baber/WOPTO huggingface dataset:
Patent CR-20170263-A (CR)
Title: Forma cristalina de sulfato acido de (s)-n- (5- ( (r)-2- (2,5-difluorofenil)-pirrolidin-1-il)-pirazolo[1,5-a]-pirimidin-3-il)-3-hidroxipirrolidina-1-carboxamida
Inventor: ARRIGO ALISHA B
IPC: C12Q1/48
Filed: 2015-11-16
Abstract: La presente invención se refiere a una novedosa forma cristalina de (S)-N- (5- ( (R)-2-(2,5-difluorofenil ) -pir rolidin-1-il )- pirazolo[1,5-a]-pirimidin-3-il) -3-hidroxipir rolidina-1-carboxamida, a composiciones farmacéuticas que contienen dicha forma cristalina, y al uso de la forma cristalina en el tratamiento del dolor, cáncer , inflamación, enfermedad neurodegenerativa o infección por Trypanosoma cruzi .
Patent CR-20190537-A (CR)
Title: Pyrazole magl inhibitors
Inventor: WIENER JOHN J M
IPC: C07D403/08
Filed: 2018-05-22
Abstract: Provided herein are pyrazole compounds and pharmaceutical compositions comprising said compounds. The subject compounds and compositions are useful as modulators of MAGL. Furthermore, the subject compounds and compositions are useful for the treatment of pain.
Patent EC-SP034765-A (EC)
Title: Derivados de bipiperidinilo y su uso como inhibidores de receptores de quimiocina
Inventor: ALBERT RAINER
IPC: C07D405/14
Filed: 2003-09-11
Abstract: Los derivados de piperidina de la fórmula I, como se dan a conocer en la memoria descriptiva, tienen interesantes propiedades farmacéuticas, por ejemplo como inhibidores de CCR5.
Patent EC-SP099330-A (EC)
Title: Compuesto de indol
Inventor: YASUMA TSNUNEO
IPC: A61K31/433
Filed: 2009-05-14
Abstract: El propósito de la presente invención es proporcionar un activador de glucocinasa útil como un agente farmacéutico tal como un agente para la profilaxis o tratamiento de diabetes, obesidad y similar. La presente invención proporciona un activador de glucocinasa que contiene un compuesto representado por la fórmula (I): en donde R1 es un átomo de hidrógeno o un átomo de halógeno; R2 es un grupo representado en donde cada símbolo se define en la especificación, o su sal o su profármaco.
Patent EC-SP109961-A (EC)
Title: Derivados de indol-2-ona disustituidos en 3, su preparación y su aplicación en terapéutica
Inventor: BARONI MARCO
IPC: A61K31/454
Filed: 2010-02-12
Abstract: La presente invención tiene por objeto los derivados de indol-2-ona disustituidos en 3, de fórmula general (I) : en la que , R1, R2, R3, R4, R5, Ar y n son tales como se han definido en la reivindicación 1, el procedimiento de preparación y la aplicación terapéutica de dichos compuestos. (I)
Patent EC-SP982437-A (EC)
Title: Metodo y aparato mejorados para recuperar la energia de desechos mediante combustion de los mismos en hornos industriales
Inventor: ARROYAVE GARCIA JOSE LUIS
IPC: F23G7/00
Filed: 1998-03-03
Abstract: Se divulga y se reivindica un método y aparato mejorados, para recuperar la energía de desechos mediante la combustión de los mismos en hornos industriales, particularmente de tipo rotatorio, que tienen un calcinador externo, alimentando tales desechos al ducto, para aprovechar eficientemente la energía producida por tal combustión, como una contribución al gasto total de combustibles necesarios para operar el horno industrial. Asi mismo, el método y aparato de la invención permiten la eliminación de desechos peligrosos que son desintegrados eficientemente al quemarlos y destruirlos hasta tener afluentes no tóxicos, queno producen contaminación atmosférica, ni tampoco ningun daño ambiental.
Patent FI-20050306-A (FI)
Inventor: LASTUNEN TURKKA
IPC: B27L1/10
Filed: 2005-03-22
Abstract: A method and an apparatus for harvesting wood by using a working machine (30, 31, 32) moving on terrain, according to which method the felled tree trunk (11) is caused to move through a harvester head (10). At least one debarking roller (20, 21) is adjusted relative to the longitudinal axis of the tree trunk (11) to an angle such that, when the cut tree trunk is being moved through the harvester head, there is created between the wood part of the tree trunk and the bark on it a shear force of a desired magnitude detaching the bark from the wood part and the desired debarking result of the tree trunk is achieved.
Patent FI-20125471-A (FI)
Inventor: PESONEN LAURI
IPC: B07B1/00
Filed: 2012-04-27
Abstract: The utility model provides equipment for supply powdered solid matters to a concentrate burner. The equipment comprises a screening device which is provided with a plurality of holes, wherein each hole has preset hole size, so that coarse components of which sizes are larger than the preset hole size can be screened out from the powdered solid matter flow, a screening position of the screening device is located in a channel of a powdered solid matter supply pipe device, and the screening device in the screening position is at least partially arranged in the powdered solid matter flow in the channel of the powered solid matter supply pipe device, so that the coarse components of which the sizes are larger than the preset hole size are screened out from the powered solid matter flow. According to the equipment disclosed by the utility model, the influence of the coarse components possibly existing in the powdered solid matters on the distribution of the powdered solid matters is reduced.
Patent GB-1050518-A (GB)
IPC: G05D23/19
Abstract: 1,050,518. Automatic temperature control. HITACHI SEISAKUSHO KABUSHIKI KAISHA. March 18, 1964 [March 19, 1963], No.11478/64. Heading G3R. A temperature control system for a chamber 4 comprises a main heat source 1 and a temperature sensing device 3 so arranged that that supply of current to the source 1 from a supply 5 is such as to maintain the chamber 4 at a predetermined temperature. Should however the temperature of the chamber deviate by two large a value from the desired value the value of current flowing from the supply 5 to the source 1 by way of the operating coil of a relay 7 will be sufficient to cause the relay to close its contact 8 to energize an auxiliary heat source 2 to rapidly restore the temperature of the chamber 4 to normal. In a further embodiment the main heat source comprises a thermoelectric element which either heats or cools the chamber depending on the current direction through the element and the auxiliary heat source is either a heating device or a cooling device operable by a pair of transistor operated relays.
Patent GB-1053318-A (GB)
IPC: H01F5/02
Abstract: 1,053,318. Coil formers. TELEDICTOR Ltd. Nov. 25, 1965 [Nov. 25, 1964], No. 47844/64. Heading,B8M. A coil former comprises a pair of hollow outer cover members 10a and 10b, each with enlargements 101 at their ends, and at least one intermediate member - 10c, each having oppositely disposed cavities separated by means of partition 107, and each having enlargements 102 at their ends; complementary locating devices 103 and 104 (Fig. 1, not shown) are provided on each member in order that any desired assembly of cover members and intermediate members may be built up into a compartmented former. In the preferred embodiment, the hollowed portion of each cover member is of semi-circular cross-section, and each intermediate member is of substantially H configuration in cross-section. The complementary locating devices are preferably diagonally disposed conical dowels and holes, but other means may be provided. In the preferred embodiment, two intermediate members are used, the compartments so produced housing a bar magnet 13 and two enclosures 12 for the contacts of reed relays, Fig. 4 (not shown). The assembly is held together by insulating tape prior to the winding of an electric coil, the cover members and intermediate members preferably being moulded from a synthetic plastics material.
Patent GB-1053991-A (GB)
IPC: H04Q9/06
Abstract: 1,053,991. Electric selective signalling. MANNESMANN - LEICHTBAU G.m.b.H. March 20, 1964, No. 11989/64. Heading G4H. An electrical system for transmitting a plurality of control commands utilizing two leads and an A.C. source, further comprises a doublecontact, three-position relay and a switch for selectively connecting the circuit of the relay via a rectifier in a polarity selected by the switch to energize the relay to close one of its contacts. In the particular embodiment, a mobile work platform is controlled by positioning a ganged set of eight-position rotary switches to connect one or both of two double-contact, threeposition relays across an A.C. source, each relay so connected being placed in series with one of two oppositely-poled diodes by the rotary switches to cause the relay to connect with a corresponding one of its contacts. A relay not connected in series with the A.C. source connects with neither contact. The four contacts are in the energization paths of four further relays controlling relay circuitry to energize one of seven control lines, relating respectively to down, up, forward, reverse, left, right movement and emergency stop of the platform. Either of two positions of the rotary switches produces the emergency stop, one also enabling a bell to be rung by pressing a button and the other connecting telephone line into the control cable running from the rotary switches and diodes to the three-position relays.
Patent GB-1063900-A (GB)
Abstract: 1,063,900. Calculating machines. K. DIEHL. Oct. 14, 1964 [Oct. 17, 1963 ; Oct. 26, 1963 (2); Jan. 30, 1964], No. 41825/64. Heading G4B. A four-rules calculating machine has a programme shaft 71 provided with a number of cam 207, 208, 209 &c. to control the various mechanisms and the shaft is moved stepwise by steps of 30 degrees or 60 degrees through half a revolution in one of two sequences according to whether a multiplication or a division operation is taking place. For division, the dividend is set up on a pin carriage and the " divide " key 6 is depressed. This switches on the motor and engages a onerevolution clutch through linkage described with respect to Fig. 5 (not shown). Depression of the key also lifts the end 112 of a slide 81 thus releasing a latch 108 from a fixed rail 110. The key is held depressed by a pivoted arm engaging a detent in a lever 122 pivoted to the key shank. The main shaft 27 rotates and thus pivots a rod 99 clockwise about a shaft 100 through the action of a cam 103. The slide 81 moves rearwardly following the rod 99 and a pawl 84 on the slide passes under a toothed wheel 73. As the follower 102 rises on the cam 103 again the slide is moved forwardly and the pawl 84 rotates the toothed wheel 73 through 30 degrees. The programme shaft is held in this adjusted position by a pawl (not shown) engaging a toothed wheel 131. During this cycle the dividend is fed into the totalizer and at the finish the key 6 is released, thus re-engaging the latch 108. The divisor is now set up and the result key 7 depressed. This again engages the clutch and also frees a second slide 82 in the manner described above. This slide then follows the rod 99 rearwardly and on its return movement a pawl 85 engages a toothed wheel 74 and moves the programme shaft through 60 degrees (two teeth of the wheel 74). During this cycle the divisor is fed into the register and the other function keys 5, 6 are locked so that they cannot be inadvertently depressed. During the next cycle of the main shaft the slide 82 moves the programme shaft 71 through a further 60 degrees and the remainder is printed. Finally, the slide 82 moves the shaft 71 through 30 degrees, there being one tooth missing from the toothed wheel 74, and the quotient is printed. During multiplication, the programme shaft is moved initially through 60 degrees by a third slide 80 engaging a toothed wheel 72 which has one tooth staggered by 30 degrees from that on the wheel 73. Thereafter, the programme shaft is moved twice through steps of 60 degrees by the slide 82. Thus only three steps are provided in which the multiplicand is input, the multiplier is input, and the product is printed. Tne calculating operations are also controlled by cams (not shown) on the shaft 71. The manner in which the various function keys are locked is fully described with reference to Fig. 4 (not shown). A storage result key is also provided which, when depressed, actuates the result key 7 thus starting the calculating operation as above. In this case however, the result is set into a storage register as well as being printed.
Patent GB-1074382-A (GB)
Abstract: 1,074,382. Burner control systems. HONEYWELL Inc. June 11, 1964 [June 12, 1963], No. 24324/64. Heading F4T. A fuel burner control system has a programme timer to give a purging time prior to ignition, a main burner ignition period, and a running period and is also provided with a manual switch which can only operate during the purging period to stop the timer to enable adjustments to be made to the burner system. When the START switch 27 is closed, current flows through the normally closed timer contacts T2 and contacts 2R1 through the heater 32ofthesafetyswitch,thelowerpart 30of the relay 1R, the contacts 34, 39 back to the other supply line 23. Energization of relay 1R closes contacts 1R3 to complete the circuit through contacts T9, manual switch 41 to start the timer motor and to energize the relay 3R to close contacts 3R1 which complete the circuit to the fan 13 and provide purging. The closing of contacts 1R1 by the relay 1R provides a holding circuit for this relay through the STOP switch when the START button is released. After a given time interval the timer contacts T5 are closed and the completion of a circuit through the STOP switch, previously closed contacts 1R2, closed contacts T8 energizes the ignition transformer 17 and pilot fuel valve 15 to light pilot burner 12. If a flame is established the sensor 26 operates the flame detector 20 to energize the relay 4R, thus closing the contacts 4R1 to energize the secondary flame relay 2R, thereby opening contacts 2R1 to disconnect the heater 32 in the safety switch, and closing contacts 2R3 to shunt contacts T8 and closing contacts 2R4 to open the main burner fuel valve 14. After a suitable interval timer opens contacts T5 to switch-off pilot ignition and valve. Should a pilot flame not be established the main burner will not be operated and the current through the heater 32 in the safety switch will cause the lower end of the bimetal 33 to release the pivoted switch arm 36 to open contacts 34, 39, and shut-off the pilot burner ignition system and complete the circuit through contacts 38, 35 to the alarm.
Patent GB-1143630-A (GB)
IPC: B66C17/00
Abstract: 1,143,630. Bridge cranes. VSESOJUZNY NAUCHNO - ISSLEDOVATELSK IPROEKTNO - KONSTRUKTORSKY INSTITUT PODEMNO - TRANDORTOGO MASHINOSTROENIA, POGRUZOCHNO - RASGRUZOCHNOGO I SKLADSKOGO OBORUDOVANIA I KONTEINEROV, and VSESOJUZNY NAUCHNO - ISSLEDOVATELSKY I PROEKTNOKONSTRUKTORSKY INSTITUT METALLURGICHESKOGO MASHINOSTROENIA. 28 June, 1967, No. 29745/67. Heading B8B. A bridge crane which revolves round a circular track 3, Fig. 1, has its axis 4 disposed along a chord of the circle. The bridge comprises girders 4, 5, 6, 7 supported by rollers 9-12 and guided by horizontal rollers. Motors 14, 15 drive the rollers on the track. Trolleys 16, 17 travel on a track on the beams 5, 6 and carry hoisting gear 22. Fig. 4 shows an embodiment in which a trolley track 28, 29 is at right angles to supporting girders 26, 27. The latter have end carriages with rollers supported on a monorail track 3. The trolley moves along radii of the circular track.
Patent GB-1227767-A (GB)
Inventor: MACKRLE SVATOPLUK
IPC: C02F1/52
Filed: 1968-06-13
Abstract: 1,227,767. Sewage filter. RUDNE A NERUDNE DOLY, NARODNI PODNIK. 13 June, 1968 [30 June, 1967], No. 28163/68. Heading B1D. [Also in Division C1] A suspension of sewage treated with a coagulating agent is stirred by grate 15 in homogenising space A. The homogenised suspension is fed through space B through the floating sludge blanket and clear water from space D passes to the graded multi layer filter bed F and is discharged at 8. Liquid from thickening space C can also pass to filter F via conduit 7. The enclosing vessel is spherical.
Patent GB-1229227-A (GB)
IPC: G02B13/04
Filed: 1968-11-25
Abstract: 1,229,227. Lenses. NIPPON KOGAKU K.K. Nov.25, 1968 [Nov.25, 1967], No.55872/68. Heading G2J. A wide angle camera lens of large aperture ratio and having a long back focus comprises from front to rear two negative meniscii L 1  L 2 , a lens doublet L 3  consisting of bi-convex and bi-concave lens elements cemented together, a bi-concave lens L 5  and a positive meniscus lens L 6  whose concave surface faces the object, either of lenses L 5  or L 6  being cemented lens doublets, and two positive lens elements L 7  and L 8 , the lens system satisfying the following conditions:- where f is the focal length of the whole lens system, fL 1  and fL 2  are the focal lengths of the negative meniscii L 1 , L 2 , d 2  and d 4  are respectively the air spaces between L 1  and L 2 , and L 2  and L 3 , n 3  and n 4  are the refractive indices of the lenses L 3  and L 4  and R 4  is the radius of curvature of the cemented surface therebetween. Optical data are provided for three examples.
Patent GB-1230238-A (GB)
IPC: C04B14/48
Filed: 1969-09-15
Abstract: 1,230,238. Cement compositions. GLANZSTOFF A.G. 15 Sept., 1969 [5 Oct., 1968], No. 45312/69. Heading C1H.  2À5-10% of brass coated steel fibres 0À15 mm diameter and 5-15 mm long are added to cement-sand mix.
Patent GB-1230446-A (GB)
IPC: G03C1/61
Filed: 1968-11-27
Abstract: 1,230,446. Diazotype processes and materials. KALLE AG. Nov.27, 1968 [Nov. 29, 1967], No.56274/68. Heading G2C. A diazotype process wherein a layer including a diazonium compound and a water-soluble zinc salt in a ratio of at least 2 moles of the salt per mole of the compound or a zinc chloride double salt of a diazonium compound in which case the proportion of the zinc salt may be correspondingly reduced, is imagewise exposed and developed to give a blue image in the presence of 2, 3- dihydroxyhyridine as coupler. The coupler may be in the layer or the developer. Preferred diazonium compounds are those containing alkoxy groups.
Patent GB-1232736-A (GB)
IPC: C07F9/535
Filed: 1969-10-02
Abstract: 1,232,736. Carbalkoxy-phosphoranes. R. J. REYNOLDS TOBACCO CO. 2 Oct., 1969 [24 Oct., 1968], No. 48571/69. Heading C2C. 1-Carbalkoxy-alkylidene triaryl phosphoranes are prepared by reacting in an aqueous medium an amine with a 1-carbalkoxyalkyltriarylphosphonium halide. The amine is preferably employed in at least an equimolar amount with respect to the phosphonium halide, and the reaction may be carried out at ambient or elevated temperature. Preferred products have the formula where R is C 1-18  alkyl, cycloalkyl, or substituted alkyl, R 1  is as R or may be H, and R 2 , R 3  and R 4  are aryl or substituted aryl.
Patent GB-1232781-A (GB)
IPC: B65B25/02
Filed: 1967-05-01
Abstract: 1,232,781. Bundling. HAMPSHIRE WATERCRESS Ltd. 24 July, 1968 [1 May, 1967], No. 20106/67. Heading B8C. An apparatus which forms masses of longstemmed articles, e.g. watercress, into individual bundles which are cleaned and trimmed before ejection comprises lower and optional upper conveyer belts 24, 26, Fig. 2, which compress and feed the watercress, lying across the lower belts, to a spring-biased gate 4 pivoted on a shaft (60), Fig. 4 (not shown). The force of the watercress on the gate 4 effects clockwise rotation of the shaft (60) which causes interengagement of fingers 34, 38, on transverse rows of bars 32, 40 which are indirectly pivoted upon the shaft (60), so separating a quantity of watercress between the fingers and the gate 4. The gate 4 pivots upwardly, the rotation of the shaft (60) activating a microswitch (62), Fig. 5 (not shown), which stops the drive for the belts 24. A horizontally movable carrier 42 pushes the bars 40, and hence the watercress, past a delivery table 6, Fig. 1, to a back-up plate 8 where the watercress is compressed by a pivotable baffle plate (90), Fig. 7 (not shown), whereupon a vertical pusher 10 descends to transfer the quantity of watercress into an uppermost cup 12 of a carrier 14 indexed in an anti-clockwise direction, this cup 12 having had a metal strip placed along its inside surface at the preceding station. Reciprocating dies 16 cold weld the ends of the metal strip around the cress to form a bundle. The dies 16 may be replaced by gluing or stapling means. At the next station the bundle of watercress is held in position by a clamp 18 whilst the stems are cleaned and trimmed, Figs. 11-14 (not shown). At the next station the bundles fall on to a conveyer 20 for delivery. If little or no watercress lies on the lower belts 24 then excessive anti-clockwise rotation of the gate 4 operates a second microswitch (not shown) to switch off a main drive motor but to leave the conveyer drive motor running. The amount of spring bias on the gate 4 can be altered to vary the size of bundles made.
Patent GB-1233482-A (GB)
IPC: B66F3/42
Filed: 1969-03-06
Abstract: 1,233,482. Hydraulic jacks. ARMSTRONG PATENTS CO. Ltd. 5 March, 1970 [6 March, 1969], No. 11853/69. Heading B8J. An hydraulic jack is manually operated by a lever 26 pivoted intermediate its ends at 28 to a pump piston-rod 22 and oscillated in a selected vertical plane about a reaction point formed by a ball 36 in a hole 34 in an arm 32 attached to a collar 30. The collar 30 is rotatably mounted on the pump body so that the lever 26 may be swivelled about the axis of the pump body to a convenient position.
Patent GB-1234514-A (GB)
IPC: B30B9/30
Filed: 1969-04-09
Abstract: 1,234,514. Packaging garbage. KOMPRIMATOR A.B. 9 April, 1969 [11 April, 1968; 23 Sept., 1968], No. 18268/69. Heading B8C. [Also in Division H1] A press for compressing refuse in a container (not shown) comprises a piston 19, Fig. 3, driven driven from an electric motor 10 through a chain 14 or belt drive, the increased tension in which controls a reversing switch of the motor 10 to withdraw the piston 19 when the required compression force has been reached. A pin 31 on a bell crank 26, 27 is yieldingly held against the chain 14 by spring 28 and is moved down by the chain at a preset tension whereby an arm 32 extending from arm 27 engages the switch actuator 30 to reverse the drive. Sprocket wheel 16 drives the piston-rod 17 by engagement with a chain 18 held under tension in a longitudinal groove of the piston-rod 17.
Patent GB-1250331-A (GB)
IPC: G03B21/20
Filed: 1968-10-14
Abstract: 1,250,331. Lamps. EASTMAN KODAK CO. 14 Oct., 1968 [12 Oct., 1967], No. 48540/68. Heading F4R. [Also in Divisions E2 and G2- G3] In a film projector, an ellipsoidal reflector 2 and coaxial halogen lamp 1 are formed as one unit which is accurately and detachably located in a holder 3 by engagement of the rim of the reflector with the inside face of a recess 3c in the holder, and with an abutment 3c under the action of springs 4, 5. A boss 2a on the rim diametrically opposite abutment 3e enters a recess 3d in the holder. Side extensions of the holder engage the reflector laterally. The locating means may be alternatively placed for lateral insertion of the unit into the projector.
Patent GB-1250797-A (GB)
IPC: H05B33/12
Filed: 1968-12-24
Abstract: 1,250,797. Electroluminescence. MATSUSHITA ELECTRIC INDUSTRIAL CO. Ltd. 24 Dec., 1968 [28 Dec., 1967], No. 61286/68. Heading C4S. A flexible electroluminescent display system comprises an EL layer 4, a flexible support film sheet of dielectric material 3, plate electrode 5, foraminous electrode 2 and a conductive material, e.g. a low resistance liquid such as water, or moisture, applied to and in electrical contact with a selected area of the foraminous electrode and closing the openings in such area. Letter and figure displays are specified, sheet 3 is preferably of high dielectric constant and strength and may be polyethylene terephthalate, electrode 5 may be evaporated Al or a transparent Au layer, layer 4 of green emitting ZnS: Cu or Al in a plastic binder such as urea resin, 50 Á thick, optional resin layer 1 of epoxy resin, and electrode 2 may be of 10 Á W wires spaced 100 Á, desirably a dimension greater than the spacing of electrodes 2 and 5, or a plurality of Al strips or may be reticulate e.g. a mesh or evaporated reticulate film, and layers 4 and 3 together may be 60 Á thick.