pin 68 extending forward from its face. Yoke 70 is pivoted on pivot 72 and has a slot 74 which engages upon crank pin 68. Connector pin 76 extends forward from the yoke adjacent to pivot 72 and engages in cross link 36. As the pulley is rotated, gear 64 rotates in a clockwise direction. This causes angular oscillating motion of link 70 about its pivot pin 72 with yoke 70 moving more slowly while crank pin 68 is farther away from pin 72 and returning relatively fast in anti-clockwise direction as pin 68 is close to pin 72. This causes the eyes to sweep slowly in the reading direction and return rapidly in the opposite direction.