baber/WOPTO huggingface dataset:
Patent CO-6180443-A2 (CO)
Title: Antagonistas del receptor de progesterona
Inventor: FUHRMANN ULRIKE
IPC: C07J21/00
Filed: 2009-05-15
Abstract: 1.- Un antagonista de receptor de progesterona de la fórmula general I:en la que R1 puede ser un átomo de hidrógeno y R2 puede ser un grupo hidroxilo o R1 y R2 pueden ser juntos un grupo oxo. 2.- 11ß-[4-(1,2-Dihidroxietil)fenil]-20,20,21,21,21- pentafluoro-17-hidroxi-19-nor-17a -pregna-4,9-dien-3-ona. 3.- 11ß-[4-[(1R) -1,2-Dihidroxietil]fenil] -20, 20, 21, 21, 21-pentafluoro-17-hidroxi-19-nor-17a -pregna-4,9-dien-3-ona. 4.- 11ß-[4-[(1S)-1,2-Dihidroxietil]fenil]-20,20,21,21, 21-pentafluoro-17-hidroxi-19-nor-17a-pregna-4,9-dien-3-ona. 5.- 20,20,21,21,21-Pentafluoro-17-hidroxi-11ß-[4-(hidroxiacetil) fenil]-19-nor-17a-pregna-4,9-dien--3-ona. 6.- Un fármaco que contiene antagonistas del receptor de progesterona de acuerdo con la reivindicación 1. 7.- El fármaco de acuerdo con la reivindicación 6 que contiene 11ß-[4-(1,2-dihidroxietil) fenil] -20, 20, 21, 21, 21- pentafluoro-17-hidroxi-19-nor-17a-pregna-4,9-dien-3-ona. 8.- El fármaco de acuerdo con la reivindicación 7 que contiene 11ß-[4-[(1R)-1,2-dihidroxietil]fenil]-20, 20, 21, 21, 21-pentafluoro-17-hidroxi-19-nor-17a-pregna-4,9-dien-3-ona. 9.- El fármaco de acuerdo con la reivindicación 7 que contiene 11ß-[4-[(1S)-1,2-dihidroxietil]fenil]-20,20,21,21, 21-pentafluoro-17-hidroxi-19-nor-17a-pregna-4,9-dien-3-ona. 10.- El fármaco de acuerdo con la reivindicación 6 que contiene 20, 20, 21, 21, 21-pentafluoro-17-hidroxi-11ß-[4- hidroxiacetil)fenil]-19-nor-17a -pregna-4,9-dien-3-ona.
Patent CO-6290623-A2 (CO)
Title: Composicion efervescente que comprende una sal fisiologicamente aceptable de un amino acido basico, una fuente de acido y una sal de carbonato soluble
Inventor: PRENCIPE MICHAEL
IPC: A61K8/36
Filed: 2010-09-03
Abstract: La presente invención se refiere a composiciones efervescentes que comprenden un aminoácido básico.1.- Una composición efervescente que comprende un aminoácido básico en forma libre o en forma de sal fisiológicamente aceptable, una fuente de ácido y una sal de carbonato soluble.2.- La composición de la reivindicación 1 donde el aminoácido básico es arginina, lisina, citrulina, ornitina, creatina, histidina, ácido diaminobutanoico, ácido diaminopropiónico, sales de los mismos y/o combinaciones de estos.3.- La composición de cualquiera de las reivindicaciones anteriores, donde el aminoácido básico presenta la configuración-L.4.- La composición de cualquiera de las reivindicaciones anteriores, donde el aminoácido básico es arginina.5.- La composición de cualquiera de las reivindicaciones anteriores, donde el aminoácido básico se presenta en forma de un carbonato.6.- La composición de cualquiera de las reivindicaciones anteriores, donde el aminoácido básico es bicarbonato de arginina.
Patent CO-6351688-A2 (CO)
Title: Derivados de benzoimidazol e inhibidores de glucogeno sintasa cinasa 3-beta que contienen los mismos.
Inventor: OHTANI MITSUAKI
IPC: A01N43/30
Filed: 2011-02-08
Abstract: La presente invención se relaciona con un compuesto de fórmula (I) y una sal aceptable farmacéuticamente, hidrato, solvato o isómero del mismo:donde,el anillo A es (II), (III), (IV), (V) o (VI)donde,X es halógeno o hidroxilo;Y es hidrógeno, fenilo, tiofen-2-ilo, furan-2-ilo, ciclopropilo o ciclopentilo;Z es un carbonilamino sustituido con un heterociclo de 5-10 miembros; y el anillo A está sustituido por -L1-(CH2)a-L2-M en la posición *;L1 es CONH-, -NHCO- o un enlace sencillo; L2 es seleccionado del grupo que consiste de -NH-, O, -CH(COOR1)-, -CH(CH2OH)-, -CH=CH- y un enlace sencillo, donde R1 es hidrógeno o C1-C6 alquilo;M es seleccionado del grupo que consiste de hidroxilo, carboxilo, amida, C1-C6 alquilo, C1-C6 alquilcarbonilo, C6-C14 arilo, C6-C14 aril C1-C6 alquilo, C6-C14 arilcarbonilo, C6-C14 arilsulfonilo, -NR2R3 entre otros; donde R2 y R3 son independientemente C1 -C6 alquilo;los grupos alquilo y aromáticos sustituyentes se encuentran, a su vez, sustituidos opcionalmente por 1-3 sustituyentes cada uno independientemente seleccionados del grupo A; donde el grupo A consiste de hidroxilo, oxo, nitro, amino, amida, halógeno, sulfamoilo, trifluorometilo, p-toluensulfonilamino, C1-C6 alquilo, C1-C6 alcoxi, C1-C6 alquilcarbonilamino y C1-C6 alquilsulfonilamino; y a es un número entero de 0-5.
Patent CO-6460767-A2 (CO)
Title: Composiciones sublinguales de dexmedetomidina y métodos de uso de ellas
Inventor: HENWOOD GERALDIE ANNE
IPC: A61K9/107
Filed: 2011-11-15
Abstract: Se provee una composición farmacéutica analgésica, transmucosal oral que comprende dexmedetomidina, o una sa farmacéuticamente aceptable de ella y un excipiente farmacéuticamente aceptable, y el uso de dichas composiciones en el tratamiento o prevención del dolor sin sedación importante.
Patent CO-6571858-A2 (CO)
Title: Proceso de flotacion con espuma para la preparacion de silicatos y carbonatos de metal alcalino terreo usando un recolector que comprende al menos una polialquilenimina hidrofobicamente modificada
Inventor: GANE PATRICK AC
IPC: C01B32/60
Filed: 2012-09-14
Abstract: La invención se refiere a un proceso para separar silicatos y carbonatos de metal alcalino térreo que implementa al menos polialquilenimina hidrofóbicamente modificada, en donde:i) la polialquilenimina es hidrofóbicamente modificada por reemplazo de todos o parte de los hidrógenos de sus grupos amino primarios y/o secundarios por el grupo funcional R, donde R comprende un grupo alquilo lineal, ramificado o cíclico y/o arilo, y contiene 1 a 32 átomos de carbono;ii) antes de la modificación, la polialquilenimina tiene al menos 3 unidades de repetición de alquilenimina y un peso molecular de entre 140 y 100 000 g/mol;iii) la modificación de la polialquilenimina produce un aumento de la cantidad de C atómico, con relación a la polialquilenimina no modificada, de entre 1 y 80%.Adicionalmente, la invención se refiere a un producto que contiene silicato y un producto que contiene carbonato de metal alcalino térreo obtenido mediante el proceso de la invención, y a sus usos.
Patent CO-6690780-A2 (CO)
Title: Formulaciones para el factor estimulante de colonias de granulocitos bovino y variantes de las mismas
Inventor: KHA CATHERINE NGAN
IPC: A61K38/19
Filed: 2013-03-22
Abstract: La presente invención se refiere a formulaciones acuosas estables que comprenden un polipéptido bG-CSF o una variante del mismo, una sustancia amortiguadora y un excipiente, en donde la formulación está sustancialmente libre de monolaurato de polioxietilen (20) sorbitán. La invención también proporciona métodos de uso, una forma liofilizada o en polvo de, y un proceso para, preparar la formulación.
Patent EP-1020627-A2 (EP)
Inventor: FUWA NAOHIDE
IPC: F02F1/24
Filed: 2000-01-11
Abstract: A controller (92) for an internal combustion engine
(11) that switches combustion modes in accordance with the
running conditions of the engine (11). When there is a need
to reduce the engine torque, the controller (92) decreases
the torque by a predetermined torque reduction method. The
controller (92) decreases the engine torque by a first
torque reduction method when the engine (11) is in a first
combustion mode. When the engine (11) is in a second
combustion mode, the controller (92) reduces the torque by a
second torque reduction method. The controller (92) sets a
first control amount, which corresponds to the torque
reduction requirement, according to one of the first and
second torque reduction methods. The controller (92)
converts the first control amount into a second control
amount, which corresponds to the other torque reduction
method. When controlling the engine torque with the first
torque reduction method, the control is based on the first
control amount. When controlling the engine torque with the
second method, the control is based on the second control
amount.
Patent EP-1044750-A2 (EP)
Inventor: FREMBGEN FRITZ-HERBERT
IPC: B23H9/16
Filed: 2000-02-25
Abstract: In the method, after shutting off a pressure reservoir, a high liquid pressure is set up using a high pressure pump (34) via regulating valve (38) and calibration is started. The pump replenishes an electrolyte stream during calibration through a liquid stream in a liquid compartment and maintains a constant high pressure. Process for electrochemically processing workpieces comprises using a pressure reservoir (20) having an electrolyte compart (18) and a liquid compartment (24) with a separator (22). The electrolyte is passed from a tank (12) under low pressure to the electrolyte compartment whilst a corresponding amount of liquid is passed to a pressure-less reservoir (32) from the liquid compartment. After shutting off the pressure reservoir a high liquid pressure is set up using a high pressure pump (34) via a regulating valve (38) and the calibrating process can be started. The pump replenishes the electrolyte stream during the calibra through a liquid stream in the liquid compartment and maintains a constant high pressure.
Patent EP-1035172-A2 (EP)
Inventor: YAMAKAWA KATSUYOSHI
IPC: C09B55/00
Filed: 2000-02-29
Abstract: An azomethine compound is represented by the formula (I).
 
and R 1 , L 1 , L 2 , R 3  and R 4  have 20 to 50 carbon
atoms in total.
Patent EP-1046833-A2 (EP)
Inventor: HASSELMEYER ALFRED DIPL-ING
IPC: F16F13/14
Filed: 2000-03-10
Abstract: The hydrolastic bearing comprises an inner (2) and outer (1) bearing ring with an elastic component (3) between them which f chambers for fluid. This has a throttle channel (5) at the bottom and an overflow channel (6) at the top. This contains a valve component (7) with a sealing pad, part of which is flexible.
Patent EP-1041172-A2 (EP)
Inventor: YAMARTINO JOHN M
IPC: H01L21/302
Filed: 2000-03-30
Abstract: A method of eliminating charging resulting from plasma
processing a semiconductor wafer comprising the steps of plasma
processing the semiconductor wafer in a manner that may result
in topographically dependent charging and exposing, during at
least a portion of a time in which the semiconductor wafer is
being plasma processed, the semiconductor wafer to particles
that remove charge from the semiconductor wafer and reduce
topographically dependent charging.
Patent EP-1049362-A2 (EP)
Inventor: KOSTELNIK JAN DR
IPC: H05K3/46
Filed: 2000-04-20
Abstract: A carrier (1) has the shape of a flat plate. On the carrier's topside a printed circuit board (4) is bonded with an adhesive foil (3). This board has a coupling area containing multiple micro-vias (6) passing through from the open topside (7) to the bottom s (8) turned to the carrier.
Patent EP-1075883-A2 (EP)
Title: Vorrichtung zum Lochen von Werkstücken beim Innenhochdruckumformen
Inventor: RECKTENWALD PAUL
IPC: B21D28/28
Filed: 2000-07-12
Abstract: Die Erfindung betrifft eine Vorrichtung zum Lochen von Werkstücken beim Innenhochdruckumformen,
mit einem aus der Formhohlraumwand in den Formhohlraum hinein vorschiebbaren
Lochstempel. Erfindungsgemäß ist zur Befestigung des Lochstempels ein Halterungsblock
mit einem Steckloch vorgesehen, in welches der Lochstempel unter Rastbefestigung
an dem Halterungsblock entgegen der Vorschubrichtung des Lochstempels einführbar
und aus dem der Lochstempel nach Lösung der Rastbefestigung in Vorschub-richtung
ausziehbar ist. Vorteilhaft erlaubt diese Erfindungslösung, verschliessene Loch-stempel mit
geringem Montageaufwand auszuwechseln.
Patent EP-1077302-A2 (EP)
Inventor: HOFF AXEL DR DIPL
IPC: E06B3/67
Filed: 2000-07-29
Abstract: The vacuum insulation element comprises at least two parallel plates (1, 2) which are joined to another only along their edges, surround an evacuat-able space (4) between them, and are provided with electrical and/or magnetic means (3) serving to substantially compensate the force produced on the plates by the surrounding atmosphere. Also claimed are a multipane window with such vacuum insulation elements, and a method for contactless support of plate shaped structural elementse The claimed heat insulating windows are characterized by the fact that the materials of foils and bipolar force com-pensating elements used are transparent.
Patent EP-1078749-A2 (EP)
Inventor: AONO KIYOMI
IPC: B41J2/05
Filed: 2000-08-22
Abstract: An ink jet recording apparatus includes an ink jet recording head provided with a discharge port (205) for discharging ink, an ink flow path (202) communicating with the discharge port, and at least two heat generating elements (501,502) provided in the ink flow path along the direction thereof, wherein the ink is pigment-based ink and the recording head comprises drive signal supply means for varying the supply timing of drive signals to the plural heat generating elements for ink discharge in such a manner that the drive signal is at first given to the heat generating element at the side of the discharge port at room temperature and the supply timings to the plural heat generating members become simultaneous or closer thereto with an increase in the temperature of the recording head.  <IMAGE>
Patent EP-1098440-A2 (EP)
Title: Zeitbasisgenerator
Inventor: THOLLET ALEXANDRE
IPC: G04G7/00
Filed: 2000-10-26
Abstract: Dargestellt und beschrieben ist eine Anordnung zum Erzeugen eines ersten zeitlich alternierenden Signals und eines zweiten zeitlich alternierenden Signals, das zum ersten Signal in einem vorbestimmten festen Frequenzverhältnis steht, mit einem ersten Oszillator (1), einem zweiten Oszillator (2) und einem dritten Oszillator (3), wobei der erste Oszillator (1) ein seiner Schwingungsfrequenz entsprechendes Schwingungssignal an einen ersten digitalen Frequenzteiler (4 ) liefert, der daraus das erste Signal erzeugt und ein seiner Schwingungsfrequenz entsprechendes Schwingungssignal an einen zweiten digitalen Frequenzteiler (5 ) liefert, der daraus ein erstes Synchronisationssignal erzeugt, wobei der zweite Oszillator (2) ein seiner Schwingungsfrequenz entsprechendes Schwingungssignal an einen dritten digitalen Frequenzteiler (6) liefert, der daraus ein zweites Synchronisationssignal erzeugt und ein seiner Schwingungsfrequenz entsprechendes Schwingungssignal an einen vierten digitalen Frequenzteiler (7) liefert, der daraus ein drittes Synchronisationssignal erzeugt, wobei der dritte Oszillator (3) ein seiner Schwingungsfrequenz entsprechendes Schwingungssignal an eine fünften digitalen Frequenzteiler (8) liefert, der daraus ein viertes Synchronisationssignal erzeugt und ein seiner Schwingungsfrequenz entsprechendes Schwingungssignal an einen sechsten digitalen Frequenzteiler (9) liefert, der daraus das zweite Signal erzeugt, wobei das erste Synchronisationssignal und das zweite Synchronisationssignal einem ersten Phasenvergleicher (10) zugeführt werden, der in Abhängigkeit von der Phasendifferenz des ersten Synchronisationssignals zum zweiten Synchronisationssignal eine Spannung an einen ersten spannungsgesteuerten Oszillator (11) ausgibt, der die Schwingungsfrequenz des zweiten Oszillators (2) derart regelt, daß diese zur Schwingungsfrequenz des ersten Oszillators (1) in einem vorbestimmten festen Verhältnis steht, und wobei das dritte Synchronisationssignal und das vierte Synchronisationssignal einem zweiten Phasenvergleicher (12) zugeführt werden, der in Abhängigkeit von der Phasendifferenz des dritten Synchronisationssignals zum vierten Synchronisationssignal eine Spannung an einen zweiten spannungsgesteuerten Oszillator (13) ausgibt, der die Schwingungsfrequenz des dritten Oszillators (3) derart regelt, daß diese zur Schwingungsfrequenz des zweiten Oszillators (2) in einem vorbestimmten festen Verhältnis steht.
Patent EP-1136840-A2 (EP)
Inventor: LOCHTE GUIDO
IPC: G01S13/931
Filed: 2000-12-04
Abstract: The device has a visual display unit (5) driven by the sound generator output (4) of a controler (3) and the visual display unit has an evaluation device (11) for converting the sound generator signals into control signals for the visual display unit. The evaluation device is a microcontroller or an electronic evaluation circuit. Independent claims are also included for the following: a display unit and the use of a controler with a sound generator output for controling a visual display unit.
Patent EP-1090836-A2 (EP)
Inventor: FENNY CARLOS ALEXANDER
IPC: B64C29/00
Filed: 2000-09-27
Abstract: The tilt rotor aircraft comprises an airframe, a
pair of wing members coupled to the airframe, a pair of
cooperating tilt rotor assemblies carried by the pair of
wing members operate in a plurality of modes of operation,
a flexible and elongated rotating shaft (201) extending between
the pair of cooperating tilt rotor assemblies, a plurality
of assemblies (215,217,219,221) for generating at least one signal
indicative of an amount of twist on the flexible and elongated shaft,
a controller (211) for receiving the at least one signal and
generating command signals, and a plurality of actuators (207,209)
for receiving the command signals and for compensating for
the twist in the flexible and elongated shaft.
Patent EP-1022668-A2 (EP)
Inventor: WILLIAMS MARVIN L
IPC: G06Q10/10
Filed: 2000-01-11
Abstract: For use with an electronic mail (e-mail) program, a
system for, and method of, establishing relationships between
hypertext references contained in e-mail messages received by
the e-mail program and an e-mail program containing the
system or the method. In one embodiment, the system
includes: (1) a message parser that locates hypertext
references in first and second e-mail messages received by
the e-mail program and (2) a message organizer that allows a
user to choose to display the first and second e-mail
messages in an order that is based on the hypertext
references.
Patent EP-1027932-A2 (EP)
Inventor: JACOBS MERRIT N
IPC: B01L3/02
Filed: 2000-02-11
Abstract: Apparatus and a method for mixing a liquid
within a disposable aspirating probe tip so that most of
the liquid is forced to move past a transition zone
between two different inside diameters to cause
rotational mixing. The apparatus and method can be used
to provide agglutination of blood, which in turn can be
used for blood typing. The probe tip can comprise a
single integral piece, or two separate portions.
The transition zone can comprise a sharp demarcation
between inside diameters, or a smooth one.
Patent EP-1048479-A2 (EP)
Inventor: ASANO SHINICHI
IPC: B41M5/00
Filed: 2000-04-25
Abstract: An ink jet recording material having excellent gloss
and capable of recording thereon clear ink images having
a high color density includes a multi-layered ink fixing
layer, formed on a substrate material and composed of an
outermost ink fixing layer, and one or more intermediate
ink fixing layers superposed on each other, and each
includes a binder and a pigment selected from silica,
aluminosilicate, alumina and zeolite, the pigment in each
ink fixing layer being in the form of fine secondary
particles having an average secondary particles size of
1 µm or less and each secondary particle is composed of a
plurality of primary particles agglomerated with each
other, and the outermost ink fixing layer being one
formed by a cast-coating procedure using a specular
casting surface.
Patent EP-1067298-A2 (EP)
Inventor: GEACH PETER WILLIAM
IPC: F16B5/01
Filed: 2000-05-03
Abstract: A composite component, for example for use in ship
building, comprises a composite panel 4 to which is
secured a metal extension 2. The metal extension 2 has
a groove within which a rib 28 at an edge region of the
composite panel 4 is fitted. The groove has an
interior width which is larger than the width of the
mouth of the groove, to prevent separation of the metal
extension 2 from the composite panel 4. The metal
extension 2 enables the composite component to be
secured to metal parts, for example for the hull of a
ship, by welding.
Patent EP-1084689-A2 (EP)
Inventor: KURATA NOBUHIRO
IPC: A61F13/15
Filed: 2000-09-13
Abstract: Provided is a water-decomposable absorbent article
including a water-decomposable back sheet, a water-decomposable
absorbent layer, and a surface member covering
the absorbent layer. The surface member has a plurality of
water-retentive water-decomposable sheets laminated and
bonded to each other by integration means for permitting to
dissociate the water-decomposable sheets from each other when
wetted.
Patent EP-1099910-A2 (EP)
Inventor: AKKALA MARC W
IPC: F24D18/00
Filed: 2000-10-27
Abstract: A potable water temperature management system (10) includes a device (26) that
produces waste heat and that has a primary purpose other than heating potable water.
The waste heat from the device (26) is used to heat potable water in a tank (14). A
heat shedding system (62) is activated when the temperature of the potable water in the
tank (14) exceeds a selected maximum temperature. An auxiliary energy transfer
system (54) may be activated to heat the potable water in the tank (14) when the
potable water in the tank (14) falls below a selected minimum temperature. A
controller (42) may be used to monitor the temperature of the potable water in the tank
(14) and activate either the heat shedding system (62) or the auxiliary energy transfer
system (54) based on the potable water temperature.
Patent EP-1114813-A2 (EP)
Inventor: SAKAMOTO KAZUHIKO
IPC: C07C67/62
Filed: 2000-12-06
Abstract: It intends to prevent the reduction in quantity with
time of an N-oxyl compound in vinyl compounds. The quantity
reduction of the N-oxyl compound is suppressed by causing
an N-oxyl compound,
N-hydroxy-2,2,6,6-tetramethylpiperidine compound and a
2,2,6,6-tetramethylpiperidine compound to co-exist in vinyl
compounds.
Patent EP-1028316-A2 (EP)
Inventor: GRIFOLS LUCAS VICTOR
IPC: G01N33/53
Filed: 2000-02-10
Abstract: A device for carrying out agglutination tests. 
     The device has a microtube with a widened upper region
and a lower tubular region of smaller diameter, having
in the transition region between the upper portion which
is intended for the test sample and the lower portion of
the microtube, which lower portion carries the
agglutination reagents, a plurality of grooves on which
coincides a freely fitted ball, defining, together with
the grooves, communication passages between the upper
portion and the lower portion of the device which
prevent the free passage of the test sample, which can
pass to the region carrying the agglutination reagents
only it it is subjected to centrifugation having
predetermined characteristics.
Patent EP-1025883-A2 (EP)
Title: Pole provided with a quick-releasing interchangeable lateral support extension
Inventor: MANNINEN TAISTO
IPC: A63C11/22
Filed: 2000-02-02
Abstract: The object of the invention is a pole provided with a quick-releasing
interchangeable lateral support extension, especially a walking, skiing, alpine
skiing or other sports pole. Around the lower end of the pole (1) is injection
moulded a sleeve socket (2) from which a guide projection (3) and a locking
projection (4) protrude. The lateral support extension sleeve (6, 8) comprises a
resilient tongue (12), below which there is a receiving aperture (14) for the
locking projection (4). The sleeve also comprises a guide groove (11) for
receiving the guide projection (3). The lateral support extension (5) is easy to
detach by turning the resilient tongue (12) outwards.