baber/WOPTO huggingface dataset:
Patent AU-633858-B2 (AU)
Title: Arylpiperidine derivatives
IPC: C07D211/22
Filed: 1989-12-04
Granted: 1993-02-11
Abstract: N-alkyl or oxyalkyl arylpiperidine cpds. of formula (I) are new. In (I), Ar = Ph, fluorophenyl, chlorophenyl, trifluoromethylphenyl, methoxyphenyl, tolyl or naphthyl opt. substd. with F, Cl, CF3 or OMe; n= 2-4; X= O, S or a direct bond; R= Ph, hydroxyphenyl, methoxyphenyl, tolyl, 2-amino-4-thiazolylphenyl, 5-oxindolyl, 2-methyl-4-oxo-4H-pyrido (1,2a)pyrimidin-3-yl, 7,9-dioxo-8-azaspiro(4,5)decan-8-yl or 1,8,8-trimethyl-2,4-dioxo -3-azabicyclo(3.2.1)heptan-3-yl. - Also new are arylpiperidine cpds. (II) from which (I) are prepd.. - (I) can be prepd. by reacting (II) with at least an equiv. amt. in moles of an aralkyl (or aryloxyalkyl) or heterocyclyl ether deriv. or corresp. halide of formula: Q(CH2)nXR where Q= a leaving gp. (e.g. p-toluenesulphonyloxy or halogen) in a reaction-inert polar organic solvent (partic. acetone or MIBK), under anhydrous conditions, in the presence of at least an equiv. amt of an appropriate base (partic. Na2CO3 or K2CO3). A temp. of 50-150 deg.C for 2-24 hrs. is used.
Patent AU-671846-B2 (AU)
Title: Apparatus for simultaneous supply of particles, the apparatus provided further with a function to remove the particles by suction, and methods for production of patterned shaped articles using these apparatus
Inventor: UCHIDA HIROSHI
IPC: B28B1/00
Filed: 1993-09-06
Granted: 1996-09-12
Abstract: An apparatus for simultaneously supplying at least two kinds of particles (B, W, R, S, Br) onto a given surface (18, 30) includes a movable supply head (10) having at least one partition member (12) for partitioning the at least two kinds of particles and defining at least two supply ports (11, 11A, 11B) in conjunction with the supply head, and a device (14, 16, 32, 34, 35) for introducing the at least two kinds of particles into the supply head. A patterned shaped article is produced by a method using the apparatus. The method includes simultaneously supplying the supply ports of the supply head, with the one partition member abutting on the given surface, thereby forming a pattern course on the given surface, and allowing the pattern course to set into an integral mass. <IMAGE>
Patent AU-660108-B2 (AU)
Title: Particles for NMR imaging and method of manufacture
Inventor: TOURNIER HERVE
IPC: A61B5/055
Filed: 1993-07-30
Granted: 1995-06-08
Abstract: Magnetite particles suitable for injection into the blood stream of patients having enhanced resistance against agglomeration and uptake by the RES of the liver and spleen. The particles essentially consist of an iron oxide core and a phosphoric acid mono alkyl or alkenyl ester or glycerophospholipid/surfactant three dimensional shell surrounding the core. The core and the monoester or a micellar glycerophospholipid form an urchin-like structure which is further interlaced or intertwined with a non-ionic surfactant to produce a protective three dimensional shell which renders particles almost undetectable by the macrophages. Particles prepared according to the invention are kept in the blood circulation for long periods and represent excellent long lasting blood pool agents. Key components in the shell are (a) a polybasic mineral-organic species such as glycero phosphatidic acid in micellar form and (b) a block copolymer having successive hydrophilic and hydrophobic segments.
Patent AU-625309-B2 (AU)
Title: Flexible medical solution tubing
Inventor: MUELLER WALTER BERNDT
IPC: A61L29/08
Filed: 1990-01-11
Granted: 1992-07-09
Abstract: A medical solution tubing (20) useful in combination with medical solution packages and pouches includes an intermediate layer (24) comprising a polymeric material which imparts flexibility to the film; an inner layer (26) comprising a heat resistant polymer; and an outer layer (22) of polypropylene, ethylene propylene copolymer, or modified ethylene propylene copolymer.
Patent AU-658127-B2 (AU)
Title: Secondarily contained fluid supply system
Inventor: WEBB MICHAEL C
IPC: F16L55/00
Filed: 1989-12-22
Granted: 1995-04-06
Abstract: A secondarily contained piping system has two spaced access chambers interconnected by a secondary containment pipe to provide a sealed housing for a flexible fluid supply pipe, the ends of which are disposed within the access chamber and have a connector element at each end forming a section adaptable to be interconnected to other fluid conduits, the diameter and bending radius of the fluid supply pipe and the size of the access chamber permitting the fluid pipe after uncoupling to readily be removed from the secondary containment pipe through one of the access chambers.
Patent AU-532187-B2 (AU)
Title: Sugar derivatives of c-076 compounds
Inventor: FISHER MICHAEL HERBERT
IPC: C07H19/01
Filed: 1979-07-24
Granted: 1983-09-22
Abstract: The invention provides derivatives of C-076, which is a series of macrolides, in which the substituents are sugar or saccharide groups. The sugar groups are substituted on any of the available hydroxy groups of the C-076 molecule by various known procedures. The compounds thus produced, which have the structural formula: 
<CHEM>
 in which the broken line indicates that a single or double bond is present in the 22(23) position; R1 is hydroxy, loweralkanoyloxy, or glycosyloxy, and is present only when the borken line indicates a single bond; R2 is iso-propyl or sec-butyl; R3 is hydrogen, methyl, loweralkanoyl or glycosyl; and R is hydrogen, loweralkanoyl, glycosyl, 
<CHEM>
 where R4 is hydrogen, loweralkanoyl or glycosyl; in which the glycosyl groups are polyhydroxy (5 or 6)-membered cyclic acetals that are optionally substituted with lower alkyl and in which the hydroxy groups may be optionally substituted with lower alkyl or loweralkanoyl and their mono-unsaturated derivatives; provided that at least one of R, R1, R3 or R4 must contain a glycosyl group, and that if only R contains a glycosyl group, that group is other than  alpha -L-oleandrosyl or  alpha L-oleandrosyl- alpha -L-oleandrosyl, have profound anthelmintic, insecticidal, ectoparasiticidal and acaracidal activity and compositions for such uses are also disclosed.
Patent AU-587597-B2 (AU)
Title: Tricyclic compounds, compositions containing such compounds, processes for their preparation and method of treatment therewith
Inventor: WILLMAN NILS-ERIC
IPC: C07D409/06
Filed: 1986-01-10
Granted: 1989-08-24
Abstract: The invention concerns:Novel dibenz/b,e/oxepin and dibenz/b,e/thiepin compounds having the general formula:wherein X is 0 or S,R<sup>1</sup>, <sub>R</sub><sup>2</sup>, R3 and R<sup>4</sup> are the same or different and are each selected from the group consisting of hydrogen, lower alkyl, lower alkenyl, lower alkynyl, lower cycloalkyl, lower alkoxy, lower alkylthio, lower alkylsulphinyl, lower alkylsulphonyl, halogen, trifluoromethyl, trifluoromethylthio, lower dialkylsulphonamido, nitro, hydroxy, cyano, carbamyl, carboxy, lower alkoxycarbonyl, amino, N-lower alkylamino, N,N-diloweralkylamino, lower acylamido, lower alkanesulfonamido and lower acyl and, when on adjacent carbon atoms at the positions 2 and 3 and/or 8 and 9, two of the substituents R<sup>1</sup> and R<sup>2</sup> or R<sup>3</sup> and R<sup>4</sup> taken together may form a methylenedioxy group;R<sup>5</sup> and R<sup>6</sup> are the same or different and are selected from the group consisting of hydrogen, lower alkyl, lower alkenyl, lower aklynyl, lower cycloalkyl, aralkyl, lower hydroxyalkyl, lower aminoalkyl, lower alkylaminoalkyl, lower dialkylaminoalkyl, lower alkoxyalkyl and together with the nitrogen atom, R<sup>5</sup> and R<sup>6</sup> may form a 5- or 6-membered ring, such as pyrrolidine, piperidine, morpholine, piperazine, and N-lower alkyl or N-hydroxy lower alkyl substituted rings such as N-alkylpiperazine or N-hydroxyalkyl piperazine or the like;R<sup>7</sup> is hydrogen or lower alkyl; optionally in the form of addition salts with pharmaceutically acceptable inorganic or organic acids and optionally in the form of essentially pure enantiomers.The invention also includes compositions containing the novel compounds, processes for their preparation and a method of treatment therewith.The compounds have pharmacological effects.
Patent AU-624230-B2 (AU)
Title: Low amylose food product
Inventor: LEWIS VICTOR MARCUS
IPC: A23L29/20
Filed: 1990-03-29
Granted: 1992-06-04
Abstract: The invention concerns a cereal food product comprising a "waxy" cereal chosen from barley, corn, rice or sorghum or from other starchy seed or tissue material wherein less than about 10% of the starch present is amylose, and preferably the starch contains substantially no amylose. Preferably the cereal is waxy barley. The major part of the starch present is also in its ungelatinised form. A process for preparing the food cereal is also described. The cereal food product is preferably a quick cooking hot porridge-like breakfast food.
Patent AU-578876-B2 (AU)
Title: Curable copolymers, a process for their preparation and their use
Inventor: JUST CHRISTOPH
IPC: C08F246/00
Filed: 1986-02-07
Granted: 1988-11-03
Abstract: Copolymers based on (A) 5-95% by weight of at least one polymerizable carbamoyloxyalkyldicarboxylic acid ester, carrying hydroxyl groups, of the general formula I   <IMAGE>   in which R1 represents hydrogen or alkyl or hydroxyalkyl having in each case 1 to 30 carbon atoms in the alkyl radical, R2 represents alkyl or hydroxyalkyl having in each case 1 to 30 carbon atoms in the alkyl radical, or the radical <IMAGE>  subject to the proviso that R1 is hydrogen and x is an integer from 2 to 10, R3 represents linear or branched alkylene having 2 to 5 carbon atoms, R4 represents hydrogen or methyl and R5 represents hydroxyalkyl or hydroxyaminoalkyl having in each case 2 to 20 carbon atoms in the alkyl radical, or an alkyl radical of this type which also contains ester groups and/or ether groups, and (B) 5-95% by weight of at least one copolymerizable monomer belonging to the group comprising (a)  alpha , beta -olefinically unsaturated monocarboxylic acid and alkyl and hydroxyalkyl esters thereof having in each case 1 to 18 carbon atoms in the alkyl radical, and amides and nitriles thereof, and also monoalkyl and dialkyl esters of  alpha , beta -olefinically unsaturated dicarboxylic acids having 1 to 18 carbon atoms in the alkyl radical, (b) vinyl-aromatic monomers, (c) vinyl esters of organic monocarboxylic acids having 1 to 18 carbon atoms in the carboxylic acid radical, and (d) glycidyl esters of unsaturated monocarboxylic and/or dicarboxylic acids, the sum of the components (A) and (B) being in all cases 100% by weight, and a process for their preparation. The copolymers are used for the preparation of shaped articles and/or coatings which have excellent properties.
Patent AU-755115-B2 (AU)
Title: New cyclic compounds having a cycloalkylene chain, a process for their preparation and pharmaceutical compositions containing them
Inventor: LANGLOIS MICHEL
IPC: A61K31/395
Filed: 1999-10-12
Granted: 2002-12-05
Abstract: Cycloalkene substituted cyclic derivatives (I) are new. Cycloalkene substituted cyclic derivatives of formula (I), their enantiomers, diastereoisomers and their acid or base addition salts are new. A = a group of formula (i) or (ii) (optionally substituted by Ra, ORa, OH, CORa, formyl, COORa, COOH or OCORa; Ra = 1-6C alkyl, 2-6C alkenyl, 2-6C alkynyl, 1-6C polyhaloalkyl, 3-8C cycloalkyl, 3-8C cycloalkyl-(1-6C) alkyl, 3-8C cycloalkenyl, 3-8C cycloalkenyl-(1-6C) alkyl (all optionally substituted with at least one OH, 1-6C alkoxy, 1-6C alkyl, 1-6C polyhaloalkyl, amino or halo), aryl, aryl-(1-6C) alkyl, heteroaryl or heteroaryl-(1-6C) alkyl; X, Y' = O, S or CH2; D' = benzene or naphthalene; a-d = single or double bond; Z = O, S, CH2 or NR<1>; R<1> = H, 1-6C alkyl, aryl or aryl-(1-6C) alkyl; D'' = benzene or pyridine; R = H, halo, OH, SH, Ra, ORa, S(O)nRa or a (un)saturated 5- to 7-membered ring of formula (iii) (optionally substituted with at least one 1-6C alkyl, 1-6C alkoxy, carboxy, 1-6C alkoxycarbonyl, OH or =O); n = 0-2; E = O or -S(O)n-; G1, G2 = single bond, -(CH2)t- (optionally substituted with at least one OH, COOH, formyl, Ra, ORa, COORa, CORa or halo; p, q = 0-4; p + q = 1-4; B' = -NR<1>aC(Q)R<2>a, -NR<1>aC(Q)NR<2>aR<3>a or -C(Q)NR<1>aR<2>a; R<1>a-R<3>a = H or Ra; Q = O or S; aryl = phenyl, naphthyl, biphenyl (all optionally substituted with at least one OH, 1-6C alkoxy, 1-6C alkyl, 1-6C polyhaloalkyl, CN, COOH, 1-6C alkoxycarbonyl, NO2, amino or halo); heteroaryl = 5- to 10-membered mono- or polycyclic aromatic ring containing 1-3 N, O or S (optionally substituted with at least one OH, 1-6C alkoxy, 1-6C alkyl, 1-6C polyhaloalkyl, CN, COOH, 1-6C alkoxycarbonyl, NO2, amino or halo); and provided that q = 0 and p = 4, or q = 4 and p = 0 do not apply, when A is naphthyl (optionally substituted with methoxy or methyl), G1 and G2 are single bonds and B' is a group of formula (iv) or NHCOCH3; that A is other than halo substituted naphthyl, when G1 is a single bond and p + q is 1; B' is other than urea, when A is indolyl substituted on position 2 with a group of formula (v); and that B' is other than CONH-aryl, when A is indolyl substituted on position 2 with carboxyl or alkoxycarbonyl, p is 1, q is 0 (p is 0 and q is 1) and G1 is single bond. A Independent claim is also included for the preparation of (I).
Patent AU-645752-B2 (AU)
Title: N-phenylalkyl substituted alpha-amino carboxamide derivatives and process for their preparation
Inventor: DOSTERT PHILIPPE
IPC: C07C231/10
Filed: 1990-05-25
Granted: 1994-01-27
Abstract: N-phenylalkyl substituted  alpha -amino carboxamide derivatives of formula (I) <CHEM> wherein R is C1-C8 alkyl, C3-C8 cycloalkyl, furyl, thienyl, pyridyl or unsubstituted or substituted phenyl; A is a -(CH2)m- or -(CH2)p-X-(CH2)q- group wherein X is -O-, -S- or -NR4-; R1, R2, R3, R min 3, R4, n, m, p and q are as herein defined; and each of R5 and R6 is independently hydrogen or C1-C6 alkyl, and the pharmaceutically acceptable salts thereof, are active on the central nervous system and can be used as anti-epileptic, anti-Parkinson, neuroprotective, antidepressant, antispastic and/or hypnotic agents in mammals.
Patent AU-671023-B2 (AU)
Title: Bearing free spring free throttle position sensor
Inventor: PFAFFENBERGER DAVID S
IPC: G01D11/20
Filed: 1994-06-23
Granted: 1996-08-08
Abstract: The rotor of a rotary position sensor mounts directly upon the rotary shaft to be sensed. The rotor prior to installation is retained in position by a pair of small protrusions extending from the rotor that cooperatively engage a pair of small indentations formed in a pair of supporting arms. During the installation process, the rotor is slipped onto the shaft and the protrusions are released from the engaged position. During operation of the position sensor, the rotor is free from direct contact with either the supporting arms or any other stationary part of the position sensor. Only the contactors engage the stationary components. This design eliminates the need for bearings and return springs prevalent in the prior art. <IMAGE>
Patent AU-583440-B2 (AU)
Title: Device and method for switching communications among taxis
Inventor: NORMAN BALDUIN
IPC: H04Q7/22
Filed: 1986-12-08
Granted: 1989-04-27
Abstract: A user connected by telephone to a central telephone exchange can inform an automatic switching communications device directly of his own telephone number by dialing on his telephone set, which determines the corresponding address and all other possible characteristics from an on-line directory. The available taxis are entered in a stand-by memory. The taxis in first place in the stand-by memory is provided with the assigned address by the switching communications device via radio. The total area serviced by the device for the switching communications exchange of the taxis, can be partitioned into individual sectors, whereby each sector then corresponds to its own stand-by memory. Therefore, a very quick and efficient switching communications exchange is possible without a large expenditure for personnel.
Patent AU-749907-B2 (AU)
Title: Process for the determination of CTp11 and for determining whether a tumor sample has metastatic potential
Inventor: MUIJEN GOOS N P VAN
IPC: C12Q1/6886
Filed: 2000-10-25
Granted: 2002-07-04
Abstract: A process for the determination of CTp11 and for determining whether a tumor sample has metastatic potential is provided.
Patent AU-629443-B2 (AU)
Title: Composition and method for the treatment of osteoporosis in mammals
Inventor: BURK ROBERT R
IPC: A61K38/00
Filed: 1990-12-27
Granted: 1992-10-01
Abstract: A composition for the treatment of osteoporosis in mammals comprising Insulin-like Growth Factor I (IGF-I) and method of treating osteoporosis therewith is disclosed.
Patent AU-763859-B2 (AU)
Title: Cable sheave for cableway systems
Inventor: BERND MEINDL
IPC: B61B7/00
Filed: 2000-10-31
Granted: 2003-07-31
Abstract: The sheave has a hub (2), a sheave surface which extends from the hub and may be configured, if appropriate, in the form of spokes (12a-12d). The sheave further is formed with a cable groove on its circumference, and it has fastening devices with flanges (14a-14d) and bolts (15) which are provided on the sheave surface and along which two or sheave parts can be connected to one another to form the complete cable sheave. The cable sheave body parting lines extend along a secant of the cable sheave body at defined positions.
Patent AU-683898-B2 (AU)
Title: Method and apparatus for producing fibrous material batts
Inventor: NEWTON LINDSAY JOHN
IPC: D06M13/50
Filed: 1994-06-28
Granted: 1997-11-27
Abstract: Fibrous material batts are produced from a mixture of natural and synthetic fibres. A sliver (10) of the fibres is fed through a lapping device (11) onto a moving conveyor to form a continuous mat. The sliver is sprayed with a bonding agent and other optional substances during lapping. The mat is then compressed to a required thickness before curing the bonding agent, and is then cut to form batts of a low density. Resilience and fire retardance properties may be imparted to the fibrous material by including an octaborate salt among the substances sprayed with the bonding agent.
Patent AU-542234-B2 (AU)
Title: Belt conveyor for concrete
Inventor: THENAUD RENE
IPC: B65G15/60
Filed: 1981-08-07
Granted: 1985-02-14
Abstract: 1. Concrete conveyor comprising a metal frame mounted in an articulated manner on a support which can be the chassis of a concrete-mixer lorry, an endless conveyor belt (1), a roller driving the said belt and actuated by a motor, and at least one return roller, supporting means on which the belt slides on it outward trip, that is to say during the time when it is loaded with concrete, and rollers for supporting the belt on its return trip, the said rollers and the said supporting means being supported by the said frame, characterised in that the said supporting means consist of slides (3, 4, 5) elongated in the direction of movement and made of an aluminium alloy resistant to the action of the concrete, each slide being in the form of one or more successive portions, the accumulated length of which is at least equal to 85% of the length of the frame, and the accumulated width of the slides being between 25 and 45% of the width of the belt, in that the slides as a whole from a trough of rounded cross-section, the edges of which form an angle of between 30 and 50 degrees with the horizontal, and in that the face of the belt which is in contact with the said slides has a coefficient of adhesion on the latter which is less than 0.20.
Patent AU-637495-B2 (AU)
Title: Medical valve assembly
IPC: A61M39/00
Filed: 1991-04-09
Granted: 1993-05-27
Abstract: A medical valve assembly is described in which the valve assembly has a female luer lock portion on an inlet end of the device and a male luer lock portion on the outlet portion of the valve. A movable piston seals the inlet portion of the valve from the outlet portion when the piston is in the closed position. When a syringe is attached to the inlet portion of the valve assembly, the piston is displaced in a manner that unseals a fluid channel inlet. This connects the end of the syringe to the fluid channel which is connected, at its outlet end, to a catheter or other device, connected to a patient. Thus, medication can be introduced to, or fluids aspirated from, a patient's bloodstream, without the use of a syringe having a needle. When the syringe is removed from the inlet to the valve assembly, the piston is urged by a biasing means into its original closed position creating a seal between the inlet portion of the valve and the outlet portion of the valve. This feature maintains catheter patency. The top surface of the piston along with the area of the female luer lock connector does not have any fluid reservoir and can be easily cleaned to prevent the possibility of bacterial infection as a result of repeated uses of the valve assembly.
Patent AU-676773-B2 (AU)
Title: Chiral nitriles, their preparation and their use for the manufacture of verapamil and analogues
Inventor: MCCAGUE RAYMOND
IPC: C07C255/43
Filed: 1994-09-26
Granted: 1997-03-20
Abstract: A process for preparing a substantially single enantiomer (R &cir& _ or S &cir& _) of R'-NH-(CH2)3-C(Ar) (CN)-R, the process comprising reacting together R-CH(Ar)-CN and X-(CH2)3-A to give X-(CH2)3-CH(Ar) (CN)-R, reacting that with methylamine to give R'-NH-(CH2)3-C(Ar) (CN)-R, and resolving that into a substantially single enantiomer thereof, wherein Ar is aryl, R and R' are each independently C1-20 alkyl, X is a halo atom and A is a leaving group and the resolution is carried out using a chiral acid. The process is particularly useful for preparing verapamil, and analogues thereof, in single enantiomeric form.
Patent AU-641515-B2 (AU)
Title: Aids for filtration and/or dehydration of mineral and coal suspensions
Inventor: KOSTER RITA
IPC: C09K23/42
Filed: 1991-06-06
Granted: 1993-09-23
Abstract: PCT No. PCT/EP91/01049 Sec. 371 Date Dec. 15, 1992 Sec. 102(e) Date Dec. 15, 1992 PCT Filed Jun. 6, 1991 PCT Pub. No. WO91/19556 PCT Pub. Date Dec. 26, 1991.Addition of alkyl and/or alkenyl polyalkylene glycol ethers as filtration aids in the filtration and/or dehydration of mineral or coal suspensions reduces the dehydration time, and filter cakes with a low residual moisture content are obtained.
Patent AU-778359-B2 (AU)
Title: Sustained-release drug formulations for implantation
Inventor: SANO AKIHIKO
IPC: A61K47/02
Filed: 2000-10-31
Granted: 2004-12-02
Abstract: The present invention relates to a formulation for implantation having a novel constitution, which accomplishes controlled releases of active ingredients. The formulation comprises one of combinations (a), (b) and (c), as well as a carrier comprising a hydrophobic polymer, wherein the particle combination is dispersed into the carrier: (a) particles comprising an active ingredient, particles comprising a carbonate, and particles comprising a substance which is reacted with the carbonate in an aqueous solution to generate carbon dioxide (substance such as an acid); (b) particles comprising an active ingredient and a carbonate, and particles comprising a substance such as an acid; and (c) particles comprising a carbonate, and particles comprising an active ingredient and a substance such as an acid.
Patent AU-603838-B2 (AU)
Title: Preparing polyethylene articles of high tensile strength and modulus and low creep
Inventor: BASTIAANSEN CORNELIS WILHELMUS
IPC: C08L23/04
Filed: 1987-10-27
Granted: 1990-11-29
Abstract: Polyethylene articles having a high tensile strength above 2.0 GPa, a modulus above 70 GPa and a creep below 3 x 10<-><7> sec<-><1> are obtained via thermoreversible gelation of a solution of polyethylene with a Mv above 5 x 10<5> kg/kmole, followed by ultradrawing. As polyethylene a copolymer or a blend is used containing 2-20 lower alkyl side chains per 1000 carbon atoms.