baber/WOPTO huggingface dataset:
Patent CZ-304045-B6 (CZ)
Title: Use of copper complexes containing 2-phenyl-3-hydroxyquinolin-4(1H)-one and 1,10-phenanthroline derivatives for preparing medicaments intended for the treatment of tumor diseases
Inventor: TRAVNICEK ZDENEK
IPC: A61K31/4709
Filed: 2012-04-10
Abstract: In the present invention, there is disclosed the use of copper complexes in oxidation stage +II and crystalline solvates thereof of the general formula [Cu(qui)(Rinphen)]X as expressed by a structural formula (I), in which the symbol qui represents 2-phenyl-3-hydroxyquinolin-4(1H)-onate anion, the symbol Rin, wherein n = 1to 4, represents a substituent or substituents on 1,10-phenanthroline(phen), in which R1 denotes a substituent being selected from the group consisting of: hydrogen, 4-methyl, 5-methyl, 5-nitro, 5-chloro, and/or if R1 is 5-methyl, then R2 is 6-methyl, if R1 is 4-phenyl, then R2 is 7-phenyl, if R1 is 3-methyl, then R2 is 4-methyl, R3 is 7-methyl and R4 is 8-methyl, as expressed by the corresponding formulae [Cu(qui)(4-methylphen)]X, [Cu(qui)(5-methylphen)]X, [Cu(qui)(5-nitrophen)]X, [Cu(qui)(5-chlorophen)]X, [Cu(qui)(5,6-dimethylphen)]X, [Cu(qui)(4,7-diphenylphen)]X, [Cu(qui)(3,4,7,8-tetramethylphen)]X, and where the X represents a monoanion of an acid being selected from the group consisting of: Fe-, Cle-, Bre-, Ie-, NOi3e-, BFi4e-, BPhi4e-, HCOOe-, CHi3COOe-, ClOi4e-, HSOi4e-, for the preparation of medicaments intended for the treatment of lung carcionoma and/or for the treatment of a malignant melanoma and/or for the treatment of cancer of the cervix and/or carcinoma of the ovary and/or cisplatin-resistant human tumor line of carcinoma of the ovary and/or for the treatment of prostatic carcinoma.
Patent CZ-307272-B6 (CZ)
Title: A compact unit for accumulation of electricity with a closed cooling system with condensation of air humidity located beneath the earth's surface and its functions
Inventor: CHLEBIŠ PETR
IPC: H02B7/08
Filed: 2014-11-30
Abstract: A compact unit for accumulation of electricity with a closed cooling system with condensation of air humidity located beneath the earth's surface. It solves the conceptual arrangement of the subsurface earth accumulating station of electrical energy using electrochemical accumulators (3) and a semiconductor converter (4). From the construction perspective, all technologies are combined into a mechanically compact unit, which is placed in an underground pit (1) by means of a lifting mechanism (17). This solves the problems connected with the complicated building and architectural placement of the accumulating stations of electricity, and it further solves the main problem of cooling the whole technology by dehumidifying the air in the underground space. The compact mechanical arrangement addresses the problem of simple handling of the accumulating station of electrical energy, both during the assembly and the maintenance. The subject of the invention is also a method of cooling the technology.
Patent CZ-307705-B6 (CZ)
Title: A stent loader
Inventor: VOLENEC KAREL
IPC: A61F2/95
Filed: 2017-07-25
Abstract: The stent loader consists of an insertion tube and running inside it a smaller tube (5) with an olive (6). The insertion tube consists of a spreading piece (1) made of controllable segments (1.1) and an extending piece (2) connected to this spreading piece (1). The controllable segments (1.1) are connected together by interlocking coupling elements connected with a sliding release (1.3). The spreading piece (1) is usually connected to the extending piece (2) by a separating piece (3) and the spreading piece (1) is preferably made of absorbent material capable of physically absorbing or chemically bonding the therapeutic agent.
Patent SK-288910-B6 (SK)
Title: Measuring assembly with conical calorimeter for measuring the fire risk of flammable liquids.
Inventor: MARTINKA JOZEF
IPC: G01N37/00
Filed: 2017-11-22
Abstract: Conical calorimeter measuring device for measuring the fire risk of flammable liquids consists of a conical calorimeter (15) made according to ISO 5660-1: 2015. A sample of combustible liquid is exposed to heat from the conical emitter (10) in the sample vessel (1). The sample vessel (1) is placed on the first fixed substrate (9) by means of a first adjustable height stand (8). The combustion products are fed through the digester (11) to the suction line (12) where the concentration of oxygen, carbon monoxide, carbon dioxide and optionally other gases is measured by the combustion gas analyzer (13) and the fuming coefficient of the burning products by the light beam intensity meter (14). A conical radiator (10), a digester (11), a suction line (12), a gas analyzer (13), and a light beam drop meter (14) are part of a conical calorimeter (15). The sample vessel (1) is sampled by means of a flexible hose (2) connected to the container (3) so as to form coupled containers. The diameter of the container (3) is greater than the diameter of the container (1) on the sample. The hopper container (3) is placed on the scales (5) by means of a second height-adjustable stand (4) which continuously weighs the weight loss of the sample. The scales (5) are located on the second fixed support (7). The edge of the sample vessel (1) is protected by the radiation shield (6) from exposure to the radiation from the conical emitter (10) so that only the surface of the combustible test fluid, but not the walls of the container (1), is exposed to the heat radiation from the conical emitter (10) on the sample.
Patent SK-285861-B6 (SK)
Title: Fungicide mixtures based on pyridine carboxamides and method of fighting fungi
Inventor: SCHELBERGER KLAUS
IPC: A01N37/00
Filed: 1998-12-15
Abstract: Fungicide mixtures containing as active components a) an amide compound of formula (Ib) wherein R4 represents halogen and R11 represents phenyl which is substituted by halogen and b) fungicides from the group of dicarboximides of formula (IIa) to (IId) and/or c) pyrimidine derivatives of formula (III) in which R represents methyl, propyne-1-yl or cyclopropyl and/or d) at least one active components of formula (IV) or (V) and/or e) derivates from the group of formula (VIa), (VIb) and (VII) and/or f) dinitroaniline of formula (VIII) and/or g) arylsulfamide of formula (IXa) or (IXb). The active components are provided in a synergistically effective quantity. It is described method of controlling harmful fungi.
Patent CZ-289241-B6 (CZ)
Title: Cutting and transporting mechanism for stalk agricultural products
Inventor: ARNOLD RUDOLF
IPC: A01D43/08
Filed: 2001-05-24
Abstract: The pivot axle (11) of the rotary discharger (12,13) is situated inside the circumference of the conveyor disc(s) (4,5) and is driven in the same rotary direction as the conveyor disc(s). The periphery of each coaxial conveyor disc has tines (7). The discharger is in the form of a toothed (14) disc above or below the conveyor disc, each of which has its own discharger. At right angles to the plane of the conveyor discs is a wall (15) spaced a little apart from the conveyor discs and the dischargers, and forming a conveyor duct (17).
Patent CZ-300315-B6 (CZ)
Title: Bicyclic derivatives of imidazo-3-yl-amine, substituted on a six-membered ring
Inventor: GERLACH MATTHIAS
IPC: B29D30/52
Filed: 2000-09-18
Abstract: The present invention relates to bicyclic imidazo-3-yl-amines of the general formula (I) being substituted on a six-membered ring, exhibiting analgesic activity, and being provided in the form of bases or of pharmaceutically acceptable salts thereof. The invention also relates to a process of their preparation, their use, and to medicaments containing them.
Patent CZ-305079-B6 (CZ)
Title: Burner air/fuel ratio regulation method and apparatus
Inventor: TESAR MICHAEL G
IPC: F23N5/18
Filed: 2000-10-17
Abstract: Control system and method for regulating the air/fuel mix of a burner for a web dryer or a regenerative or recuperative oxidizer, for example. Differential air pressure is monitored between the air chamber (21) of the burner and the enclosure (15) into which the burner fires (such as a flotation dryer or the combustion chamber of a regenerative thermal oxidizer). Fuel flow is monitored by a differential pressure measurement between the fuel chamber (22) of the burner (10) and the enclosure (15) into which the burner (10) fires. Signals obtained from these measurements are compared to non-linear predetermined values, and based on the comparison, the flow of air and fuel to said burner via the fuel and airflow control means in response to said comparison are regulated.
Patent CZ-303003-B6 (CZ)
Title: Fiber-reinforced pressure vessel and process for producing thereof
Inventor: DEBECKER ANDY
IPC: B32B5/02
Filed: 2001-02-01
Abstract: The present invention relates to a fiber-reinforced pressure vessel (1, 6) comprising a rigid gas- or fluid-tight body (2, 7, 13, 19) overwound with fiber filaments (3, 10, 11, 18), whereby the fiber filaments (3, 10, 11, 18) are wound such that at least a number of fiber filaments can freely move in respect of one another and when the pressure vessel (1, 6) is under internal pressure the fiber filaments are strained exactly in their longitudinal direction. The invention also relates to a method of manufacturing the above-described fiber-reinforced pressure vessel (1, 6) comprising a rigid gas-or fluid-tight body (2, 7, 13, 19) overwound with fiber filaments (3, 10, 11, 18), whereby the method comprises the steps of: a) providing a rigid gas-or fluid-tight body (2, 7, 13, 19), fiber filaments (3, 10, 11, 18) and a winding apparatus; b) overwinding the rigid body (2, 7, 13, 19) such that at least a number of fiber filaments (3, 10, 11, 18) can move freely with respect to one another and the fiber filaments (3, 10, 11, 18) are wound such that when the pressure vessel (1, 6) is under internal pressure the fiber filaments (3, 10, 11, 18) are loaded exactly in their longitudinal direction; whereby no matrix material (for example, resin) is provided such that the fiber filaments (3, 10, 11, 18) would be incorporated in a matrix for that section of the pressure vessel (1, 6) in which the fiber filaments (3, 10, 11, 18) can move freely with respect to one another.
Patent SK-285679-B6 (SK)
Title: Benzamide derivative and medicament containing the same and their use
Inventor: KATO HIDEO
IPC: A61K31/00
Filed: 2000-02-02
Abstract: It is described a benzamide derivative of the general formula (I), in which R represents C3-6 alkyl, or salts thereof and drugs containing these derivatives as the active ingredient and a use these derivatives for a manufacture of a medicament for therapeutic or preventive of a digestive disease.
Patent SK-287549-B6 (SK)
Title: Pharmaceutical composition and products comprising acryloyl distamycin derivative as active ingredient and use of said derivative
Inventor: GERONI MARIA CRISTINA ROSA
IPC: A61P35/00
Filed: 2001-06-20
Abstract: A pharmaceutical composition comprising an antineoplastic topoisomerase inhibitor of type I or II and acryloyl distamycin derivative of formula (I) wherein R1 is bromine or chlorine atom and R2 is distamycin or a defined derivative thereof. Brostallicin is the preferred acryloyl distamycin derivative of formula (I). As the preferred topoisomerase inhibitors of type II are in the pharmaceutical composition present doxorubicin or etoposide. Also disclosed are products comprising aforementioned active substances as combined preparations for simultaneous, separate or sequential use in the treatment of tumors and the use of acryloyl distamycin derivative of formula (I) for the preparation of a medicament for use in the combination therapy with an antineoplastic inhibitor of type I or II in the treatment of tumors, in the prevention or the treatment of metastasis or in the treatment of tumors by inhibition of angiogenesis.
Patent CH-704112-B8 (CH)
Title: Verfahren und Überwachungssystem zum Bestimmen der Turbinenschaufelverformung.
Inventor: HOYTE SCOTT
IPC: F01D21/04
Filed: 2008-05-27
Abstract: Verfahren zum Bestimmen der radialen Verformung einer Schaufel (4, 9) in einer Gasturbine (2), das Folgendes einschliesst: 1) Vornehmen einer anfänglichen Messung der Schaufel (4, 9) mit einem oder mehreren Näherungssensoren, die um den Umfang einer Stufe von Schaufeln (4, 9) angeordnet sind, 2) nach der anfänglichen Messung, Vornehmen einer zweiten Messung der Schaufel (4, 9) mit dem einen oder den mehreren Näherungssensoren, und 3) Durchführen einer Bestimmung der radialen Verformung der Schaufel (4, 9) durch Vergleichen der anfänglichen Messung mit der zweiten Messung. Die anfängliche Messung und die zweite Messung können vorgenommen werden, während die Turbine (2) arbeitet.
Patent CH-703554-B8 (CH)
Title: Einlassmischerhalterung für einen Strahlpumpeneinspannaufbau eines Siedewasserreaktors (SWR) und Verfahren zum Anbringen einer Einlassmischerhalterung.
Inventor: DEFILIPPIS MICHAEL S
IPC: G21C15/25
Filed: 2011-08-02
Abstract: Die erfindungsgemässe Einlassmischer-Halterung (30) für einen Strahlpumpeneinspannaufbau eines Siedewasserreaktors umfasst ein Halteband (40) mit Anbringungsblöcken(32, 34) und eine Einspannklammer (12). Das Halteband (40) wird durch die Mischerhalterungs-Anbringungsblöcke (32, 34), die direkt an der Einspannklammer (12) angebracht werden können und das Halteband (40) an der Einspannklammer (12) fixieren, an seiner Stelle gehalten. Durch das Befestigen des Haltebands (40) an der Einspannklammer (12) stellt das Halteband einen einstellbaren Kontaktpunkt zwischen der Einspannklammer (12) und dem Einlassmischer (2) bereit, wodurch der Einlassmischer (2) auch dann stabilisiert wird, falls die herkömmlichen Stellschrauben an der Einspannklammer (12) versagen. Daher wird die Einlassmischer-Position selbst dann aufrecht gehalten, wenn sich die Stellschrauben aus ihrer Position bewegen. Zudem wird die Abtrennung und/oder die teure und zeitaufwändige Reparatur der Stellschrauben, falls die Stellschrauben versagen sollten oder anderweitig eine Wartung erfordern, verhindert. Weiter betrifft die Erfindung ein Verfahren zum Anbringen der Einlassmischer-Halterung.
Patent EP-0913955-B8 (EP)
Inventor: BROWN PAUL A
IPC: H04B3/54
Filed: 1995-04-20
Granted: 2006-06-07
Abstract: Communications apparatus is disclosed which is adapted for use with a mains electricity transmission and/or distribution network, and includes signal transmission and/or reception means (232), and frequency conversion means (200-208) for converting the frequency of a signal transmitted or received by signal transmission and/or reception means to a frequency which facilitates improved propagation of the signal on the network. Preferably the signal transmission and/or reception means is adapted to operate according to a telephony standard which uses a relatively high carrier frequency (e.g. CT2), and the frequency conversion means is usable to convert a signal having a relatively high carrier frequency to a signal having a lower carrier frequency. <IMAGE>
Patent BR-PI0204125-B8 (BR)
Title: processo de obtenção de micro e nanoesferas de poli (e - caprolactona) na incorporação de isoniazida, composto com atividade antimicobacteriana
Inventor: AMANDA FERNANDES DE OLIVEIRA
IPC: A61K9/52
Filed: 2002-09-25
Abstract: "processo de obtenção de micro e nanoesferas de poli (<sym>-caprolactona) na incorporação de isoniazida, composto com atividade antimicobacteriana". este processo descreve a preparação de micro e nanoesferas de polímero biodegradável poli(<sym>-caprolactona) pelo método modificado de emulsificação com evaporação de solvente e pelo método modificado de emulsificação e difusão espontânea de solvente. esta técnica foi aplicada à incorporação, pela matriz polimérica, de isoniazida, composto com atividade antituberculose. neste processo, dissolve-se o tensoativo (tween 40) em água, sob agitação, até se formar uma solução. em outro recipiente dissolve-se o polímero juntamente com isoniazida em acetato de etila (no caso das microesferas) ou em uma mistura de etanol e acetona (no caso das nanoesferas). a solução de polímero com isoniazida é adicionada gota a gota utilizando-se um dispositivo construído por adaptação de um bulbo de borracha na parte superior de uma microseringa de 1,00 ml. após a adição, a microemulão é formada, o solvente é evaporado por agitação mecânica, as partículas são recolhidas por centrifugação e liofilizadas. este sistema foi caracterizado quanto às suas propriedades físico-químicas utilizando-se as técnicas microscopia eletrônica de varredura, em que se observou formas arredondadas com superfície lisa e baixa polidispersidade e microscopia de epifluorescência, que confirmou a presença de isoniazida incorporada ao polímero.
Patent BR-PI0410996-B8 (BR)
Title: sistema de filme de fixação, conjunto, métodos de preparar um sistema de filme de fixação e um conjunto e artigo absorvente descartável
Inventor: JOHANN F PETERSEN
IPC: A44B18/00
Filed: 2004-05-10
Abstract: "sistema de filme de fixação, conjunto, métodos de preparar um sistema de filme de fixação e um conjunto e artigo absorvente descartavel". a presente invenção refere-se a um sistema de filme de fixação (1) compreendendo um costado (7) e uma camada adesiva (6) sobre uma das duas superfícies principais do costado (7), o costado (7) portando sobre sua superfície principal exposta 3a, oposta à camada adesiva (6), uma pluralidade de elementos de fixação machos (4) capaz de se encaixar com materiais fibrosos (32) tendo uma pluralidade de elementos de fixação fêmeas complementares, e uma pluralidade de furos traspassantes (2) se estendendo através da espessura 11 do costado (7), de modo que a camada adesiva (6) ligada ao costado (7) seja exposta através desses furos traspassantes (2), onde pelo menos um dos mencionados furos traspassantes (2) é circundado pelo costado (7), e onde o sistema de filme de fixação (1) adere de modo liberável aos mencionados materiais fibrosos (32) através de uma combinação de um mecanismo de colagem mecânica e adesiva.
Patent BR-PI0518368-B8 (BR)
Title: artigo absorvente descartável tendo envoltórios para as pernas e método de fabricar o mesmo
Inventor: ANDREW WRIGHT
IPC: A61F13/15
Filed: 2005-12-06
Abstract: artigo absorvente descartável tendo envoltórios para as pernas e método de fabricar o mesmo. uma estrutura de envoltório para perna é fornecida em um traje absorvente descartável tal como uma fralda ou calças de treinamento. a estrutura de envoltório para perna tem uma camada base, uma camada superior, e uma construção de elástico disposta entre elas. a construção de elástico inclui uma pluralidade de elementos elásticos (por exemplo, faixas ou fios) espaçados uns dos outros (por exemplo, geralmente igualmente espaçados) que são alinhados em uma relação geralmente paralela. adicionalmente, a camada superior e de base definem uma região de inelasticidade. a estrutura de envoltório para perna fornece formação eficiente de um reservatório e uma pluralidade de barragens de fluido, cada uma capturando uma quantidade de fluido para minimizar a ocorrência de vazamentos de fluido a partir do artigo absor- vente. métodos de formar tais artigos absorventes são descritos.
Patent BR-PI0520049-B8 (BR)
Inventor: CHANG-KWON KO
IPC: A61K35/32
Filed: 2005-08-03
Abstract: A method for producing the fibrin contained semi-solid osteoblast composition has developed for treating the bone fracture. The method is comprised of: isolating osteoblasts from a bone tissue and culturing/proliferating the isolated osteoblasts in Dulbecco's Modified Eagle's Medium (DMEM) or Minimum Essential Medium, Alpha Modification (alpha-MEM) to prepare an osteoblast suspension. Then, mixing the resulting osteoblast suspension with a coagulation factor to prepare an osteoblast therapeutic agent. Accordingly, the fibrin contained semi-solid osteoblast composition of the present invention has capability to achieve the bone grafting for performing bone union without the clinical graft rejection. It is possible to uniformly distribute the fibrin mixed semi-solid osteoblast composition into the affected area of the bone fracture via injection. Therefore, the fibrin contained semi-solid osteoblast composition is effectively and rapidly cure the bone fracture via constant injection of into the affected area.
Patent ES-2362525-B8 (ES)
Title: Formulación de medicamentos en forma de agujas percutaneas penetrantes.
Inventor: GARCIA DE CASTRO ANDREWS ARCADIO
IPC: A61K9/00
Filed: 2009-10-08
Granted: 2013-01-03
Abstract: La invención se refiere a formulaciones de medicamentos para su administración en forma de agujas percutáneas penetrantes sólidas, “agujas inyectables”, fabricadas mediante procesos de polimerización por adición. El proceso de polimerización implica la transformación de una fase líquida que contiene monómeros en un cuerpo sólido monolítico, que contiene el medicamento, con la forma, dureza y rigidez requeridas para ser inyectadas en el tejido subcutáneo mediante sencillos dispositivos empujadores o inyectores. Estos procedimientos permiten la incorporación directa del medicamento a las agujas inyectables, o su incorporación en nano- o micro-partículas preformuladas para preservar la integridad y acción terapéutica del medicamento que contienen, así como de agentes modificadores de la velocidad de degradación, perfil de liberación del medicamento, dureza y rigidez, o inmunogenicidad.
Patent AU-2006282762-B8 (AU)
Title: Reconstruction render farm used in motion capture
Inventor: DEMIAN GORDON
IPC: G06T7/00
Filed: 2006-08-28
Granted: 2011-11-17
Abstract: Motion capturing markers coupled to at least one motion capture object, comprising: generating a plurality of Configurations, each Configuration including partitioning parameters; partitioning a motion capture beat into beat partitions using the plurality of Configurations; reconstructing the beat partitions, wherein each beat partition is reconstructed using each Configuration and corresponding motion capture camera calibration information to generate point data representing a marker; and merging the point data to form at least one master point file.
Patent BR-112012015016-B8 (BR)
Title: formulação farmacêutica, forma de dosagem farmacêutica entérica e uso de uma formulação
Inventor: GUILLAUME SABATE
IPC: A61K9/48
Filed: 2010-12-17
Abstract: formulação farmacêutica, forma de dosagem farmacêutica entérica e uso de uma formulação. a presente invenção refere-se á formulação farmacêutica destinada para administração oral que contém um oligossacarídeo dotado de uma a 18 unidades de monossacarídeo e que tem uma atividade terapêutica ou um sal de adições farmaceuticamente aceitável ou solvato do mesmo, em que a formulação contém: a) o oligossacarídeo (a) em uma quantidade de até 5% em peso do peso total da formulação, vantajosamente, até 1 % em peso do peso total da formulação, b) uma fase lipofílica (b) que consiste em triglicerídeo de ácidos graxos em uma quantidade de 50 a 80% em peso do peso total da formulação, vantajosamente, de 50 a 70 % em peso do peso total da formulação, c) pelo menos um tensoativo lipofílico (c) com hlb abaixo de 7 que consiste com em ésteres parciais de poliol e ácidos graxos em uma quantidade de 10 a 30% em peso do peso total da formulação, vantajosamente, de 15 a 30% em peso do peso total da formulação, d) pelo menos um tensoativo hidrofílico (d) com hlb acima de 7 em uma quantidade de até 20% em peso do peso total da formulação, vantajosamente, até 15% em peso do peso total da formulação, e) opcionalmente, pelo menos um solvente hidrofílico (e) em uma quantidade de até 15% em peso do peso total da formulação, vantajosamente, até 10% em peso do peso total da formulação, f) entre 0 e 30% em peso do peso total da formulação de um agente de estabilização químico e/ou físico (f), vantajosamente, entre 0 e 20 % em peso do peso total da formulação, em que, quando a formulação está em uma forma de uma microemulsão ou emulsão reversa e contém pelo menos um solvente hidrofílico (e), 0 agente de estabilização físico está presente e é dióxido de sílico.