baber/WOPTO huggingface dataset:
Patent HU-T67395-A (HU)
Title: Method for the n-cyclopropylation of primary and secondary aromatic amines
Inventor: SOMFAI EVA
IPC: C07C227/08
Filed: 1993-07-13
Abstract: Process for the introduction of a cyclopropyl group into a primary or secondary aromatic amine or into heterocyclic compounds containing a secondary nitrogen atom reacting to the corresponding amines or their salts so as to form the corresponding N-cyclopropyl-(1'-carboxy)-derivatives either with the reagent of general formula (I), optionally in the presence of an acid binding agent or with 2,4-dihalogen-butyric acid ester or with chloroacetic acid ester, whereupon the resulting N-(alkoxy-carbonyl)-methyl-derivative is treated with alkali alkylate and dihalogen-ethane to convert the alkoxy-carbonyl-methyl group into a carbalkoxy-cyclopropyl group and subsequently optionally hydrolysing the ester groups if present and optionally eliminating the 1'-carboxyl group introduced in the course of the first step, whereby the last step is carried out optionally after introducing other substituents into the aromatic ring or after eliminating other substituents from the aromatic group. The method is suitable to synthesize 1-cyclopropyl-7-piperazine-1,4-dihydro-quinolone-3-carboxylic acid derivatives. New biologically active compounds are formed including compounds of formula (IV) and their salts which are used in pharmaceutical and veterinary compositions.
Patent HU-T71487-A (HU)
Title: Substituted benzothiazepine derivatives process for preparing them and pharmaceutical compositions of hypolididaemic activity containing said compounds
Inventor: BRIEADDY LAWRENCE EDWARD
IPC: A61K31/55
Filed: 1993-02-16
Abstract: PCT No. PCT/GB93/00328 Sec. 371 Date Dec. 5, 1994 Sec. 102(e) Date Dec. 5, 1994 PCT Filed Feb. 16, 1993 PCT Pub. No. WO93/16055 PCT Pub. Date Aug. 19, 1993The present invention is directed to the following compounds of formula (I):    <IMAGE>  (I)  wherein l is an integer of from 0 to 4; m is an integer of from 0 to 5; n is an integer of from 0 to 2; R and R' are atoms or groups independently selected from halogen, nitro, phenylalkoxy, C1-4 alkoxy, C1-6 alkyl and -O(CH2)pSO3R'' wherein p is an integer of from 1 to 4 and R'' is hydrogen or C1-6 alkyl, wherein said phenylalkoxy, alkoxy and alkyl groups are optionally substituted by one or more halogen atoms; R4 is a C1-6 straight alkyl group; and R5 is a C2-6 straight alkyl group; and their salts, solvates and physiologically functional derivatives, with processes and novel intermediates for their preparation, with pharmaceutical compositions containing them and with their use in medicine, particularly in the prophylaxis and treatment of hyperlipidaemic conditions, such as atherosclerosis.
Patent HU-T68677-A (HU)
Title: Fluidization fermentor
Inventor: DONNER CHRISTOPH
IPC: C02F3/02
Filed: 1993-05-05
Abstract: PCT No. PCT/DE93/00414 Sec. 371 Date Feb. 3, 1995 Sec. 102(e) Date Feb. 3, 1995 PCT Filed May 5, 1993 PCT Pub. No. WO93/22246 PCT Pub. Date Nov. 11, 1993A fluidized-bed fermenter is described, which is characterized by an inverted cone-shaped fermentation space (1) with two feed pipes (2 and 3) optionally provided with control valves (4 and 5), of which one (2) is vertically aligned to the cone vertex and the second (3) is nonvertically aligned to the shell of the cone in 0.1 to 0.3 times the height of the fermentation space and a sedimentation space (6) above fermentation space (1), which has one or two drainpipes (7 and 8) optionally provided with control valves (9 and 10).
Patent IL-42707-A (IL)
Title: Device for the administration of medicaments by oral inhalation
IPC: A61M15/00
Filed: 1973-07-10
Abstract: 1404338 Administering medicines BEECHAM GROUP Ltd 2 Aug 1973 [4 Aug 1972] 36428/72 Heading A5T A device for the oral inhalation of finely divided solid medicaments comprises a hollow housing and a capsule holder fixed to an elongated vibratable member which is fixed at one end within the housing at a point remote from the capsule holder, the housing having inlet and outlet vents permitting air to flow through the housing, and means causing the member to vibrate, the outlet vents being adapted for application to or insertion into the mouth, and positioned such that the finely divided medicament is carried through the outlet vents at the intake of breath by the user of the device. As shown in Fig. 1, a hollow, generally cylindrical housing 1 has a flat reed 4 mounted on a projection 5 at the end of the housing. A capsule 3, containing finely divided medicament, is held in a holder 2 at the other end of reed 4. In use, the patient inhales at the outlet vents 7, so that air flows in through vents 6 to baffles 8 in the body and baffle 9 on reed 4. The baffles 8, 9 are arranged with a small gap between them, so that turbulence occurs in their vicinity. The reed is vibrated, and powder is shaken out of the capsule, which is pierced for the purpose, before loading or in situ. A constriction 10 is formed near the capsule to provide for low pressure to help disperse the powder. The housing 1 is made in two parts, with screw threads or a snap fastening at X, for placing the capsule in holder 2. Vents 6 may be omitted and air enters by a single vent or opposed vents in the side of the housing, co-operating with the reed or baffles mounted on opposite sides of the reed parallel to the housing walls. Vents 7 may be replaced by a plug drilled with a hole which has a cross-sectional area approximately equal to the area of the annular gap between a side vent and the reed at their greatest separation. In another embodiment, Fig. 6, air enters by tangential vents 406 (see also Fig. 7, not shown), and a vent 406a. A piercing member 421 slides coaxially in housing 401. As the patient inhales through the vent 407, a vortex is formed around holder 402, which rotates orbitally and strikes the inside of housing 401 successive light blows. Air is also drawn through vent 406a, passing partly through passage 417 and through capsule 403, adding to the turbulence. Consequently, powder issues from the capsule in a helical path. Lighter particles are inhaled through the vent 407; heavier particles whirl round in a trough 422 surrounding vent 407 until they are abraded to a size such that they also pass out through vent 407. The vibrating rod may be mounted on a spring-biassed pushbutton, and the capsule impaled on a hollow piercing member of the holder, so that it may be pushed on to a second piercing member by pressing the button. Where the patient is unable to suck sufficiently hard, his efforts may be supplemented by a rubber squeeze bulb.
[GB1404338A]
Patent IL-44046-A (IL)
Title: Process and inhibitor removing bath for direct positive color photographic development
IPC: G03C7/30
Filed: 1974-01-21
Abstract: 1451422 Photographic dye formation inhibitor removing bath MINNESOTA MINING & MFG CO 21 Jan 1974 [22 Jan 1973 28 Dec 1973] 02786/74 Heading G2C A photographic bath comprises (A) a colour accelerating agent (i.e. materials which accelerate colour dye formation in the development of photographic silver halide reversal films) at at least 0.05 moles/litre, (B) a contrast control agent (i.e. materials which control the gradation of the intensity of dye images in colour photographic silver halide processing) at at least 4 x 10<SP>-3</SP> moles/litre and (C) a buffering agent to provide a pH within the bath of 11-13, the bath containing less than 0.05 moles/litre phosphate and less than one half the molar concentration of colour developer required for full colour development i.e. to generate an optical density of 3À0. The bath may contain no colour developer. Component (A) may be ethylene diamine or (3-phenylethyl amine. Component (B) may be citrazinic acid or potassium iodide or bromide. Component (C) may be trisodium phosphate. The bath may also contain (D) a colour reversal agent (i.e. a nucleating or fogging agent) at at least 1À6 x 10<SP>-</SP><SP>3</SP> moles/litre e.g. a borohydride, amine-complexed borane or hydrazine. A colour photographic reversal development process comprises (1) treating a colour photographic element having a hydrophilic colloid silver halide layer bearing a latent image with a bath comprising in aqueous solution of pH 8À5-14 (a) at least 0À02 moles/litre photographic colour developing agent capable, upon oxidation, of reacting with a colour coupler to form a dye and having a polarographic half-wave potential at pH 11À0 of -159 to -305 mV, (b) at least one black and white developing agent having a polarographic half-wave potential at pH 10À0 of -10 to -187 mV and (c) a water-soluble, dye formation inhibitor at at least 0À10 moles/litre present in sufficient quantity so that all dye formation of a silver halide photographic element is restrained in the bath after the element has been exposed to light, the mole ratio of (c) to (a) being a least 0À97, to develop solely a negative black and white silver image therein, (2) fogging and (3) treating with a bath as defined in the previous paragraph to reduce the inhibiting effect of (c). Fogging (2) may be effected by colour reversal agent (d) in bath (3). Specification 1403408 is referred to.
[GB1451422A]
Patent IL-66378-A (IL)
Title: Mixing valve with water modulation sealing means
IPC: F16K11/078
Filed: 1982-07-23
Abstract: A mixing valve utilizes a sleeve having hot and cold water inlet ports and outlet ports therein. A valve member is reciprocal and rotatable within the sleeve to control the temperature and volume of water passing through the outlet ports. There are port seals positioned in the sleeve hot and cold water inlet ports, which port seals are in sealing contact with the valve member and have openings therein through which pass the inlet water flow of the valve. The cold water port seal opening has a cross sectional area less than that of the hot water port seal opening and there is a restricted passage in the cold water port seal controlling the access of water to the cold water port seal opening.
Patent IL-71478-A (IL)
Title: Pyrimidine derivatives,their manufacture and pharmaceutical compositions containing them
IPC: C07D451/14
Filed: 1984-04-09
Abstract: The pyrimidine derivatives of formula I    <IMAGE>  I  wherein R1 is naphthyl, substituted naphthyl or substituted phenyl; R2 is hydrogen or lower alkoxy; and A is an optionally present ethylene or 1,3-propylene, and wherein the diaminopyridine group has the exo-configuration when A is present, are described. These compounds are useful as antibacterial agents, antimalarial agents and antitumor agents, and can be used in combination with sulfonamides in the control of bacterial infections.
Patent IL-74066-A (IL)
Title: 6,6-ethylene-15,16-methylene-3-oxo-17alpha-pregn-4-ene-21,17-carbolactones,processes for the production thereof and pharmaceutical preparations containing them
IPC: C07J53/00
Filed: 1985-01-16
Abstract: 6,6-ethylene-15,16-methylene-3-oxo-17 alpha -pregn-4-ene-21,17 alpha -carbolactones of general Formula I    <IMAGE>  (I)  wherein <IMAGE>   is a CC-single of CC-double bond, R1 is a hydrogen atom or a methyl group, R2 is a methyl or ethyl group, and   <IMAGE> exhibit strong gestagen potency and an aldosterone-antagonistic activity.
Patent IL-94326-A (IL)
Title: Pyranyl cyanoguanidine derivatives and pharmaceutical compositions containing the same
IPC: C07D311/70
Filed: 1990-05-08
Abstract: Novel compounds having the formula <CHEM>  wherein <CHEM> are disclosed. These compounds have potassium channel activating activity and are useful, for example, as cardiovascular agents, especially as antiischemic agents.
Patent IL-95185-A (IL)
Title: Lighting device
IPC: H05B/
Filed: 1990-07-25
Abstract: A novel lighting device comprises an argon lamp (AL) and a power source (AC). The argon lamp (AL) is connected to an output terminal of the power source (AC) and the power source (AC) is capable of supplying to the argon lamp (AL) a voltage exceeding the rating of the argon lamp (AL). The argon lamp (AL) emits a natural light when lighted by being energized by a voltage exceeding the rating. Such a light has superior color rendering properties, as well as a color temperature of about 2,900K or higher which is very close to that of early morning sunlight. Thus, the lighting device is advantageously used in the luminares in general.
Patent JP-S58130125-A (JP)
Title: Formation of glass plate
Inventor: MIWA MASAYUKI
IPC: C03B23/023
Filed: 1982-01-27
Abstract: PURPOSE:To obtain glass plate moldings of intricate shapes with good productivity by bending a glass plate shapely along the curved line parts thereof, butting the end parts where notched parts face each other to each other, and melt sticking and joining parts to each other by heating. CONSTITUTION:Notched parts B are provided in the corner parts of a glass plate 1 and are cut in such a way that such shapes as parts A where the 3 or 4 sides of a glass plate molding are bent shaprly. The plate 1 cut to prescribed sizes and shapes is put into a heating furnace and is heated. Thereafter, the desired curved line S, S1, S2 parts of the plate 1 are heated locally to the softening point temp. or above of the glass plate and are bent sharply to butt the end parts C, D of the glass plate where the notched parts B in the upper part face each other are butted to each other, whereby a preliminarly glass plate molding for the purpose of obtaining the glass plate molding is manufactured. The parts where the end parts C, D of the preliminarly glass molding are butted are heated locally to the softening point temp. or above of the glass plate and the butted end parts C, D of the glass plate are joined to each other by melt sticking, whereby the final shape is obtained.
Patent JP-H06117645-A (JP)
Title: Combustion device
Inventor: TANI HIDEKI
IPC: A47J37/06
Filed: 1993-01-25
Abstract: PURPOSE:To burn smoke generated in a combustion device and enable non- smoke and non-odor state to be made without increasing a size of an entire combustion device. CONSTITUTION:A main body 1 of a combustion device is provided with a door 7 at its front opening which can be opened or closed and the main body 1 is further provided with a combustion housing 2 including a heating source 8 for cooking operation the same. A smoke discharging passage 3 is guided out of a rear upper part of the combustion housing 2. A bottom plate 3c is projected from a horizontal part of the smoke discharging passage 3 into the combustion housing 2. A part between a projecting part 3c-1 of the bottom plate 3c and the heating source 4 arranged above the projecting portion 3c-1 with a certain clearance being left in the same is formed as a projected discharging passage 5 formed at a front end of the smoke discharging passage 3.
Patent JP-H03214481-A (JP)
Title: Head arm locking device for disk device
Inventor: MIIKE MASAMI
IPC: G11B21/22
Filed: 1990-01-19
Abstract: PURPOSE:To improve assembling workability and reliability for connection by inserting a connector at the tip of a flexible printed board drawn out from a circuit board to the terminal of the coil of an electromagnetic means after the electromagnetic means is assembled. CONSTITUTION:The connector 32 is mounted at the tip 31a of the flexible printed board 31 drawn out from a prescribed circuit board 41 mounted at the inside or outside of a chassis in advance. After the electromagnetic means 15 is assembled in the tip of a mounting plate 10, the connector 32 at the tip 31a of the board 31 is inserted to the pair of terminals 44 of a pair of coils 14. Thereby, a part between both terminals 44 and the board 41 can be connected electrically with the board 31 and the connector 32. The board 31 and the connector 32 are separated sufficiently to a position not disturbing the assembling work of the electromagnetic means 15 while it is being performed, and the connector 32 is inserted to the terminals 44, therefore, no disturbance for the work occurs, which improves the assembling workability.
Patent JP-H07215392-A (JP)
Title: Storage bag
Inventor: ABE HIDEMI
IPC: B65D30/10
Filed: 1994-02-01
Abstract: PURPOSE:To move a flexible storage bag to the place of storage or usage by directly loading on and unloading from a container by a lifting device without using any pallet. CONSTITUTION:A flexible storage bag 1 is provided at its lower or side part with a plurality of recess parts 4 for receiving the prongs 12 of a lifting device 10. The storage bag 1 is also provided with a plurality of hanging straps at the side part and the hanging straps are engaged with a part of a raising and lowering part 11 of the lifting device 10.
Patent JP-S63178653-A (JP)
Title: Howler tone sending system
Inventor: YOSHINO HARUYUKI
IPC: H04M19/02
Filed: 1987-01-20
Abstract: PURPOSE:To eliminate the need for a large sized howler tone source device by preparing a general-purpose digital signal source behind a digital network and sending a howler tone in a route of a PCM highway, a standby subscriber circuit and a voice amplifier so as to attain the transmission of howler tone suitable for the accommodation of a few subscribers. CONSTITUTION:A digital signal from a digitized howler tone source device 27 is inputted to a main body section 21 in a standby subscriber circuit 20 via a PCM highway 26, converted into an analog signal by a PCM-CODEC in the section 21 and inputted to an input terminal 29 of a voice amplifier 28 via a feeding circuit and a switch 23. The howler tone is sent to a subscriber terminal device 1 via a switch 5 in a subscriber circuit 3 from an output terminal 30 of the amplifier 28. In this case, switches 7, 6 in the circuit 3 are kept cut off. When off state of a handset takes over in the device 1 in this way, a disconnection switch 7 is cut off at first and the digitized howler tone (from a normal large sized howler tone source device) is inputted to an access line 8 in terms of a signal of the same level as that of a conventional system through the said route.
Patent JP-2000209941-A (JP)
Title: Soil blasting ground material and soil blasting method using the ground material
Inventor: TANNO KATSUJI
IPC: E02D17/20
Filed: 1999-01-19
Abstract: PROBLEM TO BE SOLVED: To provide a soil blasting ground material and soil blasting method enabling the adjustment of the blasting amount of three kinds of materials comprising a grounding material, water and a binder through a nozzle of a blasting machine without stirring with water and the binder and the blasting of these materials at the same time while preventing the blasted soil from sagging and flowing even by applying the ground material to a thickness of about 3-5 cm and enabling easy application of the soil by mixing 45% high- quality soil and 45% fertile soil as a soil blasting ground material (ecological material) and mixing 10% dried grass into the mixture. SOLUTION: This soil blasting ground material 2 and the soil blasting method using the material comprise the mixing of sludge, dried grass, charcoal, powdered oyster shell, chicken manure, rice bran and cut root of tree, the fermentation of the mixture in a short time using a fermenting agent, the mixing of 45% fertile soil produced by the above method with 45% high-quality soil, 10% dried grass having a length of 1-3 cm as a binder and plant seeds and the application of the produced soil blasting ground material to a thickness sufficient for the growth of a plant by a single blasting work.
Patent JP-S58130112-A (JP)
Title: Manufacture of silicon carbide
Inventor: OOSAKI YOSHIHIKO
IPC: C01B31/36
Filed: 1982-01-25
Abstract: PURPOSE:To increase the space factor of starting materials and a heat insulating effect and to relieve the thermal loads of a coil frame and a stand in the manufacture of SiC by induction heating, by charging the starting materials into the inside and outside of an electrically conductive tube. CONSTITUTION:An electrically conductive cylindrical crucible 12 to be placed in a coil frame 15 holding a buried induction heating coil 14 is made small to leave a space B between the crusible 12 and a heat insulator 13. Starting materials 11 are filled into the space A and the crucible 12, and by induction-heating the crucible 12, SiC is manufactured. Thus, the space factor of starting materials is increased, and since the starting materials 11 show a heat insulating effect, the thickness of the heat insulator 13 can be reduced.
Patent JP-S58127314-A (JP)
Inventor: OONISHI AKITERU
IPC: H01G4/12
Filed: 1982-01-25
Abstract: (57)【要約】本公報は電子出願前の出願データであるた め要約のデータは記録されません。
Patent JP-H09203588-A (JP)
Title: Comminuting and sucking conveyor for deposit
Inventor: TAKAGI ATSUSHI
IPC: C21D1/00
Filed: 1996-01-25
Abstract: PROBLEM TO BE SOLVED: To attempt to improve the operating efficiency by comminuting and delivering scale and the like by one unit, and making it possible to all suck and deliver the scale and the like of the comminuting range while comminuting it. SOLUTION: A duct 2 connected to a vacuum sucking unit is elevationally tiltably mounted at a moving vehicle 1, and tilted by an air cylinder 3. A hood 5 is mounted at the suction port of the duct 2, and a spiral blade 6 to be rotatably driven by an air motor 7 is supported to a shaft in the hood. The blade 6 has a spiral blade for right-hand threads and a spiral blade for left-hand threads via the suction port, has comminuting pawls in the spiral direction, and moves the excavated scale to the central suction port to suck and convey it while excavating the scale layer by the rotation.
Patent JP-S61171902-A (JP)
Title: Hydraulic control circuit of multiple actuator
Inventor: HIDAKA YUKIO
IPC: B66D1/44
Filed: 1985-01-22
Abstract: PURPOSE:To improve work efficiency and operability by providing a pilot control circuit with a pilot controlled directional control valve which is switched by the secondary pressure of a remote-controlled valve and adapted to selectively connect a flow control portion of a variable pump to a tank or a select valve. CONSTITUTION:A pilot control circuit is provided with a select valve 16 for selectively connecting an intermediate circuit to a hydraulic pump 13 or a tank 9 and a pilot controlled directional control valve 20 for selectively connecting a flow control portion 1a of a variable pump 1 to the tank 9 or the select valve 16. A pilot portion of the pilot controlled directional control valve 20 is connected to secondary side circuits 10a, 10b, 11a, 11b of remote-controlled valves 10, 11 through shuttle valves 21, 22, 23. In this arrangement, just a little operation for one of the remote-controlled valves 10, 11 will increase the discharge flow of the variable pump 1 to the maximum, so that work efficiency can be improved. The respective actuators can be controlled independently to improve the operability.
Patent JP-S61168602-A (JP)
Title: Curing by polymerization with laser irradiation
Inventor: KUMAZAKI MAMORU
IPC: C08F2/46
Filed: 1985-01-22
Abstract: PURPOSE:To decrease a required energy dose, by adding a substance which can selectively absorb light in the infrared region in heat-curing a composition containing an active double bond-containing polymerizable compound and a polymerization initiator by irradiation with laser beam. CONSTITUTION:A polymerizable compound having at least one double bond (e.g., methyl acrylate or 2-hydroxyethyl acrylate) is mixed with a polymerization initiator (e.g., benzoyl peroxide or azobisisobutyronitrile) and a substance which can selectively absorb light in the infrared region and has a high transmittance to light in the visible region (e.g., fine powder of an IR absorption filter glass comprising a phosphate salt). The resulting polymerizable composition is heat- cured in good energy efficiency by irradiation with laser beam. This process can be used suitably in curing a filling material for restoring carious teeth.
Patent JP-S61170378-A (JP)
Inventor: SUZUKI MAMORU
IPC: A24F13/14
Filed: 1985-01-25
Abstract: (57)【要約】本公報は電子出願前の出願データであるた め要約のデータは記録されません。