baber/WOPTO huggingface dataset:
Patent EP-0820982-A1 (EP)
Inventor: YOKURA SUSUMU
IPC: C07D295/112
Filed: 1996-04-12
Abstract: 4-amino-5-oxy-2,6,6-trimethyl-2-cycloheptene compounds
represented by the following general formula:
 
(wherein R 1  and R 2  each independently represent a hydrogen
atom, an alkyl group which may have a substituent, or a
phenyl group which may have a hydroxyl group, lower
alkoxy group, amino group, nitro group, carboxyl group,
lower alkoxycarbonyl group or halogen atom, or R 1 , R 2  and
the nitrogen atom together represent a saturated nitrogen
heterocyclic group; R 3  represents a hydrogen atom, a
lower alkyl group or a lower aliphatic acyl group); and W
represents an oxo group, oxime group or oxime ether group;
and their pharmacologically acceptable salts and
solvates. 
     The 4-amino-5-oxy-2,6,6-trimethyl-2-cycloheptene
compounds exhibit an effect against rat peripheral
arterial occlusion models, spontaneous hypertensive rats
and histamine-induced airway contraction models, and are
thus useful as remedy for hypertension, peripheral 
arterial occlusion and bronchial asthma.
Patent EP-0822813-A1 (EP)
Inventor: EVENDEN JOHN
IPC: A61K31/445
Filed: 1996-04-23
Abstract: L'invention se rapporte à une combinaison d'un premier composant (a) qui est un inhibiteur de fixation de 5-HT et d'un second composant (b) qui est un antagoniste de 5-HT1A sélectif de la formule générale (I) dans laquelle R1 représente n-propyle ou cyclobutyle, R2 représente isopropyle, butyle tertiaire, cyclobutyle, cyclopentyle ou cyclohexyle, R3 représente hydrogène; R4 représente hydrogène ou méthyle; cet antagoniste 5-HT1A étant un (R)-énantiomère se présentant sous la forme d'une base libre. L'invention se rapporte également aux sels pharmaceutiquement acceptables de cette combinaison, à sa préparation, aux formulations pharmaceutiques la contenant, à son utilisation et au procédé de traitement de troubles affectifs tels que la dépression, l'anxiété et les troubles obsessionnels impulsifs au moyen de cette combinaison, ainsi qu'à un nécessaire contenant cette combinaison.
Patent EP-0826256-A1 (EP)
Inventor: STEGMUELLER BERNHARD
IPC: H01S5/12
Filed: 1996-05-03
Abstract: It is possible with the process of the invention to produce MRCW high-temperature laser diodes with coupled optical waveguides in four epitaxy steps, in which preferably the first and last two epitaxies are performed virtually immediately after one another and an interruption is needed only to produce a grid. It is possible to make other components, e.g. photodiodes, using the process of the invention.
Patent EP-0832200-A1 (EP)
Inventor: FOSTER W BARRY
IPC: C12N9/64
Filed: 1996-05-21
Abstract: Provided by the present invention are novel methods of factor IX protein recovery and purification, making use of anion exchange chromatography heparin-like resins, hydroxyapatite and immobilized metal affinity chromatography.
Patent EP-0830427-A1 (EP)
Inventor: HUGHES O RICHARD
IPC: C08L71/00
Filed: 1996-06-03
Abstract: L'invention porte sur des composites polymères avec charge élevée, moulables par injection, présentant une grande stabilité dimensionnelle à des températures supérieures à celle de la transition vitreuse de la matrice. La température de déformation à chaud des composites se rapproche de celle de fusion cristalline de la matrice. Le composite comporte une matrice polyaryléthercétone et au moins deux types de matière de charge, offrant chacune des propriétés uniques en leur genre. La première matière de charge est une charge de fibre renforçante, apportant des caractéristiques de résistance mécanique et de rigidité. La seconde est une matière de charge immobilisante non thermoplastique qui immobilise la partie amorphe du polymère polyaryléthercétone partiellement cristallin et procure une résistance à une déformation à haute température. Nonobstant ses propriétés de résistance mécanique et thermique, ce composite reste moulable par injection et, partant, susceptible d'être produit à de faibles coûts de fabrication.
Patent EP-0853484-A1 (EP)
Inventor: DOOLEY COLETTE T
IPC: C07K5/087
Filed: 1996-06-06
Abstract: The present invention provides novel opioid peptides. Disclosed are opioid peptides having the general structure Ac-Phe-Arg-Trp-Trp-Tyr-Xaa-NH2 (SEQ ID No. 1); Ac-Arg-Trp-Ile-Gly-Trp-Xaa-NH2 (SEQ ID No. 2); Trp-Trp-Pro-Lys/Arg-Hisz-Xaaz-NH2 (SEQ ID No. 222); Tyr-Pro-Phe-Gly-Phe-Xaa-NH2 (SEQ ID No. 5); (D)Ile-(D)Met-(D)Ser-(D)Trp-(D)Trp-Glyn-Xaa-NH2 (SEQ ID No. 6); and (D)Ile-(D)Met-(D)Thr-(D)Trp-Gly-Xaa-NH2 (SEQ ID No. 7). Within each genus, Xaa is substituted by a specific amino acid. The invention also relates to an opioid peptide having general structure Tyr-A1-B2-C3-NH2 (SEQ ID No. 8), wherein A is D-Nve or D-Nle, B is Gly, Phe, or Trp, and C is Trp or Nap. Also included within the invention are opioid compounds of the general structure MexHyN-Tyr-Tyr-Phez-Proz-NH2 (SEQ ID No. 221) which are peptides modified by permethylation, perallylation, perethylation, perbenzylation or pernaphthylation and which be further modified by reduction.
Patent EP-0837631-A1 (EP)
Inventor: WHITTEMORE MARILYN S
IPC: A01N43/36
Filed: 1996-05-28
Abstract: L'invention se rapporte à des compositions microbicides qui comprennent: (a) de la 2-(thiocyanométhylthio)benzothiazole et (b) un composé hétérocyclique N-alkyle de formule (I). Dans ladite formule, la variable 'n' a une valeur comprise entre 5 et 17, et l'anneau hétérocyclique qui est défini par (1) est un anneau substitué ou non substitué ayant entre 4 et 8 éléments. Les constituants (a) et (b) sont présents dans des proportions combinées efficaces pour contrôler la croissance d'au moins un micro-organisme. On décrit par ailleurs des procédés qui permettent de contrôler la croissance des micro-organismes sur différents substrats ou dans des systèmes aqueux. On décrit enfin l'application industrielle de ce type de composition microbicide dans l'industrie du cuir, l'industrie forestière, l'industrie du papier, l'industrie textile, l'agriculture, l'industrie du revêtement et les techniques des systèmes aqueux.
Patent EP-0841999-A1 (EP)
Inventor: SCHULTZ ROBERT E
IPC: B21D13/04
Filed: 1996-07-17
Abstract: On décrit une machine (90) destinée à former un panneau (50) métallique de toiture, de longueur indéterminée, à partir d'une bande (96) alimentatrice, de largeur uniforme, d'une tôle présentant une paire de bords (98, 100) longitudinaux droits et parallèles. Cette machine (90) présente une série de postes (102) de formage, espacés, possédant chacun des rouleaux supérieurs et inférieurs de mise en forme, entre lesquels on fait passer la bande (96) de tôle, de manière à donner à celle-ci une forme désirée qui soit uniforme sur sa longueur après sa sortie de la machine. Un poste (104) à estamper, placé sur le trajet de ladite bande (96) avant la série de postes (102) de formage, est efficace pour former des impressions (74) linéaires dans cette bande (96), lesquelles sont transversales par rapport aux bords (98, 100) longitudinaux de la bande (96) et sont limitées chacune en extension latérale, de manière à ce que la série suivante de rouleaux de mise en forme ne heurtent pas ces impressions.
Patent EP-0843671-A1 (EP)
Inventor: COCKERILL GEORGE STUART
IPC: A61P43/00
Filed: 1996-07-11
Abstract: The invention is directed toward substituted heteroaromatic compounds which are protein tyrosine kinase inhibitors, in particular to substituted quinolines and quinazolines. Methods for their preparation, pharmaceutical compositions including such compounds and their use in medicine, for example in the treatment of psoriasis, fibrosis, atherosclerosis, restenosis, auto-immune disease, allergy, asthma, transplantation rejection, inflammation, thrombosis, nervous system diseases, and cancer.
Patent EP-0837895-A1 (EP)
Inventor: EVANS RANDALL K
IPC: C08L23/16
Filed: 1996-07-08
Abstract: A compound comprising a blend of polypropylene with the reaction of a functionalized polypropylene and polyether amine in which the polyetheramine is grafted into the functionalized polypropylene in a customary mixing apparatus is disclosed. The blend may include an elastomer such as EP rubber and/or a filler such as glass. A process for producing the reaction product of the functionalized polypropylene and the polyether amine by melting with polypropylene in a customary mixing apparatus is also disclosed. Blends of the present invention are advantageously useful to prepare paintable automotive body parts.
Patent EP-0858522-A1 (EP)
Inventor: FERGUSON JAMES
IPC: D01F6/18
Filed: 1996-09-12
Abstract: A method of manufacture of solid-walled hollow polymeric fibres comprises the steps of dissolving polymeric material in a suitable solvent liquid to form a dope solution (44), extruding the dope solution through an aperture in a spinneret (41) to form a narrow jet of liquid, injecting a coagulant (46) through an aperture (53) in the centre of the liquid dope jet as it leaves the spinneret, directing the jet through an air gap into a coagulant bath containing a further coagulant; and directing the fibre through a drawing bath to reduce the diameter; each coagulant solution being a mixture of a coagulant liquid capable of causing gelation and solidification of the liquid dope jet and between 20 % and 80 % of the solvent liquid.
Patent EP-0851807-A1 (EP)
Title: Procede et dispositif de thermoretraction electrique
Inventor: KATZ ODED
IPC: B29C65/00
Filed: 1996-09-18
Abstract: La présente invention concerne un procédé permettant de raccorder un premier tuyau (P1) en matière plastique à un second tuyau (P2) en un matériau qui n'adhère pas bien à la matière plastique. Ce procédé consiste à utiliser un manchon de thermorétraction électrique (2) en matière plastique adhérant bien à la matière plastique du premier tuyau. Ce manchon est pourvu, sur la face interne de l'une de ses extrémités permettant de recevoir le premier tuyau (P1), d'un premier enroulement (6) de fil électrique chauffant. Ce manchon est également pourvu, sur la face interne l'extrémité opposée permettant de recevoir le second tuyau (P2), d'un second enroulement (7) de fil électrique chauffant. L'extrémité opposée du manchon est garnie de matériau de liaison capable de produire, sous l'effet de la chaleur, une bonne liaison entre les matières du manchon (2) et le second tuyau (P2). Une fois que les tuyaux ont été introduits aux deux extrémités du manchon, l'application d'un courant électrique aux deux enroulements provoque l'adhésion de la première extrémité du manchon sur le premier tuyau (P1) par thermorétraction électrique, et l'adhésion de la seconde extrémité du manchon sur le second tuyau (P2) sous l'effet conjugué de la thermorétraction électrique et du comportement du matériau de liaison.
Patent EP-0861082-A1 (EP)
Inventor: WEISZ PAUL B
IPC: A61K35/32
Filed: 1996-09-17
Abstract: Disclosed are methods of therapy applicable to pathologies that involve loss of integrity of tissue and organ membranes that lead to abnormal permeation of proteinic and other agents and their elimination or penetration of other anatomical functions. Such deficiencies are associated directly or indirectly, for example, with inflammatory diseases, with diabetes and others. The therapeutic method involves administering to the membrane in need of treatment a therapeutic amount of an oligosaccharide, preferably a cyclic oligosaccharide, having up to about 10 sugar units per molecule and having at least 1.4 anionic substituents per sugar unit. The anionic substituents are preferably the residues of strong acids.
Patent EP-0886913-A1 (EP)
Inventor: BROWN ANTHONY KEVIN DALE
IPC: H03H11/18
Filed: 1996-11-20
Abstract: Un amplificateur différentiel hyperfréquence comprend des premier et second dispositifs CMOS adaptés, chacun étant connecté par la source à un noeud de polarisation commun, par la grille à un port d'entrée pour recevoir un signal d'entrée différentiel et par les drains à un port de sortie, pour émettre un signal différentiel de sortie. Des condensateurs Miller de chaque dispositif assurent la rétroaction nécessaire entre les ports d'entrée et de sortie, pour décaler de 45° la phase du signal différentiel de sortie, par rapport à la phase du signal différentiel d'entrée, à une fréquence prédéterminée. Le point de fonctionnement des dispositifs NMOS est maintenu dans une région linéaire de la caractéristique de transfert respective, à l'aide de charges adaptées et d'un courant de polarisation correspondant. Les charges peuvent être des résistances, auquel cas on utilise une commande de gain automatique pour conserver un courant de polarisation constant, ou des charges actives. Un oscillateur, commandé en tension et réalisé avec quatre de ces amplificateurs différentiels dans une configuration de gyrateur, oscille à la fréquence prédéterminée et possède huit signaux de sortie. L'oscillateur commandé en tension peut être utilisé dans des circuits assurant une régénération des données polyphasées, où le nombre de transitions de données dépasse le nombre de transitions d'horloge, pendant une durée donnée.
Patent EP-0867027-A1 (EP)
Title: Druckbehälter, insbesondere einer siedewasser-kernkraftanlage
Inventor: MATTERN JEAN
IPC: G21C13/10
Filed: 1996-12-05
Abstract: Die Erfindung betrifft einen Druckbehälter (1), insbesondere einen Sicherheitsbehälter einer Siedewasser-Kernkraftanlage, welcher aus Stahlbeton und einer metallischen Dichtstruktur (3) aufgebaut ist. Der Druckbehälter (1) besteht aus einem Innenzylinder (16) und einem den Innenzylinder (16) umschließenden Außenzylinder (14), wobei zwischen Innenzylinder (16) und Außenzylinder (14) ein Ringraum (2) zur Aufnahme der Kondensationskammer (17) und eines Flutbeckens (19) gebildet ist. Der Druckbehälter (1) ist geeignet, einem Innendruck von beispielsweise bis zu 20 bar standzuhalten.
Patent EP-0814942-A1 (EP)
Title: Outil pneumatique et supports antivibratoires associes
Inventor: SIENKIEWYCZ ROBERT A
IPC: B25F5/00
Filed: 1996-12-20
Abstract: L'invention porte sur un outil pneumatique (10) comportant des éléments antivibratoires (32) réduisant l'intensité des vibrations transmises à l'utilisateur. Ledit outil comporte une paire de supports (60) et au moins un amortisseur antivibratoire élastique (32) reliant les supports (60) de façon à les maintenir à distance l'un de l'autre. Un conduit d'air comprimé (54) traversant les ouvertures pratiquées dans les éléments de supports ne se trouve directement fixé qu'à l'un des éléments de support (58) et (60).
Patent EP-0791622-A1 (EP)
Inventor: SANDSTROM PAUL HARRY
IPC: C08K5/36
Filed: 1997-02-11
Abstract: The invention relates to a rubber composition containing silica reinforcement and to pneumatic tires having treads comprised of such rubber composition. 
     The rubber composition comprises at least one elastomer, silica, carbon black and a silica coupler comprised of 3,3'-tetrathiodipropanol polysulfide mixture.
Patent EP-0813316-A1 (EP)
Inventor: DELLAVERSON LOUIS P
IPC: H04Q11/04
Filed: 1997-06-09
Abstract: A method of establishing a spatially normalized communications path between a mobile subscriber unit and a base station in a wireless communications network comprising a plurality of communication slots. The method comprises the steps of transmitting (12) a control packet message that comprises an identity of a dedicated one of the plurality of communication slots to the mobile subscriber unit via the wireless communication network, receiving (14) the control packet message at the mobile subscriber unit, transmitting (16) a request service message to the base station via the dedicated one of the plurality of communication slots, receiving (18) the request service message at the base station, determining (20) a time distance measurement based at least in part on the step of receiving the request service message, communicating (22) the time distance measurement to the mobile subscriber unit via the communication network, and using (26) the time distance measurement to cause the mobile subscriber unit to transmit a subscriber unit data packet message via the communications network at a predetermined time relative to the start of the dedicated one of the plurality of communication slots. In this manner a spatially normalized communication path between the base station and the mobile subscriber unit is established.
Patent EP-0886306-A1 (EP)
Inventor: BAERT KRIS
IPC: G02F1/1362
Filed: 1997-06-16
Abstract: A method of bonding a first substrate (10) to a second substrate (30) is described,
comprising the steps of:
   coating an adhesive (28) onto a first major surface of said first substrate (10);   aligning said first and second substrates (10, 30) so that said coated first major surface of
said first substrate (10) is facing said second substrate (30) and is separated therefrom by a
gap (47) ;   deflecting at least one of said first and second substrates (10, 30) by exerting a pressure
between said first and second substrates (10, 30) substantially at the center thereof so that
the adhesive coating (28) substantially at the center of said first substrate (10) comes into
contact with said second substrate (30); and   allowing the remaining parts of said adhesive coated first major surface of said first
substrate (10) to come into contact with said second substrate (30).    
     Use of the method to produce composites, in particular transmissive liquid crytal
display panels is also described.
Patent EP-0834531-A1 (EP)
Inventor: SCHUBART RUEDIGER DR
IPC: C08J3/22
Filed: 1997-09-24
Abstract: Mixtures (I) of (A) halogenated butyl rubber and (B) polymer compounds, in which rubber (A) has a halogen content of 0.5-2.5% and a residual content of more than 0.7 mol% unhalogenated double bonds, the content of anti-agglomerate-/vulcanisation control additives is 1.0-2.2 wt% based on total (A), and (B) consists of (a) cyclic and/or acyclic amidines, (b) mercapto compounds and zinc salts of mercapto compounds of benzthiazole, benzimidazole, benzpyrimidine and/or benztriazine and (c) ethylene-propylene rubber, ethylene-propylene-diene rubber (EPDM), ethylene-vinyl acetate rubber, butadiene rubber (BR), styrene-butadiene rubber (SBR), natural rubber, butadiene-acrylonitrile rubber (NBR) and/or butyl rubber. In component (B), mol. ratio (a):(b) = (0.25:1)-(2:1) and the content of binder (c) is 90-10 wt%, and the amount of (B) in (I) is 0.1-20 (preferably 0.5-10) pts. wt. to 100 pts. wt. (A) (i.e. phr).
Patent EP-0837432-A1 (EP)
Inventor: STOCKS DAVID
IPC: G08B13/24
Filed: 1997-10-02
Abstract: The device (1) consists of a transmitter (4) which transmits at least one periodic interrogation signal into an interrogation zone (3). The interrogation signal stimulates a security element (2) to transmit an identity signal which is received by a receiver (5). A computer/control unit (7) evaluates the received identity signal and triggers an alarm if the security element is identified. The computer/control unit evaluates the received identity signal wrt. its amplitude and phase, detects a noise signal contained in the received signal and frees the received signal from the noise signal.
Patent EP-0894733-A1 (EP)
Inventor: HART JOSEPH J
IPC: B65D71/68
Filed: 1997-11-08
Abstract: A carrier (1) is provided which is made of a carrier box (3) and a
separate partition assembly (5) which is secured in the carrier box. The
partition assembly is made from transverse and cross partitions (71,73)
which have interengaging slots and tabs (83,84) which lock together to
form the partition assembly without the use of glue. The carrier box is
formed from a simple blank (21) having wall panels (7,9,11,13) and
bottom panels (15). The bottom panels are glued together to form a glued
bottom and are shaped so that the outer of the bottom panels meet along
a junction that is offset from the center of the carrier bottom. In an
alternative, and preferred embodiment, the carrier box is formed from a
one piece blank and the partition is formed from a one piece blank. The
partition includes a transverse partition or devider and at least one
cross-partition or devider. The partition (205) is formed from a blank
(261), which is preferably a one-piece blanks. The blank includes a
first body section (287a), a second body section (287b), and a handle
forming section (263). The first and second body sections are hingedly
connected to each other at a bottom of the partition and form the
transverse divider of the partition. The handle forming section is
hingedly connected to the first body section at a top of the first body
section. The first and second body portions each include at least one
fold-out section (289a,b) to define at least one cross-divider of
the partition. Also shown are two embodiments of the carrier itself
which includes locking means for holding the bottom of the carrier in
place substantially without the use of glue.
Patent EP-0854304-A1 (EP)
Inventor: STRADA VITO PIETRO
IPC: F16D13/04
Filed: 1997-12-16
Abstract: The clutch wheel (2) moves in relation to the clutch core (3), thereby reducing the frictional force of the clutch. The core has at least three lead ramps (16) matching the number of counter ramps (20) on the clutch wheel. The lead ramps each hold a ball (18) in contact with the counter ramp. The ramps and counter ramps each have a pre-set lead angle sloping in relation to the rotary direction of a clutch cage (4) and positioned so that, when braking torque occurs, the clutch wheel moves axially away from the core, and reduces the pressure force of the clutch. The lead ramp and counter ramp are in the form of grooves (17,19) with semicircular cross-section.
Patent EP-0852370-A1 (EP)
Inventor: KUPERUS LOUIS
IPC: E04F15/02
Filed: 1997-01-07
Abstract: A device comprising a rigid plate part to which plate part a
print has been applied, which print is protected at its top
side by means of a transparent plastic layer having a bottom
surface and a top surface, of which plastic layer the
dimensions substantially correspond to the dimensions of the
rigid plate part, the device comprising fastening means for
anchoring the device in a floor so that the top surface
substantially aligns with the floor surface.
Patent EP-0837458-A1 (EP)
Inventor: CHAPMAN DEREK DAVID
IPC: G11B7/246
Filed: 1997-10-04
Abstract: The present invention discloses optical
recording elements having optical recording layers
containing tetra dyes. The dyes have metallized azo
dianionic dye with cationic dye counterions. The
recording layer has a thickness from 225 to 300 nm.
Patent EP-0843137-A1 (EP)
Inventor: WATANABE HIDEO
IPC: F25D11/00
Filed: 1997-11-17
Abstract: A thermoelectric refrigerator is provided with a
casing (51) formed of a heat-insulating layer, thermal
conductors (53,54) arranged in the casing (51) and having
a heat transfer surface located facing a storage
space in the casing, a Peltier device (55) thermally
connected with the thermal conductors (53,54), a device
power supply (61) for supplying electric power to the
Peltier device (55), an interior fan (57) for causing
interior air (A) to flow in the storage space, a fan
power supply (62) for supplying electric power to the
interior fan (57), and a control unit (63) for controlling
a quantity of electric power to be supplied to the
interior fan (57) in accordance with a quantity of
electric power to be supplied to the Peltier device
(55).
Patent EP-0787431-A1 (EP)
Inventor: SUNTER ADRIAN MEREDITH
IPC: A21C9/04
Filed: 1997-01-29
Abstract: Material, e.g. for pizza topping, is applied (e.g. in a weighed amount) to an upper shutter assembly (207) whence it is dropped through a predetermined (and preferably variable) height onto iris blades (316) of a (larger) lower shutter assembly (206). The resulting deposit is of controlled diameter, possibly influenced by a mask (308). Rapid opening of the iris blades (316) allows the deposit to fall a short distance onto a substrate such as a pizza base.