baber/WOPTO huggingface dataset:
Patent EP-2301916-A2 (EP)
Inventor: BERNIAC JOEL
IPC: A61K31/65
Filed: 2005-10-25
Abstract: A compound of formula I:
     
wherein: 
R 2'  and R 2"  are each independently hydrogen, alkyl, alkenyl, alkynyl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, alkylamino, arylalkyl, aryl, heterocyclic, heteroaromatic or a prodrug moiety; 
R 10 , R 11  and R 12  are each independently hydrogen, alkyl, aryl, benzyl, arylalkyl, or a pro-drug moiety; 
R 3'  is hydroxyl, hydrogen, or a pro-drug moiety; 
R 4  is N-OH; 
R 5  and R 5'  are each independently hydroxyl, hydrogen, thiol, alkanoyl, aroyl, alkaroyl, aryl, heteroaromatic, alkyl, alkenyl, alkynyl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, alkylamino, arylalkyl, alkyl carbonyloxy, or aryl carbonyloxy; 
R 6  and R 6'  are each independently hydrogen, methylene, absent, hydroxyl, halogen, thiol, alkyl, alkenyl, alkynyl, aryl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, alkylamino, or an arylalkyl; 
R 7  is hydrogen, hydroxyl, halogen, thiol, nitro, alkyl, alkenyl, alkynyl, aryl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, arylalkyl, amino, arylalkenyl, arylalkynyl, acyl, aminoalkyl, heterocyclic, thionitroso, or-(CH 2 ) 0-3 (NR 7c ) 0-1 C(=W')WR 7a ; 
R 8  is hydrogen, hydroxyl, halogen, thiol, nitro, alkyl, alkenyl, alkynyl, aryl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, alkylamino, amino, arylalkenyl, arylalkynyl, acyl, aminoalkyl, heterocyclic, thionitroso, or-(CH 2 ) 0-3 (NR 8c ) 0-1 C (=E')ER 8a ; 
R 9  is hydrogen, hydroxyl, halogen, thiol, nitro, alkyl, alkenyl, alkynyl, aryl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, arylalkyl, amino, arylalkenyl, arylalkynyl, acyl, aminoalkyl, heterocyclic, thionitroso, or -(CH 2 ) 0-3 (NR 9c ) 0-1 C(=Z')ZR 9a ; 
R 7a , R 7b , R 7c , R 7d , R 7e , R 7f , R 8a , R 8b , R 8c , R 8d , R 8e , R 8f , R 9a , R 9b , R 9c , R 9d , R 9e , and R 9f  are each independently hydrogen, acyl, alkyl, alkenyl, alkynyl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, alkylamino, arylalkyl, aryl, heterocyclic, heteroaromatic or a prodrug moiety; 
R 13  is hydrogen, hydroxy, alkyl, alkenyl, alkynyl, alkoxy, alkylthio, aryl, alkylsulfinyl, alkylsulfonyl, alkylamino, or an arylalkyl; 
E is CR 8d R 8e , S, NR 8b  or O; 
E' is O, NR 8f , or S; 
W is CR 7d R 7e , S, NR 7b  or O; 
W' is O, NR 7f , or S; 
X is CHC(R 13 Y'Y), C=CR 13 Y, CR 6' R 6 , S, NR 6 , or O; 
Y' and Y are each independently hydrogen, halogen, hydroxyl, cyano, sulfhydryl, amino, alkyl, alkenyl, alkynyl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, alkylamino, or an arylalkyl; 
Z is CR 9d R 9e , S, NR 9b  or O; 
Z' is O, S, or NR 9f , or a pharmaceutically acceptable salt, ester or enantiomer thereof.
Patent EP-2325739-A2 (EP)
Inventor: KASAHARA SHUNICHI
IPC: G06F3/041
Filed: 2010-11-11
Abstract: An device and method provide logic for processing information. In one implementation, an information processing device includes a detection unit configured to detect a speed of selection of information. The information processing device also includes a generation unit configured to generate a signal specifying a display format, based on the speed of information selection, and a display unit configured to display the selection of information according to the signal.
Patent EP-2338616-A2 (EP)
Inventor: JANUTIN ANDREAS
IPC: B08B1/02
Filed: 2010-11-30
Abstract: The cleaner (1) has cleaning member carriers (16, 17), each comprising a cleaning member. A parallel drive moves the cleaning members and a support rail (2) relative to each other and moves transversely relative to longitudinal axis (5) of the support rail to remove deposits from the support rail by the units of the cleaning member. A transverse drive periodically moves the cleaning member carriers and the support rail toward and away from each other and transversely relative to lateral longitudinal faces (6, 7) of the support rail. An independent claim is also included for a method for cleaning a mechanical support rail of a workpiece support in a machine tool.
Patent EP-2336952-A2 (EP)
Inventor: ADDY KENNETH
IPC: H01Q1/22
Filed: 2010-12-07
Abstract: A method of printing comprising the steps of: providing a print media (158) having a printing surface; measuring at least one parameter of the print media (214); calculating (218) an optimal configuration for a radio frequency identification (RFID) transponder (170) circuit for obtaining a desired RFID transponder resonant frequency; configuring the RFID transponder circuit and printing (222) the RFID transponder circuit onto the print media.
Patent EP-2339871-A2 (EP)
Inventor: SOLUM JEFFREY PAUL
IPC: H04R25/00
Filed: 2010-12-21
Abstract: The present disclosure relates to the wireless communication of analog and digital information using a modulator adapted to communicate analog information in an analog mode and to communicate digital information in a digital mode using frequency modulated transmissions. A demodulator adapted to receive the modulated information is provided. The present subject matter can be used with hearing assistance devices to communicate voice and data information. Applications of the system include communications with assistive listening devices, hearing aids, and other hearing assistance devices.
Patent EP-2239214-A2 (EP)
Inventor: ROTH HEINZ ING
IPC: B65G47/54
Filed: 2010-04-07
Abstract: The device (1) has a transferring device (2) for transferring pieces of goods (8) to a transverse transporter at an input side, and an output (3) for outputting the pieces of goods to a longitudinal transporter. An acceleration device (4) accelerates the pieces of goods in a longitudinal direction (91) for retaining the pieces of goods in a truncated cone shaped roller (41). Axes (42) of the roller are arranged proximate to the output at a side (43) turned towards the transferring device than at a side (44) turned away from the transferring device.
Patent EP-2396499-A2 (EP)
Inventor: RITCHIE DARREN JOHN
IPC: E21B23/00
Filed: 2010-02-11
Abstract: The present invention relates to downhole tools, and in particular an underreamer tool (1) for use in a wellbore of an oil or gas well and a method of actuation. In an embodiment, the underreamer tool (1) has body (10) having a longitudinal axis(18) and a fluid conduit, a tool element (20) and an actuation device (90) configured to urge the tool element (20) relative to the body (10) from a first configuration into a second configuration. In this embodiment, a portion (30) of the tool (1) has a curved actuation surface (30e) and as the tool element (20) is urged across the curved actuation surface (30e), the tool element (20) is moved radially with respect to the body (10) of the tool (1). Typically, the actuation device (90) may include a piston (60) driven by pressure of fluid circulated through the fluid flow conduit (16).
Patent EP-2456476-A2 (EP)
Inventor: BOSLEY JR RODNEY W
IPC: A61L27/14
Filed: 2010-07-21
Abstract: Disclosed are tissue graft compositions made of particles having different densities, methods of making these compositions, and methods of using these compositions for promoting tissue restoration in a patient.
Patent EP-2395100-A2 (EP)
Inventor: PARK SANG GYU
IPC: G01N33/53
Filed: 2010-02-05
Abstract: The present invention provides, as a novel diagnosis marker for type 1 diabetes mellitus, a type 1 diabetes mellitus diagnostic composition comprising alanyl-tRNA synthetase, glycyl-tRNA synthetase, asparaginyl-tRNA synthetase, or tryptophanyl-tRNA synthetase, a diagnostic kit comprising the same, and a diagnostic method using the same. The composition, the kit, and the method, according to the present invention, may be used for early diagnosis and confirmed diagnosis of type 1 diabetes mellitus because type 1 diabetes mellitus can be easily diagnosed from a patient sample.
Patent EP-2421997-A2 (EP)
Inventor: EIBISCH HARALD
IPC: C22C23/00
Filed: 2010-02-25
Abstract: Die Erfindung betrifft eine Vorrichtung zur Vorrichtung zur Herstellung von rundlichen Metallpartikeln hoher Größen- und Form-Uniformität aus einer Schmelze sowie Verfahren zur Herstellung von rundlichen Metallpartikeln aus einer hochreaktiven Metallschmelze hoher Größen- und Form-Uniformität mit folgenden Schritten: Schmelzen des metallischen Ausgangsmaterials unter einer Luftabschluss; Transportieren der Metallschmelze in einem geschlossenen Granulierrohr aus dem Schmelzeofen zu mindestens einem Schmelzeauslaß; Austritt der Schmelze aus dem Schmelzeauslaß über einem Drehteller in Form von diskreten Tropfen bis als Schmelzestrahl, der bis zum Auftreffen auf den Drehteller zu Tropfen zerfällt; Leiten eines Schutzgasstroms in den Bereich der aus dem Schmelzeauslass austretenden Schmelze, Auffangen der zu Schmelze auf dem Drehteller in Form von diskreten Schmelzetropfen, Erstarren der Schmelzetropfen zu Granulatpartikeln durch Kontakt mit der kälteren Oberfläche des Drehtellers, und Leiten der Granulatpartikel zur Verpackung/Weiterverarbeitung vom Drehteller.
Patent EP-2473523-A2 (EP)
Inventor: LANGERMANN SOLOMON
IPC: A61K47/48
Filed: 2010-08-31
Abstract: Methods for modulating immune responses in a subject are provided. A preferred embodiment provides methods and compositions for reducing or inhibiting transplant rejection in a subject, preferably a human subject. Transplant rejection can be inhibited or reduced in a subject by administering an effective amount of B7-H4 polypeptide, fragments or fusions thereof to inhibit or reduce the biological activity of an immune cell or to reduce the amounts of proinflammatory molecules at a site of transplant. Th1, Th17 and Th22 cells are exemplary T cells that can be targeted for inhibition by B7-H4 polypeptides, fusion proteins or fragments thereof to inhibit or reduce inflammation.
Patent EP-2510198-A2 (EP)
Title: Verfahren und vorrichtung zum regeln einer dampferzeugung in einer dampfkraftanlage
Inventor: BACKI CHRISTOPH
IPC: F22D5/26
Filed: 2010-09-28
Abstract: Die Erfindung geht aus von einem Verfahren zum Regeln der Erzeugung von Dampf (16) aus Speisewasser (10) in einem Verdampfer (6) einer Dampf kraftanlage, bei dem ein Zustandsregler (30) mehrere Mediumszustände im Verdampfer (6) mit Hilfe eines Beobachters (42) berechnet und daraus einen Speisewassermassenstrom (m s ) als Stellgröße ermittelt. Um eine stabile und genaue Regelung der Dampftemperatur zu erreichen, wird vorgeschlagen, dass der Zustandsregler (30) ein linear-quadratischer Regler ist.
Patent EP-2478085-A2 (EP)
Inventor: SAMSON ARNAUD
IPC: C12M1/18
Filed: 2010-09-10
Abstract: The subject of the present invention is a microplate, or microtitration plate, having an invagination consisting of a continuous peripheral channel making it possible to add thereto, in a single delivery step, a liquid acting as "evaporation curtain". The invention also relates to a device comprising such a microplate, to a manufacturing process and to the use of such a microplate.
Patent EP-2485830-A2 (EP)
Inventor: MILLER OLIVER JON
IPC: G01N1/28
Filed: 2010-10-07
Abstract: La présente invention concerne des systèmes et des procédés pour générer des microgouttelettes avec des concentrations variables d'un soluté particulier à partir d'une solution à concentration fixée.
Patent EP-2425550-A2 (EP)
Inventor: RAMAKRISHNA SUDHIR
IPC: H04B7/26
Filed: 2010-04-27
Abstract: A base station comprising a transmitter for transmitting a downlink frame. The downlink frame comprises a resource allocation region, and the resource allocation region comprises a set of resource allocation messages comprising at least one resource allocation message. Each of resource allocation messages for a particular subscriber station comprises a field including an indicator, to the indicator indicates a number of the resource allocation messages for a particular subscriber station in the resource allocation region.
Patent EP-2424885-A2 (EP)
Title: Compositions et procédés pour le traitement de troubles mettant en jeu une apoptose de cellules épithéliales
Inventor: POLK D BRENT
IPC: A61K38/16
Filed: 2010-04-28
Abstract: La présente invention porte sur des compositions thérapeutiques et prophylactiques pour une utilisation dans le traitement et la prévention de troubles mettant en jeu une apoptose de cellules épithéliales, tels que des troubles gastro-intestinaux (par exemple, une maladie intestinale inflammatoire, la maladie de Crohn ou une colite ulcéreuse), chez un sujet tel qu'un patient humain.
Patent EP-2438079-A2 (EP)
Title: Compositions pour l'administration d'acides nucléiques et procédés pour les utiliser
Inventor: DOWDY STEVEN F
IPC: A61K48/00
Filed: 2010-06-01
Abstract: Cette invention concerne des constructions d'acide nucléique modifiées afin de réduire leur charge anionique nette. Les constructions comprennent des groupes protecteurs de phosphotriester et/ou de phosphothioate. Cette invention concerne également des procédés de préparation et d'utilisation de ces constructions.
Patent EP-2459954-A2 (EP)
Title: Tube d'échangeur thermique
Inventor: SINGH GHANSHYAM
IPC: F28F13/12
Filed: 2010-07-29
Abstract: L'invention concerne un tube d'échangeur thermique (700) dont le corps tubulaire (702) est délimité par une paroi présentant une surface extérieure (704), une surface intérieure (706) et un conduit. Plusieurs dépressions ovales (718) sont formées sur la paroi, prolongeant la surface extérieure (704) et sortant en saillie à travers la surface intérieure (706) de la paroi. Le tube d'échangeur thermique (700) améliore l'efficience du transfert thermique et fonctionne efficacement sur une gamme étendue d'effets du nombre de Reynolds avec de faibles pertes de charge dues au frottement. Le tube d'échangeur thermique (700) est en outre efficient et économique en fonctionnement.
Patent EP-2460034-A2 (EP)
Title: Système de mesure atmosphérique
Inventor: TCHORYK PETER JR
IPC: G01P13/02
Filed: 2010-07-29
Abstract: Linvention concerne un système permettant de déterminer la grandeur et la direction, ou une mesure permettant de les obtenir, dune vitesse (V) dune première partie (17) dune atmosphère (20) grâce à au moins une première partie et une seconde partie dune lumière diffusée (30) générée le long dun faisceau commun de lumière (28) à lintérieur de la première partie (17) de latmosphère (20) et reçue le long de directions linéairement indépendantes à des emplacements relativement éloignés les uns des autres, parmi lesquels au moins un est relativement éloigné dune source (11) du faisceau de lumière (28).
Patent EP-2517324-A2 (EP)
Inventor: GUILLANTON ERWAN
IPC: H02G3/04
Filed: 2010-12-21
Abstract: The cable junction (106) comprises at least two electrical cables (120, 122) extending side by side, each comprising its own independent shield (128, 130) and a front end section (136, 138) where its independent shield (128, 130) is stripped off, a common shield (148) surrounding the front end sections (136, 138) and the independent shields (128, 130) of the cables (120, 122), and a clamping device (162) for clamping the common shield (148) on the independent shields (128, 130). The clamping device (162) comprises internal clamping means (176, 178) for for clamping the common shield (148) on flanks (180, 182) of the independent shield sheaths (128, 130).
Patent EP-2472374-A2 (EP)
Title: Method for providing a ui using motions, and device adopting the method
Inventor: PARK YONG-GOOK
IPC: G06F3/01
Filed: 2010-08-24
Abstract: Provided is a method for providing a UI, in which a common function is mapped to a plurality of motions, and a device adopting the method. The method of the present invention for providing a UI involves performing the function which is commonly mapped to a plurality of motions when a user motion falls within any one of the plurality of motions. Thus, as a plurality of motions for instructing a specific function exists, a user may input a familiar or desired motion, to thereby enable the user to input a command for a function in a more convenient and free manner.
Patent EP-2485614-A2 (EP)
Inventor: MATHIS MICHAEL P
IPC: D06M14/18
Filed: 2010-08-25
Abstract: The present invention is generally directed to a method of treating a folded garment to achieve good alcohol repellency on the innermost layers of the folded garment.
Patent EP-2504805-A2 (EP)
Title: Procédé et dispositif pour guider le conducteur d'un véhicule
Inventor: ERKKILAE KIMMO
IPC: B60W40/02
Filed: 2010-11-23
Abstract: L'invention concerne une solution pour guider le conducteur d'un véhicule. Cette solution consiste à définir un profil cible pour un itinéraire pour déterminer le style de conduite optimal dans différentes parties de l'itinéraire et à recevoir des informations concernant un ou plusieurs paramètres associés au véhicule et la localisation du véhicule au cours d'un événement de conduite. Cette solution consiste en outre à déterminer la conduite réelle par rapport au profil cible au cours de l'événement de conduite et à guider le conducteur du véhicule au moyen d'un dispositif de guidage de conduite au cours de l'événement de conduite d'après le profil cible, un ou plusieurs paramètres associés au véhicule, la localisation du véhicule et la conduite réelle par rapport au profil cible.
Patent EP-2354109-A2 (EP)
Inventor: DENNERT FRANK
IPC: C04B28/18
Filed: 2011-01-21
Abstract: Mineral molding comprises at least one hydrophobing agent exhibiting partially hydrophobic pores and/or capillaries, which are homogeneously distributed in the molding. The water absorption capacity of the mineral molding exhibiting a base surface of 40 cm length, 25 cm width and a height of 8 cm, after 30 minutes of immersion in water at a depth of 1 cm, is 1400-4000 g/m 2>. Independent claims are also included for: (1) a component comprising at least one mineral molding; and (2) producing the mineral molding, comprising (a) mixing at least one liquid phase, at least one mineral binder, at least one hydrophobing agent and at least one pore former to obtain a crude mixture, (b) molding the crude mixture and (c) hardening and/or drying the molded crude mixture to obtain the molding.
Patent EP-2487282-A2 (EP)
Inventor: WINZEN LOTHAR
IPC: D01H4/38
Filed: 2011-12-06
Abstract: The device has a fiber guide channel body (14) fixed in an opening roller housing. The body has a receiving opening (15) for a fiber guide channel insert (27) defining a central fiber guide channel (13) for pneumatically transporting individual fibers. The body is made of a plastics material. The insert is made of a highly abrasion-resistant material as a sleeve-like component fully closed in its annular extent. The fibers are combed by an opening roller from a feed sliver to a spinning rotor revolving at a high rotational speed in a negative pressure-loadable rotor housing.
Patent EP-2368789-A2 (EP)
Inventor: YAMADA HIROSHI
IPC: F02M37/50
Filed: 2011-03-10
Abstract: A motor scooter type vehicule (10) wherein the fuel filter (52) is located on a lateral side of a cylinder unit (54) projectingly provided at a crankcase (53) of a unit swing type engine (28), and is disposed in a space surrounded by a main frame (21) and a rear frame (29) in side view of the vehicle.
Patent EP-2380564-A2 (EP)
Inventor: COULTER IVAN
IPC: A61P37/06
Filed: 2008-04-04
Abstract: An oral composition comprising minicapsules wherein the minicapsules comprise one or more therapeutic or prophylactic substances in a liquid, semi-liquid, or solid core. The minicapsules have release profiles to release the substance in an active form at one or more sites along the gastro-intestinal tract to maximise absorption and/or therapeutic efficiency.
Patent EP-2437016-A2 (EP)
Title: Verfahren zum Trocknen von Hausmüll sowie Trocknertrommel hierzu
IPC: F26B11/04
Filed: 2011-09-30
Abstract: Die Erfindung betrifft ein Verfahren und eine Trocknertrommel (1) zum Trocknen von Hausmüll (14), der eine Leichtstofffraktion (16) und eine Schwerstofffraktion (18) umfasst. Der zu trocknende Hausmüll wird in einer rotierenden Trocknertrommel (1) mit Abwurfschaufeln (42) eingebracht. Ein entlang der Trocknertrommel gerichteter Heißluftstrom (4) transportiert die Leichtstofffraktion durch die Trocknertrommel. Der Innenraum der Trocknertrommel ist durch Schottwände (22) unterteilt, die einen sich durchgängig von der Einlass- (8) zur Auslassöffnung (10) erstreckenden Strömungskanal (17) begrenzen. Um die Verschleißfestigkeit der Trocknertrommel zu erhöhen, ist erfindungsgemäß vorgesehen, dass die Schwerstofffraktion (18) zumindest zu einem Teil an den Abwurfschaufeln (42) der Trocknertrommel (1) vorbei transportiert wird. Dies wird dadurch erreicht, dass sich wenigstens ein im Wesentlichen durchgängiger Schwerstofftransportkanal (32) entlang einer Trommelwand (20) der Trocknertrommel von der Einlassöffnung (8) zur Auslassöffnung (10) erstreckt.
Patent EP-2511021-A2 (EP)
Inventor: KIM SANG WOO
IPC: B21D13/02
Filed: 2011-11-28
Abstract: The present invention provides an apparatus for manufacturing a truss structure using multi-point pins, a method of manufacturing a truss structure using the apparatus, a truss core sandwich panel having the truss structure, and a method of manufacturing the truss core sandwich panel. The apparatus includes a metal plate, clamps, an upper die and a lower die. The clamps hold the metal plate. The upper die has upper multi-point pins which press the metal plate downwards. The lower die has lower multi-point pins which press the metal plate upwards. The metal plate has first and second points that respectively correspond to the upper and lower multi-point pins. The first points are extended downwards by the upper multi-point pins, and the second points are extended upwards by the lower multi-point pins. Thereby, many symmetrical sides are formed in the truss structure, thus increasing the stability of the truss structure.
Patent EP-2460916-A2 (EP)
Inventor: KAWAI MOTOHIRO
IPC: D01H1/241
Filed: 2011-12-02
Abstract: A draft device in the prespinning process includes a bottom roller whose roller gauge is adjustable, a belt for driving the bottom roller, a tension pulley that can urge the belt downward, a support member for supporting the tension pulley, an urging member that can urge the support member downward so as to provide a desired tension to the belt through the tension pulley and an urging force releasing device for releasing an urging force of the urging member. The urging force releasing device is provided above the tension pulley so as to be operable above the tension pulley.
Patent EP-2531035-A2 (EP)
Title: Composition herbicide synergique contenant du penoxsulam et du flazasulfuron
Inventor: HUFNAGL ANDREA
IPC: A01N47/36
Filed: 2011-02-01
Abstract: La présente invention a trait à une composition herbicide contenant (a) du penoxsulam et (b) du flazasulfuron qui permet un contrôle synergique des mauvaises herbes sélectionnées.
Patent EP-2542582-A2 (EP)
Inventor: LI YINGCHUN
IPC: C07K16/18
Filed: 2011-02-28
Abstract: DLL4 binding proteins are described herein, including antibodies, CDR-grafted antibodies, humanized antibodies, and DLL4 binding fragments thereof, proteins that bind DLL4 with high affinity, and DLL4 binding proteins that neutralize DLL4 and/or VEGF activity. The DLL4 binding proteins are useful for treating or preventing cancers and tumors and especially for treating or preventing tumor angiogenesis.