baber/WOPTO huggingface dataset:
Patent JP-3727569-B2 (JP)
IPC: C07D401/06
Filed: 2001-11-02
Granted: 2005-12-14
Abstract: The present invention relates to tetrahydroquinazoline-2,4-diones derivatives of the formula (I):  <CHEM>  pharmaceutically acceptable salts thereof, wherein A is (CH2)n where n is equal to 0, 1 or 2; U is CH2, NH, or NR<3>, R<1> and R<2> are selected independently from H, (C1-C6)alkyl, Cl, F, CN, nitro, CF3, -NHC(O)R<6> and -OR<7>, or R<1> and R<2>, together with the atoms to which they are attached, form a carbocyclic or heterocyclic five- or six-membered ring, R<3> is selected from the group consisting of H, (C1-C6)malkyl, C(=O)-(C1-C6)alkyl, where m=1 or 2; R<4> and R<5> are selected from H, (C1-C6)alkyl, Cl, F,-CF3, -CN, -NHC(=O)R<6>, -OR, a 5-to 7-membered aryl or heteroaryl ring, where m, R<6> and R<7> are as defined above; and R<6> and R<7> are selected independently from H, (C1-C6)alkyl or a 5- to 7-membered aryl or heteroaryl ring; V is CH, CR<3>, or N; W is CH2, C(O), or S(O)2; X is C or N; and Y is CH, CR<1>, CR<2>, or N. The invention also relates to pharmaceutical compositions containing the same and to methods of use thereof, including in the inhibition of serotonin reuptake, the inhibition of the binding of 5-HT2A serotonin receptors and the treatment of diseases, conditions or disorders of the central nervous system. Further, the present invention is also directed to methods for the preparation of 4-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)-propyl-1,2,3,4-tetrahydroq uinazoline-2,4-dione compounds and intermediates useful therefor.
Patent JP-4610827-B2 (JP)
IPC: G01F11/04
Filed: 1999-09-10
Granted: 2011-01-12
Abstract: Apparatus for metering one or more liquids contained in respective reservoirs (2, 6) into one or more collecting containers is characterized in that it comprises, for each liquid: a cylinder (2) for the liquid to be metered, the cylinder having a movable piston member (8) in contact with the surface of the liquid in the cylinder (2), pressure means (12) for exerting a constant force on the piston (8), means (14, 16, 18, 20) for the transfer of the liquid from the cylinder (2) to the collecting container, the transfer means comprising a duct having an inlet opening (16) for the withdrawal of the liquid from the cylinder and a delivery opening (20), the transfer means being movable in dependence on the level of liquid in the cylinder (2) and being arranged to keep the geometrical height difference H1 between the withdrawal point and the delivery point proportional to the hydrostatic head of liquid H2 above the withdrawal point with variations in the level of liquid in the cylinder so as to keep the delivery flow-rate constant, and valve means (22) associated with the transfer means for controlling the flow of liquid in the transfer means.
Patent JP-3686373-B2 (JP)
IPC: A61F9/008
Filed: 2000-11-14
Granted: 2005-08-24
Abstract: Methods and devices for performing corrective eye surgery generally direct a laser beam at a target region of a patient's eye with the laser beam having a non-uniform energy distribution profile. As ablation rates vary locally across the beam cross-section, the energy distribution profile is tailored to effect a uniform ablation depth with each laser pulse of an excimer laser system.
Patent JP-5399597-B2 (JP)
IPC: B66B5/22
Filed: 2001-05-23
Granted: 2014-01-29
Abstract: A braking device acts on a guide rail and consists of a housing that is arranged at an elevator car yoke and serves as a support for spring packets and/or for adjusting packets. The housing also serves as a support and guide for chock guide elements that in turn retain and guide brake chocks with brake linings. Pushrods engage at one end at the brake chocks, and at the other end are pivotably connected to an actuating fork. Upon braking of the elevator car, the actuating fork is moved at the pushrod end in the direction of the braking device. The guided brake chocks with the brake linings slide in the braking device. At the same time the brake linings are moved at the guide leg of the guide rail. The brake chocks are moved in the braking device and the spring and adjusting packets are stressed, whereby a braking force for stopping an elevator car or a counterweight is generated.
Patent JP-4197231-B2 (JP)
IPC: C07D231/38
Filed: 2002-02-28
Granted: 2008-12-17
Abstract: 4,5-diaminopyrazole compounds and their salts with organic or inorganic acids are new. 4,5-diaminopyrazole compounds of formula (I) and their salts with organic or inorganic acids are new. R<1> = H, 1-6C alkyl, 1-4C hydroxyalkyl, 1-4C aminoalcohol, 1-8C alkylamino, di(1-8C) alkylamino, 1-4C alkylamino-(1-4C) alkyl, di(1-4C)alkylamino-(1-4C) alkyl, aryl or heteroaryl; R<2>, R<3> = H, 1-6C alkyl, aryl, heteroaryl, carboxylic acid or ester, optionally substituted carboxylic acid amide, hydroxyl or 1-4C hydroxylalkyl or R<2> and R<3> together form a 1-6C alkylene, optionally substituted; Z = 1-10 alkyl, optionally containing heteroatoms, a mono- or di benzocondensed aromatic or heteroaromatic, optionally substituted by hydroxyl or (1-6C) alkyl or a diradical Ar-(Alk)n-Ar; Ar = arylene or heteroarylene, optionally substituted; Alk = CH2; n = 0-6; x, y = 0 or 1 An Independent claim is included for a composition for the oxidative coloring of keratin fibers containing a 4,5-diaminopyrazole compound of formula (I).
Patent JP-4274776-B2 (JP)
IPC: H04B10/2525
Filed: 2002-11-12
Granted: 2009-06-10
Abstract: A chromatic dispersion compensating optical fibre (12i) has ring refractive index profile with low index ring and negative chromatic dispersion slope, low curved loss and dispersion to loss ratio with cutoff frequency suitable for operation in Band U.
Patent JP-5000064-B2 (JP)
IPC: C08G65/333
Filed: 2001-07-11
Granted: 2012-08-15
Abstract: The present invention relates to a process for forming polymer conjugates which are useful as enzyme inhibitors. The process of the present invention comprises the steps of:a) reacting a polymer or copolymer alcohol to form a chloroformate;b) combining a substituted or unsubstituted anthranilic acid comprising an enzyme interaction attenuating unit; and a base catalyst wherein the base catalyst is a supported base catalyst, to form a substrate reactive admixture; andc) adding to said chloroformate formed in step (a) said substrate reactive admixture formed in step (b) to form a benzoxazin-4-one conjugate.
Patent JP-4768210-B2 (JP)
IPC: G02F1/1335
Filed: 2001-09-18
Granted: 2011-09-07
Abstract: A viewing screen for increasing the viewing angle of a display, such as a liquid crystal, having metallised tapered waveguides (43).
Patent JP-4057419-B2 (JP)
IPC: A21D13/00
Filed: 2001-10-23
Granted: 2008-03-05
Abstract: A food product, such as a baked good, having either high molecular weight starch hydrolysate or a crystalline hydrate producing sugar as a sweetening agent. Preferably, the starch hydrolysate has a dextrose equivalent of about 5 to 30 DE, and the crystalline hydrate former is raffinose or trehalose. The high molecular weight starch hydrolysate, the crystalline hydrate former, or combination thereof, increases the crispiness of the product at higher moisture levels. The food product can be a baked good such as an ice cream cone, cookie, wafer, or the like.
Patent JP-4606698-B2 (JP)
IPC: C07D333/62
Filed: 2002-05-07
Granted: 2011-01-05
Abstract: The present invention provides a method of treating ocular hypertension or glaucoma which comprises administering to an animal having ocular hypertension or glaucoma therapeutically effective amount of a compound represented by the general formula I;wherein hatched lines represent the alpha configuration, a triangle represents the beta configuration and a dotted line represents the presence or absence of a double bond;A and B are CH2;D represents a covalent bond or CH2, O, S or NH;X is CO2R, CONR2, CH2OR, P(O)(OR)2, CONRSO2R SONR2 orY is O, OH, OCOR<2>, halogen or cyano;Z is CH2 or a covalent bond;R is H or R<2>;R<1 >is H, R<2>, phenyl, or COR<2>;R<2 >is C1-C5 lower alkyl or alkenyl and R3 is benzothienyl, benzofuranyl, naphthyl or substituted derivatives thereof, wherein the substituents maybe selected from the group consisting of C1-C5 alkyl, halogen, CF3, CN, NO2, NR2, CO2R and OR.
Patent JP-4206320-B2 (JP)
IPC: H01L21/56
Filed: 2003-09-19
Granted: 2009-01-07
Abstract: Productivity is to be improved in assembling a semiconductor integrated circuit device. A matrix substrate is provided and semiconductor chips are disposed on a first heating stage, then the matrix substrate is disposed above the semiconductor chips on the first heating stage, subsequently the semiconductor chips and the matrix substrate are bonded to each other temporarily by thermocompression bonding while heating the chips directly by the first heating stage, thereafter the temporarily bonded matrix substrate is disposed on a second heating stage adjacent to the first heating stage, and then on the second heating stage the semiconductor chips are thermocompression-bonded to the matrix substrate while being heated directly by the second heating stage.
Patent JP-4055691-B2 (JP)
IPC: B25J19/00
Filed: 2003-10-03
Granted: 2008-03-05
Abstract: In origin adjustment between two members which rotate relatively at a joint of an industrial robot, an origin adjustment apparatus is provided which is inexpensive and highly accurate and which requires extremely few man hours. In addition, an origin adjustment apparatus is provided which is so small in size as to be easily used even on a distal end shaft of a wrist of the robot and which requires no special signal line for origin adjustment. A mount member 23 where a positioning member 22 is embedded and a guide portion 24 along which the positioning member 22 slides in such a manner as to protrude are provided on either one or both of the two members which rotate relatively.
Patent JP-4358608-B2 (JP)
IPC: B60L15/42
Filed: 2003-11-25
Granted: 2009-11-04
Abstract: An information transmission system with high reliablility by which transmission can be continued even when multiple failures occurs. Two main transmission lines (21 and 22) are provided, and transmission terminals (111 to 124) are connected to both of main transmission lines. Each of transmission terminals (111 to 124) transmits the data received other transmission terminals to both of main transmission lines (21 and 22) when the data of the transmission terminal is transmitted. Because each of transmission terminals (111 to 124) transmits data repeatedly, the data can be transmitted even at multiple troubles like two line disruptions.
Patent JP-4068558-B2 (JP)
IPC: B65D47/26
Filed: 2002-07-24
Granted: 2008-03-26
Abstract: A reclosable lid 10 for a container holding a flowable substance has a first piece or cover 12 , and a movable second piece or disk 50 . The cover 10 has a top wall 14 , a side wall 16 and a mounting portion 22 for connecting the lid 10 on the container. The cover 12 has an opening 28 adapted to permit the flow of the substance through the lid 10 . The cover 12 further includes a slot 30 located in the top wall 14 . The disk 50 has at least one aperture 78 , a post 54 , and a projection 52 . The aperture 78 and the projection 52 are each cooperatively dimensioned with the opening 28 . The post 54 is adapted to be received by the slot 30 in the cover 12 . The disk 50 is movable between a first position wherein at least a portion of the projection 52 is received in the opening 28 in the first position, and a second position wherein the aperture 78 is aligned with the opening 28 in the second position. A support ledge 102 and a support edge 104 on an inner surface 100 of the cover 12 are adapted to provide rotatable support to the disk 50.
Patent JP-4056006-B2 (JP)
IPC: F24H1/10
Filed: 2002-08-12
Granted: 2008-03-05
Abstract: Apparatus for rapidly heating fluid includes a fluid circuit (12) having electrodes (16, 17, 18) between which the fluid flows. A voltage is applied between a pair of electrodes (16, 17, 18) whereby current is caused to flow through the fluid. The inlet and outlet fluid temperatures are measured and the current controlled by varying the applied voltage to produce a desired temperature rise in the fluid in accordance with measured fluid flow rate.
Patent JP-4271030-B2 (JP)
IPC: A61M60/122
Filed: 2002-08-26
Granted: 2009-06-03
Abstract: The invention relates to a magnetically hard object and to a method for adjusting a magnetic vector of a magnetically hard object. The aim of the invention is to provide a magnetically hard object and a method for producing the same, said object having a desired resulting magnetic vector which moves within a pre-determined tolerance range, without influence from an external magnetic circuit. Furthermore, the magnetically hard object is to have a higher maximum energy density in relation to prior art. According to the invention, a magnetically hard object having a magnetic vector which moves in the open magnetic circuit, to a large extent within a pre-determined tolerance range, consists of at least one magnetically hard moulded part (1) and at least one other moulded element (11) which are combined in such a way that a pre-determined direction and position of the magnetic vector of the magnetically hard object are achieved by forming, combining and orienting the moulded part (1) and the moulded element (11). The magnetic vector of the magnetically hard object is the resulting magnetic vector of the magnetic vectors (4, 14) of the magnetically hard moulded part (1) and the moulded element (11).
Patent JP-4304075-B2 (JP)
IPC: F02N99/00
Filed: 2003-01-08
Granted: 2009-07-29
Abstract: The invention relates to a starting system ( 1 ) for an internal combustion engine comprising pressurized fuel supply means ( 3 ), an accumulator means ( 2 ), which is supplied with pressurized fuel by said supply means, and at least one injection means ( 4 ) which is supplied with fuel by the accumulator means ( 2 ). According to the invention, the system also comprises a device for storing pressurized fuel ( 5 ), which is supplied due to the pressure in the accumulator means. At start-up, the aforementioned fuel storage device can supply the stored fuel in such a way as to provide a second fuel compression means which enables the engine to start up more rapidly. The invention is particularly suitable for use in the area of common-rail engines.
Patent JP-4170916-B2 (JP)
IPC: A61F2/24
Filed: 2001-12-27
Granted: 2008-10-22
Abstract: A trileaflet biological prosthetic heart valve comprising a thin, rigid annular outer frame which supports three elastic, laminated spring inner frames which in turn provide consistent geometric form and structure for attachment of tissue leaflets.
Patent JP-4103799-B2 (JP)
IPC: H02N2/02
Filed: 2003-02-28
Granted: 2008-06-18
Abstract: A linear actuator is an actuator for directly driving (moving) a slider. The linear actuator has an actuator unit constituted by the slider and an actuator body on which the slider is movably provided for linear movement. The actuator body has a base, a vibrating element for moving the slider, two rollers to movably support the slider, pushing means for pushing the vibrating element into contact with the slider, and a conducting circuit for conducting each of electrodes of the vibrating element by selecting a conducting pattern to each of the electrodes. Grooves are respectively formed in outer circumferential surfaces of the rollers, and the slider is arranged inside each of the grooves.
Patent JP-4901084-B2 (JP)
IPC: B62D1/18
Filed: 2004-09-08
Granted: 2012-03-21
Abstract: The module has a motor (5) to adjust position of a steering wheel along a transverse pivoting axis for adjustment of a tilt of the wheel and along a longitudinal axis for adjustment of a distance of the wheel. A controller receives information representing a state of one threaded joint unit that is driven by the motor. An incremental position sensor is driven by the motor for sending a position signal to the controller.
Patent JP-4414309-B2 (JP)
IPC: F16D65/28
Filed: 2004-09-16
Granted: 2010-02-10
Abstract: <P>PROBLEM TO BE SOLVED: To provide an electric parking brake device is equipped with a motor-operated driving means having an electric motor to exert the power to change over a parking drum brake between the braking condition and non-braking condition and able to hold the braking condition of the parking drum brake and a control unit to control the actuation of the driving means by making possible to select the automatic disengage mode in which the driving means is actuated so that the parking drum brake is put in the non-braking condition automatically in accordance with the vehicle starting operation in the parking condition, whereby capable of executing easily the abutting whether the automatic disengage mode is selected or not.  <P>SOLUTION: When the abutting mode to execute the initial abutting of a brake shoe is selected by an abutting mode selecting means, the control unit controls the actuation of the motor-operated driving means so that the parking drum brake exerts a specified braking force smaller than the braking force required to maintain the parking condition until the vehicle has run for a specified distance even if the automatic disengage mode is in selection.  <P>COPYRIGHT: (C)2006,JPO&NCIPI
Patent JP-4426445-B2 (JP)
IPC: H01M8/06
Filed: 2003-05-16
Granted: 2010-03-03
Abstract: The regulation method has characteristic measured values for the liquid quantity or liquid quantity variation in the fuel cell system determined for corresponding adjustment of the cooling output of a fluid condensation device, the condensed liquid fed to the anode circuit of the fuel cell system.  An Independent claim for a fuel cell system is also included.
Patent JP-4931389-B2 (JP)
IPC: B06B1/02
Filed: 2005-09-12
Granted: 2012-05-16
Abstract: <P>PROBLEM TO BE SOLVED: To provide a pressure wave generator having high durability and quality, and a method for driving the pressure wave generator.  <P>SOLUTION: The pressure wave generator according to the present invention is a pressure wave generator 1 for generating a pressure wave, and comprises a silicon substrate 11, a heat insulating layer 13 disposed on the silicon substrate 11, a heating element film 14 formed on the heat insulating layer 13, and a driving unit 17 connecting to the heating element film 14 and supplying a driving current to the heating element film 14, wherein the driving current is composed of a pulse train with intervals of amplitudes and pulses, or a pulse width being modulated. Accordingly, the pressure wave generator according to the present invention generates and outputs a pressure wave corresponding to the modulated pulse train.  <P>COPYRIGHT: (C)2007,JPO&INPIT
Patent JP-5027397-B2 (JP)
IPC: G06F3/0482
Filed: 2005-09-21
Granted: 2012-09-19
Abstract: A method of representing user tasks to be performed by one or more of a plurality of electronic devices in a task orchestration system. Each device includes therein a function description specifying a function that the device can perform. The function descriptions are obtained from one or more of the devices, task descriptions that describe device functionalities required for certain tasks are obtained, and task suggestion are generated based on the obtained device function descriptions and task descriptions. Each task suggestion represents a user task as an abstraction of on or more of the obtained device descriptions and task descriptions. The tasks suggestion are displayed on a display for the user to select from, wherein the user selected task suggestion is to be performed by orchestration (automation) of one or more of the devices based on task descriptions that use device functionalities described in the device function descriptions.
Patent JP-4842609-B2 (JP)
IPC: H01L29/78
Filed: 2005-10-06
Granted: 2011-12-21
Abstract: In a semiconductor device including a core transistor and an I/O transistor on the same semiconductor substrate, the core transistor includes a gate insulating film, a gate electrode, sidewalls, extension diffusion layers, and source/drain diffusion layers. The I/O transistor includes a gate insulating film, a gate electrode, sidewalls, and source/drain diffusion layers. In the I/O transistor, the source/drain diffusion region is offset relative to a channel region located beneath the gate insulating film in regions below the sidewalls.
Patent JP-4217234-B2 (JP)
IPC: B60W10/10
Filed: 2005-10-06
Granted: 2009-01-28
Abstract: <P>PROBLEM TO BE SOLVED: To properly perform the continuous operation of an internal combustion engine when an intermittent operation is inhibited.  <P>SOLUTION: When the intermittent operation of an engine 22 is inhibited, and a speed from a speed sensor 88 is within a high vehicle speed region, a motoring mode is executed to operate the motoring of the engine 22 by a motor MG1 by cutting the fuel of the engine 22, and to output a torque matched with a request torque to a ring gear shaft 32a as a drive axle, and when the speed is within a low vehicle speed region, an independent operation mode is executed to operate the independent operation of the engine 22 by stopping the motor MG1, and to output a torque matched with the request torque to a ring gear shaft 32a. Thus, it is possible to improve energy efficiency by executing the motoring mode which is more efficient than the independent operation mode, and to prevent inconvenience due to the execution of the motoring mode in the low vehicle speed region, for example, the continuous discharging of a battery 50.  <P>COPYRIGHT: (C)2007,JPO&INPIT
Patent JP-5392968-B2 (JP)
IPC: C40B60/00
Filed: 2005-10-18
Granted: 2014-01-22
Abstract: An inkjet nozzle arrangement is provided. The arrangement comprises a nozzle chamber having an ink ejection port defined in a wall of the nozzle chamber, an ink supply channel for the supply of ink to the nozzle chamber, and an actuator located in the nozzle chamber, between the ink supply channel and the ink ejection port. The actuator is adapted to cause ejection of ink from the nozzle chamber upon activation.
Patent JP-4892228-B2 (JP)
IPC: B60R11/02
Filed: 2005-11-15
Granted: 2012-03-07
Abstract: <P>PROBLEM TO BE SOLVED: To satisfy requirements for improving convenience of a wireless terminal device mounted to an emergency vehicle and the like because realization of a convenience wireless terminal device is desired in a one-station and two-device constitution, in particular, an emergency condition is predicted in fire sites, accident sites and the like.  <P>SOLUTION: This wireless terminal device has a vehicle-mounted walkie-talkie 101 and a mobile walkie-talkie 110. The vehicle-mounted walkie-talkie has a terminal for outputting on/off information of a power source of a vehicle-mounted walkie-talkie to a mobile walkie-talkie for detachably mounting the mobile walkie-talkie and a mobile walkie-talkie housing part. The mobile walkie-talkie has a control unit 113 for controlling on/off of the power source of the mobile walkie-talkie, and a detection terminal for detecting on/off information of the power source of the vehicle-mounted walkie-talkie. When, the mobile walkie-talkie is mounted to the mobile walkie-talkie housing part, the control unit 113 of the mobile walkie-talkie is constituted to turn on/off the power source of the mobile walkie-talkie based on the information from the terminal outputting the on/off information of the power source of the vehicle-mounted walkie-talkie.  <P>COPYRIGHT: (C)2007,JPO&INPIT