baber/WOPTO huggingface dataset:
Patent SK-283541-B6 (SK)
Title: Nonapeptide bombesin antagonists, pharmaceutical composition and use
Inventor: SCHALLY ANDREW V
IPC: A61K38/08
Filed: 1991-11-15
Abstract: The novel pseudo polypeptides of this invention are potent bombesin antagonists. There are provided processes for their production, pharmaceutical compositions comprising said polypeptides and their use as pharmaceutically active agents. More particularly the present invention provides pseudopeptides comprising a nonapeptide moiety of formula (I): X-A1-A2-A3-A4-A5- A6-A7-A8-psi-A9-Q, wherein Q is NH2 or OQ1 where Q1 is hydrogen, C1-10alkyl, phenyl or phenyl-C7-10-alkyl; X is hydrogen or a single bond linking to A2, the acyl residue of an organic acid, or a group of formula R1CO- wherein 1) R1 is hydrogen, C1-10alkyl, phenyl or phenyl-C7-10-alkyl; 2) R1CO- is a) R2.N(R3)-CO- wherein R2 is hydrogen, C1-10alkyl, phenyl or C7-10phenyl-C7-10-alkyl, R3 is hydrogen or C1-10 alkyl; b) R4-O-CO- wherein R4 is C1-10alkyl, phenyl or phenyl-C7-10-alkyl. A1 is D-, L- or DL-pGlu, Nal, Phe, Thi, Tyr, Tpi, Hca, Hpp, Mpp, Trp or Trp substituted in the benzene ring by one or more members selected from the group consisting of halogen, NO2, NH2, OH, C1-3 alkyl and C1-3 alkoxy wherein halogen is fluorine, chlorine and bromine, A2 is Asn, Dpa, Gln, His, MeHis, His(Bz), His(Z) or a group of formula Dpa (X), Asp (Y), Glu [-] and Glu (Y); wherein X is as above, Y is -OR5 or R6-NR7 wherein R5 is hydrogen, C1-3alkyl or phenyl; R6 is hydrogen or C1-3alkyl; R7 is hydrogen, C1-3alkyl or -NHCONH2 and [-] is a single bond linking the side carboxyl group with the alpha amino group of A1 where X is a single bond, A3 is Nal, Pal, Tpi, Trp, MeTrp, Trp(For) or Trp substituted in the benzene ring by one or more members selected from the group consisting of halogen, NO2, NH2, OH, C1-3 alkyl and C1-3 alkoxy wherein halogen is fluorine, chlorine and bromine; A4 is Ala, MeAla or Gln; A5 is Val or MeVal; A6 is Gly, Phe or D-Ala; A7 is His, MeHis, His(Bz), His(Z), Lys(Z) or Pal; A8 is a reduced isostere of Leu or Phe; A9 is Leu, Phe, Tpi, Trp or Trp substituted in the benzene ring by one or more members selected from the group consisting of halogen, NO2, NH2, OH, C1-3alkyl and C1-3alkoxy wherein halogen is fluorine, chlorine and bromine; provided that where A9 is Leu or Phe, A1 is other than D-Nal or DL-Phe and where A1 is D-Nal or DL-Phe, A9 is other than Leu or Phe and the salts thereof with pharmaceutically acceptable acids.
Patent SK-281650-B6 (SK)
Title: N-methylamides, process and imtermediates for their preparation and their use as pesticides
Inventor: BAYER HERBERT
IPC: A01N37/50
Filed: 1993-08-27
Abstract: N-methylamides of the formula I <IMAGE>  in which     R denotes alkyl or cyclopropyl, the radicals A denote hydrogen, halogen, cyano, nitro, alkyl, cycloalkyl, OR<1>, cycloalkyloxy, haloalkyl, haloalkyloxy, alkenyl, alkenyloxy, alkynyl, alkoxyalkyl, cyanoalkyl, nitroalkyl, phenyl, phenoxy, C(O)R<1>, CO2R<1>, C(O)NR<1>R<2>, C(S)NR<1>R<2>, NR<1>R <2>, NR<1>C(O)R<2>, NR<1>CO2R<2>, OC(O)R<1>, SR<1>, S(O)R<1>, S(O)2R<1>, the groups -C(R<1>)=NR<2>, -N=CR <1>R<2>, <IMAGE> where the radicals R<1>, R<2> and R<3> denote hydrogen or C1-C6-alkyl or X denotes S, O and NR<3> and n denotes the numbers 0 or 1, or two of the groups Am in adjacent positions together denote the group -CH=CH-CH=CH and   m represents the numbers 1, 2 or 3, and fungicides containing these compounds.
Patent CZ-285102-B6 (CZ)
Inventor: RASEHORN HANS-JUERGEN DR ING
IPC: B02B5/02
Filed: 1991-08-14
Abstract: Třídění se provádí do více frakcí. První frakce jader se získává přímo z druhého stupně třídění. První frakce slupek a frakce nevyloupnutých jader, která se opětovně loupe, se získávají z prvního stupně třídění. Z druhého stupně třídění a jednoduché elektroseparace se získává druhá frakce slupek, druhá frakce jader a frakce směsná, která se vytřídí do třetí frakce jader a třetí frakce slupek. Ze všech tří frakcí slupek se pak znovu oddělí čtvrtá frakce jader a konečná frakce slupek. Zařízení sestává z loupacího stroje (1) prvního a druhého stupně loupání a separátoru (2) slupek, který sestává z dvojité síťové plochy (2a) a dvojitého elektroseparátoru (2b), k němuž je dále připojen elektrický odlučovač (3).ŕ
Patent CZ-283079-B6 (CZ)
Inventor: FOHL ARTUR
IPC: B60R22/32
Filed: 1992-08-17
Abstract: Vybavovací mechanismus  pro napínací ústrojí  pásů má snímací hmotu, která reaguje jak při  čelním, tak i při zadním nárazu vozdla. Snímací  hmota může být uložena vykývnutelně a může být  tvořena funkčními částmi pohonu napínacího  ústrojí. U napínacího ústrojí pásu, které je  sdruženo s navijákem (10) pásu do jedné  konstrukční skupiny a které má pyrotechnický  pístový a válcový pohon, sestává snímací hmota z  podstavce (12), na kterém je vykývnutelně uložen  nosný blok (40), na němž je upevněn vodicí válec  (42) a v něm uložený píst. Na podstavci (12)  vykývnutelně uložená úderníková páka (50) je  uvolňována pro aktivaci úderníkového zapalovače  na plynové generátorové patroně (44), pokud je  nosný blok (40) sensitivně vykývnut v jednom  nebo opačném směru jízdy.ŕ
Patent CZ-279842-B6 (CZ)
Title: Valve seat integral with cylinder head casting
Inventor: NOVOTNY OTTO ING
IPC: C22C37/00
Filed: 1990-07-03
Abstract: A casting of an integral valve seat with cylinder head casting from grey iron with a structure of lamellar pearlite with laminated graphite with grain size of 60 to 200 microns and containing a max. of 0.08 % by weight of sulphur consisting of 2.8 to 3.7 % by weight carbon, 1.4 to 2.4 % by weight silica, 0.5 to 1.0 % by weight manganese, 0.03 to 0.1 % by weight of aluminium, whereas the valve seat is formed by eutectic cementite at a max. depth of 3 mm from the active surface of the seat. The casting can also contain 0.2 to 0.4 % by weight nickel and 0.25 to 0.5 % by weight chrome, or an additive of 0.04 to 0.1 % by weight stibium and a max. of 0.1 % by weight titanium. The process of production is based on the fact that the active surface of the valve seat, after preheating the casting to 450 to 650 degrees C under a protective atmosphere, is gradually locally melted with subsequent cooling rate lower than 50 degrees C/h.
Patent CZ-288577-B6 (CZ)
Title: Process for producing composite product
Inventor: BOISSONNAT PHILIPPE
IPC: B29C48/285
Filed: 1992-11-09
Abstract: The proposed process for producing a composite product formed by conjunction of organic thermoplastic material, reinforcing fibers such as glass fibers and optionally mineral materials and organic additives, and obtained by extrusion from or injection moulding in an extruder is characterized in that at least a portion of the organic thermoplastic material is introduced in the extruder in the form of endless fibers or threads of endless fibers. The introduced organic thermoplastic material is then melted and mixed with reinforcing fibers and a moulding machine to a section or a body of a defined shape subsequently converts the obtained mixture.
Patent CZ-279563-B6 (CZ)
Title: Heating wall of a coke oven
Inventor: KYNCL JIRI ING
IPC: C10B29/02
Filed: 1992-12-17
Abstract: The heating wall of a coke oven is formed from inbound baffles (1) and outbound layers (2). The connection of the blocks (6) in the bedded joints (31) is performed by mortise joints (4), consisting of bowls (41) and pins (42), which have the form of a truncated cone. The surface of the bowls (41) and pins (42) is rounded by transient radii (5). The dimensioning of the mortise joints (4) is determined by a precise relationship between the size of the surface of the base (422) of the pin (42) and size of the surface of the perpendicular cross-section (62) through the block (6).<IMAGE>
Patent CZ-284329-B6 (CZ)
Inventor: VORWERK DIERK
IPC: A61B17/11
Filed: 1994-12-15
Abstract: Endovaskulární implantovaná protéza pro instalaci do nebo v blízkosti bufurkace v cévním systému pacienta, například z důvodu nápravy vydutí nebo bifurkace aorty, zahrnuje trubkové hlavní těleso pro umístění do horní cévy, jako je aorta, nad bifurkaci a trubkových ramen spojených s hlavním tělesem v bifurkaci a procházejících do každé ze dvou větví cév, jako jsou stehenní cévy. Hlavní těleso (8) má tvar váčku s otevřeným proximálním horním koncem a s distální dolní dnovou oblastí, ve které jsou vytvořeny dva výstupní otvory (9, 10), přičemž toto hlavní těleso (8) je radiálně roztažitelné a upevnitelné v radiálně roztaženém stavu k vnitřní straně horní cévy (2) nad bifurkací prostřednictvím fixačních prostředků (11). Ramena jsou vytvořena jako samostatná pružná a radiálně roztažitelná ramenová napínací zařízení (15, 16) upravená pro vložení ve složeném stavu do větví cév a do výstupních otvorů (9, 10), a přičemž každé z napínacích zařízení (15, 16) zabírá ve svém radiálně roztaženém staŕ
Patent CZ-280096-B6 (CZ)
Inventor: MACKRLE SVATOPLUK ING CSC
IPC: B01D21/00
Filed: 1993-10-14
Abstract: Reaktor pro chemickou úpravu vody s mechanickou homogenizací vločkovité suspenze a její následnou separací fluidní filtrací. Pro homogenizaci je vybaven homogenizačním prostorem (10), který je propojen se separačním prostorem (12) převáděcím kanálem (25) vytvořeným mezi uzavírací stěnou (7) homogenizačního prostoru (10) a k ní přiřazenou vnitřní usměrňovací stěnou (23). Tato usměrňovací stěna (23) přesahuje přitom propojovací pasáž (9) provedenou v uzavírací stěně (7) pro spojení homogenizačního prostoru (10) se separačním prostorem (12). V homogenizačním prostoru (10) je uspořádáno míchací ústrojí a čerpadlo.
ŕ
Patent CZ-286861-B6 (CZ)
Title: Gearless belt winding device
Inventor: FOREJT JIRI ING
IPC: B65H75/48
Filed: 1996-07-26
Abstract: The invented gearless strip coiler is usable particularly for coiling metal strips (22) in cold rolling mills of high rolling speeds, where there is no gear drive between a driving motor and a winding drum (2). On the side opposite to the winding drum (2) there is performed in a hollow shaft (4) a bore (15) for Belleville washers (5) mounted on the winding drum (2) axle (3). The Belleville washers (5) are in permanent contact with the axle (3) a prestressing nut (6) behind which there is arranged an adjustable nut (7) with an external recess (16) for fixing balls (8) corresponding to radial openings (17) of a guide bush (9) being fixedly coupled with a hollow shaft (4), whereby on the adjustable nut (7) and on the guide bush (9) there is mounted a slidably sprung sleeve (10) being provided on its inside diameter with a shaped recess (18) and on its outside diameter with a circumferential groove (19) for rollers (11) being in kinematic connection with at least one control element (13) attached to the coiler casing (1). A locking ball mechanism enables prior introduction of the strip beginning  opening of the winding drum (2) and during coiling a single retraction thereof.
Patent CZ-294856-B6 (CZ)
Title: Intranasal pharmaceutical preparations for treating sexual disorders and sildenafil mesylate
Inventor: BILLOTTE ANNE
IPC: C07D487/04
Filed: 1999-06-21
Abstract: In the present invention, there is disclosed an intranasal pharmaceutical formulation for the treatment of male erectile dysfunction or female sexual disorders, which formulation comprises sildenafil mesylate, together with a pharmaceutically acceptable diluent or carrier in a form adapted for intranasal administration. Disclosed is also sildenafil mesylate.
Patent SK-284932-B6 (SK)
Title: Monoclonal antibody, fragment thereof, method for its preparation and use, pharmaceutical composition, hybridoma cell line, amino acid sequence and DNA sequence
Inventor: MITJANS FRANCESC
IPC: A61K39/00
Filed: 1995-12-19
Abstract: Described is a monoclonal antibody and its fragment comprising amino acid sequence of the basic framework regions (FR) and the complementarity determining regions (CDR) of the light chain of SEQ ID NO:1 and of the heavy chain SEQ ID NO:9. A hybridoma cell line capable of producing thereof, amino acid sequence comprising the sequence given in SEQ ID NO:1 or SEQ ID NO:9. Adequate DNA sequence, pharmaceutical composition comprising said antibody, method for its preparation and use for the manufacture of a drug for the treatment of tumors.
Patent SK-278628-B6 (SK)
Title: 0-3-trimethylammonium-2-hydroxypropyl derivative of hemicelluloses of the type of (1->4)-beta-d-xylan and preparation method thereof
Inventor: EBRINGEROVA ANNA
IPC: C08B37/14
Filed: 1989-06-14
Abstract: This patent describes the derivatives of hemicellulose closed to the type of (1->4)-beta-D-xylan with the structural units represented by formulas (I) and (II) and/or (II) where R1 and R2, which can be the same or different, mean hydrogen or the group with a general formula (IV), where X means hydroxyl, dihydrogenphosphate, hydrogensulphate, chloride or acetate anion, R3 means the structural unit closed to 4-O-methyl-aplpha- -D-glucoronic acid with a general formula (V), in which Y means hydrogen, sodium or potassium, R4 means the unit closed to alpha-L-arabinofuranose with a formula (VI), while the average degree of polymerisation closed to (1->4)-beta-D-xylan is 20 up to 200. The derivatives of hemicellulose are prepared based on that principle, that in the first stage hemicellulose closed to the type of (1->4)-beta-D-xylan with the structural unit represented by the formula (VII) and (II) and / or (III) are being activated wit 1 up to 25 weight percent water solution of alkaline metal hydroxide at the temperature of 15 up to 25 Celsius degrees, for 30 up to 60 minutes, in the second stage they are undertaken to alkylation with the use of 3-chlorine-2-hydroxypropylmethylammonium chloride, at the temperature of 30 up to 80 Celsius degrees, for 2 up to 6 hours, while the molar ratio closed to hemicellulose : alkaline metal hydroxide is 1: 0,2 up to 3: 0,1 up to 2 a dialysed and dried. The prepared product can be applied as the flocculating agent, when talking about water purification and it also can be used as the auxiliary additive in the production of paper.
Patent SK-288892-B6 (SK)
Title: Modular assembly for collective clamping of the small parts for the optical 3D scanning
Inventor: BURANSKÝ IVAN
IPC: H04N13/00
Filed: 2018-05-14
Abstract: The modular assembly for mass alignment and clamping of small optical scanning components is designed so that the rectangular frame (1) is formed by a hexagonal profile, wherein two permanent magnets (3) are inserted into each side of the frame (1). Each side of the frame (1) is provided with a horizontally oriented fitting pin (4) and a fitting hole (5) that alternate regularly on the sides of the frame (1). On each side of the frame (1) between each fitting pin (4) and the fitting hole (5) is a clamping rod (6) with a locking screw (7) inserted horizontally and adjustable. The permanent magnets (3) in the fitting pins (4) have the opposite magnetic orientation as the permanent magnets (3) at the fitting holes (5). Clamping holes (9) are vertically matched with corners of the frame (1). The clamping rods (6) may be of variable size.
Patent SK-288850-B6 (SK)
Title: Continuous controlling method of temperature profile of soldering paste remelting in environment of saturated vapors of boiling liquid
Inventor: LIVOVSKÝ ĽUBOMÍR
IPC: B23K1/012
Filed: 2017-08-16
Abstract: The method is based on monitoring of temperature change at printed circuit board surface. The monitoring is realized by means of 32-bit industrial micro-controller with application of software regulator with simultaneous continual regulation of the horizontal position of a printed circuit board above the level of boiling water by means of a step motor, as well as the regulation of heating of the liquid. Thereby significant time reduction is achieved at adjusting of parameters in order to meet the defined line of temperature profile for remelting of solder paste. The method also saves energy at keeping required conditions for remelting of solder pastes in electronics.
Patent CZ-300120-B6 (CZ)
Title: Pharmaceutical composition intended for administration by injection
Inventor: FRANC ALES
IPC: A61K33/243
Filed: 2006-06-20
Abstract: In the present invention, there is disclosed an injectable pharmaceutical composition comprising a mixture of platinum complex of the general formula I, in which A and A' represent independently on each other the group NHi3 or an amine or diamine group containing 1 to 18 carbon atoms, B and B' represent independently on each other a halogen atom or a hydroxyl group or they can represent the group -O-C(O)-R optionally the group -O-C(O)-R', in which R and R' denote independently on each other a hydrogen atom, an alkyl group, an alkenyl group, an aryl group, an aralkyl group, an alkylamino group or an alkoxyl group, whereby these groups contain 1 to 10 carbon atoms, or functional derivatives of these groups, X and X' represent independently on each other a halogen atom or a monocarboxylate group having 1 to 20 carbon atoms or X and X' together form a dicarboxylate group containing 2 to 20 carbon atoms, and at least one cyclodextrin and/or at least one cyclodextrin derivative and optionally at least one pharmaceutically acceptable adjuvant.
Patent CZ-306586-B6 (CZ)
Title: A trigger mechanism for automatic and semiautomatic guns
Inventor: INDRUCH JIŘÍ
IPC: F41A19/37
Filed: 2015-11-11
Abstract: The trigger mechanism for automatic and semiautomatic guns contains the trigger lever (53), the trigger (50) connected to the trigger lever (53) and the container (302) for guiding the rear part of the breech (304). The trigger lever (53) is rotatably connected to the trigger (50) and comprises two arms (54, 55) between which there is a space which the magazine of the gun goes through, connected by the transverse strip (56) onto which there is attached the vertical plate (57), on whose upper side there is the upper claw (59) for tensioning the firing pin (1) and the projection (49) for unlocking the safety lock (46) of the firing pin (1). The trigger (50), the vertical plate (57) and the firing pin (1) are located in a vertical plane of symmetry of the gun and the arms (54, 55) are located symmetrically with respect to this plane.
Patent CZ-307698-B6 (CZ)
Inventor: KÁŇA PAVEL
IPC: A62D1/00
Filed: 2018-05-15
Abstract: Hasicí zařízení využívající k hašení kapaliny a její přeměny v plyn, kdehasicí zařízení či systém má nejméně jedno zařízení pro předehřev hasicí kapaliny, která je aplikována přímo bez rozprašovacích trysek, nebo za pomoci trysek .
Patent CZ-308048-B6 (CZ)
Title: Prefabricated construction system, especially reinforced concrete highway roads
Inventor: ZÁRUBA-PFEFFERMANN JAN
IPC: E01C5/06
Filed: 2018-10-31
Abstract: The system consists of transverse and longitudinal support thresholds (2) and (3) below the joint gaps of the road panels (1) with at least one nut grommet (6) along the longitudinal axis, and are simultaneously used as part of the lifting means for lifting the panels (1) into the desired grade line before they are poured with cement bedding (16). The panels (1) have on the side edge walls of the nut grommets (6) and transverse and longitudinal support thresholds (2) and (3) have openings on the sides of the nut grommets (6). The recesses and holes accommodate the removable plastic plugs (18) and (19) have the shape of the lower portion of the assembly lifting means, which after inserting the plastic plugs into the recesses and openings are inserted for lifting the construction into the desired grade line prior to injection.
Patent CZ-309340-B6 (CZ)
Title: Respirator or face mask
Inventor: HAVRÁNEK PETR
IPC: A62B9/06
Filed: 2020-04-15
Abstract: The respirator or face mask contains a support part (1) for the filter fabric (4) and is formed by a flat flexible structure adapted to be folded into the form of a hollow spatial body. The supporting part (1) has at least one opening (3) for breathing covered with at least one filter layer and at least a pair of protrusions (2) for the clamping element. The support part (1) has a semicircular surface with a pair of radial protrusions (2) approximately a 1/4 of the total length (L) of the circular arc between the radial edges (10) of the support part (1). In the central region of the semi-circular planar shape of the support part (1) there is a moulding (11) and a flap (12) forming the peak (V) of the respirator or face mask when folded into a three-dimensional shape and the radial edges (10) of the support part (1) are adapted to mutual folding and subsequent surface connection to create a conical hollow body of a respirator or face mask. The surface connection of the radial edges (10) is in the direction of the surface of the created spatial body of the respirator or face mask.
Patent SK-278022-B6 (SK)
Title: Catalyst for polymerization of olefins
Inventor: TAKAHASHI TSUTOMU
IPC: C08F4/642
Filed: 1984-12-21
Abstract: Catalyst is preparable by reaction of reactive product I of organoaluminium compound with donor of electrons and titanium(IV) chloride with consecutive reaction of resultant solid product II with donor of electrons and acceptor of electrons and mixing of resultant product III with organoaluminium compound in inert solution at creating of disperse of catalyst, into which is at temperature in range 0 to 70 degrees of Celsius absorbed 2-olefin in mass 0,10 to 0,5 of weight of mass of solid product III with contents 500 and 50 000 ppm carbonylsulfide by preliminary polymerization, which after the organoaluminium compound is added at which the molar ratio of organoaluminium compound to titanium in solid product III in resultant dispersion of catalyst is higher then 13,0 and then is to dispersion of catalyst added reactive product of I'organoaluminium compound and donor of electrons, gained by reaction of 0,1 to 8,0 mols of at least one compound from group of methyl-p-toluylat, triamide of hexamethylphosphoric acid, diphenyl, ethylbenzoat and ethylanisate with 1,0 mol of organoaluminium compound at temperature 20 to 200 degrees of Celsius during 30 second to 5 hours.
Patent SK-285925-B6 (SK)
Title: Method of producing fibres on basis of polyvinyl alcohol and/or partially saponified polyvinyl acetate
Inventor: ALEXY PAVEL
IPC: C08L29/00
Filed: 2003-04-07
Abstract: Method of producing fibres on the basis of polyvinyl alcohol and/or partially saponified polyvinyl acetate with high Young's modulus of elasticity at tension and high strength of fibre consists in the reaction of dry powdered mixture of polyvinyl alcohol and/or partially saponified polyvinyl acetate having a degree of hydrolysis of 95 to 99.9 % mole and a viscosity of 4 % by weight aqueous solution and/or a sol-gel at 20 °C, of 3 to 30 mPas, with a softener in an amount of 3 to 12 % by weight and eventually with peptidic modifier which is an oligomer to polymer having an average molecular weight of 3000 to 30000, containing from 2 to 16 % by weight of nitrogen in an amount of 15 % by weight.
Patent CZ-301178-B6 (CZ)
Title: Process for preparing supported catalyst and use of such a catalyst
Inventor: OHISHI JUNZO
IPC: C07B61/00
Filed: 2000-09-13
Abstract: The present invention relates to a process for preparing a supported catalyst by deposition of a catalytically active component having the composition defined by the formula Moi12ViaWibCuicSbidXieYifZigOih, in which the general symbols have specific meanings, to an inert support. The invention is characterized in that an aqueous solution or a dispersion containing compounds of elements of the catalytically active component is dried wherein said aqueous solution or dispersion contain antimony acetate as a source of antimony, to obtain a composition of the catalytically effective component, the composition of the catalytically effective component is calcined to obtain calcined powder, which is then applied to the support together with crystalline cellulose used as a binder and optionally with a strength-enhancing compound. The invention also relates to the use of the above-described catalyst when preparing acrylic acid.