baber/WOPTO huggingface dataset:
Patent IL-67275-A0 (IL)
Title: Preparation of 5-(4-trifluoromethylphenoxy)-and 5-(2-halo-4-trifluoromethylphenoxy)-2-nitrobenzoic acid and salts,esters and amides thereof
IPC: C07C255/14
Filed: 1982-11-16
Abstract: Certain trifluoromethyl substituted diphenyl ethers can be prepared three of herbicidally inactive impurities by a process which comprises:
 (A) reacting 
<CHEM>
 to form a compound: 
<CHEM>
 wherein X<1> is halo and R is hydrogen, alkyl, alkenyl, alkynyl, hydroxyalkyl, carboxyalkyl, carbalkoxyalkyl, cyanoalkyl, alkoxyalkyl, haloalkyl, alkali metal cation, alkaline earth metal cation, quaternary ammonium cation, amino or mono-R amino or di-R amino, and/or (B) reacting (I) with a halogenating agent to form a compound: 
<CHEM>
 wherein X is halo and R is as defined above. 
<??>Compounds (III), which are herbicidally active may be converted to other herbicidally active compounds by hydrolysis whereby R becomes alkali metal cation and, further reaction to form the free acid.
Patent IL-69098-A0 (IL)
Title: Gnrh antagonist peptides and pharmaceutical compositions containing them
IPC: C07K7/06
Filed: 1983-06-28
Abstract: Peptides which inhibit the secretion of gonadotropins by the pituitary gland and inhibit the release of steroids by the gonads. Administration of an effective amount prevents ovulation of female mammalian eggs and/or the release of steroids by the gonads. The peptides have the structure: X-β-D-2NAL-R<sub>2</sub>-D-Trp-Ser-R<sub>5</sub>-R<sub>6</sub>-R<sub>7</sub>-Arg-Pro-R wherein X is hydrogen or an acyl group having 7 or less carbon atoms; R<sub>2</sub> is Cl-D-Phe, F-D-Phe, N0<sub>2</sub>-D-Phe, Cl<sub>2</sub>-D-Phe or Br-D-Phe; R<sub>5</sub> is Tyr or Cl-Phe; R<sub>6</sub> is 4-NH<sub>2</sub>-D-Phe or D-Arg; R<sub>7</sub> is Leu or N<sup>α</sup>Me-Leu; and R<sub>10</sub> is Gly-NH<sub>2</sub>, NHCH<sub>2</sub>CH<sub>3</sub> or D-Ala-NH<sub>2</sub>.
Patent IL-78910-A0 (IL)
Title: Anti-cancer quinazoline derivatives
IPC: C07D333/00
Filed: 1986-05-26
Abstract: Quinazoline derivatives of the formula 
<CHEM>
 wherein R is
 1) hydrogen
 or 2) a straight or branched chain saturated or unsaturated hydrocarbon group, or 
 3) a straight or branched chain saturated or unsaturated hydrocarbon group which is substituted by at least one heteroatom, the or each heteroatom being halogeno when R is a C1 hydrocarbon group, by a saturated carbocyclic group or by a group containing at least one heteroatom, the or each heteroatom being O, N or S when R contains a cyclic group;
 n is 0, 1 or 2; Z represents-CH=CH- or -O- or -S-; X or,when n is an integer of at least 2, each X independently, represents a halogeno, C1-C4 alkyl, aryl or aralkyl group or a group including at least one heteroatom and Y represents a group of formula: 
<CHEM>
Patent IL-81230-A0 (IL)
Title: Microplastic structures,their manufacture and photomask suitable for use therein
IPC: H01L21/30
Filed: 1987-01-12
Abstract: Microplastic structures, thermally stable up to at least 200 deg.C are produced by (a) coating a substrate with a photosensitive compsn. contg. 40-99.9 wt.% crosslinkable polymer and 0.1-60 wt.% photoacid generator, (b) exposing the coating through one or more photomasks to light, (c) heating to 70-120 deg.C to crosslink the exposed coating(s), and (d) removing portions of the coating with an aq. base soln. Pref. the microplastic structure is in the positive or negative mode and the coating is exposed to a near UV light source. The compsn. pref. contains (i) 3-50 wt.% aminoplast, 90-40 wt.% of reactive H-contg. cpd. and 2-30 wt.% photoacid generator sensitive to near UV light or (ii) 50-95 wt.% phenoplast, 40-3 wt.% HCHO generating cpd. and 2-30 wt.% photoacid generator sensitive to near UV light, (iii) 95.99.9 wt.% acid-hardening resin, 0.1-5 wt.% photoacid generator sensitive to deep UV light at an exposure dosage of 10Mj/sq.cm.
Patent IL-84425-A0 (IL)
Title: Ibuprofen-containing medicament
IPC: A61K9/00
Filed: 1987-11-10
Abstract: 1. An ibuprofen-containing medicament containing ibuprofen only in the (S)-(+)-form, in the usual carriers and diluents, characterized in that it is in sustained-release form.
Patent IL-96408-A0 (IL)
Title: Homodyne receiver for cable television converter
IPC: H04B1/26
Filed: 1990-11-19
Abstract: A carrier is received containing a plurality of signals within a first frequency band, for example television signals within the cable television band. The signals are upconverted to a second frequency band above the first band wherein a selected one of the upconverted signals will reside at an intermediate frequency within the second band. The selected upconverted signal is input to a homodyne detector operating at or near intermediate frequency. In-phase and quadrature signals output from the homodyne detector are digitally processed to recover a baseband signal. <IMAGE>
Patent IL-98565-A0 (IL)
Title: Benzotriazolesulfonic acid derivatives,their preparation and their use for protecting plants against phytopathogenic microorganisms
IPC: A01N43/647
Filed: 1991-06-19
Abstract: Novel benzotriazolesulphonic acid derivatives of the formula <IMAGE>  in which:   R1 is hydrogen, halogen, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkoxy having at least two identical or different halogen atoms, furthermore CF3, nitro or the group N(R')R'' where R' and R'' independently of one another are C1-C4-alkyl; R2 is phenoxy or phenylthio, each of which is unsubstituted or monosubstituted to trisubstituted by halogen, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkoxy having at least two identical or different halogen atoms, furthermore substituted by cyano, nitro, C2-C4-alkenyl, C2-C4-alkynyl, phenyl, 2-phenylethynyl or a further phenoxy radical which is unsubstituted or substituted by halogen, C1-C4-alkyl and/or C1-C4-alkoxy; or R2 is the radical O-CH2-O; R3 is alkyl, aryl or aralkyl having not more than 14 atoms, these radicals being substituted by halogen, C1-C4-alkyl and/or nitro; including the position isomers of R1 and R2 if these substituents occupy position 5 or 6. The novel active substances have crop-protecting properties and are particularly suitable for protecting plants against attack by phytopathogenic microorganisms such as fungi, in particular Oomycetes.
Patent AU-PP366398-A0 (AU)
Title: Ventilatory assistance for treatment of cardiac failure and cheyne-stokes breathing
IPC: A61B5/087
Filed: 1998-05-22
Abstract: Method and apparatus for the treatment of cardiac failure, Cheyne-Stokes breathing or central sleep apnea are disclosed. A subject is provided with ventilatory support, for example positive pressure ventilatory support using a blower and mask. Respiratory airflow is determined. From the respiratory airflow are derived a measure of instantaneous ventilation (for example half the absolute value of the respiratory airflow) and a measure of longterm average ventilation (for example the instantaneous ventilation low pass filtered with a 100 second time constant). A target ventilation is taken as 95 % of the longterm average ventilation. The instantaneous ventilation is fed as the input signal to a clipped integral controller, with the target ventilation as the reference signal. The output of the controller determines the degree of ventilatory support. Clipping is typically to between half and double the degree of support that would do all the respiratory work. A third measure of ventilation, for example instantaneous ventilation low pass filtered with a time constant of 5 seconds, is calculated. Ventilatory support is in phase with the subject's respiratory airflow to the fuzzy extent that this ventilation is above target, and at a preset rate conversely.
Patent AU-PS300602-A0 (AU)
Title: Methods of minimising the effect of integrity loss in hollow fibre membrane modules
IPC: B01D65/10
Filed: 2002-06-18
Abstract: A method and apparatus for reducing the effect of integrity loss in a hollow fiber membrane module, said module including a plurality of hollow fiber membranes (5), at least one end of the fiber membranes (5) being supported in a pot (6), the method including the step of increasing flow resistance of the liquid through the lumen (8) of the fiber membrane (5) in the region of the pot (6).
Patent FI-20000907-A0 (FI)
Inventor: PITKAENEN VEIJO
IPC: B28B7/02
Filed: 2000-04-17
Abstract: The object of this invention is the method of manufacture of a symmetric element of a round ring and cone-shaped ring applicable in serial production. The application area of the invention is particularly the prefabrication of ceramic coating elements, which match together and which are assembled in straight walls, a surface coating containing cylinder rings and cone-shaped rings. Good application objects are for example the cyclones and the ducts of circulating bed boilers, carburetor plants, etc. various combustion chambers and high temperature devices. The concerned elements have special conditions concerning their tightness, so that their seam surfaces must be shaped so that they are profile surfaces differing from plane surfaces, profile surfaces having the capacity to resist to leakage through seam better than straight surfaces.
Patent FI-20010170-A0 (FI)
Inventor: RUNOLA ESA
IPC: G08B5/36
Filed: 2001-01-29
Abstract: The present invention relates to a system comprising: mobile stations (MS1-MS4), and means for locating the mobile stations. To allow the users of the mobile stations to find a partner, the system further comprises: a database (2) in which information is stored about parameters determined by persons seeking a partner, and monitoring means (3) that monitor the locations of the mobile stations (MS1-MS4) used by the persons seeking a partner and transmit information indicating that a partner corresponding to the parameters has been found, provided that the mobile stations of two persons seeking a partner are located close to each other and that the parameters stored in the database (2) indicate that the persons in question are compatible.
Patent FI-20020950-A0 (FI)
Inventor: MONONEN HEIKKI
IPC: B66C1/22
Filed: 2002-05-21
Abstract: A lifting device for cellulose bales comprising a beam fi-amework (2) to be detacbably fixed in crane (1) as-d its hydraulic system and claw wagons (3) ennnected to the beam framework and furnished with gripping means (4)< >to grasp and move cellulose halos (5). In the lifting apparatus as per the invention the claw wagons include booms (6) fixed movably to the beam framework, to which booms the claw wagon frame (7) is fixed.
Patent FI-20030258-A0 (FI)
Inventor: MAEKI MAARIT
IPC: A23L19/20
Filed: 2003-02-21
Abstract: The present invention relates to fermentation of plant-derived material with a starter comprising a lactic acid bacterium, Lactobacillus sp.96/142 isolated from sauerkraut. Said Lactobacillus strain is likely to belong to the species Lactobacilllus sakei. The lactic acid bacterium of the invention degrades glucosinolates contained in the plant material. The degradation products produced by the bacterium exhibit among other things antimicrobial properties, and may possess a health-promoting effect. The invention further relates to the use of said Lactobacillus strain in the production of exopolysaccharides applicable to improving of food structure.
Patent FI-20110006-A0 (FI)
Inventor: LOMMI JUKKA RAFAEL
IPC: E04B/
Filed: 2011-01-11
Abstract: The present invention concerns a method for joining longitudinal wooden elements (1, 2), cut from board material, to each other one after another and one above another as a construction piece, and a joint of such elements. The invention is characterized in that both ends of elements (1, resp. 2) located one after another in a same layer of a construction piece have one vertical drilling (3, 4) at a first distance from the concerned end, and one end of the element (1, 2) has still another vertical drilling (5) at distance in the elements longitudinal direction from the first vertical drilling (3), being twice as long as the first distance, and in the elements of the next layer the end equipped with two vertical drillings (3, 5) is at the opposite side of the element (2, 1), whereby in the joint the elements (1, 2) of two successive layers fit together such displaced that the outer vertical drilling (3) of the end equipped with two vertical drillings (3, 5) of successive elements (1, 2) is aligned with an outer vertical drilling (3) of an end equipped with two vertical drillings (3, 5) of an element of the other (2, 1) layer, so that at each joint there are three vertical drillings 5, 3, 4; 4, 3, 5) next to each other at an uniform distance from each other, to which vertical drillings (5, 4, 3) wooden pegs (6) extending through the overlapping elements (1,2) are fitted.
Patent IL-103666-A0 (IL)
Title: Zinc borate
IPC: C01B35/12
Filed: 1992-11-06
Abstract: Zinc borate compositions having a ZnO:B2O3 ratio of 4:1. The hydrated zinc borate 4ZnO.B2O3.H2O and anhydrous zinc borate 4ZnO.B2O3 are especially useful as fire-retardants and smoke-suppressant additives for polymeric compositions.
Patent IL-106536-A0 (IL)
Title: An insert for a milling cutter
IPC: C23G5/00
Filed: 1993-08-02
Abstract: A cutting insert (1) for use with a rotary milling cutter tool and having at least one major cutting edge (5) comprising first, second and third successive component cutting edges (5a, 5b, 5c), each second component cutting edge being substantially coextensive with a bore (1a) and being of substantially greater length than the length of each of said first and third component cutting edges (5a, 5c) and defining with respect to said axis of rotation of the cutter tool an axial rake angle which is substantially less positive than the axial rake angles defined respectively by said first and third component cutting edges (5a, 5c) with respect to said axis of rotation. <IMAGE>
Patent IL-106676-A0 (IL)
Title: Novel 7-(substituted)-8-(substituted-9-(substituted glycyl)amido)-6-demethyl-6-deoxytetracyclines
IPC: C07C237/26
Filed: 1993-08-12
Abstract: The invention provides compounds of the formula: <CHEM> wherein R, R<3>, R<4>, X and W are defined in the specification. These compounds are useful as antibiotic agents.
Patent IL-110089-A0 (IL)
Title: Sulphonylaminapyridines, their preparation and pharmaceutical compositions containing them
IPC: C07D417/12
Filed: 1994-06-22
Abstract: Compounds of the formula <IMAGE> in which R<1> to R<9>, R<a>, R<b>, X, Y, Z, m and n have the meaning given in the description, can be used as medicines, in particular for the treatment and prophylaxis of conditions associated with endothelin activities.
Patent IL-113782-A0 (IL)
Title: Compositions containing flubendazole their preparation and their use
IPC: A61K31/41
Filed: 1995-05-18
Abstract: PCT No. PCT/EP95/01801 Sec. 371 Date Oct. 31, 1996 Sec. 102(e) Date Oct. 31, 1996 PCT Filed May 12, 1995 PCT Pub. No. WO95/31963 PCT Pub. Date Nov. 30, 1995The present invention relates to compositions comprising flubendazole of formula (I), which are palatable to companion animals, especially dogs.anthelmintic compositions for the treatment of helminthiasis.
Patent IL-114726-A0 (IL)
Title: Noribogaine derivatives and pharmaceutical compositions containing the same
IPC: C07D487/22
Filed: 1995-07-25
Abstract: An essentially pure noribogaine compound having the formula:wherein R is hydrogen or a hydrolyzable group of the formula:wherein X is an unsubstituted C1-C12 group or a C1-C12 group substituted by lower alkyl or lower alkoxy groups, wherein the noribogaine compound having the hydrolyzable group hydrolyzes in vivo to form 12-hydroxy ibogamine.
Patent IL-115688-A0 (IL)
Title: Preparation of a tetrazole derivative in two crystalline forms and crystalline form of said derivative
IPC: A61K31/415
Filed: 1995-10-19
Abstract: Prepn. of 2-n-butyl-3-((2'-(tetrazol-5-yl)-biphenyl-4-yl)methyl)-1,3-diaza- -spiro(4.4)-non-1-ene-4-one (I) comprises: (a) treating 2-n-butyl-3-((2'-cyanobiphenyl-4-yl)methyl)-1,3-diazaspiro(4.4) non-1-ene-4-one (II) with an alkaline azide and Et3N.HCl in an inert, polar, aprotic solvent and recovering (I) in the form of an alkaline salt in aq. soln; (b) neutralising to pH 4.7-5.3, and (c) crystallising the pptd. prod. (i) in a solvent contg. < 10 vol.% water to obtain (I) in form A (i.e. (IA)) having a specified X-ray diffraction pattern; or (ii) in a solvent miscible with water contg. > 10 vol.% water to isolate (I) in form B (i.e. IB)) which has a different specified X-ray diffraction pattern. Also claimed is the prepn. of (IB) comprising recrystallising (IA) or (I) in a solvent miscible with water contg. ≥ 10% water. (IB) having a specified X-ray diffraction pattern, m.pt. 185-186 degrees C. and IR absorption at 1537,1200 and 745 cm<-1> or obtd. by the above processes is new.
Patent IL-116887-A0 (IL)
Title: Cationic copolymers of vinyl amine and vinyl alcohol for the delivery of oligonucleotides
IPC: A61K31/70
Filed: 1996-01-24
Abstract: The present invention relates to an improved method for the cytoplasmic delivery of oligonucleotides using cationic copolymers based on vinyl alcohol with low levels of vinyl amine (PVAVAMs). Improved compositions for use in such method are also provided.
Patent IL-120517-A0 (IL)
Title: Pyrazole derivatives
IPC: C07D403/12
Filed: 1997-03-25
Abstract: The subject of the invention is pyrazole derivatives of formula I:   <IMAGE>  in which   - g2, g3, g4, g5, g6 and w2, w3, w4, w5 and w6 are identical or different and independently represent hydrogen, a chlorine or bromine atom, a (C1-C3)alkyl, a (C1-C3)alkoxy, a trifluoromethyl or a nitro group and g4 optionally represents a phenyl group;   - R4 represents hydrogen or a (C1-C3)alkyl; - X represents either a direct bond or a group -(CH2)x-N(R3)- in which R3 represents hydrogen or a (C1-C3)alkyl and x represents zero or one;   - R represents   . a group -NR1R2, in which R1 and R2 independently represent a (C1-C6)alkyl group; an optionally substituted, nonaromatic (C3-C15)carbocyclic radical; an amino(C1-C4)alkyl group in which the amino is optionally disubstituted by a (C1-C3)alkyl; a cycloalkyl(C1-C3)alkyl in which the cycloalkyl is (C3-C12); a phenyl which is unsubstituted or substituted one or more times by a halogen, by a (C1-C5)alkyl or by a (C1-C5)alkoxy; a phenyl(C1-C3)alkyl; a diphenyl(C1-C3)alkyl; a naphthyl; an anthryl; a saturated, 5- to 8-membered heterocyclic radical which is unsubstituted or substituted by a (C1-C3)alkyl, hydroxyl or benzyl; a 1-adamantylmethyl; an aromatic heterocycle which is unsubstituted or substituted one or more times by a halogen, a (C1-C5)alkyl or a (C1-C5)alkoxy; a (C1-C3)alkyl which is substituted by an aromatic heterocycle which is unsubstituted or substituted one or more times by a halogen, a (C1-C5)alkyl or a (C1-C5)alkoxy; or else R1 is hydrogen and R2 is as defined above; or yet again R1 and R2 constitute, with the nitrogen atom to which they are bonded, a saturated, 5- to 8-membered heterocyclic radical, the said heterocyclic radical being other than morpholinyl when w2, w3, w4, w5, w6, g2, g3, g4, g5 and g6 are all hydrogen;   . a group R2 as defined above when X represents -(CH2)xN(R3)-; . a group R5 when X represents a direct bond, R5 being represented by a (C1-C3)alkyl; a (C3-C12)cycloalkyl which is unsubstituted or substituted by a (C1-C5)alkyl; a phenyl(C1-C3)alkyl which is unsubstituted or substituted by a halogen or by a (C1-C5)alkyl; a cycloalkyl(C1-C3)alkyl in which the cycloalkyl is C3-C12 and is unsubstituted or substituted by a (C1-C5)alkyl; or a 2-norbornylmethyl;    or one of their optional salts. Application: therapeutic treatment of pathological conditions where cannabis is involved.
Patent IL-123732-A0 (IL)
Title: Method and apparatus for off-hook signaling between telephones
IPC: H04M3/42
Filed: 1996-09-19
Abstract: When two or more telephone sets are in use on the same subscriber's loop, their activities may not be properly detected or monitored by the central office switch. The present invention provides a method of, and an apparatus for, coordinating the signaling activities so that a hook flash or "Link" can work. A telephone set of the invention senses and synchronizes hook flashes of another set on the same loop so that a coordinated hook flash or "LINK" can be properly detected by the office switch.
Patent IL-126422-A0 (IL)
Title: Acidic polylactic polymers
IPC: C08G63/08
Filed: 1997-04-22
Abstract: Methods of preparing biodegradable polyesters containing lactic acid units and/or glycolic acid units and optionally other hydroxy acids are provided, as well as biodegradable polyesters comprising lactic acid units and glycolic acid units and an initiator.
Patent IL-130276-A0 (IL)
Title: Process for the production of sulphonamides
IPC: C07C311/03
Filed: 1997-11-27
Abstract: PCT No. PCT/GB97/03272 Sec. 371 Date May 24, 1999 Sec. 102(e) Date May 24, 1999 PCT Filed Nov. 27, 1997 PCT Pub. No. WO98/25890 PCT Pub. Date Jun. 18, 1998A process for the preparation of a sulfonamide of formula: RSO2NR1R2 wherein R represents C1-C10 alkyl; and R1 and R2 independently represent hydrogen, C1-C10 alkyl or C6-C10 aryl; which comprises reacting the corresponding alkane- or arenesulfonyl halide of formula: RSO2Hal wherein Hal represents halogen; with the corresponding compound of formula: NHR1R2 in an aqueous solvent and extracting the sulfonamide from the resulting mixture into a polar organic solvent.
Patent IL-131797-A0 (IL)
Title: Dry powder inhaler
IPC: A61M16/00
Filed: 1998-03-16
Abstract: A dry powder inhaler has a lid pivotally attached to an inhaler housing. A medicine containing cartridge is attached to the top of the housing and includes a cartridge ring with apertures for holding dry powdered medicine. A slide-groove assembly located on the underside of the lid advances the cartridge ring to a next aperture when a user first opens, then closes the lid. A venturi air passageway assembly is contained within the housing of the dry powdered inhaler. The venturi air passageway assembly includes a tapered inlet section, a throat section, and a tapered outlet section. A pressure switch is advantageously located within the housing for actuating the mixing process within the mixing chamber. During inhalation, the pressure switch contained within the housing actuates the motor driven impeller within the mixing chamber of the inhaler when the pressure within the venturi air passageway reaches a predetermined level. The pressure at which the pressure switch closes corresponds to a specifically calibrated inhalation flow rate.
Patent IL-136603-A0 (IL)
Title: N-benzyl-3-indenylacetamide derivatives for treating neoplasia
IPC: A61P35/00
Filed: 1998-12-11
Abstract: Substituted condensation products of N-benzyl-3-indenylacetamides with heterocyclic aldehydes are useful for inducing or promoting apotosis and for arresting uncontrolled neoplastic cell proliferation, and are specifically useful in the arresting and treatment of neoplasias, including precancerous and cancerous lesions.
Patent IL-139709-A0 (IL)
Title: A method of permanent flourescent assay
IPC: C12Q1/28
Filed: 2000-03-17
Abstract: A method for performing a peroxidase-based assay by reacting a peroxidase enzyme with a soluble organic p-hydroxyphenyl-containing compound having the formula:wherein Q is a linear or branched 1-12 heteroatom alkyl wherein the heteroatoms are selected from C, N, O, and S, wherein the bonds connecting the heteroatom alkyl chain are single or double, wherein any carbon atom in the heteroatom alkyl chain optionally includes a substituent selected from -OH, -COOH, -NH2, and -SH, and wherein R is selected from -OH, -COOH, -NH2, and -CH3; and converting the soluble organic p-hydroxyphenyl-containing compound into a stable insoluble product which becomes highly fluorescent after illumination, upon excitation.