baber/WOPTO huggingface dataset:
Patent CZ-133998-A3 (CZ)
Title: Thrommbin inhibitors, process of their preparation and pharmaceutical composition containing thereof
Inventor: ADANG ANTON EGBERT PETER
IPC: C07K5/02
Filed: 1996-10-30
Abstract: The invention relates to non-slow-binding thrombin inhibitors of the formula: A-B-C-Lys-D wherein A is H, 2-hydroxy-3-cyclohexyl-propionyl-, R1, R1-O-CO-, R1-CO-, R1-SO2-, -(CHR2)nCOOR3, or an N-protecting group, wherein R1 is selected from -(1-6C)alkylene-COOH, (1-12C)alkyl, (2-12C)alkenyl, (6-14C)aryl, (7-15C)aralkyl and (8-16C)aralkenyl, the aryl group of which may be substituted with (1-6C)alkyl, (2-12C)alkoxy, hydroxy, or halogen; R2 is H or has the same meaning as R1, R3 is selected from H, (1-12C)alkyl, (2-12C)alkenyl, (6-14C)aryl, (7-15C)aralkyl and (8-16C)aralkenyl, the aryl group of which may be substituted with (1-6C)alkyl, (2-12C)alkoxy, hydroxy or halogen; n is an integer of 1 to 3; B is a bond, L-Asp or an ester derivative thereof, Leu, norLeu, -N(benzyl)-CH2-CO-, -N(2-indane)-CH2-CO-, D-1-Piq, D-3-Piq, D-Tiq, Atc or a D-amino acid having a hydrophobic aromatic side chain; C is Azt, Pro, Pec, norLeu(cyclo)Gly, an amino acid of one of the formulae -N[(3-8C)cycloalkyl]-CH2-CO- or -N(benzyl)-CH2-CO-, D is selected from COOH, tetrazole, oxazole, thiazole and benzothiazole, or A and C have the aforesaid meanings, B is D-(3-8C)cycloalkylalanine, and D is tetrazole, oxazole, thiazole or benzothiazole; or a prodrug thereof; or a pharmaceutically acceptable salt thereof; with the exception of the compound Me-D-Phe-Pro-Lys-COOH. The compounds can be used as antithrombotic agents.
Patent CZ-146398-A3 (CZ)
Title: Agricultural soil treating implementing entral adjusting device for adjusting working depth
Inventor: GEBBEKEN MARTIN DIPL-ING
IPC: A01B33/02
Filed: 1998-05-12
Abstract: The soil cultivator is especially in the form of a circular spike harrow. It has at least two implement units (2) which fold over inwards and have rollers positioned after them. The rollers (3) are swivel-connected by arms (4) to the implement units and have depth-adjusters (6,7) for the unit. Each roller is joined to its implement unit by at least two arms which have one adjustment acting as a depth-restrictor and or stop-piece and have a central adjustment (30).
Patent CZ-157494-A3 (CZ)
Title: Derivative of 5-amino-8-methyl-7-pyrrolidinylquinoline-3-carboxylic acid, stereoisomer and salt thereof, process for preparing said derivative and pharmaceutical composition containing thereof
Inventor: YASUO ITO
IPC: C07D215/56
Filed: 1994-06-27
Abstract: A 5-amino-8-methyl-7-pyrrolidinylquinoline-3-carboxylic acid derivative represented by the general formula: <CHEM> wherein R<1> is a hydrogen atom or a lower alkyl group; R<2> is a hydrogen atom, a lower alkyl group, a lower alkanoyl group, a halogenated lower alkanoyl group or a residue of carboxylic acid ester; R<3> is a hydrogen atom or a lower alkyl group; R<4> , R<5> or R<6> are each independently a hydrogen atom or a lower alkyl group; or two of R<4>, R<5> and R<6> may be taken together to form a -(CH2) n - group wherein n is 1 or 2, a stereoisomer thereof, or a pharmacologically acceptable salt thereof, the process for preparing these compounds, a pharmaceutical composition comprising an effective amount of these compounds and methods for the treatment of infectious diseases through the administration to patients of an effective amount of these compounds, and intermediates of these compounds are disclosed. These compounds are effective as antibacterial agents.
Patent CZ-160697-A3 (CZ)
Title: Waste water or sewage disposal plant
Inventor: TOPOL JAN ING
IPC: E03F1/00
Filed: 1997-05-26
Abstract: In the present invention there is disclosed a waste water disposal plant consisting of waste water treatment plants being connected to local sources of waste water, where a tank (4) of treated water with a pump (5) for pumping purified water into a pressurized branch (9) and further to a collecting piping (11) being provided with a central checking place (12) and leading out in a recipient forms an integral part of each domestic sewage plant (3). The pressurized branch (9) is provided in front of connection to the collecting piping with a ground closing fitting (10). The purified water tank (4) can be represented by an existing cleaned up cesspool, respectively a septic tank.
Patent CZ-201339-A3 (CZ)
Inventor: WOLF JAN
IPC: G01N33/50
Filed: 2013-01-18
Abstract: ﻿Řešení popisuje způsob manipulace se vzorky biologického materiálu, zejména pro molekulární diagnostiku nebo pro izolaci nukleových kyselin. Vzorek biologického materiálu se na počátku procesu vloží do vkládací komory (11) prostředku pro manipulaci se vzorky biologického materiálu, v jehož zásobních komorách (12) byly před tím odděleně od sebe uloženy všechny pro příslušný proces potřebné reagenční chemikálie, přičemž následující etapy procesu probíhají uvnitř prostředku bez přímé manipulace obsluhy s reagenčními chemikáliemi, které se postupně mísí a reagují, přičemž nežádoucí zbytky z reakcí se ukládají do odpadní komory (41), která se nachází rovněž uvnitř prostředku a je bezpečně oddělena od ostatních prostor prostředku, obsluhy i okolí.
Patent CZ-9602691-A3 (CZ)
Title: Expanding dowel
Inventor: SCHAFFER MARC DIPL ING
IPC: F16B13/06
Filed: 1996-09-13
Abstract: The dowel consists of a sleeve (1) the end of which has longitudinal slits (4). The end with slits is spread on mounting by a bolt with conical head which is forced into the sleeve. The sleeve further incorporates a zone which allows the sleeve to be compressed endways.   The compression zone is formed by two sets of sicked shaped slots in the sleeve wall. The pointed ends of the slots face one another and slightly overlap so that strips (12) are formed which are bent when force is applied to the end of the sleeve by the bolt.
Patent CZ-283194-A3 (CZ)
Title: System of extensible rods with electomagnets for control device of a rotary dobby machine
Inventor: VINCIGUERRA COSTANTINO
IPC: D03C1/00
Filed: 1994-11-17
Abstract: An electromagnet-striker bar system for the control device of a rotary dobby comprising an amagnetic container (13) of extremely rigid box structure into which the iron cores (14) of the electromagnets are equidistantly inserted and irreversibly locked, on the electromagnet pole pieces (14') there being mounted amagnetic spools (18) for supporting the electrical windings (19), said container (13) being provided in that side further from the hinging axis (2) of said striker bars (1) with a longitudinal groove (11) into which are inserted the amagnetic support and slide shoulders (10) for the free ends (1'') of the striker bars hardened by heat treatment. <IMAGE>
Patent CZ-9403256-A3 (CZ)
Inventor: STEFAN LIBOR ING
IPC: B04B9/10
Filed: 1994-12-21
Abstract: Způsob řízení otáček rotoru odstředivky s ohledem na velikost
mechanického kmitání odstředivky, kdy řízení otáček rotoru se
provádí na základě technologického řídícího systému a na
základě aktuální zjištěné úrovně mechanického kmitání
odstředivky, kdy se rozlišují tři, předem stanovené, vzestupně
uspořádané úrovně mechanického kmitání odstředivky, nárůst
otáček )10) rotoru (2) se provádí pokud aktuální velikost
mechanického kmitání (6) odstředivky (1) je nižší než druhá,
střední, předem stanovená hodnota úrovně (8) mechanického
kmitání odstředivky (1), přičemž po předchozím překročení
druhé, střední, úrovně (8) mechanického kmitání se provádí
nárůst otáček (10) rotoru (2) pokud aktuální velikost
mechanického kmitání (6) odstředivky (1) není vyšší než
první, nejnižší, předem stanovená hodnota úrovně (7)
mechanického kmitání odstředivky (1), že snižování otáček
(10) rotoru (2) se provádí, pokud aktuální velikost
mechanického kmitání (6) odstředivky (1) překročí třetí,
nejvyšší, předem stanovenou hodnotu úrovně (9)
mechanického kmitání odstředivky (1) a to do té doby, pokud
aktuální velikost mechanického kmitání (6) odstředivky (1)
není nižší než druhá, střední, předem stanovená hodnota
úrovně )8) mechanického kmitání odstředivky (1).
Patent CZ-338997-A3 (CZ)
Title: 9-n-ethylene derivatives of 9(s)-erythromycylamine
Inventor: KUJUNDZIC NEDJELJKO D SC
IPC: A61K31/7042
Filed: 1997-10-24
Abstract: The invention relates to 9-N-ethenyl derivatives of 9(S)-erythromycylamine, new semisynthetic antibiotics of the macrolide class of the general formula (I) <CHEM> wherein R<1> and R<2> are the same or different and represent nitryl, a carboxyl group of the formula COOR<3>, wherein R<3> represents a C1-C4 alkyl group, or a keto group of the formula COR<4>, wherein R<4> represents a C1-C4 alkyl group, to their pharmaceutically acceptable addition salts with inorganic or organic acids, to a process for their preparation, to a process for the preparation of the pharmaceutical compositions as well as to the use of the obtained pharmaceutical compositions in the treatment of bacterial infections.
Patent SK-126197-A3 (SK)
Title: Stent with variable features to optimize support and method of making such stent
Inventor: RICHTER JACOB
IPC: A61F2/82
Filed: 1997-09-18
Abstract: An intravascular stent especially suited for implanting in curved arterial portions or ostial regions. The stent can include an end region which is fabricated to have a greater radial strength than the remaining axial length of the stent. Such a stent is particularly suited for use in ostial regions, which require greater support near the end of the stent. The stent alternatively can include sections adjacent the end of the stent with greater bending flexibility than the remaining axial length of the stent. Such a stent is particularly suited for use in curved arteries. The stent can also be constructed with an end that has greater radial strength and sections adjacent the end with greater bending flexibility. Such a stent prevents flaring of the stent end during insertion. <IMAGE>
Patent SK-136898-A3 (SK)
Title: Safety circuit
Inventor: BRITZ WOLFGANG
IPC: F15B20/00
Filed: 1997-01-17
Abstract: The invention relates to a safety circuit for controlling a hydraulic drive (10) with a drive part (12) movable in at least two different directions of movement and controllable for any movement  by a control switching circuit. A safety circuit which ensures the required safety function in an absolutely safe manner, even in the event of a power failure, is obtained in that at least one safety switching circuit is hydraulically combined with the control switching circuit in such a manner that when the latter is switched off the drive part (12) can only be controlled by the respective safety switching circuit. Consequently, the highest-priority operation provided in an emergency, for example in the form of the defined closing or opening of a vapour control valve, is safely executed and the otherwise usual control process is interrupted by the control switching circuit.
Patent SK-152195-A3 (SK)
Title: Compounds of the secomacrolide and secoazalide class and preparaton method thereof
Inventor: LAZAREVSKI GORJANA
IPC: C07D407/12
Filed: 1995-12-01
Abstract: The present invention refers to the new compounds of formula (I) of the secomacrolide and secoazalide class, a process for the preparation thereof as well as to new intermediates of formula (II) for the preparation of these seco derivatives.
Patent SK-163898-A3 (SK)
Title: Absorbent structure, and production of absorbent structure by mat formation together with adhesive-bonded layer
Inventor: ROSSELAND BERIT
IPC: D04H1/425
Filed: 1997-05-23
Abstract: Absorbent structure (1) consisting of an absorbent material layer (2) of adhesive-free cellulose fibres (4) and an airlaid material layer (3) of adhesive-bonded cellulose fibres (5), and a method for producing an absorbent structure (1) which is intended for use in an absorbent article. The layers are bonded together by means of the adhesive of the airlaid material (3) functioning as a binding material and fibres (4) from the absorbent material layer (2) extending into the airlaid material (3). In the method, the absorbent material (2) is mat-formed on an airlaid material (3). Alternatively, the absorbent material (2) is mat-formed and an airlaid material (13) is then laid on top of it. After the material layers have been laid together, they are compressed (24) at a temperature in excess of 100  DEG C. During the compression (24), the adhesive of the airlaid material is softened, and the two layers are bonded together. Some of the fibres (4) from the absorption material (2) also penetrate down into the airlaid material (3) and further connection between the layers is achieved.
Patent SK-175198-A3 (SK)
Title: Bisphosphonate derivatives of hydroxy steroids, process for their preparation and pharmaceutical composition containing them
Inventor: GALLAGHER JAMES A
IPC: A61K31/565
Filed: 1997-06-26
Abstract: Bisphosphonate derivatives of hydroxy steroids which are bone resorption inhibitors or bone formation stimulators, the derivatives having at least one group A in place of a hydroxy group on the steroid molecule, where A is a group of formula (A) where X is: (i) St-O-CO- where St is the residue of the hydroxy steroid given by removal of an OH group; (ii) R<1>-O-CO- where R<1> is an alkyl, alkenyl, cycloalkyl, aralkyl or aryl group, any of which may optionally be substituted; or (iii) a hydrogen atom, and the salts and solvates of these compounds. The steroid is typically 17 beta -oestradiol, oestrone, testosterone, norethindrone, androsterone, norethandrolone or nandrolone. The derivatives can be used in the treatment of bone disorders such as osteoporosis.
Patent SK-622021-A3 (SK)
Title: Waste container lid with vertical information surface
Inventor: VORONIČOVÁ ADRIANA
IPC: B65F1/16
Filed: 2021-08-17
Abstract: Waste container with a vertical information surface has a lid (3), while a panel (1) is attached to the underside of the lid (3) with the help of a movable joint (2), which is a carrier of information.
Patent WO-9322720-A3 (WO)
Inventor: VACARIU CORNELL
IPC: G06F7/52
Filed: 1993-04-29
Abstract: A novel process and a pure hardware and architecturally symmetrical division circuit is described which recursively and bidirectionally finds a quotient from a dividend and a divisor by approximation. It is thus possible to start the calculation with the highest or lowest position value or at the same time with the two extremes of the divisor/divident/quotient, in a parallel process. The division circuit therefore consists of four parts, with two symmetrical pairs. The left-hand main circuit (1), which is symmetrical with the right-hand sub-circuit (3), processes the divisor and, via the two control signals D/I and AS, controls the left hand sub-circuit (2) which is symmetrical with the right-hand sub-circuit (4) and processes the dividend in order to find the quotient. The two symmetrical parts can operate mutually independently, i.e. separately, thus making it possible to perform two different division operations at the same time via the two symmetrical halves. The division process can thus be performed bidirectionally or on one side (left or right). The operands may be represented in a non-redundant format or in a digit format with a sign, where 'carry-ripple' transfer can be prevented by the representation strategy of the 'non-neighbouring non-zero trits' and a region centred on '1' will be alocated to the absolute value of the mantissa (M) after the standardisation process.
Patent WO-9415566-A3 (WO)
Title: Train de roulement
Inventor: DU-BOIS ROBERT LEO
IPC: B62B3/02
Filed: 1994-01-04
Abstract: Train de roulement, en particulier pour civière, qui possède un système permettant le réglage à différentes hauteurs, et que le manipulateur n'a pas à élever ou à abaisser manuellement lorsque ladite civière est chargée dans une ambulance, ou lorsqu'elle en est déchargée. Ledit train de roulement comporte une structure (10) de support rectangulaire, un châssis (11) réglable en hauteur muni de roulettes et doté d'une première et d'une seconde paires de jambes pliables (23, 24; 31, 32) et un dispositif de réglage de la hauteur. Ledit dispositif de réglage de la hauteur comporte une ou plusieurs courroies de liaison (46, 47) reliées aux première et seconde paires de jambes et à la structure de support, qui peuvent se rétracter ou s'étendre de manière à étirer ou à plier les première et seconde paires de jambes pour régler la hauteur de la structure de support.
Patent WO-0212799-A3 (WO)
Title: Dispositif pour l'utilisation d'energie solaire concentree
IPC: F24S23/79
Filed: 2001-08-06
Abstract: L'invention concerne un dispositif pour l'utilisation d'énergie solaire concentrée. Ce dispositif comporte un concentrateur (1) primaire linéaire constitué d'un ou de plusieurs miroirs, qui collecte le rayonnement solaire et le réfléchit vers un absorbeur (2) oblong placé parallèlement au concentrateur primaire ; et un concentrateur (3) secondaire placé au-dessus de cet absorbeur. Le concentrateur (1) primaire est dirigé vers l'absorbeur (2) de manière à former trois lignes (20, 21, 22) focales parallèles à l'absorbeur (2).
Patent BE-1003077-A3 (BE)
Title: Copolymeres lineaires a sequences alternees et procede pour les preparer.
Inventor: AGOSTINIS ENRICO
IPC: C08L53/00
Filed: 1989-11-24
Granted: 1991-11-12
Abstract: L'invention concerne des copolymères linéaires comportant quatre séquences alternées, représentés par la formule suivante : B1 - T - A1 - B2 - A2 dans laquelle A1 et A2 sont des séquences poly(vinyl-aromatique), B1 et B2 sont des séquences constituées de copolymères d'éthylène et de butène-1 ou d'éthylène et de propylène, et T est un segment terpolymère statistique formé de motifs de monomères éthylène, propylène et vinyl-arène ou éthylène, butène-1 et vinyl-arène. Ces copolymères présentent une masse moléculaire moyenne en poids comprise entre 20.000 et 300.000, et une teneur totale en motifs vinyl-aromatiques comprise entre 10 et 60% en poids.
Patent BE-1004813-A3 (BE)
Title: Optische zender/ontvangerinrichting.
Inventor: SIERENS CHRISTIAAN HENDRIK JOZ
IPC: H04J14/08
Filed: 1991-05-08
Granted: 1993-02-02
Abstract: Optische zender/ontvangerinrichting voor het overdragen van informatiesignalen (S1, Sn), van een zenderinrichting (T) naar een ontvangerinrichting (R) over een optsiche golfgeleider (L). Dit gebeurt door elektrische subdraaggolven, aan de hand van modulatiemiddelen (M1,.Mn) te moduleren met deze informatiesignalen (S1,., Sn) en om te zetten naar optische signalen aan de hand van omzetters (E/01,., E/01n) en deze gebruik maken van tijdmultiplexeermiddelen (TDM1,., TDMn) over te dragen in verschillende tijdssleuven (t1,., tn) wanneer deze subdraaggolven dezelfe frekwentie hebben. De modulatie- en tijdsmultiplexeermiddelen worden gestuurd door bijbehorende individuele besturingsmodules /c1,., Cn) onder toezicht van een centrale besturingsmodule (CC) welke zich in de ontvangerinrichting (R) bevindt.
Patent BE-1005752-A3 (BE)
Title: Acoustic screen device
IPC: E04B1/84
Filed: 1992-03-24
Granted: 1994-01-18
Abstract: An acoustic screen device with a supporting system (1) which has niches(10) for the incorporation of sound-absorbing elements (3), with apre-determined mass, whereby at least one elastic element is fitted betweeneach sound absorbing element (3) and the corresponding niche (3) for theelastic suspension of the said sound absorbing element (3), in such afashion that this results in an individual frequency which is dependant onthe pre-determined mass and the elasticity of the stated elastic element(s).<IMAGE>
Patent BE-1007612-A3 (BE)
Title: Schakelinrichting.
Inventor: OVERGOOR BERNARDUS J M
IPC: H02H9/02
Filed: 1993-10-11
Granted: 1995-08-22
Abstract: De uitvinding heeft betrekking op een schakelinrichting voor het bedrijven van een last (La) met behulp van een voedingsspanning voorzien van -ingangsklemmen (K1,K2) voor aansluiting op polen van een voedingspanningsbron, - een circuitdeel V voor het beperken van een tijdens bedrijf ten gevolge van de voedingsspanning door de ingangsklemmen vloeiende ingangsstroom, bevattende een eerste veldeffecttransistor S1 voorzien van twee hoofdelectrodes en een stuurelectrode en zodanig gekoppeld met een ingangsklem dat de ingangsstroom tijdens bedrijf door beide hoofd electrodes (K3,K4) van de veldeffecttransistor S1 vloeit. Volgens de uitvinding is de eerste veldeffecttransistor S1 van het type ''depletion FET'' en uitsluitend via de hoofdelectrodes gekoppeld met de ingangsklemmen. Hiermee is bereikt dat de ingangstroom met behulp van relatief eenvoudige middelen wordt begrensd.
Patent BE-1011595-A3 (BE)
Title: Improved heat exchanger and method to realise such a heat exchanger
Inventor: WAUMANS ERIK
IPC: F28D9/04
Filed: 1997-12-09
Granted: 1999-11-09
Abstract: An improved heat exchanger, characterised by the fact that it mainly consists of at least one path formed by a layer of flexible foil (2) on which at least one side of local sealing or swellings (4-11-13-14-15-18-19) are applied in order to form the inlets and outlets (8-9-20-21), where this (these) path (paths) is (are) rolled in such a way that the windings wound next to each other form passages (3) for two or more liquids.<IMAGE>
Patent WO-0127630-A3 (WO)
Title: Procede permettant d'identifier des composants modulant l'activite neuronale
Inventor: SNUTCH TERRANCE P
IPC: A61P25/28
Filed: 2000-10-13
Abstract: On a démontré qu'une séquence d'acides aminés spécifique, située du côté proximal de la terminaison carboxy des canaux ioniques de type P/Q régule, en se liant avec la protéine Homer, l'expression du gène codant pour la syntaxine-1A. Cette région du canal ionique du calcium du type P/Q comprend des peptides qui peuvent être utilisés pour l'identification de composants modulateurs du système nerveux central.
Patent WO-0172607-A3 (WO)
Title: Corps de conteneur pour vehicule de collecte de dechets recyclables
Inventor: DURON ALAIN
IPC: B65F3/08
Filed: 2001-03-26
Abstract: L'invention concerne un conteneur de collecte de déchets monté sur un véhicule. Le conteneur est particulièrement adapté pour séparer et compacter des matériaux recyclables en raison de la présence d'un séparateur diagonal s'étendant de façon longitudinale. Le conteneur possède une paire de godets de réception de déchets adaptés de préférence pour être levés afin de se trouver en alignement avec des ouvertures situées dans la paroi frontale du conteneur. Les matériaux recyclables, triés par type dans les godets, sont ensuite introduits dans le conteneur par une lame de compactage placée dans chaque godet. Le déchargement des matériaux est facilité par un mouvement pivotant du séparateur avant que le véhicule ne soit placé en position de déversement. Le séparateur est extensible de sorte que, quant il est placé diagonalement par rapport aux parois latérales du conteneur, le séparateur s'étend jusqu'à l'extrémité de décharge du conteneur.
Patent CZ-2000408-A3 (CZ)
Title: Process for producing steel rolling-contact bearing rings
Inventor: TENBRACK KARL
IPC: F16C33/64
Filed: 1998-07-01
Abstract: A method for producing steel rolling bearing rings, starting from a hot-rolled tube, the structure of which is similar to a spheroidized structure and from which rings of the same continuous length are hot-cut while supplying a lubricant and, after cooling, are further processed. The hot-cutting takes place at a temperature below the transformation temperature of the rolling bearing steel used but above 720° C., with subsequent cooling in static air. From the blank ring a green or soft ring of a rolling bearing ring is produced with narrow tolerances of its shaped elements by an optimally timed multistage machining type of cold further processing operation, the main element of the cold further processing being a turning operation.
Patent CZ-2002900-A3 (CZ)
Title: Protective film based on modified polymer mixture
Inventor: SCHOTTA MIROSLAV
IPC: C09D129/04
Filed: 2002-03-13
Abstract: The protective film with enhanced adhesion to the skin constitutes of a modified compound on the basis of a alcoholic polyvinilalchol solution of the following proportion: 1 to 50 weight perc. of polyvinilalcohol, 5 to 70 weight perc. of alcohol C1 to C10 series, to 40 weight perc. of magnesium chloride, 0.1 weight perc. of acticide preservant and distilled water to 100 weight perc.