baber/WOPTO huggingface dataset:
Patent CO-5540316-A2 (CO)
Title: Pirimidinas inhibidoras de cdk, su preparacion y uso como medicamento
Inventor: BRUMBY THOMAS
IPC: A61K31/513
Filed: 2003-12-26
Abstract: 1.- 	Compuestos de la fórmula general I dondeR1 es hidrógeno, halógeno, alquilo C1-C6, nitro o es el grupo -COR5, -OCF3 , - (CH2)nR5, -S-CF3 o -SO2CF3, R2 es alquilo-C1-C10, alquenilo-C2-C10, alquinilo-C2-C10 o cicloalquilo-C3-C10 o es alquilo-C1-C10, alquenilo-C2-C10, alquinilo-C2-C10 o cicloalquilo-C3-C10 mono o polisustituido de manera igual o diferente por hidroxi, halógeno, C1-C6-alcoxi, alquiltio-C1-C6, amino, ciano, alquilo-C1-C6, cicloalquilo-NH-(CH2)n-C3-C10, cicloalquilo-C3-C10, hidroxialquilo-C1-C6, alquenilo-C2-C6, alquinilo-C2-C6, C1-C6-alcoxi-C1-C6-alquilo-C1-C6, alcoxi-C1-C6-alcoxi-C1-C6- alquilo-C1-C6, -NHC1-C6-alquilo, -N(C1-C6-alquilo)2, -SO(C1-C6-alquilo), -SO2(C1-C6-alquilo), alcanoílo-C1-C6, -CONR3R4, -COR5, alquilo C1-C6OAc, carboxi, arilo, heteroarilo, -(CH2)n-arilo, -(CH2)n-heteroarilo, fenil-(CH2)n-R5, -(CH2)nPO3(R5)2 o por el grupo -R6 o -NR3R4 y el propio fenilo, cicloalquilo-C3-C10, arilo, heteroarilo, -(CH2)n-arilo y -(CH2)n-heteroarílo puede estar opcionalmente mono o polisustituido de manera igual o diferente por halógeno, hidroxi, alquilo-C1-C6, alcoxi-C1-C6, heteroarilo, benzoxi o por el grupo -CF3 o -OCF3, yel anillo del cicloalquilo-C3-C10 y el alquilo-C1-C10 puede estar interrumpido opcionalmente por uno o varios átomos de nitrógeno, oxígeno y/o de azufre y/o por uno o varios grupos =C=O y/o opcionalmente el anillo puede contener una o varias uniones dobles, oR2 es el grupo X. es oxígeno o es el grupo -NH-, -N(C1-C3-alquilo) o es -OC3-C10-cicloalquilo, el que puede estar mono o poli-sustituido, de manera igual o diferente por un heteroaromáticosoX y R2 forman juntos un anillo cicloalquilo-C3-C10, que opcionalmente puede contener uno o varios heteroátomos y opcionalmente puede estar mono o polisustituido por hidroxi, alquilo-C1-C6, alcoxi-C1-C6 o halógeno, ...
Patent CO-5660300-A2 (CO)
Title: Composicion limpiadora antimicrobial
Inventor: ZOCCHI GERMAINE
IPC: C11D3/38
Filed: 2006-03-16
Abstract: 1.- Una composición limpiadora antimicrobial la cual comprende:(a) 0,01% a 5% de polihexametileno biguanida hidrocloruro; (b) 0,01% a 5% de biopolímero aniónico; y (c) el resto siendo agua.2.- La composición tal y como se reivindica en la cláusula 1, caracterizada porque el biopolímero aniónico es mucina.3.- La composición tal y como se reivindica en la cláusula 1, caracterizada además porque incluye 0,01% por peso a 5% por peso de un surfactante seleccionado del grupo que consiste de surfactantes aniónicos, surfactantes de poliglucosido dé alquilo, surfactantes de óxido de amina, surfactantes zwitteriónicos y surfactantes no iónicos y mezclas de los mismos.
Patent CO-6150144-A2 (CO)
Title: Inhibidores de proteina tirosina fosfatasa humana y metodos de uso
Inventor: GRAY JEFFREY LYLE
IPC: C07D277/28
Filed: 2009-01-27
Abstract: 1.- Un compuesto que tiene la fórmula:en donde R es una unidad tiazolilo sustituida o no sustituida que tiene la fórmula:R4 y R5 se escogen cada uno independientemente de: i) hidrógeno; ii) alquilo C1-C6 lineal, ramificada o cíclico sustituido o no sustituido; iii) fenilo sustituido o no sustituido; iv) heteroarilo sustituido o no sustituido; o R4 y R5 se pueden tomar juntos para formar un anillo saturado o insaturado que tiene de 5 a 7 átomos; dichas sustituciones se escogen independientemente de una o más unidades alquilo C1-C6 lineal, cíclico o ramificado, halógeno, hidroxilo, o ciano; R6 es una unidad escogida de: i) hidrógeno; ii) alquilo C1-C6 lineal, ramificado o cíclico sustituido o no sustituido; iii) fenilo sustituido o no sustituido; y iv) heteroarilo sustituido o no sustituido; R1 se escoge de: i) hidrógeno; ii) alquilo lineal o ramificado C1-C6; iii) fenilo sustituido o no sustituido; o iv) bencilo sustituido o no sustituido; R2 se escoge de: i) alquilo lineal o ramificado C1-C6; o ii) alcoxi lineal o ramificado C1-C6; R3 es hidrógeno o alquilo lineal o ramificado C1-C4. 2.- Un compuesto de acuerdo con la Reivindicación 1 en donde R tiene la fórmula:3.- Un compuesto de acuerdo con la Reivindicación 2, en donde R4 y R5 son cada uno hidrógeno.
Patent CO-6220930-A2 (CO)
Title: Inhibidores de la actividad de akt
Inventor: SEEFELD MARK A
IPC: A61K31/12
Filed: 2009-08-06
Abstract: 1.- Un compuesto de Fórmula (I):en la que: R41 y R42 se seleccionan independientemente entre: hidrógeno, , halógeno, alquilo C1-4, alquilo C1-4 sustituido, alquiloxi C1-4, alquiloxi C1-4 sustituido, furano, furano sustituido, tiofeno y tiofeno sustituido, donde Q y Y se seleccionan independientemente entre: nitrógeno y -C(R70)-, y Z se selecciona entre: nitrógeno y -C(R48)-, con la condición de que al menos uno y como mucho 2 de Q, Y y Z sean nitrógeno, y R30 se selecciona entre: alquilo C1-4 y alquilo C1-4 sustituido con uno a tres átomos de flúor, donde R70 se selecciona entre: hidrógeno, y halógeno, y R48 se selecciona entre: hidrógeno, alquilo C1-4, alquilo C1-4 sustituido, arilo, arilo sustituido, heteroarilo, heteroarilo sustituido, cicloalquilo, cicloalquilo sustituido, heterocicloalquilo, heterocicloalquilo sustituido y halógeno; R43 se selecciona entre: hidrógeno, halógeno, alquilo C1-4, alquilo C1-4 sustituido, alquiloxi C1-4, alquiloxi C1-4 sustituido,furano y tiofeno; R44 está ausente o se selecciona entre: -(CR60R61)mAR donde el grupo AR está sin sustituir, -(CR60R61)mAR donde el grupo AR está sustituido y alquilo C1-6, donde m es de 0 a 3 y AR es un anillo, aromático o no aromático, saturado o insaturado, cíclico o policíclico, que contiene de 3 a 16 átomos de carbono y que contiene opcionalmente de uno a tres heteroátomos, con la condición de que cuando el anillo es aromático y el número de átomos de carbono es 3, el anillo contenga al menos dos heteroátomos y cuando el anillo es aromático y el número de átomos de carbono es 4, el anillo contenga al menos un heteroátomo, y R60 y R61 se seleccionan independientemente entre: hidrógeno y alquilo C1-4, con la condición de que cuando m es 3, no más de 4 de R60 y R61, cuando se añaden juntos, sean alquilo C1-4, R45 se selecciona entre hidrógeno y alquilo C1-4; R20 se selecciona entre hidrógeno alquilo C1-4 e hidroxi;X se selecciona entre O, S y NR49,donde R49 se selecciona entre hidrógeno y alquilo C1-4; y n es de 0 a 2 y este resto está opcionalmente, si es aplicable, sustituido con hidroxialquilo C1-4; con la condición de que uno y sólo uno de R41 y R42 sea y/o una sal farmacéuticamente aceptable del mismo.
Patent CO-6331300-A2 (CO)
Title: Composicion que comprende un anticuerpo monoclonal o el anticuerpo scfv enlazado a un epitopo en la region de tallo de la proteina de hemaglutinina (ha)
Inventor: LIDDINGTON ROBERT C
IPC: A61K39/395
Filed: 2010-07-06
Abstract: La invención proporciona anticuerpos humanos scFV y anticuerpos monoclonales que neutralizan el virus de influenza. También proporciona métodos de tratamiento y/o prevención de influenza relacionada con una enfermedad o trastorno de dicha influenza. La invención también provee el método de vacunación a un paciente contra la influenza. También proporciona métodos de diagnóstico de influenza - relacionados con enfermedades o trastornos y métodos de detección de la presencia de influenza en una muestra.
Patent CO-6390005-A2 (CO)
Title: Conversion de aceites vegetales a aceites base y combustibles para transporte
Inventor: MILLER STEPHEN J
IPC: C10G3/00
Filed: 2011-02-01
Abstract: La presente invención está dirigida a métodos (procesos) y sistemas para procesar aceites biológicamente derivados que contienen triglicéridos para dar lugar a aceites base y combustibles para transporte, en donde la oligomerización parcial de los ácidos grasos allí contenidos da lugar a una mezcla oligomerizada a partir de la cual se pueden extraer los aceites base y combustibles para transporte. Dichos métodos y sistemas pueden involucrar una etapa inicial de hidrotratamiento o una isomerización directa de la mezcla oligomerizada.
Patent CO-6440516-A2 (CO)
Title: Formulaciones concentradas en suspensión acuosa que contienen saflufenacilo
Inventor: KRAPP MICHAEL
IPC: A01N43/54
Filed: 2012-02-27
Abstract: Una formulación concentrada en suspensión acuosa para la protección de plantas, que comprende: - 2-cloro-5-[3,6-dihidro-3-metil-2,6-dioxo-4-(trifluorometil)-1-(2H)pirimidinil]-4-fluoro-N-[[metil(1-metiletil)amino]sulfonil]benzamida en forma de su anhidrato cristalino;- al menos un tensioactivo no iónico seleccionado de copolímeros de bloque de polioxietileno-polioxi-alquileno C3-C4;- al menos un tensioactivo aniónico que comprende al menos un grupo arilsulfonato; y - agua;en donde el valor pH de la formulación está en el rango de 3 a 7.
Patent CO-7101250-A2 (CO)
Title: Formulación de tensioactivos para la liberación de fluidos fósiles subterráneos
Inventor: SALAZAR LUIS C
IPC: B32B15/02
Filed: 2014-10-10
Abstract: La presente descripción proporciona una formulación de tensioactivos para uso en el tratamiento y recuperación de fluidos fósiles de una formación subterránea. La formulación de tensioactivos incluye un tensioactivo primario, un agente de estabilidad de la formulación y agua de inyección. La formulación de tensioactivos puede ser inyectada en uno o más pozos de inyección situados dentro de la formación subterránea y posteriormente pueden recuperarse fluidos fósiles a partir de uno o más pozos de producción.
Patent DD-158860-A2 (DD)
Title: Verfahren zum einziehen rotationssymmetrischer hohlkoerper
Inventor: WENKE KARLHEINZ
IPC: B21D22/16
Filed: 1981-05-12
Abstract: Das Verfahren zum Einziehen rotationssymmetrischer Hohlkoerper bezieht sich auf das Gebiet der Blechumformung und stellt eine Zusatzerfindung analog PS 141630 dar. Infolge durchmesserabhaengiger variabler Wanddickenreduzierung wird ein groesserer Umformgrad erreicht. Anwendungsgebiet ist die Konsumgueterindustrie, der Fahrzeug- und Apparatebau.
Patent EP-1035354-A2 (EP)
Inventor: COCCOLO ENZO
IPC: B29C48/355
Filed: 2000-03-02
Abstract: A chain-operated traction unit for drawing, comprising a
pair of chains (15, 16) which are arranged on opposite sides
with respect to the product to be drawn (30), each being
constituted by a plurality of elements (17) which are mutually
concatenated so as to form a closed loop which has a
substantially straight active portion, which is parallel to the
drawing axis (13), and pusher means (46) which are suitable to
push toward each other said active portions of said chains (15,
16) in order to impart to said product to be drawn (30) a given
traction force, said chains (15, 16) lying on two planes which
are substantially parallel to each other, being disposed on
opposite sides with respect to said drawing axis (13), and being
suitable to cooperate with the product to be drawn (30) by
virtue of the opposite lateral surfaces (22) of said
concatenated elements (17).
Patent EP-1033797-A2 (EP)
Inventor: KIE-HYUNG CHUNG
IPC: H05H1/24
Filed: 2000-03-02
Abstract: A pulse power system includes an energy storing device for storing
electric energy; a high power arc switch comprising: a cylindrical housing having a
central axis and defining a predetermined discharging region; a first electrode disposed
within the cylindrical housing to be movable in a direction of the central axis; a second
electrode disposed within the cylindrical housing and spaced away from the first
electrode at a predetermined distance, an arc generating between the first and second
electrodes as the first electrode approaches the second electrode; an insulating member
formed at a portion between the first and second electrodes except for the discharging
region; and a solenoid coil for forming a magnetic field within the discharging region in
a direction of the central axis, the arc formed between the first and second electrodes
being spirally moved in a direction of the central axis by a magnetic field formed in a
circular direction by the arc and the magnetic field formed by the solenoid coil in the
direction of the central axis, thereby electrically interconnecting the first and second
electrodes; a load excited by the electric energy stored in the energy storing device
according to an operation of the switch; and a transmission line for connecting the
switch and the load.
Patent EP-1041440-A2 (EP)
Inventor: CARPI ENIO LUIZ
IPC: G03F1/78
Filed: 2000-03-04
Abstract: A method for fabricating mask patterns in accordance with the present invention includes the steps of providing a mask blank (122) for patterning, propagating a laser/electron beam (120) having an elliptical cross-sectional shape onto the mask blank, the elliptical cross-sectional shape having an elongated axis and edges at opposite ends of the elongated axis and positioning the mask blank to write a pattern on the mask blank wherein the positioning includes employing the edges of the elliptical cross-sectional shape of the laser/electron beam to write corners (124) of the pattern. A system is also included. <IMAGE>
Patent EP-1039247-A2 (EP)
Inventor: BESSER ULRICH
IPC: F24H1/36
Filed: 2000-03-14
Abstract: A heating device has a burner (10) fed by a fuel-air mixture, a combustion chamber (12), a heat exchanger unit (14) for cooling combustion gas in a low performance range below steam dew point and a bypass device (20) for linking the combustion chamber to a combustion gas eduction device (18) so as to re-heat the combustion gas to a value acceptable for a flue connection by introducing heat from the combustion gas.  Fitted in the combustion gas eduction device upstream from a bypass channel (20) opening (22), an adjusting element (32) affects the mass flow rate of combustion gases reaching the combustion gas eduction device via the bypass channel.
Patent EP-1038666-A2 (EP)
Inventor: FUKINO KIYOTAKA
IPC: G03F7/004
Filed: 2000-03-21
Abstract: A heat mode type lithographic printing plate precursor
which can be directly mounted on a printing press without
development processing after scanning exposure for a short time
to conduct plate-making, has excellent press life and also gives
few print stains onto a printed face, which comprises a substrate
having provided thereon an image recording layer containing fine
light-heat convertible particles which are hydrophilic in their
surfaces, the layer being made hydrophobic by the action of heat.
Patent EP-1048938-A2 (EP)
Inventor: MAY JOE T
IPC: G01J1/02
Filed: 2000-03-16
Abstract: A UV sensor design which virtually eliminates solarization effects
on optical components and photodetector and is effective for both broad
area and collimated light sources. The sensor design reduces the number of
photons striking a unit area of any of the materials in the light path
sensitive to UV light to a level which does not produce appreciable
solarization over very long periods of time. The UV sensor has as the first
optical element in the viewing path a UV transmitting, extremely low
solarization window. The back surface of this window is frosted to
produce some diffusion of the UV rays. A small metal disc with a very
small aperture is the next optical element and reduces the total amount of
energy admitted to the optical measurement system. A second frosted UV
transmitting, extremely low solarization window further diffuses the light
beam passing through the aperture. The UV light from this second window
travels toward to two UV filters and is further dispersed to produce low
intensity level UV light which impinges on a silicon photodetector.
Patent EP-1054013-A2 (EP)
Inventor: JUNG IL NAM
IPC: C07F7/12
Filed: 2000-05-11
Abstract: The present invention is organosilicon compounds described by formula (1) and formula (2) were R<sup>1</sup> is selected from hydrogen, dichlorosilyl, trichlorosilyl, methyldichlorosilyl, dimethylchlorosilyl or trimethylsilyl, each R<sup>2</sup>, R<sup>3</sup> and R<sup>4</sup> are independently selected from hydrogen, chlorine and alkoxy radicals having 1 to 12 carbon atoms, aryloxy radicals having up to 12 carbon atoms, aryl radicals having up to 12 carbon atoms or saturated hydrocarbon radicals having 1 to 12 carbon atoms, n=2 to 6 and methods for the making of organosilicon compounds described by formulas (1) and (2).
Patent EP-1056134-A2 (EP)
Inventor: BRUSH LINDA
IPC: H01L21/336
Filed: 2000-05-17
Abstract: A trench-gated power device (100) comprises a substrate (101) having
an overlying epitaxial layer disposed on an upper layer of the
substrate, well regions containing source (110) and body regions (111),
a trench gate, and a drain region (113). The gate trench (105) having
sidewalls (106) that comprise selectively grown epitaxial material. A
dielectric layer (102) having an upper surface and thickness and width
dimensions that substantially correspond to the height and width
dimensions of a gate trench is formed on an upper layer of the
substrate. A layer (103) of epitaxial material is grown on the upper
layer of the substrate and the dielectric layer (102) and planarized to
be substantially coplanar with the upper surface of the dielectric layer
(102), which is than removed, so as to form gate trench sidewalls (106)
that comprise selectively grown epitaxial material. The process
comprising lining the trench (105) with a dielectric material (107) and
filling the lined trench with a conductive material (108).
Patent EP-1056220-A2 (EP)
Inventor: AIHARA YASUO
IPC: H04B1/3822
Filed: 2000-05-23
Abstract: Since a flip part for protecting an operation surface
is provided, with a patch antenna provided on the front surface
of the flip part, in the case the device is disposed laterally
on a desk with the operation surface upward, the patch antenna
is oriented vertically (zenith direction), and thus the optimum
antenna directivity can be provided with respect to the
counterpart of the electric wave transmission and receipt so
as to ensure the stable electric field strength.
Patent EP-1069326-A2 (EP)
Inventor: GOMBERT STEPHANE
IPC: F16B21/16
Filed: 2000-06-21
Abstract: The rigid elastic plastic holder element comprises a container-cage (1) pressed onto the plastic, longitudinally ribbed bolt (5). The cage's inner wall (2) is placed on the bolt. A support arm (3) is molded on the opposite side of the cage and is pointed contrary to the pressure direction (A) at an obtuse angle onto the opposite inner wall. The free end of the support arm has an acute-angled support edge (13) whose distance from the inner wall is less than the outer diameter of the ribbed bolt. Above the acute-angled support edge is a support lug (14) resting on the lengthwise ridges (11).
Patent EP-1077104-A2 (EP)
Inventor: SCHUETZ UDO
IPC: B21D1/08
Filed: 2000-08-05
Abstract: Beim Rekonditionieren von Spundfässern (1) zu Deckelfässern wird durch einen konzentrisch zur Faßlängsachse durch den Übergangsbereich (16) zwischen Bodenscheibe (17) und Innenrand (18) des Oberbodens (7) eines Spundfasses (1) geführten Kreisschnitt (19) mittels einer Schneidrolle (20) die Bodenscheibe (17) des Oberbodens (7) von dem Faßmantel abgetrennt, und anschließend wird der untere Abschnitt (18a) des Innenrandes (18) des Oberbodens (7) mit einem Profilierwerkzeug in eine ringförmig umlaufende Innensicke des Faßhalses (5) ausgeformt. Anschließend wird auf dem Öffnungsrand (6) des Faßmantels (2) ein Spunddeckel oder ein einfacher Deckel mit einem Spannring befestigt.
Patent EP-1106344-A2 (EP)
Inventor: MOECK CHRISTOF DR
IPC: B60R13/02
Filed: 2000-11-10
Abstract: A sandwich sheet (I) comprises: (A) a core layer of polypropylene particulate foam; (B) cover layers of fiber reinforced polypropylene as well as optionally; and (C) decorative layers. The core layer (A) contains 1-30 wt.% recycled particles from components (A), (B) and optionally (C). Independent claims are included for: (i) a process for the production of a foam sheet by comminuting waste pieces of sandwich sheets comprising (A), (B) and optionally (C) to an average particle size of 5-10 mm and bonding 1-20 wt.% of the comminuted material with 80-99 wt.% of polypropylene foam particles in a mold; and (ii) a process for the production of the sandwich sheet (I) by deep drawing of components (A), (B) and optionally (C) at above the softening point of polypropylene.
Patent EP-1103950-A2 (EP)
Inventor: STERGIOPOULOS STERGIOS
IPC: G06T1/00
Filed: 2000-11-16
Abstract: An adaptive multidimensional beamformer having near-instantaneous convergence for
ultrasound imaging systems deploying multidimensional sensor arrays is disclosed. In a first step,
the multidimensional beamformer is decomposed into sub-apertures. Each sub-aperture is then
again decomposed into two coherent subsets of circular and/or line array beamformers in different
coordinate directions of the multidimensional array. Implementation of the multidimensional
beamformer according to the present invention provides the basis for a 3D ultrasound imaging
system according to the present invention comprising a compact multidimensional sensor array
and a compact processing unit that is field deployable and generates high resolution three-dimensional
images in real time. It is also possible to capture four-dimensional images, the
fourth dimension being time and the resulting images forming a video image of a volume of a
moving organ.
Patent EP-1045243-A2 (EP)
Inventor: NAGANAWA RYUICHI
IPC: G01N33/00
Filed: 2000-03-30
Abstract: In a method of analyzing a concentration of a target
substance contained in a fluid using a quartz oscillator
having a surface covered with a layer capable of absorbing
the target substance, the temperature of the fluid and the
quartz oscillator is controlled at substantially the same
predetermined temperature selected according to the
concentration of the target substance in said fluid, so
that the analysis can be made with optimum sensitivity. A
device for analyzing a concentration of a target substance
contained in a fluid, includes a contacting chamber
accommodating a quartz oscillator, a temperature
controller, disposed in a feed passage for feeding the
fluid into said contacting chamber, for adjusting a
temperature of the fluid at a desired predetermined
temperature; and a detector of a frequency of the quartz
oscillator.
Patent EP-1087315-A2 (EP)
Inventor: BLOTT STEPHEN MICHAEL
IPC: G06Q10/00
Filed: 2000-09-11
Abstract: A method and apparatus for verifying email attachments are disclosed.
Upon a user initiating a send of an email message, the message is scanned to
determine if the message contains an attachment indicator term. Attachment
indicator terms are terms which, if present in an email message, would generally
indicate that an attachment should be present in the message. If the message
contains an attachment indicator term, then it is determined whether the message
actually contains an attachment. If not, then the user is prompted with a send
verification request which gives the user an opportunity to send the message
notwithstanding the prompt, or to return to a composition screen in order to attach
an inadvertently omitted attachment. In one embodiment, the attachment indicator
term(s) is identified to the user (e.g. via highlighting) upon return to the composition
screen.
Patent EP-1094619-A2 (EP)
Inventor: NARUSE TETSUYA
IPC: H04B1/707
Filed: 2000-10-16
Abstract: A signal receiving apparatus of the global positioning
system and a mobile wireless terminal apparatus execute the
synchronization acquisition to the satellite signal at high speed
and reduce the consumption of electric power. According to the
present invention, since the spread spectrum signal from the base
station of the cellular system, that is synchronized with the
satellite signal to be transmitted from the GPS satellite, is
received and based on the spread spectrum signal the system time
signal as a reference signal used to synchronize with the
satellite signal is generated, and receiving the satellite signal,
the synchronization acquisition with the PN code in the satellite
signal can be executed in a short period of time in synchronism
with the system time signal. And thereby the consumption of
electric power can be further reduced.