baber/WOPTO huggingface dataset:
Patent CO-6190619-A2 (CO)
Title: Derivados de 2- quinolinona y 2-quinoxalinona y su uso como agentes antibacterianos
Inventor: COMITA-PREVOIR JANELLE
IPC: C07D493/04
Filed: 2009-07-02
Abstract: 1.- Un compuesto de la fórmula (I):o una sal farmaceuticamente aceptable del mismo, en donde el compuesto de la fórmula es sustancialmente libre de una mezcla cis (±) de sus enantiómeros, y en donde A se selecciona a partir de CH y N; D se selecciona a partir de C- R7 y N; en donde al menos uno entre A y D es carbono; E se selecciona a partir de O, NH, y S, en donde: i) E es NH si R8 y R9 juntos forman =O; y ii) E es O o S si R8 y R9 son cada uno H; G se selecciona a partir de O y S; J se selecciona a partir de C- R4 y N; R1 se selecciona a partir de H, halo, ciano, C1-6alquilo, C2-6alquenilo, y C2-6alquinilo R1a y - N(R1a), en donde dichos C1-6alquilo, C2-6alquenilo, y C2-6alquinilo son opcionalmente sustituidos con uno o más R10;R1a en cada ocurrencia se selecciona independientemente a partir de H y C1-6alquilo, en donde dicho C1-6alquilo es opcionalmente sustituido con uno o más R20;R2 se selecciona a partir de halo, ciano, C1-6alquilo, C2-6alquenilo, C2-6alquinilo, -OR2a, -N(R2a) en donde dichos C1-6alquilo, C2-6alquenilo, y C2-6alquinilo son opcionalmente sustituidos con uno o más R20;R2a en cada ocurrencia se selecciona independientemente a partir de H y C1-6alquilo, en donde dicho C1-6alquilo es opcionalmente sustituido con uno o más R20; R3 se selecciona a partir de H, halo, ciano, C1-6alquilo, C2-6alquenilo, y C2-6alquinilo, OR3a y -N(R3a) 2, en donde dichos C1-6alquilo, C2-6alquenilo, y C2-6alquinilo son opcionalmente sustituidos con uno o más R30;R3a en cada ocurrencia se selecciona independientemente a partir de H y C1-6alquilo, en donde dicho C1-6alquilo es opcionalmente sustituido con uno o más R30;R4 se selecciona a partir de H, halo, ciano, -CO2H, C1-6alquilo, C2-6alquenilo, y C2-6 alquinilo, en donde dicho C1- 6alquilo, C2-6alquenilo, y C2-6alquinilo son opcionalmente sustituidos con uno o más R40;R6 se selecciona a partir de fluoro, C1-6alquilo, C2-6alquenilo, C2-6alquinilo, -OR6a, en donde dichos C1-6alquilo, C2-6alquenilo, y C2-6alquinilo son opcionalmente sustituidos con uno o más R60; ...
Patent CO-6220937-A2 (CO)
Title: Compuestos triciclicos composiciones y procedimientos
Inventor: CHENG HENGMIAO
IPC: A61K31/44
Filed: 2009-07-31
Abstract: En una realización, la invención se refiere a un compuesto de Fórmula I:en la que R1 es -H o -P(O)(OH)2; o una sal del mismo. En otra realización, la invención se refiere a composiciones que comprenden un compuesto de Fórmula I y un vehículo. En otra realización, la invención se refiere a un procedimiento de poner en contacto un receptor de glucocorticosteroides con un compuesto de Fórmula I. Una realización adicional incluye procedimientos de tratamiento de una afección en un sujeto mediado por la actividad del receptor de glucocorticosteroides mediante la administración al sujeto de un compuesto de Fórmula I. 1.- Un compuesto de fórmula I:en la que R1 es -H; o sal del mismo. 2.- El compuesto de la reivindicación 1, en el que el compuesto es:o sal del mismo. 3.- El compuesto de la reivindicación 1, en el que el compuesto es:4.- Una sal clorhidrato del compuesto de la reivindicación 1.5.- Una composición que comprende el compuesto de la reivindicación 1 o sal del mismo y un vehículo. 6.- Un procedimiento que comprende poner en contacto un receptor de glucocorticosteroides con el compuesto de la reivindicación 1 o sal del mismo.
Patent CO-6260119-A2 (CO)
Title: Paquete doble con conector integral
Inventor: BOURGOIN PHILIPPE
IPC: B65D5/00
Filed: 2010-02-18
Abstract: 1.- Un recipiente para artículos para fumar comprendiendo al menos dos paquetes conectados de manera engoznada (2, 5), cada uno para alojar un haz separado de artículos para fumar, en donde en una posición inicial el recipiente comprende: un primer paquete (2) teniendo una primera pared (11, 51) con primero y segundo bordes opuestos y un conector integral (17, 57) que se extiende a través de la primera pared (11, 51), el conector integral (17, 57) que comprende una primera sección (18, 58) engoznada alrededor del primer borde de la primera pared (11, 51) y una segunda sección (19, 59) engoznada alrededor del segundo borde de la primera pared (11, 51); yun segundo paquete (5) teniendo una primera pared (31, 71) con primero y segundo bordes opuestos y un conector integral (37, 77) que se extiende a través de la primera pared (31, 71), el conector integral (37, 77) comprendiendo una primera sección (38, 78) engoznada alrededor del segundo borde de la primera pared (31, 71) y una segunda sección (39, 79) engoznada alrededor del primer borde de la primera pared (31, 71), en donde la primera sección (18, 58) del conector integral (17, 57) del primer paquete (2) se fija a la primera sección (38, 78) del conector integral (37 77) del segundo paquete y la segunda sección (19, 59) del conector integral (17, 57) del primer paquete se fija a la segunda sección (38, 78) del conector integral (37, 77) del segundo paquete, de manera que los primeros bordes de las primeras paredes (11, 51, 31, 71) del primero (2) y segundo (5) paquetes están adyacentes y los segundos bordes de las primeras paredes (11, 51, 31, 71) del primero (2) y segundo (5) paquetes están adyacentes.
Patent CO-6511246-A2 (CO)
Title: Dispositivo de distribución de liquido
Inventor: PAINCHAUD GAETAN
IPC: A61F9/00
Filed: 2012-03-15
Abstract: La presente invención se refiere a un dispositivo de distribución de líquido que comprende: - un depósito (12) para el almacenamiento del líquido a ser distribuido, - una contera (10) de distribución colocada sobre el depósito, provista de un soporte (14) y de una valva (16) de distribución de líquido, pudiendo dicha valva tomar una configuración de bloqueo y una configuración de paso de líquido, por cooperación con soporte (14), - un órgano (20) denominado de reducción de flujo, que comprende una forma (74) de desviación de líquido que delimita un canal (76) de reducción de flujo, siendo tal órgano (20) de reducción de flujo una pieza distinta del soporte (14) y distinta de la valva (16).
Patent CO-6531459-A2 (CO)
Title: Uso de 4-[etil(dimetil)amonio] butanoato en el tratamiento de enfermedades cardiovasculares
Inventor: KALVINS IVARS
IPC: C07C229/12
Filed: 2012-04-20
Abstract: Nuevo compuesto 4-[etil(dimetil)amonio]butanoato, método de preparación del mismo y su uso en el tratamiento de enfermedades cardiovasculares.
Patent CO-6771403-A2 (CO)
Title: Derivado de acilbenceno
Inventor: YAMANOI SHIGEO
IPC: A61K31/4245
Filed: 2013-05-10
Abstract: Se proveen compuestos que tienen una excelente acción hipoglucémica y una acción protectora de las células ß o el páncreas, o una sal farmacéuticamente aceptable de los mismos; y una composición farmacéutica que tiene un excelente efecto terapéutico y/o efecto profiláctico sobre la diabetes de tipo 1, la diabetes de tipo 2, etcétera, que causan un aumento del nivel de azúcar en la sangre debido al metabolismo anormal del azúcar; se describe un compuesto representado por la fórmula general (I), o una sal farmacéuticamente del mismo.
Patent CO-6761386-A2 (CO)
Title: Derivados de pirrolopiridina y pirrolopirimidina sustituidos con ciclobutilo como inhibidores de jak
Inventor: RODGERS JAMES D
IPC: C07D471/04
Filed: 2013-05-31
Abstract: La presente invención provee pirrolopirimidinas y pirrolopiridinas sustituidas con ciclobutilo de la fórmula I:en donde X, Y, Z, L, A, R5, n y m se definen con anterioridad, así como sus composiciones y métodos de uso que modulan la actividad de Janus quinasas (JAKs) y son de utilidad en el tratamiento de enfermedades relacionadas con la actividad de JAKs que incluyen, por ejemplo, trastornos inflamatorios, trastornos autoinmunes, cáncer y otras enfermedades
Patent CO-6781549-A2 (CO)
Title: Uso de ligandos sigma en dolor por cáncer de huesos
Inventor: ZAMANILLO-CASTANEDO DANIEL
IPC: A61K31/4152
Filed: 2013-07-02
Abstract: La invención se refiere al uso de un ligando sigma, particularmente un ligando sigma de fórmula (1) para prevenir y/o tratar dolor asociado a cáncer de huesos.
Patent CO-7141449-A2 (CO)
Title: Escobilla limpiaparabrisas
Inventor: TOLENTINO VAMBI RAYMUNDO
IPC: B60S1/38
Filed: 2014-09-23
Abstract: Se presenta una escobilla limpiaparabrisas que tiene una regleta limpiadora, un marco primario, y un par de marcos secundarios. El marco primario tiene un dispositivo de unión capaz de unir la escobilla limpiaparabrisas con un brazo limpiador dispuesto en un lado superior del marco primario, y una estructura de unión dispuesta en extremos opuestos del marco primario. En el par de marcos secundarios, cada uno tiene una parte de unión de pivote central y dos partes de brazos que se extienden desde la parte de unión de pivote central, una estructura de pivote dispuesta en la parte de unión de pivote central de los marcos secundarios en donde la estructura de pivote de los marcos secundarios está unida a las estructuras de unión en los extremos del marco primario. También se presenta una escobilla limpiaparabrisas que tiene una regleta limpiadora, una estructura de distribución de fuerza que tiene extremos opuestos, y una cubierta.
Patent EP-1039145-A2 (EP)
Inventor: KOETTER WOLFGANG
IPC: F15B13/044
Filed: 2000-01-04
Abstract: The controller controls the flow of hydraulic medium to a hydraulic control motor depending on electrical input signals to a magnetic drive that displaces a control sliding element in a valve housing from a spring-centered central position into working positions on either side. The sliding element is centered by a dual action restoring device, whereby inner and outer springs are arranged mutually concentrically on the same side of the control sliding element. A first adjuster has a first spring plate (34) in the form of a toothed wheel (43) and an externally adjustable setting spindle (45). A second spring plate (36) in the form of a toothed wheel (53) forms part of a transmission (57) externally adjustable via a second setting spindle (56).
Patent EP-0999571-A2 (EP)
Inventor: REYAL JEAN-PIERRE
IPC: H01J9/46
Filed: 1997-05-15
Abstract: Device for fixing the element on the frame wall comprises: upright (56) attached to plate having at least 2 locking tabs (60a, 60b) on the side of the frame (61) wall (62); spring (57) projecting on to an internal face of upright (56) coming into contact with the frame wall; and at least one strip (59a, 59b) comprising fixing bar (59'a, 59'b) at its end to attach the element on frame by clipping. The fixing bars (59'a, 59'b) of the strip (59a, 59b) are engaged on an element for retention of the frame (61) and the spring (57) compressed between the upright (56) and the wall (62) of the frame (61). The suspension element consists of a thin metal strip cut out and bent.
Patent EP-1038759-A2 (EP)
Inventor: TEAL RICHARD DONALD
IPC: B62D7/10
Filed: 2000-03-27
Abstract: The device includes a steering wheel (28) and means for restricting and/or changing the maximum steering range of the steering wheel. The steering wheel can be swivelled right and left of a neutral position up to a maximum of 90, 135, 180 or 270 degrees.  The maximum steering angle can be restricted by a stop (172) whose position can be changed relative to the vehicle and/or steering wheel or a transfer device in active connection therewith. The transfer device can have a steering spindle connected to a swivel-mounted sector toothed wheel.
Patent EP-1045194-A2 (EP)
Inventor: BRUEGGEMANN JUERGEN
IPC: F21V21/04
Filed: 2000-04-11
Abstract: A procedure for renovating a built-in ceiling lamp is described. On an old ceiling lamp (2-101) which is mounted on or in a ceiling is fastened a renovation lamp (11-100) which has one or more housing parts with one or more light exit openings. The renovation lamp has a cladding which extends to the side edges of the renovation lamp and forms, at least outside the region of light exit openings, a screen against being seen from below. The renovation lamp has a greater length and width than the old lam The renovation lamp is mounted so that the cladding comes to lie below the old lamp so that it screens the housing of the hold l at least outside the region of the light exit openings, essentially completely against being seen from below.
Patent EP-1048762-A2 (EP)
Inventor: ITO SYUNJI
IPC: D01H5/32
Filed: 2000-04-20
Abstract: Spinning machine includes draft rollers 3, 4 and 5
and a drive device for driving the draft rollers. The
drive device has a drive unit 6 for driving the front
draft roller 5, and a drive unit 7 for driving the back
and middle draft rollers 3 and 4. Each drive unit has a
variable speed motor M2 or M3 and a transmission
mechanism, and the variable speed motor of the drive
unit 6 for driving the front draft roller 5 is a
synchronous AC motor having permanent magnets. A reverse
rotation preventing device including a ratchet wheel and
a pawl is arranged in the drive unit 6 for preventing a
reverse rotation of the front draft roller 5, occurring
with a reverse rotation of the synchronous motor M2,
caused by the action of the permanent magnets in the
synchronous motor upon starting the synchronous motor.
Patent EP-1065473-A2 (EP)
Inventor: HAMAOKA TAKASHI
IPC: G01B7/30
Filed: 2000-06-27
Abstract: A stator core (25) has a detecting portion (37) located
at a center of a gap (30) penetrating the stator core in a diametric
direction and a Hall IC (31) arranged in the detecting portion.
Large gap portions (38) each having a distance G3 wider than a
distance G2 of the detecting portion are formed on both sides of
the detecting portion. Therefore, a magnetic flux passing through
the stator core is concentrated into the detecting portion (37),
and the magnetic flux density passing through the Hall IC is increased.
As a result, an output of the Hall IC is increased. The large gap
portion is formed to have a narrower distance G4 at an outer side
of the stator core, and the distance G4 is wider than an air gap
G1 between the permanent magnet (27) and the stator core (25).
Patent EP-1064865-A2 (EP)
Inventor: KURAHASHI CHITARO
IPC: A45C13/08
Filed: 2000-07-03
Abstract: A ring attachment structure for attaching a ring to an object to be
adorned includes an opening formed in the object for passage of a
band of a ring, a first attachment means formed with a through-hole
that is fitted in an area surrounded by the band of the ring, a second
attachment means formed with a hole that is fixed to the object at a
location adjacent to the opening in the object, the hole being positioned
to align with the through-hole of the first attachment means when the
first attachment means is fitted in the area surrounded by the band of
the ring and the band of the ring is passed through the opening, and a
locking member that passes through the aligned through-hole and
hole. The ring attachment structure facilitates use of rings in
unconventional ways.
Patent EP-1069617-A2 (EP)
Inventor: TANAKA SHINJI
IPC: H05K1/11
Filed: 2000-07-14
Abstract: A wiring layer on which X-directional signal lines
20 to 22 are arranged is formed on a multilayer board.
Rectangular power-source conductive patterns 10c are
arranged each in which via holes 120 are formed
longitudinally or in the wiring direction of the X-directional
signal lines 20 to 22. The area (batched with
broken lines) acts as a wiring channel for the X-directional
signal line 22.
Patent EP-1086934-A2 (EP)
Title: Zementzusammensetzungen, enthaltend redispergierbare Polymerisatpulver
Inventor: DREHER STEFAN DR
IPC: C09D1/08
Filed: 2000-08-09
Abstract: Zusammensetzungen auf Basis von Zement, enthaltend 1 bis 500 Gewichtsteile, bezogen auf 100 Gewichtsteile Zement, eines Polymerisats, aufgebaut aus a) 30 - 99,5 Gew.-% mindestens eines Alkylesters der (Meth)acrylsäure, b) 0 - 70 Gew.-% mindestens eines Vinylaromaten, c) 0,5 - 10 Gew.-% mindestens eines Alkylpolyethoxy(meth)acrylats der Formel <IMAGE> wobei R1 für eine H-Atom oder eine Methylgruppe , R2 für eine C1 bis C4 Alkylgruppe und n für eine ganze Zahl von 1 bis 55 steht. d) 0 - 10 Gew.-% mindestens einer ethylenisch ungesättigten Mono- oder Dicarbonsäuren wie Acrylsäure, Methacrylsäure, Maleinsäure, Itakonsäure, deren Anhydride, Amide oder Hydroxyalkylamide, e) 0 - 10 Gew.-% Acrylnitril oder Methacrylnitril, und f) 0 - 50 Gew.-% weiteren, von a) bis e) verschiedenen ethylenisch ungesättigten Verbindungen.
Patent EP-1085354-A2 (EP)
Inventor: NISHIMURA MASAYUKI
IPC: G02B6/34
Filed: 2000-09-07
Abstract: A planar lightwave circuit (PLC) of a PLC module
is provided with many waveguides including a plurality
of input (output) optical waveguide on a substrate.
Junction faces between these input (output) optical
waveguide and input (output) optical fibers are slant
against the optical axis thereof. The PLC module has
photodetectors opposed to corresponding junction
faces disposed at the input-optical-fiber's-side
(output-optical-waveguide's-side).
Patent EP-1085623-A2 (EP)
Inventor: KAKIZAKI KOJI
IPC: H01S3/0971
Filed: 2000-09-15
Abstract: The oscillation pulse width is extended in a gas
laser apparatus emitting ultraviolet radiation by a high-repetition
rate oscillating operation. The gas laser
apparatus has a pair of laser discharge electrodes (3, 4)
connected to the output terminals of a magnetic pulse
compression circuit and disposed in a laser chamber (1). The
pulse width is extended by determining circuit constants
so that the period of the oscillating current flowing
between the discharge electrodes is shortened and, at the
same time, the peak value of the current is increased,
whereby the laser gas is continuously excited even during
at least one half-cycle subsequent to the first half-cycle
of the oscillating current to sustain the laser
oscillating operation.
Patent EP-1094308-A2 (EP)
Inventor: STATON KENNETH L
IPC: G01J1/46
Filed: 2000-10-04
Abstract: High quantum efficiency point detector system. The system includes a light source
generating a light beam having an area and includes a CCD detector (10) with a cell size
comparable to the light beam area. The CCD cell may include a single pixel or at least two
pixels.
Patent EP-1111249-A2 (EP)
Inventor: JAKSIC DAVORIN
IPC: F16B2/06
Filed: 2000-10-18
Abstract: The clamp for fixing a sensor (26) to a mounting bar (24) has jaws (11, 12) which fit around the bar and have a slot at the sensor end into which a mounting plate (32) fits. A bolt (22) is screwed into a bore at the other end to fasten the clamp.
Patent EP-1106587-A2 (EP)
Inventor: THIELE LOTHAR DR
IPC: C04B26/10
Filed: 2000-11-30
Abstract: A composite article comprises a mineral molded article having a solid adhesively bonded layer of gravel. An Independent claim is included for a process for the preparation of the article by coating a mineral molded article with a layer of gravel and binding agent and hardening the layer, optionally by heating.
Patent EP-1151825-A2 (EP)
Inventor: LIN FRANK S
IPC: B24B53/12
Filed: 2000-12-04
Abstract: The present invention discloses a CMP pad dresser which has a plurality of
uniformly spaced abrasive particles (180) protruding therefrom. The abrasive particles
(180) are super hard materials, and are typically diamond, polycrystalline diamond
(PCD), cubic boron nitride (cBN), or polycrystalline cubic boron nitride (PcBN). The
abrasive particles (180) are attacked to a substrate (40) which may be then coated with
an additional anti-corrosive layer (130). The anti-corrosive layer (130) is usually a
diamond or diamond-like carbon which is coated over the surface of the disk to prevent
erosion of the brazing alloy (90) by the chemical slurry used in conjunction with the
CMP pad. This immunity to chemical attack allows the CMP pad dresser to dress the
pad while it is polishing a workpiece. In addition to even spacing on the substrate (40),
the abrasive particles (180) extend for a uniform distance away from the substrate (40),
allowing for even grooming or dressing of a CMP pad both in vertical and horizontal
directions. A method of producing such a CMP pad dresser is also disclosed.
Patent EP-1108888-A2 (EP)
Inventor: BOLCICH ALEJANDRO JUAN ALFREDO
IPC: F03D1/04
Filed: 2000-12-12
Abstract: The invention provides a wind energy converter comprising a wind actuated rotor assembly rotatably mounted around a horizontal axis on the top of a support tower, the rotor assembly comprising two axially aligned and spaced apart rotors, each rotor comprising a plurality of blades, wherein the blades of one of the rotors have a pitch opposite to the pitch of the blades of the other rotor whereby the rotors rotate in opposite directions. <IMAGE>
Patent EP-1041551-A2 (EP)
Inventor: MUELLER ROBERT L
IPC: G11B17/22
Filed: 2000-03-14
Abstract: Data cartridge exchange apparatus (10) for allowing
a user to access a data cartridge (14) contained in a data
storage system (12) may comprise a cartridge engaging
assembly (16) mounted within the data storage system (12)
so that the cartridge engaging assembly (16) is moveable
along a displacement path (50). A panel (32) located
adjacent a portion of the displacement path (50) is
provided with a cartridge exchange aperture (34) therein
that is sized to pass the data cartridge (14).
Patent EP-1041288-A2 (EP)
Inventor: MAEJIMA YASUSHI
IPC: F04D19/04
Filed: 2000-03-28
Abstract: To facilitate the fabrication work of a stator column
assembly and improve full and wise use of resources, as well as
to prevent contact accident between a mold portion of a stator column
and a rotor shaft due to the thermal inflation. A first
electromagnet unit (30), a stator coil unit (20), and a second
electromagnet unit (40) are engaged to and arranged in a cylindrical
stator column (11) in the order stated, the first electromagnet
unit (30) comprising an electromagnet (31) of a first active radial
magnetic bearing and a radial displacement sensor (32) for the
electromagnet (31) which are attached in a first circular holding
member (30c) to be coated and molded with a resin mold (30d), the
stator coil unit (20) comprising a stator coil (21a) that is attached
in a circular yoke member (20c) to be coated and molded with a resin
mold (20d), the second electromagnet unit (40) comprising an
electromagnet (41) of a second active radial magnetic bearing and
a radial displacement sensor (42) for the electromagnet (41) which
are attached in a second circular holding member (40c) to be coated
and molded with a resin mold (40d).
Patent EP-1059372-A2 (EP)
Inventor: OCHI TAKASHI
IPC: D03D15/56
Filed: 2000-06-06
Abstract: A soft stretch yarn substantially comprising polyester
fibres has a stress, at 50% yarn stretch, of no more
than 30x10 -3  cN/dtex and, at the same time, a percentage
recovery of at least 60%. Preferably, the Uster
unevenness is no more than 2.0% and the crimp diameter
is no more than 250 µm. This soft stretch yarn can be
produced by spinning yarn of conjugate fibres comprising
two types of polyester in which one component is PTT at
a take-up velocity of at least 1200 m/min, drawing at a
drawing temperature of 50 to 80°C at a draw ratio such
that the drawn yarn tensile elongation is 20 to 45%, and
then heat setting.
Patent EP-1143967-A2 (EP)
Inventor: CARRAZANA ENRIQUE
IPC: A61P25/06
Filed: 2000-01-13
Abstract: Anticonvulsant derivatives useful in treating cluster headaches are disclosed.