baber/WOPTO huggingface dataset:
Patent ES-510015-A0 (ES)
IPC: C07D271/04
Filed: 1982-03-01
Abstract: Pharmacologically-active 3-aminosydnonimines (which are optionally substituted in the N6-position) and their physiologically-acceptable acid-addition salts are compounded into standard dosage-form medicament compositions and are useful for prophylaxis for and treatment of cardiovascular-system disorders, such as high blood pressure and angina pectoris. The 3-aminosydnonimines are 3-[4-(lower alkoxy)carbonylpiperazin-1-yl]sydnonimines and 3-[N-(lower alkyl)-N-(tetrahydro-3-thienyl S,S-dioxide)]-sydnonimines.
Patent ES-522740-A0 (ES)
IPC: C07C59/56
Filed: 1983-05-26
Abstract: (d)-2-(6-Methoxy-2-naphthyl)propionic acid and pharmaceutically acceptable salts thereof are prepared by resolving mixtures of (d)- and (1)-enantiomers of 2-(6-methoxy-2-naphthyl)propionic precursor acids or salts thereof with N-alkyl- or N-cycloalkyl-D-glucamines or salts thereof to isolate the corresponding (d)-2-(6-methoxy-2-naphthyl)propionic precursor acid which can be readily converted into (d)-2-(6-methoxy-2-naphthyl)propionic acid or a pharmaceutically acceptable salt thereof.
Patent ES-527717-A0 (ES)
IPC: H02H3/33
Filed: 1983-12-01
Abstract: 1. In use, an earth leakage circuit breaker with a sum current transformer (3) having a primary winding of magnitude sufficient at 50 Hz, in whose secondary circuit is arranged a triggering device (4) following the principle of a holding magnet and wherein the secondary circuit between the sum current transformer (3) and the triggering device (4) contains a rectifier arrangement (7), the circuit serving as a frequency-independent earth leakage circuit breaker in a frequency range from 16 2/3 Hz to 30 kHz.
Patent ES-534321-A0 (ES)
IPC: A61K38/27
Filed: 1984-07-13
Abstract: Disclosed is an improved plasmid which upon introduction into a suitable Escherichia coli host cell containing the thermolabile repressor CI, renders the host cell capable, upon increasing the temperature of the host cell to a temerature at which the repressor is destroyed, of effecting expression of a gene encoding superoxide dismutase inserted into the vector, and production of the superoxide dismutase encoded by the gene.
Patent ES-546602-A0 (ES)
IPC: C07D209/12
Filed: 1985-08-30
Abstract: A compound represented by the formulawherein R, represents a lower alkyl group; each of R<sub>2</sub> and R<sub>3</sub> represents an alkyl group having 1 to 3 carbon atoms; and each of R<sub>4</sub>, R<sub>5</sub> and R<sub>6</sub> represents a hydrogen atom, a halogen atom, a lower alkyl group, a lower alkoxy group, a lower alkanoyloxy group, an aralkyloxy group, a lower alkylthio group, a lower haloalkyl group, a hydroxyl group, a cyano group, a nitro group, an amino group, a mono- or di-(lower alkyl or aralkyl)amino group or a group of the formulaorin which R<sub>7</sub> represents a lower alkylene group having at least 2 carbon atoms, one of R<sub>8</sub> and R<sub>s</sub> represents a hydrogen atom or a lower alkyl group and the other represents a lower alkyl group, and R<sub>10</sub> represents a hydrogen atom or a lower alkyl group; or any two of R<sub>4</sub>, R<sub>5</sub> and R<sub>6</sub> which are adjacent to each other, together, represent a lower alkylenedioxy group, and a salt thereof; and a process for production thereof. This compound has 5-lipoxygenase inhibiting activity and is useful as a medicament.
Patent ES-555134-A0 (ES)
IPC: C08F4/634
Filed: 1986-05-20
Abstract: A process for removing one or more contaminants of the formula TiCl<sub>3</sub>OR, in which R is an alkyl or aryl group, from a liquid phase comrising TiCl<sub>4</sub>, characterized in that the contaminants are reacted with an organic acid halide R'-C" O Cl, in which R' is an aryl or alkyl group, to precipitate an addition complex of the formula nTiCl<sub>4</sub>.R'-C "O OR, in which n is a number of from 0.3 to 3.0, and the addition complex is separated from the liquid phase.
Patent FI-864269-A0 (FI)
Inventor: SCHMALENBACH WERNER
IPC: H01H13/14
Filed: 1986-10-22
Abstract: 1. Electric pushbutton switch, especially in a flush-mounted design for house installations, comprising at least one internal and at least one external pushbutton and also a rotatable, non-positively coupled height-controlling element arranged centrally between the inner and outer pushbuttons, through the rotation of which element a variation in the clearance between the inner and outer pushbuttons can be carried out, characterized in that the height-controlling element (7) has a lower part (19) facing the internal pushbutton (2) and an upper part (20) facing the external pushbutton (3), at least n = 2 multiple-step first stairways (9) of mutually identical shape, and running in the form of spiral stairway along an associated circular arc b = 2 r pi /n, being constructed on the lower part (19) to run peripherally along a base circle (18), and second stairways (10) being constructed on the upper part (20) correspondingly to and interlocking with the first stairways (9), in such a way that the meeting of the respective uppermost stairway steps (9a) of the first stairway steps (9a) of the first stairways (9) with the respective lowermost stairway steps (10b) of the second stairways (10) produces the minimum clearance, and the meeting of the respective uppermost stairway steps (9a) of the first stairways (9) with the respective uppermost stairway steps (10a) of the second stairways (10) produces the maximum clearance.
Patent FI-870100-A0 (FI)
Inventor: TOMCUFCIK ANDREW STEPHEN
IPC: C07D417/12
Filed: 1987-01-12
Abstract: Omega-[(hetero)alkyl]benz[cd]indol-2-amines useful in inhibition of thromboxane synthetase and in treatment of hypertension in warm-blooded animals are disclosed.
Patent FI-881016-A0 (FI)
Inventor: ROSELLE BRIAN JOSEPH
IPC: C11D3/395
Filed: 1988-03-04
Abstract: Detergent compositions suitable for use in automatic dishwashing machines are disclosed. The compositions contain detergency builder materials, a chlorine bleach component, an optional low-foaming, bleach-stable surfactant and a relatively water-soluble stilbene dye which is color-stable with respect to said chlorine bleach component and which does not stain dishes etc.
Patent FI-881270-A0 (FI)
Inventor: MANUSCH CHRISTOPH
IPC: B43M11/06
Filed: 1988-03-17
Abstract: The device, suitable for use in a hand roller, for transferring a film from a carrier tape to a substrate is a cartridge containing a feed reel and a windup reel. The tape travels by way of a protruding stiff applicator bar which has a pressure-applying edge for pressing the tape against the substrate. The stiff applicator bar is on a spring support member which can be deflected until a protrusion on the bar encounters a detent fixed on the housing. The application bar has its pressure-applying edge appropriately shaped to facilitate the transfer action.
Patent FI-890713-A0 (FI)
Inventor: MARUYAMA HIROSHI
IPC: G03F1/90
Filed: 1989-02-15
Abstract: A lightsafe masking film is disclosed which comprises a substrate, and a peelable lightsafe layer provided over the surface of the substrate and including a lightsafe substance, a copolymer containing vinyl chloride, and a mixture of a first nitrile rubber containing 25-30 % by weight of acrylonitrile and a second nitrile rubber containing 31-35 % by weight of acrylonitrile.
Patent FI-891865-A0 (FI)
Inventor: HETTCHE HELMUT
IPC: A61K9/32
Filed: 1989-04-19
Abstract: Azelastine-containing pharmaceutical compositions with controlled release of active substance using a release-delaying component, there being 0.001 to 800 parts of release-delaying component for one part by weight of azelastine (as base), and it also being possible for the azelastine to be in the form of its physiologically tolerated salts, and the rate of azelastine release being between 0.05 and 5 mg per hour.
Patent FI-900271-A0 (FI)
Inventor: GUICHARD PHILIPPE
IPC: H04N7/015
Filed: 1990-01-17
Abstract: PCT No. PCT/NL89/00037 Sec. 371 Date Mar. 20, 1990 Sec. 102(e) Date Mar. 20, 1990 PCT Filed May 19, 1989 PCT Pub. No. WO89/11767 PCT Pub. Date Nov. 30, 1989.In order to reduce the digital data throughput, the transmission system comprises means for determining, for each image, in the set of speed vectors, a subset containing the vectors which are encountered most frequently in this image, and means for digitally transmitting, once per image, the characteristics of all the vectors of this subset, and if the speed vector of an image part to be transmitted is an element of the subset, it is defined by reference to the subset, while, if it is not an element of the subset, another transmission mode is used for the current image part, being a mode in which the speed vector is not used, but in which the analog video data are transmitted with a lower spatial definition but with a higher frame rate.
Patent FI-902327-A0 (FI)
Inventor: LUDLOW IAN KEITH
IPC: G01N/
Filed: 1990-05-09
Abstract: An apparatus and method which provides a measure of the asymmetry as well as the size of individual fluid borne particles. Laser-light scattering techniques are employed to obtain data on the particles, which is then compared to data on known particle shapes to ascribe an asymmetry factor to the particles.
Patent FI-905138-A0 (FI)
Inventor: NEUHAUS ALFRED
IPC: C08J9/08
Filed: 1990-10-18
Abstract: A process for the production of moulded articles having a density of at least 250 kg/m<3> from polyurethane foams having a compact surface by expansion, in a mould, of a reaction mixture of a polyisocyanate component, a reactive component consisting of at least one organic polyhydroxy compound, blowing agents and optionally further auxiliaries and additives, the blowing agents used being salts of (i) organic carboxylic acids and (ii) nitrogen bases having at least one N-H bond, and moulded articles obtained by this process.
Patent FI-911282-A0 (FI)
Inventor: MARCINIAK GILBERT
IPC: A61P29/00
Filed: 1991-03-15
Abstract: This invention relates to derivatives of certain 3,4-dihydroxy-2,5-dihydrofuran-5-ones, to the intermediates and processes useful for their preparation, to their free-radical scavenger and cellular protective properties, and to their end-use application as therapeutic agents.
Patent FI-912937-A0 (FI)
Inventor: BRAX VEIKKO
IPC: H04W88/06
Filed: 1991-06-17
Abstract: A method for handling a call coming via a digital transmission system in terminal equipment suitable for speech and data service, the transmission system including at least one connection element which is a speech transmission connection when the call is in speech service mode and which is a data transmission connection rate-adapted in compliance with the CCITT recommendation V.110 or in a like manner and preferably attached to V.24 interfaces when the call is in data service mode. The terminal equipment starts the connection in speech service mode and automatically changes over to data service mode and initiates a procedure for changing the at least one connection element to a data transmission connection upon receipt, in speech mode, of a predetermined audio signal from the connection. The method can make use of a mobile telephone.
Patent FI-913428-A0 (FI)
Inventor: ARNOLD ALAN FREDERICK
IPC: G11B19/04
Filed: 1991-07-16
Abstract: This invention relates to personal computers, and particularly to a personal computer having provision for identifying the storage capability of a removable media direct access storage device used with the computer. At least certain ones of a plurality of signal communicating pathways extending between a storage device and a controller for the storage device are used to identify to the controller the type of device with which the controller is communicating. The apparatus disclosed distinguishes among a plurality of types of removable media potentially used in removable media direct access storage devices using at least certain ones of a plurality of signal communicating pathways extending between a storage device and a controller for the storage device to identify to the controller the type of media inserted into the device with which the controller is communicating.
Patent FI-925525-A0 (FI)
Inventor: BYRD ALAN EUGENE
IPC: A61F13/472
Filed: 1992-12-04
Abstract: Disclosed is a sanitary napkin and releasable wrapper package. The releasable wrapper is folded about the longitudinal side margins of the sanitary napkin in a C-fold so that both faces of the sanitary napkin are protected and a relatively smaller package is produced than if the releasable wrapper extends laterally beyond the longitudinal side margins of the sanitary napkin. The releasable wrapper and sanitary napkin may be trifolded about spaced-apart, laterally oriented fold lines to produce a discrete single use package. Several variations, including flapped and asymmetric embodiments, are illustrated.
Patent FI-930092-A0 (FI)
Inventor: CHEN YUHPYNG L
IPC: A61P25/28
Filed: 1993-01-11
Abstract: Compounds of formula (I) wherein W is (a) or (b) and R<7>, R<8>, R<9>, R<10>, R<11>, R<6>, R<5> and R<1> are as described herein.
Patent FI-941933-A0 (FI)
Inventor: KLOEBER JOHANNES
IPC: E04D1/36
Filed: 1994-04-26
Abstract: The roof-ridge-sealing strip has a central air-permeable zone (8) of fabric structure, and two edge areas (9) adaptable to the corrugations of the tiles by stretchable stabilising inlay(s) of metal or other material. The strip is in one piece of fabric extends for the full width, and is extensible in the lengthwise direction at least at the edge areas. The inlay has undulating wires or strips running parallel to the edge (10'), and which are secured to the fabric surface in a holder allowing variation of the undulating pattern.
Patent FI-945248-A0 (FI)
Inventor: BARSOUM JAMES G
IPC: C12N15/87
Filed: 1994-11-08
Abstract: This invention relates to delivery of biologically active cargo molecules such as polypeptides and nucleic acids into the cytoplasm and nuclei of cells  in vitro  and  in vivo.  Intracellular delivery of cargo molecules according to this invention is accomplished by the use of novel transport polypeptides which comprise one or more portions of HIV tat protein and which are covalently attached to cargo molecules. The transport polypeptides of this invention are characterized by the presence of the tat basic region (amino acids 49-57), the absence of the tat cysteine-rich region (amino acids 22-36) and the absence of the tat exon 2-encoded carboxy-terminal domain (amino acids 73-86) of the naturally-occurring tat protein. By virtue of the absence of the cysteine-rich region found in conventional tat proteins, transport polypeptides of this invention solve the problems of spurious trans-activation and disulfide aggregation. The reduced size of the transport polypeptides of this invention also minimizes interference with the biological activity of the cargo molecule.
Patent FI-954413-A0 (FI)
Inventor: HEINZMANN HELMUT
IPC: D21F1/00
Filed: 1995-09-19
Abstract: The dispenser has a flow chamber with inlet and outlet and, built into the chamber, a segment comprising many channels with a surface structure for turbulence generation. In cross-section perpendicular to the flow the channels are in length at least double that of their breadth. Also claimed is the application of the above dispenser in a multi-layer pulp dispenser. Pref. the channels, each dimensioned to match approx. the turbulent flow regime, are approx. vertical, alternatively inclined to the vertical or they run horizontally, each extending at maximum to half, or a third or a quarter of machine width.
Patent FI-961125-A0 (FI)
Inventor: KIVIPELTO PEKKA
IPC: F16K3/26
Filed: 1996-03-11
Abstract: PCT No. PCT/FI97/00158 Sec. 371 Date Apr. 21, 1999 Sec. 102(e) Date Apr. 21, 1999 PCT Filed Mar. 11, 1997 PCT Pub. No. WO97/34097 PCT Pub. Date Sep. 18, 1997A control valve comprises a valve body (1) including two flow channels (2, 2'); a cup-formed, steplessly turnable closure member (5); and a shaft (6) for turning the closure member. On the sides of the closure member there is at least one opening (14). The second flow channel (2') has in the valve body (1) an extension (10), the outer surface of which forms a surface of revolution concentric with the inner surface of the closure member (5), and which extends within the closure member. On the sides of the flow channel extension there is at least one opening (21). The opening or openings (14) of the closure member are located so that in the open position of the valve they at least partly overlap the opening or openings (21) of the flow channel extension (10). In the closed position of the valve the openings of the flow channel are covered by the closure member.
Patent AP-9600905-A0 (AP)
Title: Methods of producing effective recombinant serine protease inhibitors and uses of these inhibitors.
Inventor: RUBIN HARVEY
IPC: C12N15/63
Filed: 1995-04-11
Abstract: A method of producing a recombinant serine protease inhibitor capable of effectively modulating serine protease activity is provided. Compositions capable of modulating serine protease activity and use of such compositions to regulate inflammatory processes in cells are also provided.
Patent IL-61689-A0 (IL)
Title: Reaction vessel
IPC: B01J3/06
Filed: 1980-12-11
Abstract: The present invention relates to a reaction vessel adapted to withstand pressures and temperatures of the magnitude associated with the manufacture of diamond products and boron nitride (BN) and similar hard materials. The reaction vessel has an outer chamber or shell formed from steel and an inner reaction chamber. Known vessels of this type must be provided with a thick layer of insulating material between the reaction chamber and the outer steel shell to protect the outer shell from the heat of the diamond-forming process carried on in the reaction chamber. The quantity of insulating material required within the vessel for adequate protection of the outer shell is relatively large as compared to the area of the outer shell. Accordingly, the amount of available space remaining within the vessel for the diamond-forming reaction is limited, thus limiting the size of the diamonds formed. The present invention provides a reaction vessel with a cooling system which eliminates the need for the large quantity of insulating material in the known vessels. As such, the reaction vessel provides a significantly larger reaction chamber for the diamond-forming process, and the resultant diamonds are up to a thousand times larger than those formed from known reaction vessels. In one embodiment of the invention, the cooling system includes a plurality of truncated steel pyramids arranged to form flow passages or channels for a cooling fluid adjacent to the inner wall of the vessel's outer steel shell to absorb and disperse heat before it penetrates the outer steel shell.
Patent IL-61805-A0 (IL)
Title: Preparation of oxiranes
IPC: C07D301/12
Filed: 1980-12-26
Abstract: 1. Process for the preparation of oxiranes from olefines and hydrogen peroxide in the presence of orthoboric acid, characterized in that a) an olefine of the general formula  see diagramm : EP0031537,P8,F1 wherein R1 , R2 , R3  and R4  independently of one another denote hydrogen, C1 - to C30 -alkyl, C1 -to C15  -alkenyl, C3 -C1 -cycloalkyl, phenyl or naphthyl, and/or wherein R1  and R2  can be linked to one another by a hydrocarbon chain with up to 12 carbon atoms, and/or wherein R1  and R3 , together with the double bond to be epoxidized can form a mono- di- or tri-cyclic ring system with up to 12 carbon atoms, and wherein R1 , R2 , R3  and R4  can optionally contain as substituents C1 - to C4 -alkyl, C3 -to C6 -cycloalkyl, C1 - to C4 - alkenyl, phenyl, C1 - to C4 -alkoxy, hydroxyl, carboxyl or halogen, there being at least one further carbon atom between the carbon atom which contains alkoxy, hydroxyl, carboxyl or halogen as a substituent and the double bond to be epoxidised, is reacted with a solution, containing less than 0,1 % by weight of water, of hydrogen peroxide in a solvent at a temperature of 30 to 110 degrees C and for a reaction time which, depending on the reactivity of the olefin introduced, is between 15 minutes and 5 hours, b) the oxirane formed and the unreacted olefine are separated off, c) the amount of hydrogen peroxide which has been consumed during the reaction is added to the reaction mixture before, during and/or after separating off the oxirane and olefine, d) after carrying out steps b) and c), the water is largely removed from the reaction mixture and e) the resulting solution, containing less than 0.1 % by weight of water, of hydrogen peroxide and orthoboric acid in the solvent is reacted again with the olefine.
Patent IL-71863-A0 (IL)
Title: Aryloxy-and arylthio-hydroxypropylene-piperazinylacetanilides,their preparation and pharmaceutical compositions containing them
IPC: A61P9/08
Filed: 1984-05-17
Abstract: Novel compounds of the general formula   <IMAGE> (I)  and the pharmaceutically acceptable esters and acid addition salts thereof, wherein: R1, R2, R3, R4 and R5 are each independently hydrogen, lower alkyl, lower alkoxy, cyano, trifluoromethyl, halo, lower alkylthio, lower alkyl sulfinyl, lower alkyl sulfonyl, N-optionally substituted alkylamido, except that when R1 is methyl, R4 is not methyl; or R2 and R3 together form -OCH2O-; R6, R7, R8, R9 and R10 are each independently hydrogen, lower acyl, aminocarbonylmethyl, cyano, lower alkyl, lower alkoxy, trifluoromethyl, halo, lower alkylthio, lower alkyl sulfinyl, lower alkyl sulfonyl, di-lower alkyl amino; or R6 and R7 together form -CH=CH-CH=CH-; R7 and R8 together form -OCH2O-; R11 and R12 are each independently hydrogen or lower alkyl; and W is oxygen or sulfur. These cardioselective compounds have calcium entry blockade properties and therefore are useful in therapy in the treatment of cardiovascular diseases, including arrhythmias, variant and exercise induced angina and myocardial infarction.
Patent IL-83132-A0 (IL)
Title: 6-or 7-methylenandrosta-1,4-diene-3,17-dione derivatives,their preparation and pharmaceutical compositions containing them
IPC: C07J71/00
Filed: 1987-07-08
Abstract: The invention relates to new 6- or 7-methylenandrosta-1,4-diene-3,17-diones of the following formula <CHEM> wherein R is hydrogen or fluorine; R1 is hydrogen or C1-C6 alkyl; R2 is hydrogen or halogen; one of R3 and R4 is =CH2 and the other is hydrogen or C1-C4 alkyl, and when R3 is =CH2, at least one of R and R4 is other than hydrogen; and the symbol @ @@ represents a double bond and the symbol @@@ represents a single bond when R3 is =CH2 or the symbol @@@ represents a single bond and the symbol @@@ represents a double bond when R4 is =CH2, which are useful in therapy, in particular as anti-cancer agents.
Patent IL-85002-A0 (IL)
Title: Flat seal
IPC: H05K5/06
Filed: 1988-01-01
Abstract: A seal, particularly a flat seal to be arranged between two bodies, in particular a magnetic head and a plug socket with one part having at least one electrical plug and another part in which the plug is engageable and with at least one structural element, the seal comprises an electrical conductor printed circuit board arranged to provide an electrical contact between the electrical structural element and the plug, and a sealing mass in which the electrical printed circuit board is arranged, the sealing mass being formed as a pre-formed frame in which the printed circuit board is insertable.
Patent IL-91756-A0 (IL)
Title: Pyridoindole derivatives,processes for the preparation thereof and pharmaceutical compositions containing the same
IPC: A61K31/435
Filed: 1989-09-24
Abstract: A compound of the formula : <CHEM>  wherein  R<1> is hydrogen, lower alkyl or lower alkenyl  R<2> is hydrogen, lower alkyl or halogen, R<3> is imidazolyl or pyridyl, each of which may have suitable substituent(s), and R<4> is hydrogen, lower alkyl, lower alkenyl or hydroxy(lower)alkyl and R<5> is hydrogen, hydroxy or acyloxy, or  R<4> and R<5> are linked together to form an additional bond, and pharmaceutically acceptable salts thereof, processes for their preparation and pharmaceutical compositions comprising them in association with the pharmaceutically acceptable, substantially non-toxic carrier or excipient.