baber/WOPTO huggingface dataset:
Patent NO-20030624-D0 (NO)
Inventor: HENNEQUIN LAURENT FRANCOIS AND
IPC: A61K31/541
Filed: 2003-02-07
Abstract: The invention relatest to compounds of the formula (I) wherein either any one of G<SUB>1</SUB>, G<SUB>2</SUB>, G<SUB>3</SUB>, G<SUB>4 </SUB>and G<SUB>5 </SUB>is nitrogen and the other four are -CH-, or G<SUB>1</SUB>, G<SUB>2</SUB>, G<SUB>3</SUB>, G<SUB>4 </SUB>and G<SUB>5 </SUB>are all -CH-; Z is -O-, -NH-, -S-, -CH<SUB>2</SUB>- or a direct bond; Z is linked to any one of G<SUB>1</SUB>, G<SUB>2</SUB>, G<SUB>3 </SUB>and G<SUB>4 </SUB>which is a free carbon atom; n is an integer from 0 to 5; any of the substitutents R<SUP>1 </SUP>may be attached at any free carbon atom of the indole, azaindole or indazole group; m is an integer from 0 to 3; R<SUP>a </SUP>represents hydrogen; R<SUP>b </SUP>represents hydrogen or another value as defined herein; R<SUP>1 </SUP>represents hydrogen, oxo, hydroxy, halogeno, C<SUB>1-4</SUB>alkyl, C<SUB>1-4</SUB>alkoxy, C<SUB>1-4</SUB>alkoxy, C<SUB>1-4</SUB>-alkyl, aminoC<SUB>1-4</SUB>alkyl, C<SUB>1-3</SUB>alkylaminoC<SUB>1-4</SUB>alkyl, di(C<SUB>1-3</SUB>alkyl)aminoC<SUB>1-4</SUB>alkyl, -C<SUB>1-5</SUB>alkyl(ring B) wherein ring B is selected from azetidinyl, pyrrolidinyl, piperidinyl, piperazinyl, N-methylpiperazinly, N-ethylpiperazinyl, morpholino and thiomorpholino; R<SUP>2 </SUP>represents hydrogen, hydroxy, halogeno, cyano, nitro, trifluoromethyl, C<SUB>1-3</SUB>alkyl, C<SUB>1-3</SUB>alkoxy, C<SUB>1-3</SUB>aklylsulphanyl, -NR<SUP>3</SUP>R<SUP>4 </SUP>(wherein R<SUP>3 </SUP>and R<SUP>4</SUP>, which may be the same or different, each represents hydrogen or C<SUB>1-3</SUB>alkyl), or R<SUP>5</SUP>X<SUP>1</SUP>- (wherein R<SUP>5 </SUP>and X<SUP>1 </SUP>are as defined herein) and salts thereof, processes for the preparation of such compounds, pharmaceutical compositions containing a compound of formula I or a pharmaceutically acceptable salt thereof as active ingredient and the use of a compound of formula I in the manufacture of medicament for the production of an antiangiogenic and/or vascular permeability reducing effect in warm-blooded animals. The compounds of formula I and the pharmaceutically acceptable salts thereof inhibit the effects of VEGF, a property of value in the treatment of a number of disease states including cancer and rheumatoid arthritis.
Patent NO-20030828-D0 (NO)
Inventor: BUCHANAN JERRY E
IPC: B31B50/64
Filed: 2003-02-21
Abstract: A flexible container and method for making same are provided. The container comprises a base portion including a bottom, side walls, and an interior, the bottom defining a substantially flat planar surface when the container houses product and the container rests on its bottom, an upper panel portion, that is designed to be received within the interior of the base portion and includes side panels that define a closure member, the upper panel being so constructed and arranged to define a substantially flat surface when the closure member is closed and portions of the upper panel are folded over, the upper panel includes a portion that is sealed to the base portion, and a pair of handles may also be coupled to the base portion.
Patent NO-20030883-D0 (NO)
Inventor: HEAD PHILIP
IPC: E21B17/02
Filed: 2003-02-25
Abstract: A generally tubular drill string has a conductive path over a plurality of drill pipe section ( 10 ). Each drill pipe section has a first end and a second end, and a wall, and the first end has a first radial sealing surfaces ( 11 ) and the second end has a corresponding second radial surfaces ( 59 ), such that when the first or second end of one drill pipe section is engaged with the second or first end respectively of another drill pipe section, at least one seal is formed. The drill pipe includes at least one conductor ( 21 ) disposed inside it, this conductor being connected to a first contact means at the first end and a corresponding contact means at the second end of each drill pipe section. Ingress protection means ( 240 ) are provided to protect the contact means from ingress from inside or outside of the drill pipe section. The ingress protection means comprises a sealed volume surrounding the contact means.
Patent NO-20034672-D0 (NO)
Inventor: KANIOS DAVID P
IPC: B65D81/26
Filed: 2003-10-17
Abstract: A device and method for stabilizing a drug, particularly a chiral drug or the active enantiomer(s) thereof, in a carrier composition of a transdermal delivery system prior to the systems use by providing a product packaging system (14) to prevent or control degradation reactions that can result from certain packaging materials and moisture contamination, while at the same time providing a child-resistant wrapping (9) for the transdermal system.
Patent NO-20035173-D0 (NO)
Inventor: RIXON MARK W
IPC: C12N15/09
Filed: 2003-11-21
Abstract: Molecules that interfere with the binding of a tumor necrosis factor receptor with its ligand, such as a soluble receptor, have proven usefulness in both basic research and as therapeutics. The present invention provides improved soluble transmembrane activator and calcium modulator and cyclophilin ligand-interactor (TACI) receptors.
Patent NO-20052711-D0 (NO)
Inventor: SHIRLEY IAN MALCOLM
IPC: A01N25/00
Filed: 2005-06-06
Abstract: The stability of a particulate suspension comprising an aqueous phase containing substantially no miscible organic solvent having suspended therein an agrochemical solid substantially insoluble in said aqueous phase is enhanced by (i) forming a polymeric stabiliser having a hydrophilic moiety and a hydrophobic moiety by polymerising a plurality of vinylic monomers, not being exclusively vinylic esters or their hydrolysed products, at least some of which contain functional groups capable of undergoing cross-linking reactions and (ii) reacting said polymeric stabiliser with one or more substances contained (dissolved or suspended) in the aqueous phase capable of undergoing a cross-linking reaction with said functional groups, wherein the ratio by weight of (a) the polymeric stabiliser prior to cross-linking to (b) the suspended agrochemical is less than 1 part of polymeric stabiliser per 5 parts of suspended agrochemical.
Patent NO-20053713-D0 (NO)
Inventor: SIMONELLI DAVID
IPC: B25C1/00
Filed: 2005-08-01
Abstract: A fastener driving tool includes a housing assembly with a nosepiece assembly defining a drive track. A safety trip assembly includes a trigger enabling portion and a workpiece engaging portion and is movable between an extended disabling position and a retracted enabling position. The safety trip assembly is biased toward the extended position and is moved toward the retracted position by engagement between a workpiece and the workpiece engaging member. The workpiece engaging portion is movable to permit adjustment of a length of the safety trip assembly. The workpiece engaging portion may be removed from the safety trip assembly and exchanged with another different workpiece engaging portion. A workpiece engaging portion usable with the fastener driving tool includes a positioning mechanism having an opening locating structure and a guiding structure.
Patent GB-201019204-D0 (GB)
Title: An electro-optic waveguide polarisation modulator and a method of modulation
Filed: 2010-11-15
Abstract: An electro-optic waveguide polarisation modulator comprising 
first and second spaced apart cladding layers; 
a waveguide core sandwiched between the first and second cladding layers, the waveguide core having a higher refractive index than the cladding layers; 
a plurality of primary electrodes arranged on the opposite side of the first cladding layer to the core; and, 
at least one secondary electrode arranged on the opposite side of the second cladding layer to the core; 
the electrodes being arranged to provide an electric field having field components in two substantially perpendicular directions within the waveguide core so as to modulate the refractive index thereof such that electromagnetic radiation propagating through the core is converted from a first polarisation state to a second polarisation state; 
characterised in that 
the modulator further comprises at least one grading layer sandwiched between at least one of the first and second cladding layers and the core, the grading layer having an effective refractive index intermediate between that of the waveguide core and the cladding layer.
Patent GB-201021997-D0 (GB)
Title: Signal detection in noise
Filed: 2010-12-24
Abstract: A method of detecting a transmission. The method comprises: measuring, from a first portion of a received spread-spectrum signal, a first code-phase of a spreading-code; measuring, from a second portion of the signal, a second code-phase of the spreading-code; comparing the first and second code-phases; and detecting whether the transmission is present according to the result of the comparison. Also disclosed are corresponding methods and apparatus for transmission and reception of signals.
Patent GB-201109399-D0 (GB)
Title: Applicator with extendable implement
Filed: 2011-06-03
Abstract: An applicator system for applying a product to a surface includes an extendable implement comprising a stem (110) and an applicator (116) including a brush (118) and a tip (120) attached distally to the brush. A cap (122) is securely disposed on the top of the stem (110). A push button (124) is arranged on the top of the cap and is connected by a linkage (128) housed in the stem (110) to the tip (120) and may be actuated to extend the tip (120) relative to the brush (118) to facilitate application of the product. Optionally the system may include a locking mechanism. Preferably the brush comprises a blub shaped unit of bristles overmoulded to a shaft shaped unit of bristles and the tip is stretchably extendible from the brush.
Patent GB-201111116-D0 (GB)
Title: Pallet handling
Filed: 2011-06-29
Abstract: Pallet puller apparatus 801 comprises a rigid hook element 802 for hooking onto a pallet for example at a spacer 114 and a flexible elongate strap element 803 for securing between the rigid hook element 802 and a pulling device such as a fork lift truck, the flexible elongate strap element 803 comprising a first securing element such as a safety hook 806 at a first location and a second securing element such as a ring 808 at a second location, the first and second securing elements releasably engaging to form a portion of the flexible elongate strap element into a loop for securing the flexible elongate strap element 803 to the pulling device. The strap element may 803 include several second securing elements (108, 110 fig. 1) to allow loops of different circumference to be formed. The apparatus may include two rigid hooks (609, 610 fig. 7) secured to two tails of the strap (603 fig. 7). A pulling device mounting element such as a mounting post or a ring (1110 fig. 11) may be secured to a pulling device for releasably engaging with the flexible elongate strap element (1103 fig. 11) of a pallet puller apparatus.
Patent GB-201209599-D0 (GB)
Title: Noise variance estimation and interference detection
Filed: 2012-05-30
Abstract: Noise variance estimation and interference detection is described. In one example, a method of estimating noise variance is described in which the pilots within a received OFDM signal are divided into bands and then a noise variance estimate is calculated on a per-band basis by averaging the noise estimates for those pilots within the band. In some examples, the pilots are divided into bands in frequency and in other examples, the pilots are divided into bands in frequency and time, such that noise estimates from more than one OFDM symbol are used in calculating the per-band noise variance estimates. The noise variance estimate for a pilot is then set to the noise variance estimate for the band which contains the pilot. The noise variance estimate for a data sub-carrier can then be determined by interpolating between the values for the pilots.
Patent GB-201215894-D0 (GB)
Title: Child safety seat
Filed: 2012-09-06
Abstract: A child safety seat includes a seat back and a head rest disposed on the seat back. When a child sits on the child safety seat, his back is against the seat back, and his head is against the head rest. The child safety seat also includes two sliding slot structures, formed on the seat back, and two sliding rods. The two sliding rod are connected to two opposite sides of the head rest corresponding to the two sliding slot structures and slidably disposed in the corresponding sliding slot structures. When the sliding rod is at a first restraining position of the sliding slot structure and the child safety seat shakes because of an impact, the head rest moves relative to the seat back, so that the sliding rod slides to a second restraining position sliding slot structure, which reduces possible harm to the head of the child.
Patent GB-201218643-D0 (GB)
Title: Pre-chamber
Filed: 2009-02-24
Abstract: A pre-chamber is provided. In one embodiment, the pre-chamber is part of a two-stroke combustion engine having a cylinder head with a sparkplug receptacle that has a generally frustoconical shape, and the pre-chamber is coupled to the sparkplug receptacle. The pre-chamber may include a cooling jacket with a generally frustoconical shape and a combustion chamber having an upper zone and a lower zone, which may be narrower than the upper zone.
Patent GB-201307242-D0 (GB)
Title: Tool for deforming threads at a particular location on a fastener
Filed: 2011-08-01
Abstract: Some embodiments pertain to a tool that includes a first arm and a second arm that is rotatably connected to the first arm. The first arm includes an opening and the second arm includes a projection that engages threads on a fastener which is installed within the opening in the first arm. During operation of the tool, a fastener is inserted into the opening in the first arm. Pressure is applied to bring the first and second arms together such that the projection engages the threads of the fastener and then deforms the threads. The first arm may include a plurality of threaded openings such that each opening is adapted to receive a different diameter fastener. In addition, the second arm may include a plurality of projections such that each projection is a different size and is aligned relative to one of the openings in the first arm.
Patent IT-BO20020503-D0 (IT)
Inventor: LAMBERTINI MARCO
IPC: E05B63/00
Filed: 2002-07-31
Abstract: A handle (1) for doors or windows comprises: a handle body (2) attachable to a door or window sash (A); an operating handgrip (4) protruding from one side of the handle body (2); drive elements (5) protruding from the opposite side of the handle body (2) and being connectable to operating devices (6, 7) for opening and closing the door or window; the drive elements (5) comprising a slider element (10) connected to kinematic means (8) and constituting the element that drives the operating devices (6, 7), and means (11) for locking the single slider element (10) in the different positions corresponding to the tilt opened and turn opened configurations of the sash; the locking means (11) being mounted on the slider element (10) detachably, that is to say, in such a way that they can be separated. <IMAGE>
Patent IT-CO20000027-D0 (IT)
Inventor: GIACOMINI LUCA
IPC: F16K35/00
Filed: 2000-12-29
Abstract: An improved ball valve (1), in particular for gas systems, includes a tampering indicating seal (25) made by injection molding a synthetic or metal material into cavities (19; 21; 22) formed in the screw-clamping nut assembly (11, 13) and including a cap outer portion (29) which substantially covers the surface of the outer face of the nut (13) and/or extending (29A) on the side surface of the nut (13).
Patent IT-RE20010021-D0 (IT)
Inventor: MAZZANTI VASCO
IPC: C03C8/16
Filed: 2001-03-09
Abstract: Method of glazing ceramic articles, consisting of preparing a glaze compound in liquid suspension, preferably aqueous; feeding the glaze compound in liquid suspension, preferably aqueous, into the forming cavity of a porous mould, for the time required to create a glaze film of desired thickness on the surface of the cavity by absorption of the liquid phase; feeding the slip into the same cavity for the time required to create the wall of the article by absorption of the liquid phase.
Patent IT-RM20010279-D0 (IT)
Inventor: SOLURI ALESSANDRO
IPC: G01T1/202
Filed: 2001-05-23
Abstract: A miniaturised scintigraphic device comprising a collimator (1), internally having a multiplicity of equal conduits (10) of determined length, identified and separated by septa (11) of minimum thickness in relation to the energy of the radiation, terminating in a common end plane (12) on the side opposite to the source of the event to be measured, comprising a scintillation crystal structure (2) and at least a photomultiplier (3), in which the scintillation crystal structure is constituted by a multiplicity of individual crystals (20) with polygonal section, each integrally integrated in proximity to the end, oriented towards the photomultiplier (3), of each conduit (10) of the collimator (1), having conforming polygonal section, and arranged in such a way that all the base faces (21) of the crystals (20) oriented towards the photomultiplier (3) are mutually coplanar and lying on a plane parallel to said common end plane (12) of the collimator (1). <IMAGE>
Patent DE-2966095-D1 (DE)
Title: Dental rontgen-opaque products based on organic synthetics in paste form
Inventor: WALKOWIAK MICHAEL DR
IPC: A61K6/884
Filed: 1979-11-06
Granted: 1983-09-29
Abstract: The invention provides dental materials which are opaque to X-rays and are based on organic plastics in paste form, which comprises (a) a polymerizable binder, (b) a crosslinked bead polymer and (c) an X-ray contrast medium. The materials can also contain as an additional component (d) a fine-particled inorganic filler which is not opaque to X-rays. The materials are useful, inter alia, for filing dental cavities.
Patent DE-3060340-D1 (DE)
Title: Process for the preparation of acetaldehyde
Inventor: GAUTHIER-LAFAYE JEAN
IPC: C07C45/49
Filed: 1980-07-02
Granted: 1982-06-09
Abstract: A process for the carbonylation of methanol to produce acetaldehyde comprising reacting methanol in the presence of hydrogen, cobalt, ruthenium, at least one ionic halide, and at least one alkyl halide, the molar ratio Ru/Co being at most equal to about 2, and the cobalt concentration being at most about 50 milligram atoms per liter of reaction medium.
Patent DE-3169348-D1 (DE)
Title: New substituted 3-phenoxy-1-alkoxycarbonyl-alkylamino-propanol-2-s having beta receptor blocking properties
Inventor: CARLSSON ENAR INGEMAR
IPC: C07C227/14
Filed: 1981-05-27
Granted: 1985-04-25
Abstract: The present invention relates to new compounds of the formula I <IMAGE> (I)  as well as their preparation, pharmaceutical preparations containing same, and method of treating acute myocardial infarction. The compounds which possess beta-adrenoceptor blocking activity are very shortacting and are preferably intended for treatment of acute myocardial infarction by administration by means of injection.
Patent DE-3261566-D1 (DE)
Title: Apparatus for recovery of heat from waste water and method of its operation
Inventor: KALBERER FELIX
IPC: F24D11/02
Filed: 1982-02-04
Granted: 1985-01-31
Abstract: Waste water is led into a container (1) through a inlet (4) at the top. A connection (20) between the inlet (4) and an outlet (21) having a check valve (22) comprises adjacent to the inlet (4) two inverted frusto-conical hollow bodies (24, 25) which are directly connected to each other. The connecting surface between the two hollow bodies (24, 25) is formed as a coarse screen (26). A round fine screen (30), which diverges downwardly, surrounds the hollow bodies (24, 25). Heat exchangers (31) are located in the space between the fine screen (30) and the wall (2) of the container (1). An outlet (5) terminates at the bottom of the container and connects with a riser (6) and via a bend (7) with the sewerage conduit (8). Through the coarse screen (26) the waste water reaches the container, and the heat can reach the heat exchangers (31) through the fine screen (30 ), so that practically uncontaminated water is present at the heat exchangers, and the need for cleansing is substantially diminished.
Patent DE-3263084-D1 (DE)
Title: Method and device for the non destructive determination of the thickness of the iron-tin intermediate layer of electrolytically tinned sheet metal
Inventor: KOPINECK HERMANN JOSEF PROF DR
IPC: G01N23/20
Filed: 1982-05-03
Granted: 1985-05-23
Abstract: 1. Method for the non-destructive determination of the thickness of the iron-tin intermediate layer on electrolytically-tinned sheet steel by means of X-ray or gamma-ray radiation, wherein the radiation issuing from the sheet is measured on the same side of the sheet as the one which is irradiated, characterized in that, in the measurement, an energy is selected for the incident radiation which is higher than 7.111 keV which has a constant magnitude and the measuring is effected at an angle which lies between 6 to 20 degrees for the incident beam and for the beam issuing at the same side of the sheet, wherein the angle lies between the beam and the sheet surface or, with a curved surface, between the tangent and the beam, and moreover the measured values are taken simultaneously in the energydispersive mode from the fluorescence radiation of the iron and from one or more of the other enery regions of the diffracted beam, so that the measured values of the fluorescence radiation are representative of the thickness of the tin layer and the values of the iron-tin intermediate layer are computed from the other measured values with reference to the values for the thickness of the tin layer.
Patent DE-3264532-D1 (DE)
Title: Compounds with gaba-like activity, process for their preparation and pharmaceutical compositions containing them
Inventor: CURTI MARIA
IPC: A61K31/195
Filed: 1982-04-16
Granted: 1985-08-08
Abstract: The present invention relates to compounds of general formula:
 R1OOC-(CH2)2-NH-(CH2)3-COOR2 (I)
 wherein R1 and R2 = H or a lower alkyl, and a process for their preparation, characterized in that it comprises a condensation of a substrate selected from: gamma-amino butyric acid (II) or (GABA), its lactam pyrrolidine-2-one (II) min , or its esters, with a reagent selected from: acrylonitrile, acrylic acid or its esters. 
<??>The invention also relates to pharmaceutical compositions containing said compounds and adapted to provide a GABA-like activity in the brain.
Patent DE-3266657-D1 (DE)
Title: Fireplace with an opening to a furnace
Inventor: AEBERHARD HANS
IPC: F24B7/02
Filed: 1982-06-04
Granted: 1985-11-07
Abstract: 1. Fire place with an open combustion chamber (1), a chimney breeching (9) and a fresh air chamber (28) traversed by an additional gas flue tube system (19, 22a, 22b, 23) which coming from the combustion chamber enters into the fresh air chamber and after having traversed it, discharging into the chimney breeching characterized in that - the gas flue tube system (19, 22a, 22b, 23) traverses meander-shaped the fresh air chamber (28) and that - a closable louver (11) for the opening of the combustion chamber and a hinged cover (13) for the chimney breeching (9) between the combustion chamber and the entrance of the gas flue tube system as well as - means for conducting the combustion air into the combustion chamber (1) bypassing the closable louver are forseen.