baber/WOPTO huggingface dataset:
Patent IL-45340-A (IL)
Title: 3,4-dihydro-1-benzoxepin-5-one amino-alkyloxime derivatives their preparation and pharmaceutical compositions containing them
IPC: C07D313/08
Filed: 1974-07-24
Abstract: 1449406 Amine ethers of 3,4-dihydro-1- benzoxepin-5-one oximes CERPHA 31 July 1974 [31 July 1973 22 May 1974] 33750/74 Heading C2C Novel compounds are the free amines of Formula I and their acid addition salts wherein R is halogen or C 1-4 alkoxy, n is 2 or 3 and Z 1 and Z 2 , which may be the same or different, are C 1-4 alkyl or Z 1 and Z 2 together with the common nitrogen atom form a 5 to 7 membered ring optionally containing a second hetero atom, the compounds having either the cis or trans configuration relative to the benzene nucleus. The compounds of Formula I are obtained by effecting intramolecular acylation on a γ- phenoxybutyric acid which is R-substituted in the para-position to produce a compound of Formula II reacting the latter with a compound of formula H 2 N-O-A, in which A is H or the group -(CH 2 )n-NZ 1 Z 2 , the reaction when A is -(CH 2 ) n -NZ 1 Z 2 being carried out in an alcoholic solvent in an acid medium and at the reflux temperature of the solvent and when A is H being effected in pyridine or ethanol; and reacting the resulting intermediate, obtained when A is H, with a compound of formula X-(CH 2 ) n -NZ 1 Z 2 , in which X is halogen, in the presence of a base. The products of this preparation are at least 95% in the cis configuration and the cis isomer may be isolated by recrystallization of a cis/trans mixture of acid addition salts of the free amine. The trans isomer may be isolated similarly by fractional crystallization following partial isomerization in an anhydrous acid medium (e.g. HCl/ChCl 3 ) after the introduction of the oxime function. Examples describe the preparation of compounds of Formula I and intermediate ketones and oximes wherein R is Cl, Br, or CH 3 O and Z 1 and Z 2 are each CH 3 or C 2 H 5 or -NZ 1 Z 2 represents a morpholino or pyrrolidino group. Salts prepared are those with HCl, oxalic and fumaric acids. The compounds of Formula I and their pharmaceutically acceptable acid addition salts are used in therapeutic applications as muscle relaxants.
[GB1449406A]
Patent IL-92407-A (IL)
Title: Bis-arylphosphate ester antagonists of platelet activating factor and their preparation
IPC: C07F9/62
Filed: 1989-11-23
Abstract: The invention is novel compounds of the formula: <CHEM> which are antagonists of platelet activating factor.
[EP0374513A2]
Patent IL-94652-A (IL)
Title: Carboplatin composition
IPC: A61K9/00
Filed: 1990-06-06
Abstract: A carboplatin composition is provided in the form of an aqueous solution of carboplatin buffered at a pH of 2-6.5. Such a ready to use solution possesses a remarkable stability.
Patent IL-95121-A (IL)
Title: N-n'bis (alkoxyalkyl)-pyridine-2,4-dicarboxylic acid diamides, process for their preparation and pharmaceutical compositions containing them
IPC: A61K31/455
Filed: 1990-07-18
Abstract: N,N'-bis(alkoxyalkyl)pyridine-2,4-dicarboxylic acid diamides of the formula I <IMAGE>  where     R<1> is linear or branched C1-C4-alkanediyl,   R<2> is unbranched C1-C4-alkyl or hydrogen and   n is 1 or 2 and R<1'>, R<2'> and n' have the same meanings as R<1>, R<2> and n, where R<1> and R<1'>, R<2> and R<2'>, and n and n' are identical or different, and their physiologically acceptable salts with the exception of N,N'-bis(2-methoxyethyl)pyridine-2,4-dicarboxylic acid diamide and N,N'-bis(2-hydroxyethyl)pyridine-2,4-dicarboxylic acid diamide. The compounds of the formula I inhibit prolin hydroxylase and lysin hydroxylase and are suitable as fibrosuppressants and immunosuppressants.
Patent IL-97028-A (IL)
Title: Propellant gas mixtures and pharmaceutical compositions containing them
IPC: A61K9/72
Filed: 1991-01-24
Abstract: Novel advantageous vehicle gas mixtures contain two or more components, at least one of which is a partly fluorinated lower alkane, and may be used in medical preparations.
[DE4003272A1]
Patent IL-99167-A (IL)
Title: Carbamoyl-1-(pyridinylalkyl)-1h-indoles indoles and related analogs process for their preparation and pharmaceutical compositions containing them
IPC: A61K31/47
Filed: 1991-08-12
Abstract: This invention relates to compounds of the formula <CHEM>  where   R1   is hydrogen, loweralkyl, arylloweralkyl, loweralkenyl or loweralkynyl; R2   is hydrogen, loweralkyl, loweralkenyl, formyl or cyano; R3   is hydrogen or loweralkyl; R4   is loweralkyl, arylloweralkyl, cycloalkyl, aryl, heteroaryl, heteroarylloweralkyl, <CHEM>  or NR3R4 taken together constitute <CHEM>   R5   is hydrogen, loweralkyl or aryl; R6   is hydrogen, loweralkyl, aryl, arylloweralkyl, formyl, loweralkanoyl or arylloweralkanoyl, X and Y   are independently hydrogen, nitro, amino, halogen, loweralkyl, loweralkoxy or hydroxy; or the pharmaceutically acceptable acid addition salts thereof, and where applicable, the geometric and optical isomers and racemic mixtures thereof.   The compounds of this invention are useful for the treatment of various memory dysfunctions characterized by a decreased cholinergic function, such as Alzheimer's disease.
Patent IL-99598-A (IL)
Title: INTERLEUKIN-1beta PROTEASE INHIBITORS AND PHARMACEUTICAL COMPOSITIONS THEREOF
IPC: C07K5/065
Filed: 1991-09-27
Abstract: There is disclosed an isolated polypeptide and derivatives thereof having protease biological activity for human precursor IL-1 beta  and for a substrate comprising : R1-Asp-R2-R3 wherein R1 and R3 are independently any D or L isomer amino acid, R2 is Ala or Gly, and wherein the specific protease cleavage site is between Asp and R2. Inhibitor compounds, compositions and methods for inhibiting Interleukin 1 beta  protease activity are also disclosed. The inhibitor compounds comprise an amino acid sequence of from 1 to about 5 amino acids having an N-terminal blocking group and a C-terminal Asp residue connected to an electronegative leaving group, wherein the amino acid sequence corresponds to the sequence Ala-Tyr-Val-His-Asp.
Patent JP-S61170002-A (JP)
Title: Manufacture of anisotropic resin binding type magnet
Inventor: YAMASHITA FUMITOSHI
IPC: H01F1/032
Filed: 1985-01-23
Abstract: PURPOSE:To specify a minimum melt viscosity of ferromagnetic powder of a high magnetic anisotropic constant, and to fill a large quantity of the ferromagnetic powder and to stabilize magnetic characteristics by injection-molding a compound magnetic material with a thermal polymerizational resin compound in a magnetic field. CONSTITUTION:After a compound magnetic material of both a ferromagnetic powder of a high magnetic anisotropic constant and 0.5-100 poise of a minimum viscosity of a thermal polymerizational compound is injection-molded in a magnetic field in a comparatively low temperature, an anisotropic resin bonding type magnet is obtained. When a minimum melt viscosity is at most 0.5 poise, in using a ferromagnetic powder and a compound magnetic material by an extruding process, or in inject-moding this in the magnetic field, a shear rate grade is generated on walls of each portion of a die and devices like that, and a shearing flow is easily made. While on the other hand, when a minimum melt viscosity is over 100 poise, it becomes difficult to fill the ferromagnetic powder in great quantity and to heighten an orientational rate of the ferromagnetic powder in inject-molding in the magnetic field.
Patent JP-S60154455-A (JP)
Inventor: INADA AKIISA
IPC: H01K1/38
Filed: 1984-01-25
Abstract: (57)【要約】本公報は電子出願前の出願データであるた め要約のデータは記録されません。
Patent JP-S54102213-A (JP)
Title: Manufacture of al-mg-si type corrosion resistant, free cutting aluminum alloy pipe or rod with little residual stress
Inventor: MIZOGUCHI MASAO
IPC: C22F1/04
Filed: 1978-01-31
Abstract: PURPOSE: To manufacture an Al alloy pipe or rod with little residual stress by hardening an Al-Mg-Si type corrosion resistant, free cutting alloy, followed by stretch leveling, drawing, roll leveling and tempering under specific conditions.  
     CONSTITUTION: An Al-Mg-Si type corrosion resistant, free cutting alloy is hardened and stretch leveled at a stretch ratio of 1.0W3.0% to relieve the residual stress, and cold drawn at a working ratio of 10W30% to enhance the dimensional accuracy such as roundness. The drawn alloy is then roll leveled and held at 210W250°C for 1W2 hr to be tempered to relieve the residual strees formed by the cold working and roll leveling. By this method an Al-Mg-Si type corrosion resistant, free cutting Al alloy pipe or rod with little residual stress is obtd. without lowering the strength, and it is used for parts of optical instruments, etc. 
     COPYRIGHT: (C)1979,JPO&Japio
Patent JP-H05198576-A (JP)
Title: Manufacture of semiconductor device
Inventor: WATANABE KUNIO
IPC: H01L21/3205
Filed: 1992-01-23
Abstract: PURPOSE:To stably form high melting point metallic silicide having a small sheet resistance on polycrystalline silicon by a method wherein the polycrystalline silicon containing no impurities on the polycrystalline silicon containing impurities having a high density to form the high melting point metallic silicide by using it. CONSTITUTION:On a semiconductor substrate 1 forming an element separating silicon oxide film 2, a polycrystalline silicon film 3 is formed to ion-implant impurities such as arsenic or the like onto the entire plane. Next, a polycrystalline silicon layer 4 added no impurities thereto is formed thereon. Next, the polycrystalline silicon layers 3, 4 are patterned with photoresist 5 to remove the polycrystalline silicon layers by dry-etching. Next, titanium 6 is formed on the entire plane of a semiconductor substrate to react polycrystalline silicon with titanium at a high temperature to form titanium silicide 7. Thus, silicide having a small sheet resistance can stably be formed.
Patent JP-S5294994-A (JP)
Title: Double line control system
Inventor: AMI YURIO
IPC: G05B15/02
Filed: 1976-02-04
Abstract: PURPOSE: Out of two lines each of which can operate independently, complete separation of the line in trouble for repairment is designed to largely increase the reliability of the lines at this two line control system. 
     COPYRIGHT: (C)1977,JPO&Japio
Patent JP-S54100456-A (JP)
Title: Molded article free from sink marks and mold for producing the same
Inventor: YAMADA FUMIHIKO
IPC: B29C45/44
Filed: 1978-01-23
Abstract: PURPOSE: To prepare the title article having excellent appearance and surface flatness, by integrating a thick-walled part separated from the main part of the molded article to a rib of a thin-walled part at the side face of the thick-walled part.  
     CONSTITUTION: The base of a thick-walled part 2 is separated from the main part 4 of a molded article, and the side face of the thick-walled part 2 is bonded to a thin-walled rib 3 protruded from the main part 4. The length of the bonded part is made to be sufficiently long to attain highly enough strength. The bonding can be carried out by the use of molds 5, 5', wherein a core 1 which blocks the thick-walled part during molding can be removed by pulling out to the direction of the arrow or by turning. 
     COPYRIGHT: (C)1979,JPO&Japio
Patent JP-H01186365-A (JP)
Title: Multicolor ink ribbon
Inventor: KANBAYASHI KENICHI
IPC: B41J31/00
Filed: 1988-01-20
Abstract: PURPOSE:To make ink have various functions by enabling various dyes to be used by coating a dye fixing agent on a ribbon foundation before coating the ink. CONSTITUTION:As a dye fixing agent to be used, a cyclic cation polymer, quaternary salt type cation polymer, etc. which are derived from diallylamine are exemplified. It is generally used, when fiber is dyed by the dye, as a resist printing agent for preventing dyeing of other fiber after dyeing. Then though a dye having a migration property is used as ink, mixture of color to an adjacent color is not generated by coating this dye fixing agent on a ribbon foundation before coating the ink. Therefore, various dyes can be used as the ink. Consequently, various functions, for instance, having long life, making a wire little abrasive, etc. can be given to the ink.
Patent JP-H05206236-A (JP)
Title: Measuring method for particle in vacuum equipment
Inventor: NITTAMI KENJI
IPC: H01L21/66
Filed: 1992-01-24
Abstract: PURPOSE:To obtain the size of a particle, by measuring the intensity difference of scattered light, from when a particle begins to intersect a laser beam until the particle completely leaves the laser beam region, and estimating the particle velocity on the basis of the change of intensity. CONSTITUTION:In the measuring method of a particle in a vacuum equipment wherein a particle 11 is irradiated with a laser beam and scattered light generated at this time is measured, thereby detecting the particle, the scattered light is received with a CCD photosensor 12 having surface resolving power. The received scattered light is subjected to surface resolution, and scattered light intensity distribution is obtained. On the basis of the scattered light intensity distribution, the speed and the size of the particle 11 are detected.
Patent JP-H09262772-A (JP)
Title: Grindstone for polishing stone and the like, and manufacture thereof
Inventor: SUNAKAWA KATSUJI
IPC: B24D11/00
Filed: 1997-01-23
Abstract: PROBLEM TO BE SOLVED: To provide a stone polishing grindstone having more elasticity at the contacting point with a processed object (such as a stone) than the existing vertrified quality polishing tool and a segment making a smooth contact with curvatures and polishing without colliding against the stone. SOLUTION: A segment 6a is provided by filling a metal mold 12a with materials which is made in a granulated chips 10 by sintering a metallic powder 9 containing diamond abrasive particle 8, in a density of the chips individually contacting each other and filling the gap between the granulated chips 10 contacting each other with a resin 11 by pressure, while a sheet shaped polishing grindstone E arranged with a plural number of segments 6e in a preferable shape at sufficient intervals needed to obtain flexibility is made.
Patent JP-H04244857-A (JP)
Title: Printing element for wire dot printer
Inventor: ITO KYOSHI
IPC: B41J2/26
Filed: 1991-01-31
Abstract: PURPOSE:To keep high printing quality by enhancing the strength of a plate- shaped lever and stabilizing printing operation by providing a reinforcing constriction equipped with a centroid wherein reaction force coincides with the acting surface of the center in a thickness direction to the plate-shaped lever supporting a printing wire at one end part thereof and revolving around the other end part thereof to allow the printing wire to advance and recede. CONSTITUTION:A plate-shaped lever 13 supports a printing wire 8 at one end part thereof and revolves around the other end part thereof through an armature 6 to allow the printing wire 8 to advance and recede. Reinforcing constrictions 14 equipped with the centroid wherein the stricking reaction force due to the printing wire 18 coincides with the acting surface 13a of the center in a thickness direction, for example, the wavy constrictions alternately protruding on both sides centering around the acting surface are provided to the plate-shaped lever 13. By this constitution, when the plate-shaped lever 13 is struck, the reinforcing constrictions 14 develop reinforcing effect and no torsional vibration is induced.
Patent JP-H09202788-A (JP)
Title: Asymmetric dioxazine compound, its intermediate compound and application of asymmetric dioxazine compound
Inventor: INOUE MASAHITO
IPC: D06P1/382
Filed: 1996-01-24
Abstract: PROBLEM TO BE SOLVED: To obtain an asymmetric dioxazine compound useful for dyeing and printing a fibrous material, especially a reactive dye for a cellulosic fibrous material. SOLUTION: This asymmetric dioxazine compound is represented by formula I (T1 and T2 are each H, Cl, a lower alkyl, phenoxy, etc.; A1 is an alkyl, Cl, carboxyl, etc.; A2 is H, an alkyl, Cl, carboxyl, etc.; R is H or a lower alkyl; X and Y are each a halogen, a fiber reactive group, etc.). The compound represented by formula I is obtained by condensing an asymmetric triphenedioxazine compound represented by formula II, a compound represented by the formula H-X' (X' is a lower alkoxy, amino, etc.) and a compound represented by the formula H-Y' (Y' is a lower alkyl, amino, etc.) in an optional order with a 2,4,6-trihalogeno-s-triazine.  The compound has good color fastnesses to light, perspiration and sunlight, wet color, chlorine and NOx fastnesses, color fastness to rubbing and ironing fastness and is useful for providing a blue dyed or printed material excellent in especially chlorine fastness.
Patent JP-H08203321-A (JP)
Title: Luminaire
Inventor: NAGAO HITOSHI
IPC: F21V21/02
Filed: 1995-01-26
Abstract: PURPOSE: To prevent the careless dropping of a globe at the time of attaching and detaching it. CONSTITUTION: This luminaire is provided with an appliance main body 1 in which an edge 1b is provided upright toward on the front side in the circumferential end, a reflecting plate 8 mounted on the front side of the appliance main body 1 and a translucent globe 3 which has an opening part 3a on one side and is installed by making the vicinity of the circumferential end part 3b of the opening part nearly abut on the edge part 1b of the appliance main body 1, and one end 1c of the appliance main body 1 is mounted sideways toward the upper side.  In the luminaire, the end part 8a of one end side of the reflecting plate 8 is projected into the inside of the globe 3 so that the distance between the other end side of the appliance main body 1 and the tip 1d of the edge part becomes longer than the distance between the tip 1d of the edge part of the other end side of the appliance main body 1 and the circumferential end part 3b of the opening part of the one end side of the globe 3.
Patent JP-H04244951-A (JP)
Title: Dewing sensor and preparation thereof
Inventor: IZEKI TAKESHI
IPC: H01B5/14
Filed: 1991-01-31
Abstract: PURPOSE:To obtain a resin dispersion type dewing sensor excellent in dewing responsiveness used in various electric machineries by solving such a problem that dewing responsiveness can not be made fast heretofore by making a humidity-sensitive resistance film thin. CONSTITUTION:A humidity-sensitive resistance film 12 is formed on a ceramic substrate 11 and a comb-shape opposed electrode 13 is formed on the humidity- sensitive resistance film 12 and, since humidity-sensitive resistance paste is not applied to the stepped part of the comb-shape opposed electrode and the ceramic substrate as is conventional but can be printed on the plane of the substrate, the thinner humidity-sensitive resistance film can be formed and a resin dispersion type dewing sensor excellent in dewing responsiveness is obtained.
Patent JP-S62166858-A (JP)
Title: Powdery whipping cream
Inventor: NAGAHARA HIROSHI
IPC: A23L9/20
Filed: 1986-01-20
Abstract: PURPOSE:To improve the frothing property, shape-retainability, etc., of a pow dery whipping cream, by mixing a powdery whipping cream with an (acetylated) sucrose fatty acid ester, a glycerol fatty acid ester, lecithin and carrageenan at specific weight ratios. CONSTITUTION:A powdery whipping cream composed mainly of an oil or fat (e.g. palm kernel oil), a sugar (e.g. sucrose) and a protein (e.g. casein sodium) is mixed with 3-50(wt)% acetylated sucrose fatty acid ester (based on the oil or fat), 0.9-5.5% sucrose fatty acid ester, 0.2-1.6% glycerol fatty acid ester and 0.6-4% lecithin. The sum of the above 4 kinds of food emulsifiers is 2-10% based on the oil or fat. The objective powdery whipping cream can be produced by adding 0.1-1wt% carrageenan to the above mixture based on the whole powdery whipping cream.
Patent JP-2000205652-A (JP)
Title: Hot water supplying device
Inventor: TABATA SETSUYOSHI
IPC: F24H1/10
Filed: 1999-01-19
Abstract: PROBLEM TO BE SOLVED: To ensure to prevent hot temperature water from running, by controlling the valve travel of a bypass flow quantity control valve suitably for a form in the case of a water and hot water mixed using form, and by controlling the valve travel of a bypass flow quantity control valve suitably for the form in the case of a single water using form on the basis of the comparison result of a set temperature of running hot water and a threshold temperature. SOLUTION: A bypass channel 13, which bypasses a hot water supplying heat exchanger 2 to provide communication between a water supply channel 6 and a hot water supply channel 10, is provided, and a bypass flow quantity control valve (GM) 14 is interposed in the channel. A hot water supplying mode can be selected from a water/hot water supplying condition in which a mixing faucet is connected for use, and a water supplying condition in which a single faucet is connected for use. When running of hot water is started from the operation condition, in which the temperature of the hot water residing in the hot water supplying heat exchanger 2 rises during the shutdown of hot water running, comparison is made between a set temperature of running hot water and a threshold temperature.  When the set temperature of the running hot water is higher than the threshold temperature, the valve travel control of the GM 14 that is suitable for the water/hot water supplying condition is done. When the set temperature of the running hot water is lower than the threshold temperature, the valve travel control of the GM 14 that is suitable for the single faucet using form is done.
Patent JP-S59136780-A (JP)
Inventor: YAMAMOTO YOSHITAKA
IPC: G09F11/23
Filed: 1983-01-26
Abstract: (57)【要約】本公報は電子出願前の出願データであるた め要約のデータは記録されません。
Patent JP-H09194517-A (JP)
Title: Olefin polymerization catalyst and production of olefin polymer using the catalyst
Inventor: ISOBE EIJI
IPC: C08F4/6392
Filed: 1996-01-25
Abstract: PROBLEM TO BE SOLVED: To provide a new olefin polymerization catalyst and a process for producing an olefin polymer using the catalyst. SOLUTION: The objective olefin polymerization catalyst (A) can be produced by successively performing the following steps (I) to (IV); (I) a step to produce a solid product by contacting a compound selected from a clay, a clay mineral and an ion-exchanging laminar compound with a salt soluble in water or in an acidic aqueous solution and composed of a cation containing a group 4-6 transition metal atom and an anion selected from anion of a halogen, an inorganic acid and an organic acid, (II) a step to wash the solid product until the pH of the washing liquid becomes 3-7, (III) a step to dry the water-washed solid product and (IV) a step to contact the dried solid product with an organic Al compound. An olefin polymer can be produced by polymerizing an olefin in the presence of (A) the catalyst or (A) the catalyst and (B) the organic Al compound.
Patent JP-S57124448-A (JP)
Title: Semiconductor device
Inventor: TABUCHI MASAYUKI
IPC: H01L21/60
Filed: 1981-01-26
Abstract: PURPOSE:To shorten time for construction and reduce the external dimensions of an insulating substrate by a method wherein a plural number of unit semiconductor chips of a kind remaining unseparated is installed on a substrate as a single sheet of multiple semiconductor chips. CONSTITUTION:A pair of unit semiconductor chips remaining unseparated forms a sheet of unified semiconductor chips 7. Each unit chip is connected face down by a bump 6 to a corresponding part on the surface of a conductor pattern exemplifiedly of a thick film covering an insulating substrate 8. This results in the reduction of the number of jobs of installing semiconductor chips, shortening time required for the process.