baber/WOPTO huggingface dataset:
Patent IL-186551-A0 (IL)
Title: Quinoline and quinoxaline derivatives as inhibitors of kinase enzymatic activity
IPC: C07D215/22
Filed: 2007-10-10
Abstract: Compounds of formula (IA) or (IB), are inhibitors of aurora kinase activity: Formula (IA), (IB) wherein -L1Y1-[CH2]z- is a linker radical wherein Y1, L1 and z are as defined in the claims; R6 is C1-C4alkoxy, hydrogen or halo; W represents a bond, —CH2—, —O—, —S—, —S(═O)2—, or —NR5— where R5 is hydrogen or C1-C4 alkyl; Q is ═N—, ═CH— or ═C(X1)— wherein X1 is cyano, cyclopropyl or halo; linker radicals L2 are as defined in the claims; R is a radical of formula (X) or (Y): wherein R1 is a carboxylic acid group (—COOH), or an ester group which is hydrolysable by one or more intracellular carboxylesterase enzymes to a carboxylic acid group; R4 is hydrogen; or optionally substituted C1-C6 alkyl, C3-C7 cycloalkyl, aryl, aryl(C1-C6 alkyl)-, heteroaryl, heteroaryl(C1-C6 alkyl)-, —(C═O)R3, —(C═O)OR3, or —(C═O)NR3 wherein R3 is hydrogen or optionally substituted (C1-C6)alkyl, C3-C7 cycloalkyl, aryl, aryl(C1-C6 alkyl)-, heteroaryl, or heteroaryl(C1-C6 alkyl)-; R41 is hydrogen or optionally substituted C1-C6 alkyl; and D is a mono-cyclic heterocyclic ring of 5 or 6 ring atoms.
Patent IL-189595-A0 (IL)
Title: Hydrogel functionalized with a polymerizable moiety and their uses as biosensors or bioreactors
Filed: 2008-02-18
Abstract: The present invention relates to a new hydrogel functionalized with a polymerizable moiety, the polymerized hydrogels, films and gels comprising the same and their use for cells, proteins, DNA or other molecules encapsulation, including use as biosensors or bioreactors.
Patent IL-198621-A0 (IL)
Title: Systems and methods for posterior dynamic stabilization of the spine
Filed: 2009-05-07
Abstract: Devices, systems and methods for dynamically stabilizing the spine are provided. The devices include an expandable spacer having an undeployed configuration and a deployed configuration, wherein the spacer has axial and radial dimensions for positioning between the spinous processes of adjacent vertebrae. The systems include one or more spacers and a mechanical actuation means for delivering and deploying the spacer. The methods involve the implantation of one or more spacers within the interspinous space.
Patent IL-206759-A0 (IL)
Title: Liquid formulation of fsh
Filed: 2010-07-01
Abstract: The present invention relates to a liquid pharmaceutical composition comprising a follicle stimulating hormone polypeptide and benzalkonium chloride and benzyl alcohol as preservatives. The composition further comprises optionally one or more other pharmaceutically acceptable excipients. In one embodiment, the composition contains methionine as an antioxidant. The composition shows a good storage stability and is especially useful for the prophylaxis and treatment of disorders and medical indications where follicle stimulating hormone preparations are considered as useful remedies.
Patent IL-217332-A0 (IL)
Title: Rnai modulation of rsv therapeutic uses thereof
IPC: C12N15/113
Filed: 2012-01-02
Abstract: The present invention relates to a method of reducing the levels of a viral protein, viral mRNA or viral titer in a cell in a subject comprising the step of administering an iRNA agent to said subject, wherein the iRNA agent comprising a sense strand having at least 15 or more contiguous nucleotides complementary to gene from a first mammalian respiratory virus and an antisense strand having at least 15 or more contiguous nucleotides complementary to said sense strand, wherein said gene is selected from the group consisting of the P N or L gene of RSV.
Patent RO-126026-A0 (RO)
Title: Convertible motor vehicle body system
Inventor: OANCEA NECULAI DORIN
IPC: B60J7/02
Filed: 2010-08-23
Abstract: The invention relates to a convertible motor vehicle body system. According to the invention, the body system intended, in particular, to close/release a motor vehicle load carrying compartment (1), comprises a roof assembly (3) which is fixed as to slide along some upper slides (12, 13) mounted on a vehicle cabin (2), two lateral dump shutters (38, 39) sliding under the roof assembly (3), some rear pillars (18) assembled with the roof (3) and fixed as to slide along some slides (7) mounted on the lateral sides of the load carrying compartment (1), and a tail gate (5) vertically foldable in relation to the rear pillars (18), so that the slides (12, 13) are fixed, in the front part, onto the cabin (2), by some resilient means, while, in the rear part, they are fixed by some resilient means onto a front wall (10) integral with the motor vehicle load carrying compartment (1), the roof assembly (3) being provided with some front and rear male means for relative blocking on the vertical and transverse direction, which cooperate with some front female blocking means provided on the motor vehicle cabin (2) and some rear female blocking means, respectively, provided on the front wall (10) integral with the load carrying compartment (1), a central lock (58), whose tongue is locked within a pocket (62) located at the top of the front wall (10), blocking the body system on the longitudinal direction, in the position with the fully released load carrying compartment (1).
Patent RO-126565-A0 (RO)
Title: Technical products made of rubber and thermoplastic polyurethane and process for manufacturing the same
Inventor: DAVID VIOREL
IPC: C08L9/02
Filed: 2010-12-02
Abstract: The invention relates to a range of technical products and to a process for manufacturing the same. According to the invention, the products consist of vulcanizable rubbers, reinforcing elements and active surfaces of thermoplastic polyurethane-type. According to the invention, the process consists in heating a thermoplastic polyurethane sheet at a temperature of 130...150°C, thereafter the sheet is treated successively with a 15% solution of rubber in N-methylpyrrolidone, then with 5% solution of thermoplastic polyurethane in N-methylpyrrolidone and with an adherence agent, the thus treated sheet, rolled in a polyethylene foil, is subjected to a maturation process, thereafter the sheet is doubled on a calendering machine with a mixture of vulcanizable rubber and then it is used for manufacturing technical products which are vulcanized at a temperature of 145...148°C, for 20...50 min at a pressure of 80...150 at.
Patent RO-131719-A0 (RO)
Title: Method and equipment for numerical control and regulation of multi-motor electric drives with brake energy recovery, to be used in high capacity extraction installations
Inventor: HUREZEANU ADRIAN-IONUŢ
IPC: B60T8/172
Filed: 2016-10-24
Abstract: The invention relates to a method for numerical control and regulation of multi-motor electric drives with brake energy recovery and to an equipment for applying the same, intended to be used in high-capacity extraction installations. According to the invention, the method consists in supplying three inverters (A, B and C) for the control of traction motors and a braking inverter (D) for the recovery of braking energy from the same intermediate direct current circuit (1), where the output signal of a torque regulator (13) of the first inverter ensures the unitary control of the other inverters, for equalizing the torques in the operation of three traction motors (5, 6, 7), by means of a common data bus (15) which takes over the output data of the torque regulator (13) and applies them to the width-modulated pulse generators (14, 16, 17) of the three inverters, while permanently adjusting the reference quantities, to prevent shocks in the drive control process, and, when the energy stored in the intermediate circuit (1) exceeds the nominal value, the braking inverter is controlled as to convert the direct current energy resulting from the operation in braking condition into alternating current energy the frequency, phase and level parameters of which are compatible with the three-phase network (RST), using therefore a software control and an output filter (23)
Patent RO-135172-A0 (RO)
Title: Pair of rotors used in oil injection screw compressors
Inventor: NIŢULESCU MARIAN
IPC: F04C29/00
Filed: 2021-04-15
Abstract: The invention relates to a pair of rotors for oil-injection screw compressors to be used for compressing gases. According to the invention, the pair of rotors consists of two rotors (1 and 2), a driving one and a driven one, having two parallel axes (3 and 4), where the driving rotor (1) has five (5) lobes and the driven rotor (2) has seven (6) recesses, they gearing to one another, with reduced backlash between the rotors, the two rotors (1 and 2) being covered with a temperature-resistant material, which has an expansion coefficient close to that of the rotor material, and a hardness lower than that of the rotor material.
Patent AP-2004003047-A0 (AP)
Title: Gravitational energy driven fluid mixer
Inventor: CAWOOD DESMOND EDWARD
Filed: 2004-05-21
Abstract: This invention relates to a gravitational energy utilizing displaceable fluid dispensing apparatus for filtering fluid in an apparatus displacing fashion. Although not so limited the invention finds useful application when used in the field of water filtration
Patent MW-5886-A1 (MW)
Title: Substituted bridged-diazabicycloalkyl quinolone carboxylic acids
IPC: C07D215/56
Filed: 1986-08-28
Abstract: Antibacterial compounds have the formula <CHEM> wherein R<1> is hydrogen, a pharmaceutically acceptable cation, or alkyl; A is CH, CF, CCl or N; Y is alkyl, haloalkyl, cyclopropyl, vinyl, methoxy, N-methylamino, p-fluorophenyl, p-hydroxyphenyl or p-aminophenyl; or A is carbon and is taken together with Y and the carbon and nitrogen to which A and Y are attached to form a five to seven membered ring which is optionally substituted; and R<2> is a bridged-diazabicycloalkyl group.
Patent IE-910976-A1 (IE)
Title: Compositions comprising cytotoxic agent and permeation¹enhancers
IPC: A61K47/26
Filed: 1991-03-25
Abstract: The present invention is directed to a composition of matter for the percutaneous administration of a cytotoxic agent, and particularly to the percutaneous administration of 5-fluorouracil. The composition comprises, in combination, the cytotoxic agent to be administered and a permeation-enhancing mixture that includes a lower alkanol, propylene glycol or a mixture of polyethylene glycols, a third permeation enhancer and, optionally, a covehicle. The invention is also directed to a method for treating malignant and non-malignant skin disorders and comprises applying to an area of skin affected by a skin disorder, a therapeutically effective amount of the composition of this invention.
Patent MA-27427-A1 (MA)
Title: Composes de benzimidazole-1-yl-thiophene utilises en cancerotherapie
Inventor: ANDREWS III CLARENCE W
IPC: A61K39/00
Filed: 2005-03-04
Abstract: L'invention concerne des composés représentés pas la formule (I), des compositions pharmaceutiques qui renferment ces composés, des procédés de préparation de ces composés ainsi que leur utilisation comme agents pharmaceutiques
Patent MA-46809-A1 (MA)
Title: Ralentisseur actif producteur d’electricité (rape)
Inventor: ABBOU Ahmed
IPC: H02K7/18
Filed: 2019-09-03
Abstract: Ralentisseur actif producteur d’electricité (rape) joue un double rôle : permet de limiter les vitesses des véhicules sur les trajets à forte utilisation et produire de l’électricité de façon permanente. Cette innovation donne l’opportunité de récupérer l’énergie électrique à partir de l’énergie cinétique issue du passage des véhicules au-dessus du ralentisseur proposé, l’énergie produite sera utilisée immédiatement ou stockée sur des batteries pour une utilisation ultérieure.
Patent UY-25345-A1 (UY)
Title: Sal de bisulfato del inhibidor de la vih-proteasa
Inventor: LINDRUD JANAK SINGH MADHUSUDHA
IPC: A61K31/44
Filed: 1999-01-12
Abstract: La presente invención proporciona la sal de bisulfato cristalina de la fórmula (ver) que se encuentra que tiene una velocidad de solubilidad/disolución inesperadamente alta y biodisponibilidad oral alta con relación a la forma de base libre de este compuesto inhibidor de la azapeptido-vih-proteasa.
Patent UY-26365-A1 (UY)
Title: Sales de disodio, monohidratos, solvatos de etanol para la liberación de agentes activos
Inventor: BAY WILLIAM E
Filed: 2000-10-04
Abstract: La presente invención provee un solvato de alcohol, como solvato de etanol, de una sal de disodio de un agente de liberación de fórmula I, un hidrato de sal de disodio de un agente de liberación de dicha fórmula. Preferentemente los agentes de liberación incluyen, pero no están limitados a ácido N (5-clorosalisiloil) -8-aminocaprilico (5-CNAC), ácido N- (10-(2-hidroxibenzoil) amino) decanoico (SNAD),y caprilato de sodio N-(8-(2-hidroxibenzoil)amino (SNAC). También provee métodos de preparación de sal de disodio, el solvato de etanol, y el hidrato y composiciones que contiene a la sal de disodio, el solvato de etanol, y/o el hidrato.-
Patent UY-29894-A1 (UY)
Title: Derivados del ácido (2-((2s)-2-hidroxipropil)oxi)fenil)acético y del ácido (2-((2s)-2-hidroxipropil)oxi)fenil) propanoico sustituidos, composiciones farmacéuticas conteniéndolo, procesos de preparación y aplicaciones
Inventor: ASA SJOHOLM TIMEN
IPC: A61P37/00
Filed: 2006-11-01
Abstract: La invención proporciona compuestos de fórmula general en donde m, n, q, R1, R2, R3, R4, R5 y R6 son como se define en la memoria descriptiva, procesos para su preparación, composiciones farmacéuticas que los contienen y su uso en terapia.
Patent ES-151077-A1 (ES)
Title: Mecanismo impulsor de disco oscilante
Filed: 1940-12-09
Abstract: Un mecanismo impulsor de disco oscilantecuyo disco se provee de una corona dentada de rueda cónica que engrana en otra corona dentada fija de igual magnitud y rueda sobre ellacaracterizada porque la corona dentada fija (11) se apoya mediante un disco (12) sobre el eje (5) del disco oscilantegiratoria respecto a éste y centrada con el mismo y se sujeta en dirección axial respecto al eje mediante topes adecuados (1516) fijos sobre el mismo eje (5) y porque dicha corona dentada (11) se une de tal modo por medios adecuados de sujección (2133) a una parte fija de la máquina (1)que se impide tenga rotación propia.
Patent ES-181836-A1 (ES)
Title: Dispositivos de capacitancia negativa
Filed: 1948-01-24
Abstract: Dispositivo para producir una capacitancia negativa, que comprende, en combinación, una válvula termoiónica que tiene un cátodo, una placa y por lo menos una rejilla, una fuente de potencial positivo de corriente continua para la referida placa, y una fuente de tensión de variación de tiempo, caracterizado por un transformador que acopla la referida fuente con la rejilla, estando la fuente de variación de tiempo, acoplada también capacitivamente a la placa, por lo que se presenta una capacitancia negativa a la fuente de variación de tiempo.
Patent ES-182832-A1 (ES)
Title: MEJORAS INTRODUCIDAS EN LA CONSTRUCCIoN DE COLMENAS
Filed: 1948-02-18
Abstract: Mejoras introducidas en la construcción de colmenas caracterizadas por el hecho de constituir a los elementos que la configuran, mediante placas formadas por planchas de aglomerado de corcho recubiertas preferentemente en su total superficie por una capa de adecuado grosor de fibro-cemento o materia similar.
Patent ES-187497-A1 (ES)
Title: Sistema de elementos tubulares de agua y de humos para cambiadores de calor, y especialmente para calderas de vapor
Filed: 1949-03-10
Abstract: Sistema de elementos tubulares de agua y de humos para cambiadores de calor y especialmente para calderas de vapor caracterizados por comprender un cuerpo tubular atravesado al menos en parte por un tubo de humos que presenta en sus extremos aberturas de entrada y salida para el agua y el vapor 1as cuales desembocan en un colector o en varios en los que desembocan también las aberturas correspondientes a los restantes elementos constitutivos de la caldera.
Patent ES-196577-A1 (ES)
Title: UN PROCEDIMIENTO PARA LA OBTENCIoN DE ELECTRODOS NEGATIVOS DESTINADOS A LOS ACUMULADORES DE ELECTRoLITO ALCALINO
Filed: 1951-02-16
Abstract: Procedimiento para la obtención de electrodos negativos destinados a los acumuladores de electrolito alcalino compuestos de un armazón porosa. obtenida mediante concreción de polvos metálicos y en cuyos poros se introduce una masa activa preferentemente en forma de cadmio. caracterizado porque la armazón se compone de niquel-hierro
Patent ES-197147-A1 (ES)
Title: Un pricedimiento para la fabricacion de productos biologicos de tipo antigenos y vacunas integrales para su uso terapeutico e inmunizantes
Filed: 1951-03-27
Abstract: Un procedimiento para la fabricación de productos biológicos de tipo-antígenos y vacunas integrales para su uso terapéutico como preventivos desensibilizantes e inmunizantes que se caracteriza por la obtención de los virus o bacterias etio-patogénicas de infecciones por medios idóneos y en medios de cultivo acondicionados sintéticamente a fin de que sus factores pH y RH sean idénticos a los correspondientes del sitio plasma o mucosa humanos en donde aquellos virus o bacterias se desarrollan reproducen y provocan las reacciones características de las infecciones se caracteriza por la selectividad de los virus cepas o bacterias en cuanto a su poder inmunizante en soluciones tamponadas se caracteriza por la preparación del antíngeno o vacuna integralmente o sea a partir del mismo medio de cultivo en el que se encuentra la bacteria o virus con sus toxinas de excresión y constitución y los productos reaccionales y metabólicos se caracteriza por la esterilización por procedimientos físico-eléctricos y térmicos reforzada o no por sustancias químicas y se caracteriza por la conservación del producto antígeno integral por liofilia con la consiguiente presentación en polvo del antígeno integral base en la confección de fórmulas y especialidades biológicas.
Patent ES-199287-A1 (ES)
Title: PROCEDIMIENTO PARA LA OBTENCIoN DE UN PRODUCTO COSMÉTICO
Filed: 1951-08-22
Abstract: Procedimiento de obtención de un producto cosmético caracterizado por el hecho de que contiene al menos un proteinato metálico y un diluente destinado a favorecer la penetración del mencionado proteinato en la piel o sus anejos.
Patent ES-199925-A1 (ES)
Title: PROCEDIMIENTO DE FABRICACIoN DE UN PRODUCTOPARA LA TRANSFORMACIoN DE RESIDUOS VEGETALES EN ESTIÉRCOL
Filed: 1951-10-09
Abstract: Procedimiento de fabricación de un producto para la transformación de residuos vegetales en estiércol, caracterizado por la formación de una composición integrada de nitrógeno, urea, potasa, cloro, fósforo, azufre, sodio, sulfato de manganeso y hormonas.
Patent ES-303777-A1 (ES)
Title: Steam surface condenser
IPC: F28B1/06
Filed: 1964-09-04
Abstract: An air-cooled steam surface condenser having steam-condensate lanes (16) branching from a steam distribution chamber 4 and in communication with a condensate collecting tank 5 is characterized by baffles 17 disposed in the steam-condensate lanes to establish lower and upper condensing zones and to provide tapered steam paths and the lower condensing zones are separated from subcooling zones 20 by condensate collection trays 21. In the form shown, steam enters through a pipe 3 extending through the tank 5 and flows through the lower condensing zones and up over the baffles 17, through the upper condensing zones and the saturated uncondensable gases reach a chamber 18 at which point the cross-sectional area of the steam path is between 8 and 10% of that at the inlet. Pipes 19 convey these gases to subcooling zones 20, located at the cooling air inlet, where entrained water vapour is finally condensed out, before the uncondensable gases leave via pipes 24. Cooling air 13 is drawn through finned ducts (151) (Figs. 2 and 8, not shown), by a variable speed fan 11. In one form (Fig. 3, not shown) the inclination of the trays (21) is reversed so that the condensate and steam flow concurrently in the lower cooling zone, the condensate being collected in tanks (511) arranged at the outer ends of the lanes and in communication with central tank (51) through pipes (28). In another form (Fig. 4, not shown), baffle plates (32) are placed in the steam distribution chamber (4) to constrain the incoming steam to enter the upper parts of the lower condensing zones.
Patent ES-315496-A1 (ES)
Title: Electric starter motors
IPC: H02K7/12
Filed: 1965-07-06
Abstract: In engine starting apparatus the motor includes a yoke 18 and a plurality of polepieces each having one end rounded, adjacent polepieces having their rounded ends at opposite axial ends of the yoke. The field system of the motor consists of a single field coil 17 extending around the inside of the yoke and shaped to define portions which extend substantially axially relative to the yoke and are joined by curved end portions which extend around the rounded ends of the polepieces. At least one of the polepieces has a part 19a, 21a fixed relative to the yoke and including the rounded end and a movable part 19b, 21b resiliently urged away from the fixed part in a direction parallel to the motor shaft. The apparatus further includes means 28, 29 connecting the movable part to the pinion, the arrangement being such that when the field system of the motor is energized the movable part will be attracted by the fixed part and the pinion will be moved from its inoperative position to its operative position. The fixed and movable parts of the polepieces may be formed with complementary inter-engaging faces of part conical form.
Patent ES-335300-A1 (ES)
Title: A digging wheel assembly for a reclaimer or other digging machine
IPC: E02F3/22
Filed: 1967-01-05
Abstract: In a bearing assembly balls bear on circular races formed from rods or wires of circular cross-section.
Patent ES-338904-A1 (ES)
Title: Coating Materials and Methods for their Application
IPC: C09D7/63
Filed: 1967-04-04
Abstract: A coating composition, especially for heat fusion processes, comprises (a) polyvinyl chloride, an acetal resin or a polyamide, (b) Pb, Cr, Mn, Ti or Fe or an oxide or salt thereof and (c) a nitrogen compound selected from dicyandiamide (except in combination with Ti or Fe or compounds thereof), hydrazine a hydrazide, thiohydrazide, dihydrazide dithiohydrazide or hydrazone or polyethylene hydrazide, hydrazodicarbonthioamide urazine, guanazole, or azodicarbonamide. Optionally there may also be added tris (dimethylaminomethyl) phenol and/or a pigment. The PVC compositions may be used as plastisols in fluidised bed coating of steel or copper sheets or as an organosol, which is baked after drying, to coat aluminium or steel. Nylon 6 (particle size 210Á) with lead silicochromate and dicyandiamide is used in a fluidised bed coating process. An acetal resin with titanium dioxide and adipic dihydrazide is dusted over a heated steel panel and postheated.
Patent ES-344598-A1 (ES)
Title: Improvements relating to Electrolytic Capacitors.
IPC: H01G9/00
Filed: 1967-08-30
Abstract: Aluminium electrode foil having an enlarged effective surface is produced by a method including electrolytically etching hard aluminium foil. The foil may then be subjected to thermal treatment prior to anodic oxidation thereof. The capacitance of the foil is measured with respect to a platinum-coated silver cathode in the electrolyte in which forming was carried out.