baber/WOPTO huggingface dataset:
Patent MA-21028-A1 (MA)
IPC: C07D513/04
Filed: 1987-07-02
Abstract: A compound of the general formula I:    <IMAGE>  (I)  in which Ar is a pyridyl, quinolinyl, isoquinolinyl, naphthyridinyl, pyrimidyl, quinazolinyl, thiazolyl, benzothiazolyl, imidazolyl, benzimidazolyl, oxazolyl, benzoxazolyl, thienyl, benzothienyl or naphthyl group; optionally substituted with one or more halogen or alkyl, alkyloxy, alkylthio, trifluoromethyl, amino, alkylamino, dialkylamino, hydroxy, cyano, alkylsulphinyl, alkylsulphonyl, sulphamido, alkylsulphamido, dialkylsulphamido, alkylcarbonyl, benzoyl, alkyloxycarbonyl, carboxy, phenoxycarbonyl, alkylcabonyloxy, benzoyloxy, alkylcarbonylamino, benzamido, phenyl, benzyl, phenoxy or phenylthio group, provided that (i) when Ar is a pyridyl group, the pyridyl group must be substituted, (ii) an alkyl moiety contains 1 to 4 straight- or branched chain carbon atoms; (iii) a phenyl moiety may be unsubstituted or substituted with one or more halogen or alkyl, alkyloxy, alkylthio, trifluoromethyl, amino, alkylamino, dialkylamino, hydroxy, cyano, phenyl or benzyl group in separate enantiomeric form or mixtures thereof, or a pharmaceutically acceptable salt thereof is useful in the treatment of all pathological conditions in which PAF-acether may be implicated directly or indirectly.
Patent MA-24456-A1 (MA)
IPC: D06L4/75
Filed: 1998-01-23
Abstract: Disclosed are photochemical super oxide generators useful as photobleaches for laundry detergent compositions and as photobleaches or photodisinfectants for use in hard surface cleaning compositions. The compounds described herein comprise an amino-containing electron transfer moiety bonded to the photosensitizing unit wherein the amino-containing moiety is capable of transferring an electron to the photochemically excited pi electron cloud of the photosensitizer unit thereby enabling superoxide formation.
Patent MA-27111-A1 (MA)
Inventor: ZHANG CHENGZHI
IPC: C07D407/06
Filed: 2004-09-22
Abstract: This invention relates to novel benzofuran and benzothiophene derivatives of the general formula and their use for the treatment of hyper-proliferative disorders.
Patent MA-27475-A1 (MA)
Inventor: ALLEN DAVID GEORGE
IPC: A61P29/00
Filed: 2005-04-15
Abstract: The invention relates to a compound of formula (I) or a salt thereof: wherein: R<SUP>1 </SUP>is C<SUB>1-4</SUB>alkyl, C<SUB>1-3</SUB>fluoroalkyl, -CH<SUB>2</SUB>CH<SUB>2</SUB>OH or -CH<SUB>2</SUB>CH<SUB>2</SUB>CO<SUB>2</SUB>C<SUB>1-2</SUB>alkyl; R<SUP>2 </SUP>is a hydrogen atom (H), methyl or C<SUB>1</SUB>fluoroalkyl; R<SUP>3 </SUP>is optionally substituted C<SUB>3-8</SUB>cycloalkyl or optionally substituted mono-unsaturated-C<SUB>5-7</SUB>cycloalkenyl or an optionally substituted heterocyclic group of sub-formula (aa), (bb) or (cc); in which n<SUP>1 </SUP>and n<SUP>2 </SUP>independently are 1 or 2; and in which Y is O, S, SO<SUB>2</SUB>, or NR<SUP>10</SUP>; or R<SUP>3 </SUP>is a bicyclic group (dd) or (ee): and wherein X is NR<SUP>4</SUP>R<SUP>5 </SUP>or OR<SUP>5a</SUP>. The compounds are phosphodiesterase (PDE) inhibitors, in particular PDE 4 inhibitors. Also provided is the use of a compound of formula (I), or a pharmaceutically acceptable salt thereof, in the manufacture of a medicament for the treatment and/or prophylaxis of an inflammatory and/or allergic disease in a mammal such as a human, for example chronic obstructive pulmonary disease (COPD), asthma, or allergic rhinitis.
Patent MA-37748-A1 (MA)
Title: Composés d'azétidine et de pipéridine utiles comme inhibiteurs de pde10
Inventor: ALLEN JENNIFER R
IPC: C07D403/14
Filed: 2015-01-09
Abstract: L'invention concerne des composés d'azétidine et de pipéridine de formule (i) tels que définis dans le descriptif, des compositions les contenant, et des procédés de préparation de ces composés et leurs intermédiaires. L'invention concerne également des méthodes de traitement des maladies ou troubles cognitifs pouvant être traités par inhibition de pde10, tels que la maladie de huntington, la schizophrénie, les troubles bipolaires, les troubles obsessionnels-compulsifs et analogue.
Patent MA-39181-A1 (MA)
Title: Connecteur pour dispositif jetable à usage unique
Inventor: SOKOLOV RICHARD
IPC: A61M5/168
Filed: 2015-01-09
Abstract: La présente invention concerne un connecteur médical pour la mise en place d'une connexion stérile entre une portion à usages multiples et une portion à usage unique d'un système de distribution fluidique. Le connecteur médical inclut un port d'entrée fluidique configuré pour s'engager de façon amovible avec un port de connexion d'un dispositif jetable à usages multiples ou muds (multi-use disposable set) pour établir une connexion fluidique avec ce dernier et un port de sortie de déchets configuré pour s'engager de façon amovible avec un port d'entrée de déchets du dispositif muds et établir une connexion fluidique avec ce dernier. Une ligne fluidique de patient est connectée au niveau d'une première extrémité au port d'entrée fluidique et au niveau d'une deuxième extrémité au port de sortie de déchets. Le débit fluidique à travers la ligne fluidique de patient est unidirectionnel entre la première extrémité et la deuxième extrémité. La ligne fluidique de patient est configurée pour se déconnecter du port de sortie de déchets pour la distribution de fluide à un patient. La présente invention concerne également un système de distribution multi-fluidique comportant le connecteur médical et le dispositif muds.
Patent MA-40160-A1 (MA)
Title: Procédé de construction d'un renforcement fibreux en forme de bande pour un mur de soutènement de sol renforcé
Inventor: LEE JEUNG SU
IPC: E02D29/02
Filed: 2015-03-12
Abstract: La présente invention concerne une structure de mur de soutènement de sol renforcé qui permet la liaison rapide et facile d'un matériau de renforcement de fibre de type bande, qui peut fournir divers procédés de liaison associés, et qui empêche une contrainte de se concentrer dans une partie de liaison avec un élément de parement pendant l'enfoncement d'un corps de sol renforcé, la structure de mur de soutènement de sol renforcé comprenant : un élément de parement (10) ayant un trou d'insertion de matériau de renforcement (20) incorporé dans celui-ci ; un matériau de renforcement de fibre de type bande (30) qui est ajusté dans le trou d'insertion de matériau de renforcement (20) de l'élément de parement (10) et qui est disposé sur un corps de sol renforcé (g), le trou d'insertion de matériau de renforcement (20) comportant : deux entrées (21, 22), qui sont chacune ouvertes vers le côté arrière (12) de l'élément de parement (10) et qui sont espacées d'un côté à l'autre ; un passage traversant (23) dans lequel un rayon de courbure prédéterminé est formé des deux entrées (21, 22) jusqu'à l'intérieur du côté arrière (12) de l'élément de parement (10), les deux entrées (21, 22) ayant une surface interne (21a, 22a) ouverte perpendiculairement au côté arrière (12) de l'élément de parement (10) et ayant une surface externe (21b, 22b) ouverte, le côté avant de celle-ci étant large et son côté arrière étant étroit par rapport au côté arrière (12) de l'élément de parement (10), un matériau de renforcement de fibre de type bande flexible (30) étant inséré dans une entrée (21 ou 22) et tiré par l'autre entrée (22 ou 21), puis étant ensuite relié, disposé sur le corps de sol renforcé et enterré.
Patent UY-23845-A1 (UY)
Title: Aparato para verificacion e identificacion de cheques y/o tarjetas magnéticas
IPC: G06V30/224
Filed: 1994-10-19
Abstract: La presente invención trata de un aparato especialmente desarrollado para efectuar la verificación e identificación de cheques bancarios o tarjetas magnéticas. El aparato que ejecuta estas funciones a partir de la lectura del código de barras, comprende basicamente una Unidad Central de Procesamiento UCP (10), la cual incorpora oscilador interno, memoria, líneas de entrada y salida, comunicación en serie y temporizadores, y es responsable por la operacionalidad del aparato, el cual consiste en un lector de tarjeta magnética (4) y un lector de código de barras (2), además de un teclado (1), que son las unidades de entrada en el aparato y están interligadas a la UCP (10), la cual recibe las señales y los decodifican y los procesan a través de correlación de algorítmos de criptografía de forma totalmente independiente de cualquier línea de comunicación, siendo también a la dicha UCP (10) interligados diodos emisores de luz (8), un display (7) y una bocina (6) de orientación de operación, además de la memoria (9) mantenedora de las configuraciones posibles del aparato, de comunicación en serie (3) con otros equipamientos y un cargador de baterías (11), siendo que dicho aparato es alimentado por una batería/fuente de alimentación (5). La figura 1 es un diagrama de los bloques funcionales del aparato.
Patent UY-24143-A1 (UY)
Title: Elemento calentador de resistencia polimerico
Inventor: CHARLES M ECKMAN
IPC: H05B3/04
Filed: 1995-12-29
Abstract: Mediante esta invención se proporciona elementos calentadores poliméricos y calentadores de agua que contienen estos elementos. Los elementos calentadores incluyen un material de resistencia eléctricamente conductivo capaz de calentar fluido cuando es energizado. La serpentina está aislada y protegida por una capa de polímero íntegramente dispuesta por encima del material de resistencia. Los elementos son livianos, de bajo costo para producir y usar, y minimizan la corrosión galvánica y los depósitos de cal sin sacrificar la capacidad de calentamiento.
Patent UY-28989-A1 (UY)
Title: Dispositivo para suministrar senales electromagneticas a cuello de utero
Inventor: PICCALUGA DR ALVARO VERGARA
Filed: 2005-06-27
Abstract: El dispositivo se muestra compuesto de Parte a- que puede detectar frecuencia de senal electromagnetica celular por:1- 1-Fenómeno de coincidencia de fase (versión biológica de resonancia). 2-Resonancia a campo electromagnético. 3-Detección directa por pantallas conductoras y amplificación posterior. NOTS- El fénomono 1 es el más simple de aplicar. Parte b- Consta de: a- Eje de flexion de cobre, achatado transversalmente b-Cuerpo de teflón c-Cable de cobre revestido en teflón d-contacto de cobre e-salida hembra a generador de ondas. Es autoclavable y/o descartable. 3-Detección directa 3-Detección directa por pantallas conductoras y amplificación posterior. NOTA- El fenómeno 1 es el más simple de aplicar. Parte b- Consta de:
Patent UY-29595-A1 (UY)
Title: Derivados de benzooxazol-2-ona como inhibidores de lipasas y de fosfolipasas
Inventor: HEUER DR HUBERT
IPC: C07D263/58
Filed: 2006-06-09
Abstract: La presente invención se refiere a derivados de benzooxazol-2-ona de fórmula general I con los significados indicados en la descripción, a sus sales farmacéuticamente utilizables y a su uso como sustancias medicinales.
Patent UY-30815-A1 (UY)
Title: Moduladores no esteroidales del receptor de progesterona
Inventor: KIRKLAND THOMAS ADREW
IPC: A61K31/167
Filed: 2007-12-19
Abstract: Moduladores no esteroidales del receptor de progesterona de la formula general I el uso de los moduladores del receptor de progesterona en la preparacion de medicamentos, y composiciones farmacéuticas que contienen estos compuestos. Los compuestos de acuerdo con la invencion son apropiados para la terapia y la profilaxis de enfermedades ginecologicas, tales como endometriosis, el leimioma uterino, la hemorragia disfuncional y la dismenorrea, y también para la terapia y la profilaxis tumores dependientes de hormonas, y para usarlos en el control de la fertilidad femenina y la terapia de reemplazo de hormonas femeninas.
Patent AT-516824-A1 (AT)
Title: Verfahren und Vorrichtung zur Prüfung von OVI-Merkmalen
IPC: G07D7/20
Filed: 2015-01-23
Abstract: Die Erfindung betrifft ein Verfahren zur Prüfung eines bedruckten Objekts (1) auf einen Aufdruck mit einer vorgegebenen OVI-Tinte, die bei Weißlicht-Bestrahlung einer mit ihr bedruckten Oberfläche unter einem vorgegebenen ersten Winkel (a) Licht mit einem ersten Spektrum (S1) abgibt und bei Weißlicht-Bestrahlung einer mit ihr bedruckten Oberfläche unter einem vorgegebenen vom ersten Winkel (a) abweichenden zweiten Winkel (ß) Licht mit einem zweiten Spektrum (S2) abgibt, Es ist vorgesehen, dass für eine Anzahl von Oberflächenpunkten (2) innerhalb eines Oberflächenbereichs (5) des Objekts jeweils die folgenden Schritte durchgeführt werden, nämlich dass -der Sahstrahl (11) eines Helligkeitssensors (10) auf den jeweiligen Oberflächenpunkt (2) des Objekts (1) gerichtet wird, wobei mit dem Helligkeitssensor (1 0) Licht in zumindest zwei voneinander unterschiedlichen Wellenlängenbereichen (1. .. 1, A.2) detektiert wird, - der von einer ersten Lichtquelle (21) abgegebene erste Lichtstrahl (22) auf den Oberflächenpunkt (2) des Objekts (1) gerichtet wird, wobei der Sahstrahl (11) und der erste Lichtstrahl (22) in einem Winkel der Größe des ersten Winkels (a) zueinander angeordnet werden, - der von einer zweiten Lichtquelle (31) abgegebene zweite Lichtstrahl (32) auf den Oberflächenpunkt (2) des Objekts (1) gerichtet wird, wobei der Sahstrahl (11) und der zweite Lichtstrahl (32) in einem Winkel der Größe des zweiten Winkels (ß) zueinander angeordnet werden, und - jeweils mit dem Helligkeitssensor (1 0) sowohl Licht im ersten Wellenlängenbereich (A.1) als auch im zweiten Wellenlängenbereich (A.2) jeweils ein Intensitätswert ermittelt und dem jeweiligen Oberflächenpunkt (2) ein Intensitätsvektor (V) umfassend die beiden Intensitätswerte (l1, l2) zugewiesen wird. Anschließend wird überprüft, ob innerhalb der für den jeweiligen Oberflächenbereich (5) Helligkeitswerte ermittelten und den einzelnen Oberflächenpunkten (2) zugewiesenen Intensitätswerte (l1, b) bei den beiden Wellenlängen (A-1, A-2) zwei voneinander abweichende Häufungen (H1, H2) bestehen.
Patent ES-193444-A1 (ES)
Title: Un sistema para producir humos a fines de propaganda comercial en los aviones o avionetas
Filed: 1950-06-15
Abstract: Un sistema para producir humos a fines de propaganda comercial en los aviones o avionetas, esencialmente caracterizado por la circunstancia de disponer en lugar apropiado del avión un tanque o depósito que ha de contener un líquido o materia de fácil combustión y que por sus cualidades químicas sea gran productora de humos a cuya finalidad podrá añadirse mediante el catalizador adecuado otra sustancia tanto para pigmentar los humos en la tonalidad que se desee si estos han de ser de color determinado como para acrecentar su combustibilidad.
Patent ES-279708-A1 (ES)
Title: Improvements in or relating to self-oscillating mixer circuits
IPC: H03D7/10
Filed: 1962-08-01
Abstract: A self-oscillating frequency changer utilizes a mixer valve having a planar cathode 2 surrounded by a control grid 1 and a screen grid 3 and having two independent anodes 4, 5 each co-operating with a respective side of the cathode, one anode being included in the oscillator circuit and the other being connected to an IF circuit. The valve may have in addition a screen 5 and the grids may be of " frame grid " form.
Patent ES-317190-A1 (ES)
Title: Improvements in or relating to machines for peeling tomatoes
IPC: A23N7/00
Filed: 1965-09-07
Abstract: A tomato peeling machine includes a plurality of peeling devices 4 each comprising a hollow, open ended body 27 carried by a moving support 28, a perforated wall 29 mounted within the body 27 with an annular space 30 therebetween, an elastic jacket 32 with a roughened inner surface secured by enlarged end flanges 33 within the perforated wall 29, means 41, 37 for supplying air under pressure to within and outside the jacket 32, and a cutting device over which the support 28 is moved to cut the skin of a tomato 8 supported in a deformed jacket 321. In operation, tomatoes are fed singly from a hopper 26 into the jacket 32 and compressed air from a toroidal channel 41 urges the tomato 8 to the middle of the jacket. Compressed air is then passed through an inlet 37 to act on the outer surface of the jacket 32 and deform it, as at 321, to a tomato skin gripping position. The lower, stem end of the tomato has its skin cut so that the skinned tomato is ejected from the jacket 32 and the skin remains adhered to the jacket 32. The hollow body may be of cylindrical form (Figs. 9, 10) and is selectively fitted with one of a number of alternative perforated walls (44) and jackets (46) according to the size of the tomatoes being skinned. The moving support 28 may be in the form of a rotary disc (3) or an endless conveyer (12) each carrying a plurality of rows of peeling devices 4, the tomatoes being fed to the support by a conveyer system which is advanced synchronously with the operation of the peeling devices. An electronic device senses the difference in ripeness between the zone of the stem of the tomato and the tomato itself and energizes an elecromagnet which rotates the peeling device through 180 degrees if the tomato is wrongly oriented therein.
Patent ES-322183-A1 (ES)
Title: Waterproofing and decorating building materials
IPC: C04B41/63
Filed: 1966-01-24
Abstract: Compositions suitable for water-proofing or decorating building materials which may contain free lime comprise (a) 100 parts by weight of a film-forming copolymer of an acrylic or methacrylic ester with another such ester or a copolymer of such an ester with styrene (b) 0.5 - 12.5 parts by weight of a dispersion agent selected from sodium methylene-bisnaphthalene sulphonate, condensates of 8 - 14 mols ethylene oxide with 1 mol -naphthol, condensates of 2 - 8 mols ethylene oxide with 1 mol stearic or palmitic acid, condensates of 4 - 10 mols ethylene oxide with 1 mol cetyl, lauryl or oleyl alcohol, and fatty acid amides or alkylamines having 12 - 18 carbon atoms (c) 0.5 - 12.5 parts by weight of a water-proofing agent selected from fatty acid amides or alkylamines having 12 - 18 carbon atoms, fatty acid - alkylene oxide condensates having 2 - 8 alkylene oxide units, *-acylamino-butyric acids having 12 - 18 carbon atoms in the acyl radical, butyl, ammonium or amine stearates or oleates, dialkyl ketones having 7 - 18 carbon atoms in each alkyl group, or a wax or 0.5 - 40 parts by weight of a microcrystalline wax (d) 150 - 250 parts by weight of an aqueous or organic solvent (e) 0 - 200 parts by weight of a pigment and/or inorganic filler (f) 0 - 1.5 parts by weight of an anti-foaming agent and (g) 0 - 10 parts by weight of a coalescing agent. The consistency of the composition may be adjusted, if desired, by the addition of a further quantity of solvent. The (meth) acrylic ester components) of the copolymers may be derived from an aliphatic, araliphatic or cycloaliphatic alcohol. Where component (c) of the composition is a wax, this may be polyethylene wax, ceresin or a paraffin wax. Suitable organic solvents (d) include aliphatic or aromatic hydrocarbons, and aliphatic esters, alcohols and ketones. Components (e) specified are red or black iron oxide, titanium dioxide, burnt sienna, ochre, green chromium, oxide, gypsum, magnesium silicate, magnesium carbonate, calcium carbonate, pyrophyllite, mica, pumice, silica, diatomite, barium sulphate and alumina. The anti-foam (f) may be tributyl phosphate or 2-ethyl hexanol, and the coalescing agent may be ethylene glycol monoethyl ether acetate, diethylene glycol monobutyl ether acetate or hexylene glycol. The compositions are particularly suitable for application to asbestoscement agglomerates in the form of plane or corrugated boards, wall boards, tiles &c. The compositions can be applied by means of a spray gun, scraper or brush, or by the curtain painting method. In a preferred procedure, the substrate material is preheated to 40 - 60 C. and then coated, the coated material left to stand for 0.5 - 1 minute, and then dried in an oven at 40 - 60 C for 2 - 10 minutes. The weight of dry film coating may be from 30 - 85 g. per sq. m.
Patent ES-335270-A1 (ES)
Title: New Benzimidazole Derivatives
IPC: D06M16/00
Filed: 1967-01-04
Abstract: A pesticidal composition contains as active ingredient a 2-trifluoromethyl benzimidazole of the formula:- wherein R 1 is a halogen atom or a halogenalkyl radical, R 2 is a halogen atom or a C 1 , to C 4 alkyl or C 2 to C 4 alkenyl radical optionally bound to the benzene nucleus by way of an oxygen or sulphur atom or a sulphinyl or sulphonyl radical, R 3 is a halogen atom, X is an oxygen or sulphur atom or a sulphinyl or sulphonyl group, m is from 0 to 3, n is from 0 to 2 and p is from I to 3, the halogeno radicals being those having atomic weights below 100, or a salt thereof. The composition may also contain a solid or liquid carrier or distributing agent and may be in the form of a dust, sprinkling agent, granulates, aqueous dispersion, wettable powder, paste, emulsion concentrate, solution or aerosol. The composition may also contain other active substances, e.g. halogenated diphenyl ureas, halogenated phenoxydiphenyl ureas, 2- chloro-methyl-sulphonylamino polychlorodiphenyl ethers. halogenated N - alkylsulphonyl anthranilic acid anilides, phosphoric, phosphonic, thiophosphoric or dithiophosphoric acid esters and amides, carbamic acid esters, halogenated hydrocarbons, analogues of D.D.T., and pyrethrins, and synergists or auxilliaries, e.g. succinic acid dibutyl ester, piperonyl butoxide, olive oil or peanut oil. The compositions may be used for protecting materials, particularly keratin materials, e.g. wool, other animal hair, fells and furs, against pesticidal attack. The textile materials may be impregnated using textile finishing processes, e.g. hot or cold, aqueous dye, bleaching chroming, pad dyeing or after treatment baths.
Patent ES-338250-A1 (ES)
Title: Lubricant
IPC: C10M169/00
Filed: 1967-03-20
Abstract: A sol of a nitrate, acetate, laurate, formate or salicylate of calcium, magnesium or barium, particularly of calcium acetate, in a predominantly naphthenic heavy hydrocarbon fraction, together with calcium sulphonate as an emulsifying agent, is included in lubricants. The sol can be used as an anti-rust protection, for the lubrication of slow, very hot bearings and pivots and as an addition to lubricants e.g. a diesel oil containing anti-oxidation additives, colloidal graphite and molybdenum disulphide.
Patent ES-338348-A1 (ES)
Title: Method and device for producing high-power light pulses of short duration
IPC: H01S3/11
Filed: 1967-03-22
Abstract: Coherent light generated in a laser resonant cavity is concentrated into a wave packet having a length which is less than the length of the cavity and is then extracted from the cavity. The active medium 9 is initially pumped while cavity reflector 2 is non-parallel to reflector 13. With the reflectors parallel, electro-optical modulator M, consisting of a Pockels cell 12 and a Glan prism 10, is energized with A.C. so that its instant of maximum transmission recurs with a period equal to the time taken for light to travel from the modulator to reflector 2 and back to the modulator. As a result photons emitted from the active medium tend to concentrate in a wave packet which is transmitted by the modulator at the instant of maximum transmission. When this wave packet has formed a D.C. voltage is applied to electrooptical switch C, also consisting of a Pockels cell and Glan prism, to deflect the wave packet out of the cavity. In a second embodiment the modulator and switch are combined in a single unit and in a third embodiment this unit also performs the same function as the rotating prism 2, the cavity being initially give a low Q by applying a D.C. voltage to the electro-optical cell. The prism is in this embodiment replaced by a plane mirror.