baber/WOPTO huggingface dataset:
Patent IE-40660-L (IE)
Title: 2-deoxy-2-nicotinamido-1-o-nicotinoylglucopyranose¹derivatives
IPC: C07H13/10
Filed: 1975-01-20
Abstract: 1451181 2 - Nicotinamides - 1 - nicotinoyloxy- 0-glycopyranoses F HOFFMAN-LA ROCHE AG 24 Jan 1975 [25 Jan 1974] 3180/75 Heading C2C Novel compounds I in which R is C 1-6 alkanoyl, C 1-6 alkoxy C 1-6 alkanoyl or aryl are prepared by replacing X in a compound II where X is halogen or optionally protected hydroxy, by a nicotinoyloxy group in known manner. Compounds I (R=acetyl, propionyl, benzoyl) are prepared. Compound II (X=Cl, R=acetyl) is prepared by reacting N-nicotinoyl-D-glucosamine with acetyl chloride. Compound II (X=acetoxy, R=acetyl) is prepared by reacting 1,3,4,6- tetra - O - acetyl - D - glucosamine with nicotinic acid. Compounds I have plasma lipid-lowering activity and form with a carrier a pharmaceutical composition which may be administered orally, parenterally or rectally.
[GB1451181A]
Patent IE-900142-L (IE)
Title: Cyclic amine compounds and their use
IPC: C07D521/00
Filed: 1990-01-12
Abstract: A cyclic amine compound of the formula <CHEM> wherein B means a saturated or unsaturated 5- to 7-membered aza-heterocyclic group which may be substituted; A means a bond or an alkylene or alkenylene group which may be substituted by hydrocarbon residues, oxo, hydroxyimino, and/or hydroxy, ___ means either a single bond or a double bond (provided that when A means a bond, ___ means a single bond); R2 and R3 independently mean a hydrogen atom or a hydrocarbon residue which may be substituted (provided that both of R2 and R3 are not hydrogen atoms) or jointly form a cyclic amino group together with the adjacent nitrogen atom, n is 0, 1 or 2 and p is 1 or 2 or a physiologically acceptable salt thereof. The compounds are useful for therapy of cerebral edema, acute symptoms in cerebral apoplexy and protection of brain and nerve cell, or useful as anticholinesterase or as brain function-improving agent.
[EP0378207A1]
Patent IE-890153-L (IE)
Title: Dideoxydidehydrocarbocylic nucleosides
IPC: C07D473/16
Filed: 1989-01-19
Abstract: Disclosed are compounds of formula (see fig. I) wherein X is H, NRR1, SR, OR or halogen; Z is H, OR2 or NRR1; R,R1,R2 are H, C1-4alkyl or aryl and pharmaceutically acceptable derivatives thereof. Also disclosed are use of the compounds as antiviral and anti-tumor agents, pharmaceutical formulations, methods for the preparation of the compounds and intermediates thereto.
[CA1339896C]
Patent IE-880198-L (IE)
Title: Plasminogen activator.
IPC: A61K38/46
Filed: 1988-01-26
Abstract: A fibrinolytically active tissue-type plasminogen activator which has been modified: (a) in the region of the growth factor domain, and (b) to provide an amino acid other than arginine or lysine at position 275. i
[EP0277751A2]
Patent IE-790217-L (IE)
Title: Stoma adaptor
IPC: A61F5/445
Filed: 1979-02-06
Abstract: A stoma adaptor (1) comprising an open tube (2) of non-toxic material, having a proximal end (3) for insertion into the lumen of a body orifice (4) at a stoma site; a distal end at which the rim is turned outwards to form an annular lip (6) having a concave underside (7) geometrically continuous with the rest of the tube whereby an open live intestine advanced over the tube from the proximal end will take up a similarly flared configuration for attachment to the external periphery of the orifice; means for securing an open intestine to the outer surface of the tube; means for securing the tube to the body wall (5); and means for attachment to the tube at the distal end thereof, of a fluid-tight stoma closure.
[EP0003671A1]
Patent IE-840290-L (IE)
Title: Moulding plastics.
IPC: B29C37/00
Filed: 1984-02-08
Abstract: A process is described of coating the interior wall of a mould heated at a temperature of 130 DEG  to 180 DEG  C. with a dry powder of an aminoplast or phenoplast resin, in particular melamine-formaldehyde, having a grain size distribution of 10 to 100 mu , whose particles gel in contact with the walls without running, then introducing into the mould a moulding composition comprising a thermosetting resin, mineral fillers and a catalyst, hardening and polymerizing by heat and pressure the contents of the mould and releasing the article whose coating is solidly anchored in the moulding composition. Sanitary ware articles of polyester-based substrate and melamine-formaldehyde-based coating, and refrigerator boxes consisting of polyurethane foam substrate and melamine-formaldehyde coating can be produced.
Patent IE-780582-L (IE)
Title: PYRIDO [2,1-b] QUINAZOLINES
IPC: C07D213/61
Filed: 1978-03-23
Abstract: The present invention relates to novel chemical compounds. 
[FR2384771A1]
Patent IE-900645-L (IE)
Title: Derivatives of N-phenylbenzamide with anti-ulcer and¹anti-allergy activity and a method for their preparation
IPC: C07C255/60
Filed: 1990-02-22
Abstract: PCT No. PCT/EP90/00270 Sec. 371 Date Aug. 19, 1991 Sec. 102(e) Date Aug. 19, 1991 PCT Filed Feb. 19, 1990 PCT Pub. No. WO90/09989 PCT Pub. Date Sep. 7, 1990.Derivatives of N-phenylbenzamide with general formula (1) in which R1 is a cyano, nitro, halogen, hydrozy, C1-C4 alkyl methyl, methoxy or tetrazol-5-yl group, R2 is hydrogen, hydroxy, or methoxy, R3 is a tetrazol-5-yl group or hydrogen, R4 and R5 are hydrogen if R3 is tetrazolyl but are independently selected from the group consisting of carboxy, methoxycarbonyl, ethoxycarbonyl and carbamoyl if R3 is hydrogen, and R6 is hydrogen or methyl. The derivatives have an anti-ulcer and anti-allergy activity.
Patent IE-36492-L (IE)
Title: Tyre mould
IPC: B29D30/06
Filed: 1971-05-24
Abstract: 1356062 Moulding tyres DUNLOP HOLDINGS Ltd 1 June 1971 [1 June 1970] 18602/71 Heading B5A A tyre mould comprises adjustably spaced mould plates 12, 13 with heating channels 11 between which radially movable tread forming mould segments 14 with heating channels 15 are located. Frusto-conical surfaces on the segments engage corresponding surfaces on a depending member 17 to urge the segments radially inwardly when the mould is closed. The segment heating channels are supplied with heating medium e.g. hot water or steam via flexible hose lines 16 which may be arranged as spirals between adjacent segments. The lower edge of the member 17 may sealingly clamp against the plate 13 providing a sealed mould chamber which may be evacuated and to which a heating medium may be fed. Upstanding spacers between adjacent segments prevent their being clamped between the mould plates.
[GB1356062A]
Patent IE-820782-L (IE)
Title: Scanning an object by means of ultrasonic radiation
IPC: G10K11/20
Filed: 1982-04-02
Abstract: A scanner for periodically scanning an object to be examined with a beam of ultrasonic radiation. A transducer mounted within a housing emits a beam of ultrasonic radiation. The beam is guided and deflected respectively to a continuously rotating scanning reflector which is disposed opposite a stationary object reflector, from which the beam is directed to the object. The beam propagation path further includes a first focussing member adapted to focus the beam to a focal point within the housing, and a second focussing member adapted to focus the beam to a focal point within the object. In a preferred embodiment the first focussing member can be selectively adjusted. Thereby the focal area of the beam in the object can be conveniently shifted.
Patent IE-35481-L (IE)
Title: Dentrifrice package
IPC: B65D35/08
Filed: 1971-07-29
Abstract: 1342755 Packaging toothpaste COLGATEPALMOLIVE CO 27 July 1971 [5 Aug 1970] 35143/71 Heading B8C Toothpaste, comprising a homogeneous paste or gel which is clear or includes particles, speckles, stripes or bubbles, is packaged in a clear thermoplastics squeezable tube. The tube may be of polythene coated with an epoxide or polyvinylidene chloride, or of unplasticized polyvinyl chloride co-polymerized with 3-8% by weight of polypropylene. Again, the tube may be of a nitrile-rubber modified acrylonitrilemethyl acrylate copolymer.
Patent FI-822864-L (FI)
Inventor: MIYADERA TETSUO
IPC: C07D477/00
Filed: 1982-08-18
Abstract: Compounds of the formula: <CHEM>  wherein: R<1> represents a hydrogen atom, a C2-3 alkyl group, a 1-hydroxyethyl group or a 1-hydroxy-1-methylethyl group;  R<2> represents a group of formula: <CHEM> in which, X represents a hydrogen atom, an alkyl group, a cyanoalkyl group, a haloalkyl group, an alkoxyalkyl group, an alkylthioalkyl group, an alkoxycarbonylalkyl group, an alkoxy group, an alkylthio group, an alkylsulphinyl group, an alkylsulphonyl group, a hydroxy group or a halogen atom, where each alkyl or alkoxy has 1-4 carbon atoms; Y represents a hydrogen atom, a C1-4 alkyl group, a C1-4 alkyl group substituted by a hydroxy, amino, carboxy or C1-4 alkoxy group, a C1-5 aliphatic acyl group, a C1-5 aliphatic acyl group substituted by a hydroxy, amino, carboxy or C1-4 alkoxy group, a group of formula -C(R<5>)=N-R<6> (R<5> and R<6> each represents a hydrogen or C1-4 alkyl). <CHEM> represents a 2- or 3-azetidinyl, a 2- or 3-pyrrolidinyl, a 2-, 3- or 4-piperidyl or a 3,4,5,6-tetrahydropyrimidin-5-yl. R<3> represents a carboxy group or a protected carboxy group, and pharmaceutically acceptable salts thereof, provided that when the group <CHEM>  is a 4-piperidyl group then Y is not a C1-4 alkyl group and when <CHEM> is a 3-pyrrolidinyl group Y is not a group then Y is not a group -C(R<5>)=n-R<6>, are useful antibiotics.
Patent FI-823043-L (FI)
Inventor: LANSBERGEN GABRIEL JACOBUS THE
IPC: C11B7/00
Filed: 1982-09-03
Abstract: A process for the fractionation of hardened butterfat resulting in a fraction (i) enriched in triglycerides comprising two fatty acid residues having each at least 16 carbon atoms and 1 fatty acid residue with 2 to 8 carbon atoms, said triglycerides having a carbonnumber ranging from 24 to 42 and a fraction (ii) enriched in triglycerides having a carbonnumber greater than 42. Fractionation is preferable carried out in the presence of a solvent such as acetone or hexane. Margarine fat blends containing fraction (i) display improved butterlike properties.
Patent FI-830630-L (FI)
Inventor: REICHEN FREDY
IPC: F16L27/00
Filed: 1983-02-25
Abstract: Two rigid cylindrical sleeves are interconnected by a spring bellows. Each cylindrical sleeve carries a flange section. Such flange section is provided with joint plates. The joint plates are a forklike interconnecting structure. A rolling contact wedge member is located in a first number of joint plates and a rolling contact prism member is located in a second number of joint plates. This provides for a hinge-like joint of a rolling contact rocker structure having a line contact only of the parts moving relative to each other. Because no friction exists in such hinge joint, a cold welding is not possible. Accordingly, no additional stresses due to such cold welding will be able to exist in the pipe conduit sections interconnected by this apparatus.
Patent FI-843648-L (FI)
Inventor: HONEGGER WERNER
IPC: B65H29/51
Filed: 1984-09-18
Abstract: Before winding-up the printed products arriving in imbricated product formation, the thickness of the imbricated product formation travelling toward a winding mandrel, respectively toward a product coil or package forming thereupon, is regulated to a prescribed value. This is effected by spreading or compacting the printed products within the imbricated product formation. For this purpose a first conveyor device is driven at higher or lower speed than a second preceding conveyor device. The imbricated product formation of prescribed thickness is wound-up upon the winding mandrel together with a winding strap maintained under tension which always lies upon the outer side of the coil layer being formed. By regulating the thickness of the imbricated product formation to be wound-up so as to have a prescribed value which remains essentially constant throughout the winding-up procedure, it is possible to form product coils of essentially constant diameter with a prescribed constant length of winding strap independently of the thickness of the arriving printed products.
Patent IE-32349-L (IE)
Title: Central heating boilers
IPC: F24H9/02
Filed: 1968-09-11
Abstract: 1,242,215. Hot water boilers. J. C. W. O'BRIEN. 9 Sept., 1968 [12 Sept., 1967], No. 41611/67. Heading F4A. In a domestic boiler having a casing 6 including a lagged water section 8 and an extension section 9 housing a burner 10, e.g. oil or gas, and ancillary equipment, the combustion chamber is a continuously curved tube 11 in the water section having its inlet and outlet facing the extension section. The sections 8 and 9 are separated by a partition 7 welded to the casing 6. The tube 11 may be provided with one or two semicircular tubes 21 and/or outwardly projecting fins 15. The casing 6 may be circular. The water section is adapted to be mounted in the cavity wall 5 of a dwelling with a short portion inside the dwelling covered by a square cover plate 16 finished by a stove enamelling or with a decorative laminate and carrying a thermostat, an indicating light and a switch. The extension section 9 exterior of the dwelling is provided with a louvred detachable cover 18. Water pipe connections 26 to the boiler are connected to pipes passing through the wall 5.
[GB1242215A]
Patent IE-841358-L (IE)
Title: A space-divided optical switch assembly
IPC: H04Q3/52
Filed: 1984-05-30
Abstract: 1. A device for an optical spatial switching being accesses of a first group (GA) of N first distinct optical elements (fa) and a second group (GP) of P second distinct optical elements (fp), characterized in that it comprises : - an optical selection assembly (10) constituted by a stack of N rigid, flat optical plates (1) interposed and each maintained in a fixed position face to the access of one of the N first optical elements (fa) which are mounted according to the pitch of the optical plates (1) in their stack in a network which is transverse to these plates, each optical plate (1) in the assembly (10) comprising P distinct waveguides (g), first ends of which are coupled in common to the access of the first optical element which faces it and to which this optical plate is associated, second aligned ends of the P distinct waveguides (g) emerging on one of the edges, each optical plate being associated to an opaque tape (5, 7) presenting at least one perforation (I) and being movable in front of the second ends of the P waveguides of this optical plate, and all the optical plates (1) in this assembly having the second ends of their waveguides with their N tapes associated to the same side of the optical selection assembly (10), - an optical distribution assembly (20) constituted by a stack of P optical distribution plates (21) in which the plates (21) are mounted transversely to the optical plates (1) of the optical selection assembly (10) and at the same pitch as that between the second ends of the waveguides of each of the optical plates (1) of the optical selection assembly (10), and each one incorporating N individual waveguides (h) having their first ends coupled in common to the access of said second optical element (fp) to which the respective plate (21) is associated, whereas second aligned ends emerge on one of the edges of the plate, the first ends of the guides (h) of the different plates (21) being disposed at the same side of the stack and being coupled to the accesses of the second optical elements (fp), the second ends of the waveguides of the different plates (21) emerging at a common side of the stack and being arranged in N rows perpendicularly to the planes of the plates (21) of the distribution assembly, these second ends facing on each row second ends of the P waveguides respectively of one of said plates of the selection assembly (10) and being separated from said plate by the associated tape (5, 7).
[EP0131131A1]
Patent IE-881666-L (IE)
Title: Peptide boronic acid inhibitors of trypsin-like proteases
IPC: A61K38/00
Filed: 1988-06-03
Abstract: Peptides comprising C-terminal boronic acid derivatives of lysine, ornithine, and arginine, homoarginine and corresponding isothiouronium analogs thereof, of the formula <CHEM> are reversible inhibitors of trypsin-like serine proteases such as thrombin, plasma kallikrein and plasmin.
[EP0293881A2]
Patent IE-37206-L (IE)
Title: Attachable leg
IPC: A47B91/00
Filed: 1972-12-11
Abstract: 1362075 Separate feet MARDON ILLING- WORTH Ltd 5 Dec 1972 [8 Jan 1972] 969/72 Heading A4U [Also in Division B8] A leg 12 is detachably clamped to a base 10 of a container such as a box of corrugated or solid board or a pallet by a device having a body 18 and a flange 19, the leg and the device having teeth 16, 20 which adjustably inter-engage so that the distance between the flange 19 and the leg 12 can be varied to suit the thickness of the base 10. The teeth 20 are flexible and so can be resiliently forced past the tooth 16 by a ratchet-type action. The flange 19 may have a diameter which reaches as far as the side wall of the leg, andthe body 18 may be slit to make it flexible so as to facilitate the tooth inter-engagement. In a second embodiment, Fig. 3, (not shown), the top of the leg has a recess into which the base 10 is deformed by the flange 19 and which also receives the flange 19. In a third embodiment, Figs. 5 and 6, (not shown), the leg has an upper flange having slots and is attached to a base having complementary slots by elongate clamping plates having flanges which are passed through the aligned slots and have flexible teeth for adjustably engaging a tooth in the slot in the leg flange. Each leg and each clamping device may be a moulding of plastics material, e.g. polystyrene or polyethylene. Each leg may be internally stiffened.
[GB1362075A]
Patent IE-801780-L (IE)
Title: Scaffolding joint
IPC: E04G7/30
Filed: 1980-08-22
Abstract: A scaffolding joint for connecting together a pair of scaffolding members (1) and (2) has a lug (4) on one member for co-operation with a bracket (5) on the other, and a wedge (6) arranged to retain the bracket (5) and lug (4) tightly in engagement. The wedge (6) has guide surfaces (23) arranged to cooperate with surfaces (25) on the bracket (5) to guide the wedge (6) to a retracted position and retention surfaces (24) arranged to co-operate with corresponding surfaces (26) on the bracket (5) to retain the wedge (6) in that position.
[EP0024865A1]
Patent IE-44179-L (IE)
Title: Compositions for inhibiting absorption of cholesterol
IPC: A23L33/20
Filed: 1976-10-18
Abstract: Polyol fatty acid polyesters having at least four fatty acid ester groups are fortified with fat-soluble vitamins and used in pharmaceutical compositions for treating and/or preventing hypercholesterolemia in animals, especially humans, and in low-calorie foods.
[US4034083A]
Patent IE-802421-L (IE)
Title: Quinazoline derivatives
IPC: C07D239/74
Filed: 1980-11-21
Abstract: The quinazoline derivatives have the formula: 
<CHEM>
 wherein R<1>a and R<1>b are esterified carboxy, R<2> and R<3> are hydrogen, alkyl, halogen, nitro, amino, alkoxy, aryloxy, alkylthio, alkylpiperazinyl, acylamino or dialkylamino which may be substituted with hydroxy,
 A<1> is a group of the formula: 
<CHEM>
 in which R<4> is hydrogen, alkyl, hydroxy, alkoxy, alkenyloxy, dialkylamino or 2,2-dialkoxycarbonylvinylamino, and R<3> is alkyl or alkenyl; or the formula: 
<CHEM>
 wherein R<1> is hydrogen, carboxy or esterifed carboxy, A<2> is a group of the formula: 
<CHEM>
 in which R<4>a is hydrogen, alkyl, hydroxy, alkoxy, alkenyloxy or dialkylamino, R<6> is carboxy or esterified carboxy R<2>, R<3> and R<5> are each as defined above. The quinazoline derivatives are useful as antiallergy agents.
Patent IE-832767-L (IE)
Title: Sand trap
IPC: B01D21/04
Filed: 1983-11-25
Abstract: 1. Sand collector for the recovery of sand suspended in water, having a trough (1), which is provided with an entry (4) for the water/sand mixture and a water outlet (8) and into which at least one drivable bucket wheel (2) dips, wo which the sand settling on the floor (5) of the trough (1) may be conducted by means of at least one drivable worm (3) arranged coaxially to the bucket wheel (2), characterized in that each bucket wheel (2) is drivable independently of the respective associated worm or worms (3) and that at least one of the two drive speeds is variable.
Patent IE-44488-L (IE)
Title: 2,6-dinitroanilines
IPC: C07C67/00
Filed: 1976-12-21
Abstract: This invention relates to certain novel substituted 2,6-dinitroaniline compounds of formula (I) wherein R2 is sec-alkyl C3-C7; monochloro-sec-alkyl C3-C4 or methoxy-sec-alkyl C3-C4; Z is -CHR3OCH3, R3 being hydrogen or-CH3 and Y is chloro or alkyl selected from the group consisting of -CH3, -C2H5, n-Pr, i-Pr, sec-Bu and i-Bu, and compounds of formula (I) selected from the group wherein: z is -CH3; and R2 and Y respectively are -CH(C2H5)2 and i-Pr or -CH(C2H5)2 and -C2H5 or -CH(C2H5)2 and sec-Bu or -CH(C2H5)2 and n-Pr or-CH(C2H5)2 and n-Bu or i-Pr and -C2H5 or sec-Bu and -C2H5 or i-Pr and i-Pr or i-Pr and n-Pr or sec-Bu and i-Pr or -CH(C2H5)-CH2Cl and -Cl or sec-Bu and n-Pr and compounds of formula (I) selected from the group wherein: R2 is i-C4H9 or n-Pr, Z is-CH2OCH3 and Y is i-Pr or -CH3 or -C2H5; R2 is -CH(C2H5)2, Y is n-Bu and Z is CH2OCH3; or R2 is n-Bu, Z is -CH2OCH3 and Y is i-Pr; R2 is i-Pr, Z is -CH2OCH3 and Y is n-C4H9; R2 is CH(C2H5)2, Z is CH2OC2H5 and Y is CH3. It further relates to certain novel preemergence herbicidal methods and compositions employing substituted 2,6-dinitroaniline compounds.
[CA1100998A]
Patent IE-853198-L (IE)
Title: Antibiotic derivatives
IPC: C07D413/04
Filed: 1985-12-17
Abstract: The compounds of the formula: <CHEM> wherein R<1> is amino or an organic residue bonded through nitrogen; R<2> is carboxy or a group derivable therefrom; X is hydrogen, methoxy or formylamino, provided that when R<1> is acetylamino or amino and X is hydrogen, R<2> is not paranitrobenzyloxycarbonyl or benzhydryloxycarbonyl or salts thereof exhibit excellent antimicrobial activity, and are utilized as antimicrobial agents.
Patent IE-922401-L (IE)
Title: An injectable pharmaceutical composition for the¹protectionof tissue damaged by ischemia
IPC: A61K31/765
Filed: 1987-05-14
Abstract: "IMPROVED FIBRINOLYTIC COMPOSITION" of the Invention In accordance with the present invention, a composition is provided that is effective in dissolving blood clots and reestablishing and maintaining blood flow through thrombosed coronary or other blood vessels. The fibrinolytic composition of the present invention comprises an enzyme, such as streptokinase, urokinase, tissue plasminogen activator or other fibrinolytic enzyme, and a surface-active copolymer. The surface-active copolymer can be an ethylene oxide-propylene oxide condensation product with the following general formula: HO(C2H4O)b(C3H6O)a(C2H4O)bH wherein a is an integer such that the hydrophobe represented by (C3H6O) has a molecular weight of approximately 950 to 4000, preferably approximately 1750 to 3500, and b is an integer such that the hydrophile portion represented by (C2H4O) constitutes approximately 50% to 90% by weight of the compound.
[CA1297792C]
Patent NO-762741-L (NO)
Inventor: BALZER M
IPC: B29C65/02
Filed: 1976-08-06
Abstract: Fremgangsmåte til forbinding av baner, plater eller fomdeler av termoplastiske kunststoffer.
Patent NO-811908-L (NO)
Inventor: DERUNGS ROMANO
IPC: C07D405/04
Filed: 1981-06-04
Abstract: Imidazole derivatives of the formula    <IMAGE>  I  wherein X is hydrogen or C1-4-n-alkyl and Y is thienyl, optionally substituted by methyl or fluorine, or a group of the formula    <IMAGE> Y1  wherein R1, R2 and R3 independently are hydrogen, methyl, fluorine, hydroxy or methoxy, or two of R1, R2 and R3 on adjacent carbon atoms taken together are methylenedioxy or ethylenedioxy, or one of R1, R2 and R3 is mono- or di-(C1-4-n-alkyl)-amino and the other two are hydrogen, and physiologically compatible or pharmaceutically acceptable acid addition salts thereof, are described. These compounds of formula I inhibit the aggregation of the blood platelets.