baber/WOPTO huggingface dataset:
Patent DK-1481966-T3 (DK)
Inventor: OJIMA KATSUJI
IPC: A61K31/44
Filed: 2003-03-04
Granted: 2011-10-24
Abstract: Arylamide derivatives (I) are new. Arylamide derivatives of formula (I) and their salts are new. [Image] X : optionally substituted lower alkylene or alkenylene; G 1O, S or NH; G 2C or N; R aH, halo or optionally substituted alkyl, cycloalkyl or alkoxy; R 1optionally protected or substituted amidino; R 2NR 3R 4, NR 5YNR 6R 7 or a group of formula (i); R 3H, amino protecting group, a group of formula (ii) or optionally substituted cycloalkyl or alkenyl; W : a bond or optionally substituted alkylene; Y coptionally substituted 2-4C alkylene; Y c1optionally substituted 1-4C alkylene; R 7bH, amino protecting group, a group of formula (iii) or optionally substituted alkyl, cycloalkyl or alkenyl; Z : optionally substituted lower alkylene or alkenylene; G 3O, S, NH or bond; G 5C or N; R bH, halo or optionally substituted alkyl, cycloalkyl or alkoxy; R 8para or meta to G 3 and is optionally protected or substituted amidino; R 4-R 6H, amino protecting group or optionally substituted alkyl, cycloalkyl or alkenyl; Y : optionally substituted 2-6C alkyelene or 3-6C alkenylene; R 7R 4 or (iii); Y aoptionally substituted 2-4C alkylene; Y boptionally substituted 1-4C alkylene; G 4C or N; R 7aalkyl (optionally substituted by at least one CN, NO 2, halo, sulfo, phosphoryl, lower alkenyl, lower alkoxy, heterocyclyl, cycloalkyl, lower alkylidene, SH, amidinophenylaryloxy, aryloxy, lower alkylthio, lower alkylsulfinyl, lower alkylsulfonyl, lower alkylcarbamoyl, lower alkylsulfonylamino, lower alkylaminosulfonyl, lower carboxylalkenyl, lower alkoxyimino or optionally protected hydroxyl, amino, carbamoyl, hydrocarbamoyl, aminosulfonyl, cyclic amino or lower alkylamino), (iii) or optionally substituted phenyl, cycloalkyl or alkenyl, provided that when G 1 = NH, then X = optionally substituted 3-6C alkylene or alkenylene. [Image] ACTIVITY : Fungicide. In cytotoxicity assays, 4-[2-[1-(3-[4-[amino(imino)methyl]phenoxy]propyl)-4-piperidinyl]ethoxy]benzamidine hydrochloride (Ia) had an IC 50 value for Candida albicans TIMM1623 of 0.0039 mu g/ml. MECHANISM OF ACTION : None given.
Patent DK-1490052-T3 (DK)
Inventor: BREITENBACH ARMIN
IPC: A61K31/381
Filed: 2003-12-24
Granted: 2007-10-01
Abstract: The invention relates to a polymer matrix suitable for the transdermal administration of rotigotine [(-)-5, 6, 7, 8-tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-1-naphtol], containing a matrix for the transdermal administration of rotigotine [(-)-5, 6, 7, 8-tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-1 naphtol], containing a matrix polymer which is supersaturated with a rotigotine base. Said polymer matrix is characterised in that the part of the rotigotine which is not dissolved in the matrix polymer is dispersed in the matrix polymer as amorphous particles having a maximum mean diameter of 30 mum, and the matrix is free of solubilisers, crystallisation inhibitors and dispersants. The invention also relates to a flat device for the transdermal administration of rotigotine, containing the above-mentioned, preferably silicon-based polymer matrix which is supersaturated with rotigotine, and a rear layer which is impermeable to the active ingredient.
Patent DK-1536999-T3 (DK)
Inventor: GRUENBAUM JOERG
IPC: B61C17/04
Filed: 2003-09-11
Granted: 2009-03-09
Abstract: The invention relates to a rail vehicle (SCH) having an emergency exit (NOT) located at the front (FRO), whereby a driver's console (FAP) and a driver's seat (FAS) are mounted in an end area (END) of the rail vehicle (SCH) that is located in front of the emergency exit (NOT). The emergency exit (NOT) is located essentially in the middle of the front (FRO), and the driver's seat (FAS) and at least one middle section of the driver's console (FAP) are mounted in a manner that enable them to be moved toward a side wall (SEI) out of a middle driving position (Fig. 1) located in front of the emergency exit (NOT) and into an emergency position (Fig. 2). When the driver's seat and the at least one middle section of the driver's console are in the emergency position (NOP), an escape space (FLR) is formed in the front end area (END). This escape space corresponds at least to the width of the emergency exit (NOT) and runs parallel to the longitudinal extension of the rail vehicle.
Patent DK-1496341-T3 (DK)
Inventor: STORM RALF
IPC: G01F1/84
Filed: 2004-05-19
Granted: 2011-03-14
Abstract: A Coriolis mass flow meter has a measurement tube (1) with vibrator (2) and vibration sensor (3) and controller (4) and control signal path with vibration sensor (10) amplifier (11) and analogue to digital converter (12) connecting the excitation signal path directly to the processor (5) from immediately before the vibrator. Includes INDEPENDENT CLAIMs for the procedures used by the meter and for equipment with multiple multiplexed excitation and control signal paths.
Patent DK-1592853-T3 (DK)
Inventor: SORIANO HOYUELOS ESTHER
IPC: D04H1/4209
Filed: 2004-02-04
Granted: 2008-08-25
Abstract: The invention relates to a mineral wool panel of increased structural strength, of the type of those used for the manufacture of air ducts, particularly airconditioning ducts, which are composed of a central core made of mineral wool, especially glass wool, coated on both faces with coatings, said core incorporating a web on the face located on the inside of the duct obtained, the panel of the invention being characterized in that it comprises a core ( 1 ) the surface faces of which, both the inner face and the outer face, each incorporate a respective web ( 2 ) extending over the totality of said faces, the two webs ( 2 ) being bonded to the surfaces of the core ( 1 ) by means of binders that can cure through the action of heat.
Patent DK-1612146-T3 (DK)
Inventor: YUYAMA SHOJI
IPC: B65B5/08
Filed: 2004-03-25
Granted: 2009-11-16
Abstract: The present invention prevents tablets from bouncing in a tablet drop guide path so that dropping time can be shortened so as to be ready in time for packing. In a tablet packing apparatus provided with a tablet drop guide path 12 that guides tablets to a packing unit, the tablets drop obliquely downward from each of tablet outlets 10 of tablet feeders 8 provided in an up and down direction in a manner of multistage shelf, wherein a bounce preventing member 14 is provided in a position opposing to the tablet outlets or the tablet drop guide path, and wherein the bounce preventing member 14 is obliquely provided so that it recedes from the tablet outlets 10 toward the lower end.
Patent DK-1618046-T3 (DK)
Inventor: PASBRIG ERWIN
IPC: B65D75/36
Filed: 2004-04-05
Granted: 2007-05-29
Abstract: A tropical blister pack (10) having a heat-shaped plastic blister base section (12) and a covering foil (16) over the blisters (14) and against the package edge (20), sealed against the reverse side of the blister base, is new. The base is covered by a further foil (18) as a sealing trough. A tropical blister pack (10) having a heat-shaped plastics blister base section (12) and a covering foil (16) over the blisters (14) and against the package edge (20), sealed against the reverse side of the blister base, is new. The base is covered by a further foil (18) as a sealing trough. Between the under foil and the blister base there is a peelable varnish as a hot seal applied at a rate of 2-20 g/m 2> and preferably 7-15 g/m 2>, or a peelable plastics film with a thickness of 10-40 Microm and preferably 15-30 Microm, or a peelable plastics coating at a rate of 5-40 g/m 2> and preferably 7-20 g/m 2>. When the lower shrouding has been peeled away, the blister contents can be seen. The plastics material of the blister base incorporates a barrier against the entry of water vapor or gas.
Patent DK-1654178-T3 (DK)
Inventor: DEVINE DANIEL
IPC: B65D83/04
Filed: 2004-08-04
Granted: 2009-01-19
Abstract: A package assembly 10 for the storage and distribution of a plurality of stacked mints 12 is provided. The package assembly 10 includes a cylindrical outer shell 14 including a shell sidewall 16 , a shell bottom surface 18 , and a shell open top 20 . The shell sidewall 16 includes a sidewall inner surface 22 and a sidewall outer surface 24 . A vertical control slot 28 is formed in the shell sidewall 16 , the vertical control slot 28 having a control slot height 40 and a control slot width 42 . At least one retention protrusion 78 is formed onto a slot side edge 34 such that the control slot width 42 is reduced in the location of the at least one retention protrusion 78 . A cylindrical inner insert 26 including an insert sidewall 44 , an insert top surface 46 , and an insert open bottom 48 , is formed to house the plurality of stacked mints 12 . The cylindrical inner insert 26 is positioned within the cylindrical outer shell 14 such that the insert open bottom 48 faces the shell bottom surface 18 . A control pad 52 is formed onto and protrudes outwards from the insert sidewall 44 . The control pad 52 is positioned within the vertical control slot 28 and is movable such that the cylindrical inner insert 26 can be moved between a closed position 68 and an open position 70 . The control pad 52 has a control pad width 54 such that said control pad 52 engages the at least one retention protrusion 78 when in the closed position 68 and such that the cylindrical inner insert 26 is resisted from moving into the open position 70 . A dispensing chamber 72 is formed in the insert sidewall 44 adjoining the insert top surface 46 . The dispensing chamber 72 is covered by the shell sidewall 16 when the cylindrical inner insert 26 is in the closed position 68 . The dispensing chamber 72 is positioned outside the cylindrical outer shell 14 when the cylindrical inner insert 26 is in the open position 70 . The dispensing chamber 72 has a dispensing chamber height 74 sufficient to allow one of the plurality of stacked mints 12 to be removed from the cylindrical inner insert 26.
Patent DK-1690805-T3 (DK)
Inventor: BURCHARD JOERN
IPC: B65D51/24
Filed: 2005-02-11
Granted: 2009-01-05
Abstract: A mug of tea sold from a mobile vending station is prepared by the release of hot water into a mug containing a tea bag suspended from a draw string under a plastic lid. The lid has a stepped central detent and an aperture through which the tea bag may be withdrawn onto the step when the tea has brewed to the desired concentration.
Patent DK-1723829-T3 (DK)
Inventor: KAULBERG THOMAS
IPC: H04R25/00
Filed: 2005-02-28
Granted: 2011-07-18
Abstract: The invention regards a method for noise reduction in an audio device whereby an electrical and/or digital signal which represents sound is routed simultaneously through:-a signal analysis path, and-a signal processing path wherein the signal amplification is individually controllable in specific frequency bands by attenuation values derived from the signal analysis path, whereby the signal in the signal analysis path is routed simultaneously through:-a first detector which identifies the presence of speech indicators in the overall signal, and-a second detector which in a predefined number of frequency bands detects the modulation amplitude, and-where attenuation values in each of the predefined frequency bands are calculated based on the combined results of the first detector and the modulation amplitude in the specific frequency band detected by the second detector,-where the attenuation values in the predefined number of frequency bands are routed to the signal processing path in order to attenuate the signal level in corresponding frequency bands.
Patent DK-1812207-T3 (DK)
Inventor: MOELLER LARRY M
IPC: B25C1/00
Filed: 2005-10-10
Granted: 2011-01-03
Abstract: A modular magazine assembly in a fastener-driving tool having a nosepiece includes a first magazine housing portion secured to the tool and at least partially defining a chamber for fasteners. An extension portion is configured for releasable attachment to the first magazine housing portion. Upon assembly of the extension portion, a resulting large capacity magazine is defined and dimensioned to accommodate at least two fastener strips.
Patent DK-1809320-T3 (DK)
Inventor: MARGOLIN ALEXEY L
IPC: A61K38/46
Filed: 2005-10-14
Granted: 2010-11-15
Abstract: The present invention relates to compositions for the treatment of conditions, including pancreatic insufficiency. The compositions of the present invention comprise lipase, protease and amylase in a particular ratio that provides beneficial results in patients, such as those afflicted with pancreatic insufficiency. This invention also relates to methods using such compositions for the treatment of pancreatic insufficiency.
Patent DK-1915767-T3 (DK)
Inventor: HENDRIX JULES DR
IPC: H01J35/10
Filed: 2006-08-18
Granted: 2010-02-08
Abstract: The cooling arrangement (100) has firing path (11) and storage part (15) in rotating anode (10). The electron current meets on the firing path. Fluid (13) is present between firing path and storage part. The storage part forms simultaneously a condensation area (16) as well as evaporation area on the firing area. The evaporation area vaporizes the fluid as vapor (18) to arrive at condensation area to condense and return back to the firing path as condensate (22) due to the centrifugal forces of the rotating anode.
Patent DK-2173371-T3 (DK)
Inventor: HIGAZI ABD AL-ROOF
IPC: A61K38/08
Filed: 2008-07-24
Granted: 2012-02-06
Abstract: The present invention relates to isolated 18-mer peptides corresponding to amino acid residues 369-386 of human plasminogen activator inhibitor 1 (PAI-1) and fragments thereof, compositions comprising same, and uses thereof for treating thromboembolic diseases and pathological conditions associated with neurological damage.
Patent DK-2219954-T3 (DK)
Inventor: AGELING WERNER
IPC: B65B11/12
Filed: 2009-10-08
Granted: 2012-04-10
Abstract: A packaged unit includes a cluster of products and a shrink film that secures the products to each other. The shrink film is wrapped around the cluster, thereby forming a lateral opening that would otherwise result in a shrink eye. A closure formed by placing a portion of the shrink film against the cluster at in the region of the lateral opening forms a closed surface with overlapping fold regions of the shrink film, thus avoiding the shrink eye.
Patent DK-2620153-T3 (DK)
Inventor: YAN GUANGMEI
IPC: A61P25/00
Filed: 2011-07-08
Granted: 2018-07-23
Abstract: A 5α-androstane-3β,5,6β-triol injection and its preparation are disclosed. The injection uses hydroxypropyl-β-cyclodextrin as a solubilizing agent and the active ingredient is present at a weight ratio of 1-20:40-500 to the hydroxypropyl-β-cyclodextrin. The injection may also comprise, by weight, 1-100 parts of at least one isotonic adjusting agent, 0-200 parts of at least one freeze drying filler, and 0-2000 parts of at least one solvent. The preparation method comprises dissolving hydroxypropyl-β-cyclodextrin solution, 5α-androstane-3β,5,6β-triol and at least one additional soluble excipient in water for injection in sequence to obtain a raw injection solution, and subjecting the raw injection solution to decolorization, depyrogenation, filtration and sterilization to obtain the injection. Drying the filtrate yields a solid for injection.
Patent DK-2694043-T3 (DK)
Inventor: HIROSE TSUYOSHI
IPC: A61K31/00
Filed: 2012-04-04
Granted: 2018-01-15
Abstract: The present invention provides a medicament having a wider treatment spectrum, causing a fewer side effects and superior in tolerability and safety, as compared to known typical antipsychotic agents and atypical antipsychotic agents. The present invention related to a medicament containing (I) a compound which is 7-[4-(4-benzo[b]thiophen-4-yl-piperazin-1-yl)butoxy]-1H-quinolin-2-one or a salt thereof, and (II) one or more antianxiety drugs, in combination.
Patent DK-3072524-T3 (DK)
Inventor: MAZMANIAN SARKIS K
IPC: A61K35/741
Filed: 2011-10-06
Granted: 2018-04-09
Abstract: Provided is a method and a composition for improving behavioral performance in an individual comprising identifying an individual in need of treatment, and providing such an individual a composition comprising bacteria within the genus Bacteroides.
Patent DK-3419205-T3 (DK)
Inventor: SUZUKI TAKASHI
IPC: H04L1/18
Filed: 2007-02-14
Granted: 2020-05-04
Abstract: A method for Discontinuous Reception ('DRX') operation, comprising waking up a receiver at a radio frame if the radio frame number is equal to a radio frame offset plus N times a DRX interval, wherein N is an integer greater than or equal to zero is described.
Patent DK-0387507-T3 (DK)
Inventor: KRAKER ALFRED
IPC: H03H17/06
Filed: 1990-01-26
Granted: 1994-06-27
Abstract: Conversion of the sampling rates of digital signals by means of an interpolation computer which calculates from interpolation points derived from input sample values and from time differences between input and output sampling times, measured by means of a timer, the output sample values. Difference structure computers form from the interpolation points special difference structures of second, fourth and further even-numbered orders, from which the sample values are obtained in accordance with the Everett interpolation formula.
Patent DK-0378255-T3 (DK)
Inventor: VANDENBERK JAN
IPC: A61K31/519
Filed: 1990-01-03
Granted: 1994-05-24
Abstract: Novel 2-aminopyrimidinone derivatives of formula <CHEM>  wherein R<1> is <CHEM>  R<3> is hydrogen or C1-6alkyl;  R<4> is hydrogen, C1-6alkyl or substituted C1-6alkyl; R<5> is hydrogen, C1-6alkyl, C1-6alkylaminocarbonyl, Ar-aminocarbonyl, C1-6alkylcarbonyl or Ar-carbonyl; R<6> is hydrogen, C1-6alkyl or Ar-C1-6alkyl; or R<5> and R<6> taken together is -CH2-CH2-, -CH2-CH2-CH2-, -CH=CH-, -CH=N-, -N=CH- or -N=CH-CH2-; the pharmaceutically acceptable acid addition salts and possible stereochemically isomeric forms thereof; pharmaceutical compositions containing such compounds as an active ingredient and methods of preparing said compounds and pharmaceutical compositions.
Patent DK-0419165-T3 (DK)
Inventor: JANSSEN HERWIG
IPC: A61K47/22
Filed: 1990-09-17
Granted: 1994-05-02
Abstract: An ophthalmic formulation comprising a salt of sepazonium or a similar imidazolium compound as a preservative is provided.
Patent DK-0461554-T3 (DK)
Inventor: CANOVA LUCIANO DR
IPC: C07C43/21
Filed: 1991-06-07
Granted: 1994-01-31
Abstract: The fluidity at low temperatures of compositions based on liquid refinery hydrocarbons can be improved by adding thereto substituted [l4]-metacyclophanes, e.g., those obtained from the condensation reaction of a resorcin with an aldehyde, followed by a reaction with halides or organic acids or alkyl halides.
Patent DK-0506919-T3 (DK)
Inventor: HENNEUSE HENRY
IPC: E21B47/00
Filed: 1991-10-17
Granted: 1995-09-04
Abstract: PCT No. PCT/FR91/00812 Sec. 371 Date Aug. 7, 1992 Sec. 102(e) Date Aug. 7, 1992 PCT Filed Oct. 17, 1991 PCT Pub. No. WO92/07162 PCT Pub. Date Apr. 30, 1992.A motorised rotary swivel for driving drill pipe in rotation is disclosed. The swivel includes a measuring unit for measuring a dynamometric behavior of the drill pipe which is mounted adjacent to the output of the motor between the motor and a torque wench assembly.
Patent DK-0558834-T3 (DK)
Inventor: JOUWSMA WIJBREN
IPC: G01F15/12
Filed: 1992-12-14
Granted: 1996-07-29
Abstract: Device for measuring pressure differences or mass portions in a fluid flow - gas or liquid - and/or for implementing processes for mixing fluids, whereby when in use the fluid flows into the device, then passes a part therein where the fluid flow is laminar and the flow measurement is made, and finally flows out of the device, whereby the device has a turbulence filter which is integrated therein, with a settling chamber behind it. The fluid then first flows through that filter, so that a laminar flow leads to the flow measuring element. <IMAGE>
Patent DK-0541410-T3 (DK)
Inventor: BILLON THIERRY
IPC: H04L12/43
Filed: 1992-10-05
Granted: 1996-06-03
Abstract: The installation usable in particular in accordance with the GSM standard, comprises a master station (10) equipped with time-division multiplex links with slaves (14). The slave stations constitute at least one group and each have a cross-connection unit which is controllable so as either to insert a specified channel of order i into the respective station, or route it while passing the station. Each cross-connection unit (2) and the master station contain an identifier of a signalling channel assigned to the cross-connection unit; the cross-connection units of all the slave stations contain means of associating all the pairs each consisting of counterpart channels on two links so as to pass all the stations and carry out complete routing; the master station is devised so as to transmit, over the signalling channel of each respective slave station, the order of insertion of the channel or of the channels to be assigned to the station. <IMAGE>
Patent DK-0562504-T3 (DK)
Inventor: CONNEMANN JOOSTEN DR ING
IPC: C07C69/52
Filed: 1993-03-22
Granted: 1996-03-04
Abstract: Production of lower alkyl esters of higher fatty acids from an oil phase and lower alcohols by catalytic transesterification at reaction temperatures of up to 100 DEG  C. in the presence of an alkaline catalyst, includes a) introducing a mixture of oil phase, alcohol and catalyst at reaction temperature into the top of a first reactor column, at a rate of flow which is lower than the sinking rate of the glycerine separated from the reaction mixture, b) the reaction mixture is passed into a second reactor for further transesterification, c) the thus obtained reaction mixture is further freed of glycerine in an initial separating stage by means of a short-term washing, d) the reaction mixture is passed into a third reactor with addition of further alcohol and catalyst, and at a rate of flow conforming to the first stage of the process, e) the reaction mixture is further transesterified, f) reaction product is freed of the remaining methanol, glycerine, soaps formed and catalyst in a second separating stage, under addition of an aqueous extraction buffer solution, and g) the reaction mixture is freed of lower alcohols by stripping, washed with suitable extraction and washing solutions and dried.
Patent DK-0577107-T3 (DK)
Inventor: HOERMANN STEPHAN DIPL-PHYS
IPC: E06B9/58
Filed: 1993-06-30
Granted: 1998-09-28
Abstract: The invention relates to a guide rail (1) of a rolling shutter door, having a number of securing devices which are distributed at intervals over the longitudinal extent of said rail and each have a claw upper part (3). In adaptation to different spacings, having dimensions dependent on the respective rolling-shutter-door reel thickness, of the guide rails from the border surface (4) enclosing the door opening, said claw upper part is provided with an underlay with the aid of underparts (2) which can be optionally introduced and stacked and each of which forms the securing means for a correspondingly dimensioned sheet-metal strip which can be clipped on and covers the respective gap, towards the door-opening side, between guide rail and border surface. <IMAGE>
Patent DK-0576090-T3 (DK)
Inventor: THOMSON JAMES
IPC: G01T1/203
Filed: 1993-06-21
Granted: 2001-11-12
Abstract: An adhesive plastic scintillator which can be attached onto a solid support medium, either by melting it in and/or on a solid support medium when the plastic scintillator is capable of being changed between solid and liquid phases, whichever is desired, by temperature control, or by deposition from a solution of said adhesive plastic scintillator. The plastic scintillator comprises fluorescent substances and optionally energy transfer compounds for converting radiation energy into light energy. The plastic scintillator remains transparent upon transition from the liquid to the solid state, and upon the same transition adheres to the solid support medium.
Patent DK-0586013-T3 (DK)
Inventor: CHIURLO PAOLO
IPC: C03C1/00
Filed: 1993-08-27
Granted: 1998-04-06
Abstract: The preparation of objects, in particular optical components and/or devices, is described using, as precursors of optical materials, amorphous monolithic aerogels for high-precision mechanical machining.