baber/WOPTO huggingface dataset:
Patent EA-015444-B1 (EA)
Title: Process for the coating of polymer particles and
Inventor: BREMER LEONARDUS GERARDUS JACOBUS
IPC: C08J7/043
Filed: 2006-09-26
Abstract: Process for the coating of polymer particles, comprising contacting the particles with a composition comprising an additive, a film-forming binder that is miscible with the polymer, and a distributing agent, removing the distributing agent at a particle temperature at which the binder can form a film and that is below the softening temperature Tof the polymer, and forming and consolidating an additive-containing layer of binder on the polymer particles, the polymer particles being kept in mutual motion while they are being contacted with the composition and while the additive-containing layer of binder is being formed and consolidated. The binder is miscible with the polymer if it satisfy the followings. Equal amounts of polymer and dried binder are mixed in the melt in a kneader or extruder. A sample of the resulting mixture is placed in a standard DSC pan and heated in a DSC apparatus at a heating rate of 10°C per minute. If a single glass transition temperature peak is visible in the heating curve, situated between the corresponding values of the binder and the polymer by themselves, then the binder is considered to be miscible with the polymer or a mixture of a quantity of a dispersion or solution of the binder as intended for use in the process with an equal amount of polymer powder is heated to Tin a DSC apparatus, with evaporation of the distributing agent. Binder and polymer are also considered to be miscible in the framework of the invention if the glass transition temperature of the binder, as measured in the second heating curve, has been increased due to the heating together with the polymer by at least 5% of the difference between the values of the glass transition temperature of the binder and the polymer by themselves. An additive-containing polymeric objects, in which polymer particles coated according to the above-mentioned process are processed at a temperature that lies above the melting point of the polymer.
Patent EA-015526-B1 (EA)
Title: Antagonist antibodies directed against calcitonin gene-related peptide and methods using same
Inventor: ZELLER JOERG
IPC: A61K39/395
Filed: 2006-11-02
Abstract: The invention features methods for preventing or treating CGRP associated disorders such as vasomotor symptoms, including headaches (e.g., migraine, cluster headache, and tension headache) and hot flushes, by administering an anti-CGRP antagonist antibody. Antagonist antibody G1 and antibodies derived from G1 directed to CGRP are also described.
Patent EA-012930-B1 (EA)
Title: Selective vpac2 receptor peptide agonists
Inventor: BOKVIST BENGT KRISTER
IPC: C07K14/575
Filed: 2006-10-24
Abstract: The present invention encompasses peptides that selectively activate the VPAC2 receptor and are useful in the treatment of diabetes.
Patent EA-015991-B1 (EA)
Title: Template-fixed peptidomimetics
Inventor: GOMBERT FRANK
IPC: A61K38/04
Filed: 2007-01-15
Abstract: Template-fixed β hairpin peptidomimetics of the general formulawhereisPro-Pro orPro-Pro; and Z is a template-fixed chain of 12 α- amino acid residues, which, depending on their positions in the chain (counted starting from the N-terminal amino acid), wherein said amino acid residues in positions P1-P12 areand salts thereof, have the property to selectively inhibit the growth of or to kill microorganisms such as Pseudomonas aeruginosa. They can be used as disinfectants for foodstuffs, cosmetics, medicaments or other nutrient-containing materials, or as medicaments to treat or prevent infections. These β-hairpin peptidomimetics can be manufactured by processes which are based on a mixed solid- and Solution phase synthetic strategy.
Patent EA-016073-B1 (EA)
Title: A composition for inactivating an enveloped virus (variants), composition based thereon for preparing a medicament against virus disease, for preparing pharmaceutically amount of biocompatible disinfectant and for preparing coating agent comprising a kit for inactivating an enveloped virus and method therefor
Inventor: PELET THIERRY
IPC: A61K9/127
Filed: 2007-05-18
Abstract: The present invention relates generally to the field of prevention of diseases caused by enveloped viruses. More particularly, this invention concerns a composition for inactivating an enveloped virus comprising at least one non phospholipid Lipid Vesicle (nPLV) able to interact with said enveloped virus and an agent that enhances the lipid exchange between said nPLV and the membrane of said enveloped virus.
Patent EA-021050-B1 (EA)
Title: Synergistic preservative blends
Inventor: NUNEZ ROSITA
IPC: A61Q17/00
Filed: 2009-05-20
Abstract: The present invention discloses a preservative formulation comprising the combination of at least two compounds having bactericidal and/or fungicidal properties, wherein the respective combination is selected from the group consisting of methylisothiazolinone/piroctone olamine; caprylyl glycol/dehydroacetic acid and lauryl alcohol/sorbic acid.
Patent EA-020988-B1 (EA)
Title: Method for stripping voltametric determination of platinum in nitrite medium
Inventor: SCHEGLOVA NATALIYA VENEDIKTOVNA
IPC: G01N27/48
Filed: 2012-05-23
Abstract: A method for stripping voltametric determination of platinum in nitrite medium relates to analytical chemistry of platinum metals. Determination of palladium(II) in an analysed solution of a nitrite complex involves a step for its electrochemical reduction on a carbon-containing electrode and then electrochemical stripping of the reduced platinum while plotting the current-voltage curve. Concentration of platinum(II) in the nitrite solution is determined from the value of the anodic peak of electrochemical stripping of preliminarily reduced platinum. The background electrolyte used is 1 M KNOor 1 M HSO. Electrochemical stripping of the reduced platinum is carried out while varying potential of the working carbon-containing electrode at a rate of 50 mV/s and the current-voltage curve is plotted. For a carbon-containing electrode, the range of the determined concentration of platinum(II) is on a 1 M KNObackground - 0.1-2.0 mg/l, 1 M HSO- 0.01-1.00 mg/l. The analytical signal for determining platinum is the height of the anodic peak of its electrochemical stripping on the current-voltage curve in the potential region from 0.10 to 0.45 V. The invention enables to determine concentration of platinum directly in a nitrite medium without sample preparation.
Patent EA-023981-B1 (EA)
Title: Androgen receptor modulators and uses thereof
Inventor: SMITH NICHOLAS D
IPC: C07D487/04
Filed: 2011-02-16
Abstract: Described herein are compounds that are androgen receptor modulators, wherein said compounds correspond to formula (Ia)wherein ring A is pyridinyl, ring B is phenyl, Ris substituted or unsubstituted C-Cheterocycloalkyl attached to phenyl by a binding group, and R, R, R, X, m and n are defined in the claims. Also described are pharmaceutical compositions and medicaments that include the compounds described herein, as well as methods of using such androgen receptor modulators, alone and in combination with other compounds, for treating diseases or conditions that are mediated or dependent upon androgen receptors.
Patent EA-019612-B1 (EA)
Title: Substituted phenyl(oxy/thio)alkanol derivatives
Inventor: NISING CARL FRIEDRICH
IPC: A01N43/54
Filed: 2010-06-25
Abstract: The present invention relates to novel substituted phenyl(oxy/thio)alkanol derivatives, to a method for producing said compounds, to agents comprising said compounds, and to the use thereof as biological active compounds, in particular for combating harmful microorganisms in crop protection and material protection and as plant growth regulators.
Patent EA-026342-B1 (EA)
Title: Water purification device comprising a gravity-fed filter
Inventor: MISTRY MAHENDRAKUMAR MAGANLAL
IPC: C02F1/76
Filed: 2011-08-02
Abstract: The present invention relates to water purification devices, particularly to gravity-fed water purification devices that operate without electricity and pressurised water. The invention relates to a gravity-fed water purification device comprising a chamber (3) that has the sediment filter (6), also has a compartment (7) that surrounds the sediment filter (6). The compartment (7) has sidewalls (16) rising upwardly from bottom of the chamber (3) to define an open top with a rim having a notch (7a). The compartment (7) is spaced apart from the walls of the chamber (3) to define a space around the compartment (7). Preferred devices were surprisingly found to solve the problem of tapering-off of the flow-rate from the device over a period of use, and the need to frequently back wash the carbon block filter (9), particularly under conditions of poor water quality and at the same time provide the required residence time for the chemical purifying agent to act on the pathogens.
Patent EA-023739-B1 (EA)
Title: Cleaner of fibrous material
Inventor: KARIMOV SUNDET SMAKHANOVICH
IPC: D01G9/14
Filed: 2013-02-04
Abstract: The invention relates to textile industry and can be used in machines for cleaning fibrous materials, in particular, raw cotton. In the proposed invention enhancement of cleaning effect is achieved by using rubber T-shaped nozzles inserted into movable splittings with attached rubber rods, having compliance, not exceeding cotton seed and strength of cotton fiber for compression, thus providing to create adaptive conditions of interconnection with raw cotton for preserving seed strength and increasing fiber loosenability aimed at increasing effect of removing trashes from the treated material. The nozzle is provided to have a single-row or multi-row arrangement of rubber rods, wherein bend of working members occurs not only in rubber rods, but also in rubber nozzle itself, thus enhancing cleaning effect.
Patent EA-023932-B1 (EA)
Title: Treatment of vascular hyperpermeability-associated diseases
Inventor: BAR-OR DAVID
IPC: B65D69/00
Filed: 2011-09-07
Abstract: The invention provides a method of inhibiting vascular hyperpermeability in an animal in need thereof. The method comprises administering an effective amount of a diketopiperazine or a pharmaceutically acceptable salt thereof to the animal, wherein the diketopiperazine has the following formula:wherein (a) Ris a side chain of an aspartic acid and Ris a side chain of alanine (DA-DKP); (b) Ris a side chain of methionine and Ris a side chain of arginine (MR-DKP); (c) R1 is a side chain of tyrosine and Ris a side chain of a glutamic acid (YE-DKP).
Patent EA-028396-B1 (EA)
Title: Formulation for the preparation of pharmaceutical fluorocarbon-linked peptide formulation and method for obtaining such formulation
Inventor: BROWN CARLTON BRADLEY
IPC: A61K39/385
Filed: 2011-12-30
Abstract: The invention relates to a visually clear aqueous acidic formulation suitable for use in the preparation of a pharmaceutically acceptable fluorocarbon-linked peptide formulation, which aqueous formulation comprises a) at least one fluorocarbon-linked peptide, wherein i) the peptide linked to the fluorocarbon is at least 20 amino acid residues long, comprises at least 50% hydrophobic amino acid residues and has an isoelectric point greater than or equal to 7; and ii) the fluorocarbon-linked peptide is present in micelles; and b) acetic acid in the concentration of at least 10% (v/v). Also provided is a method for obtaining a pharmaceutically acceptable fluorocarbon-linked peptide formulation. The method comprises solubilising a fluorocarbon-linked peptide in acetic acid to obtain said formulation; filter-sterilising the solubilised fluorocarbon-linked peptide; and drying the filter-sterilised fluorocarbon-linked peptide.
Patent EA-026258-B1 (EA)
Title: Device and process for improved recovery of deionised water
Inventor: ALENCHERRY TINTO JOHNICHAN
IPC: C02F1/469
Filed: 2012-07-18
Abstract: Disclosed is a process for improved recovery of deionised water from a feed water stream, comprising the steps of: (i) delivering the feed water stream in to a capacitive deionisation cell; (ii) measuring the salt concentration of the water exiting the capacitive deionisation cell; (iii) collecting the water exiting the cell, when the salt concentration is lower than a predetermined lower set point, to prepare purified water or rejecting the water exiting the cell when the salt concentration is higher than a predetermined upper set point; wherein the water exiting the cell is recycled with the feed water stream when the salt concentration of the water exiting the cell is between the lower set point and the upper set point. By this process the waste water produced during capacitive deionization can be recycled so as to improve total recovery of water as well as to enhance the life of the electrodes of the capacitive deionisation cell.
Patent EA-027675-B1 (EA)
Title: Urea production process and plant
Inventor: MENNEN JOHANNES HENRICUS
IPC: C07C273/04
Filed: 2013-05-02
Abstract: The invention relates to a plant for the production of urea. The plant comprises conventional sections for synthesis and recovery, for evaporation and condensation, for urea finishing, and for dust scrubbing. According to the invention, the plant also comprises an additional evaporation and condensation recirculating loop comprising and additional evaporation section placed downstream of the dust scrubbing section and being in fluid communication with the finishing section, wherein the additional evaporation section has a gas flow line to an additional condensation section which is in fluid communication with the dust scrubbing section. This recirculating loop results in a more favorable energy consumption of the plant. The invention also relates to a corresponding process for the preparation of urea.
Patent EA-026701-B1 (EA)
Title: Substituted annellated pyrimidines, method of production thereof, use thereof and medicine for treating and/or preventing diseases
Inventor: FOLLMANN MARKUS
IPC: C07D519/00
Filed: 2012-08-30
Abstract: The present application relates to substituted annellated pyrimidines of general formula (I)wherein all the substituents are disclosed in the claims, a method for the production thereof, the use thereof for the treatment and/or prophylaxis of diseases, and also for the use thereof to produce medicines for the treatment and/or prophylaxis of diseases, in particular for the treatment and/or prophylaxis of cardiovascular diseases, and a stimulator of soluble guanylate cyclase which is a compound of formula (I).
Patent EA-036434-B1 (EA)
Title: Method of treating lung cancer using a combination of aurora kinase inhibitor and paclitaxel
Inventor: CHAKRAVARTY ARIJIT
IPC: A61K35/00
Filed: 2013-03-19
Abstract: Disclosed is a method for the treatment of small-cell lung cancer by administering a selective inhibitor of Aurora A kinase alisertib in combination with paclitaxel. A specified dosage regimen allows to use increased alisertib doses with acceptable tolerability without losing efficacy.
Patent EA-028169-B1 (EA)
Title: Method for wear-fatigue tests of materials
Inventor: BOGDANOVICH ALEXANDER VALDEMAROVICH
IPC: G01N3/56
Filed: 2015-06-30
Abstract: The invention is related to the field of wear-fatigue tests of materials and can be used for assessment of operability of mechanical systems involving sliding friction or rolling friction and that take up simultaneously repeatedly varying contactless load. The objective of the invention is performance of cyclic loading of a specimen with simultaneous provision of sliding friction or rolling friction between the specimen and counter-specimens using a single vibration-type force actuator that allows also higher test rate due to higher loading frequency. The set objective is attained by that in the known wear-fatigue test method, the specimen is fixed vertically in the vibrator clamp, a weight of mass m is fastened to the other end of the specimen, counter-specimens in the form of inserts or rollers are pressed to the working surface of the specimen using a dynamometric cramp, and the specimen is imparted, through the clamp, longitudinal oscillations of velocity v and frequency f close to the natural oscillation frequency of the entire mechanical system; masses of the specimen, the weight at its free end and the dynamometric cramp with counter-specimens are selected so as to provide, under cyclic resonance loading, preset levels of the amplitude of normal σ and frictional stresses (specific friction force) τin the dangerous cross-section of the specimen at the appropriate amplitude of reciprocate motion of the counter-specimens relative to the median point located on the line of the initial contact of counter-specimens with the specimen.
Patent EA-032481-B1 (EA)
Title: Progesterone receptor antagonist dosage form
Inventor: SCHUTT BARBARA
IPC: A61P15/00
Filed: 2014-04-09
Abstract: The invention relates to a method for the treatment or prophylaxis of gynaecological diseases, such as fibroids of the uterus (myomas, uterine leiomyoma), endometriosis or excessive menstrual bleeds, that comprises administering a progesterone receptor antagonist, namely (11β,17β)-17-hydroxy-11-[4-(methylsulphonyl)phenyl]-17-(pentafluoroethyl)estra-4,9-dien-3-one at the dosage of about 2 to 4 mg and more particularly 2 mg.
Patent EA-029818-B1 (EA)
Title: Cytotoxic and anti-mitotic compounds, and methods of using the same
Inventor: WINTERS GEOFFREY C
IPC: A61P35/00
Filed: 2014-03-14
Abstract: Compounds having cytotoxic and/or anti-mitotic activity are disclosed. Methods associated with preparation and use of such compounds, as well as pharmaceutical compositions comprising such compounds, are also disclosed. Also disclosed are compositions having the structure (T)-(L)-(D), wherein (T) is a targeting moiety, (L) is an optional linker, and (D) is a compound having cytotoxic and/or anti-mitotic activity.
Patent EA-032627-B1 (EA)
Title: Device for the manual blocking of the wheel of a truck on a lane in front of a facade with a loading and unloading platform
Inventor: STROET FRANCISCUS JOHANNES
IPC: B60T3/00
Filed: 2015-12-04
Abstract: Device for manual locking of the wheel of a truck on a lane in front of a facade with a loading and unloading platform, comprising a guide provided alongside and parallel to the lane, extending from a road side to a facade side, and a carriage movable on the guide, provided with a locking arm that is moveable between a starting position, in which the locking arm extends alongside the lane, and an end position; wherein said device comprises locking means for bringing about a locking of the carriage to the guide, whereby by moving of the locking arm from the starting position to the end position, the locking means are operated.
Patent EA-032160-B1 (EA)
Title: Apparatus and method for laser engraving foodstuffs
Inventor: LEACH JAMES RICHARD HUGHES
IPC: A23G3/34
Filed: 2015-06-02
Abstract: Provided is a wafer product decorating apparatus comprising a laser, a collimator, at least one galvanometer driven mirror, and an aspheric scan lens, the apparatus being positionable relative to the wafer product to be decorated wherein the apparatus is configured to provide a laser beam having a spot size of from 100 to 750 μm in diameter on the surface of the product to be decorated and a substantially flat focal plane, characterised in that the focal plane has a depth of field of from 5 to 20 mm and that the focal plane of the laser beam is from 5 to 30 mm above or below the surface of the product to be decorated. Also provided is a process for decorating a wafer product.
Patent EA-036661-B1 (EA)
Title: Oxaborole esters and method of treating parasitic infection
Inventor: AKAMA TSUTOMU
IPC: C07F5/02
Filed: 2017-05-01
Abstract: The present invention provides oxaborole ester compounds and method of treating parasitic infection using the same, including diseases associated with parasites, such as Chagas Disease and African Animal Trypanosomosis.
Patent EA-039260-B1 (EA)
Title: Wall construction for a building and method for manufacturing same
Inventor: HALLDORSSON HALLDOR GUNNAR
Filed: 2018-01-09
Abstract: A wall construction (1) for a building and a method for manufacturing same are described, the wall construction (1) comprising a wooden structural frame (3), the structural frame (3) comprising at least vertical studs (5) which are fixed, at their end portions, to plates (7) at the top and bottom, and the structural frame (3) constituting at least a portion of a wall that has an external side and an internal side, the external side of the structural frame (3) being provided with a vapour barrier (9). The wall construction (1) may be manufactured by means of at least one module element (10).
Patent ES-2192917-B1 (ES)
Title: Particulas de poliacrilonitrilo obtenidas mediante polimerizacion de surfmer y separacion de sodio por intercambio quimico.
Inventor: WADE BRUCE E
IPC: C08F228/02
Filed: 1999-03-29
Granted: 2005-02-16
Abstract: Partículas de poliacrilonitrilo obtenidas
mediante polimerización de surfmer y separación de sodio por
intercambio químico. 
     La presente invención es una partícula de
polímero  acrílico que es consistente y sustancialmente de  forma
esférica y que tiene un diámetro medio que  puede estar
predeterminado desde aproximadamente  30 micrómetros de diámetro a
aproximadamente 5  micrómetros o menos. El poliacrilonitrilo es
sintetizado en una polimerización en dispersión acuosa con un
monómero iónico o "surfmer" para conseguir una  distribución
estrecha del tamaño de partículas con un diámetro medio tan bajo
como aproximadamente 3+1,5 micrómetros que es característico de una
polimerización en emulsión. El polímero comprende el monómero iónico
y, opcionalmente, un comonómero neutro. El tamaño medio de
partículas depende de  la concentración del monómero iónico
presente, del monómero o monómeros iónicos particulares
seleccionados y del contraión asociado con los monómeros  iónicos,
el iniciador de persulfato y el activador de bisulfito. Los
contraiones, a menudo iones de sodio, pueden ser separados de las
partículas de polímero  por intercambio iónico con compuestos de
amonio cuaternario.
Patent ES-2199010-B1 (ES)
Inventor: GALAN VALIENTE MIGUEL
IPC: G02B7/02
Filed: 2001-02-06
Granted: 2005-05-01
Abstract: This device includes: an outer ring (1) provided with: a truncated cone-shaped inner surface (11), one or more wedges (2) provided with an inner surface (22) designed to exercise pressure on the glass (3) to be immobilised and an outer truncated cone-shaped surface (21), which acts upon the truncated cone-shaped surface (11) of the outer ring (1) and, optionally, an additional ring (4) designed to be positioned between the outer ring (1) and the wedges (2), increasing the range of glass sizes (3) which the device can accept. <IMAGE>
Patent ES-2188377-B1 (ES)
Title: Conjunto de espejo y placa portaespejos de retrovisores exteriores de vehiculos automoviles.
Inventor: CLARIMON FELIP JOAQUIM
IPC: B60R1/06
Filed: 2001-06-04
Granted: 2004-10-16
Abstract: Conjunto de espejo y placa portaespejos de retrovisores exteriores de vehículos automóviles. Este conjunto de espejo y placa portaespejos es aplicable a retrovisores exteriores del tipo constituido por una carcasa adaptada para contener el conjunto y un mecanismo de posicionamiento de la placa portaespejos, siendo la carcasa acoplable a un soporte fijado a la carrocería del vehículo. El conjunto comprende una primera capa (2) de material eléctricamente aislante y una segunda capa (3) de material adhesivo dispuestas entre la cara interior (5) del espejo (1) y la placa portaespejos (4), quedando la primera capa (2) entre la cara interior (5) del espejo (1) y la segunda capa (3). Entre la cara interior (5) del espejo (1) y la primera capa (2) de material eléctricamente aislante el conjunto está provisto de un dispositivo calefactor (6, 7).