baber/WOPTO huggingface dataset:
Patent EA-001880-B1 (EA)
Title: Insect-repellent formulations
Inventor: SCHULZ DARREN JOHN
IPC: C07D209/52
Filed: 1997-09-09
Abstract: 1. An insect- or acarid-repellent formulation comprising a compound of formula I   wherein R represents straight or branched chain C2-10 alkyl, straight or branched chain C2-10 alkenyl, or straight or branched chain C2-10 alkynyl, which groups are optionally substituted by one or more groups selected from halogen, C4-8 cycloalkyl and C4-8 cycloalkenyl; and a suitable adjuvant, diluent or carrier. 2. A formulation as claimed in claim 1, wherein R represents straight chain C2-10 alkenyl. 3. A formulation as claimed in claim 2, wherein R represents 6-hepten-1-yl. 4. A formulation as claimed in claim 1, wherein R represents straight chain C2-10 alkyl, optionally substituted by chlorine. 5. A formulation as claimed in claim 1, wherein R comprises a C4-6 cycloalkyl group. 6. A formulation as claimed in any one of the preceding claims, which is a cream or a lotion. 7. A compound of formula I, as defined in claim 1, with the proviso that R does not represent n-butyl or n-octyl. 8. A method of repelling insects or acarids, which comprises applying a compound of formula I, as defined in claim 1, to the exterior of a mammal. 9. The method as claimed in claim 8, wherein the mammal is a human, a companion animal or a livestock animal. 10. The method as claimed in claim 8 or claim 9, wherein the insects are mosquitoes, gnats or midges. 11. The method as claimed in claim 8 or claim 9, wherein the acarids are ticks. 12. A process for the production of a compound of formula I, as defined in claim 7, which comprises: reacting the compound of formula II   with a compound of formula RX, wherein R is as defined in claim 1, and X is halogen, in the presence of a base. 13. A process for the production of a compound of formula I, as defined in claim 7, which comprises: reacting the compound of formula III   with a compound of formula RNH2, wherein R is as defined in claim 1. 14. A process for the production of a compound of formula I, as defined in claim 7, which comprises: reacting the compound of formula II   with diethyl azodicarboxylate, triphenylphosphine and a compound of formula ROH, wherein R is as defined above, in a Mitsunobu reaction. 15. A process for the production of a compound of formula I, as defined in claim 7, which comprises: reacting the compound of formula IV   in which R<d> has the same definition as R in claim 1 except that it is substituted by OH or oxo, with diethylaminosulfurtrifluoride to give a corresponding compound of formula I in which each OH or oxo group is replaced with one or two fluorine atoms, respectively. 16. A compound of formula IV, as defined in claim 15.
Patent EA-006154-B1 (EA)
Title: N-phenpropylcyclopentyl-substituted glutaramide derivatives as nep inhibitors for fsad
Inventor: CHALLENGER STEPHEN
IPC: C07D317/62
Filed: 2002-03-18
Abstract: The invention relates to compounds of formula (I) for treating for example sexual dysfunction, wherein R<1> is optionally substituted C1-6alkyl, optionally substituted carbocyclyl, optionally substituted heterocyclyl, hydrogen, C1-6alkoxy, -NR2R<3> or -NR<4>SO2R<5>; X is the linkage -(CH2)n- or -(CH2)q-O- (wherein Y is attached to the oxygen); wherein one or more hydrogen atoms in linkage X may be replaced independently by C1-4alkoxy; hydroxy; hydroxy(C1-3alkyl); C3-7cycloalkyl; carbocyclyl; heterocyclyl; or by C1-4alkyl optionally substituted by one or more fluoro or phenyl groups; n is 3, 4, 5, 6, or 7; and q is 2, 3, 4, 5 or 6; and Y is phenyl or pyridyl, each of which may be substituted; or two R<8> groups on adjacent carbon atoms together with the interconnecting carbon atoms may form a fused optionally substituted 5- or 6-membered carbocyclic or heterocyclic ring.
Patent EA-007024-B1 (EA)
Title: Multistorey apartment building with floor parking places
Inventor: PRUS IGOR VLADIMIROVICH
IPC: E04H14/00
Filed: 2005-03-09
Abstract: A structure of a multistorey apartment building, comprising one central and two extreme butt-adjacent to it at least on a part of a blank wall surface multistorey blocks, longitudinal and/or transverse axes of which, not necessarily, coincide, in which each of the extreme blocks is executed with a possibility of placement in it on each floor of apartments, kand k, correspondingly, and is supplied with at least one people transportation facility connected with each floor, a central block is executed with a possibility of placement of N parking places, where N=α(k+k) provided α1, the central block being executed open, at least, on a part of the sides, non-adjacent to the side blocks and is supplied with connected with each floor at least one selected floor vehicle entry facility, at least one selected floor vehicle exit facility, and at least one people transportation facility, each of the side blocks on each of the floors being supplied with at least one coupler with the central block, executed as a door system, the blocks having equal number of storeys, is claimed.In a preferable variant of implementation, at least one side block has a L-shaped form, the central block being executed adjacent with the side block of L-shaped form on the L-shaped form surface.
Patent EA-008193-B1 (EA)
Title: Method of manufacturing glimepiride and the respective intermediate
Inventor: RADL STANISLAV
IPC: C07C211/35
Filed: 2004-02-20
Abstract: A method of manufacturing glimepiride of formula Iwherein trans-4-methylcyclohexylamine pivalate of formula VIIis reacted, either directly or after conversion to trans-4-methylcyclohexylamine or to its another salt, with an alkyl [4-(2-{[(3-ethyl-4-methyl-2-oxo-2,5-dihydro-lH-pyrrol-l yl)carbonyl]amino)ethyl)phenyl]-sulfonyl carbamate of general formula IVwherein R is a Calkyl, giving glimepiride of formula I.trans-4-Methylcyclohexylamine pivalate of formula VII.
Patent EA-009107-B1 (EA)
Title: Recovery of metal values from cermet
Inventor: HALPIN PETER T
IPC: C22B11/02
Filed: 2004-03-12
Abstract: Cermet material obtained from unused inert anodes, used inert anodes and cermet used in the production of inert anodes is beneficiated into a nonferrous metal concentrate composition from which metal values contained in the composition may be readily recovered by using a conventional smelting process. The invention also relates to the use of the composition in a smelting process for the recovery of metal values from the cermet composition of the invention.
Patent EA-013321-B1 (EA)
Title: Bio-herbicidal composition and use thereof
Inventor: AUTKO ALEXANDER ALEXANDROVICH
IPC: A01N43/22
Filed: 2006-08-02
Abstract: The invention relates to the agriculture, namely to a bio-herbicidal composition and method of its application for the weed control in plant cultivation. The task of the present invention is a bio-herbicidal composition for increasing the agrochemical herbicide efficiency and thus decreasing their rate of application using highly effective bioactive compounds – brassinosteroids (BS). The problem is solved by a bio-herbicidal composition containing a herbicide and brassinosteroids as bioactive constituent having the following structure (I-III):I Brassinolide, R = α-Me (BR)II Epibrassinolide, R = β-Me (EBR)III Homobrassinolide, R = α-Et (HBR)with the mass component ratio 400000-800000 : 1-10 (BS mass is 1,25×10-2,25×10%).
Patent EA-014334-B1 (EA)
Title: Device for authentification of articles
Inventor: MILLINGTON ROGER BRADLEY
IPC: B42D15/00
Filed: 2005-06-06
Abstract: A holographic or diffraction device responsive to interrogation, the device comprising an image-former and an image-concealer; wherein the image-former is adapted such that light reflected from or transmitted through it forms at least one image; wherein the image-concealer acts to attenuate the image; and wherein the attenuation of the image by the image-concealer is alterable responsive to interrogation.
Patent EA-011591-B1 (EA)
Title: Method of assaying a hydrocarbon-containing feedstock
Inventor: VOELKENING JOACHIM
IPC: G01N33/28
Filed: 2005-09-15
Abstract: Disclosed herein is a method of assaying a crude oil, the method includes measuring at least two selected properties of the crude oil with one or more laboratory-independent devices using at least two different techniques wherein each technique is predictive of each respective property, transmitting the measured properties to a processor capable of reconstructing a determinative assay of the crude oil from the measured properties, and reconstructing a determinative assay of the crude oil from the measured properties. The disclosed method provides real-time information of a refinery feedstock such that, for example, a trader negotiating the sale of the product has accurate assay information on which to determine whether to sell or purchase the product.
Patent EA-011110-B1 (EA)
Title: Method for producing metal by molten salt electrolysis and method for producing metal titanium
Inventor: YAMAGUCHI MASANORI
IPC: C25C3/28
Filed: 2005-10-05
Abstract: Disclosed is a method for producing a metal by molten salt electrolysis wherein metal production is performed while filling an electrolysis vessel having an anode and a cathode with a molten salt containing a metal chloride. This method is characterized by using such a molten salt which decreases the solubility of the metal in the molten salt.
Patent EA-012788-B1 (EA)
Title: Method of recycling fibers from sewage sludge and means thereof
Inventor: AHARON REFAEL
IPC: D21C5/02
Filed: 2006-03-09
Abstract: The present invention generally relates to a method of recycling and producing fibers from sewage sludge, such as streams of municipal, agricultural and industrial flowing wastes to be further processed. The present invention also relates to industrial means adapted for recycling the same. The present invention discloses environmentally friendly processes and means for recovering valuable fibers and especially cellulose fibers and the like from agricultural and/or urban sewage sludge, waste and/or industrial effluents to decrease its volume especially BOD and TSS, obtaining valuable raw materials and decreasing environmental damages
Patent EA-014118-B1 (EA)
Title: Method and equipment relating to input of data into equipment for performing animal-related operation
Inventor: AXELLSON LARS-ARNE
IPC: A01K11/00
Filed: 2007-12-18
Abstract: The present invention provides a manual input arrangement, whereby on the entry of an initial piece of data, the apparatus will suggest one or more possible animal identification numbers. As a further data input is made, the suggestions made by the apparatus are refined.
Patent EA-014032-B1 (EA)
Title: Tightening means for anti-skid devices and traction enhancement devices
Inventor: BOZKURT EMRAH
IPC: B60C27/10
Filed: 2006-11-17
Abstract: A tightening system (135) for use with anti-skid and traction enhancement devices for wheeled vehicles comprising a sealed tightening mechanism (130) which can clutch and ratchet the rotational movement applied by the user on a knob (212). The system further comprises at least one connection assembly (134) which is adapted to be pivotably and releasably attached to a proximal end of a surface contact member (63; 71) and which is adapted to be connected to the tightening mechanism. The tightening mechanism comprises a locking component (193) which has a base plate (240), an inner sidewall (195) and an outer sidewall (194) standing perpendicular to said base plate (240). The inner sidewall recessed portion has a plurality of recesses (230; 231) which are adapted to engage with a peripheral projection of the upper clutch (206) for holding the knob in place during locked and unlocked positions of the knob. The outer sidewall enters fully or partly, respectively in locked and unlocked positions of the knob, into a corresponding slot (210) of said knob (212) for sealing inner volume of the tightening mechanism from outside conditions.
Patent EA-013771-B1 (EA)
Title: Control valve with profiled packing element
Inventor: BEREZNAI JOZSEF
IPC: F16K47/10
Filed: 2007-03-12
Abstract: Control valve with profiled packing element for making bidirectional flow-through with asymmetric intensity possible in a flow area, the packing element (1) has a first surface (3) which can be abutted against a second surface (4) formed within the valve housing (2), said packing element (1) has a first position in which said first surface (3) and said second surface (4) abut against one another, and a second position in which said first surface (3) and said second surface (4) are distant from one another; characterized in that at least one of the surfaces from said first surface (3) of said packing element (1) and said second surface (4) within said valve housing (2) is provided with a damage (5) by means of which when said packing element (1) is in its first position a first cross-section of flow is ensured between said abutting first and second surfaces (3, 4), said first cross-section of flow being smaller than a second cross-section of flow ensured by said packing element (1) when it is in its second position, and one of said first (3) and second surfaces (4) is a hard surface formed from metal, plastic or ceramic material, the other is formed from plastic, rubber or other elastic material, where the compressed elastic material is narrowing down said damage (5) due to a pressure difference on the two sides of the packing element (1) in its first position.
Patent EA-014744-B1 (EA)
Title: Electrolysis cell for production of aluminium
Inventor: OVSTETIN FRANK
IPC: C25C3/06
Filed: 2007-09-12
Abstract: An electrolysis cell and a method for operating thereof comprising horizontal cathode (4) of an electronic conducting material and further have current leads such as horizontal collector bars embedded therein. The cell further comprises a bus bar system. The cell can be operated by improved distribution of electrical current, while said cathode comprises at least one substantial vertical electrical current outlet (6).
Patent EA-016171-B1 (EA)
Title: Agricultural machine having dedicated multi-section fan unit
Inventor: VANDIKE NATHAN R
IPC: A01D41/12
Filed: 2009-07-01
Abstract: A fan unit for an agricultural machine includes a fan housing configured to define a plurality of fan chambers. Each fan chamber of the plurality of fan chambers has a respective air inlet port and a respective air outlet port. A shaft is rotatably mounted to the fan housing. The shaft has an axis of rotation that intersects the plurality of fan chambers. A plurality of fans is attached to the shaft for rotation with the shaft. Each fan of the plurality of fans is located in a separate respective fan chamber of the plurality of fan chambers.
Patent EA-016900-B1 (EA)
Title: System and method (variants) of cleaning river, lake, sea and ocean water areas from accumulation of solid man-made wastes being uncapable of natural decomposition
Inventor: PRUS IGOR VLADIMIROVICH
IPC: B09B3/00
Filed: 2009-11-11
Abstract: The claimed invention relates to solid wastes disposal into useful and/or safe products. A system of the river, lake, sea, ocean water areas cleaning from accumulation of the solid man-made wastes being incapable of natural decomposition comprises at least one waste collection device, placed in the waste accumulation area and at least one service craft, whereon the sequentially interconnected means of storing and preprocessing of wastes, a unit of waste disposal by thermolysis, comprising at least one thermolysis reactor, at least one single-stage thermolysis products purification means and the thermolysis products storing and offloading means, comprising a liquid product dispensing device and the thermolysis solid inert residue offloading means, are placed, the waste collection device being configured to interact with the means of storing and preprocessing of wastes of the service crafts. The system and variants of the method provide for environmentally sound, efficient and cost-effective utilization in continuously cyclic operation of the waste accumulation in the water area regardless of the accumulation scopes and their remoteness from the coast.
Patent EA-017286-B1 (EA)
Title: Gamma-secretase inhibitors
Inventor: MILLER MELINDA JOY HOPE
IPC: A61K31/55
Filed: 2008-08-04
Abstract: Compounds of formula (I)pharmaceutical compositions comprising them, and methods for their use are described.
Patent EA-018242-B1 (EA)
Title: Methods of treating a wellbore and method and system for breaking a filtercake formed on a surface of a wellbore
Inventor: BALLARD DAVID ANTONY
IPC: E21B21/00
Filed: 2009-03-06
Abstract: A method of treating a wellbore including emplacing at least one electrolytic tool in a desired section of the wellbore, applying an electric charge to wellbore fluids present in the desired section of the wellbore, and generating oxidants in situ by electrolyzing components of the wellbore fluids. A method of breaking a filtercake formed in a wellbore, comprising: generating oxidants in situ by electrolyzing components of a wellbore fluid present in the wellbore; and allowing the oxidants to degrade filtercake components. A system for breaking a filtercake formed on a surface of a wellbore, comprising: a wellbore having a filtercake formed thereon; a fluid supply source for supplying an aqueous solution into the wellbore; and at least one electrolytic tool for generating oxidants in the wellbore.
Patent EA-018540-B1 (EA)
Title: Method of shaft sinking in mellow soils that occur from the land surface
Inventor: SMYCHNIK ANATOLIJ DANILOVICH
IPC: E21D1/16
Filed: 2011-03-29
Abstract: This invention relates to the mining industry and it can be applied, in particular, to construction of sealing curtains for vertical shaft sinking and open-pit mine development. This invention is aimed at improvement of shaft sinking in mellow soils by applying backfilling method and reducing slurry losses. The aim of this invention is achieved by mine shaft backfilling through main grouting holes arranged along the contour of the shaft. Furthermore, backfilling is applied to construction of a solid horizontally-mounted sealing curtain of a variable thickness by using a network of reliever holes. The thickness of the curtain is determined from the formula, depending on the distance to the nearest grout injection hole. An additional hydraulic hole is drilled in the middle of the shaft contour to ensure hydraulic liquid backing during backfilling of the main grout holes. The backfilling contributes to replacement of slurry to the area of a vertical sealing curtain construction. It also reduces slurry losses, prevents heavy cementation (hardening) of mellow soils within the mine shaft contour, facilitates mining and reduces the time of sinking operations.
Patent EA-022107-B1 (EA)
Title: Method for recovering oil using elastic vibration energy and assembly therefor
Inventor: ABRAMOVA ANNA VLADIMIROVNA
IPC: E21B43/25
Filed: 2010-04-16
Abstract: The invention relates to the field of oil recovery and, more specifically, to the recovery of oil using elastic vibration energy. The method for recovering oil using elastic vibration energy involves placing a downhole apparatus in a well, which downhole apparatus is connected to aboveground power supply units and contains an ultrasonic transducer that provides for the generation of high frequency elastic vibrations, exciting elastic vibrations of different frequencies and then repeatedly applying the elastic vibrations to the oil formation, wherein both high and low frequency vibrations are applied to the formation. The low frequency vibrations are generated with the aid of an electric pulse device which is connected to an aboveground power supply and comprises the following electrically interconnected components: a charger, a unit of energy storage capacitors, a discharge unit with electrodes, and two switching means. The invention makes it possible to recover oil from depths of over 2000 metres and to act effectively on the formation being treated.
Patent EA-021055-B1 (EA)
Title: Method of enhancing the speed of absorption of tryptans and method for treating the complications or symptoms of migraine
Inventor: POLVINO WILLIAM J
IPC: A61K45/06
Filed: 2010-03-01
Abstract: A method of enhancing the speed of absorption of sumatriptan, rizatriptan, naratriptan, zolmitriptan, eletriptan, almotriptan or frovatriptan, compring administering to the subject having a migraine an effective amount of anamorelin or a pharmaceutically acceptable salt thereof. The invention also relates to a method of treating the complications or symptoms of migraine, wherein said complications or symptoms are selected from gastric stasis, nausea, vomiting, photophobia and phonophobia, comprising administering to a subject suffering from one or more of said complications or symptoms an effective amount of anamorelin or a pharmaceutically acceptable salt thereof and sumatriptan, rizatriptan, naratriptan, zolmitriptan, eletriptan, almotriptan or frovatriptan. The invention provides to enhance the speed of absorption of tryptans.
Patent EA-023838-B1 (EA)
Title: SUBSTITUTED PIPERIDINES THAT INCREASE p53 ACTIVITY AND THE USES THEREOF
Inventor: BOGEN STEPHANE L
IPC: A61K31/445
Filed: 2010-10-05
Abstract: The present invention provides a compound of Formula (1) as described herein or a pharmaceutically acceptable salt thereof. The compounds are useful as inhibitors of the HDM2 protein. Also disclosed are pharmaceutical compositions comprising the above compounds and methods of treating cancer using these compounds.
Patent EA-028975-B1 (EA)
Title: Method for producing a closure for containers and polymer compound for a sealing element of a closure
Inventor: POEL CHRISTIANE
IPC: C08L53/00
Filed: 2009-11-20
Abstract: The invention relates to a polymer compound for a sealing insert for container closures, in particular for fat-containing filling materials, which has a composition such that the migration of constituents of the compound into the filling material is reduced, and also to a method for producing "Press-on Twist-off" caps for containers comprising a sealing element based on the polymer compound. The proposed polymer compound is PVC-free and comprises two different polymers, one of which is a copolymer which comprises polyethylene units and alkene, selected from propene, butene, hexene and, in particular, octene, and the other is a random copolymer, that is composed of a linear or branched interpolymer of ethylene and at least one C-Calpha-olefin. The Shore A hardness of the proposed compound is in the range of 40 to 90. The proposed compound shows a compression set between 30 and 70% in the compressive deformation test according to ASTM after 22 hours at 70°C and a compression of 25%.