baber/WOPTO huggingface dataset:
Patent BG-65277-B1 (BG)
Title: Cyclothiocarbamate derivatives as modulators of progesterone receptors
Inventor: ZHANG PUWEN
IPC: A61P15/00
Filed: 2001-11-02
Abstract: The invention relates to compounds which are agonists of the progesterone receptor and have a structure (I), wherein R1 and R2 are independent substituents selected from the group consisting of H, optionally substituted C1 to C6 alkyl, alkenyl, alkynyl, or alkynyl groups C3 to C8 cycloalkyl, aryl, substituted aryl, or heterocyclic groups, or CORA, or NRBCORA; or R1 and R2 are fused to form an optionally substituted 3 to 8 membered spirocyclic alkyl or alkenyl ring, or a spirocyclic ring containing one to three heteroatoms selected from the group consisting of O, S and N; RA is selected from the group consisting of H, amino, or optionally substituted C1 to C3 alkyl, aryl, C1 to C3 alkoxy, or C1 to C6 aminoalkyl groups; RB is H, C1 to C3 alkyl, or substituted C1 to C3 alkyl; R3 is H, OH, NH2, CORC, or optionally substituted C1 to C6 alkyl, C3 to C6 alkenyl, alkynyl, or alkynyl groups; RC is substituted by H, optionally substituted C1 to C3 alkyl, aryl, C1 to C3 alkoxy, or C1 to C3 aminolkyl groups; Q1 is S, NR7; or CR8R9, R5 is an optionally trisubstituted benzene ring, or optionally substituted five or six membered heterocyclic ring with 1, 2 or 3 ring heteroatoms selected from the group consisting of O, S, SO, SO2, or NR6. The invention relates also to pharmaceutically acceptable salts thereof, as well as to the use of such compounds for the preparation of medicines for contraception and for the treatment of progesterone-related maladies.
Patent BG-66576-B1 (BG)
Title: Grinding body
Inventor: PENCHEV TODOR
IPC: B02C17/20
Filed: 2010-10-13
Abstract: The present invention relates to a grinding body for crushing and grinding of ores, rock or earth mass, inert or any other materials, in drums and other mills. It is used in the enrichment of ores, production of construction materials, waste treatment and in other industries. The grinding body is a spheroidal cone (1) whose generating arc (5) is the result of a circle or another geometric curve and peak (6) and base (2), which is part of a sphere or another volumetric figure formed by the rotation of geometrical curves and an edge (4) between them. In one version the cone (1) and the base (2) are interconnected via a cylinder (9). For better manufacturability in elaborating the body, on the surface of the base (2), a flat spot (3) is formed, of circular or of another form. In another version the flat spots (7, 8) are located on the surface of the cone (1) and on the surface of the cylinder (9) between the base (2) and the cone (1). In the next version, the tip (6a) of the cone (1) is flat-sloped by a plane, perpendicular or inclined towards the axis of the body. In other versions, between the cone (1) and the base (2) there are more or less convex peripheral rings (10, 11, 12), whose cross-section is of a from close to a circle, triangle or rectangle. In a next version, on the base (2) and on the flat-sloped tip (6a) there are short cylinders (13) protruded, with flat fronts (14). All edges and the vertex of the body can be rounded along a part of a circle, spiral or another geometric shape. The grinding body has a larger surface than the spherical grinding bodies and a greater density in a specific volume, and the presence of an edge and vertex allows increasing the grinding productivity.
Patent BG-67128-B1 (BG)
Title: Acoustic fiber optic sensor system
Inventor: STOYANOV DIMITAR
IPC: G01D5/353
Filed: 2016-06-08
Abstract: The invention relates to an acoustic fiber optic system, in which the acoustic sensor can be located over long distances (10-20 km or more) from the transceiver unit, which along with the information processing and data interpretation unit form the acoustic monitoring system for marine and ground areas. The connection of the acoustic sensor to the transceiver unit is performed entirely (all optical) via an optic cable without the need to supply electrical energy to the remote acoustic sensor. High sensitivity is achieved with the use of coherent detection, and the required efficiency is ensured by accurate aligning of the optical paths in the reference and signal channels. These are prerequisites for the realization of remote monitoring systems with remote sensors. It is shown that the coherence length of the laser source may be smaller than the distance between the transceiver unit and the acoustic sensor. This allows, by appropriate choice of a laser with a certain length of coherence, to create unique multiplexed networks of a large number of remote independent acoustic sensors while maintaining the high quality of coherent detection. Various embodiments of the invention have been described which allow for the implementation of flexible approaches, both in the construction of the acoustic monitoring systems and in the choice of the sensor arrangement of the sensor elements depending on the particular environment. The marine aquatory monitoring systems based on the proposed invention can be applied to simultaneously monitor a large number of water surface and underwater moving objects via the acoustic noises they make. The latter can be directly controlled by an operator combined with powerful computer signal processing, whereby maximum performance can be ensured in the functioning of the monitoring systems.
Patent CH-715597-B1 (CH)
Title: Gasturbomaschine, insbesondere Radialgasturbomaschine, mit einer Berstschutzvorrichtung.
Inventor: BORIS THASER
IPC: F01D25/24
Filed: 2019-10-24
Abstract: Die Erfindung betrifft eine Gasturbomaschine (10), insbesondere Radialgasturbomaschine, mit einer Berstschutzvorrichtung (1) und mit einem Turbinengehäuse (20), das ein in dem Turbinengehäuse (20) drehbar angeordnetes Turbinenrad (21) vollumfänglich umfasst, wobei die Berstschutzvorrichtung (1) als Einsatzstück ausgebildet ist und um eine zentrale Achse (A) in Umfangsrichtung ringförmig an der Turbinengehäuseinnenwand (22) angeordnet ist, um das Turbinenrad (21) zumindest teilweise zu umgreifen, wobei die Berstschutzvorrichtung (1) wenigstens eine/n erste/n Aussparung/Hohlraum (2) aufweist, wobei diese/r Aussparung/Hohlraum (2) in der Berstschutzvorrichtung (1) so ausgebildet ist, dass die kinetische Energie von Bruchstücken des Turbinenrads (21) bei dessen Zerbersten durch die Berstschutzvorrichtung (1) aufgrund plastischen Verformens im Bereich der/des Aussparung/Hohlraums (2) aufgenommen wird und dazu die/der erste Aussparung/Hohlraum (2) einseitig in Richtung des Turbinengehäuses (20) geöffnet ist.
Patent CH-713285-B1 (CH)
Title: Temporärer Landeplatz.
Inventor: RICHARD STEGER
IPC: E04F15/02
Filed: 2016-12-23
Abstract: Es wird ein temporärer Landeplatz (10') für Hubschrauber, umfassend mindestens zwei verlegbare faserverstärkte Kunststoffplatten (1e-1l), sowie Verbinder zum lösbaren Verbinden von benachbarten Kunststoffplatten 1e-1l) beschrieben. Die Kunststoffplatten (1e-1l) weisen jeweils einen inneren Bereich und einen umlaufenden, äusseren Bereich auf. Der innere Bereich weist regelmässige Positiv- und Negativerhebungen auf. Der äussere Bereich weist erste und zweite Überlappungsbereiche auf, welche sich jeweils entlang zwei Rändern der Kunststoffplatte ( 1e-1l) erstrecken und Öffnungen zur Aufnahme der Verbinder aufweisen, wobei der erste Überlappungsbereich gegenüber dem zweiten Überlappungsbereich um mindestens eine Dicke der Überlappungsbereiche versetzt ausgebildet ist. Die ersten bzw. zweiten Überlappungsbereiche einer Kunststoffplatte (1e-1l) sind jeweils mit zweiten bzw. ersten Überlappungsbereichen) einer benachbarten Kunststoffplatte (1e-1l) derart in Überlappung gebracht, dass die Öffnungen fluchten und die Verbinder jeweils mit zwei fluchtend überlappenden Öffnungen form -und/oder kraftschlüssig in Eingriff gebracht sind.
Patent CU-24307-B1 (CU)
Title: Válvula dosificadora
Inventor: BODET HERVÉ
IPC: B65D83/54
Filed: 2014-01-14
Abstract: <p>La invención se refiere a una válvula dosificadora para un recipiente de aerosol, que tiene una cara interna destinada a colocarse en el interior del recipiente de aerosol y una cara externa destinada a colocarse en el exterior del recipiente de aerosol. La válvula está provista de</p> <p>- un cuerpo de válvula que tiene una cámara interna (17) capaz de ponerse en contacto o bien con la cara interna de la válvula o con la cara externa de la válvula,</p> <p>- un vástago (41) provisto de medios de cierre (42) y colocado parcialmente en el interior de la cámara interna (17) capaz de moverse entre dos posiciones, a saber, una posición cerrada en la que la cámara interna está en contacto con la cara interna de la válvula, pero aislada de la cara externa de la válvula, y una posición abierta en la que la cámara interna está en contacto con la cara externa de la válvula pero aislada de la cara interna de la válvula,</p> <p>- un depósito (R) que puede llenarse cuando el vástago está en la posición cerrada y vaciarse cuando el vástago está en la posición abierta.</p> <p>De acuerdo con la invención, el depósito está localizado en el lado de la cara interna de la válvula, en el exterior del cuerpo de válvula, el depósito está en contacto con la cámara interna del cuerpo de válvula, y el depósito está formado por al menos una membrana flexible (2).</p> <p>Figura para el resumen: figura 2</p>
Patent EP-1067193-B1 (EP)
Inventor: KREUTZER CAROLINE
IPC: C07K14/34
Filed: 2000-07-06
Granted: 2005-10-19
Abstract: New L-lysine producing coryneform bacteria (A) contain amplified pyc (pyruvate carboxylase) and dapA (dihydrodipicolinate) genes, where the promoter of the dapA gene contains the mutation MC20 or MA16 (as shown in respective sequences of 79 or 80 bases given in the specification as SEQ-ID-NO: 5 and SEQ-ID-NO: 6). (A) optionally also contains amplified lycC, lysE and/or dapB gene(s). An independent claim is included for the preparation of L-lysine by fermentation of coryneform bacteria having an amplified pyc gene, where the bacteria additionally contain the amplified dapA gene as specified for (A).
Patent EP-1042952-B1 (EP)
Inventor: VAN DER LELY CORNELIS
IPC: A01K11/00
Filed: 1994-08-05
Granted: 2003-10-29
Abstract: A construction for automatically milking animals, such as cows, comprising a milking box (2) and a milking robot (19). The construction includes two boxes (1, 2) which are contiguous to each other via their ends, the first (1) of these boxes being arranged for selecting and/or supplying animals with concentrate and the second (2) being arranged as milking box. <IMAGE>
Patent EP-1099829-B1 (EP)
Inventor: KESS ROLAND
IPC: F01N1/02
Filed: 2000-11-09
Granted: 2006-01-25
Abstract: The inlet (6) of the silencer (1) has a tapered reducing piece (4,5) leading into the perforated tube (2). The concentric space (8) between the inner and outer tubes acts as an expansion chamber. Some of the exhaust gases flow through the perforations and are released to the outside through vanes (17) at the outlet (19) end of the silencer. There may be a large-diameter pipe surrounding these vanes. The vanes are made by bending the edges of discs (14) which have openings (11,18) in them to allow exhaust gases to flow through.
Patent EP-1109346-B1 (EP)
Inventor: ARTUN BERKAN
IPC: H04L1/22
Filed: 2000-12-12
Granted: 2007-11-07
Abstract: Detection and handling of transmission errors occurring on a bus system with several stations during access contention can lead to discontinuation of data transmission unless a redundant bus-system can be brought into use and switched over in order to continue data transmission via the bus system, thus resulting in adaptive error detection and corresponding correction. Improved detection and handling of erroneous data results when several stations (14-17) connected to the bus-system (18) send a test pattern which recognizes when a further access contention is carried out, and where each station wishing to send the test pattern is allowed to take part in the following access contentions at different times.
Patent EP-1072407-B1 (EP)
Inventor: FUKUMORI HIROTSUGU
IPC: B41F9/00
Filed: 2000-07-26
Granted: 2005-05-25
Abstract: A photogravure printing method and machine for printing films (7) uses a water based ink and avoids customary problems associated with wetting of the plate, bleed, fogging and drying by using a printing drum (3) having between 200 and 400 mesh lines with a depth between 10 and 17  mu . Left-over ink may be reduced by having an ink reservoir formed with a trough (4) into which the inking roller (2) dips the trough (4) being associated with a drip tray (1a) located beneath the printing drum (3). Printing may be improved further by using a doctor blade assembly (5) having two blades of differing resilience. In a modification two inking rollers are used in spaced relationship at the lower part of the printing drum.  <IMAGE>
Patent EP-1069052-B1 (EP)
Inventor: BETHUNE ALAIN
IPC: B65D41/04
Filed: 2000-07-12
Granted: 2003-05-21
Abstract: The bottle has a threaded neck which is covered by a top which consists of an inner seal cap and an outer trim cap (6) fixed to it. The bottle is made with a projecting stop adjacent to its neck, and the outer cap has at least one inner surface (30) shaped to engage with it to position the cap symmetrically with the bottle when closed. The shaped inner surface (30) of the cap is formed in the thickness of a tubular skirt (22) made in one piece with the outer cap and designed for fixing it to the inner seal cap. The skirt's lower edge is covered by a metal ring (12).
Patent EP-1152843-B1 (EP)
Inventor: MORPHY GARY EARLE
IPC: B21D41/02
Filed: 2000-02-08
Granted: 2003-01-22
Abstract: A method and apparatus for sealing the net shape of the end of a final product tube to eliminate or minimize scrap for a wide range of shapes of the end of the product. A sealing tool has a neck, and a coining portion comprising a shoulder extending outwardly from the neck. The sealing tool is inserted into the deformed end of the tube while the end is being laterally engaged by a clamp pressing inwardly against the outer surface of the tube. The end is then sealed by coining a surface of the tube by axially pressing the sealing tool into the end while laterally inwardly pressing the end with the clamp.
Patent EP-1177217-B1 (EP)
Inventor: AUZELY-VELTY RACHEL
IPC: A61K47/48
Filed: 2000-04-26
Granted: 2004-10-13
Abstract: The invention provides cyclodextrin derivatives that may be used to transport hydrophobic molecules for pharmaceutical or cosmetic applications, by forming organised systems in an aqueous medium, alone or with phospholipids. The cyclodextrin derivatives of the present invention have the formula:in which, R<1 >represents a steroid, R<2 >represents an alkyl or aryl group, substituted if applicable, R<3 >represents H or R<2>, all the R<4 >represent OR<2>, or one of the R<4 >represents -NHCO(CH2)mCONHR<1>, m is an integer ranging from 1 to 8, and n is equal to 5, 6 or 7.
Patent EP-1173448-B1 (EP)
Inventor: YUNLU KENAN
IPC: C07F9/02
Filed: 2000-04-25
Granted: 2004-02-25
Abstract: Stable rare earth tris (organophosphate) solutions comprise a rare earth tris (organophosphate) and a hydrocarbon solvent. From about 2 % to about 10 % rare earth element, preferably from about 3 % to about 8 %, is present in the solutions. The rare earth tris (organophosphate) solutions are stable from precipitation of the rare earth tris (organophosphate) for at least about fifteen (15) days, preferably for at least about twenty (20) days and most preferably at least about thirty (30) days. A process for preparing these solutions is described herein. A stabilizing additive, acid, glycol or mixtures thereof, is utilized to inhibit precipitation. The molar ratios of free acid, glycol and/or water to the rare earth element are controlled to inhibit precipitation.
Patent EP-1144124-B1 (EP)
Inventor: FOSTER PETER D
IPC: B05C13/02
Filed: 2000-05-09
Granted: 2008-01-23
Abstract: A process and an apparatus are disclosed for coating at least one surface of an article such as a paper plate with a liquid coating. The surface to be coated is passed through a wave of liquid coating, such as an aqueous dispersion, followed by removal of the excess coating. The coating and coating removal steps are carried out in an environment which is vaporous with the vehicle of the liquid coating, which prevents premature drying of the coating and allows for a smooth, even application of the coating to the surface.
Patent EP-1186054-B1 (EP)
Inventor: THORNTON TREVOR J
IPC: H01L29/76
Filed: 2000-05-31
Granted: 2003-11-12
Abstract: Various emdodiments include a transistor device that is controlled by a gate current and that exhibits low power consumption as well as high speed characteristics. In various embodiments, an enhancement mode MESFET device exhibits channel drain current that is controlled by the application of bias current into the gate. Complementary n- and p-channel devices can be realized for, for example, micropower analog and digital circuit applications.
Patent EP-1209262-B1 (EP)
Inventor: FUJIMOTO KATSUHIRO
IPC: D01F6/92
Filed: 2000-07-12
Granted: 2006-11-02
Abstract: A polytrimethylene terephthalate fiber, a method for producing the same, a cheese-shaped package formed thereof, a false-twist textured yarn using the fiber and a fabric using the false-twist textured yarn are provided. The fiber is composed of 90 mol% or more of trimethylene terephthalate repeating units having a density in a range from 1.320 to 1.340 g/cm<3>, a birefringence in a range from 0.030 to 0.070, a peak value of thermal stress in a range from 0.01 to 0.12 cN/dtex, a boiling water shrinkage in a range from 3 to 40%, and an elongation at break in a range from 40 to 140%. The inventive polytrimethylene terephthalate fiber has both of proper crystallinity and orientation and is free from the package tightness due to yarn shrinkage and the bulge. The inventive fiber can be produced on an industrial scale.
Patent EP-1220892-B1 (EP)
Inventor: LIAO JAMES C
IPC: C12P7/02
Filed: 2000-07-27
Granted: 2008-02-13
Abstract: The invention features a method of producing heterologous molecules in cells under the regulatory control of a metabolite and metabolic flux. The method can enhance the synthesis of heterologous polypeptides and metabolites.
Patent EP-1202964-B1 (EP)
Inventor: ROFFEY JONATHAN RICHARD ANTHON
IPC: C07D491/04
Filed: 2000-08-04
Granted: 2005-10-12
Abstract: Cette invention a trait à un composé chimique correspondant à la formule (I) dans laquelle R1 et R2 sont choisis de manière indépendante entre un hydrogène et un alkyle, R3 représente un alkyle, R4 et R5 sont choisis entre un hydrogène et un alkyle, R6 et R7 sont choisis, de manière indépendante, dans le groupe constitué par un hydrogène, un halogène, un hydroxy, un alkyle, un aryle, un amino, un alkylamino, un dialkylamino, un alcoxy, un aryloxy, un alkylthio, un alkylsulfoxyle, un alkylsulfonyle, un nitro, un carbonitrile, un carbo-alcoxy, un carbo-aryloxy et un carboxyle, et A représente un noyau à 5 ou 6 chaînons contenant éventuellement un ou plusieurs hétéroatomes, les atomes du noyau A, autres que des atomes de carbone insaturés du noyau phényle avec lequel fusionne le noyau A, sont saturés ou insaturés. L'invention concerne également les sels acceptables du point de vue pharmaceutique de ce composé, ses composés d'addition ainsi que se promédicaments. Elle porte, en outre, sur l'usage qui en est fait en thérapeutique, notamment en tant qu'agoniste ou antagoniste du récepteur 5HT, en particulier du récepteur 5HT2C, par exemple dans le traitement de troubles du système nerveux central, de dégâts occasionnés au système nerveux central, de troubles cardio-vasculaires, de troubles gastro-intestinaux, du diabète insipide, ainsi que de l'apnée du sommeil et tout particulièrement dans le traitement de l'obésité.
Patent EP-1214108-B1 (EP)
Title: Prothese poreuse et procede de depot de substances dans les pores
Inventor: HOSSAINY SYED F A
IPC: A61L31/14
Filed: 2000-08-23
Granted: 2007-01-10
Abstract: La présente invention concerne une prothèse implantable, par exemple une endoprothèse vasculaire, que l'on peut remplir de substances destinées à une application ultérieure sur des tissus biologiques. Dans une réalisation, la prothèse possède un corps de forme cylindrique comportant une formation de dépôts ou de pores. Les dépôts peuvent être formés à des emplacements présélectionnés sur le corps de la prothèse et peuvent présenter une profondeur, une taille et une forme présélectionnées, y comprise cylindrique ou conique. De substances telles que des substances thérapeutiques, des matériaux polymériques, des matériaux polymériques contenant des substances thérapeutiques, des isotopes radioactifs, et des matériaux de contraste peuvent être déposés dans ces dépôts. L'invention concerne aussi un procédé de chargement d'une substance dans la prothèse contenant des dépôts ou des pores. Un premier fluide en combinaison avec une substance ajoutée est appliqué à la prothèse poreuse. Lors de l'application, le premier fluide contenant la substance peut pénétrer dans les pores de la prothèse. Le premier fluide est éliminé et un deuxième fluide est appliqué à la prothèse. Le deuxième fluide n'est pas capable de pénétrer sensiblement dans les pores. Avant l'application du deuxième fluide, la prothèse peut être immergée dans un troisième fluide et agitée au moyen de techniques mécaniques de perturbation de façon à ce qu'aucune quantité de substance amassée sur la surface du corps, après application du premier fluide, soit éliminée. Le troisième fluide ne doit pas pouvoir dissoudre la substance.
Patent EP-1214369-B1 (EP)
Title: Solution ou dispersion aqueuse d'un sel acide de polyetheramine
Inventor: SCHMIDT DALE C
IPC: C08J3/03
Filed: 2000-09-01
Granted: 2005-05-18
Abstract: La présente invention concerne une solution et une dispersion aqueuse stable d'un sel acide de polyéthéramine, qui peuvent être préparées par la neutralisation au moins partielle de la polyéthéramine avec un acide. Cette solution et cette dispersion sont utiles sous forme de revêtement, en particulier dans des applications où il convient de disposer d'une barrière contre les petites molécules.
Patent EP-1238156-B1 (EP)
Inventor: TORVI TIMO
IPC: D21G1/00
Filed: 2000-11-01
Granted: 2004-06-02
Abstract: Higher-gloss paper grades, in particular paper grades with a Hunter gloss % above 40, are produced in an arrangement having pairs of calendering units ( 1, 3 ) disposed in the machine direction one after the other and apart from one another, which pairs are each formed of separate and different calendering units ( 1, 3 ) and in each of which the nip load in the latter calendering unit ( 3 ) is higher than the nip load in the preceding calendering unit ( 1 ). Advantageously, the calendering unit ( 1 ) placed first in the machine direction is an on-line long-nip calendering unit ( 1 ) and the calendering unit ( 3 ) placed after that in the machine direction is an on-line or off-line supercalender.
Patent EP-1216286-B1 (EP)
Inventor: DE LIMA PFX
IPC: C10B29/00
Filed: 2000-07-17
Granted: 2010-09-15
Abstract: This invention comprises a complete arrangement of ovens, underflues, cooling air ducts under the oven, the feeder flue, to control dampers in the feeder flues, the common flues, the charge car operating over the ovens the ram car operating on one side of the ovens and the hot coke car operating on the other side of the ovens, the oven doors, the door opening/closing mechanism, the coal bin tower with the weighbridge, the quench tower and the feed of the flue gases to boilers of the power plant. The oven is a specially designed structure made of various qualities and shapes of refractory bricks designed to withstand the high temperatures. The combustion is controlled by allowing air in and the hot waste gases are led to a common flue refractory lined inside to withstand the high temperature. The waste gases are led to the boiler for producing steam and electric power in a turbine/generator for energy recovery or alternatively led to an oven stack of sufficient height to maintain a draft in the oven to sustain the coking process.