baber/WOPTO huggingface dataset:
Patent BR-112022017727-A2 (BR)
Title: Inibidores de eif4e e usos dos mesmos
Inventor: CHRISTOPHER L VANDEUSEN
IPC: C07D417/04
Filed: 2021-03-03
Abstract: INIBIDORES DE EIF4E E USOS DOS MESMOS. A presente invenção refere-se a compostos que inibem a atividade de eIF4E e composições e métodos de uso dos mesmos.
Patent BR-112022020904-A2 (BR)
Title: Método e aparelho para dispensar uma bebida super-refrigerada
Inventor: PETRUS JOHANNES VAN GEIJLSWIJK
IPC: B67D1/08
Filed: 2021-04-16
Abstract: MÉTODO E APARELHO PARA DISPENSAR UMA BEBIDA SUPER-REFRIGERADA. Um método e dispositivo são fornecidos para dispensar uma bebida. O método compreende resfriar uma bebida a uma primeira temperatura abaixo de um ponto de fusão da bebida, receber um recipiente de bebida com um volume de armazenamento para receber a bebida, pressurizar o volume de armazenamento do recipiente de bebida até uma primeira pressão, dispensar a bebida no volume de armazenamento pressurizado do recipiente de bebida, e diminuir a pressão no volume de armazenamento do recipiente de bebida até a pressão ambiente, em que a bebida é resfriada a uma primeira temperatura abaixo de um ponto de fusão da bebida antes de diminuir a pressão no volume de armazenamento do recipiente de bebida à pressão ambiente. O dispositivo pode ser disposto para realizar partes do método.
Patent BR-112022021299-A2 (BR)
Title: Microesferas termicamente expansíveis e processo de preparo de microesferas termicamente expansíveis
Inventor: BO ANDREASSON
IPC: B01J13/04
Filed: 2021-05-19
Abstract: MICROESFERAS TERMICAMENTE EXPANSÍVEIS E PROCESSO DE PREPARO DE MICROESFERAS TERMICAMENTE EXPANSÍVEIS. A invenção se refere a microesferas termicamente expansíveis que compreendem uma casca polimérica em torno de um núcleo oco, em que o núcleo oco compreende um agente de expansão, e a casca polimérica compreende uma celulose funcionalizada com carboxilato, em que as microesferas termicamente expansíveis têm uma temperatura na qual a expansão começa, TInício, de 80°C a menos de 135°C. A invenção se refere ainda a um processo para preparar microesferas expansíveis, bem como microesferas termicamente expansíveis obtidas por tal processo, em que o processo compreende misturar uma celulose funcionalizada com carboxilato, um solvente orgânico, um agente de expansão e, opcionalmente, um potencializador da casca de polímero e, em seguida, pulverizar a mistura assim obtida em um equipamento de secagem para produzir as microesferas termicamente expansíveis tendo uma casca polimérica em torno de um núcleo oco, em que a casca polimérica compreende a celulose funcionalizada com carboxilato, e o núcleo oco compreende o agente de expansão.
Patent BR-112022024697-A2 (BR)
Title: Agente antimicrobiano para animal não humano
Inventor: HIROSHI SHIKAMA
IPC: A61K31/4164
Filed: 2021-06-02
Abstract: AGENTE ANTIMICROBIANO PARA ANIMAL NÃO HUMANO. Um novo agente antimicrobiano é provido e um composto representado pela fórmula (I) ou (II) ou um sal do mesmo é usado como um agente antimicrobiano para um animal não humano.
Patent BR-112023001634-A2 (BR)
Title: Método de preservação de um composto ativo reativo, cápsula e formulação
Inventor: TOM KAMPERMAN
IPC: A61K9/107
Filed: 2021-08-03
Abstract: MÉTODO DE PRESERVAÇÃO DE UM COMPOSTO ATIVO REATIVO, CÁPSULA E FORMULAÇÃO. Um composto ativo reativo é colocado em um líquido. O referido líquido, contendo o referido composto ativo, é encapsulado por uma camada de revestimento circundante e compreende uma emulsão de um primeiro líquido em um segundo líquido. O referido composto ativo é disperso no referido primeiro líquido. O referido primeiro líquido, contendo o referido composto ativo, é disperso em um segundo líquido que é substancialmente imiscível com o referido primeiro líquido para formar a referida emulsão. A referida emulsão é encapsulada pela referida camada de revestimento para preservar o referido composto ativo reativo em uma ou mais cápsulas que podem ser aplicadas em uma formulação.
Patent BR-122015014056-A2 (BR)
Title: âncora de fixação, segmento de torre, arranjo de preensão para prender um segmento de torre, e, processo para produção de um segmento de torre
Inventor: GÜNTHER HORN
IPC: E04H12/12
Filed: 2012-06-14
Abstract: 1/1 resumo âãncora de fixaãão, segmento de torre, arranjo de preensão para prender um segmento de torre, e, processo para produãão de um segmento de torreâ a presente invenã§ã£o se refere a um mã©todo para produzir um segmento de torre de uma torre de concreto de uma instalaã§ã£o de energia eã³lica, compreendendo as etapas: prover um molde de segmento tendo pelo menos um isolamento para definir um molde do segmento de torre que deve ser produzido e encher com concreto; encher o molde de segmento com concreto a fim de formar o segmento de torre pelo subsequente endurecimento do concreto; medir o segmento de torre entã£o endurecido para criar um modelo atual virtual tridimensional do dito segmento de torre; produzir o dito modelo atual tridimensional; comparar o modelo atual tridimensional com um molde prã©-definido, em particular um modelo alvo virtual tridimensional armazenado; e determinar um desvio entre ambos os modelos virtuais e alterar o molde de segmento, em particular alterar o pelo menos um isolamento quando o desvio excede um primeiro valor limite prã©- definido.
Patent CZ-25694-A3 (CZ)
Title: Process of removing methoxyaromatic contaminants from vapour phase of natural mixtures of cresolic acid
Inventor: STRUNK MARVIN H
IPC: C07C37/70
Filed: 1992-07-09
Abstract: A process for removing guaiacols from naturally-occurring cresylic acid mixtures by pyrolysis is described.
Patent CZ-51999-A3 (CZ)
Title: 25-methylene and 24,25 epoxymarcfortines and paraherquamides
Inventor: LEE BYUNG H
IPC: A61P33/00
Filed: 1997-09-05
Abstract: The present invention are marcfortines and paraherquamides where the 7-member oxygenated ring has been modified to produce 25-methylene compounds (VII) and 24,25-epoxy compounds (VIII) all of which are useful as antiparasitic agents against endo and ecto parasites, particularly helminths and arthropods.
Patent SK-12397-A3 (SK)
Title: Pinned connection
Inventor: SMORADEK PETER
IPC: F16B5/02
Filed: 1997-01-28
Abstract: Two-part pin (1) consists of an external adjustable body (6) provided with a coaxial orifice. The orifice has an inside thread to admit an inside anchoring shackle (11) which is, on the other hand, provided with an external thread (12). An anchoring side (7) of the pin (1) is provided with a recess (10) and the front side (4) contains a groove (5). Said front side (4) has its cross-section smaller than the external adjustable body (6) of the pin (1) but is bigger than the groove (5).
Patent SK-24494-A3 (SK)
Title: Medicinal device for inhalation of dosed aerosols
Inventor: KLEIN CHRISTOPH
IPC: A61M16/12
Filed: 1992-08-28
Abstract: PCT No. PCT/DE92/00723 Sec. 371 Date Jun. 29, 1994 Sec. 102(e) Date Jun. 29, 1994 PCT Filed Aug. 28, 1992 PCT Pub. No. WO93/04718 PCT Pub. Date Mar. 18, 1993.A medical device for inhaling metered aerosol has a cylindrical housing with a receiving chamber for receiving an aerosol container and first main air channels extending axially within the housing. A mouthpiece is coaxially connected to the housing. An atomizing and vortexing chamber is delimited by the housing and the mouthpiece. Second main air channels extend within the mouthpiece and communicate with the first main air channels. A partition is positioned between the receiving chamber and the atomizing and vortexing chamber. The partition has a stepped bore with a first section and a second section, the first section having a larger diameter than the second section. The first section opens into the receiving chamber and the second section opens into the atomizing and vortexing chamber to form an aerosol outlet. Branch air channels extend at a slant to an axial direction of the medical device within the partition so as to surround the stepped bore. The branch air channels are connected to the first main air channels and open into the atomizing and vortexing chamber.
Patent SK-43393-A3 (SK)
Title: A lifting platform and method of its production
Inventor: BAR GERD
IPC: B60P1/44
Filed: 1993-05-04
Abstract: Loading wall especially for the rear of a trailer or a goods vehicle which is rectangular when viewed from above or below, but triangular when viewed from the side. The underside of the triangle, which has a very sharp peak, is formed by a loading bearing sheet (18). The underside sheet is essentially flat from the peak to the connection head (12, 13) near the cross beam (29). The cross beam and longitudinal beam configuration (68, 69) is placed between the upper and lower sheets and connected together by welded joints. USE/ADVANTAGE - Triangular section loading wall for goods vehicle can be made of steel or aluminium and avoids the danger of corrosion from entrapped water.
Patent SK-56496-A3 (SK)
Title: 5-arylisoxazol-4-yl-substituted 2-amino carboxylic acid compounds, pharmaceutical composition containing them and their use
Inventor: MOLTZEN LENZ S
IPC: A61K31/496
Filed: 1994-11-02
Abstract: 2-Aminocarboxylic acid compounds substituted with 5-arylisoxazol-4-yl or 5-arylisothiazol-4-yl and having general formula (I), wherein A is a bond or a spacer group; B is a group -CH(NR'R'')-COOH wherein R' and R'' are independently hydrogen or C1-6 alkyl, or B is a group of formula (II), wherein R2, R3 and R4 are substituents; or R3 and R4 or R4 and R2 are connected in order to form a ring; E is O, S, COO, (CH2)n-COO, O-(CH2)n-COO or S-(CH2)n-COO wherein n is 1-6, 5-tetrazolyl, 5-tetrazolyl-C1-6 alkyl, 3-hydroxyisoxazolyl or 3-hydroxyisoxazolyl-C1-6 alkyl; D is O or S; and R1 is an optionally substituted aryl or heteroaryl group; are excitatory amino acid receptor ligands useful in the treatment of cerebral ischaemia, Huntington's disease, epileptic disorders, Parkinson's disease, Alzheimer's disease, schizophrenia, pain, depression and anxiety. <CHEM>
Patent SK-84599-A3 (SK)
Title: G-rich oligo aptamers and methods of modulating an immune response
Inventor: TAM ROBERT
IPC: C12Q1/00
Filed: 1997-12-19
Abstract: Aptamer oligonucleotides specifically bind to the DNA binding site of proteins such as Sp1 and Sp1-related proteins which regulate the genes which encode costimulatory molecules such as CD28 and cytokines such as IL-2 and GMCSF. The oligonucleotides compete with the DNA-binding sites of regulatory proteins which specifically regulate molecules to modulate T-cell activation. This serves to modulate gene expression by preventing transcription of the gene. Aptamers are administered to provide therapies for diseases which involve aberrant T-cell activation such as psoriasis, Type I (insulin-dependent) diabetes mellitus, multiple sclerosis, autoimmune uveitis, rheumatoid arthritis, systemic lupus erythematosus, inflammatory bowel disease (Crohn's and ulcerative colitis), and septic shock and to regulate normal T-cell activation such as in allograft rejection.
Patent SK-92000-A3 (SK)
Title: Method and device for soldering the ends of tubular containers, specially tubes
Inventor: SATOR ALEXANDER P
IPC: B29C65/16
Filed: 1998-07-10
Abstract: Method for welding the ends of tubular containers filled with a pourable medium, in particular tubes, made from a thin-walled flat material which can be softened or melted through heat, wherein the tubular container is held in such a fashion that the end which is to be welded is accessible and the tubular container is heated at the accessible end in a peripheral region to a temperature which allows welding thereof, and the heated end is pressed together along an elongated welding seam transverse to the longitudinal extension of the container, wherein the tubular container is stationary and a laser beam is directed, via a deflection element positioned outside of the tubular container, onto the inner wall of the tubular container, and the deflection element is set into rotation for heating the peripheral region.
Patent CZ-226192-A3 (CZ)
Inventor: HINZE JAN
IPC: H04M1/74
Filed: 1992-07-21
Abstract: První vodič (a) účastnického vstupu ústředny je připojen k
prvnímu vývodu spínače (S). Jeho druhý vývod je spojen s
prvním vývodem účastnického zařízení (U), jeho druhý
vývod je připojen paralelné ke druhému vodiči (b)
účastnického vstupu ústředny a ke druhému vývodu obvodu
(F) pásmového filtru, připojeného svým prvním vývodem
ke třetímu vývodu spínače (S). Tento spínač (S) ovládá zapojení
obvodu (F) pásmového filtru k vodičům (a,b)
účastnického vstupu ústředny v době průběhu hovorového
spojení a rovněž zajišťuje odpojení, resp. nepřipojení obvodu
(F) pásmového filtru k vodičům (a,b) účastnického vstupu
ústředny v době, kdy jsou po této cestě realisovány jiné
, spojové služby, např. dekadická impulsní volba nebo
' účastnické vyzvánění.
Patent CZ-254992-A3 (CZ)
Inventor: RYBA IVAN ING
IPC: B29C48/32
Filed: 1992-08-19
Abstract: Vnitřní povrch trubky je opatřen spirálovitými drážkami s
úhlem stoupání 70 až 89 0 a hloubkou 50 až 500 lm. Trubka
je vybavena zatahovacím lankem (5) procházejícím volně
celou délkou trubky. Zařízení k výrobě této trubky pak
sestává z vytlačovacího stroje s přesazenou nebo kolmou
vytlačovací hlavou (2) s trnem (1). Kalibrační trn (1) je
volně otočný a chlazený médiem, procházejícím vytlačovací
hlavou (2), tepelně od ní oddělený izolační vložkou (3) a
na povrchuje opatřen spirálovitými drážkami odpovídajícími
drážkám na vnitřním povrchu vytlačované trubky. Vytlačovací
hlava (2) ikalibrační trn (1) jsou duté a umožňují M zavádění zatahovacího lanka (5).
Patent CZ-255892-A3 (CZ)
Inventor: NEMRAVA JIRI
IPC: E03C1/01
Filed: 1992-08-20
Abstract: Po spláchnutí WCje voda z plovákového ventilu (3) vedena
trubkou (6), usměrňována výtokovou hubicí (7) do umývátka
(8) a z něj pak odtokovou trubkou (9) do nádržky (2). Je
uvažováno s variantami způsobu provedení a umístění
umývátka (8) formou nástavby vyráběného kombi WC a zapojení
stávajících typů umývátek (8)
Patent CZ-312092-A3 (CZ)
Inventor: MALINA JOSEF
IPC: F24H1/10
Filed: 1992-10-14
Abstract: Deskový elektrický ohřívač vody, zejména pro průtokové
ohřívače, sestávající ze dvou po obvodě vodotěsně spojených
desek, vyznačující se tím, že na vnitřních k sobě přilehlých
plochách je vytvořen kanál (3) menšího průřezu
než kanál (2), který vytváří mezi stěnou kanálu (2) a trubkovým
topným tělesem (3) průtokový prostor (4), přičemž
kanál (2) je z jedné strany desky na svém začátku opařen
přítokovým otvorem (5) a na odvrácené straně výtokovým
otvorem (6).
Patent CZ-381492-A3 (CZ)
Title: Steering device of a vehicle front and rear axle wheels
Inventor: KOVAR JOSEF
IPC: B62D7/14
Filed: 1992-12-21
Abstract: The steering device for a vehicle with front axle wheels (1) and rear axle wheels (2) has the wheels (1,2) of the same axles connected by linking rods (5), which engages with the levers (4) arranged on the wheel (1,2) hubs (3). The wheel (1,2) hubs (3) on one side of the vehicle is connected with the steering levers (6), connected to the steering rods (7,8). The steering rods (7,8) are connected to the timing gear (9), formed by a rocker (16) pivoted on the vehicle around the turning axis (17). On the rocker (16), outside the turning axis (17), there is a swinging transmission member (10) of control movement and, through the joints (21), the steering rods (7,8). The joints (21) are provided with adjustment blocks (20), which are each slide fitted in one guide (18,19) of the rocker (16). The guides (18,19) have the form of circular arches, whose diameters correspond to the lengths of the corresponding steering rods (7,8). The guides (18,19) lie in two mutually varied levels and overlap with their centre parts in the area of the turning axis (17). If the adjustment blocks (20) are in the central parts of the guides (18,19), the centres of the joints (21) lie in the turning axis (17). The adjustment blocks (20) are connected to the link chains (24), guided in the guides (18,19) and each link chain (24) has a chain gear (25) pivoted on the rocker (16).<IMAGE>
Patent CZ-111399-A3 (CZ)
Title: Device for automatic transport of workpieces in multistage chipless forming machine
Inventor: STEINHAUSER ULRICH
IPC: B21K27/00
Filed: 1997-09-29
Abstract: A device for the automatic conveyance of workpieces on a multistage metal-forming machine tool with a tong case (1) located on a cross conveyor tube (2). Tong case (1) comprises a base body (10) on which interchangeable tong cartridges (12a, 12b, 12c), each with a pair of tongs enabling workpiece (W2,W3) to be gripped laterally from above, are placed. Each pair of tongs is connected via a coupling point (19) to means of transmission associated thereto. Said means interact with a control shaft (3) which is placed rotatably in the cross conveyor tube (2) to control opening and closing movement of tongs. Conveyance of a workpiece (W2, W3), grasped by one pair of tongs with twin interacting grippers (130, 140), from one metal-forming station (U1,U2,U3) to a neighbouring metal-forming station (U2,U3,U4) and the return movement of the tongs occur when the cross conveyor tube (2) moves back and forth. Tong travel can be adapted to workpieces by using tong cartridges (12a,12b, 12c) with tongs having appropriate lever ratios.
Patent CZ-142196-A3 (CZ)
Title: 2-pyrazolinone-5-derivative, process of its preparation and pharmaceutical composition containing thereof
Inventor: ARLT MICHAEL DR
IPC: C07D413/12
Filed: 1996-05-16
Abstract: 4-(Arylaminomethylidene)-2,4-dihydropyrazol-3-one cpds. of formula (I) (sic) and their salts are new. R1 = benzyl, 1-3C alkoxybenzyl, phenyl (opt. mono-, di- or tri-substd. with amino, acyl, halo, nitro, CN, OA, carboxyl, sulphonyl, COOA, NHCOA, NACOA, carbamoyl (opt. mono- or di-substd. by 1-6C alkyl), NHCOOA, NACOOA, SO2A, SO2NR4R5, SO2NHCOA, SO2NACOA, NHSO2A, NASO2A, N(SO2A)2, tetrazolyl or phosphonyl) or pyridyl; R2 = 1-5C alkyl, alkoxycarbonylalkyl, hydroxyalkyl or hydroxycarbonyl; R3 = H, 1-5C alkyl (opt. substd. by F or Cl), 1-5C alkoxy, aminoalkanoyl, aminoalkyl, carbamoyl, SO2NR4R5; R4, R5 = H or 1-6C alkyl; or NR4R5 = 5- or 6-membered ring opt. with other heteroatoms like N, S, O, and opt. substd. by A); A = 1-6C alkyl (opt. substd. by F or Cl).
Patent CZ-176797-A3 (CZ)
Title: Rail wheel with a disk connecting head and rim of the wheel
Inventor: MURAWA FRANZ ING
IPC: B60B17/00
Filed: 1995-11-20
Abstract: PCT No. PCT/EP95/04561 Sec. 371 Date Jun. 6, 1997 Sec. 102(e) Date Jun. 6, 1997 PCT Filed Nov. 20, 1995 PCT Pub. No. WO96/18512 PCT Pub. Date Jun. 20, 1996A stress-homogenized track wheel with a wheel disk (3) which connects the wheel hub (1) and wheel rim (2) and decreases in thickness from the hub (1) towards the rim (2), the disk's outer surfaces merging via three-center curves as radial generatrices tangentially with the adjacent outer surfaces of the hub (1) and rim (2) is shown. In order to suppress stress peaks and reduce the stress across the radial width of the wheel disk, the two outer surfaces of the wheel disk (3) are defined in the radial central area (1) geometrically by radial straight generatrices (Z3*,Z3**) which intersect in the area between the three-center curves on the wheel rim (2).
Patent CZ-201039-A3 (CZ)
Inventor: STACH JAN
IPC: A61K47/12
Filed: 2010-01-19
Abstract: Rešení se týká amorfní formy hemivápenaté soli (3R,5R) 7-[3-fenyl-4-fenylkarbamoyl-2-(4-fluorfenyl)-5-isopropylpyrrol-1-yl]-3,5-dihydroxyheptanové kyseliny (atorvastatinu vzorce I) s vysokým specifickým povrchem založeného na rízeném srážení a jeho použití v lékové forme.
Patent CZ-234694-A3 (CZ)
Inventor: SLABY VLADISLAV ING
IPC: A01D46/24
Filed: 1994-09-26
Abstract: Pomůcka pro trhání zejména ovocných plodů se skládá z
pevného oka (1), přítlačného oka (2), motouzu a pružiny
(3). Pomůcka je vyrobena z hliníkového drátu lehce tvarovatelného
a opatřeného v místě styku s plodem plastovou
vrstvou. Tahem za motouz se plod přitlačí přítlačným okem
(2) k pevnému oku (1) a po spuštění plodu k zemi pružina
(3) plod ze sevření uvolní.
Patent CZ-255196-A3 (CZ)
Title: Feeding automatic machine for pulverized bulk material, particularly coffee in the form of a powder
Inventor: FREUND EDGAR
IPC: G01F13/00
Filed: 1995-02-22
Abstract: An automatic metering device for powdery bulk material, in particular coffee powder, has a reservoir (1) with a wall (2) and a stationary base plate (3) for the bulk material. The base plate (3) has an opening (4) to a conveyor tube (5) which is disposed below said plate and in which a conveyor member (6) is disposed for conveying the bulk material to a delivery location. According to the invention, the wall (2) of the cylindrical reservoir (1) is rotated during the metering process, and a sensor is provided for determining the amount to be delivered by the conveyor member. The appliance of the invention enables bulk material, in particular coffee powder, to be metered simply and accurately without the risk of bridges forming inside the reservoir such that the bulk material poured in first is also dispensed first.
Patent CZ-265096-A3 (CZ)
Title: Thienoindole derivatives, their use, process of their preparation and pharmaceutical composition containing thereof
Inventor: JAKOBSEN PALLE
IPC: C07D209/18
Filed: 1995-03-10
Abstract: The present invention relates to therapeutically active heterocyclic compounds, a method of preparing the same and to pharmaceutical compositions comprising the compounds. The novel compounds are useful in treating diseases in the central nervous system related to the metabotropic glutamate receptor system.
Patent CZ-279894-A3 (CZ)
Title: Fundamental element of detachable spatial brick blocks
Inventor: PRIHODA JAROSLAV ING
IPC: A63F9/12
Filed: 1994-11-14
Abstract: The device consists of an n-block right angled prism at least three walls of which are equipped with raised joining elements (2) which are staggered along the walls. The prism is a three-side right angled prism, the main cross section of which is a right angled triangle.<IMAGE>
Patent CZ-316495-A3 (CZ)
Title: 14-substituted marcfortines and and derivatives usable as antiparasitic substances
Inventor: LEE BYUNG H
IPC: A61K31/535
Filed: 1994-06-07
Abstract: There are disclosed 14 alpha -hydroxymarcfortine derivatives of the natural products marcfortine A, B, C, and D useful in the treatment and prevention of helminth and arthropod infections of animals and plants. The synthetic derivatives are of Formula (I).
Patent CZ-325598-A3 (CZ)
Title: Process for producing liquid pig iron of liquid steel half-finished product
Inventor: WIESINGER HORST
IPC: C21B13/02
Filed: 1998-02-10
Abstract: The invention concerns a method of producing liquid crude iron or liquid steel fabricated materials from material containing iron oxide. According to this method, fine-particle material which contains iron oxide is reduced by means of a reduction gas in at least one fluid bed reduction stage (7, 8) by the fluid bed process to form fine-particle iron sponge and lumps of ore are reduced in a fixed bed reduction stage (28) to form lumps of iron sponge. The iron sponge is introduced into a fusion gasification zone (11) and melted there by the addition of carbon-carriers and oxygenous gas, a CO and H2-containing reduction gas being produced to reduce the material containing iron oxide. In order to avoid having to treat the fine-particle iron sponge separately from the lumps of iron sponge, the fine-particle iron sponge in the un-processed state and fine-particle form is introduced directly into the fusion gasification zone (11) and melted therein together with the lumps of iron sponge.