baber/WOPTO huggingface dataset:
Patent UA-123969-C2 (UA)
Title: БРОМІД 1-(4<sup>1</sup>-МЕТОКСИФЕНІЛ)-3-(4<sup>2</sup>-БІФЕНІЛ)-3-ГІДРОКСИ-2,5,6,7,8,9-ГЕКСАГІДРО-3Н-ІМІДАЗО[1,2-а]АЗЕПІНІЮ, ЩО МАЄ ПРОТИПУХЛИННІ ВЛАСТИВОСТІ
Filed: 2019-06-13
Abstract: Бромід 1-(41-метоксифеніл)-3-(42-біфеніл)-3-гідрокси-2,5,6,7,8,9-гексагідро-3H-імідазо[1,2-а]азепінію, що має протипухлинні властивості. Винахід належить до органічної та фармацевтичної хімії, а також медицини. Визначення протипухлинної активності заявленої сполуки проведено in vitro на 60 лініях ракових клітин при дії речовини в концентраціях 10-4-10-8 моль/л за стандартною процедурою оцінки мітотичної активності, виконаних у Національному інституті раку США (National Cancer Institute of Health, USA) в рамках Development Therapeutic Program. Показано, що заявлена сполука перевищує еталон на більшості лініях ракових клітин з 60, що досліджувалися. Найбільш ефективною вона виявилася відносно клітин лейкемії HL-60(TB), К-562, MOLT-4, RPMI-8226 та SR (перевищує дію 5-флуорурацилу на 91,33, 74,48, 74,30, 70,21 та 71,94 % відповідно), раку товстого кишечнику COLO 205, НСТ-116, НТ-29 та KМ12 (перевищує дію еталону на 79,43, 60,15, 63,66 та 61,80 % відповідно), клітин меланоми SK-MEL-5 перевищує дію 5-флуорурацилу на 82,61 % та клітин раку молочної залози T47D - на 84,76 %. Слід відмітити, що для клітин MDA-MB-468 раку молочної залози мітотична активність становить - 15,21 %. Тобто, заявлена сполука не тільки затримує ріст цих ракових клітин, а й знищує їх.
Patent UA-126099-C2 (UA)
Title: Novel compound exhibiting enteropeptidase inhibitory activity
Inventor: KIM YOUNG KWAN
Filed: 2019-05-08
Abstract: The present invention relates to: a novel compound exhibiting enteropeptidase inhibitory activity; a pharmaceutically acceptable salt thereof; a pharmaceutical composition for metabolic diseases such as obesity, diabetes, or hyperlipidemia, including the compound or a pharmaceutically acceptable salt thereof; and a method for preventing or treating metabolic diseases using the novel compound. The compound of the present invention enables, due to excellent enteropeptidase inhibitory activity, not only fats but also proteins to be excreted when ingested foods are excreted, not absorbed, from the body, resulting in fewer side effects such as fatty stool, and acts only on the gastrointestinal tract, thus reducing side effects such as depression. Thus, the compound of the present invention is very useful as an agent for the treatment or prevention of various metabolic diseases such as obesity, diabetes, and hyperlipidemia.
Patent UA-59771-C2 (UA)
Title: A process for producing homopolymer coarsely dispersed polyvinyl acetate dispersion
Inventor: KUNCHENKO OLEKSII PETROVYCH
IPC: C08F118/00
Filed: 2002-12-17
Abstract: A process for producing homopolymer coarsely dispersed polyvinyl acetate dispersion is performed by emulsion polymerization of vinyl acetate in the acid medium. The aqueous phase is prepared with the concentration of polyvinyl alcohol of 7.5-7.7 % by weight and sulphuric acid ferrous oxide of 1.63-2.21 % by weight, and vinylacetate is loaded simultaneously into two polymerizers.
Patent UA-78004-C2 (UA)
Title: Method for operation of sea gaslift and system for its implementation
Inventor: KYRYCHENKO YEVHEN OLEKSIIOVYCH
IPC: F04F1/20
Filed: 2004-07-26
Abstract: The group of inventions relates to the field of gaslift lift of mixes from sea depth where water is saturated with gas dissolved in it, in particular at development of underwater mineral beds. A method of operation of sea gaslift is in formation of rarefaction and gas desorption in accumulator through which saturated with gas water flows. Desorbed gas is supplied to mixer of gaslift that is placed at smaller depth compared to accumulator. At that one controls the values of accumulated released gas and compressed gas desorbed from sea water, with achieving correspondence of those through control of decrease of pressure value in accumulator through change of ratio of water flow rate for flows coming in and out. A gaslift system has a pump and accumulator with pipelines, indicators and water and gas controllers placed at depth. Depth of accumulator placement is larger than depth of gaslift pipe mixer. The pump pumps out water from the accumulator, through throttling water at outlet controlled slide rarefaction needed for gas desorption in it is formed.
Patent DE-19645488-C5 (DE)
Title: System und Verfahren zum Entnehmen von kaltem Gas aus einem Kryotank
Inventor: HETTINGER WOLFGANG
IPC: F17C7/04
Filed: 1996-11-05
Granted: 2012-08-30
Abstract: Die Erfindung sieht ein System zum Entnehmen von kaltem Gas aus einem Kryotank vor, das einen isolierten Speicherbehälter für flüssiges Gas und eine Entnahmeleitung aufweist. Die Entnahmeleitung ist außerhalb des Kryotanks bis zu einem Verdampfungsvolumen isoliert. Das Verdampfungsvolumen kann die Form einer nicht-isolierten Erweiterung der Entnahmeleitung oder eines kleinen nicht-isolierten, mit der Entnahmeleitung verbundenen Bechers haben. Von dem Verdampfungsvolumen führt eine Leitung über ein Ventil zu einem Verbraucher. Aufgrund des Druckgefälles zwischen Tank und Verbraucher kommt es zu einer Flüssigkeitsströmung in der Entnahmeleitung bis zu dem nicht-isolierten Verdampfungsvolumen außerhalb des Tanks. Dort entsteht eine spontane Verdampfung, die eine Druckerhöhung in der Entnahmeleitung bewirkt und Flüssigkeit in der Leitung und ein Teil des verdampften Gases in den Tank zurückdrückt, bis der Druck in der Entnahmeleitung wieder ausgeglichen ist. Danach strömt die Flüssigkeit wieder durch die Entnahmeleitung nach, es entsteht eine natürliche Druckschwingung, welche den durch die Entnahme bedingten Druckabfall im Kryotank kompensiert.
Patent DE-102009025474-C5 (DE)
Title: PTC-Heizstab-Anordnung und PTC-Heizgerät
Inventor: LIM JAE CHAN
IPC: H05B3/46
Filed: 2009-06-18
Granted: 2019-07-18
Abstract: Stab-Anordnung (100) mit positivem Temperaturkoeffizienten (PTC), aufweisend:
 ein kanalförmiges Stab-Gehäuse (110) mit einer offenen Seite und Flanschen (111), die von dessen einander gegenüberliegenden Rändern nach innen abstehen;
 ein PTC-Element (180), dessen untere Fläche in Kontakt mit dem Innenboden des Stab-Gehäuses (110) ist;
 einen Elektroden-Anschluss (170), der von den Flanschen (111) umgeben ist, der in Kontakt mit der oberen Fläche des PTC-Elements (180) ist und der in dem Innenraum des Stab-Gehäuses (110) derart untergebracht ist, dass sich der Elektroden-Anschluss (170) unter die Flansche (111) erstreckt;
 einen Isolator (120), der an einer nicht in Kontakt mit dem PTC-Element (180) stehenden Außenfläche des Elektroden-Anschlusses (170) angebracht ist; und
 einen Radiator (200), der zwischen die Flansche (111) des Stab-Gehäuses (110) eingesetzt ist und in direktem Kontakt ist mit dem Isolator (120) des Elektroden-Anschlusses (170).
Patent RU-2440376-C9 (RU)
Inventor: SARPESHKAR ASHOK M
IPC: C08G18/42
Filed: 2006-10-23
Granted: 2013-01-20
Abstract: FIELD: chemistry. 
     SUBSTANCE: in one version, polyurethaneurea contains a product of reaction of: (A) at least one (cyclo)aliphatic polyisocyanate prepolymer, having content of NCO groups from approximately 4 to approximately 50%, and average functionality from approximately 2 to approximately 3, which is a product of reaction of (1) at least one (cyclo)aliphatic polyisocyanate and (2) at least one organic compound which contains at least approximately two hydroxylic groups and has molecular weight from approximately 100 to approximately 4000; with (B) an isocyanate-reactive component containing: (1) one or more aromatic diamine compounds containing two primary aromatic amine groups and having molecular weight from approximately 100 to approximately 1000, (2) one or more isocyanate-reactive compounds containing two secondary amine groups and having molecular weight from approximately 100 to approximately 750, where the secondary amine groups are bonded to the (cyclo)aliphatic and/or aromatic groups; if necessary, in the presence of (C) one or more catalysts; where the ratio of the amount of (A) and (B) is such that the isocyanate index ranges from approximately 95 to approximately 110, the equivalent ratio of NCO to OH in the prepolymer ranges from approximately 2.25:1.0 to approximately 20.0:1.0, and the equivalent ratio of NH 2  to NCO ranges from approximately 0.6:1.0 to approximately 0.95:1.0. In another version, polyurethaneurea, besides the above-mentioned components, contains B)(3) one or more compounds with hydroxyl functional groups, having functionality from approximately 2.0 to approximately 3.0 and molecular weight from approximately 100 to approximately 4000. 
     EFFECT: obtaining optically transparent solid lightfast polyurethaneurea which demonstrates very high shrink resistance at high temperature and does not have creep even in a lower hardness interval. 
     42 cl, 17 ex, 7 tbl
Patent RU-2659796-C9 (RU)
Title: Flexible rotor with constant magnets
Inventor: MIKHAJLOV VALERIJ MIKHAJLOVICH
IPC: H02K1/27
Filed: 2017-09-26
Granted: 2021-12-08
Abstract: FIELD: electrical equipment. 
     SUBSTANCE: invention relates to electrical equipment. Rotor of the electric machine contains a core and radially magnetized permanent magnets of alternating polarity. Rotor is made unit-construction and consists of a pack of magnetic blocks fixed by axial pins and stems. Each of the magnetic blocks is a disk of ferromagnetic (magnetically conductive) material, on the periphery of which are installed and fixed by a bandage, which is a hollow cylinder of a non-ferromagnetic material, magnetized in the radial direction, permanent magnets of alternating polarity. On the ends of the pack of magnetic blocks shafts with bearing necks are installed. 
     EFFECT: increased rotor reliability. 
     1 cl, 2 dwg
Patent RU-2711465-C9 (RU)
Inventor: UILYAMS RODNI OUEN
IPC: A24F40/90
Filed: 2016-10-27
Granted: 2020-11-24
Abstract: Изобретение относится к устройствам доставки аэрозоля. Устройство доставки аэрозоля содержит по меньшей мере один кожух и находящийся внутри указанного по меньшей мере одного кожуха нагревательный элемент, выполненный с возможностью активации и испарения компонентов композиции предшественника аэрозоля при обнаружении прохождения потока воздуха по меньшей мере через часть кожуха, причем воздух пригоден для смешивания с образованным таким образом паром для получения аэрозоля; и специализированную интегральную схему (ASIC), которая содержит системные блоки, выполненные с возможностью реализации соответствующих функций устройства доставки аэрозоля и включающие в себя по меньшей мере: блок управления батареей, выполненный с возможностью управления батареей, выполненной с возможностью питания устройства доставки аэрозоля; интерфейсный блок датчика потока, выполненный с возможностью обнаружения потока воздуха, проходящего по меньшей мере через часть кожуха; и блок возбуждения, выполненный с возможностью вызова активации нагревательного элемента в ответ на входной сигнал от интерфейсного блока датчика потока, который указывает на обнаружение воздушного потока, проходящего по меньшей мере через часть кожуха. Техническим результатом изобретения является создание специализированной интегральной схемы, обеспечивающей более высокий уровень интеграции функциональных возможностей для устройства доставки аэрозоля за счет выполнения различных функций посредством однокристальной интегральной схемы и, таким образом, снижающей производственные затраты. 2 н. и 19 з.п. ф-лы, 9 ил.
Patent RU-2725506-C9 (RU)
Title: Method and system for optimizing laboratory analysis of rock samples
Inventor: Orlov Denis Mikhajlovich
IPC: G01N35/00
Filed: 2019-08-21
Granted: 2020-07-27
Abstract: FIELD: mining; data processing. 
     SUBSTANCE: group of inventions relates to means of optimizing laboratory analysis of rock samples taken from an oil-and-gas bearing formation. Essence: standard laboratory studies of rock samples are performed, the results of which are used to form a database on analysis of formations. Using the obtained results of standard laboratory studies of rock samples as input data, basic predicative models are used to predict missing rock characteristics for each sample using machine learning algorithms. Using as input data obtained results of standard studies of rock samples and results of prediction of missing characteristics of rocks, obtained using basic predictive models, machine learning creates predictive models of the second group to determine corrections to formation conditions and to predict rock characteristics in thermobaric conditions. Using as input data obtained results of rock samples analysis, results of prediction of missing rock characteristics, obtained using basic predictive models, and the results of prediction of rock characteristics in thermobaric conditions, obtained using predictive models of the second group, by means of machine training create predictive models of the third group for prediction of multidimensional characteristics of reservoir rocks. Using all created predictive models, rock characteristics are predicted. All obtained results of forecasting rock characteristics are entered into a database on analysis of formations. Current degree of reservoir study is assessed based on accuracy of obtained prediction results and significance of new investigations is evaluated to increase current degree of study of formation. Based on the evaluation results of the current study of the formation, the program and the volume of laboratory tests of the samples are corrected. System for method implementation comprises base (1) of formation survey data, module (2) for rock characteristics prediction, module (3) for evaluation of formation investigation degree and module (4) for program optimization and volume of laboratory tests of samples, designed to correct program and volume of laboratory studies based on evaluation of current degree of study of formation. 
     EFFECT: technical result: providing fast and high-quality processing of laboratory research results with possibility of scaling these results on entire section of productive deposits of oil-and-gas bearing formation. 
     8 cl, 4 dwg
Patent RU-2723787-C9 (RU)
Inventor: Pateyuk Sergej Andreevich
IPC: B03D1/02
Filed: 2019-11-29
Granted: 2020-12-08
Abstract: FIELD: technological processes. 
     SUBSTANCE: invention relates to chemical processing of gypsum-containing raw materials and man-made wastes, particularly to methods of separating silicon concentrate from boric acid production wastes (borogypsum), which can be used as reinforcing filler of synthetic and polymer materials in tire, rubber, chemical, light and other industries, production of construction materials, as well as gypsum concentrate used in construction industry. Method of borogypsum processing includes repulping of borogypsum to ratio of liquid to solid L:S=4:1, agitation of minerals with flotation reagent for 2–3 minutes, flotation for 8–9 minutes and drying of obtained products. Floatation reagent used is sodium oleyl sarcosinate, which is added in amount of 1 kg/t of borogypsum. Flotation process is carried out at temperature of 30–35 °C in neutral medium. 
     EFFECT: recycling wastes from production of boric acid and their use as technogenic raw material for production of commodity concentrates (gypsum and silicic). 
     1 cl, 1 dwg, 5 ex
Patent DK-7185-D0 (DK)
Inventor: RADVAN BRONISLAW
IPC: B29C67/20
Filed: 1985-01-04
Abstract: A fibre reinforced plastics structure comprising a porous matrix of thermoplastics material and reinforcing fibres, the pores of said matrix being wholly or partly invested with a thermosetting plastics material.
Patent DK-42286-D0 (DK)
Inventor: WRIGHT EARL H
IPC: B05B11/02
Filed: 1986-01-28
Abstract: A device for use with foamable liquids includes a reservoir (13) adapted to contain a quantity of a foamable liquid and an air pump (77) for supplying air to be mixed with the foamable liquid to form a foam. The foamable liquid reservoir is isolated from the air from the air supplying pump. A mixing chamber (53) is provided in which the foamable liquid and air from the air supplying pump can interact to create the foam. A first passage (37,55) leads from the reservoir of foamable liquid to the mixing chamber and a pump (43) is provided for pumping the foamable liquid from the reservoir through the passage to the mixing chamber. A second passage (51) is provided from the air supplying pump to the mixing chamber to introduce air into the mixing chamber.
Patent DK-49893-D0 (DK)
Inventor: PALMASON JON ARNAR
IPC: A22C/
Filed: 1993-04-30
Abstract: Fish to be processed are moved through succesive fish processing stations located along a predetermined path of movement. The path of movement is defined by a pair of transversely spaced guide rails (4) and the free end parts of the guide rails or pins are inserted through the head of the fish. The free end of the guide rails may, for example, be inserted through the eyes and through the tongue of the fish, beneath the lower jaw bone of the head of the fish and out through the mouth of the fish, through the thin skin of the cheeks along the tongue and through the lower jaw of the fish, through the mouth beneath the tongue and out behind the tongue, through the cheeks and out through the mouth of the fish or through the mouth and out behind the tongue and across square bones of the fish.
Patent HU-9300801-D0 (HU)
Title: Dna-sequence resulting male sterility, mitochondrial genom nucleus genom, mitochondrion and plant containing such sequence as well as method for producing said hybrides
Inventor: BONHOMME SANDRINE
IPC: C12Q1/68
Filed: 1991-09-20
Abstract: Ogura sterility DNA (I) is carried by a DNA sequence defined by nucleotides 928-2273 of a 2428 base sequence reproduced in the specification. When present in mitochondrial or nuclear genome of a plant it confers cytoplasmic male sterility (CMS). Also included are sequences with at least 50% homology with (I). Also new are (1) recombinant plant nuclear and mitochrondrial genome contg. a DNA sequence defined by nucleotides 928-1569 of the specified sequence (or its homologues); (2) cytoplasm contg. sucha as mitochrondrial genome; (3) Brassica plants or hybrids contg. (I); (4) DNA probes of at least 10 bases form the 928-1569 sequences.
Patent DK-110891-D0 (DK)
Inventor: BLOOM JOY S
IPC: C08G14/00
Filed: 1991-06-11
Abstract: A thermoformable polyaryletherketone sheet of a thickness of about 625-5000 micrometers, having repeating units derived from diphenyl ether and terephthalyl and isophthalyl groups, especially a polyetherketoneketone in which the terephthalyl to isophthalyl isomer ratio is about 70:30 to 0:100, especially 60:40 to 50:50, which thermoformable sheet has a crystallinity of 5% of less, can be fabricated into three-dimensional articles such as, e.g., panels and ducts for aircraft interiors having good formability and mold replication.
Patent DK-131193-D0 (DK)
IPC: D21C5/00
Filed: 1993-11-23
Abstract: PCT No. PCT/DK94/00437 Sec. 371 Date May 15, 1996 Sec. 102(e) Date May 15, 1996 PCT Filed Nov. 23, 1994 PCT Pub. No. WO95/14807 PCT Pub. Date Jun. 1, 1995In the production of pulp and paper from starch-coated paper, the deinking effect can be improved by including a treatment with a starch-degrading enzyme e.g. amylase or a debranching enzyme. The process comprises enzyme treatment before, during or after disintegration of the paper to produce pulp, followed by separation of ink particles.
Patent DK-184985-D0 (DK)
Inventor: EDWARDS PHILIP NEIL
IPC: C07D233/64
Filed: 1985-04-25
Abstract: A phenol derivative of the formulawherein NU is a defined bis-phenolic nucleus including a hydroxyphenyl-hydroxynaphthyl; hydroxyphenyl-hydroxyin- danyl, hydroxyphenyl-hydroxybenzothienyl or di-hydroxyphenyl-ethylene or vinylene nucleus; wherein A is alkylene, alkenylene or cycloalkylene which is interrupted by a heterocyclene linkage, wherein R<sup>1</sup> is hydrogen, or alkyl, alkenyl, cycloalkyl, halogenoalkyl, aryl or arylalkyl, or R is joined to R<sup>2</sup>, and wherein X is -CONR<sup>2-</sup>, -CSNR<sup>2-</sup>, -NR<sup>12</sup>CO-, -NR<sup>12</sup>CS-, -NR<sup>12</sup>CONR<sup>2</sup>-,-SO<sub>2</sub>NR<sup>2</sup>- or -CO-, or, when R<sup>1</sup> is not hydrogen, is -NR<sup>12</sup>COO-, -S-, -SO- or -S0<sub>2</sub>-, wherein R<sup>2</sup> is hydrogen or alkyl, or R<sup>1</sup> and R<sup>2</sup> together form alkylene; wherein R<sup>12</sup> is hydrogen or alkyl, and wherein R<sup>22</sup> is hydrogen, cyano or nitro; or a salt thereof when appropriate. The compounds possess antioestrogenic activity and may be used for the treatment of hormone-dependent breast tumours or of anovulatory infertility.
Patent DK-476988-D0 (DK)
Inventor: ROSE DAVID
IPC: A61K8/41
Filed: 1988-08-26
Abstract: The composition contains oxidation dye precursors in a vehicle and, besides customary developer substances, coupler compounds of the formula I 
<IMAGE>
 or the salts thereof. The compounds are suitable as red couplers for developer substances of the 2,4,5,6-tetraaminopyrimidine type or derivatives thereof.
Patent DK-480487-D0 (DK)
Inventor: NEWKIRK MARC S
IPC: C04B35/65
Filed: 1987-09-15
Abstract: A method for producing an alumina of high purity, which comprises forming an oxidation reaction product of an aluminum parent metal and an oxygen-containing vapor-phase oxidant, comminuting the resultiang ceramic body, and leaching any non-alumina materials therefrom, and recovering said substantially pure alumina material.
Patent DK-516687-D0 (DK)
Inventor: GOODE HENRY CLAUDE
IPC: C03B3/00
Filed: 1987-10-01
Abstract: A pulverulent batch stream is fed into a liquefying vessel by means of an angled feed tube so as to direct the stream tangentially onto side wall portions. The tube may be rotated so as to change the location onto which the batch stream is impinged.
Patent DK-649789-D0 (DK)
Inventor: GUPTA PRAMOD
IPC: C08K5/13
Filed: 1989-12-20
Abstract: The present invention relates to a method for stabilizing a polyether polyol having a molecular weight of from about 300 to about 10,000 comprising adding 3,5-di-tert-butyl-4-hydroxyphenylpropionic acid as an antioxidant stabilizer, optionally in combination with other antioxidants, to said polyether polyol. This invention further relates to polyols stabilized by the method of this invention and to stabilized polyurethanes prepared from such stabilized polyols.
Patent IT-9002952-D0 (IT)
Inventor: CARRARA SERGIO
IPC: F16J15/22
Filed: 1990-10-23
Abstract: A compound for making packing seals (4) comprises a plurality of yarns (3) braided together and consisting of twisted spinning of pieces of different and random lengths of stainless steel filaments (1) and filaments of other materials (2) such as carbon, pure graphite, aramidic fibers and others. The technique used comprises an action of tear spinning or intermittant twisting and traction on said filaments (1). <IMAGE>
Patent NO-862552-D0 (NO)
Inventor: KASAI KAZUMI
IPC: A44B19/36
Filed: 1986-06-25
Abstract: A bottom-end-stop assembly for a slide fastener comprises a pair of intercoupling male and female members (1), (2) of thermoplastic synthetic resin adapted to be molded on adjacent bottom ends of opposed fastener stringers (19), (20). The male member (1) has an inner longitudinal projection (5) and a pivot pin (6). The female member (2) has an inner longitudinal groove (8) receptive of the projection (5), and an inwardly opening support hole (10) receptive of the pivot pin (6) for pivotal movement of the male member (1). The male member (1) has at least one aperture (4) in the projection (5) so that the stringer tape (19) is clamped between a pair of mold members (22), (23) so as not to become wavy during the molding. The male member (1) also has on opposite surfaces a pair of reinforcing ridges (7), (7) remote from the inner longitudinal side of the male member (1).
Patent NO-883763-D0 (NO)
Inventor: BEACHEY EDWIN H
IPC: C12N15/31
Filed: 1988-08-23
Abstract: Non-virulent bacteria are disclosed into which have been cloned heterologous nucleotide sequences encoded for the expression of Streptococcal M protein antigens, which are effective to elicit opsonic antibodies against Streptococcal infections. These bacteria are useful for vaccination against Streptococcus pyogenes bacteria.