baber/WOPTO huggingface dataset:
Patent BR-112023017280-A2 (BR)
Title: Estimação de canal para múltiplas tecnologias de radioacesso em um cenário de alta velocidade
Inventor: CHINMAY SHANKAR VAZE
IPC: H04W36/08
Filed: 2021-03-05
Abstract: estimação de canal para múltiplas tecnologias de radioacesso em um cenário de alta velocidade. trata-se de métodos, sistemas e dispositivos para comunicações sem fio. as técnicas descritas fornecem um equipamento de usuário (ue) que usa informações identificadas por meio de tecnologia de radioacesso (rat) (por exemplo, evolução a longo prazo (lte)) para suportar comunicações em uma outra rat (por exemplo, novo rádio (nr)). por exemplo, o ue pode receber, de uma primeira estação-base que opera de acordo com uma primeira tecnologia de radioacesso, uma indicação de uma alta velocidade associada a uma primeira conexão sem fio do ue com a primeira estação-base. o ue pode realizar um procedimento de estimação de canal para a primeira conexão sem fio para gerar um valor de doppler com base no recebimento da indicação. o ue pode aplicar o valor de doppler gerado a um loop de rastreamento de frequência ou um loop de rastreamento de tempo para comunicações com uma segunda estação-base por meio de uma segunda conexão sem fio, em que a segunda estação-base está operando de acordo com uma segunda rat.
Patent BR-112023020826-A2 (BR)
Title: Cocristais de upadacitinibe
Inventor: MATTEI ALESSANDRA
IPC: A61K31/395
Filed: 2022-04-07
Abstract: cocristais de upadacitinibe. a revelação refere-se a cocristais de formas de estado sólido de (3s,4r)-3-etil-4-(3h-imidazo[1,2-a]pirrolo[2,3-e]-pirazin-8-il)-n -(2,2,2-trifluoroetil)pirrolidina-1-carboxamida (composto 1). especificamente, a presente revelação refere-se a cocristais do composto 1 e a um coformador adequado, como um ácido benzoico substituído.
Patent CU-21554-A3 (CU)
Title: Obtainment procedure of imidazobenzodiacepine
Inventor: HUNKELER WALTER
IPC: C07D487/14
Filed: 1983-07-21
Abstract: There are described novel pharmaceutically active substances which have a pronounced affinity to the central benzodiazepine receptors and which have only a low toxicity. These active substances, namely imidazobenzodiazepines of the formula    <IMAGE>  I  wherein A is lower alkylene, n is zero or 1, R1 is lower alkynyl, lower alkenyl, aryl, (C3-8)-cycloalkyl optionally substituted by lower alkyl or (C5-8)-cycloalkenyl optionally substituted by lower alkyl, or a 5- or 6-membered saturated or unsaturated heterocycle which contains an oxygen or sulphur atom as a ring member and which is optionally substituted by lower alkyl, R4 and R5 each are hydrogen, halogen, trifluoromethyl, cyano, nitro, amino or lower alkyl and either R2 is hydrogen and R3 is lower alkyl or R2 and R3 together are dimethylene, trimethylene or propenylene, the compounds of formula I in which R2 and R3 together are dimethylene, trimethylene or propenylene having the (S) or (R,S) configuration with reference to the carbon atom denoted by  gamma , and their pharmaceutically acceptable acid addition salts, can be used as medicaments in the form of pharmaceutical preparations, especially in the control of convulsions and anxiety states and/or in the partial or complete antagonization of some or all activities which 1,4-benzodiazepines having tranquillizing activity or other substances display via the central benzodiazepine receptors.
Patent CZ-26199-A3 (CZ)
Title: 1,4-diaryl-3-fluoro-2-butene compounds for protecting animals and humans from attack and infection by arthropodious parasites
Inventor: DOSCHER MARY EHLERS
IPC: A61P33/00
Filed: 1999-01-26
Abstract: The present invention relates to methods and compositions for treating animals and humans, and controlling, and preventing and protecting animals and humans from infestation and infection by arthropod parasites by administering or applying to the animals, humans or their environment a 1,4-diaryl-3-fluoro-2-butene compound having the structural formula <CHEM>
Patent CZ-91093-A3 (CZ)
Title: Collapsible container
Inventor: PASEK LUBOS ING
IPC: B65D88/52
Filed: 1993-05-17
Abstract: A collapsible container, consisting of a base frame (1) with upwards projecting corner stands (11), which has, between the stands (11),  collapsible attached walls (2,3). Each wall (2,3) has at least one stabilising device, formed by the projection (12,13) of the base frame (1) and recess, arranged opposite it from below on the wall (2,3). Furthermore, each wall (2,3) has a two-piece collapsible guide, whose one side is formed by a groove (4a,4b) and second by a pin (5). One part of the two-piece collapsible guide is arranged on the sides of the walls (2,3), and the second on the corresponding opposite sides of the stands (11).<IMAGE>
Patent SK-24694-A3 (SK)
Title: Pharmaceutical composition
Inventor: REED MICHAEL JOHN
IPC: A61K31/56
Filed: 1992-08-28
Abstract: The use of purified composition for production of medicament to inhibit the activity of steroid sulphatase, containing circle system comprising a circle, to which there is bonded a sulphamate group of formula (I), wherein each of R1 and R2 are independently selected from the group comprising H, alkyl, alkenyl, cycloalkyl and aryl or together represent alkylene containing either one or more heteroatoms, or groups in alkylene chain and wherein the composition is an inhibitor of the enzyme with the activity of steroid sulphatase (E.C.3.1.6.2) and wherein, if the sulphamate group was replaced in the composition by sulphate group to make a sulphate composition and incubated with the enzyme of steroid sulphatase (E.C.3.1.6.2) with pH 7.4 and temperature 37  C, the value Km less than 50 umol would be obtained.
Patent SK-50299-A3 (SK)
Title: Thienopyrimidine with phosphodiesterase v inhibiting effect
Inventor: JONAS ROCHUS
IPC: C07D495/04
Filed: 1997-10-08
Abstract: The invention relates to thienopyrimidine of the formula (I) as well as to their physiologically acceptable salts, wherein R<1>, R<2>, R<3>, R<4>, X and n have the meaning cited in Claim 1. Said compounds exhibit a phosphodiesterase V inhibition and can be used in the treatment of cardiovascular diseases and for the treatment and/or therapy potency disorders.
Patent SK-50499-A3 (SK)
Title: Bis(acridinecarboxamide) and bis(phenazinecarboxamide) as antitumour agents
Inventor: DENNY WILLIAM ALEXANDER
IPC: C07D219/04
Filed: 1997-10-17
Abstract: PCT No. PCT/GB97/02886 Sec. 371 Date Jun. 18, 1999 Sec. 102(e) Date Jun. 18, 1999 PCT Filed Oct. 17, 1997 PCT Pub. No. WO98/17650 PCT Pub. Date Apr. 30, 1998A compound which is a bis(acridinecarboxamide) or bis(phenazinecarboxamide) derivative of formula (I): wherein each X, which may be the same or different in a given molecule, is -CH= or -N= each of R1 to R4 which may be the same or different, H, C1-C4 alkyl, OH, SH, NH2, C1-C4 alkoxy, aryloxy, NHR, N(R)2, SR, SO2R wherein R is C1-C4 alkyl, CF3, NO2 or halogen, or R1 and R2 together form a methylenedioxy group; each of R5 and R6, which may be the same or different, is H or C1-C4 alkyl; Z is (CH2)n, (CH2)nO(CH2)n, (CH2)nN(R7)(CH2)n, (CH2)nN(R7)(CH2)mN(R7)(CH2)n or (CH2)nN(CH2CH2)2N(CH2)n wherein R7 is H or C1-C4 alkyl and n and m, which may be the same or different, are each an integer of 1 to 4; or a pharmaceutically acceptable acid addition salt or N-oxide thereof; has activity as an antitumor and antibacterial agent.
Patent CH-629934G-A3 (CH)
IPC: G10H1/06
Filed: 1978-07-17
Abstract: An electronic tone generator capable of providing improved musical and tone quality by providing a primary melody and a secondary melody such as an accompaniment or the like is provided. The electronic tone generator of the instant invention is characterized by the use of a primary electronic scale generator circuit for producing a primary scale signal representative of a primary melody scale and a secondary electronic scale generator circuit for producing a secondary scale signal that is representative of a secondary melody and that is distinct from the primary scale signal. The primary scale signal and second scale signal are respectively shaped and summed and thereafter applied to an electro-acoustic transducer in order to produce music having a primary melody and secondary melody of considerable musical quality.
Patent CZ-261990-A3 (CZ)
Inventor: HEMZAL BOLESLAV
IPC: A47C1/022
Filed: 1990-05-29
Abstract: Na nosném rámu (3), který nese sedák (4), je přestavitelné
uložena objímka (7), na jejichž protilehlých bočních stěnách
jsou prostřednictvím čepů (8) výkyvné uloženy protilehlé
vzpěry (9). Opačné konce těchto vzpěr (9) jsou
prostřednictvím dalších čepů (10) vykyvně uloženy v závěsech
(11), upevněných na spodní straně sedáku (4). Přitom
objímka (7) je opatřena polohovacím aretačním zařízením
(12).
Patent CZ-295292-A3 (CZ)
Title: Container for storing record carriers
Inventor: NEHL WOLFGANG
IPC: B65D85/575
Filed: 1992-09-25
Abstract: 2.1 In the case of known storage devices, the recording medium is transported by a slide, which can be displaced by means of spring force, into a removal position on the front side of the storage device, the slide being extended with the recording medium placed on it out of the housing to such an extent that the recording medium can be grasped. After removal of the recording medium, the slide is pushed back again to avoid projecting parts. 2.2 In order to be able to dispense with pushing back the slide after removal of the recording carrier, the storage device is equipped with a locking mechanism which, in the storage position, engages in the housing of the recording medium. Furthermore, even in the removal position, the entire slide is in a withdrawn location in the storage device. <IMAGE>
Patent CZ-374692-A3 (CZ)
Title: Proteolytic enzymes inhibitors based on saccharin derivatives
Inventor: HLASTA DENIS JOHN
IPC: A61K31/428
Filed: 1992-12-18
Abstract: Compounds having the structural formula <CHEM> which inhibit the enzymatic activity of proteolytic enzymes, and processes for preparation thereof, method of use thereof in treatment of degenerative diseases and pharmaceutical compositions thereof are disclosed.
Patent CZ-548884-A3 (CZ)
Title: Process for preparing human proinsulin
Inventor: BELL GRAEME
IPC: C12N1/00
Filed: 1984-07-16
Abstract: A DNA having a base sequence coding for human proinsulin and a DNA having a base sequence coding for human pre-proinsulin have been cloned, and novel recombinant DNA transfer vectors containing said cloned DNAs have been constructed. Novel microorganisms transformed by said recombinant transfer vectors have been obtained. Certain of said transformed microorganisms have demonstrated capability to express the cloned DNA's, synthesizing a protein comprising human proinsulin and a protein comprising human pre-proinsulin.
Patent CZ-190096-A3 (CZ)
Title: Wall element for high-rise buildings and process for producing thereof
Inventor: SEBALD RALF
IPC: E04G11/10
Filed: 1996-06-27
Abstract: The reinforcement (7,8) which is embedded before the casting material set protrudes over the lower end face and upper end face of the wall element to form a reinforced connection. The load-absorbing edge strips of the upper end face are flat. Length-adjustable levelling members (15) such as threaded rods and screw sleeves for the wall element are embedded spaced out from each other in the lower end face. At least the upper end face has additionally two spaced anchorage members for fixing lifting tools. Empty tubes (11) for electric cables can be embedded in the wall element to protrude over the relevant end faces of the wall element.
Patent CZ-202134-A3 (CZ)
Inventor: SOUKUP ONDŘEJ
IPC: C07D219/06
Filed: 2021-01-26
Abstract: Předkládané řešení poskytuje 7‐fenoxy‐1,2,3,4‐tetrahydroakridin‐9‐amin pro léčbu některých demencí na základě duální aktivity pro inhibici cholinesteras a jako antagonisty NMDAR
Patent CZ-205198-A3 (CZ)
Inventor: AUSTIN MARK
IPC: B28B1/32
Filed: 1996-12-27
Abstract: Způsob vytváření vzorů v litých materiálech vícebarevných provedení, zahrnující následující kroky: příprava formy k přijímání licích směsí, příprava alespoň dvou licích směsí různých barev při viskozitě, která usnadňuje jejich rovnoměrné lití, zajištění předpisu stanovícího horizontální a vertikální uspořádání pro naložení těchto licích směsí do zásobníku, zajištění zásobníku, naložení licích směsí do zásobníku podle tohoto předpisu, přenášení těchto naložených směsí ze zásobníku do formy, zpevnění směsí ve formě do fyzikálně stejnoměrné hmoty a ponechání této hmoty ztvrdnout, vytvoření litého výrobku, majícího v sobě barevný vzor, určený předpisem, podle něhož jsou licí směsi naloženy do zásobníku. Vyjímatelná matrice (1) v zadržovacím zásobníku (2) zajišťuje možnost reprodukovat vzory.
Patent CZ-208295-A3 (CZ)
Title: In line electron gun
Inventor: PONTAILLIER YVES
IPC: H01J29/48
Filed: 1995-08-15
Abstract: An improved inline electron gun (10), for use in a color picture tube, includes a plurality of electrodes (16, 18, 20, 22, 24, 26) spaced from three cathodes (14) in the direction of a longitudinal axis (Z) of the gun. The electrodes form at least a beam forming region and a main focus lens in the paths of three electron beams, a center beam and two side beams. Each of the electrodes includes three inline apertures (56, 66) therein for passage of the three electron beams. The beam forming region includes the cathodes (14) and three consecutive electrodes, a G1 electrode (16), a G2 electrode (18) and a G3 electrode (20). The improvement comprises the G2 electrode having two linear projections (58) on either side of the inline apertures (56) therein. The projections parallel the inline direction of the apertures protrude in a direction parallel to the longitudinal axis, past the apertured portion (54) of the G3 electrode in overlapping relationship therewith. On the side (52) of the G3 electrode facing the G2 electrode, the G3 electrode has two linear channels (64) therein on either side of the inline apertures (66) therein. The channels are immediately adjacent the projections on the G2 electrode and in a spaced nested relationship therewith. <MATH>
Patent CZ-245895-A3 (CZ)
Title: Coupling for wooden parts
Inventor: MAYER ROBERT
IPC: F16B12/44
Filed: 1995-09-21
Abstract: The invented connector for wooden components serving for detachable joining of wooden components (BT1, BT2) butted against one another has a connecting element (2), and a tensioning element (1) which is inserted into one of two wooden components (BT1, BT2), which are to be joined. One end of the connecting element (2) is in its functional state engaged with the tensioning element (1). The other end of the connecting element (2) can be inserted into a second tensioning element (1) that is provided on the second component (BT2), or it can be inserted directly in a hole of this second component. The connecting element (2) and the tensioning element (2), respectively tensioning elements (2), are parts that are separated from each other and at assembly place communicating with each other for mounting in the components (BT1 and BT2). The tensioning element (2) is made as a disk with an eccentric opening (1.1) performed therein for mounting and clamping said connecting element (2) and in its face it has a slit (1.2) that is symmetrical about a diameter of the disk, and which has a longitudinal axis which is roughly normal to the tensioning element (1) diameter. The clamping slit (1.2) central axis lies in the center of the tensioning element (2) and in the center of the eccentric opening (1.1). The connecting element (2) has a central part (2.1) at the ends of which there is provided an anchoring spigot (2.2, 2.3) located in both the component (BT1, BT2) and the tensioning element (1).
Patent CZ-248693-A3 (CZ)
Title: Porcelain, porcelain mass, as well as process for producing porcelain
Inventor: KREINER ROSWITHA
IPC: C04B33/32
Filed: 1993-11-19
Abstract: The invention relates to a porcelain with a transparency and strength properties of a hard porcelain, characterized by a phosphate-containing glass phase as well as the predominance of unreacted quartz grains in the matrix. The invention relates to a porcelain batch composition as well as to a method for the manufacture of the porcelain.
Patent CZ-9902668-A3 (CZ)
Inventor: SLAMA PAVEL ING
IPC: B23Q1/01
Filed: 1999-07-28
Abstract: Střední vodící dráha je tvořena dvojitou rybinovou lištou (8),
uspořádanou na loži (1) obráběcího stroje rovnoběžně s
pohybovým šroubem (9), na které jsou prostřednictvím rybiny
(7) uloženy křížové saně (2). Krajní vodící dráhy tvoří vodící
lišty (4) na loži (1) obráběcího stroje, uložené s přesahem a
nesoucí valivá tělesa (5) uspořádaná v protilehle
orientovaných dvojicích. Mezi takto orientovanými dvojicemi
valivých těles (5)je na křížových saních (2) uchycena opěrná
deska (6), opatřená na straně přivrácené vodící liště (4)
kluznou hmotou (10).
Patent CZ-304996-A3 (CZ)
Title: Reactor plates with divided flow for vertical stage polycondensation reactors
Inventor: YOUNT THOMAS LLOYD
IPC: B01D3/24
Filed: 1995-04-21
Abstract: This invention relates to a vertically disposed polymerization reactor having a series of essentially circular tray assemblies; each tray assembly having a central open vapor chimney and two split-flow paths each split-flow path containing one reverse flow path wherein the liquid polymer flow is reversed by means of a substantially semi-circular turnaround region; each tray having a liquid polymer tray inlet and a liquid polymer tray outlet for conducting a flow of the liquid polymer by means of a hydraulic gradient; each tray assembly being open at the top for escape of vapor from the liquid polymer flow to the central open vapor chimney; and each tray arranged in vertical disposition one above the other.
Patent CZ-347798-A3 (CZ)
Title: Use of interleukin-10 for preparing population of suppressor cells
Inventor: RONCAROLO MARIA-GRAZIA
IPC: A61K39/00
Filed: 1997-05-02
Abstract: Interleukin-10 for producing a population of cells which are capable of inhibiting or suppressing reactions to alloantigens, for example in graft-versus-host disease or tissue rejection, is described. Interleukin-10 for reducing responses in mixed lymphocyte response (MLR) is also described. Exogenous or induced endogenous IL-10 may be used for the inhibition or suppression of the reactions to alloantigens.
Patent CZ-366299-A3 (CZ)
Inventor: WAITE DAVID CHARLES
IPC: A61K31/404
Filed: 1998-06-16
Abstract: Podstatou řešeníje způsob výroby sloučeniny vzorce I, který
zahrnuje reakci sloučeniny vzorce II se sloučeninou vzorce ΠΙ
v přítomnosti silné báze a palladium(0)kalalyzátoru, při
zvýšené teplotě v rozpouštědle, které neovlivňuje škodlivě
reakci. Sloučeniny vzorce I mohou být dále zpracovány na
sloučeniny vzorce V, kteréjsou užitečné pň léčení, mezi
jinýmmigrény.
Patent CZ-367697-A3 (CZ)
Title: Process for preparing allyl halide and reaction vessel for making the same
Inventor: TIRTOWIDJOJO MAX M
IPC: B01J19/24
Filed: 1996-02-27
Abstract: Allyl halide is produced in high yields and purity with minimal carbon formation using a process of (1) initially reacting propylene and molecular halogen in a molar ratio of at least 2.5:1 in a "continuously stirred tank reactor" (CSTR) zone under conditions suitable to provide a reaction temperature of 400°C to 525°C to partially convert propylene and chlorine into allyl chloride; and (2) feeding an effluent from Step (1) into a plug-flow reactor zone where the reaction is continued at a temperature of 400°C to 525°C until essentially all of the chlorine is consumed. A preferred reactor for the process contains: (1) a spherical, egg-shaped or oval reactor zone (1); (2) a tubular reactor zone (2) attached to the spherical, egg-shaped or oval reactor zone (1); (3) one or more inlets (3,4) for injecting gaseous reagents into the spherical, oval or egg-shaped reactor zone (1); and (4) one or more outlets (5) from the tubular reactor zone (2) for withdrawing a gaseous product.
Patent CZ-419199-A3 (CZ)
Inventor: OTTOSEN ERIK RYTTER
IPC: C07D213/75
Filed: 1998-05-15
Abstract: Předkládané řešení se týká dosud neznámých sloučenin
charakterizovaných vzorcemI, nebojejichtautomemími
formami, přičemž připojení pyridinového kruhu bývá v poloze
3 nebo 4, a v kterých R] představujejeden nebo více
substituentů, které mohou být stejné nebo různé ajsou
vybrané ze skupiny obsahující vodík, halogen, trifluorometyl,
I karboxy, C i_4alkyl, alkoxy nebo alkoxykarbonyl, nitro, amino
1 ή ,j'nebo kyano substituenty, aQpředstavuje C9-C2o divalentní
uhlovodíkový radikál, který může být nasycený, alifatický
nebo větvený, nebo Q představuje C4-C20 divalentní
uhlovodíkový radikál, který může být cyklický nebo
nenasycený, aX představuje atom kyslíku, síry nebo dusíku,
přičemž dusíkmůže být i substituován vodíkemnebo Cμ
4alkylemaR2 představujejeden nebo více substituentů, které
mohou být stejné nebo různé ajsou vybrané ze skupiny
obsahující vodík, C i^alkyl, nebo alkoxy, hydroxy, halogen,
trifluormetyl, kyano, karboxamido, sulfámoyl, nebo nitro
substituenty; ajejich farmaceuticky přijatelné netoxické sole a
N-oxidy. Tyto sloučeniny mají významv humánní i
veterinární lékařské praxi jako inhibitory nežádoucí buněčné
proliferace.
Patent CZ-433898-A3 (CZ)
Title: Nonaqueous protic peptide formulations
Inventor: ECKENHOFF JAMES B
IPC: A61P13/08
Filed: 1997-07-01
Abstract: This invention relates to stable non-aqueous protic formulations of peptide compounds. These stable formulations comprise peptide in non-aqueous protic solvent. They may be stored at elevated temperatures for long periods of time and are especially useful in implantable delivery devices for long term delivery of drug.
Patent CZ-456199-A3 (CZ)
Inventor: MUNKERT EDWIN
IPC: B31F1/08
Filed: 1999-12-15
Abstract: Způsob výroby skládané tiskoviny, která sestává alespoň
z jednoho přeloženého archu, přičemž počet papírových pásů,
odpovídající počtu archů, ze kterých bude po rozříznutí
tiskovina vytvořena je před tímto rozříznutím veden vedle
sebe přes oblast vysokonapěťového pole, kdy se nanese
elektrostatický náboj alespoň najeden pás papíru probíhá tak,
že se vytvoří potenciálová rovina, opatřená z obou stran
směrem ven orientovaným stejnoměrným potenciálem, a tato
se uspořádá paralelně s uvnitř tiskoviny uspořádanou rovinou
lomu, takže na každý boční díl vyráběné tiskoviny,
uspořádaný po stranách potencionálové roviny, se nanese
stejně velký a stejně orientovaný náboj. Zařízení k provádění
tohoto způsobuje opatřeno alespoň jednou oblastí s alespoň
třemi, vůči sobě a vůči rovině lomu vyráběné tiskoviny
paralelně uspořádanými a proběh alespoň jednoho
přeloženého pásu (3, 4) papíru umožňujícími, elektrodovými
jednotkami (13, 14,16), z nichž ta střední definuje rovinu
lomu tiskoviny. Elektrodové jednotky mohou tvořit též vodicí
válečky (8, 9) a/nebo vodivý plech (11).
Patent SK-107199-A3 (SK)
Title: Bicyclic aromatic amino acids
Inventor: DIEFENBACH BEATE
IPC: C07D265/36
Filed: 1998-02-06
Abstract: The invention relates to compounds of formula (I), wherein X, Y, Z, R<1>, R<2>, R<3>, R<4>, R<5>, R<7>, R<8>, R<11>, m and n have the meaning cited in Claim 1, and to their physiologically acceptable salts. Said compounds can be used as integrin inhibitors, specially for prophylaxis and treatment of circulatory diseases, thrombosis, infarcts, coronary heart diseases, arteriosclerosis, osteoporosis, pathological symptoms sustained or propagated by angiogenesis and in tumor therapy.