baber/WOPTO huggingface dataset:
Patent SG-10201809066T-A (SG)
Title: 5,6-Disubstituted Pyridine-2-Carboxamides and 5,6-Disubstituted Pyrazine-2-Carboxamides as Cannabinoid Receptor Agonists
Inventor: GOBBI LUCA
Filed: 2015-04-01
Abstract: Novel Pyridine Derivatives The invention relates to a compound of formula (I) A N R 1 R 2 N O R 3 R 4 (I) wherein A and R 1 to R 4 are defined as in the description and in the claims. The compound of formula (I) can be used as a medicament. [No Available Figure] PYRIDINE-2-AMIDES USEFUL AS CB2 AGONISTS 5,6-Disubstituted pyridine-2-carboxamides and 5,6-Disubstituted pyrazine-2-carboxamides as Cannabinoid Receptor Agonists 5,6-Disubstituted Pyridine-2-Carboxamides and 5,6-Disubstituted Pyrazine-2-Carboxamides as Cannabinoid Receptor Agonists
Patent SG-11201807677Y-A (SG)
Title: Antibodies to cd40 with enhanced agonist activity
Inventor: RAVETCH JEFFREY
IPC: C07K16/28
Filed: 2016-06-28
Abstract: INTERNATIONAL APPLICATION PUBLISHED UNDER THE PATENT COOPERATION TREATY (PCT) (19) World Intellectual Property Organization International Bureau (43) International Publication Date 8 September 2017 (08.09.2017) WIPO I PCT (10) International Publication Number WO 2017/151176 Al 11111111111111011101111111111101011111011101111111101110101111111111111111110111111 (51) International Patent Classification: C07K 16/28 (2006.01) A61K 39/00 (2006.01) (21) International Application Number: PCT/US2016/039785 (22) International Filing Date: 28 June 2016 (28.06.2016) (25) Filing Language: English (26) Publication Language: English (30) Priority Data: 62/304,012 4 March 2016 (04.03.2016) US (71) Applicant: THE ROCKEFELLER UNIVERSITY [US/US]; 1230 York Avenue, New York, NY 10065 (US). (72) Inventors: RAVETCH, Jeffrey, V.; 1230 York Avenue, New York, NY 10065 (US). DAHAN, Rony; 1230 York Avenue, New York, NY 10065 (US). (74) Agents: NORTON, Gerard, P. et al.; Fox Rothschild LLP, 997 Lenox Drive, Building 3, Lawrenceville, NJ 08648-2311 (US). (81) Designated States (unless otherwise indicated, for every kind of national protection available): AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, Fl, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JP, KE, KG, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW. (84) Designated States (unless otherwise indicated, for every kind of regional protection available): ARIPO (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW), Eurasian (AM, AZ, BY, KG, KZ, RU, TJ, TM), European (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR), OAPI (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG). Declarations under Rule 4.17: as to applicant's entitlement to apply for and be granted a patent (Rule 4.1700) as to the applicant's entitlement to claim the priority of the earlier application (Rule 4.17(iii)) Published: with international search report (Art. 21(3)) with sequence listing part of description (Rule 5.2(a)) W O 20 17 / 15 117 6 Al (54) Title: ANTIBODIES TO CD40 WITH ENHANCED AGONIST ACTIVITY (57) : Provided herein are agonistic antibodies, or antigen binding portions thereof, that bind to human CD40. Such anti- bodies optionally comprise Fc regions with enhanced specificity for FcYRIIb. The invention also provides methods of treatment of cancer or chronic infection by administering the antibodies of the invention to a subject in need thereof.
Patent SG-11201811374S-A (SG)
Title: Offline payment method and device
Inventor: SUN YUANBO
IPC: G06Q20/40
Filed: 2017-06-07
Abstract: The application an payment and device. method the obtaining, a payment an identity authentication identifier of a user that sends an offline payment request when the third-party payment application receives the request that corresponds to a target 5 payment obtaining, the payment ication, offline payment certificate issued by the target payment application to the user and stored in the device, it determined the identity identifier is verified; and providing, by the third-party payment application, the offline payment certificate for an offline payment service party, so that the offline payment 10 service party requests the target payment application to process offline payment of the user on offline certificate. present ication user's payment and secure a application selected a third-party payment application integrated into a consumer terminal device to make offline payment. 15
Patent AT-395287-B (AT)
Title: Shaped cushion, especially for use as a pillow
IPC: A47G9/10
Filed: 1991-01-08
Granted: 1992-11-10
Abstract: Shaped cushion, especially for use as a pillow, comprising a preferably seamed sleeve and a filling, the filling consisting of material which can be shaped or which consists of small pieces, and the filled sleeve having the shape of a cylindrical roll 1 with a wedge 2 attached to the circumference 3 of the cylinder, parallel to its axis. <IMAGE>
Patent AT-398008-B (AT)
Title: Holographic sundial
IPC: G03H1/24
Filed: 1992-03-27
Granted: 1994-08-25
Abstract: The sundial consists of two reflection holograms 1, 2 which reconstruct a virtual scale 6 with indications of time of day and of season, as well as a virtual pointer 5 which in this case does not throw a shadow on the scale but functions as a kind of sight. The observer looks, as through an aiming device, along the hour pointer 5 which points to a given point on the scale. As the sun 3, as the reconstruction light source, travels on its course during the day, the pointer 5 will point in different directions at different times of the day. If the position of the sun and the behaviour of the holograms 1, 2 is calculated at different angles of incidence of the reconstruction light source, the direction in which the pointer 5 points, or the position of the scale 6, is known. The direction of the pointer 5 must be intersected by the scale plane 6 in order to obtain the point of inscription for a given time of day or season. <IMAGE>
Patent DK-164374-B (DK)
Inventor: ROLIN INGMAR ERIK
IPC: F24F13/068
Filed: 1988-01-26
Abstract: A method of introducing supply air into a lower portion of a room space (3) directly to an occupied zone (7) by means of at least one elongated air distribution means (1) provided with a plurality of outflow openings (2) for supply air. In order to blow supply air into the occupied zone without draught and without drawing impurities from the upper portion of the room space, supply air is blown from the air distribution means at a high speed but through outflow openings so small that the speed of the air jets (A) from the openings is reduced essentially over a short distance (X) and the entrance of secondary air (B) from the room space into the air jets is prevented in the vertical direction of the room space over said distance (X) and at least at one end of the air distribution means. The air distribution means (1) is provided with a plurality of small outflow openings (2) the distance of which from each other in the longitudinal direction of the air distribution means is great as compared with the size of the outflow opening for enabling secondary air to flow from the room space in between the outflow openings, and to mix with the air jets from all sides.
Patent DK-151627-B (DK)
Inventor: KARJALAINEN ARTO JOHANNES
IPC: C07D263/32
Filed: 1981-02-11
Abstract: The invention provides compounds of the formula:wherein each of R<sub>1</sub>, R<sub>2</sub> and R<sub>3</sub>, which can be the same or different is hydrogen, chloro, bromo, fluoro, methyl, ethyl, methoxv, amino, hydroxy or nitro; R<sub>4</sub> is hydrogen or alkyl of 1 to 7 carbon atoms; X is(R<sub>5</sub> is hydrogen or hydroxy) and n is 1-4; and their non-toxic pharmaceutically acceptable acid addition salts. These compounds exhibitvaluable pharmacological activity and are useful in the treatment of mammals, especially as anti- hypertensive agents. Furthermore, some of the compounds have proved to possess diuretic, ß-blocking activity and/or antithrombotic activity. The compounds may be made by a variety of methods and may be incorporated in pharmaceutical compositions also comprising a compatible pharmaceutically acceptable carrier.
Patent DK-157146-B (DK)
Inventor: ERIKSSON INGEMAR
IPC: G01M3/26
Filed: 1985-02-07
Abstract: A method and a device for testing the tightness of an engine of the kind having at least one cylinder (1 ),a piston (2) movable therein and a crankcase (3) with crank means (4, 5), which are drivable by the piston, is based on measuring of the leakage of gases passing the piston into the crankcase by connection of a measuring apparatus (8) so that it communicates with the interior of the crank case.
Patent HU-183347-B (HU)
Inventor: KRIEGLER JANOS
IPC: H03K17/14
Filed: 1981-03-02
Abstract: A találmány olyan tápegység, amelynek bemenőkapcsára vagy áramforrására kapcsolt olvadóbiztosítéka, bekapcsoló beavatkozó-, és/vagy kezelőszerv útján vezérelt bekapcsolóegységből, és üzemi kikapcsoló beavatkozó-, és/vagy kezelőszerv útján, továbbá feszültségérzékelő által vezérelt feszültségeséskikapcsoló egységből álló vezérlő egysége van, úgy kialakítva, hogy az üzemáramkapcsolóval párhuzamosan újabb (belső) feszültségesésérzékelő van kötve, amelynek kimenete jelfeldolgozó egység bemenetére csatlakozik, mely utóbbi további bemenete vészkikapcsoló vezérlő kimenetére csatlakozik, a kimenet pedig vészkikapcsoló bemenetére van kapcsolva. A találmány szerinti tápegység robbanásveszélyes helyeken is működtethető.  -1-
Patent HU-203137-B (HU)
Inventor: DEME EVA
IPC: D06P5/00
Filed: 1987-02-10
Abstract: Eljárás nyomott textilkelmék előállítására, rotációs filmnyomógépen, habfázisű technológia alkalmazásával, úgy, hogy az alkalmazott textilszínezékek viszkozitását textilsűrítökkel és/vagy hígítókkal a habfázisú nyomógépek esetén 15-30 dPas, a nem habfázisú díszítő színezékek esetén pedig 35-70 dPas értékre beállítjuk. A textilkelmét a nagyobb felületet takaró színekkel, rotációs filmnyomógépen, habfázisű színezékeket tartalmazó nyomópéppel nyomjuk, majd a nem habfázisú díszítő színekkel tovább mintázzuk. Végül a textilkelmét ismert módon szárítjuk, színrögzítjük. Az eljárás alkalmas marőnyomott hatású, akár mindkét oldalán több színnel is mintázott textilkelmék előállítására.
Patent HU-196344-B (HU)
Title: Process and apparatus for treating liquide materials containing organic materials first of all waste materials, liquide manure and sewage-sludge
Inventor: CSEPREGI LASZLO
IPC: C02F11/00
Filed: 1986-02-12
Abstract: Liquids contg. organic materials, esp. wastes such as dilute manure and sewage sludge, to be treated are routed to concentric reactor spaces. The raw liquid is introduced from below, under pressure into the first reactor space. Acidic fermentation takes place and hydrogen gas is developed which is fed to the lower part of the second reactor space to produce floatation in the liquid. Liquid is intermittently withdrawn from the first reactor space by overflowing into discharge throats. It is routed into the second reactor space where methanogen decomposition occurs. The methane developed is piped away and the liquid overflows into the third reactor space, where it is sterilised at 50-55 deg.C and discharged from the reactor.
Patent HU-193103-B (HU)
Inventor: FARKAS JOZSEF
IPC: B23B5/44
Filed: 1985-02-21
Abstract: A találmány lehetővé teszi törtvonalas profilok forgácsolását elektronikus zárthurkú szabályozással; az üzem közben szükséges leállások esetén is fenntartható a szöghelyes együttfutás, kedvezőbb feltételek között és hosszú élettartamon át biztosítható a pontosság; elmaradnak az ilyen típusú mechanikai szabályozórendszereknél elkerülhetetlen járulékos zajkomponensek és bonyolult, eszközés időigényes manuális beavatkozó műveletek. A sokszögforgácsolás ismert elve szerint— a töréspontok számának megfelelő áttétellel— futtatunk együtt fő orsót és excci ter orsókat, de indítás előtt az excenter orsókat a kiindulási szöghelyzetbe, a fő orsót előírt mértékű szögkésésnek megfelelő helyzetbe állítjuk, és ehhez a kiindulási állapothoz időzítjük az együttfutást és spirálalkotójú profilok esetén az előtoló szerkezet mozgását is. Két zárthurkú szabályozó láncot alkalmazunk, amelyek fő ágai egy-egy szervomotort működtetnek. A szervomotorok (35, 317) egyfelől ellenőrzőjelet szolgáltató visszavezető hurkon (la, Ila), másfelől impulzusadót (37, 319) és vezérlő egységgel (320) csatolt digitális eszközt tartalmazó visszavezető hurkon (lb, Ilb) át vannak a megfelelő fő ág különbségképzőjével (32, 315) csatolva, és az első szabályozó lánc impulzusadójával (37) csatolt illesztő szerven át van a két lánc egymással csatolva. (3. ábra)  -1-
Patent HU-193280-B (HU)
Inventor: CALDWELL ALBERT GORDON
IPC: C07D233/88
Filed: 1984-02-17
Abstract: A találmány tárgya eljárás az (I) általános képletű új hidantoinszármazékok, valamint az ezeket hatóanyagként tartalmazó gyógyászati készítmények előállítására. A képletben Z jelentése hidrogénatom vagy alkilcsoport, Z1 jelentése karbonsavcsoport és Z2 jelentése helyettesített aminocsoport. Az eljárás során egy (II) általános képletű vegyületet reagáltatnak egy (III) általános képletű vegyülettel, és a kapott (I) általános képletű vegyületet kívánt esetben más (I) általános képletű vegyületté alakítják. Az (I) általános képletű vegyületek a természetes prosztaglandinokéhoz hasonló farmakológiai tulajdonságokkal bírnak, azok mimetikumaiként vagy antagonistáiként alkalmazhatóak.  -1-
Patent HU-207831-B (HU)
Title: Process for producing enanthiomere mixtures of nitrogen-containing bases dividing raceme composition
Inventor: ACS MARIA
IPC: C07B57/00
Filed: 1991-02-27
Abstract: This method simplifies the usual long and material consuming procedures by sepg. one enatiometer by addn. of a royal cpd., leaving the other enantiometer, which comprises the optical isomer, behind. The royal cpd. is then removal by usual methods
Patent HU-206460-B (HU)
Title: Apparatus for settling sludge or/and water containing scale originating from metallurgy of ferrous metals
Inventor: ADAMIS GEZA
IPC: B03D3/00
Filed: 1990-02-06
Abstract: The equipment comprises a settling space, liq. feed and clarified water and sludge discharge, to deal with slurry and/or water effluent of iron smelting activities. The settling space is a basin with pref. circular cross section which decreases in the downward direction. It has an outer wall (2b), bottom (2a) and a central downcomer (31). The bottom of the downcomer is set at a distance above the bottom plate (2a). Its top end is extended above the liq. level (V2) of the basin (2). The cross section of the basin decreases more rapidly below the bottom of the downcomer (31). The inlet channel (1) is joined to the downcomer (31), pref. above the liq. level (V2). The outside of the downcomer (31) is joined to a conical inner wall (4) which forms the boundary of the clarified water space (37). The top of this inner wall carries a collector trough (36) with a stilling/level control weir. A divider wall (41) is also located between the downcomer (31) and the inner wall (4). This carries a feed trough (5), also equipped with a level control weir, which is fed from the collector trough (36). Clarified water is removed by a submersible pump (52) located on the side of the divider wall (41) which is opposite the feed trough (5).(Dwg.1/19)
Patent HU-202905-B (HU)
Title: Process for reducing temperature in the regeneration zone of fluidized catalytic cracking process
Inventor: LENGEMANN ROBERT A
IPC: C10G11/14
Filed: 1986-02-19
Abstract: A method for operating a fluid catalytic cracking unit comprising a regeneration zone and a reaction zone with a relatively reduced temperature in the regeneration zone while processing a high-coke-making hydrocarbon feedstock having a 50 volume percent distillation temperature greater than about 500 DEG F (260 DEG C) which method comprises contacting at conversion conditions the feedstock in a reaction zone with a fluidizable mixture of regenerated cracking catalyst and low-coke-make non-catalytic solid particles, comprising a refractory inorganic oxide, in a ratio of low-coke-make solid particles to cracking catalyst from about 1:100 to about 10:1, the low-coke-make solid particles having a surface area of less than about 5 m<2>/g and a coke making capability of less than about 0.2 weight percent coke in the ASTM standard method for testing cracking catalyst by microactivity (MAT); separating the resulting hydrocarbon products from the mixture of deactivated cracking catalyst and low-coke-make solid particles; recovering the hydrocarbon products; passing the mixture of cracking catalyst and low-coke-make solid particles to the regeneration zone for generation by removal of coke; and passing the resulting regenerated mixture of cracking catalyst and low-coke-make solid particles from the regeneration zone to the reaction zone to contact the feedstock as described above whereby the regeneration zone temperature is maintained at a reduced temperature as compared to an equivalent operation without the use of the low-cake-make solid particles while simultaneously not reducing the coke burning capacity of the regeneration zone or affecting the operation of the reaction zone.
Patent HU-189124-B (HU)
Title: Process for producing chloromethyl-ester of penicillanic acid
Inventor: JASYS VYTAUTAS J
IPC: C07D519/00
Filed: 1982-03-22
Abstract: A process for the preparation of chloromethyl esters of penicillanic acids, using iodochloromethane or bromochloromethane and a tetraalkylammonium salt of the penicillanic acid, and their use in processes for the synthesis of penicillanic acid esters, using a halomethyl ester and the tetraalkylammonium salt of the penicillanic acid, which readily hydrolyze in vivo to antibacterial penicillins and the beta-lactamase inhibitor penicillanic acid sulfone.
Patent HU-203136-B (HU)
Title: Clouded mixture for producing textiles lasting form
Inventor: KALIJADA VALENTINA GRIGORIEVNA
IPC: F17D1/20
Filed: 1987-03-05
Abstract: Knitted fabrics of natural and synthetic fibres and cotton based underwear are dimensionally stabilised by a foamed mix. Treated articles are crease- and shrink-proof and are easily handled while cutting and sewing. The foamed mix contains a benzene-sulphonate of a methyl-di:amino-methyl deriv. of a di:ethylene-glycol-ester of a long chain fatt acid (ALKAMON OC-2) and of a polyethylene-glycol-ester of stearic acid (STEAROX 920) and consists of the following ingredients (g/l): 100-120 precondensate of a thermosetting resin, 3-5 ammonium-chloride, 3-5 urea, 10-21 ALKAMON OC-2, 10-20 STEAROX 920, Water: to 1l.
Patent LT-3989-B (LT)
Title: Cement flour - binding aggregate of materials, device and method for its preparing
Inventor: CHARTSCHENKO IGOR
IPC: C04B28/02
Filed: 1995-08-07
Abstract: A dry mix, for producing a cement suspension for filling and/or injecting pore spaces and cavities in loose rock or cavities and/or cracks in rock or in concrete components, is in the form of a ready mix containing (a) sulphate additive-free finely ground clinker and/or smelter sand powder; (b) additives; and (c) an ettringite-forming swelling component which produces swelling during strength development of the fine cement-binder mixture while the matrix is still soft after the filling and/or injection operation. The entire homogeneous dry mix has a continuous graduated particle distribution with sieve pass values of d95 = ≤ 24 (preferably ≤ 16) microns and d50 = ≤ 7 (preferably ≤ 5) microns, the d50/d95 ratio preferably being 0.33 plus or minus 0.04. Preferably, the mix contains a naphthalene sulphonate-formaldehyde condensate as plasticiser. Also claimed are: (a) preparation of the above dry mix, in which all the components have the above defined fineness and particle distribution and are stored separately in storage silos, certain components being dosed from the corresponding silos for delivery to a mixer and the components being homogenised and mixed in the mixer to form the ready mix; and (b) apparatus for carrying out the above process, in which a storage silo (7-12) is provided for each component and is combined with a dosing device, the silos being followed by a mixer (14).
Patent LT-3228-B (LT)
Title: Device for moulding of tubular thin-wall article, manufactured of concrete
Inventor: PASKEVICIUS VYTAUTAS
IPC: B28B1/08
Filed: 1993-05-11
Abstract: This invention belongs to the construction, fine-wall, and tubular product formation industry.This formation device consists of two parts, connected with screws, inner falsework and a punch. We choose the type of the form and the punch according to what kind of tubular product we want to form. The abovementioned are smooth, pointed-cone shaped with a fixed drill shaped element, orbicular, 3/4 truncated sphere shaped smooth - elastic, filled with mortises.The technological process of the product formation proceeds according to the technical solution of the punch type and the shape used.Using the inner plastic falsework, the outer form is removed immediately after product formation.With these technical formation solutions, we can form awry concrete tubular products of different diameters and wall thicknesses. They can be straight, muff, cloven, three-way, tetra-way, muffs, ramification, with passages for mounting plumbing manifolds.
Patent YU-48504-B (YU)
Inventor: MILAN VUKOJEVIC
Filed: 1995-03-13
Abstract: Uređaj za pretvaranje signalizacije D2/D2 u PCM signal 2Mb/s, naznačen time, što se izlazni PCM signal u HDB-3 kodu sa izlaza 2 kola (7) vodi na izlaz preko kola za uobličavanja impulsa (6) transformatora (5) i rastavnog konektora (4). - Prijava sadrži još 9 zavisnih zahteva.
Patent ZA-83773-B (ZA)
Title: Substituted dibenzodiazepinones,processes for their preparation,and pharmaceutical compositions containing these compounds
Inventor: WOLFHARD ENGEL DR
IPC: C07D451/06
Filed: 1983-02-04
Abstract: This invention relates to compounds of the formula   <IMAGE> wherein X is oxygen, -NH-, or-NCH3-and R is 1-methyl-4-piperidinyl, 4-methyl-1-piperazinyl, endo-8-methyl-8-azabicyclo[3.2.1]oct-3-yl, or exo-8-methyl-8-acabicyclo[3.2.1]oct-3-yl, each of which may optionally have an additional methyl substitutent, a diastereomer or enantiomer thereof, or a non-toxic, pharmacologically acceptable acid addition salt thereof with an inorganic or organic acid.
Patent ZA-84292-B (ZA)
Title: Process for the manufacture of beta-lactams
Inventor: SCHMID GERARD
IPC: C07D205/085
Filed: 1984-01-13
Abstract: 1. A process for the manufacture of optically uniform beta -lactams of the general formula  see diagramm : EP0116854,P10,F1  wherein R**1 signifies lower alkanoyl, lower alkoxycarbonyl or benzoyl, R**2 signifies hydrogen, lower alkyl, lower alkanoyl, lower alkoxycarbonyl or cyano, R**3 signifies hydrogen or lower alkyl, B signifies lower alkylidene, lower cycloalkylidene or carbonyl and Z signifies lower 2-alkenyl or 2,4-di(lower alkoxy)benzyl, whereby the residues denoted as lower have a maximum of 7 carbon atoms, and their corresponding optical antipodes, characterized by reacting a salt of a carboxylic acid of the general formula  see diagramm : EP0116854,P10,F2  wherein R**1, R**3 have the above significance, in the presence of a reactive derivative of an organic sulphonic acid and a base with an optically uniform compound of the general formula  see diagramm : EP0116854,P11,F3  wherein B and Z have the above significance, or the optical antipode thereof.