baber/WOPTO huggingface dataset:
Patent IL-139277-A0 (IL)
Title: Method for producing isoxazoline-3-yl acyl benzene
IPC: C07C205/44
Filed: 1999-05-04
Abstract: 3-(2-Alkylthio-5-acylphenyl)-isoxazoles (I) are prepared by a multi-stage process via 3-(2-aminophenyl)-isoxazole intermediates (VI). Also new are various oxime and isoxazole derivative intermediates, including (VI); and methods for preparing oximes (XV) and thioethers (XIX) . Preparation of 3-(2-alkylthio-5-acylphenyl)-isoxazoles of formula (I) involves preparing a 3-(2-aminophenyl)-isoxazole intermediate of formula (VI), then halogenating, thioalkylating, oxidizing and acylating to give (I). [Image] R 1, R 3-R 5 : H or 1-6C alkyl; or R 4+R 5 : a bond; R 2 : 1-6C alkyl; R 6 : heterocycle; n : 0-2. Independent claims are included for: (i) new oxime and isoxazole derivative intermediates of formulae (III), (X) (including (VI)) and (XII); (ii) the preparation of benzaldoxime derivatives of formula (XV), involving the reaction of toluene derivatives of formula (XVI) with an organic nitrite of formula R-ONO in presence of a base, where the process optionally further includes the conversion of the oxime group of (XV) into aldehyde, nitrile or nitrile oxide; (iii) the preparation of thioethers of formula (XIX), involving the reaction of an aniline of formula (XX) with a dialkylsulfide of formula R 2SSR 2 (VII) in presence of a catalyst; and (iv) new benzaldoxime compounds of formula (XV'). [Image] [Image] A : NO 2, NH 2 or SR 2; X : NO 2 or SO 2R y; R x, R y : inert substituents; m : 0-4; p : 0-5; R' 1 : H, 1-6C alkyl, halo, 1-6C alkoxy or 1-6C alkylthio; X' : S(O) nR' y; R' y : H, Cl or Br '' in the para position of the phenyl ring to X' '' (sic). ACTIVITY : Herbicidal. MECHANISM OF ACTION : None given.
Patent IL-144956-A0 (IL)
Title: Pesticide and/or plant growth regulating compositions
IPC: A01P21/00
Filed: 2000-03-07
Abstract: The invention concerns pesticide and/or insecticide and/or plant growth regulating compositions comprising specific dendrimers, said compositions being, in particular, useable for agriculture and/or public health or domestic hygiene; the invention also concerns methods for treating and/or protecting crops and/or for public health and domestic hygiene using said compositions. The invention further concerns specific dendrimers.
Patent IL-146878-A0 (IL)
Title: Interfaces between terminal users, satellites and hubs in a two-way satellite system
IPC: H01Q3/08
Filed: 2001-03-30
Abstract: A two-way satellite communication system that includes a terminal having a receiver unit and a transmitter unit is disclosed. The terminal is configured to transmit and receive signals to and from a hub via a satellite. A terminal interface is configured to permit exchange of data between the receiver unit and the transmitter unit, wherein the receiver unit is configured to translate data received from a host to a data frame that conforms to a predetermined protocol format that is supported by the hub. A demodulator interface is coupled to an antenna associated with the terminal and is configured to permit exchange of the data frame between the terminal and the satellite. The data frame conforms with a return channel frame format. A satellite-to-hub interface is configured to permit receipt of the data frame at the hub from the satellite. The hub is configured to modify the data frame for transmission to an external packet switched network. A hub-to-terminal interface is configured to support the exchange of data from the hub to the terminal using a multi-layer protocol.
Patent IL-148902-A0 (IL)
Title: A construction for automatically milking animals
IPC: A01J5/007
Filed: 2002-03-26
Abstract: A construction for automatically milking animals is provided with a milking robot and a computer which is capable of being connected with a number of measuring instruments which are related to a number of functions of the construction. A monitoring program for said functions is installed in the computer, with the aid of which the computer is suitable for determining, on the basis of a comparison of data from one or more of the measuring instruments with reference data related to said functions, a diagnosis in relation to an anticipated fault in one or more of said functions. The early determination of a diagnosis enables to warn a user and/or a service mechanic, who is then able to take in time the possibly required measures to avoid the anticipated malfunction.
Patent IL-150846-A0 (IL)
Title: Device for extracting a dental appliance
Inventor: MULLER ALEXANDRE
IPC: A61C3/16
Filed: 2001-02-02
Abstract: An instrument for removing a crown by generating a couple of forces between the occlusal surface of the stump of the tooth and the basal surface of the crown. The instrument has an indented intermediate portion and a working part extending from a tapered intermediate portion and a handle. When inserted in a groove formed at the occlusal part of the stump along a plane substantially parallel to the occlusal surface of the crown, the working portion enables, by a physical action, exertion of a couple of forces between the respective occlusal surfaces of the stump and the basal surface of the crown. The working part is rotatable integrally and correspondingly with a rotation of the handle.
Patent IL-151595-A0 (IL)
Title: Shortened synthesis of 3,3-diarylpropylamine derivatives
IPC: C07C227/08
Filed: 2001-06-11
Abstract: Optically active 3,3-diarylpropylamine derivatives are produced in six steps from 4-hydroxybenzoic acid or an alkyl 4-hydroxybenzoate and cinnamic acid via new and known phenyl-chromanone and phenyl-chromanol compounds. Production of optically active 3,3-diarylpropylamine derivatives of formula (I) comprises: (A) condensation of 4-hydroxybenzoic acid or an alkyl 4-hydroxybenzoate (II) with cinnamic acid; (B) reaction of the resulting (R,S)-2-oxo-4-phenylchromane of formula (III) with cinchonidine; (C) acidification of the (R)-2-oxo-4-phenylchromane cinchonidine salt of formula (IV) obtained; (D) isolation of the resulting (R)-6-carboxy-2-oxo-4-phenylchromane (V) and reaction of this, after conversion into an activated form, with an alcohol (VI); (E) reduction of the alkyl (R)-2-oxo-4-phenylchromane-6-carboxylate (VII) obtained with diisobutylaluminum hydride or lithium tri-tert.butoxyaluminum hydride; and (F) reductive amination of the resulting lactol (VIII) with a primary, secondary or tertiary amine. [Image] [Image] R : H; or 1-6C alkyl, preferably methyl or isopropyl, but R in compound (VI) is 1-6C alkyl); R', R'' and R 1>1-6C alkyl, preferably methyl or isopropyl. Independent claims are also included for: (a) the (R,S)-2-oxo-4-phenylchromane (III) (R = H); (b) the (R)-2-oxo-4-phenylchromane cinchonidine salt (IV); (c) the (R)-6-carboxy-2-oxo-4-phenylchromane (V); and (d) the (R)-hydroxybenzyl alcohol salt of formula (IX). [Image] - ACTIVITY : Uropathic. - MECHANISM OF ACTION : None given in the source material.
Patent IL-160940-A0 (IL)
Title: Adapter for mounting a faceplate of a first style on to an electrical outlet cavity of a second style
IPC: H01R31/02
Filed: 2001-09-25
Abstract: An adapter for mounting electrical outlet faceplates designed for mounting on rectangular junction boxes in hollow walls onto solid walls with cylindrical cavities and sleeves. Junction box mounting is popular in North America, whereas cavity mounting is popular in Europe and the Middle East. Such an adapter provides universal mounting for specialized faceplates which are designed and intended for junction box mounting. The adapter features clamps for gripping the inner surface of a wall cavity or sleeve and a rectangular plate for mounting an faceplate designed for junction box mounting. The rectangular plate has mounting points with a nominal center-to-center distance of 31/4  inches, corresponding to the requirements of junction box mounting. <IMAGE>
Patent IL-165816-A0 (IL)
Title: Use of cyclooxygenase-2 inhibitors for the manufacture of a medicament for the treatment and prevention of neoplasia
IPC: A61P43/00
Filed: 2004-12-16
Abstract: The present invention relates to a pharmaceutical composition for the treatment of a neoplasia, which comprises a compound of formula II and an anti-neoplastic agent
Patent IL-179281-A0 (IL)
Title: Rupturable opening for sealed container
IPC: B65D77/28
Filed: 2006-11-14
Abstract: A container formed from a paperboard laminate and including a rupturable opening for gaining access to the contents of the container, the opening being defined by an embossment pattern in a wall of the container. The embossment defines a weakened area which includes the layers of the laminate, but without destruction or deterioration of selected ones of the barrier/sealing layers of the laminate. A method is disclosed.
Patent IL-184051-A0 (IL)
Title: Acylated glp-1 compounds
Filed: 2007-06-19
Abstract: Protracted GLP-1 compounds and therapeutic uses thereof.
Patent IL-186504-A0 (IL)
Title: Methods and compositions for treatment of cns disorders
Filed: 2007-10-08
Abstract: The invention relates to methods and compositions for the treatment and prevention of CNS-related conditions. One of the CNS-related conditions treated by the methods and compositions of the invention is Alzheimer's disease.
Patent IL-187917-A0 (IL)
Title: Antiarrhythmic precursor compounds, methods of synthesis and methods of use
Filed: 2007-12-05
Abstract: The invention comprises compounds of Formula 1:   
wherein, R 1  is independently H or halogen; R 2  is, for example, H or --R 10 -NR 11 R 12 , and wherein R 10  is C 1 -C 6  alkyl, and R 11  and R 12  are independently H, C 1 -C 4  alkyl, and hydrates, solvates, salts and tautomers thereof. The invention further comprises methods for making the compounds of the invention and methods for making compounds useful in the treatment or prevention of cardiac arrhythmia from the compounds of the invention.
Patent IL-190056-A0 (IL)
Title: Collision safety device being applicable to infant seats
Filed: 2008-03-10
Abstract: This safety device is characterised by being made up by a chamber (1) of flexible walls being filled with air and comprising a nipple (5) being such as to facilitate the progressive outflow of the air when the chamber (1) is highly pressed. Said nipple (5) has valve means (6) being such as to prevent the accidental outflow under low pressures of the air occupying the chamber (1) and to give way when receiving a high pressure thereby facilitating the outflow of the air. Said chamber (1) will be preferentially subdivided into several departments (2, 3 and 4) each of them having a nipple (5) for the outflow of the air. The chamber (1) and the valve means (6) are arranged in the inside of the complementary side members (7) of the backrest (8) of the infant seat and in the complementary side members (9) of the headrest (10) of said backrest.
Patent RO-127175-A0 (RO)
Title: Process for the rehabilitation and corrosion protection of water supply pipes by coating with mortar
Inventor: BRAI LEON DUMITRU
IPC: B05D7/14
Filed: 2011-03-07
Abstract: The invention relates to a process for the rehabilitation and corrosion protection of water supply pipes. The claimed process consists in preparing the working site, disconnecting the pipe section to be rehabilitated, mechanically coarsely cleaning the same, visualizing the inside of the pipe with a video camera, applying the mortar paste lining by using a high pressure pump with an adjustable flow rate of up to 150 l/min and a guniting equipment driven by a motor, in-built on a frame with a mechanically-adjusted travelling speed so as to adhere and react with the pipe walls ensuring a uniform coating with low roughness, then the pipe is closed at both ends, it is filled with water up to 5...10% and, for a period of 3 to 7 days, there takes place the hydration and, after carrying out the pressure test, the connections and branches are restored, the rehabilitated pipe is inspected with a videocamera and it is put into operation.
Patent RO-135793-A0 (RO)
Title: Biostimulant for plants based on keratin hydrolyzate and eutectic solvents and process for preparing the same
Inventor: OANCEA FLORIN
IPC: A01N63/10
Filed: 2021-12-29
Abstract: The invention relates to a biostimulant composition for plants and to a process for preparing the same. According to the invention, the composition consists of 47.03 ... 51.96% soluble keratin, 30.34 ... 33.46% 2,3-butanol, 15.67 ... 17.28% choline chloride, 2.02 ... 2.23% water and has a proton pump induction activity in tomato test plants of at least 175% compared to the witness. According to the invention, the process consists of the following steps: preparing the eutectic solvent from choline chloride, 2,3-butanediol isomer 2R, 3R and water, extracting keratin from wool or feathers, filtration under pressure, ultrafiltration to recover the eutectic solvent from the filtrate, recovering the retentate which is used as a biostimulant for plants by seed treatment.
Patent AP-2004003094-A0 (AP)
Title: Metabolities of (3-{[4-tert-butyl-benzyl)-(pyridine-3-sulfonyl)-amino]-methyl}-phenoxy)-acetic acid
Inventor: CAMERON KIMBERLY O'KEEFE
IPC: A61P1/02
Filed: 2003-01-20
Abstract: the present invention relates to metabolities of (3-{[4-tert-butyl-benzyl)-(pyridine-3-sulfonyl)-amino]-methyl}-phenoxy)-acetic acid
Patent MA-23344-A1 (MA)
IPC: A61K47/44
Filed: 1994-10-06
Abstract: PCT No. PCT/SE94/00926 Sec. 371 Date Jan. 30, 1995 Sec. 102(e) Date Jan. 30, 1995 PCT Filed Oct. 5, 1994 PCT Pub. No. WO95/09609 PCT Pub. Date Apr. 13, 1995The present invention is related to a pharmaceutical formulation which is an oil-in-water emulsion for parenteral and oral use which comprises (i) an emulsion-stabilizing surface active drug in high concentration; (ii) optionally a pharmacologically inert oil; (iii) optionally a surfactant; (iv) water or a buffer; and (v) an agent giving isotonicity to the final formulation; the use of and a process for preparation of the formulation.
Patent MA-25266-A1 (MA)
Inventor: NEIL D BLAZEY
IPC: A23C19/028
Filed: 2001-06-01
Abstract: The invention relates to a simplified, rapid method which is suitable for making a variety of cheese and cheese products, including natural and processed cheese, in a single installation with common equipment. In particular, the invention concerns a method of making cheese, comprising the steps of: (a) concentrating milk or a reconstituted dry milk, having its pH adjusted to about 5.0 to 6.8, by ultrafiltration and diafiltration to produce a retentate; (b) supplementing said retentate with a protein concentrate or isolate and, optionally, fat and/or flavor; and (c) heating the mixture to produce a smooth consistency.
Patent MA-37404-A1 (MA)
Title: Dispositif et methode de controle et de validation du graissage manuel
Inventor: SAINT-MARD MICHEL
IPC: G01F11/00
Filed: 2013-03-13
Abstract: La présente invention se rapporte à un dispositif de contrôle et de validation du graissage manuel pour une installation munie d'au moins un point de graissage (12), ledit dispositif comprenant : - des moyens d'identification (4, 11) dudit point de graissage (12 ), - des moyens (8) pour mesurer la quantité de graisse injectée et, - des moyens (9) pour déterminer si la graisse injectée est bien acheminée jusqu'au point de graissage (12), lesdits moyens comportant un capteur de pression et/ou un capteur ultrason.
Patent MA-56080-A1 (MA)
Title: Plateforme collaborative de partage sécurisé de l’information dans le domaine de l’éducation
Inventor: Badr ABOU EL MAJD
IPC: G06F21/30
Filed: 2022-03-14
Abstract: La présente invention a pour objet une plateforme technologique décentralisée et sécurisée qui permet à l’apprenant l’accès et le suivi de ses parcours éducatifs. La plateforme permet à chaque apprenant de stocker ses informations d’éducation (de la maternelle jusqu’au supérieur), ses parcours éducatifs (scolaires, civique, professionnel, culturelle et artistique, santé et bien-être), ses compétences, ses activités extra-scolaire… chaque apprenant sera équipé d’une carte format carte bancaire, qu’on nomme edu@pass, avec un qr-code qui lui permet de décider de ce à quoi il donne accès et de ce qu'il souhaite récupérer. La plateforme permet la collecte, le suivi, la structuration et le partage des données d’éducation, véhiculées par les apprenants eux-mêmes pour aboutir à des modèles d'intelligence artificielle (ia) automatisés et collaboratifs de prévention et d’orientation personnalisée. Les données de chaque apprenant sont stockées sur un serveur privé de cloud connecté à d’autres espaces numériques de travail.
Patent UY-26159-A1 (UY)
Title: Método para realzar la celulosa y modificar la biosíntesis de la lignina en las plantas
Inventor: CHADRASHEKHAR VINCENT L CHIANG
IPC: C12N9/10
Filed: 2000-05-23
Abstract: Este invento se refiere a moléculas de polinucleótidos que codifican la sintasa de la celulosa, promotores de la sintasa de la celulosa y polipéptidos de la sintasa de la celulosa, métodos para, genéticamente, alterar la biosíntesis de la celulosa y de la lignina y métodos para mejorar las propiedades de fuerza de la madera joven y de las fibras en los árboles. El invento también se refiere a métodos para identificar elementos regulatorios en un promotor de la sintasa de la celulosa y los factores de transcripción que ligan o enlazan a dichos elementos reguladores y a métodos para aumentar la expresión de los polinucleótidos, imperablemente ligados o enlazados a un promotor de la sintasa de la celulosa.
Patent UY-26190-A1 (UY)
Title: Compuestos de tiazol y composiciones farmacéuticas para inhibir a las proteinquinasas y métodos para su utilización
Inventor: BENDER SHAO SON CHU LARRY ANDR
IPC: C07D417/04
Filed: 2000-06-02
Abstract: Se describen compuestos de diaminotiazol que modulan y/o inhiben la actividad de determinadas proteinquinasas. Estos compuestos y composiciones farmacéuticas que los contienen son capaces de mediar la transducción de la senal de la tirosinquinasa para modular y/o inhibir la proliferación de células no deseadas. La invención también se refiere al uso farmacéutico o profiláctico de composiciones farmacéuticas que contienen dichos compuestos y a métodos de tratamiento del cáncer y otros estados de enfermedad asociados con una angiogénesis y/o proliferación celular no deseada, como por ejemplo la retinopatía diabética, el glaucoma neovascular, la artritis reumatoide y soriasis, mediante la administración de cantidades efectivas de dichos compuestos.
Patent UY-28548-A1 (UY)
Title: Método y aparato para reducir compuestos oxígeno-metal
Inventor: KOOIJ CHRISTIAAN JOHANNES
Filed: 2004-10-04
Abstract: Método y aparato para reducir compuesto oxígeno-metal (en adelante compuesto) donde el carbono actúa como agente reductor, comprendiendo: a) Primera rezcción: pasar gas CO en cámara de reacción conteniendo dicho compuesto, bajo condiciones tales que el CO sea convertido en carbono sólido y dióxido de carbono introduciendo de esta forma carbono sólido en el compuesto,y b) Segunda etapa: que el carbono, introducido en el compuesto, reduzca dicho compuesto, donde estápresente, al menos en dicha segunda etapa de reacción, un primer material promotor efectivo para promover reducción del compuesto, comprendiendo el primer material promotor el mismo y/o un compuesto del mismo.
Patent UY-29719-A1 (UY)
Title: Mejora sobre patente de invencion ns 13.219 " nuevo picaporte cerradura y llave con sus 4 caras, 4 cantos y 8 aristas
Inventor: TOCCHIETTO DANTE VIRGILIO
IPC: E05B55/14
Filed: 2006-08-01
Abstract: mejora sobre Patente de Invencion NS 13.219 relativo a "NUEVO PICAPORTE CERRADURA Y LLAVE CON SUS 4 CARAS, 4 CANTOS Y 8 ARISTAS" caracterizado por ser un nuevo sistema de picaporte que funciona sin girar el pomo, basta para hacerlo con apretar un boton ubicado en la parte superior de este, al apretar este boton, entra a funcionar un mecanismo de empuje que llega hasta el pestillo pasador y lo desplaza hasta liberar la puerta del marco.
Patent UY-30842-A1 (UY)
Title: Derivados de n-(amino-heteroaril)-1h-pirrolopiridin-2-carboxamidas, su preparacion y su aplicacion en terapéutica
Inventor: GILLE CATHERNIE
IPC: A61K31/397
Filed: 2007-12-26
Abstract: La invencion se refiere a compuestos derivados de n-(amino-(hetero)aril)-1h-pirrolopiridin-2carboxamidas, de la formula general (I): En el estado de base o de sal de adicion a un ácido, así como en el estado de hidrato o de solvato, en la que los sustituyentes e índices están especificados en la memoria y la prevencion y el tratamiento de las patologías en las que están implicados los receptores de TRPV1.
Patent UY-30896-A1 (UY)
Title: Composicion fitosanitaria
Inventor: EGON DR HADEN
IPC: A01N43/56
Filed: 2008-02-06
Abstract: La presente invencion se refiere a una composicion que contiene (A) un fungicida de carbamato específico y (B) un insecticida específico, el uso de esta composicion para aumentar la fitosanidad y un método para aumentar la fitosanidad mediante el tratamiento a una planta, sus propágulos o el locus donde la planta está creciendo o crecerá con la composicion anterior.
Patent UY-31148-A1 (UY)
Title: Compuestos de piperazina con accion herbicida (ii)
Inventor: KIBLER ELMAR
IPC: A01N33/00
Filed: 2008-06-12
Abstract: Compuestos de piperazina de la fórmula general I en la fórmula I, las variables R1, R2, R3, R4, R5, R6, R7, R8, R9 y R10 se definen en la descripción, y a su uso como herbicidas. Además agentes destinados a la protección de plantas y un procedimiento para combatir el crecimiento de plantas indeseadas.
Patent AT-512490-A1 (AT)
Title: Hochdrucknebelanlage
IPC: B05B7/08
Filed: 2012-01-16
Abstract: Hochdrucknebelanlage (1) mit einem Kompressor (3) und einem Vernebelungsventil (5) zur Erzeugung von schwebefähigem Nebel eines flüssigen Mediums, wie z.B. Wasser, wobei das Vernebelungsventil (5) mit einer elektronischen Steuerung verbunden ist, und wobei die Hochdrucknebelanlage (1) Mittel zum Anschluß mindestens eines weiteren Vernebelungsventils (5) aufweist, die Steuerung Mittel zum Anschluß mindestens eines Sensors aufweist, und in der Steuerung ein Programm zur Umrechnung von Daten mindestens eines Sensors in getrennte Steuerbefehle mindestens zweier Vernebelungsventile (5) gespeichert ist.
Patent CH-709202-A1 (CH)
Title: Montre à dispositif de recharge en énergie électrique.
Inventor: BULGARI GIORGIO
IPC: G04G19/00
Filed: 2014-01-17
Abstract: L’invention a pour objet une montre (1) comprenant un dispositif destiné à recharger une unité de fourniture d’énergie (2), telle que, par exemple, un accumulateur ou un condensateur. Le dispositif de recharge comporte un générateur électrique (4) et une lunette tournante (5) en liaison cinématique avec le générateur (4).
Patent DZ-1427-A1 (DZ)
Inventor: PETERSEN LARS-GORAN
IPC: H04Q11/04
Filed: 1990-06-17
Granted: 2004-09-13
Abstract: A wideband connection between subscribers G and B is throughconnected in a digital time switch module. Information arriving from the transmitting subscriber G is stored in a speech store (SS) on store locations (SM) corresponding to the channel numbers (8, 11, 17, 31) of G. The receiving subscriber B is assigned channels (7, 14, 21, 26). The channel numbers of G are stored in store locations (MM) of a matrix store (MS), and can be read-out via horizontal (HI) and vertical (VI) inputs. A fixed address number (6) is stored in a pointer store (PS) on store location (PM) corresponding to the channel numbers of subscriber B. When establishing the wideband connection, an internal address number (M) is written into a difference store (OS) on a store location (OM) having the address of the fixed address number (6). A time slot counter (TSC) steps forward the time slots (7, 15, 21, 26) of subscriber B and addresses the pointer store (PS), wherein the address number (6) addresses the difference store (OS). On each addressing occasion, the internal address number (M) is read-out to one of the vertical inputs (VI = 18) and the time slot counter (TSC) addresses the horizontal inputs (HI) at the same time. The channel numbers of subscriber G in the store locations (MM) address the speech store (SS) and the content of the store locations (SM) are read-out to the channel numbers of subscriber B. Only the internal address number (M) need to be written-in when establishing the connection.