baber/WOPTO huggingface dataset:
Patent JP-H0625252-A (JP)
Title: New alpha-aminoquinolinoyl-(3)-penicillin, its production and antibacterial agent containing it
Inventor: GIZERA KUBITSUTOSHIYOORU
IPC: A61P31/04
Filed: 1992-01-22
Abstract: PURPOSE: To obtain a novel compound with an antibacterial activity, which is useful as a remedy for infectious disease.  
     CONSTITUTION: This novel compound is expressed by formula I (wherein R 1  is H, Na, K, Ca, 1-6C alkyl ammonium or the like; R 2  is H or alkoxycarbonyl; R 3  is H, 1-6C alkyl, 1-5C alkoxy, halogen or the like; R 4  is H, 1-4C alkyl or the like; R 5  is H, alkyl, methoxy or the like; R 6  is H, 1-4C alkyl, acetyl or the like; R 3  and R 4  binds together to form a condensed ring), e.g. 6-[D-(-)-α-([4'- ethoxycarbonyloxy-6'-ethyl-7'-(4"-chloro)-phenoxymethylene-quinolinoyl-3']- carboxamide)-α-phenylacetoamide]-penicillinic acid-sodium salt. The compound of formula I is obtained by converting a substituted quinoline-3-carboxylic acid of formula II, in a form of a mixed anhydride or an active ester, with an α- aminobenzylpenicillin base structure of formula III. 
     COPYRIGHT: (C)1994,JPO
Patent JP-S60154274-A (JP)
Title: Toner cartridge of developing device for copying machine
Inventor: KONISHI KEIJI
IPC: B65D83/06
Filed: 1984-01-24
Abstract: PURPOSE:To prevent toner from scattering out of a machine during the replacement of a cartridge by fixing an external cylinder to the cylindrical guide of a toner supplementing device without reference to the rotation of the internal cylinder when the cartridge is inserted. CONSTITUTION:The principal part of the toner cartridge 13 consists of the external cylinder 15 which has an opening 14 for toner discharging lengthwise and the internal cylinder 17 which is fitted rotatably in the external cylinder 15 and has an opening 16 aligned to said opening part 14 lengthwise. The opening part 16 of the internal cylinder 17 is formed to at least the same and same size with the opening 14 of the external cylinder 15, and normally positioned in the opposite direction in which its position is not coincident with that of the opening 14. Further, a knob for rotating the cylinder 17 in the external cylinder 15 is formed at one end of the internal cylinder 17.
Patent JP-S55102246-A (JP)
Title: Method for indicating defective semiconductor chip
Inventor: UMETSU TSUNENORI
IPC: H01L21/66
Filed: 1979-01-29
Abstract: PURPOSE: To increase the speed of the indication of a defective chip by providing additional pads other than bonding pads on a semiconductor chip, by wiring said bonding pads and said additional pads, and by electrically melting out the wiring if the chip is found to be defective as a result of a check.  
     CONSTITUTION: Bonding pads 11 a  and 11 b  whose configurations are different each other are formed on a semiconductor substrate 1. On said semiconductor chip 1, are formed additional Al pads 12 a  and 12 b  whose configurations are approximately the same as the configurations of said pads 11 a  and 11 b . Then, said additional pads 12 a  and 12 b  are connected to the pads 11 a  and 11 b  by using thin Al wirings 13 a  and 13 b . In this constitution, the chip is checked by contacting a probe with the pads 11 a  and 11 b . If the chip is defective, a current is flown by using the additional pads 12 a  and 12 b  and the wirings 13 a  and 13 b  and the like are burned out. In this way, the indication of the defective chip becomes clear and easy by the observation of the melted portions. 
     COPYRIGHT: (C)1980,JPO&Japio
Patent JP-H10206375-A (JP)
Title: Cover for oxygen sensor
Inventor: KIKUCHI TOMOSHI
IPC: G01N27/409
Filed: 1997-01-22
Abstract: PROBLEM TO BE SOLVED: To restrain introducing holes of the cover from being clogged by a deposit sticking to a cover for an oxygen sensor. SOLUTION: An oxygen sensor 20 installed in an intake pipe of a diesel engine has a sensor element 21 composed of solid electrolyte such as a zirconia element and a cover 22 having plural introducing holes 31. Deposit removing members 40 are arranged in the respective introducing holes 31. The deposit removing members 40 have column parts 41 inserted into the introducing holes 31 and disk parts 42 and 43 respectively formed on both end sides of the column parts 41. Outer peripheral surfaces of the column parts 41 slidingly move in the inside and outside direction of the cover 22 to an inner peripheral wall surface of the introducing holes 31 according to vibration of an engine or a vehicle.
Patent JP-S5292938-A (JP)
Title: Controlling method for correcting power in arc furnace
Inventor: MIYASHITA TETSUO
IPC: F27D11/08
Filed: 1976-01-31
Abstract: PURPOSE: To avoid excess power consumption and to prevent from production delay by means of calculating thermal loss when operation in stopping due to an accident of arc furnace. 
     COPYRIGHT: (C)1977,JPO&Japio
Patent JP-S61168477-A (JP)
Inventor: KOMURA SEIICHI
IPC: B25H1/10
Filed: 1985-01-21
Abstract: (57)【要約】本公報は電子出願前の出願データであるた め要約のデータは記録されません。
Patent JP-S63181832-A (JP)
Inventor: SEGIRI ARAO
IPC: E04B1/70
Filed: 1987-01-19
Abstract: (57)【要約】本公報は電子出願前の出願データであるた め要約のデータは記録されません。
Patent JP-H01186868-A (JP)
Title: Pyrazole compound and herbicide containing said compound as active ingredient
Inventor: TSURUYA TETSUO
IPC: A01N47/36
Filed: 1988-01-21
Abstract: NEW MATERIAL:A pyrazole compound expressed by formula I (X is halogen). EXAMPLE:5-tert-Butyl-3-(N-dimethylcarbamoyl-N-methylamino)pyrazole. USE:useful as a herbicide, capable of remarkably inhibiting growth of weeds and killing the weeds by spraying on the soil surface or mixing in soil and also controlling the weeds by spraying on foliar parts of the weeds during growth, effective against broad-leaved weeds, such as chickweed, gramineous weds, such as annual bluegrass, and cyperaceous weeds, such as flat-sedge, with low phytotoxicity to crops. PREPARATION:As shown in the reaction formula, a compound expressed by formula II is reacted with N,N-dimethylcarbamoyl chloride in the presence of an inorganic base, such as sodium carbonate, in an organic solvent, such as benzene, at 30-120 deg.C to afford the aimed compound expressed by formula I.
Patent JP-H01185719-A (JP)
Title: Coordinate detector
Inventor: UCHIYAMA BUNJI
IPC: G06F3/03
Filed: 1988-01-21
Abstract: PURPOSE:To increase the number of detection of a coordinate value and to obtain plotting data with high accuracy even at hand-writing speed by performing the detection of coordinate for only a first coordinate detection point by taking out the output signals of first and second conductor groups, and performing the detection of coordinate for the coordinate of another coordinate detecting point by taking out the output signal of the conductor group on one side. CONSTITUTION:When a line is plotted on a coordinate detecting plate 21 by an indicator 6, the coordinate value of a position on the coordinate detecting plate 21 being brought into contact first is detected by using the first and second conductor groups. And following coordinate values in the same pitch area are detected by finding the position of the indicator 6 with respect to a prescribed conductor in the conductor group on either side and computing a difference between the position and the position with respect to the prescribed conductor at a preceding coordinate detecting point and adding the difference on the coordinate value of the indicator 6 at the preceding coordinate detecting point. In such a way, it is possible to increase the number of detection of the coordinate value in a unit time.
Patent JP-H10202302-A (JP)
Title: Grooved bar for welded tube and its manufacture
Inventor: MORI YASUTOSHI
IPC: F28F1/40
Filed: 1997-01-23
Abstract: PROBLEM TO BE SOLVED: To obtain the grooved bar for a welded tube having a uniform groove shape and excellent weldability by forming a great number of grooves in the part excluding both end parts in the width direction of a bar stock and forming at least one groove each boundary in the boundary between the groove forming part and end parts in parallel with the length direction of the bar stock more deeply than grooves in the groove forming part. SOLUTION: The bar stock 10 is rolled down between a groove roll 20 and a flat roll 22, a great number of groove forming projecting parts B of the height (b) are formed in the spiral groove forming part 25 of the groove roll 20, and a great number of spiral grooves E are formed in the part excluding both end parts T on the upper surface of the bar stock 10 by the projecting parts B. Also, grooves G are formed in parallel with the length direction of the bar stock 10 in respective boundaries between the spiral groove forming part 25 and both end parts T by expanding parts K of the groove roll 20. Here, expanding parts K are formed higher than the projecting parts B and parallel grooves G are formed deeper than spiral grooves E.  The action, restraining that the material of the spiral grooves E forming part 25 is made to flow into the end parts T and whereby the groove part in the vicinity of the end parts T of the groove forming part 25 of the bar stock 10 becomes shallow, is achieved by expanding parts K.
Patent JP-H01183843-A (JP)
Title: Manufacture of semiconductor device
Inventor: HONDA HIROMI
IPC: H01L27/06
Filed: 1988-01-19
Abstract: PURPOSE:To form a semiconductor device having electric characteristics required by forming a conductive film onto an insulating film including a thin gate insulating film, applying the insulating film even when a mask layer at the time of the formation of a contact hole in a BIP (bipolar) transistor is removed and avoiding the exposure of the main surface section. CONSTITUTION:A contact hole 20 to which an electrode layer 23 for a conductive film 21 must be connected is bored to the conductive film 21 in a BIP transistor under the state in which a thin insulating film 6a as a gate insulating film is applied by the conductive film 21 shaped onto a substrate 1. Since gate electrodes 24, 25 are formed to conductive films 21, 22 shaped through the same process in a MOS transistor, sections as gate insulating films under the gate electrodes 24, 25 are protected and expected shapes are acquired even when contact holes 20 are formed. Accordingly, the MOS transistor having excellent electric characteristics is formed, thus improving the performance of a semiconductor device.
Patent LV-11884-A (LV)
Inventor: OLBRICH MATTHIAS
IPC: A61K47/14
Filed: 1997-05-14
Abstract: The invention relates to formulations of cyclosporin with high bioavailability for oral administration, which contain about 1 part by weight of one or more cyclosporin(s), preferably cyclosporin A and/or cyclosporin G, 7.5 to 7.8 parts by weight of one or more polyethylene glycol esters of saturated C10-C22hydroxy fatty acids, 0.7 to 0.85 part by weight of a monohydric alcohol as co-solvent, and 0.7 to 0.8 part by weight of a polyhydric alcohol as co-solvent. The drug form is produced by initially dissolving the cyclosporin in ethanol and, while stirring, adding propylene glycol and SOLUTOL(R) HS 15 until a clear, viscous solution results, bottled as drinkable solution or packed into capsules.
Patent ME-00557-A (ME)
Inventor: BROWN ALAN DANIEL
IPC: C07D295/03
Filed: 2005-01-12
Abstract: Pronalazak se odnosi na jedinjenja formule (1) i na postupke za njihovo dobijanje, na intermedijere koji su korišćeni za njihovo dobijanje, preparate koji sadrže ove derivate i njihova upotreba. Jedinjenja predmetnog pronalaska su korisna kod brojnih bolesti, poremećaja i stanja, posebno upalnih, alergijskih i respiratornih bolesti, poremećaja i stanja.
Patent TR-26084-A (TR)
IPC: A23D7/02
Filed: 1990-11-21
Abstract: The present invention is concerned with a stable edible dispersion comprising 95 to 86% by weight of an aqueous phase and 5 to 14% by weight of a continuous fat phase having and N20-value of at least 5. It is surprising that, provided suitable processing conditions are applied and a seeding component is employed, stable dispersions containing less than 14% by weight of a continuous fat phase having an N20-value of at least 5, and more than 86% by weight of an aqueous phase can be prepared. Another aspect of the present invention is a method of preparing a dispersion comprising 95 to 86% of an aqueous phase and 5 to 14% by weight of a continuous fat phase having an N20-value of at least 5, said method comprising cooling and working an emulsion of oil and water, the oil comprising 0.1-4%, by weight of the oil, of a solid seeding component.
Patent YU-204682-A (YU)
Title: Process for obtaining s-adenosylmethionine (sam) derivatives
Inventor: GENNARI F
IPC: C07H19/16
Filed: 1982-09-10
Abstract: New S-adenosylmethionine (SAM) salts of formula   <IMAGE> (I)  have been prepared in which R, R1, R2, m, n and A are as defined in the text. The methods of preparing the new products starting from SAM salts are described. The new products are stable and highly bioavailable, particularly when administered orally.
Patent YU-244790-A (YU)
Inventor: ANTOINE STOKBROEKX RAYMOND
IPC: A61K31/505
Filed: 1990-12-24
Abstract: Piperidinyl, pyrrolidinyl, azepinyl and piperazinyl pyridazines of formula <CHEM>  wherein X represents CH or N; R<1> represents hydrogen, C1-4alkyl, halo, hydroxy, trifluoromethyl, cyano, C1-4alkyloxy, C1-4alkylthio, C1-4alkylsulfinyl, C1-4alkylsulfonyl, C1-4alkyloxycarbonyl, C1-4alkylcarbonyl or aryl; R<2> and R<3> represent hydrogen or C1-4alkyl; Alk represents C1-4alkanediyl;  R<4> and R<5> represent hydrogen, C1-4alkyl or halo; and  Het represents <CHEM> the addition salts and stereochemically isomeric forms thereof, said compounds having antipicornaviral activity. Pharmaceutical compositions containing these compounds as active ingredient, and methods of preparing said compounds and pharmaceutical compositions.
Patent YU-64603-A (YU)
Title: Blowing erodible matrix system with controlled realease of active substance
Inventor: PETROVIC ALEKSANDAR
IPC: A61K9/30
Filed: 2003-08-12
Abstract: Invention refers to pharmaceutical products, tablets and/or film coated tablets, containing in high dosage incorporated one or more active substances of different solubility and blowing erodible polymer and/or channel of forming agent - "channeling agent" and/or agent for lubrication and sliding and/or binding agent and diluent and a layer of film coating made of film forming polymer, plasticizer, colors and/or other pharmaceutically acceptable materials. Chubbing erodible matrix system in the form of tablets and/or film coated tablets of different geometry and forms, for oral application that is characterized by controlled, continual release of active substance without any delay of time or pulsation by a permanent speed during a delayed time (12 hours minimum), by a combined mechanism of controlled diffusion of active substance through a gel layer and controlled erosion of matrix itself and procedure for obtaining thereof.
Patent YU-79401-A (YU)
Title: 1-trifluoromethyl-4-hydroxy-7-piperidinyl-aminomethylchroman derivatives
Inventor: OBACH RONALD SCOTT
Filed: 2000-04-20
Abstract: This invention relates to novel 1-trifluoromethyl-4-hydroxy-7-piperidinyl-aminomethylchroman derivatives of formula (I) wherein R1 is C1-C6 alkyl; R2 is hydrogen, C1-C6 alkyl, halo C1-C6 alkyl or phenyl; R3 is hydrogen or halo; and R4 and R5 are independently hydrogen, C1-C6 alkyl or halo C1-C6 alkyl, their pharmaceutically acceptable salts, pharmaceutical compositions containing such compounds, and the use of such compounds to treat CNS, gastrointestinal and other disorders.
Patent RS-81804-A (RS)
Title: Process for preparing crystalline form i of cabergoline
Inventor: SHEIKH AHMAD
IPC: C07D471/04
Filed: 2003-03-10
Abstract: A process for producing crystalline form I of cabergoline, which process comprises the preparation of Form V using heptane as precipitation solvent, and its exclusive conversion into crystalline Form I of cabergoline. The present crystallization process from toluene-heptane solvent system for form V involves "reverse addition" of toluene-cabergoline concentrate to cold heptane.
Patent AP-818-A (AP)
Title: Process for the preparation of a natural medicinal liquor based on carica papaya and vinca rosea.
Inventor: AIZPURUA MANUEL SESMA
IPC: A61K36/00
Filed: 1997-02-06
Granted: 2000-03-14
Abstract: The process comprises using a bacteriostatic sugar cane spirits, the latex of a fruit obtained by incision arid further collected and which is macerated appropriately in said spirits, dissolving it with a mixer until a homogenous product is obtained,- then the product is filtrated, and the same operation is carried out with flowers, both being immersed in a magnetic field during the maceration to obtain, after the final filtration, a nan toxic liquor having a anti-tumoral activity.
Patent AU-1003692-A (AU)
Title: Tube with a rectangular cross-section
Inventor: PRAHS HARALD
IPC: B65D35/12
Filed: 1992-01-03
Abstract: A plastics tube produced by blow moulding has a main section (1) with an essentially constant cross-section over its length, which is formed by an even number of level wall sections (2, 3, 4, 5) whose wall sections (2, 4; 3, 5) located opposite to each other each has the same width. At the front end of the main section there is a tubular opening section (15) with a smaller diameter than that of the main section (1). At the rear end the main section (1) converges to an essentially straight end edge (11) which lies in a plane extending through the central longitudinal axis of the main section (1) and which joins two longitudinal edges of the main section (1), the end edge (11) lying within the enveloping curve of the outer surfaces of the walls (2, 3, 4, 5) of the main section (1). <IMAGE>
Patent AU-1056383-A (AU)
Title: Welding power supply
IPC: H02M7/162
Filed: 1983-01-18
Abstract: In a three phase welding power supply, the three phase power is connected to a welding arc by a power control circuit having three conducting paths for straight polarity current and three conducting paths for reverse polarity current. The power control circuit comprises a three phase bridge rectifier circuit (112) having eight bridge arms each including a silicon controlled rectifier (1, 2, 3, 4, 5, 6, 7, 8) with the bridge circuit being connected between the three phase power source (102) and the welding arc (124) which is in turn connected to the three phase power supply neutral (103). An inductor (116) is connected across the direct current terminals of the bridge circuit so that arc currentflows in one direction through the inductor (116) regardless of the polarity of the arc current. The conducting paths are selectively activated at nonzero voltage points to conduct repetitive sequences of independent numbers of straight polarity half cycles of arc current followed by independent numbers of reverse polarity half cycles of arc current to the welding arc. Pulses are generated in synchronism with each of the three power phases and counted to determine the activation sequences of the conducting paths. By controlling the generation of the pulses and the counts of the pulses at which the paths are activated, a variety of sequences are generated.
Patent AU-1272788-A (AU)
Title: Use of metformin in the preparation of medicines
Inventor: WIERNSPERGER NICOLAS
IPC: A61K31/155
Filed: 1988-03-04
Abstract: The invention relates to the use of metformin and its salts in the preparation of medicaments. This derivative is used in the preparation of medicaments manifesting anti-ischaemic and antianoxic properties. It is also employed in the preparation of medicaments intended for the treatment or regression of neovascularisation.
Patent AU-1339088-A (AU)
Title: Electric hotplate, apparatus and method for fitting a cover plate thereto
Inventor: KICHERER ROBERT
IPC: H05B3/68
Filed: 1988-03-22
Abstract: The lower cover plate of an electric hotplate is fixed to the hotplate body by a resilient fixing structure provided on the cover plate, engaging with gripping edges on the outer face of a downwardly directed, central cast pin. The fixing structure can be defined by radial or flap-like, inwardly-directed portions of the cover plate and additionally can have portions engaging on the lower face of the pin and which are firmly held by the final screwing down of the electric hotplate.
Patent AU-1407988-A (AU)
Title: A differential hydraulic jack with damping system for the control of electric circuit-breakers
Inventor: GRATZMULLER CLAUDE ALAIN
IPC: H01H33/34
Filed: 1988-03-31
Abstract: A differential hydraulic jack with a damping system for the control of electric circuit-breakers is provided with a floating ring which produces a damping action at the end of travel and is also provided with a damping extension stud which forms part of the jack piston and penetrates into the damping ring. No provision is made on the jack piston for any packing ring forming a seal with the jack cylinder. The damping ring carries two projecting lips constituting a double valve which forms a leak-tight seal with the bottom face of the jack piston and the internal face of the cylinder end. At the end of the travel of the piston, the damping ring forms a double sealing valve for shutting-off the supply/drain orifice of the jack.
Patent AU-1521395-A (AU)
Title: Aqueous prolonged release formulation
Inventor: HAGEMAN MICHAEL J
IPC: A61K9/00
Filed: 1995-01-09
Abstract: Prolonged parenteral release into the circulatory system of a cow of a bioactive bovine somatotropin at desirably effective levels can be achieved using novel compositions in which the bovine somatotropin is present in an aqueous liquid at a dose of at least about 150 mg and at a concentration of at least about 50 mg/ml. The aqueous bovine somatotropin formulation provides for the sustained release of bovine somatotropin into the circulatory system of the animal for greater than three (3) days.
Patent AU-1637792-A (AU)
Title: Agent for transdermal administration containing ergoline derivatives
IPC: A61K31/475
Filed: 1992-05-18
Abstract: Compsn. contains ergoline derivs. opt. in combination with one or more penetration promoters.  The ergoline deriv. is of formula (I); where the dotted line represents an opt. bond; R1 = H, halo or 1-4C alkylthio; R2 = 1-4C alkyl; salt of (I) may also be used. The cpd. is esp. liswide, 2-bromoliswide, tergwide, or protergwide, or their salts.
Patent AU-1778900-A (AU)
Title: Alpha-sulfin- and alpha-sulfonamino acid amides
Inventor: JEANGUENAT ANDRE
IPC: C07C311/11
Filed: 1999-12-01
Abstract: The invention relates to alpha-sulfin- and alpha-sulfonamino acid amides of the general formula Iincluding the optical isomers thereof and mixtures of such isomers,whereinn is a number zero or one;R1 is C1-C12alkyl, C1-C12alkyl substituted with C1-C4alkoxy, C1-C4alkylthio, C1-C4alkylsulfonyl, C3-C8cycloalkyl, cyano, C1-C6alkoxycarbonyl, C3-C6alkenyloxycarbonyl or C3-C6alkynyloxycarbonyl; C3-C8cycloalkyl; C2-C12alkenyl; C2-C12alkynyl; C1-C12haloalkyl; or a group NR12R13 wherein R12 and R13 are each independently of the other hydrogen or C1-C6-alkyl, or together are tetra- or penta-methylene;R2 and R3 are each independently hydrogen; C1-C8alkyl; C1-C8alkyl substituted with hydroxy, mercapto, C1-C4alkoxy or C1-C4alkylthio; C3-C8alkenyl; C3-C8alkynyl; C3-C8cycloalkyl; C3-C8cycloalkyl-C1-C4alkyl; or the two groups R2 and R3 together with the carbon atom to which they are bonded form a three- to eight-membered hydrocarbon ring;R4, R5, R6 and R7 are each independently hydrogen or C1-C4alkyl;R8 is C1-C6alkyl, C3-C6alkenyl or C3-C6alkynyl;R9 and R10 are each independently hydrogen or C1-C4alkyl; andR11 is either in whereinR14, R,15, R16 and R17 are each independently hydrogen or C1-C4alkyl,X is oxygen, sulfur or -NR18-, wherein R18 is hydrogen or C1-C4alkyl, andA is optionally substituted mono- or polycylic aryl or heteroaryl, andto the preparation of those substances and to agrochemical compositions comprising at least one of those compounds as active ingredient. The invention relates also to the preparation of compositions and to the use of the compounds or of the compositions in controlling or preventing the infestation of plants by phytopathogenic microorganisms, especially fungi.