baber/WOPTO huggingface dataset:
Patent RU-2733393-C9 (RU)
Inventor: LU YAN
IPC: A61K31/427
Filed: 2015-05-05
Granted: 2021-09-09
Abstract: Настоящее изобретение относится к соединению, представленному формулой II, где Q представляет собой NH; Z представляет собой CH или N; A представляет собой фенил, индолил или индазолил, каждый из которых необязательно замещен по меньшей мере одним из следующего: C1-C5линейный или разветвленный алкил или их комбинация; R1независимо представляет собой водород, O-(C1-C5)алкил, O-галоген(C1-C5)алкил, галоген(C1-C5)алкил, -O(CH2)jOCH3, -O(CH2)jNHCH3, -O(CH2)jNH2, -O-(CH2)jN(CH3)2, - OC(O)CF3, -OC(O)CH2Cl, -OCH2Ph, -O(CH2)jN-фталимид или их комбинацию; R2представляет собой водород, O-(C1-C5)алкил, O-галоген(C1-C5)алкил, F, Cl, Br, I, галоген(C1-C5)алкил, CN, NO2, -CH2CN, NH2, гидроксил, COOH, C(O)H, NHCO-(C1-C5)алкил, -O(CH2)kOCH3, -O(CH2)kOH, -O(CH2)kNHCH3, -O(CH2)kNH2, -O-(CH2)kN(CH3)2, -OC(O)CF3, - OC(O)CH2Cl, -OCH2Ph или -O(CH2)kN-фталимид; j и k независимо представляют собой целые числа от 1 до 5; n представляет собой целое число от 1 до 4; или его гидрату, фармацевтически приемлемой соли или их комбинации. Соединения формулы II обладают противораковой активностью и предназначены для лечения, ослабления, снижения тяжести, снижения риска развития или подавления рака. 4 н. и 19 з.п. ф-лы, 12 ил., 4 табл., 6 пр.
Patent DK-259688-D0 (DK)
Inventor: DONN GUENTER
IPC: C12N15/01
Filed: 1988-05-11
Abstract: Callus cultures which are able to grow on nutrient medium containing no amino acids and are able to regenerate can be used for selection on inhibitor-containing nutrient media of cell lines which can be regenerated to crop plants and are resistant to the relevant inhibitor over generations. Cell suspension cultures likewise result in inhibitor-resistant cell lines under these conditions.
Patent DK-382588-D0 (DK)
Inventor: COSTALL BRENDA
IPC: A61K31/445
Filed: 1988-07-08
Abstract: Phenyl-3-aminoalkyl-4-methyl-2,6-dioxopiperidines of the Formula I   <CHEM>  wherein:      R1 represents hydrogen or C1-C4 alkyl;      n is 1 or 2; R2 represents hydrogen or methyl, provided that one R2 is hydrogen when n is 2;      R3 represents hydrogen or C1-C2 alkyl;      R4 represents C1-C2 alkyl;      R5 and R6 independently represent hydrogen or methyl;      m is 0 to 3; and each Y is in a meta or para position and independently represents hydroxy, C1-C2 alkoxy, C1-C2 alkyl, C1-C2 hydroxyalkyl, halogen, or trifluoromethyl, provided that hydroxy and alkoxy are not in the para position, and pharmacologically acceptable salts thereof have antiposychotic activity without sedative side effects. They are particularly useful in the treatment of schizophrenia. The presently preferred compound is 3-(3 min methoxyphenyl)-3-(3 sec -N,N-dimethylaminopropyl)-4,4-dimethyl-2,6-diox opiperidine (AGN 2979).
Patent DK-418089-D0 (DK)
Inventor: TAYLOR JOHN R
IPC: E04C2/54
Filed: 1989-08-24
Abstract: A glass block (14) panel construction and method of fabrication useful for decorative and functional purposes. The panel includes a frame (10) rigidly assembled from interlocking components (40,52) to form a grid-like pattern of adjacent pockets (12), each pocket (12) sized to receive and support a glass block (14) by way of support lips (39,50,60) extending around each pocket, the blocks (14) bonded to the frame (10) and therefore to one another in structurally stable and weather sealed relation. <IMAGE>
Patent DK-534484-D0 (DK)
Inventor: NARDI FRANCO
IPC: B01J19/18
Filed: 1984-11-09
Abstract: PCT No. PCT/SE83/00100 Sec. 371 Date Oct. 2, 1984 Sec. 102(e) Date Oct. 2, 1984 PCT Filed Mar. 18, 1983 PCT Pub. No. WO84/03724 PCT Pub. Date Sep. 27, 1984.The present invention provides a reactor adapted to simultaneously accomplish chemical reactions and operations of size reduction of the solid materials in suspension and particularly for treatment in the cellulose and/or paper pulp industry. The reactor provides an essentially closed working environment and is provided in the lower part with a rotor which creates turbulence with flows over essentially the whole volume of the closed environment and is adapted to realize said conditions of the size reduction of solid materials with intimate mixing of same with the suspending liquid.
Patent DK-537988-D0 (DK)
Inventor: BURNS ALAN ROBERT
IPC: B62D55/24
Filed: 1988-09-27
Abstract: A ground engaging segment providing a running surface for wheels, endless tracks and the like, which is not pneumatic in nature, thereby not susceptible to puncture, and which is resiliently flexible to offer some resistance to shock. The ground engaging segment comprises a base and a number of removable, hollow, tubular ground engaging elements which extend transversely of the direction of travel of the running surface. Said ground engaging elements include an inner face for engagement to the base and an outer face for contact with the ground surface, and angular shaped side faces between the inner and outer faces allowing for resilient flexibility under normal load conditions. It is preferable that the ground engaging elements are open at their ends to allow for dissipation of heat and are arranged in circumferential rows, defining a chevron pattern, to prevent resultant side thrust imposed upon the running surface. In addition, the ground engaging elements are constructed angularly to provide a line about which the side faces can flex, and include a flexible internal reinforcement, built in to the walls of the faces of the ground engaging element to provide reinforcement for the ground engaging element, while maintaining flexibility.
Patent DK-593785-D0 (DK)
Inventor: GALLENKAMP BERND
IPC: A01N43/56
Filed: 1985-12-19
Abstract: 1. Process for the preparation of substituted phenylhydrazines of the formula (I)  see diagramm : EP0187285,P7,F4  in which R**1 and R**2 represent hydrogen or chlorine, R**3 represents halogenoalkyl, X represents oxygen, sulphur, sulphinyl or sulphonyl and n represents a number 0 or 1, characterised in that substituted chlorobenzenes of the formula (II)  see diagramm : EP0187285,P7,F1  in which R**1 and R**2 represent hydrogen or chlorine, R**3 represents halogenoalkyl, X represents oxygen, sulphur, sulphinyl or sulphonyl and n represents a number 0 or 1, are reacted with hydrazine or hydrazine hydrate, if appropriate in the presence of a diluent and if appropriate at elevated pressure, at temperatures between 60 and 160 degrees C.
Patent DK-665887-D0 (DK)
Inventor: CIRELLI GIORGIO
IPC: A61M5/14
Filed: 1987-12-17
Abstract: The portable appliance is of use for the subcutaneous or intradermal injection of a liquid formulation of an active principle and it comprises in combination: a supply vessel for the formulation; an injection needle adapted to communicate with the vessel; pump means for emptying the vessel through the injection needle; securing means for securing the appliance to an appropriate part of the patient's body; and needle-driving means for shooting the injection needle into the patient's skin.
Patent HU-912318-D0 (HU)
Title: New trichoderma harzianum, t-39 isolate, fungicide preparations containing the isolate, and their use against b.cinerea and s.sclerotiorum
Inventor: ELAD YIAGAL
IPC: A01N63/38
Filed: 1991-07-10
Abstract: The present invention relates to a novel biologically pure culture of Trichoderma Harzianum, T-39, to biological control compositions containing same and to methods of protecting plants from the disease gray mold, caused by B. Cinerea and the disease white rot caused by S. Sclerotiorum with such compositions.
Patent IT-8309391-D0 (IT)
Inventor: ALBERTO FRULLINI
IPC: D04B9/20
Filed: 1983-04-12
Abstract: A machine for knitting tubular fabrics by using a cylindrical array of (double barbed) needles is complemented by an external concentric shell and cam with oblique edges and an adjacent peg such that for each full cycle of the machine, the shell can accelerate to one angular position and halt for the cam to control selection of needles between thread pick-up and release positions, to allow formation of partial rows of meshes, then restores the needle positions while rotating to the start position for the next cycle.
Patent NO-863206-D0 (NO)
Inventor: BONIN WULF VON
IPC: C09K21/12
Filed: 1986-08-08
Abstract: 1. Filler-containing, solid or porous intumescent compositions and construction elements which eliminate water at temperatures above 100 degrees C and can be obtained by reacting polysisocyanates with phosphorus-containing hydroxyl compounds, in particular phosphorus-containing condensation products containing at least two hydroxyl groups and obtainable by condensation of primary of secondary alphatic, araliphatic or heterocyclic monoamines and/or polyamines, carbonyl compounds and dialkyl phosphites which optionally contain OH groups, if appropriate with subsequent oxalkylation, and, if appropriate, cyanuric acid and/or cyanuric acid derivatives, in the presence of fillers which eliminate water above 100 degrees C and, if appropriate, further auxiliaries and additives, characterized in that the water-eliminating fillers used are those having means grain sizes above 5 mu m, preferably 8 - 50 mu m, and/or BET surface areas of less than 5 m**2/g, preferably 2 - 0.1 m**2/g.
Patent NO-874572-D0 (NO)
Inventor: COSSEMENT ERIC
IPC: C07D233/64
Filed: 1987-11-03
Abstract: New substituted 1H-imidazoles and their salts, processes for the preparation thereof and pharmaceutical compositions. These compounds have the formula   <IMAGE>   wherein R1, R2, R3 and R5=hydrogen or C1-C4-alkyl; R4=hydrogen, C1-C4-alkyl or C1-C4-alkoxy; Y1=hydrogen and Y2=OZ2 or the reverse; Z1=Z2=hydrogen or C1-C4-alkyl or Z1 and Z2=-CH2- or -C(CH3)2-. These compounds are prepared either by reducing a corresponding imidazole compound having a hydroxyl or alkoxy group on the methyl bridge between the imidazole and phenyl rings, or by hydrolyzing a 4-[[2,2-dimethyl-4H-1,3-benzodioxin-6(or 8)-yl]methyl]-1H-imidazole, or yet by reducing an alkyl 3-[(1H-imidazol-4-yl)methyl]-2-hydroxybenzoate. These compounds have cardiac, cerebral and tissular anti-ischemic activities.
Patent NO-875014-D0 (NO)
Inventor: DREANO CLAUDE
IPC: A23L13/70
Filed: 1987-12-01
Abstract: The process aims to tenderise the meat, to improve its behaviour and appearance on preservation, and to reduce weight losses on preservation and cooking. 
<??>It consists in subjecting the meat to vacuum/pressurisation cycles which may be repeated several times in a closed chamber (1), optionally in rotation on itself, equipped with a vacuum pump (22) and a source (20, 16) of compressed air. 
<??>The process may be applied to fresh meat or to frozen meat before, during or after freezing. 
<??>All meats may be treated, including poultry and game. The process may also be used for fish. 
<IMAGE>
Patent NO-882014-D0 (NO)
Inventor: MAECHTLE DANIEL
IPC: B25B31/00
Filed: 1988-05-09
Abstract: Expansion dowel for anchoring in a bore with an undercut, the expansion dowel consisting of an expansion sleeve (10) having an axial bore (12, 14), tapering gradually to the front, for guiding an expansion body (26), and having, in the front section of the expansion sleeve, fins (28) formed by longitudinal slots, which fins (28) have an undercut shoulder (20) at the front end and are conically tapered on their outside, from the front in the direction of the undercut shoulder. A guide tube (30) for a set bolt (40) for driving the expansion body (26) is used for connection at the rearward end of the expansion sleeve (10), the guide tube carrying an external stop (36) and the set bolt carrying an external stop (42). 
<IMAGE>
Patent NO-884269-D0 (NO)
Inventor: RAGNARSSON GERT ANDERS
IPC: A61K31/44
Filed: 1988-09-27
Abstract: Preparation giving a controlled and extended release of both a dihydropyridine, e.g. felodipine and a  beta -adrenoreceptor antagonist, namely metoprolol as well as a method for the manufacture of the new preparation.
Patent NO-893052-D0 (NO)
Inventor: KLOSSNER BOTHO
IPC: C06B35/00
Filed: 1989-07-26
Abstract: The invention provides a process for the preparation of finely grained lead azide, in which aqueous solutions of lead nitrate and sodium azide are stirred in a vessel at constant temperature, characterized in that in a first process step the aqueous solution of lead nitrate and a small amount of an aqueous solution of sodium citrate are poured into the vessel, in a second process step, the aqueous solution of sodium azide is dosed into the vessel over a period of time of 30 to 40 minutes, the aqueous solutions poured into the vessel are agitated at a peripheral stirring speed of between 0.2 m/sec and 1.0 m/sec., and the constant temperature is set to a value of 50 DEG  C. to 80 DEG  C.
Patent NO-894465-D0 (NO)
Inventor: YOSHIDA MITSUHIRO
IPC: A61K31/505
Filed: 1989-11-09
Abstract: A pharmaceutical composition comprises (a) a pharmacologically effective amount of bunazosin or a pharmacologically acceptable salt thereof and (b) a monoglyceride of a fatty acid having 8 to 12 carbon atoms and/or a lactic acid ester of an aliphatic alcohol having 12 to 18 carbon atoms and is improved in percutaneous administration.
Patent NO-902946-D0 (NO)
Inventor: JOLLEY SCOTT T
IPC: C10M105/72
Filed: 1990-07-02
Abstract: A liquid composition is described which comprises (A) a major amount of a fluorine containing hydrocarbon containing one or two carbon atoms, and (B) a minor amount of a soluble organic lubricant free of acetylenic and aromatic unsaturation and comprising at least one sulfone or sulfoxide characterized by the formulae R1(R2)SO2 (I) R1(R2)SO (II)  wherein R1 and R2 are each independently hydrocarbyl groups, -R3O(O)CR4, -NR4R5 or -R3NR4R5 groups wherein R3 is a hydrocarbylene group, and R4 and R5 are each independently hydrocarbyl groups, or R1 and R2 are hydrocarbylene groups joined together to form a cyclic moiety including the sulfur atom, or R1 is a hydrocarbyl group and R2 is OR6 wherein R6 is a hydrocarbyl group. The liquid compositions exhibit excellent thermal stability and are useful particularly as refrigeration liquids in refrigerators and air-conditioners including auto, home and industrial air-conditioners.
Patent NO-903026-D0 (NO)
Inventor: GOIRE CHRISTIAN
IPC: G06F21/24
Filed: 1990-07-06
Abstract: The invention concerns a system consisting of a terminal linked by a transmission line to a central unit, the terminal comprising a memory divided into a program memory and a RAM-type working memory, the program memory itself comprising a volatile memory, an EEPROM or battery-operated RAM-type backup memory and a ROM or PROM-type non-volatile memory, characterized in that each of the memories constituting the program memory is divided into a non-certified area, the terminal further comprising an interpreter program, which performs the interpretation between a program written in a compact high-level and universal language and the language specific to the terminal microprocessor, the interpreter program being capable of accessing each of the memory divisions and a test program of the downloading system consisting of at least one CHSB instruction, whose command word is stored in one of the registers and expresses the downloading possibilities of the different areas.
Patent NO-922269-D0 (NO)
Inventor: WINTERSTEIN DONALD F
IPC: G01V1/42
Filed: 1992-06-10
Abstract: A method for geophysical exploration by analyzing shear-wave polarization directions relative to a fixed coordinate frame is disclosed, for either vertical seismic profile data or surface seismic reflection data. Energy in a selected time window of two off-diagonal components is determined, and the source and receiver coordinate frame is then rotated, and energy is again determined. A second rotation of the source and receiver coordinate frame is followed by a third energy determination. A simple trigonometric function equation is generated to fit the determined energy values, and a minimum energy value is determined. The coordinate frame is then rotated by the angle that gives the minimum energy value, so that all of the signal is put on the diagonal components. <IMAGE>
Patent NO-933481-D0 (NO)
Inventor: EMONDS-ALT XAVIER
IPC: A61P9/00
Filed: 1993-09-29
Abstract: The invention relates to basic quaternary amides of formula <IMAGE>  in which   - Ar represents an optionally substituted mono-, di- or tricyclic heteroaromatic or aromatic group; - T represents a direct bond, a hydroxymethylene group, an alkoxymethylene group in which the alkoxy group is C1-C4 or a C1-C5 alkylene group; - Ar' represents a phenyl which is unsubstituted or substituted one or a number of times, a thienyl, a benzothienyl, a naphthyl or an indolyl; - R represents hydrogen, a C1-C4 alkyl, an  omega -(C1-C4)alkoxy(C2-C4)alkyl or an  omega -(C1-C4)alkanoyloxy(C2-C 4)alkyl,   - Q represents hydrogen; - or else Q and R, together, form a 1,2-ethylene, 1,3-propylene or 1,4-butylene group;   - Am<(+)> represents the radical <IMAGE> in which X1, X2 and X3, together and with the nitrogen atom to which they are bonded, form an azabicyclic or azatricyclic system optionally substituted by a phenyl group;   - A<(-)> is a pharmaceutically acceptable anion.   These compounds are useful in the preparation of medicaments intended for the treatment of pathologies involving the tachykinin system.
Patent NO-941021-D0 (NO)
Inventor: HOLTON ROBERT A
IPC: C07D409/12
Filed: 1994-03-22
Abstract: 10-Desacetoxytaxol and its derivs. of formula (I) are new, where R2 = H or opt. protected OH; R3, R4 = H, opt. protected OH, Me, -SH, -NH2 or -NR8R9; R5 = R10 or -OR10; R6, R7 = H, alkyl or aryl; R8, R9 = H, alkyl, alkenyl, alkynyl or aryl; R10 = alkoxy, alkyl, alkenyl, alkynyl or aryl; provided that when R2 = H then R3 and R4 are not opt. protected OH. 10-Desacetoxytaxol and 10- desoxytaxotere, are specifically claimed.
Patent NO-952674-D0 (NO)
Inventor: GAASLAND STEIN
IPC: B29C45/00
Filed: 1995-07-06
Abstract: PCT No. PCT/DK94/00045 Sec. 371 Date Nov. 6, 1995 Sec. 102(e) Date Nov. 6, 1995 PCT Filed Jan. 27, 1994 PCT Pub. No. WO94/18384 PCT Pub. Date Aug. 18, 1994The invention describes a method for dispersion of cellulose based fibers in water. The raw material, which particularly may be recycled paper, is first wetted with water. By a combination of addition of hydrocolloid which binds water, and strong kneading at high solid content, the mixture is transformed into a modulable paste. The high viscosity of the paste effectively conveys the shear forces of the kneading machine to make the fibers flexible and tear them apart. When the kneading is terminated, the hydrocolloid prevents the fibers from reassociation into fiber bundles.
Patent NO-965099-D0 (NO)
Inventor: PEET NORTON PAUL
IPC: C07K5/08
Filed: 1996-11-29
Abstract: This invention relates to acylated enol derivatives of known elastase inhibitors. These compounds are useful in the treatment of various inflammatory diseases, including cystic fibrosis and emphysema or as prodrugs of compounds which are useful in the treatment of said diseases.
Patent NO-974209-D0 (NO)
Inventor: JUNG HAE-MOOK
IPC: H04N19/625
Filed: 1997-09-12
Abstract: An apparatus for encoding a digital video signal to reduce a transmission rate of the digital video signal, which comprises a feature point based motion compensation circuit for selecting a set of feature points from the reconstructed reference frame to detect a set of motion vectors between a current frame and a original reference frame corresponding to the set of feature points by using a feature point based motion estimation, and for generating a second predicted frame based on the set of motion vectors and the reconstructed reference frame. The feature point based motion estimation employs a convergence process in which a displacement of each of the feature points are given to a motion vector thereof and the six triangles of each of the hexagon are affine-transformed independently using the displacements of their vertex feature points. If the displacements provide a better PSNR, the motion vector of the subject feature point is sequentially updated. Therefore, the inventive convergence process is very efficient in the matching process to determine the predicted image as close as possible to the original image having zooming, rotation or scaling of objects.
Patent NO-990276-D0 (NO)
Inventor: JOHNSON DAVID
IPC: A61K49/00
Filed: 1999-01-22
Abstract: Ultrasound contrast agents comprising microbubbles of biocompatible gas, e.g. a sulphur halide or a perfluorocarbon, stabilized by opsonisable amphiphilic material, e.g. a membrane-forming lipid such as a phospholipid, especially a negatively charged phospholipid such as a phosphatidylserine, may exhibit prolonged contrast-generating residence time in the liver following intravenous administration.
Patent GB-0025811-D0 (GB)
Title: Secure dispensing of materials
IPC: B65D83/14
Filed: 2000-10-20
Abstract: Secure dispensing apparatus is described which is adapted to dispense e.g. a prescription drug from an axial compression dispensing device ( 1 ). This is located in a housing ( 10 ) including a dispensing aperture ( 16 ). The axial compression dispensing device ( 1 ) is located in a central chamber of axial length slightly longer than that of the axial compression dispensing device, and structures ( 30 ) are provided at one end of the chamber movable with respect thereto to compress the axial compression dispensing device to cause dispensing via the dispensing aperture ( 16 ). The structures ( 30 ) comprises a central breakable axial stem ( 33 ) attached to a pressure plate ( 34 ), the pressure plate having a surface configuration on its side facing away from the axial compression dispensing device providing a set of surfaces ( 35 ) not in a plane transverse to the axis of the breakable stem, and apertures ( 36 ) in the end of the outer housing aligned with the set of surfaces of the pressure plate and none of the apertures ( 36 ) being coaxial with the breakable stem ( 33 ). Structures such as a wall ( 15 ) are provided to limit the amount of movement of the pressure plate ( 34 ) away from the end ( 11 ) of the outer housing containing the set of apertures ( 36 ).
Patent GB-0107175-D0 (GB)
Title: Chassis for grass treatment machine
IPC: A01B45/00
Filed: 2001-03-22
Abstract: A chassis for a grass treatment machine on which an elongate grass treatment module having opposed outer ends may be mounted, and in which the chassis is intended to be mounted in, or form part of, the frame of a grass treatment machine. The chassis has two module mountings which are laterally spaced form each other with respect to the direction of travel of the machine, and each mounting being adapted to receive a respective outer end of the module. The chassis has two chassis portions which can be assembled in order to hold the outer ends of the module in the module mountings in order to mount the module on the chassis, and which can be relatively separated in order to provide access to the module mountings for the purposes of mounting or demounting the ends of the module relative to the chassis.
Patent GB-0108435-D0 (GB)
Title: Connection of a junction to an electrical conductor track on a plate
IPC: H01L23/13
Filed: 2001-04-04
Abstract: A connection of an electrical junction (13) to a conductor track (5) applied to a glass or glass ceramic plate (1) is to be resistant to temperature change and traction and conductive. For this purpose an electrically conductive connecting element (11) is ultrasonically welded to the composite consisting of the conductor track (5) and plate (1). The connecting element (11) extends to the terminal (13) which is fastened to the plate (1).
Patent GB-0214038-D0 (GB)
Title: Electric heating element
IPC: F24C15/20
Filed: 2002-06-19
Abstract: An electric heating element (10) for an oven (2) is provided at least in part with a coating (14) of a catalyst means. <IMAGE>