baber/WOPTO huggingface dataset:
Patent CO-5560573-A2 (CO)
Title: Derivados activos de amino-ftalazinona como inhibidores de quinasa, proceso para su preparacion y composiciones farmaceuticas que los contienen
Inventor: PULICI MAURIZIO
IPC: A61P19/02
Filed: 2004-03-03
Abstract: 1.- Un método para el tratamiento de enfermedades causadas y/o asociadas con una actividad alterada de proteína quinasa que comprende la administración a un mamífero en necesidad de este, de una cantidad de un derivado de amino-ftalazinona representado por la fórmula I. en dondeRa y Rb son, cada uno independientemente, un átomo de hidrógeno o un grupo, opcionalmente substituido adicionalmente, seleccionado de alquilo C1-C6 lineal o ramificado, cicloalquilo C3-C6 o alquilo C1-C6 cicloalquilo, arilo, alquilo C1-C6 arilo, heterociclil de 5 a 7 miembros o alquilo C1-C6 heterocliclil con de 1 a 3 heteroatomos seleccionados entre nitrógeno, oxigeno o azufre; o que alguno de Ra o Rb es hidrógeno o un grupo sustituido opcionalmente de alquilo C1-C6 lineal o ramificado, y el otro es un grupo seleccionado de -CORAND#39, -CONHRAND#39, -COORAND#39, o -SO2RAND#39, en donde RAND#39 es hidrogeno o un grupo opcionalmente sustituido seleccionado entre alquilo, cicloalquilo, cicloalquilalquilo, arilo, arilalquilo, heterociclil o heterociclilalquil, como se expuso anteriormente;R1 es un grupo de formula -CHR4R5 donde R4 y R5 son, cada uno independientemente, hidrógeno o un grupo sustituido opcionalmente, seleccionado de alquilo C1-C6 lineal o ramificado, cicloalquilo C3-C6 o alquilo C1-C6 cicloalquilo, arilo, alquilo C1-C6 arilo, heterociclil de 5 a 7 miembros o alquilo C1-C6 heterociclil con de 1 a 3 heteroatomos seleccionados entre nitrógeno, oxígeno o azufre; o R1 es un grupo de formula -NHRAND#39, -NRAND#39COR", -NRAND#39CONHR" o -NRAND#39SO2R", donde RAND#39 tiene los significados anteriores diferentes de hidrógeno, y R" es hidrógeno o tiene los significados expuestos anteriormente para RAND#39;R2 es un átomo de hidrógeno o es un grupo, opcionalmente sustituido adicionalmente, seleccionado de alquilo C1-C6 lineal o ramificado, cicloalquilo C3-C6 o alquilo C1-C6 cicloalquilo, arilo, alquilo C1-C6 arilo, heterociclil de 5 a 7 miembros o alquilo C1-C6 heterociclil con 1 a 3 heteroatomos seleccionados entre nitrogeno, oxigeno o azufre;Cualquier R3, colocado en una o más de las posiciones libres 5, 6 y 8 del anillo ftalazinona es, independientemente de cada uno, halógeno, nitro, carboxi, ciano, o un grupo opcionalmente sustituido adicionalmente y seleccionado de alquilo C1-C6 lineal o ramificado, cicloalquilo C3-C6, alquilo C1-C6 cicloalquilo, arilo, alquilo C1-C6 arilo, ...
Patent CO-6321136-A2 (CO)
Title: Derivados de indazol sustituido por axadiazol para uso como agonistas de esfingosina 1 fosfato (s1p)
Inventor: AHMED MAHMOOD
IPC: A61K31/4245
Filed: 2009-10-16
Abstract: La presente invención proporciona compuestos de la fórmula (I) o sales de los mismos:que tienen actividad farmacológica, procedimientos para su preparación, composiciones farmacéuticas que los contienen y el uso de los mismos en el tratamiento de diferentes trastornos mediados por los receptores S1P1.
Patent CO-6751261-A2 (CO)
Title: Parche medicado para mejorar la penetración transdérmica del diclofenaco dietilamonio
Inventor: CILURZO FRANCESCO
IPC: A61K31/00
Filed: 2013-07-26
Abstract: Un parche medicado para mejorar la penetración transdérmica del diclofenaco dietilamonio en una composición que comprende un copolímero acrílico y un éster de ácido cítrico.
Patent CO-7151513-A2 (CO)
Title: Nuevo inhibidor de beta-lactamasa y proceso para prepararlo
Inventor: ABE TAKAO
IPC: C07D471/08
Filed: 2014-12-10
Abstract: Los inhibidores de beta-lactamasa disponibles en laactualidad son insuficientes para inhibir cada vez más lab lactamasa y se han requerido nuevos inhibidores de beta- lactamasa en la actualidad para el tratamiento difícil frlas enfermedades infecciosas bacterianas causadas porbacterias resistentes que producen b lactamasa de clase C,ß lactamasa de espectro extendido (ESBL) perteneciente a laclase A y D o KPC 2 de clase A que aun descomponecarbapenem como un último recurso para el antibiótico lactámico. Se proporcionan un compuesto representado por lafórmula (I), el proceso de preparación del mismo,inhibidores de beta-lactamasa y método para tratar lasenfermedades infecciosas bacterianas.[Fórmula química 1]
Patent EP-1031455-A2 (EP)
Inventor: BACHORSKI TOMASZ
IPC: G01D7/04
Filed: 2000-01-21
Abstract: The display device has a pointer element (50) or elements that can be brought into a neutral position in a separate display field covered by a further display element when the vehicle is operationally deactivated. This neutral position is not the display null position and the vehicle is brought back into the null position at operational start-up.  An Independent claim is also included for a method of operating a display device.
Patent EP-1037370-A2 (EP)
Inventor: ITABASHI TORU
IPC: F02D41/20
Filed: 2000-03-17
Abstract: A microcomputer (8) produces to a drive circuit (9) drive
command signals for starting to drive and braking a motor (3)
so that the position of a throttle valve (2) is controlled to
a target position. A current supplied to the motor (3) is
limited not to exceed a first current limitation value at the
time of motor drive start and braking. When the current
limitation continues for a predetermined time period (t32),
the current is further limited not to exceed a second current
limitation value. The microcomputer (8, 108 - 110) detects
switching of motor current supply direction. When the current
supply direction is switched, a reset command signal (SR) is
produced to reset a timer operation for a current limitation
continuation determination.
Patent EP-1108675-A2 (EP)
Inventor: UTSUNOMIYA HIROFUMI
IPC: B66B23/00
Filed: 2000-04-10
Abstract: In order to perform curing of the passenger conveyer
without the specifically used leg bodies to be set up on
the floor surface, a frame of the passenger conveyer
supports a curing system for covering a working position
when the passenger conveyer is being installed or repaired.
Patent EP-1046587-A2 (EP)
Inventor: PLUESCHOW DIETER
IPC: B65B61/20
Filed: 2000-04-11
Abstract: A conveyor device with numerous tong-type pincers (17) to pick up leaflets can insert a leaflet (16) between a product (14) its packaging. Near a delivery device in the conveyor path of the pincers there is a stop (18) causing a pincer to open and rele a leaflet.
Patent EP-1048224-A2 (EP)
Inventor: HATTORI TOSHIMITSU
IPC: A23L7/152
Filed: 2000-04-25
Abstract: The present invention provides a method for retaining or enriching gamma  -aminobutyric acid in green grass leaves, which comprises the step of subjecting green grass leaves or processed products thereof to at least one treatment selected from the group consisting of incubation treatment, anaerobic treatment, and microwave treatment.
Patent EP-1065337-A2 (EP)
Inventor: EISENKOECK ERWIN
IPC: E05C9/24
Filed: 2000-06-05
Abstract: A method for fitting the corner joints of an interior frame inside a window, e.g. a twist and tilt window system, has a coupling (10) fitted to the vertical section (13) of the frame and a second coupling (66) fitted to the horizontal section (60) of the frame. The first coupling has a sprung ratchet grip (48), which grips the shaped end (64) of the second coupling for a clip fastening which does not require any separate fasteners. The first coupling has a shaped inlet jaw (46), which guides the tag (64) of the second coupling into the coupling position. The tag has a slot into which the sprung grip drops.
Patent EP-1060913-A2 (EP)
Inventor: BEDERNA CHRISTOPH
IPC: B60C15/02
Filed: 2000-06-09
Abstract: The rim(1) has a radially outer emergency running face. Annular chambers(10) in the axial rim end faces have walls, the outer axial wall(23) including a radially inward facing lip(2) and an annular opening for inserting the thick bead area. When located the tyre bead contacts three walls(21,22,23) and the radially outer face of a filler ring(12). No contact is made between the axially inner chamber wall(21) and bead outer face at a point where an axial gap exists in the wall face. Preferred Features: The filler ring locks the bead(7) in position and rests on the radially inner chamber wall(20). The entire axial length of the radially inner surface of the bead rests on the filler ring. A located bead area contacts the axially inner(21), radially outer(22) and axially outer(23) walls.
Patent EP-1047100-A2 (EP)
Inventor: ANDERSON WETSON A
IPC: H05G1/04
Filed: 1995-01-09
Abstract: An X-ray tube rotating anode (14) is cooled
with a liquid metal (40) functioning as a recirculated
heat exchange fluid and/or a metal film in a gap (39)
between the anode (14) and a stationary structure. The
liquid metal (40) is confined to the gap (39) by (a) a
labyrinth (44 or 46) having a coating that is not
wetted by the liquid, (b) a magnetic structure (22),
or (c) a wick (38). The liquid metal (40)
recirculated through the anode (14) is cooled in a heat
exchanger located either outside the tube or in the
tube so it is surrounded by the anode (14). The heat
exchanger in the tube includes a mass of metal in
thermal contact with the recirculating liquid metal and
including numerous passages (36) for a cooling fluid,
e.g. water. A high thermal conductivity path (26, 48,
49) is provided between an anode region (16) bombarded
by electrons and a central region of the tube where
heat is extracted. In one embodiment the high thermal
conductivity is achieved by stacked pyrolytic
structures having crystalline axes arranged so there is
high heat conductivity radially of the region and lower
thermal heat conductivity normal to the high heat
conductivity direction.
Patent EP-1082955-A2 (EP)
Inventor: KOLLER ANDREAS DR
IPC: A61Q1/04
Filed: 2000-09-04
Abstract: Cosmetic or dermatological formulations contain water-soluble and/or water-dispersible combination polymer(s) (I), consisting of a polymer main chain and sulfonated polyester side arms attached to the main chain by ester groups. An Independent claim is also included for the use of (I) for skin care.
Patent EP-1081444-A2 (EP)
Inventor: FOSTER LORD NORMAN
IPC: F24F13/18
Filed: 2000-09-01
Abstract: The ventilator (1) is built into a partition wall (2) the plane of which coincides with the ventilator's lengthwise axis(6). Part of the ventilator protrudes into a first environmental medium (3) on the one side of the partition; another part of the ventilator protrudes into a second environmental medium (4) on the second side of the partition. The ventilator consists of an outer, immovable part with a drum shaped housing (5) and inner movable part. The inner part is turned by an adjustment (33); the outer and inner parts have ventilation slots (16,17)
Patent EP-1099845-A2 (EP)
Inventor: WELLMANN NORBERT DR
IPC: F02F3/22
Filed: 2000-09-27
Abstract: The piston (1) has a gudgeon pin bore (4) for accommodating a gudgeon pin (5) and a cooling channel (6) arranged in the region between the bore and a piston combustion surface (9), especially within an annular field (2). The cooling channel has at least one connection (7) to the gudgeon pin bore. The connection(s) can be produced after piston manufacture, especially by drilling.
Patent EP-1059392-A2 (EP)
Inventor: BERTINELLI ROMANO
IPC: B08B9/02
Filed: 2000-06-02
Abstract: The device comprises an air receiver (7) having its inlet
connected to a manually operated pumping unit (3, 33) for its
filling with compressed atmospheric air, between said pumping unit
and said receiver (7) there being interposed a valve unit
comprising a non-return valve (77) positioned to intercept the
delivery conduit of said pumping unit; a valving element (10)
slidingly housed air-tight inside a passage chamber (12) into
which said delivery conduit opens, and arranged to close the
outlet of the receiver (7); a vent valve (24), controlled by a
trigger operable from the outside, to intercept a channel (25)
which connects said passage chamber (12) to the outside; and a
duct (11) which passes through said valving element (10) and has
one end constantly connected to said passage chamber (12) and its
other end opening into the outer cylindrical surface of the
valving element (10); said valving element (10) is provided with
elastic means (15) arranged to maintain the valving element (10)
constantly urged towards its closure position, the thrust of said
elastic means (15) being overcome by the thrust produced by the
pressure downstream of the valving element (10) when the passage
chamber (12) is connected to discharge.
Patent EP-1073196-A2 (EP)
Inventor: MA ZHENGXIANG
IPC: H04L27/00
Filed: 2000-07-17
Abstract: A signal notching system reduces signal peaks by notching the peak of a signal
above a threshold to produce a notched signal. The notched signal is then filtered to
produce a resulting signal with a reduced peak amplitude. For example, in an
implementation where the signal is represented by signal samples, the peak notching
system first locates a peak sample that is beyond a threshold, such as a sample
representing a positive peak sample of a peak above the threshold. Once a peak sample is
located, the peak notching system adjusts the peak sample by an amount which is a
function of the amount that the peak sample is beyond the threshold, effectively creating
a notched signal with a one sample notch at the peak. The peak notching system filters
the notched signal to fill in the notch to produce a signal with a reduced peak.
Patent EP-1089240-A2 (EP)
Inventor: SATO TAKESHI
IPC: G07F13/06
Filed: 2000-09-20
Abstract: An automatic beverage vending machine is provided a plurality of
cartridge storing portions (10) each for storing a plurality of cartridges each of
which contains a powdery beverage material therein. A cartridge transferring
mechanism (40) transfers a particular one of the cartridges from the cartridge
storing portions to a beverage extracting position. A beverage extracting
device (20) supplies hot water into the particular cartridge at the beverage
extracting position to extract a beverage from the powdery beverage material.
Patent EP-1099841-A2 (EP)
Inventor: DOTTAVIO JAMES J
IPC: F02D9/02
Filed: 2000-11-03
Abstract: The present invention relates to an electronic throttle
control system having a housing (22) with a motor (40),
throttle valve (60), gear mechanism (100), and failsafe
mechanism (130). A spring member (150) attached between
the housing (22) and a gear member (104) attached to the
throttle valve shaft (62) biases the throttle plate (60)
towards the closed position. A spring-biased plunger
member (134) biases the throttle plate (60) from its
closed position to a default or "limp-home" position.
Patent EP-1113239-A2 (EP)
Inventor: ANG TEOH HWA
IPC: F41A25/20
Filed: 2000-11-24
Abstract: A recoil buffering apparatus for use with an artillery gun of the type comprising a
breech assembly (15) connected to a barrel (12), the breech assembly (15) having
a firing mechanism for firing a projectile through an open end of the barrel (12). The
recoil buffering apparatus comprises a recoil buffering means adapted to be fixed
to the barrel ( 12) and movable therewith during recoil action of the barrel (12)
caused by firing of the projectile, and a support means associated with the recoil
buffering means for supporting the recoil buffering means and thereby supporting
the barrel (12) and breech assembly (15) through the recoil buffering means. An
elevating apparatus and a traversing apparatus for an artillery gun are also
described. The artillery gun can also be provided with a muzzle brake (11).
Patent EP-1111844-A2 (EP)
Inventor: IZUMI MICHIHIRO
IPC: H04W28/00
Filed: 2000-12-15
Abstract: A communication apparatus automatically sets the most
appropriate communication mode in accordance with the
location at which the communication apparatus is used. For
example, the communication mode is switched between
operating as a master station and operating as a remote
station of a wireless communication system depending on
whether or not connection is made to a wired communication
line.
Patent EP-1074918-A2 (EP)
Inventor: OH HYANG-KYUN
IPC: G06F3/08
Filed: 2000-08-01
Abstract: An integrated controller for the detection and operation of both PC Cards,
smart cards and passive smart card adapter cards. In one aspect, the invention detects
the presence of standard expansion cards or passive smart card adapters 18 by
utilizing the reserved detection and voltage selection signal area defined by the PC
Card specification. In another aspect, the invention provides an integrated controller
10 that includes logic to operate either a standard expansion card or a passive smart
card adapter by reassigning certain PC Card signal lines to operate a standard
expansion card or a passive smart card adapter, thereby eliminating the need to
provide pins in addition to those defined by the PC Card specification.
Patent EP-1022596-A2 (EP)
Inventor: DUMITRIU ION
IPC: G02B6/24
Filed: 2000-01-20
Abstract: A packaging assembly for protecting splices of optical fibers comprises an inner
heat-shrinkable tube (1), an outer thinner heat-shrinkable tube (5) and a reinforcing rod
(3). The reinforcing rod has a metal layer (7) on a flat surface thereof. When heating the
assembly for applying it tightly to a splice an electrical current is passed through the
metal layer. Then heat is developed which causes the tubes to shrink. The metal layer can
be applied to have a larger resistance in its central region where it then will be heated
first, the shrinking of the tubes then also starting in the central region, as seen in the
longitudinal direction of the tubes. The metal layer (7) can be made to act like an
electrical fuse, being evaporated when the heat is sufficiently intensive and then
automatically interrupting the electrical current.
Patent EP-1181534-A2 (EP)
Inventor: CHEE MARK S
IPC: G01N21/64
Filed: 2000-05-22
Abstract: Described herein are assays and components for encoding and decoding microspheres. Each assay or component described utilizes at least one nanocrystal.
Patent EP-1218192-A2 (EP)
Inventor: PURCELL DAVID A
IPC: B41J2/165
Filed: 2000-09-21
Abstract: La présente invention concerne un système d'analyse de dépôt de gouttelettes pour une imprimante à jet d'encre. Ce système comporte un substrat souple transparent. L'imprimante peut comporter une source lumineuse d'un côté du substrat, avec un détecteur optique de l'autre côté du substrat.
Patent EP-1242975-A2 (EP)
Inventor: NENONEN PETRI
IPC: G06T5/00
Filed: 2000-12-21
Abstract: This invention provides a method and associated device an inverse histogram based pixel mapping step is combined with an edge enhancement step such as unsharp masking. In such an arrangement the inverse histogram based pixel mapping step improves the performance of the unsharp masking step, serving to minimise the enhancement of noise components while desired signal components are sharpened.
Patent EP-1242823-A2 (EP)
Inventor: LOGTENBERG TON
IPC: C07K16/00
Filed: 2000-12-21
Abstract: The invention provides a method for selecting at least one member from a library of proteinaceous molecules comprising providing at least one cell and/or a functional equivalent thereof, with at least part of said library under conditions that allow binding of any such member to an epitope in and/or on said cells and/or said functional equivalent thereof, removing unbound proteinaceous molecules and selecting said at least one member, wherein said library comprises at least one mutant of a proteinaceous molecule capable of binding to said epitope.
Patent EP-1224424-A2 (EP)
Title: Gas cooker
Inventor: MARBACH ANDREAS
IPC: A47J27/62
Filed: 2000-10-11
Abstract: A gas cooktop includes a gas supply control controlling flames applied to a cooking vessel through a control circuit connected to an infrared sensor that is directed at an infrared-radiation-generating outer surface region of the cooking vessel and receives temperature-related information from the surface of the vessel.
Patent EP-1122357-A2 (EP)
Title: Refiner zur Zerkleinerung von Faserstoffen
Inventor: ANTENSTEINER PETER DIPL ING
IPC: D21D1/38
Filed: 2001-01-25
Abstract: Die Erfindung betrifft einen Refiner zur Zerkleinerung von Faserstoffen mit auf einem Rotor 4 und einem Stator angeordneten Mahlflächen 5, 5', die einen zylindrischen oder kegelförmigen Mahlspalt 3 bilden. Sie ist vornehmlich dadurch gekennzeichnet, daß die Einstellung des Mahlspalts 3 durch am Stator und am Rotor 4 vorgesehene, gegeneinander verschiebbare Keile erfolgt. <IMAGE>
Patent EP-1134982-A2 (EP)
Inventor: FUJIWARA YUJI
IPC: H04N7/26
Filed: 2001-03-16
Abstract: An image signal encoding device has at least encoding
means of dividing a luminescence signal and color-difference
signals of image signals into macro blocks having a plurality
of sub macro blocks and encoding data of the macro blocks
with use of any one of a plurality of compression modes of
which compression rate is different each other, 
   wherein the total numbers of sub macro blocks in the
each macro block are the same for the use of the all kinds
of compression modes.
Patent EP-1138554-A2 (EP)
Inventor: OOKOSHI TETSURO
IPC: B60R16/03
Filed: 2001-03-29
Abstract: A power system where energy generated at a deceleration time
of a running vehicle such as an automobile can be accepted as
regenerative energy sufficiently and safely is provided. In a power
system 10, a non-aqueous solution system secondary battery group 1
where 10 to 11 lithium ion secondary battery cells are connected in
series and an aqueous solution system secondary battery group 2 where
18 control valve type lead-acid battery cells are connected in series
are connected in parallel. The battery capacity of the non-aqueous
solution system secondary battery group 1 is smaller than that of the
aqueous solution system secondary battery group 2. The non-aqueous
solution system secondary battery group 1 and the aqueous solution
system secondary battery group 2 are charged at a current value of
7C or less from a motor generator 3, and the ratio of the charged current
value of the aqueous solution system secondary battery group 2 to the
charged current value of the non-aqueous solution system secondary
battery group 1 is 0.05 to 1.00.
Patent EP-1164043-A2 (EP)
Inventor: TAKENAKA MASAYUKI
IPC: B60L50/16
Filed: 2001-06-06
Abstract: A hybrid driving device is provided with an engine shaft I, a
motor shaft II, and a countershaft III. A parking gear 54, which
has conventionally been placed on the countershaft, is placed on
the engine shaft I to reduce torque loads applied to parts
associated with a parking mechanism 8 and, at the same time, the
countershaft is placed so as not to overlap an engine or a motor
in a radial direction as a result of an axial length being
shortened, thereby shortening the distance between the engine
shaft and the motor shaft. The parts associated with the parking
mechanism are placed in a dead space of an oil pan near a valve
body, being supported by the valve body and a casing wall, thereby
cutting down on space required for arrangement.
Patent EP-1243377-A2 (EP)
Inventor: KOMINE TSUYOSHI
IPC: B23B3/22
Filed: 2001-07-04
Abstract: The present invention provides an automatic-tool-changer-equipped
lathe which has excellent rigidity for
holding tools, which causes no interference between a tool
and a work, and which has no limitation on the number of
changeable tools. The lathe has: a slide 15 relatively
movable in the X and Z axis directions relative to a work
head 12; a tool-rest 18 provided on the slide 15 for holding
a tool; and a tool changer 20 for storing a plurality of
tools and indexing each of the tools at a tool changing
position. The tool-rest 18 can turn on the X-Z plane and
comprises one tool spindle 19 acting as a tool insert part.
The tool spindle 19 is secured to the tool-rest 18.