baber/WOPTO huggingface dataset:
Patent PH-12015502425-A1 (PH)
Title: Novel compounds for selective histone deacetylase inhibitors, and pharmeceutical composition comprising the same
Inventor: CHANGSIK LEE
IPC: A61K31/5377
Filed: 2015-10-21
Abstract: The present invention relates to novel urea derivatives and, more particularly, to novel urea derivatives with histone deacetylase (HDAC) inhibitory activity, isomers thereof, pharmaceutically acceptable salts thereof, their use for the preparation of a medicaments comprising the same, a pharmaceutical composition comprising the same, a treatment method using the composition, and a method for preparing novel urea derivatives. The novel urea derivatives as selective histone deacetylase (HDAC) inhibitors are effective for the treatment of histone deacetylase-mediated diseases such as malignant tumors, inflammatory diseases, rheumatoid arthritis, neurodegeneration, etc.
Patent PH-12017500725-A1 (PH)
Title: Indole carboxamide compounds useful as kinase inhibitors
Inventor: AHMAD SALEEM
IPC: C07D471/04
Filed: 2017-04-20
Abstract: Disclosed are compounds of Formula (I): or a salt thereof, wherein: X is CR4 or N; R1, R2, R3, R4, and A are defined herein. Also disclosed are methods of using such compounds as inhibitors of Bruton's tyrosine kinase (Btk), and pharmaceutical compositions comprising such compounds. These compounds are useful in treating, preventing, or slowing the progression of diseases or disorders in a variety of therapeutic areas, such as autoimmune diseases and vascular disease.
Patent PH-12017501458-A1 (PH)
Title: Printhead employing data packets including address data
Inventor: BAKKER CHRIS
IPC: B41J29/38
Filed: 2017-08-14
Abstract: A printhead including an address line for communicating a set of addresses and a number of primitives, each primitive including a plurality of controllable activation devices coupled to the address line, each switch corresponding to at least one address of the set of addresses, each address corresponding to one of a number of primitive functions. A buffer receives a series of data packets, each data packet including address bits representative of one address of the set of addresses. Address logic receives the address bits from the buffer, wherein for each data packet the address logic encodes the address represented by the address bits onto the address line, and wherein the at least one switch corresponding to the address activates the primitive function corresponding to address.
Patent PH-12017501840-A1 (PH)
Title: Bidirectional reversible medical skin tension reducing closer
Inventor: YANG SHUAI
IPC: A61B17/03
Filed: 2017-10-06
Abstract: A bidirectional reversible medical skin tension reducing closer comprises left and right substrates (3, 4), left and right pawls (5, 7), and left and right racks (2, 1), the left and right substrates being horizontally and symmetrically disposed, the left and right pawls being fixedly disposed on adjacent ends of the left and right substrates (3, 4) respectively, one end of the left rack and one end of the right rack being fixedly connected to the left and right pawls (5, 7) in an upper-down side-by-side disposing manner respectively. Ratchets (9) of the left and right racks tilt towards the left and right substrates (3, 4) respectively, and the other ends of the left and right racks (2, 1) penetrate through the lower parts of the left and right pawls (5, 7) respectively and are fitted with ratchets (11) disposed at the lower parts of the left and right pawls (5, 7). Adhesive layers for fixing the left and right substrates on the surface of human skin are disposed on the bottom surfaces of the left and right substrates (3, 4). The skin tension reducing closer can apply force from two sides uniformly. Moreover, the closing degree of a tension reducing device can also be freely adjusted.
Patent PH-12018500576-A1 (PH)
Title: Mono- or di-substituted indole derivatives as dengue viral replication inhibitors
Inventor: KESTELEYN BART RUDOLF ROMANIE
IPC: C07D209/12
Filed: 2018-03-15
Abstract: The present invention concerns mono- or di-substituted indole compounds of formula (I), methods to prevent or treat dengue viral infections by using said compounds and also relates to said compounds for use as a medicine, more preferably for use as a medicine to treat or prevent dengue viral infections. The present invention furthermore relates to pharmaceutical compositions or combination preparations of the compounds, to the compositions or preparations for use as a medicine, more preferably for the prevention or treatment of dengue viral infections. The invention also relates to processes for preparation of the compounds.
Patent PH-12019000285-A1 (PH)
Title: Process for preparing l amino acids using improved strains of the enterobacteriaceae family
Inventor: RIEPING MECHTHILD
IPC: C12R1/19
Filed: 2019-08-08
Abstract: The invention relates to a recombinant, L-amino acid-secreting microorganism of the Enterobacteriaceae family, comprising an DNA fragment having promoter activity that is functionally linked to a polynucleotide coding for a membrane protein, characterized in that the DNA fragment having promoter activity comprises the SEQ ID NO: 8
Patent PH-12019501878-A1 (PH)
Title: Ventilation device for switchgear
Inventor: WAKABAYASHI TORU
IPC: H02B1/56
Filed: 2019-08-13
Abstract: A ventilation device for a switch gear according to an embodiment of the invention is provided with a pair of support members (11) and a louver (12). The pair of support members (11) are arranged at a distance from each other and are joined to a housing (2). The louver (12) is located between the pair of support members (11) and opens and closes an opening (8c) provided in the housing (2). Either the pair of support members (11) or the opposite ends (12a, 12b) of the louver (12) in the direction (D1) in which the support members (11) are arranged are provided with protrusions (12f, 12g) protruding in the arrangement direction (D1). The pair of support members (11) or the opposite ends (12a, 12b) to which the protrusions (12f, 12g) are not provided are provided with holes (11c) in which the protrusion (12f, 12g) are inserted, and also with cylindrical surfaces (11d) facing the holes (11c). The pair of support members (11) supports the louver (12) while the protrusions (12f, 12g) and the cylindrical surfaces (11d) are engaged with each other.
Patent PH-12019502805-A1 (PH)
Title: Multi-level hysteresis voltage controllers for voltage modulators and methods for control thereof
Inventor: SLEPCHENKOV MIKHAIL
IPC: H02M7/86
Filed: 2019-12-12
Abstract: Systems and methods that facilitate multilevel hysteresis voltage control methods for cascaded multilevel voltage modulators having a plurality of power cells connected in series and has any positive integer number of output voltage levels to control any unipolar voltage on the load of the voltage modulator, and transfer electrical power from an electrical grid via AC/DC converters or directly from energy storage elements of the power cells to that load. A method of operational rotation of the power cells of a multilevel voltage modulator, which ensures an equal power sharing among the power cells and voltage balancing of the energy storage elements of the power cells of the modulator.
Patent PH-12019550134-A1 (PH)
Title: Multi-signal analysis for compromised scope identification
Inventor: LUO PENGCHENG
IPC: H04L29/06
Filed: 2019-07-22
Abstract: Detecting compromised devices and user accounts within an online service via multi-signal analysis allows for fewer false positives and thus a more accurate allocation of computing resources and human analyst resources. Individual scopes of analysis, related to devices, accounts, or processes are specified and multiple behaviors over a period of time are analyzed to detect persistent (and slow acting) threats as well as brute force (and fast acting) threats. Analysts are alerted to individually affected scopes suspected of being compromised and may address them accordingly.
Patent PH-12021550477-A1 (PH)
Title: Sustained-release injectable antibiotical formulation
Inventor: FRIEDMAN MICHAEL
IPC: A61P31/04
Filed: 2021-03-05
Abstract: Provided herein are compositions of injectable antibiotics for veterinary use. The compositions are characterized by forming a gel at animal physiological temperature, said gel being characterized by a stable and repeatable release profile of the antibiotic. The compositions comprise high loading of drug in poloxamer solutions with addition of a co-solvent, and preferably with an addition of a cellulose derivative at least partially soluble in organic solvents. Methods of treatment of veterinary infections are also provided.
Patent DE-102004001933-A1 (DE)
Inventor: BREHM STEFAN
IPC: F16F9/54
Filed: 2004-01-14
Abstract: A piston rod (2) is connectable to one of the masses to which the shock absorber (1) is installed. A fixing component has a stem and a fork which are made of a single piece. The stem is fixed to the base which is fixed to the container tube. The fork is connectable to the other mass.
Patent DE-102004002795-A1 (DE)
Title: Komponente, insbesondere für ein Kraftfahrzeug, mit einem Federmittel und Fahrzeugsitz
Inventor: KIENKE INGO
IPC: B60N2/90
Filed: 2004-01-19
Abstract: Es wird eine Komponente, insbesondere für ein Kraftfahrzeug, mit einer ersten Teilkomponente und einer zweiten Teilkomponente vorgeschlagen, wobei die Teilkomponenten relativ zueinander um eine Drehachse drehbar angeordnet sind, wobei ein Federmittel derart vorgesehen ist, dass auf einem ersten Winkelstellungsbereich der Teilkomponenten zueinander wenigstens ein erstes Drehmoment zwischen den Teilkomponenten wirkt, wobei auf einem zweiten Winkelstellungsbereich der Teilkomponenten zueinander, im Wesentlichen konstant, zwischen den Teilkomponenten entweder ein zweites Drehmoment wirkt oder kein Drehmoment wirkt.
Patent DE-102004004661-A1 (DE)
Title: Searching method for locating intellectual property or specialist literature relating to a particular search area, whereby a search request comprised of search terms and information is input via a suitable interface
Inventor: BEYER WOLFGANG
IPC: G06F17/30
Filed: 2004-01-29
Abstract: Method for searching for intellectual property or specialist literature relating to a particular search area, whereby a search request is input in the form of suitable terms and information and then matching data searched for using a special search profile via generated interface connections using a computer unit and or a mobile phone connection that permits the downloading of information from the internet or from a data support. The invention also relates to a corresponding computer unit for implementation of the inventive method.
Patent DE-102004004908-A1 (DE)
Title: Controlling idling speed of vehicle engine, measures current supplied to on-board consumers and current supplied for battery charging, to calculate the necessary idling speed
Inventor: PFALLER STEFAN
IPC: F02D41/08
Filed: 2004-01-30
Abstract: The instantaneous battery charging current is measured. Together with the measured current supplied to the vehicle wiring and consumer systems, this value is used to calculate the required idling speed. The method relates to an earlier disclosure cited as 102 57 024.8. An independent claim is included for the corresponding vehicle.
Patent DE-102004006893-A1 (DE)
Title: Verfahren zur Herstellung von 1[N2-[3,5-Dibrom-N-[[4-(3,4-dihydro-2(1H)-oxochinazolin-3-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)-piperazin
Inventor: LINZ GUENTER
IPC: C07D401/14
Filed: 2004-02-12
Abstract: Gegenstand der vorliegenden Anmeldung ist ein Verfahren zur Herstellung des CGRP-Antagonisten 1-[N·2·-[3,5-Dibrom-N-[[4-(3,4-dihydro-2(1H)-oxochinazolin-3-yl)-1- DOLLAR A piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)-piperazin der Formel DOLLAR F1 mit Hilfe dessen diese Verbindung in großen Mengen, hohen Ausbeuten und hoher Reinheit hergestellt werden kann.
Patent DE-102004007298-A1 (DE)
Title: Verfahren zur Überwachung von Laborproben
Inventor: BECKER ANNETTE
IPC: G01N35/00
Filed: 2004-02-14
Abstract: Es wird ein Verfahren zur Überwachung von zu untersuchenden Proben beansprucht, die nach der Probenentnahme an einem vom Ort der Probenentnahme verschiedenen Ort untersucht werden, welches die folgenden Schritte umfasst: DOLLAR A a) Erfassen der Probe in einem Datensystem, DOLLAR A b) Aufnahme der vorzunehmenden Analyse in das Datensystem, DOLLAR A c) Melden der an der Probe vorzunehmenden Untersuchung(en) als Auftrag an ein Labor, DOLLAR A d) Melden der Probe als Transportauftrag an einen Transportdient, DOLLAR A e) Transport der Probe zum Labor und Durchführen der Untersuchung, DOLLAR A f) Melden des Untersuchungsergebnisses an den Auftraggeber.
Patent DE-102004008169-A1 (DE)
Title: Control process for a motor vehicle interior light that can operate in permanent light mode changes type of operating activity on starting the vehicle
Inventor: AIGNER KONRAD
IPC: B60Q3/02
Filed: 2004-02-19
Abstract: A control process for a motor vehicle (1) interior light (3,7) comprises switching off a first operating activity on starting the vehicle and switching on a second such activity of an opposite sense with the light modes being chosen by the driver.
Patent DE-102004008462-A1 (DE)
Title: Reflective flag for road vehicles in case of accident has square of reflective material with separate strengthening tubes and three part aluminum rod
Inventor: MISINSKI ELKE
IPC: B60Q7/00
Filed: 2004-02-20
Abstract: A reflective flag for road vehicles comprises a square of water-repellant doubled reflective material (14) visible in the dark that can be rolled up and has four equal spacing tubes (9-12) having bent wiring. A three-part aluminum rod (3,5,7) has a massive point (8) for inserting into the ground.
Patent DE-102004010636-A1 (DE)
Title: Firing range projectile catchment device comprises at least vertical side parts, rear wall and connecting plates made of horizontal lamellas backwardly inclined
Inventor: SCHUETZ ANDREAS
IPC: F41J13/00
Filed: 2004-03-02
Abstract: The firing range projectile catchment device comprises at least vertical side parts, a rear wall and connecting plates made of horizontal lamellas backwardly inclined. The front plate edge of the connecting plates has an upper part edge (12), which runs horizontally or tilts upwards by 30 degrees at most in relation to the horizontal and comprises a lower part edge (14), forming approximately a right angle to the plate under side. The lower part edge (14) has an edge height which amounts at most to half the diameter of the projectiles used. The connecting plates have a thickness of 10 to 20 mm and the lower part edge has a width of 3 to 5 mm. The upper part edge (12) is at an angle of 105 to 165 degrees to the lower part edge (14) or to the upper plate surface (13).
Patent DE-102004012399-A1 (DE)
Title: Body for a vehicle comprises a pillar in a monocoque construction with an inner and an outer skin interconnected by two flanges, and a reinforcing panel arranged between the inner and outer skins
Inventor: HOGGER THOMAS
IPC: B62D25/04
Filed: 2004-03-13
Abstract: Vehicle body comprises a pillar (1) in a monocoque construction with an inner and an outer skin (2, 3) interconnected by two flanges (4, 5), and a reinforcing panel (7) arranged between the inner and outer skins. When the pillar is viewed in the transverse direction, the reinforcing panel is connected at least twice to the inner skin and extends between the connecting regions on the inner skin toward the outer skin so that a cavity is formed between the inner skin and the reinforcing panel. Preferred Features: The flanges serve as connecting regions between the inner skin and the reinforcing panel.
Patent DE-102004012470-A1 (DE)
Title: Operating handle for insitu-foam dispenser is constructed with size suited at least partially to encompassing hand, and handle is constructed together with operating lever and delivery tube connection
IPC: B65D83/14
Filed: 2004-03-15
Abstract: The operating handle (1) for an insitu-foam dispenser (2) has an operating lever (4) for acting upon a delivery valve, and a delivery tube connection (5). The operating handle is constructed with a size suited at least partially to an encompassing hand (H). The operating handle together with an associated section of the dispenser serves for the hand-holding of the dispenser, and the handle is constructed with the operating lever and delivery tube connection. An independent claim is included for a combination comprising an insitu-foam dispenser and operating handle.
Patent DE-102004013966-A1 (DE)
Inventor: MAIER RUDOLF
IPC: F16F15/02
Filed: 2004-03-19
Abstract: The invention relates to an active element (10) for reducing the vibrations of components and in particular aircraft components. Said element comprises a support structure (11, 12) for fixing a first component to a second component, in addition to an actuator unit (13), which is mechanically coupled to the support structure (11, 12), in order to subject the support structure (11, 12) to variable forces. A regulator controls the actuator unit (13), based on a sensor signal, in order to minimise the transmission of unwanted vibrations along a transmission path through the support structure (11, 12). Said support structure (11, 12) can be regulated by the actuator unit (13) in three degrees of freedom to counteract the transmission of the unwanted vibrations. The support structure is configured by a first support plate (11), a parallel second support plate (12) and several actuators that form the actuator unit (13) and are located between the two plates. The inventive active element and method permit components to be interconnected in a soundproofed manner.
Patent DE-102004015023-A1 (DE)
Title: Verbesserter Augendiagramm-Analysator tastet niedrige DU/DT Spannungen korrekt ab
Inventor: ESKELDSON DAVID D
IPC: H04B10/08
Filed: 2004-03-26
Abstract: Ein abtastender Übergang-durch-eine-ausgewählte-Spannung-Detektor stellt zwei Latches auf unterschiedliche Werte ein, wenn ein Eingangssignalkomparator, bezogen auf die ausgewählte Spannung, während eines Abtastintervalls einen Übergang durchläuft: am Anfang des Abtastintervalls empfängt ein Latch einen Vergleichswert, wohingegen am Ende des Abtastintervalls das andere Latch einen entgegengesetzten Vergleichswert empfängt. Eine Differenz (XOR) der zwischengespeicherten Werte für die Übergangserfassungslatches zeigt einen Übergang durch die ausgewählte Spannung während des Abtastintervalls an. Eine Lösung für das Problem der Unempfindlichkeit eines derartigen Übergang-durch-eine-ausgewählte-Spannung-Erfassungsmechanismus gegenüber Dauerzustandsspannungen kann durch Einschließen eines zusätzlichen Latches gelöst werden, das durch einen zweiten Eingangssignalkomparator eingestellt wird, dessen Bezugsspannung leicht von der versetzt ist, die verwendet wird, um Übergänge durch die ausgewählte Spannung zu erfassen, und das ebenfalls am Anfang des Abtastintervalls getaktet wird. Es liegen somit zwei Latches vor, die am Anfang des Abtastintervalls getaktet werden. Wenn dieselben sich unterscheiden, wie durch eine andere XOR-Verknüpfung angezeigt ist, dann war das Eingangssignal zwischen der Bezugsspannung und ihrem leicht versetzten Gegenstück, selbst wenn sich das Eingangssignal am Beginn des Abtastintervalls nicht in einem Übergangszustand oder in einem Dauerzustand befand. ...
Patent DE-102004018843-A1 (DE)
Title: Elektronisches Steuersystem für die Vorfüllung eines Brennstoffsystems
Inventor: GRECO LUCA
IPC: F02M37/08
Filed: 2004-04-19
Abstract: Insbesondere bei einem relativ großen Motor, der für eine wesentliche Zeitperiode bei kalter Temperatur inaktiv gewesen ist, kann der Druck innerhalb eines Brennstoffsystems absinken. Vor der Einteilung eines Motorstarts können Brennstoffpumpen, die betriebsmäßig mit dem Motor gekoppelt sind, nicht den Brennstoff innerhalb des Brennstoffsystems unter Druck setzen und/oder zirkulieren. Somit kann die Zeit vernünftigerweise verzögert werden, die erforderlich ist, um die Hochdruck-Leitungen mit einem ausreichenden Brennstoffdruck zu beliefern, um den Motor zu starten und laufen zu lassen. Um die Verzögerung beim Start des Motors zu verringern, weist die vorliegende Erfindung ein elektronisches Steuermodul auf, welches einen Vorfüllungsalgorithmus aufweist. Der Vorfüllungsalgorithmus ist dahingehend wirksam, dass er eine elektrisch angetriebene Pumpe aktiviert, wenn ein Brennstoffsystem in einem nicht vorgefüllten Zustand ist. Das elektronische Steuermodul ist in Verbindung mit mindestens einem Sensor, der betreibbar ist, um den Zustand des Brennstoffsystems abzufühlen.
Patent DE-102004020632-A1 (DE)
Title: Hochfrequenz(RF)-Modulator mit schmalem Bandpassfilter
Inventor: RYU JONG GI
IPC: H04N5/38
Filed: 2004-04-27
Abstract: Es wird ein RF-Modulator mit einem schmalen Bandpassfilter (30, 30a, 30b) beschrieben. Der RF-Modulator zur Modulation von Video- und Audiosignalen in RF-Signale, entsprechend einem Frequenzband eines vorherbestimmten Kanals, umfasst eine Oszillatoreinheit (14) zur Erzeugung eines vorherbestimmten RF-Signals, das für das Frequenzband des vorherbestimmten Kanals geeignet ist; einen Mischer (15) zur Modulierung der Video- und Audiosignale unter Verwendung des RF-Signals, das von der Oszillatoreinheit (14) erzeugt wird; und einen schmalen Bandpassfilter (30, 30a, 30b) zum Empfang eines RF-modulierten Signals vom Mischer (15) und zum Durchlass nur eines Frequenzsignals des Frequenzbands des vorherbestimmten Kanals von dem RF-modulierten Signal. Deshalb kann der RF-Modulator unnötige Komponenten wie untere Seitenband- und Oberwellenfrequenz-Signale, die nach der RF-Modulierung von Video- und Audiosignalen erzeugt werden, entfernen oder sperren, sodass er die Entstehung von Interferenz zwischen Kanälen verhindern kann, wodurch besonders hervorragende Video- und Audiosignale erzeugt werden.
Patent DE-102004021285-A1 (DE)
Title: Process for the parallel generation of a secure digital and handwritten form of a will
Inventor: LEHR HARTMUTH F
IPC: G07C11/00
Filed: 2004-04-29
Abstract: The creation of a will involves both the hand written form and the generation of a digital version. The digital version is made by scanning and reproducing in precise form and colour. The document is authenticated by an identification code. The scanned information may be transmitted using a cable or wireless link.
Patent DE-102004023188-A1 (DE)
Title: Quality control process for the dairy industry, useful e.g. for selecting cultures with optimal properties, comprises detecting gene sequences indicative of quality by nucleic acid hybridization
Inventor: BLOHM DIETMAR
IPC: C12Q1/70
Filed: 2004-05-11
Abstract: Quality control method for the dairy industry in which a sample is tested simultaneously for many genes (A) relevant for quality. A prepared sample is treated with many nucleotide probes (I), each specific for a particular (A), and the resulting hybridization products are detected. Independent claims are also included for the following: (1) method for investigating cultures for simultaneous presence of genes (B1) that mediate resistance to phages; (2) method for investigating cultures for presence of desirable genes (B2) that affect milk product properties (flavor; odor; consistency of the end product); (3) microarrays for performing the new methods; and (4) methods for targeted selection of a culture, or set of cultures, for milk processing.
Patent DE-102004024144-A1 (DE)
Title: Warming up indicator, for frozen food, has two pieces of cloth impregnated with potassium hexacyanoferrate solution and with ammonium ferrous sulfate solution, respectively, which react above their melting points to form blue color
IPC: G01K11/12
Filed: 2004-05-14
Abstract: Warming up indicator (4) has two pieces of cloth (1, 2) that are impregnated with potassium hexacyanoferrite solution and with ammonium ferrous sulfate solution, respectively. The pieces are frozen separately at respective salt concentration. The pieces are placed one above the other and are fixed together by welding with a transparent foil (3). The solutions react to form a blue color above their melting points.