baber/WOPTO huggingface dataset:
Patent EC-SP067079-A (EC)
Title: Derivados de ácido carboxílico de bencimidazolona
Inventor: IGUCHI SATORU
IPC: A61P25/06
Filed: 2006-12-13
Abstract: Esta invención se refiere a compuestos de fórmula (I): (consta gráfico) en la que R1,R2, R3, A y m son cada uno de ellos como se han descrito en esta memoria descriptiva a una sal o solvato farmacéuticamente aceptable de los mismos, y las composiciones que contienen tales compuestos y el uso de tales compuestos en el tratamiento de una afección mediada por la actividad del receptor 5-HT4 tal como, pero sin limitación a, enfermedad de reflujo gastroesofágico, enfermedad gastrointestinal, trastorno de motilidad gástrica, dispepsia no ulcerosa, dispepsia funcional, síndrome de intestino irritable (IBS), estreñimiento, dispepsia, esofagitis, enfermedad gastroesofágica, nauseas, enfermedad del sistema nervioso central, enfermedad de Alzheimer, trastorno cognitivo, tmesis, migraña, enfermedad neurológico, dolor, trastornos cardiovasculares, tales como insuficiencia cardiaca y arritmia cardiaca, diabetes y síndrome de apnea.
Patent EC-SP992860-A (EC)
Title: Apoptosis auto- regulada de celulas inflamatorias mediante terapia genica
Inventor: MARLIN STEVEN D
IPC: C12N15/00
Filed: 1999-02-18
Abstract: La invención se refiere a ácidos nucléicos quiméricos y a la inducción terapéutica de la apoptosis en células inflamatorias activadas, o células en un sitio de la inflamación, al inducir en esas células el ácido nucléico quimérico. El ácido nucléico quimérico tiene al menos un reforzador del promotor de TNF alfa unido a una copia funcional de TNF alfa y está unido, además, al menos una copia de un gen inductor de la apoptosis que está unido adicionalmente a una 3ÚTR. El gen inductor de la apoptosis es Granzyme B. La invención se refiere también a métodos para preparar y utilizar ácidos nucléicos quiméricos de apoptosis auto-regulada y a composiciones farmacéuticas que los contienen para tratar enfermedades inflamatorias.
Patent FI-20022009-A (FI)
Inventor: NISSILAE SEPPO
IPC: A61B5/0245
Filed: 2002-11-08
Abstract: The invention relates to a method and an electronic device for implementing the method for measuring mental load. The electronic device generates (600) at least two different cognitively loading tasks for the person participating in the measurement, the first task determining a reference level and at least one other task determining the loading capacity level. The electronic device determines (602) the pulse parameters of the person participating in the measurement during the cognitively loading tasks. The electronic device also compares (604) the pulse parameters during the different tasks with each other. Finally, the electronic device generates (606) a value descriptive of the mental load of the person participating in the measurement on the basis of the comparison of the pulse parameters. <IMAGE>
Patent FI-20065195-A (FI)
Inventor: VITIKKA ILPO
IPC: H04L69/324
Filed: 2006-03-24
Abstract: A communication system that comprises a mobile station (17), an access point (10, 11), and a wireless interface for implementing a local connection between the mobile station and the access point. The mobile station (17) is configured with a virtual device that a virtual device that provides a serial port emulation for a terminal function and interfaces the serial port emulation with an Ethernet-based connection. simple user experience of serial connection type applications may be provided within a wider region of coverage. A user may use the familiar applications in a consistent way without worrying about the creation of IP connection or basically even needing to know which kind of radio units his or her user equipment comprises.
Patent FR-1605038-A (FR)
Title: 1,2,3,4-tetrahydroquinolines useful as - plastics stabilisers ageing preventers and
IPC: C07D215/20
Filed: 1968-12-11
Granted: 1972-08-28
Abstract: Amine (I) is reacted with formaldehyde and olefin (II) in presence of a strong acid at 0-70 degrees C, opt. in presence of a solvent, and the salt obtained is converted to the free base (III) in known way. R1,R2,R3,R4 = H, 1-4C alkyl or alkoxy, halogen (R1 pref. H), R9 = H or 1-4C alkyl (pref. H). Any of the pairs R1 & R2, R2 & R3, R3 & R4, R1 & R9 may together form part of a 6 membered ring. R6,R8 = H or 1-10C alkyl, R7 = Ph, CH2=CH or Me, Et provided R6 = H.
Patent GB-1050182-A (GB)
IPC: E04H6/18
Abstract: 1,050,182. Mechanical garages. SPEEDPARK Inc. April 13, 1965, No. 15747/65. Heading B8E. A vehicle parking structure 10, Fig. 1, comprises a vehicle passageway 12 at a first level 11, a passageway 26 extending vertically from a second level contiguous to the level 11, a lift 39 having limited movement between the two levels, a lift conveyer 27 having vertically movable members 33, 34, and parking stalls 20 disposed in tier formation on at least one side of the passageway 26, the members 33, 34 being mounted for lateral movement between the conveyer 27 and the lift 39 and the stalls 20 for transferring a vehicle between these members. The level 11 is the ground level and there is provided a pedestrian passage 17, and the passageway 12 may be extended in width to accommodate through traffic. As shown the stalls 20 are disposed on both sides of the passageway 26 in parallel rows 24, 25. The conveyer 27 comprises a frame 28, 31, 32 and has wheels 29 which run on rails 30, and the members 33, 34 are comblike, each having parallel fingers which extend toward the fingers of the other in interdigitated relationship from a backbone independently movably mounted on a side of the frame 28, 31, 32. The stalls 20 and the lift 39 have support fingers 37 and 41 for interengagement with the fingers of the members 33, 34. A safety barrier 44 is provided in the form of an upright rectangular frame vertically movable between a depressed position to stop a vehicle and a raised position to allow a vehicle to pass to the lift 39. In a second embodiment, Fig. 2 (not shown), the parking stalls are above the ground level. In a third embodiment, Figs. 3, 4 (not shown), a plurality of lifts 39A similar to the lift 39 are provided and the parking stalls are serviced by two lift conveyers 27. In a fourth embodiment, Figs. 5, 6, 7 (not shown), access to underground parking stalls is by a pair of lifts 39 situated at an indented portion 62 of a curb 61 bounding a city thoroughfare 60.
Patent GB-1054180-A (GB)
IPC: B23D45/16
Abstract: 1,054,180. Grinding. FRANCIS W. BIRKETT & SONS Ltd. March 16, 1965 [July 18, 1964], No. 29381/64. Heading B3D. [Also in Divisions B5 and F2] A portable grinding machine comprises a frame 1 having handles 2, 3 and carrying an internal combustion engine 4 which drives through belt, chain or, as shown, spur gearing 9, 10, 11 a grinding wheel 13. A throttle control 5 is provided adjacent one of the handles. A four section guard 15, 19, 25, 26 completely shrouds the wheel 13 when not in use. The lower sections 19, 26 pivot upward when the machine is lowered on to a workpiece. The lower section 19 may be locked in the position shown by a rod 22 and the sections 25, 26 removed to provide a side grinding machine.
Patent GB-1176884-A (GB)
IPC: A01N43/70
Filed: 1967-06-19
Abstract: 1,176,884. Herbicides containing triazines. GULF RESEARCH & DEVELOPMENT CO. 19 June, 1967 [27 June, 1966], No. 28115/67. Heading ASE. [Also in Division C2] Pre- and post-emergent herbicides comprise compounds of the general formula wherein X is H or CH 3  and Y is cyclopropyl, 1-methylcyclopropyl, isopropyl or ethyl. Examples illustrate the use of the compounds in the form of (a) acetone solutions, and (b) aqueous dispersions which additionally contain xylene, kerosene and a polyoxyethylated vegetable oil emulsifier.
Patent GB-1225994-A (GB)
IPC: D06F39/12
Filed: 1968-06-07
Abstract: 1,225,994. Washing machines. INDUSTRIE A. ZANUSSI S.p.A. 7 June, 1968 [14 June, 1967], No. 27302/68. Heading D1A. In a washing machine or the like, with a wheeled base, at least one stabilizing wheel 18 has a curvilinear triangular outline with rounded corners and a pedal actuated means 19 is provided to displace the machine between a position in which the stabilizing wheel 18 assists in supporting the machine and a position in which it is idle.
Patent GB-1226406-A (GB)
IPC: G08C19/28
Filed: 1968-05-08
Abstract: 1,226,406. Vehicle identification system. "FOK - GYEM" FINOMMECHANIKAI ES ELEKTRONIKUS MUSZERGYARTO KTSZ. 8 May, 1968 [10 May, 1967; 29 May, 1967], No. 21842/68. Heading B7H. In a vehicle identification system in which a column and row array of reed switch elements 11-19 at the trackside detects the position of magnets 1-3 arranged in selected positions, coded in dependence on the vehicle number, in a corresponding array of positions on the vehicle, each reed switch, e.g. 12, is associated in the detector array with a magnet 12<SP>1</SP> disposed with its direction of magnetization opposite to that of the next adjacent column and row magnets 11, 13<SP>1</SP>, 2<SP>1</SP> and each magnet, e.g. 2, in the coded array on the vehicle has the same direction of magnetization as its corresponding magnet 2<SP>1</SP> in the detector array and thus opposite to a next adjacent magnet in the coded array if present. The magnets may be permanent or electromagnets and the reed switches are provided with polepieces of larger cross-sectional area than the switch contacts. Means (not shown) are provided for sensing the signals produced by operation of the reed switches when the positions of the arrays correspond.
Patent GB-1226412-A (GB)
IPC: H01G4/20
Filed: 1968-06-11
Abstract: 1,226,412. Capacitors. GENERAL ELECTRIC CO. 11 June, 1968 [29 June, 1967], No. 27687/68. Heading H1M. Capacitor electrodes are separated by a dielectric spacer comprising a blend of a polyphenylene oxide and polystyrene. The blend preferably has about 50% by weight of each constituent. The spacer may be in the form of a biaxially oriented film. It may be used together with a strip of kraft paper, especially for impregnating with dielectric liquids, or hardenable materials, or with sheet mica. It may include fillers, e.g. alumina or silica flour. Alternatively sheets of glass cloth, asbestos or textile cloth may be impregnated or coated with the blend. The film may be wound with aluminium, tantalum or copper electrodes or metallized with tin, silver, lead, or zinc or coated with carbon for making a wound capacitor.
Patent GB-1227620-A (GB)
IPC: C07D207/404
Filed: 1968-11-28
Abstract: 1,227,620. N - (3,5 - " Dichlorophenyl) - maleimide and -succinimide. SUMITOMO CHEMICAL CO. Ltd. 28 Nov., 1968 [1 Dec., 1967], 56557/68. Heading C2C. [Also in Division A5] The invention comprises compounds of the general formula wherein A is a -CH=CH- or -CH 2 -CH 2 - group. The compounds are prepared by reacting 3,5-dichloroaniline with maleic or succinic anhydride.
Patent GB-1228194-A (GB)
IPC: B05D7/24
Filed: 1968-07-10
Abstract: 1,228,194. Polysiloxane coating. WACKERCHEMIE G.m.b.H. 10 July, 1968 [14 Feb., 1968], No. 32824/68. Heading B2E. [Also in Division C3] Coatings which repel tacky substances are produced by applying to a substrate a coating of a solution of a composition comprising 80 to 95% by weight of a diorgano polysiloxane having end groups capable of reacting with an amino-substituted silicon compound and 5 to 20% by weight of a cross-linking aminosubstituted silicon compound containing at least 3 hydrolysable groups in the molecule in a volatile organic solvent that is free from water and is inert to SiN bonds, at least at ambient temperature and curing the coating by heating it to 80‹ to 200‹C in the presence of steam. The substrate may be paper, e.g. imitation parchment, parchment, kraft or silk paper, metals such as aluminium foils and organic plastics, e.g. polyamides or regenerated cellulose, or cardboard. The diorgano polysiloxanes which may be used are those of formula: (in which R is a monovalent optionally substituted hydrocarbon radical, x has an average value of 0.99 to 1.01, y has an average value of 1.99 to 2.01, the sum of x+y is 3, and n is an integer having a value of 10 to 10,000). The hydroxyl groups may be at least partially replaced by other reactive end groups, e.g. radicals of formula R"HN-, where R" is optionally substituted hydrocarbon, alkoxy or alkoxyalkoxy radical. The diorgano polysiloxanes may be homopolymers, mixtures of various homopolymers, copolymers or mixtures of various copolymers. Preferred crosslinking amino-substituted silicone are aminosilanes of formula: (in which R is as hereinbefore defined, R<SP>1</SP> is a monovalent hydrocarbon radical, p is 0 or 1, m is 0, 1 or 2. Further examples of crosslinking amino-substituted silicone compounds are: silazanes of formula: (H m R<SP>1</SP> 2-m N) 2  SiR" (NHSiR"NH m R1 2-m ) n  NHSiR" (NH m R1 2-m ) 2  (in which R" is as R or a 1-4C alkoxy or 3-6 C alkoxyalkoxy; n' is 0 or an integer; compounds of formula: R'' r SiZ 4-r  (in which Z is aminoalkoxy; r is 0, 1, 2 or 3); and com- O pounds of formula: R" r Si(NR"'CR"') 4-r  (in which R"' is as R' or is H). The compositions can be applied by dipping, brushing, pouring, spraying or rolling. The process is particularly suitable for the production of release backings and blanket papers for self-adhesive tapes and self-adhesive films, the coating of the back of self-adhesive tapes and films, of release papers such as are used in the preparation of laminates from epoxy resins and glass fibre fabrics, for the preparation of packaging material for tacky foodstuffs such as meat, and other tacky substances such as asphalt, resins, tar and photographic films.
Patent GB-1229572-A (GB)
IPC: B60P7/00
Filed: 1967-01-20
Abstract: 1,229,572. Releasable fastenings. C. R. TYRER. 22 April, 1968 [20 Jan., 1967], No. 3106/ 67. Heading E2A. An attachment means 10 for tying down a cover sheet 14 is made of substantially rigid material and has a flat plate-like first portion 11 of trapezoidal form capable of being secured to the cover sheet and a second portion 15 of substantially triangular form, integral with the first portion and of increased thickness relative to the first portion, there being in the second portion a hole 16 for attachment thereto of a fastening rope or a hook. The device described is made of a moulded plastics material such as low density polythene and in a modification two second portions disposed side by side are provided.
Patent GB-1232089-A (GB)
IPC: H04R7/02
Filed: 1968-07-02
Abstract: 1,232,089. Moulding plastic substances. PHILIPS ELECTRONIC & ASSOCIATED INDUSTRIES Ltd. 2 July, 1968 [5 July, 1967], No. 31559/68. Heading B5A. [Also in Division H4] A multi-compartment injection mould for forming a loud-speaker diaphragm has mould walls 14, 15, 16 (Fig. 5) defining a space 20 for moulding the diaphragm rim and rim support. Walls 16, 17 define a space 21 for moulding the cone and coil support. Spaces 20, 21 are separable by a slide 19. In use, reaction mixture is fed through nozzles 27 to a chamber 23. The reaction mixture forms a foam so as to produce a foamed diaphragm. The foam spreads to fill a mould space 21, slide 19 being closed. After curing, the slide 19 is lifted. A different reaction mixture is fed through nozzles 26 to chamber 22. Foam, produced by this reaction mixture, penetrates to the space 20 and reaches the boundary 28 where it bonds to the foam in the space 21. An alternative multi-compartment mould (Fig. 6) has a space 35 which can be closed off at a boundary 34 by a slidable wall 30. A slide 43 is also provided. In use the slide 43 and boundary 34 are first closed. Foamed material is fed through a duct 46 into a mould space 40. After curing, the slide 43 and boundary 34 are opened. Foamed material is then fed through the duct 47 to form the rim and rim support in space 35 and the centring ring in space 45. Another mould (Fig. 7, not shown) has two mould walls (50, 51) and the mould spaces merge into one another. Each mould space has its own duct (54, 55). A control member (56) controls the rate of expansion of foamed material in the two mould spaces, e.g. by controlling the quantities fed. The two foams meet at the desired boundary where the two bond together and may partly mix.
Patent GB-1232787-A (GB)
IPC: C07D263/58
Filed: 1967-08-08
Abstract: 1,232,787. Substituted anilides or substituted aminobenz(oxa and thia)-zoles. JOHN WYETH & BRO. Ltd. 24 July, 1968 [8 Aug., 1967], No. 36337/67. Heading C2C. Substituted anilides or substituted aminobenz(oxa and thia)-zoles of the Formulµ I(a), I(b) and I(c) and acid addition and quaternary ammonium salts thereof, in which X is O or S; R is H, halogen, NO 2 , alkyl, alkoxy or haloalkyl; R<SP>1</SP> is CH 3  or, when X is S, R<SP>1</SP> may be a radical of the Formula II R<SP>2</SP> is (CH 2 ) n  or N (R<SP>4</SP>)R<SP>5</SP> or CH 2 -C#C-CH 2 N- (R<SP>4</SP>)R<SP>5</SP> where n is 1 to 4, and R<SP>4</SP> and R<SP>5</SP> each represent H or alkyl or together with the nitrogen atom to which they are attached complete a heterocyclic ring which may contain a further hetero atom and which may be substituted; and R<SP>3</SP> is a substituted or unsubstituted alkyl, aryl, aralkyl or aralkenyl radical, the compound of the above Formulµ Ia, Ib and Ic being novel when in compounds of Formula Ia X is O, R<SP>1</SP> is CH 3 , R<SP>3</SP> is an unsubstituted alkyl, R<SP>2</SP> is (CH 2 ) n  N (R<SP>4</SP>)R<SP>5</SP> where n is 2 or 3, and R<SP>4</SP> and R<SP>5</SP> are both alkyl or together with the nitrogen atom to which they are attached complete a heterocyclic ring, R is halogen, NO 2 , alkyl, alkoxy or haloalkyl; are prepared by reacting the corresponding compounds of the above Formulµ I(a) and I(b) in which R<SP>2</SP> is H with compounds of the formulµ or in which Z is halogen or alkyl- or aryl-sulphonyl. Alternatively compounds of the above Formulµ I(a), I(b) and I(c) in which R<SP>2</SP> is CH 2 .C#CCH 2 N(R<SP>4</SP>)R<SP>5</SP> may be obtained by reacting compounds of the above Formulµ Ia and Ib in which R<SP>2</SP> is -CH 2 C#CH with formaldehyde or paraformaldehyde and amines of the formula HN(R<SP>4</SP>)R<SP>5</SP>. p-Methylthioacetanilide is made by reacting p-methylthioaniline with acetic anhydride. 2,2<SP>1 </SP>- Diacetamidodiphenyldisulphide is obtained by acetylating 2,2<SP>1</SP>-diaminodiphenyldisulphide resulting from the treatment of a suspension of o-aminobenzenethiol in ammonium hydroxide with air. Pharmaceutical compositions having activity on the central nervous system and/or cardiovascular system and suitable for oral or parenteral administration, contain the above novel compounds and pharmaceutically acceptable carriers.
Patent GB-1239080-A (GB)
IPC: G12B11/02
Filed: 1968-07-17
Abstract: 1,239,080. Indicating-apparatus. AMETEK, Inc. July 17, 1968 [July 21, 1967], No.34092/68. Heading G1J. [Also in Division F4] An indicating instrument has a unit for illuminating light transmitting indicia 22 provided in the dial 20 thereof which unit includes a lamp chamber 16 and at least a pair of linear polarized discs 24, 26 between a lamp or lamps 18 in the chamber 16 and the dial 20 and means for rotating at least one of the discs to vary the angle between the polarization axes 72, 74 of the discs to vary the intensity of light transmitted to the indicia. A tab 30 projects from the disc 26 through an arcuate slot 32 in wall 14 whereby the disc 26 can be rotated through at least ninety degrees. Ribs 34 inside the wall 14 provide seats 36 supporting a diffusing ring 28. An indicating pointer 60 and its shank 62 are constructed from light conducting material coated with a layer of white paint covered by a layer of black paint where indicated by shading so that only the clear part 64 becomes illuminated by the lamps 18. To obtain a desired intensity of illumination of the indicia 22 or a desired ratio of brightness between the pointer and indicia, the unit is set up with a photo-meter in a darkroom, the lamps are energized by a specified voltage and the disc 26 is rotated by means of the tab 30 until the angle between the axes of the discs 24, 26 produces the desired result. A small dab of cement or adhesive e.g. silicone rubber is then applied between the tab 30 and wall 14. Lamp leads 52 pass through pairs of holes 50 in recesses 44 in a rear wall 12 to be soldered to conductor rings 46 in concentric grooves 40, 42, each ring having a hook 48 serving as a terminal.
Patent GB-1251462-A (GB)
IPC: G03C5/00
Filed: 1970-04-15
Abstract: 1,251,462. Developing photographic lightsensitive silver halide material. FUJI PHOTO FILM CO. Ltd. April 15, 1970 [April 16, 1969], No. 18053/70. Heading G2C. A silver halide developing solution comprises a silver halide developing agent and an inositolpolyphosphoric acid or an alkali metal salt thereof. The developing agent may be a colour or black and white developing agent and the additive may be inositolhexaphosphoric acid, inositolpentaphosphoric acid, inositoltetraphosphoric acid or 9Na, 11Na, or 7K inositolhexaphosphate. These compounds have very strong chelating properties which prevent stains formed during development as well as very strong aerial fog inhibiting properties without being harmful to. photographic materials and developers. The compounds are also effective as hard water softeners and preservatives.
Patent GB-1252016-A (GB)
IPC: F16B35/00
Filed: 1968-12-18
Abstract: 1,252,016. Making bolts; welding by fusion. STANDARD PRESSED STEEL CO. 18 Dec., 1968 [20 Dec., 1967], No. 60257/68. Headings B3A and B3R. [Also in Division F2] A method of making a bolt or the like comprises providing a stud 10 having a first threaded section 12 spaced from one end of the stud by an abutment shoulder 13 and engaging a nut 20 on the threaded section 12, so that an end face of the nut bears against the shoulder 13. The stud and nut are mechanically worked by conventional equipment to the desired shapes and then heat treated. After heat treatment the threads are formed on the stud and in the bore of the nut. The stud and nut are normally of stainless steel, but two different compatible alloys may be used, the stud at least being of an alloy which develops high strength properties, either by the combination of mechanical working and heat treatment or by mechanical working alone. The stud and nut may be secured by electron beam welding along a length of their threaded engagement to form a weld seam 30. Alternatively, either or both abutting surfaces may be knurled or roughened.
Patent GB-1257023-A (GB)
IPC: F24H9/00
Filed: 1968-01-31
Abstract: 1,257,023. Air supply to liquid heaters. SANTON Ltd. 14 April, 1969 [31 Jan., 1968], No. 4962/68. Heading F4W. [Also in Division H1] In a fuel-fired liquid heater, the combustion air blower 5 and a transformer connected to the electric control systems of the heater are so mounted that air passing through the blower cools the transformer. The blower 5, its drive motor 13 and the transformer are mounted in a box 6 having an inlet 7 for air and an outlet 8 connected to the blower outlet. To restrict vibrations, the outlet 8 of the box is connected to the air inlet to the combustion chamber of the heater by a flexible pipe. The box 6, together with the blower, motor and transformer, can be readily removed from the heater for servicing.
Patent GB-1257380-A (GB)
IPC: H02K33/10
Filed: 1969-07-30
Abstract: 1,257,380. Vibrators. GOSUDARSTVENNY NAUCHNO - ISSLEDOVATELSKY I PROEKTNY INSTITUT UGOLNOI PROMYSRLENNOSTI. 30 July, 1969, No. 38185/69. Heading F2X. [Also in Division H3] A vibrator, for example for a rock conveyer, comprises a thyristor type inverter 9 driving the stator winding 3 and controlled by a pick-up 6 associated with the vibrating elements 4, 5 so that the arrangement oscillates at the natural frequency of vibration. The pulsating magnetic flux created provides alternating attraction to the stator 1 of the electromagnet moving parts 4 which are connected by flexible links, e.g. springs, to the stator 1 and connected rigidly to the working element 5. The arrangement described uses a velocity sensitive pick-up 6, an amplifier 7 and a switching circuit 8. D.C. is fed to a separate stator winding 2 from a rectifier supplied from the mains or from the inverter output.