baber/WOPTO huggingface dataset:
Patent IE-810092-L (IE)
Title: Dipeptide amides
IPC: A23L27/30
Filed: 1981-01-20
Abstract: Amides of dipeptides of L-aspartyl-D-amino acids of formula <IMAGE> and their cationic and addition salts with physiologically acceptable acids where Ra is methyl, ethyl, n-propyl or isopropyl, R is a branched radical selected from the group comprising phenyl, diisopropyl carbinyl, d-methyl-t-butyl carbinyl, d-ethyl-t-butyl carbinyl, di-t-butyl carbinyl, 2-methylthio-2,4- dimethylpentane-3-yl <IMAGE> where at least one of the radicals R3, R4, R5 or R6 is alkyl having from 1 to 4 carbon atoms and the remainder are hydrogen or alkyl having from 1 to 4 carbon atoms, X is O, S, SO, SO2, C=O or CHOH, m is 0 or 1-4, n and p are each 0, 1, 2, or 3 and the sum of n + p is not greater than 3 and the sum of the carbon atoms in R3, R4, R5 and R6 is not greater than 6 and when R3 and R4 or R5 and R6 are both alkyl, they are then methyl or ethyl, <IMAGE> where one of the radicals R7, R8 or R9 is alkyl having from 1 to 4 carbon atoms and the remainder are hydrogen or alkyl having from 1 to 4 carbon atoms and the sum of the carbon atoms in R7, R8 and R9 is not greater than 6, m and q are the same or different and each has the values previously specified for m, <IMAGE> where each of the radicals R12 and R13 is methyl or ethyl or R12 is hydrogen and R13 is alkyl having from 1 to 4 carbon atoms, Z is O or NH and t is 1 or 2, <IMAGE> where w is 1-4, R14 and R16 are each alkyl having from 1 to 4 carbon atoms, R15 is H, OH, methyl or ethyl and the sum of the carbon atoms in R14, R15 and R16 is not greater than 6 and when R14 and R15 are both alkyl, then they are methyl or ethyl and <IMAGE> where R17 and R19 are alkyl having from 1 to 4 carbon atoms, R18 and R20 are H or alkyl with 1 or 2 carbon atoms, A is OH and B is H, OH or CH3 and when joined together A and B are <IMAGE> where the sum of the carbon atoms in R17, R18, R19 and R20 is not greater than 6 and when R17 and R18 or R19 and R20 are both alkyl then they are methyl or ethyl; these amides are powerful sweeteners which have advantages over those in the prior art; edible compositions containing these amides, methods for their use in edible compositions and new intermediate amines and amides useful for their production.
[ES8204413A1]
Patent IE-840130-L (IE)
Title: Benzoylureas
IPC: A01P7/04
Filed: 1984-01-20
Abstract: The invention relates to new benzoylurea compounds of the general formula <IMAGE> wherein R1 is a hydrogen atom or represents 1 or 2 substituents which are selected from the group consisting of halogen and alkyl and haloalkyl having 1-4 carbon atoms, R2 is a hydrogen atom or represents 1 or 2 substituents which are selected from the group consisting of chlorine, methyl and trifluoromethyl, and R3 is a hydrogen atom or represents 1-3 alkyl and/or alkenyl groups each having 1-6 and/or 2-6 carbon atoms respectively, or wherein R3 together with the cyclohexyl ring to which it is attached forms a bi- or polycyclic hydrocarbyl group having 8-14 carbon atoms and, if desired, substituted with 1-3 alkyl groups each having 1-4 carbon atoms. The compounds have an insecticidal and acaricidal activity. After having been processed to compositions, the compounds may be used for the control of insects and/or mites in a dosage from 1 to 5000 g of active substance per hectare.
[US4656193A]
Patent IE-800209-L (IE)
Title: Dextrorotatory 9, 10-ethanoanthracene derivative.
IPC: C07C215/38
Filed: 1980-02-01
Abstract: For all designated states : BE, CH, DE, FR, GB, IT, LU, NL, SE 1. S-(+)-alpha-[methylamino)methyl]-9-10-ethano anthracene-9(10H)-ethanol of the formula I  see diagramm : EP0014434,P11,F1  or an acid addition salt thereof. For the contracting state : AT 1. A process for the production of S-(+)-alpha-([methylamino)methyl]-9-10-ethano anthracene-9(10H)-ethanol of the formula I ad indicated in claim 1, or of an acid addition salt thereof, which process comprises a) resolving the racemic alpha-[(methylamino)-methyl]-9-10-ethanoanthracene- 9(10H)-ethanol and isolating S-(+)-alpha-[(methylamino)-methyl]-9-10-ethano anthracene-9(10H)-ethanol, if desired in the form of an acid addition salt, or b) reacting a compound of the formula II  see diagramm : EP0014434,P12,F1  with a compound of the formula III X2 -CH3 wherein one of X1  and X2  is the amino group and the other is a reactive esterified hydroxyl group, and Y1 is a free hydroxyl group, and X1 together with Y1  can also be an epoxy group, and A is the 9,10-ethanoanthracen-9(10H)-yl radical, or c) in a compound of the formula IV  see diagramm : EP0014434,P12,F2  in which at least one of Z1  and Z2  is a removable radical and the other may be hydrogen, or Z1  and Z2 together are a divalent removable radical, and A is the 9,10-ethanoanthracen-9(10H)-yl radical, removing Z1 and/or Z2 , d) reducing a compound which differs from the compound of the formula I only in that, in said compound, a carbon atom adjacent to the nitrogen atom is attached to this latter through a double bond or is substituted by a hydroxyl group or an oxo radical, optionally together with lower alkoxy, or e) adding ethylene to S-alpha-[(methylamino)-methyl]-9(10H)-anthracene, or hydrolyzing the intermediate obtained, and, if desired, converting the resultant S-(+)-alpha-[(methylamino)methyl]-9,10-ethanoanthracen- e-9(10H)-ethanol into an acid addition salt and/or liberating the base from a resultant acid addition salt.
Patent IE-800310-L (IE)
Title: Tyre bead-ring
IPC: B21F37/00
Filed: 1980-02-19
Abstract: A method of manufacturing a tire bead ring of the package type by winding metal wires on a form of revolution, the radially inner face of the tire bead ring having a frusto-conical shape of half angle alpha at the apex and of radius R with respect to the axis of rotation of the tire bead ring, in which a permanent circular deformation is effected on the wires prior to their winding on the form of revolution, is improved due to the fact that the permanent circular deformation is a radial deformation of a radius substantially equal to the radius R of the tire bead ring and is effected on the wires whose one principal axis of inertia of their cross section is inclined by one angle alpha with respect to the axis of winding of the wires on the form of revolution.
[US4305769A]
Patent IE-37351-L (IE)
Title: Saccharase inhibitor.
IPC: C12P19/22
Filed: 1973-02-28
Abstract: This invention relates to the production of saccharase inhibitors in which a polysaccharidic or oligosaccharidic amylase inhibitor is hydrolytically degraded either enzymatically or by acid hydrolysis. The invention also relates to the use of said saccharase inhibitors in pharmaceutically acceptable therapeutic compositions in the treatment of conditions indicating adiposity, hyperlipaemia (atherosclerosis), diabetes, pre-diabetes, caries and the like.
[US3879546A]
Patent IE-830332-L (IE)
Title: Vaccination for herpes simplex virus
IPC: A61K/
Filed: 1983-02-17
Abstract: Disclosed are immunologically active preparations of Herpes simplex virus envelope glycoproteins, gD-1 and gD-2. Preferably purified through use of a monoclonal anti-gD antibody immunoadsorbent, gD-1 and gD-2 preparations are incorporated in vaccines useful in generating immunological responses protective against Herpes simplex disease states. Disclosed also is the preparation and use in vaccination procedures of synthetic polypeptides comprising amino acid sequences which are: (1) substantially common to both gD-1 and gD-2; cumulatively hydrophilic in nature; and (3) specifically immunoreactive with a type common, monoclonal anti-gD antibody of Group VII classification.
[US4762708A]
Patent IE-37375-L (IE)
Title: Plastics bag
IPC: B65D33/24
Filed: 1973-03-06
Abstract: 1359099 Bags and pouches DECOFLEX Ltd 16 March 1973 [21 March 1972] 13152/72 Heading A4G [Also in Divisions B5 and B8] A transparent polythene bag includes a downwardly opening pouch 8 and an enclosed part 7 formed on its front wall. The front and back walls of the bag may be of equal depth Fig.6 (not shown) or the rear wall may be deeper than the front wall, as shown, or vice versa Fig.7 (not shown). The bag is closed by turning the pouch 8 inside out to enclose the part 7 and the free end portion of the rear wall Fig. 5 (not shown).
[GB1359099A]
Patent IE-37421-L (IE)
Title: Spring balance mechanism
IPC: G01G23/20
Filed: 1973-03-20
Abstract: 1376053 Spring balance: pointers CAMBRIAN HOUSEWARES Ltd 26 March 1973 [25 March 1972] 14133/72 Heading G1J and G1W A kitchen spring balance includes a unitary, self-contained spring balance mechanism 10 which comprises two L-shaped members 12a, 12b interconnected by a pair of leaf springs 11a, 11b, a pointer 20 or indicator disc pivotally mounted on the base part 15a of a member 12a, and a control arm 37 fastened to spring 11b so as to deflect angularly as the spring is loaded and control the rotation of the pointer or indicator disc. The pointer 20 comprises a moulded plastics inner part pivoted by means of integral trunnions 22, and a spring wire blade 29 resiliently locked to the inner part by engagement with bridge parts 31, 32 and grooved abutment 34. The pointer is rotated by a weak spring 36 until the end of a limb 27 abuts the control arm 37 and the sensitivity of the weighing is adjusted by adjusting arm 27 using screw 28. To zero or tare the balance an adjusting screw (not shown) may be provided which contacts the arm 37 or an arm 71 attached thereto.
[GB1376053A]
Patent IE-900518-L (IE)
Title: Pesticidal 3-cyano-5-alkoxy-1-arylpyrazoles
IPC: A01N57/18
Filed: 1990-02-13
Abstract: The invention describes novel 3-cyano-4-sulfenylated-5-alkoxy-1-arylpyrazoles of general formula(I) wherein typically preferred substituents are: R is C1 to C4 alkyl fully substituted by halogen; R1 is C1 to C4 alkyl, C3 to C6 alkenyl and alkynyl or aralkyl (each of which may be optionally substituted), dialkylaminocarbonyl or a group -P(=X)(Oalkyl)(Salkyl) wherein X is oxygen or sulfur; R2, R3, R5 and R6 are each hydrogen or halogen; R4 is CF3, OCF3, SCF3, SOCF3, SO2CF3, OCHF2, halogen or alkyl; and n is 0, 1 or 2. The invention further relates to intermediates and processes to make the compounds as well as to compositions thereof and to methods of control of arthopod (especially insect) nematode, helminth, and protozoan pests.
Patent IE-810696-L (IE)
Title: Plastics film with occludable strips
IPC: B31B19/90
Filed: 1981-03-27
Abstract: An apparatus for producing a plastic container having occludable closure strips comprises a source for the closure strips, a rotatable casting cylinder having a pair of spaced apart circumferential grooves defined therein, a mechanism for advancing the closure strips to the casting cylinder, an extruder for casting a plastic film onto the casting cylinder so that it becomes connected to base portions of the closure strips, and a chill roll for receiving the combination of plastic film and closure strips to provide cooling.
[US4306924A]
Patent IE-790701-L (IE)
Title: Ergot alkaloids and heparin
IPC: A61K9/00
Filed: 1979-08-08
Abstract: A pharmaceutical composition comprises a mixture of a hydrogenated ergot alkaloid of formula (I):- <IMAGE> wherein R is hydrogen or a C1-4 alkyl group other than t-butyl; R1 is methyl, ethyl or isopropyl; R2 is isopropyl, secbutyl, isobutyl or benzyl; and X is hydrogen or methoxy; together with heparin, the proportion of compound (I) in mgs. to heparin in international Units being 1:5000. The composition may be in unit dosage form containing 0.5 mgs. of the alkaloid and 2,500 I.U. of heparin, together with a pharmaceutical carrier or diluent for injection (eg. poly-N- vinyl-2-pyrrolidone).
[GB2015338A]
Patent IE-37652-L (IE)
Title: Phenylethylamines
IPC: C07C47/56
Filed: 1973-05-31
Abstract: Trifluoromethylthiophenylethylamine derivatives, made from the corresponding acid chlorides by successive reduction, condensation with nitroethane, reduction, and condensation with an amide, possess anorexigenic properties, unaccompanied by central stimulant activity or cardiovascular effects.
[US3965190A]
Patent IE-44925-L (IE)
Title: Measuring spoon set
IPC: G01F19/00
Filed: 1977-04-26
Abstract: A plurality of measuring spoons, for measuring liquid or dry materials, each having a bowl and an integral elongated handle. The bowls vary in capacity from each other. The handles of the spoons are releasably affixed to a spoon holding ring by a slot at the end of the handle. Each slot has an arcuate section so that a tubular spoon holding ring can be snapped into the slot due to flecture of the spoon handle portions defining the slot. The slots permit the spoons to be individually pivoted on the spoon holder ring, or individual spoons can be removed from the spoon holder ring. The spoons nest together to form a compact unit. The spoon holder ring is designed to permit the entire assembly to be hung up in the kitchen in a convenient location. Each spoon is clearly marked with an indication as to its bowl capacity. Several of the spoons have a measuring ledge within the bowl and these spoons can be used to measure two different capacities depending on whether the spoon is filled to the ledge or to the top. Also, spilling from these spoons is minimized if the spoon is filled only to the ledge.
[US4043203A]
Patent IE-790883-L (IE)
Title: Detergent compositions.
IPC: A61K8/00
Filed: 1979-08-08
Abstract: An improved non-irritating or low irritating detergent composition exhibiting good foaming properties is disclosed. The composition is a synergistic mixture of an amphoteric surfactant and a phosphobetaine or phosphitaine surfactant.
[US4231903A]
Patent IE-33476-L (IE)
Title: Destroying penicillin activity in an antibiotic mixture
IPC: C07D499/00
Filed: 1969-07-09
Abstract: 1,259,204. Purifying cephalosporin antibiotics. ELI LILLY & CO. 10 July, 1969 [10 July, 1968], No. 34874/69. Heading C2A. A method for freeing a mixture of cephalosporin and penicillin antibiotics from penicillin biological activity comprises treating the mixture with a 2-mercaptoamine of formula wherein R<SP>1</SP> and R<SP>2</SP> are hydrogen or C 1- C 9 alkyl, and R<SP>3</SP> is hydrogen, -COOH or a salt thereof or COOR where R is C 1 -C 9 alkyl, at a pH of 4 to 9 and a temperature of 20-40‹ C. using a molar ratio of 2-mercaptoamine to penicillin of at least 1. The process is preferably performed in aqueous medium or in a mixed aqueous-organic medium of water with ethanol or dioxane. Preferred mercapto-amines are 2-aminoethanethiol, 2-dimethylamino-ethanethiol, cysteine or its ethyl ester, N-butylcysteine and 2-(N-hexylamino)ethanethiol. The penicillin activity is destroyed due to reaction with the mercaptoamine with opening of the #-lactam ring to give an amide derivative.
[GB1259204A]
Patent IE-41041-L (IE)
Title: Removing chlorine from zinc sulphate solution.
IPC: C22B19/20
Filed: 1975-05-05
Abstract: A process for removing chlorine from a solution of zinc sulfate, in which the pH of the solution is reduced to below 2.6 with sulfuric acid. Cupric ions are established in the solution in an amount such that after removal of the chlorine by precipitation as cuprous chloride, there remains an excess of cupric copper in the solution which is greater than 0.5 g/l. The cupric ions can be added by adding cupric sulphate and zinc powder, or cupric salt and metallic copper, or cupric copper followed by cuprous oxide. The cuprous chloride precipitate is collected and washed and treated with sodium hydroxide in an amount to raise the pH to more than 7, thereby to precipitate cuprous oxide which is separated by filtration.
[US4005174A]
Patent FI-821397-L (FI)
Inventor: HABICHT ERNST
IPC: C07D317/46
Filed: 1982-04-21
Abstract: The invention relates to novel benzodioxole derivatives of the formula I    <IMAGE>  (I)  in which R1 represents an unsubstituted or substituted, aromatic or heteroaromatic radical, alk represents an alkylene or alkylidene radical having a maximum of 5 carbon atoms, n represents O or 1, R2 and R3 each represents, independently of the other, hydrogen, lower alkyl, lower alkoxy or halogen, and A represents the radical O-R4, wherein R4 represents hydrogen or an unsubstituted or substituted, aliphatic or araliphatic hydrocarbon radical, or A represents the radical   <IMAGE>   in which either R5 and R6 each represents, independently of the other, hydrogen or lower alkyl, or R5 and R6 are bonded to one another and, together with the adjacent nitrogen atom, represent unsubstituted or lower alkyl-substituted tetra- or hexa-methyleneimino or 4-morpholinyl, to salts of compounds of the formula I in which A represents OR4 wherein R4 is hydrogen, with bases, and to acid addition salts of compounds of the formula I in which the radical R1 has a basic character, and to pharmaceutical compositions that contain them. The novel substances exhibit diuretic and, in addition, uricosuric activity and may be administered, according to the invention, preferably in the form of appropriate pharmaceutical compositions, to mammals for the treatment of oedema and hypertension.
Patent IE-901233-L (IE)
Title: Disposal absorbent article
IPC: A61F13/514
Filed: 1990-04-05
Abstract: A disposable absorbent article, such as a disposable diaper, having barrier leg cuffs. The barrier leg cuffs have a distal edge which is spaced from the proximal edge so as to provide a barrier against leakage. The barrier leg cuff has a portion affixed to the diaper so that the spacing between the barrier leg cuffs is increased in selected portions to reduce irritation of the genetalia and to provide a larger area to receive bodily discharges.
Patent IE-36697-L (IE)
Title: Infusion cannula assembly.
IPC: F16L33/22
Filed: 1972-09-13
Abstract: An infusion cannula assembly has a mounting sleeve made from a thermoplastic material and having inside in the order mentioned a cylindrical mouth channel, a cylindrical mounting chamber with a diameter greater than that of the mouth channel, a connection chamber with a diameter greater than that of the mounting chamber, and an inwardly protruding snap collar, and an end section of a flexible cylindrical cannula tube, made from a polymer having a low friction coefficient extends through said mouth channel into said mounting chamber and is fastened to the mounting sleeve by being expanded into engagement with the circumferential wall of said mounting chamber by means of a tubular metal insert inserted in the cannula tube and having an outwardly directed end flange which abuts the cannula tube and is positioned between said snap collar and an annular shoulder at the merging point between said mounting chamber and said connection chamber, said end flange being movable past said snap collar with snapping action.
[US3802433A]
Patent IE-34645-L (IE)
Title: Container closures
IPC: B65D41/42
Filed: 1970-10-01
Abstract: 1277396 Container closures AMERICAN FLANGE & MFG CO Inc 1 Oct 1970 [27 Oct 1969] 46707/70 Heading B8T A metallic bottle cap comprises a top wall 2, a curved portion 3 and a skirt 4 to which is attached a pull member 8. Score lines 6 and 7 facilitate tearing. A gasket 11 comprises a solid plastics sheet 12 adhered to the underside of the cap, and a spongy annulus 17 formed in situ, which are fused together. In another embodiment, the annulus 17 is covered by the solid sheet (23), Fig. 4 (not shown).
[GB1277396A]
Patent IE-881513-L (IE)
Title: Spiro (4.5) decane derivatives
IPC: C07D498/10
Filed: 1988-05-20
Abstract: Spiro (4,5) decane compounds of the formula:   <IMAGE>   in which: X is methyl and Y is hydrogen or R'-CO- in which R' is C1-C4-alkyl or C1-C4-alkoxy,   <IMAGE>  X and Y together represent   <IMAGE>   in each of which A is hydrogen, methyl, carboxy, methoxycarbonyl or ethoxycarbonyl; R is C1-C7-alkyl optionally containing a double bond; Z is a C2-C7-polymethylene chain optionally carrying an OH group; R1 is hydrogen or methyl; and R2 is hydrogen, R'-CO- or benzyloxycarbonyl; and physiologically tolerable acid addition salts thereof. These compounds may be used therapeutically especially in the treatment of asthma, allergic phenomena and bronchopathies.
Patent IE-35903-L (IE)
Title: Guanidine derivatives, their preparation, and antiviral¹compositions containing them
IPC: A61K31/17
Filed: 1971-12-16
Abstract: 1311432 Substituted ureas IMPERIAL CHEMICAL INDUSTRIES Ltd 13 Dec 1971 [7 Jan 1971] 777/71 Heading C2C [Also in Division A5] Novel substituted ureas of the formula and pharmaceutically acceptable acid addition salts thereof, wherein either R<SP>1</SP> is ethyl, R<SP>2</SP> is bromophenyl and the group -NHCONHR<SP>2</SP> is in the meta-position, or R<SP>1</SP> is isopropyl, isobutyl, isopentyl or phenyl, R<SP>2</SP> is chlorophenyl, bromophenyl, nitrophenyl, ethoxyphenyl or tolyl and the group -NHCONHR<SP>2</SP> is in the meta- or para-position, or R<SP>1</SP> is chlorophenyl, R<SP>2</SP> is C 3-10 alkyl and the group -NHCONHR<SP>2</SP> is in the meta-position, or R<SP>1</SP> is chlorophenyl or tolyl, R<SP>2</SP> is phenyl or o-chlorophenyl and the group NHCONHR<SP>2</SP> is in the para-position are prepared by one of the following processes: (a) reacting the appropriate 1-R<SP>1</SP>-3-(aminophenyl) guanidines with isocyanates of the formula R<SP>2</SP>NCO; (b) reacting thioureido compounds of the Formula III with ammonia in the presence of a catalyst; (c) reacting alkyl or aralkyl thiourium salts derived from thioureas of the above Formula III with ammonia; or (d) oxidizing thioureido compounds of the Formula V 1 - (3 - p - Chlorophenylureido - 3 - (3 - isobutylthioureido)benzene is obtained by reacting p-chlorophenyl isocyanate with 1-isobutyl-3-mphenylaminothiourea. 1 - (p - Chlorophenyl) - 3 - (m - aminophenyl)- guanidine dihydrochloride is prepared by reacting ammonia in the presence of mercuric oxide with 1-(p-chlorophenyl)-3-(m-aminophenyl)thiourea, obtained by reacting p-chlorophenyl isothiocyanate with m-phenylenediamine. 1 - (3 - Isopropylthioureido) - 3 - (3 - p - chlorophenylureido)benzene is made by reacting isopropyl isothiocyanate with 3-(3-p-chlorophenylureido)aniline resulting from the reaction between m-phenylenediamine and p-chlorophenyl isocyanate. 1 - Isobutyl - 3 - (m - aminophenyl)guanidine dihydrochloride is prepared by reacting ammonia in the presence of mercuric oxide with 1-isobutyl-3-(m-aminophenyl)thiourea obtained by reacting isobutyl isothiocyanate with m-phenylenediamine.
[GB1311432A]
Patent IE-45459-L (IE)
Title: Cephalosporin analogues
IPC: C07F9/568
Filed: 1977-08-04
Abstract: PURPOSE:Cephalosporin analogs I(R<1> is H, halogen, lower alkoxy, sulfonyloxy, arylthio or monoheterocyclic thio;R<2> is COOH or its carboxyl derivatives; R<3> is H, or methoxy), e.g. 7beta-amino-3-chloro-1-oxa-1-dithia-3-cephem-4-carboxylic acid.
[JP53018597A]
Patent IE-44381-L (IE)
Title: Fluid-cooled moulding device.
IPC: B29C53/24
Filed: 1976-08-18
Abstract: A mold has a mold cavity centered on an axis and formed with a plurality of arrays of passages each lying at least approximately in a respective plane including the mold axis. Fluid is passed through these passages in order to cool the mold, and fluid may be passed more rapidly or under greater pressure or under lower temperature through some of the passages than through others in order to increase the cooling effect. Similarly inserts may partially insulate some of the passages for cooling some parts of the mold more or less than others. A plurality of temperature sensors each connected to a respective control valve may serve to control the fluid flow through each of the passages or sets of passages for continuous cooling control.
[US4251253A]
Patent IE-811833-L (IE)
Title: Meat replacement products
IPC: A23J1/02
Filed: 1981-08-11
Abstract: Heat replacement product to be used in mixed minced meat products, process for its preparation, and meat products comprising same, whereby the meat replacement product comprises the gluten protein and the bran fractions of whole cereal grain, preferably wheat. To the gluten-bran fraction the blood hemoglobin fraction can be added as well as a milk protein in form of a cheese foam. The meat replacer can replace up to 50 % of the meat.