Patent EP-2562174-A1 (EP)
IPC: C07D417/14
Filed: 2011-08-24
Abstract: Substituted heterocyclic compounds (I) are new. Substituted heterocyclic compounds of formula (I) and their salts are new. Q : substituted 1H-tetrazole-5-yl moieties of formula (IIa), substituted 1H-[1,2,4]triazolyl moieties of formula (IIb), substituted furazanyl moieties of formula (IIc) or substituted [1,3,4]oxadiazolyl moieties of formula (IId); either R1 : phenyl, phenylsulfonyl, W1-(phenyl), W1-(S-phenyl), W1-(SO 2-phenyl), W2-(SO 2CH 2-phenyl) or W2-(SCH 2-phenyl) (all substituted by u substituents R8), 1-10C alkyl, 2-10C alkenyl, 2-10C alkynyl, halo-1-10C alkyl, halo-2-10C alkenyl, halo-2-10C alkynyl, 3-10C cycloalkyl, halo-3-10C cycloalkyl, 1-4C alkyl-3-7C cycloalkyl, 3-7C cycloalkyl-1-6C alkyl, 3-7C cycloalkyl-3-7C cycloalkyl, halo-3-7C cycloalkyl-1-6C alkyl, 1-6C alkyl-3-7C cycloalkyl-1-6C alkyl, 3-12C cycloalkenyl, halo-3-12C cycloalkenyl, 1-6C alkoxy-1-6C alkyl, 1-6C alkoxy-2-6C alkenyl, 1-6C alkyl-3-7C cycloalkyl, 1-6C alkoxy-3-7C cycloalkyl, 3-7C cycloalkoxy-1-6C alkyl, 3-7C cycloalkoxy-1-6C alkoxy-1-6C alkyl, 1-6C alkoxy-1-6C alkoxy-1-6C alkyl, 1-6C alkylthio-1-6C alkyl, 1-6C alkylsulfinyl-1-6C alkyl, 1-6C alkylsulfonyl-1-6C alkyl, 1-6C alkylamino-1-6C alkyl, di-1-6C alkylamino-1-6C alkyl, halo-1-6C alkylamino-1-6C alkyl, 3-7C cycloalkylamino-1-6C alkyl, 1-6C alkylcarbonyl, halo-1-6C alkylcarbonyl, 3-7C cycloalkylcarbonyl, 1-6C alkoxycarbonyl, 3-7C cycloalkoxycarbonyl, 3-7C cycloalkyl-1-6C alkoxycarbonyl, 1-6C alkylaminocarbonyl, di-1-6C alkylaminocarbonyl, 3-7C cycloalkylaminocarbonyl, CN-1-6C alkyl, OH-1-6C alkyl, 3-7C cycloalkenyl-1-6C alkyl, halo-1-6C alkoxy-1-6C alkyl, 1-6C alkoxy-halo-1-6C alkyl, halo-1-6C alkoxy-halo-1-6C alkyl, halo-3-7C cycloalkoxy-1-6C alkyl, 3-7C cycloalkenyl-oxy-1-6C alkyl, halo-3-7C cycloalkenyl-oxy-1-6C alkyl, di-1-6C alkoxy-1-6C alkyl, 1-6C alkoxy-1-6C alkylcarbonyl, 1-6C alkoxycarbonyl-1-6C alkyl, halo-1-6C alkoxycarbonyl, 1-10C alkoxy, halo-1-10C alkoxy, 3-12C cycloalkoxy, halo-3-7C cycloalkoxy, 3-7C cycloalkyl-1-6C alkoxy, 2-12C alkenyloxy, halo-2-10C alkenyloxy, 2-10C alkynyloxy, halo-3-10C alkynyloxy, 1-6C alkoxy-1-6C alkoxy, 1-6C alkylcarbonyloxy, halo-2-12C alkylcarbonyloxy, 3-7C cycloalkylcarbonyloxy, 1-6C alkylcarbonyl-1-6C alkoxy, 1-10C alkylthio, halo-1-10C alkylthio, 3-12C cycloalkylthio, 1-10C alkylsulfinyl, halo-1-10C alkylsulfinyl, 1-10C alkylsulfonyl, halo-1-10C alkylsulfonyl, 3-12C cycloalkylsulfonyl, 1-6C alkyl-carbonylthio, 1-6C alkyl(thiocarbonyl)thio, 3-12C cycloalkylsulfinyl, 1-6C alkyl-aminosulfonyl, di-1-6C alkylamino-sulfonyl, 1-6C alkylamino, di-1-6C alkylamino , halo-1-6C alkylamino, halo-di-1-6C alkylamino, 3-12C cycloalkylamino, 1-6C alkylcarbonylamino, halo-1-6C alkylcarbonylamino, 1-10C alkylsulfonylamino, halo-1-10C alkylsulfonylamino, 3-7C cycloalkyl-1-6C alkylamino, CN, OH, NH 2, C(=O)OH, C(=O)NHOH, SO 2NH 2, SO2 NHCN, SO 2NHOH, NHCHO, G or W2G; and R2 : phenyl or W3-(phenyl) (both substituted by u substituents R8), G, W4G, H, CN, OH, NH 2, NO 2, CHO, C(=O)OH, C(=O)NH 2, C(=S)NH 2, C(=O)NHCN, C(=O)NHOH, SH, SO 2NH 2, SO 2NHCN, SO 2NHOH, SF 5, NHCHO, NHNH 2, NHOH, NHCN, NHC(O)NH 2, 1-10C alkyl, 2-10C alkenyl, 2-10C alkynyl, halo-1-10C alkyl, halo-2-10C alkenyl, halo-2-10C alkynyl, 3-8C cycloalkyl, halo-3-8C cycloalkyl, 1-6C alkyl-3-7C cycloalkyl, 3-7C cycloalkyl-1-6C alkyl, 1-6C cycloalkyl-1-6C cycloalkyl, halo-1-6C cycloalkyl-1-6C alkyl, 1-6C alkyl-3-7C cycloalkyl-1-6C alkyl, 3-8C cycloalkenyl, halo-3-8C cycloalkenyl, 1-6C alkoxy-1-6C alkyl , 1-6C alkoxy-1-6C alkenyl, 1-6C alkyl-3-7C cycloalkyl, 1-6C alkoxy-3-7C cycloalkyl, 1-6C cycloalkoxy-1-6C alkyl, 3-7C cycloalkoxy-1-6C alkyl, 1-6C alkoxy-1-6C alkoxy-1-6C alkyl, 2-8C alkylthioalkyl, 1-6C alkylsulfinyl-1-6C alkyl, 1-6C alkylsulfonyl-1-6C alkyl, 1-6C alkylamino-1-6C alkyl, di-1-6C alkylamino-1-6C alkyl, halo-1-6C alkylamino-1-6C alkyl, 3-7C cycloalkylamino-1-6C alkyl, 1-6C alkylcarbonyl, halo-1-6C alkylcarbonyl, 3-7C cycloalkylcarbonyl, 1-6C alkoxycarbonyl, 3-7C cycloalkoxycarbonyl, 3-7C cycloalkyl-1-6C alkoxycarbonyl, 1-6C alkylaminocarbonyl, di-1-6C alkylaminocarbonyl, 3-7C cycloalkylaminocarbonyl, CN-1-6C alkyl, OH-1-6C alkyl, 3-7C cycloalkenyl-1-6C alkyl, halo-1-6C alkoxy-1-6C alkyl, di-1-6C alkoxy-1-6C alkyl, 1-6C alkoxy-1-6C alkylcarbonyl, 1-6C alkoxycarbonyl-1-6C alkyl, halo-1-6C alkoxycarbonyl, 1-6C alkoxy, halo-1-6C alkoxy, 3-8C cycloalkoxy, halo-3-8C cycloalkoxy, 3-7C cycloalkyl-1-6C alkoxy, 2-6C alkenyloxy, halo-2-6C alkenyloxy, 2-6C alkynyloxy, halo-3-6C alkynyloxy, 1-6C alkoxy-1-6C alkoxy, 1-8C alkylcarbonyloxy, halo-1-8C alkylcarbonyloxy, 3-7C cycloalkylcarbonyloxy, 1-6C alkylcarbonyl-1-6C alkoxy, 1-6C alkylthio, halo-1-6C alkylthio, 3-8C cycloalkylthio, 1-6C alkylsulfinyl, halo-1-6C alkylsulfinyl, 1-6C alkylsulfonyl, halo-1-6C alkylsulfonyl, 3-10C cycloalkylsulfonyl, 1-6C alkyl-carbonylthio, 1-6C alkyl(thiocarbonyl)thio, 3-8C cycloalkylsulfinyl, 1-6C alkyl-aminosulfonyl, di-1-6C alkyl-aminosulfonyl, 1-6C alkylamino, di-1-6C alkylamino, halo-1-6C alkylamino, halo-di-1-6C alkylamino, 3-8C cycloalkylamino, 2-8C alkylcarbonylamino, halo-2-8C alkylcarbonylamino, 1-10C alkylsulfonylamino, halo-1-10C alkylsulfonylamino, 3-7C cycloalkyl-1-6C alkylamino or halo-tri-1-4C alkylsilyl; or R1+R2+atoms to which they are bonded : 5-, 6- or 7-membered ring (optionally saturated or partially saturated and contains m number of N, n number of O, n number of S and n number of S(O), S(O) 2or C(O), where C atoms are substituted by s number of halo, CN, 1-6C alkyl, 2-10C alkenyl, 2-10C alkynyl, 1-6C haloalkyl, 3-8C cycloalkyl, 2-8C alkoxyalkyl or phenyl (substituted by u number of CN, NO 2, halo, 1-6C (halo)alkyl or 1-6C alkoxy), and N atoms are substituted by n number of 1-6C alkyl or phenyl (substituted by u number of CN, NO 2, halo, 1-6C (halo)alkyl or 1-6C alkoxy); and X : N or C-R3. Full definitions are given in the DEFINITIONS (Full Definitions) Field. An independent claim is also included for an herbicidal agent comprising (I). [Image] [Image] ACTIVITY : Herbicide. Test details are described but no results given. MECHANISM OF ACTION : None given.