baber/WOPTO huggingface dataset:
Patent IL-152337-A0 (IL)
Title: A pyridine-1-oxide derivative, and process for its transformation into pharmaceutically effective compounds
IPC: C07B57/00
Filed: 2001-04-17
Abstract: The invention relates to N-[2-hydroxy-3-(1-piperidinyl)-propoxy]-pyridine-1-oxide-3-carboxamidine and its optically active enantiomers. (R)-(-)-N-[2-hydroxy-3-(1-piperidinyl)-propoxy]-pyridine-1-oxide-3-carboxamidine and (S)-(+)-N-[2-hydroxy-3-(1-piperidinyl)-propoxy]-pyridine-1-oxide-3-carboxamidine. Furthermore, the invention relates to the preparation of N-[2-hydroxy-3-(1-piperidinyl)-propoxy]-pyridine-1-oxide-3-carboxyimidoyl chloride, which may be used as an active ingredient of medicaments, and the preparation of the optically active enantiomers of this compound using the compounds of the invention as intermediate substances.
Patent IL-153748-A0 (IL)
Title: Processes for preparing azacycloalkanoylaminothiazole derivatives
IPC: C07D417/12
Filed: 2001-05-02
Abstract: The present invention relates to new, efficient processes for the preparation of 5-(-2-oxyazolylalkylthio)-2-azacycloalkanoylaminothiazole compounds of formula I or a pharmaceutically acceptable salt thereof, wherein: R is alkyl, aryl or heteroaryl; R<SUP>1</SUP>, R<SUP>2</SUP>, R<SUP>3</SUP>, R<SUP>4 </SUP>and R<SUP>5 </SUP>are each independently hydrogen, alkyl, aryl or heteroaryl; R<SUP>6 </SUP>and R<SUP>7 </SUP>are each independently hydrogen, alkyl, aryl, heteroaryl, halogen, hydroxy or alkoxy; R<SUP>8 </SUP>is hydrogen, alkyl, aryl, heteroaryl, CONR<SUP>9</SUP>, R<SUP>10</SUP>, COR<SUP>11 </SUP>or COOR<SUP>12</SUP>; R<SUP>9</SUP>, R<SUP>10</SUP>, R<SUP>11 </SUP>and R<SUP>12 </SUP>are each independently hydrogen, alkyl or aryl; m equals 0 to 5; and n equals 0 to 5, which are novel, potent inhibitors of cyclin dependent kinases (cdks). The present invention further concerns new key intermediate compounds, a quaternary ammonium salt of formula III' and a 2-oxazolylalkyl derivative of formula IX.
Patent IL-160468-A0 (IL)
Title: Sterile handle cover for surgical lamp
IPC: A61B19/08
Filed: 2004-02-19
Abstract: A disposable sterile handle cover uses a flexible bag, a portion of the open side of which is held snugly by a retaining ring to the inside of a conical skirt. A first set of spikes include variable length spikes protruding from the inner wall, to secure the bag against the handle. A second set of spikes protrude inwardly from the retaining ring and promote stretching and orderly application of the to the handle.
Patent IL-166103-A0 (IL)
Title: Pyrrolidine derivatives and their use
IPC: C07D403/12
Filed: 2005-01-03
Abstract: The present invention relates to novel pyrrolidine derivative of formula (I), its geometrical isomers, its optically active forms as enantiomers, diastereomers, mixtures of these and its racemate forms, as well as salts thereof, wherein R<SUP>1 </SUP>is selected from the group comprising or consisting of H and C<SUB>1</SUB>-C<SUB>6</SUB>-alkyl, for the prevention and/or treatment of preterm labor, premature birth or dysmenorrhea.
Patent IL-175748-A0 (IL)
Title: Polyamide composition comprising optical brightener, yarns made therefrom and process for heat setting such yarns
IPC: A41C3/14
Filed: 2006-05-18
Abstract: A polyamide composition, which includes an optical brightener together with either an antimicrobial agent or anti-oxidant stabilizer, or both, is suitable for making yarns, and fabrics, garments, molded articles or other articles such as carpets from these yarns. Processes for incorporating optical brighteners into polyamide compositions, polymers and yarns to make fabrics and molded articles that exhibit superior whiteness after heat-setting are also disclosed.
Patent IL-181220-A0 (IL)
Title: Floor panel and floor covering composed of such floor panels
Filed: 2007-02-08
Abstract: Floor panel consisting at least of a board-shaped element (3), whereby this floor panel (1), at least at two opposite edges (4-5), is provided with coupling parts (6-7) allowing that several of such floor panels (1) can be coupled to each other, whereby the coupling parts have contact portions forcing the floor panels (1), in the coupled condition, with a tension force (T1) at least laterally towards each other, characterized in that said coupling parts (6-7) also comprise support portions (17-18), which, in the coupled condition (8) of the respective floor panels (1), create a fixation in the mutual position of the contact portions (12-13) cooperating under tension.
Patent IL-185358-A0 (IL)
Title: Immunogens from uropathogenic escherichia coli
Filed: 2007-08-19
Abstract: Disclosed herein is a gene that can be included in immunogenic compositions specific for pathogenic  E. coli  strains. The gene is from uropathogenic strains but is absent from non-pathogenic strains, and its encoded protein has cellular locations which render it accessible to the immune system.
Patent AP-2001002122-A0 (AP)
Title: Damping arrangement.
Inventor: CLARK RICHARD ALAN
IPC: B61F5/24
Filed: 2001-04-11
Abstract: A damping arrangement for use with a three piece comprises a hydraulic damping device 20 mounted between a part of a vehicle body and a side arm 12 of the bogie, and a connector member 26 connected between the side arm 12 and support member 10 to resist lateral movement of the side arm 12 relative to the support member 10.
Patent AP-2004003065-A0 (AP)
Title: Set top box supporting cellular short message service
Inventor: BEHRENS BERNHARD AUGUST
IPC: H03M/
Filed: 2002-12-09
Abstract: A set-top box decoder arrangement (10) comprises a decoder (12) for television services (18). The decoder (12) is connectable to a monitor (21). The arrangement comprises a controller (28) for executing a short message service (SMS) application for formatting, 10 input data received from a user via remote control unit (22) into a short message. The arrangement (10) further comprises a transceiver (26) for transmitting the message to a user selectable addressee and for receiving incoming messages from a remote contact, for selective display on the monitor (21).
Patent MC-1858-A1 (MC)
IPC: A61L/
Filed: 1987-02-20
Abstract: PCT No. PCT/GB87/00125 Sec. 371 Date Sep. 7, 1988 Sec. 102(e) Date Sep. 7, 1988 PCT Filed Feb. 20, 1987 PCT Pub. No. WO87/04931 PCT Pub. Date Aug. 27, 1987.An indicator sheet for an autoclave test pack wherein a pair of porous masses (10) are held in close superimposed relationship by means of a clamp (13) with the indicator sheet (12) sandwiched between them. The indicator sheet (12) has printed thereon a pattern of markings (14) formed from one or more substances which are adapted under steam sterilizing conditions to provide an indication of the presence of air and/or excessive moisture such that each is evident and individually identifiable.
Patent MC-2190-A1 (MC)
Inventor: ALAIN BOUCHERON
IPC: G04B37/14
Filed: 1991-03-13
Abstract: PCT No. PCT/FR91/00204 Sec. 371 Date Nov. 5, 1991 Sec. 102(e) Date Nov. 5, 1991 PCT Filed Mar. 13, 1991 PCT Pub. No. WO91/14212 PCT Pub. Date Sep. 19, 1991.A bracelet watch comprises a removable flexible bracelet (2), the ends (5) of which are reinforced by an elastic tubular blade (6) or a cylindrical jaw inserted into a sleeve (7) removably fitting into a drilling (13) made in one side (1a) of the case (1) of the watch. A pawl mechanism (11, 16) is fitted for this assembly system.
Patent IE-910456-A1 (IE)
Title: Aniline derivatives of Ó-styryl carbinols as antifungal¹agents
IPC: C07D249/08
Filed: 1991-02-12
Abstract: There are provided novel aniline derivatives of alpha -styryl carbinols, pharmaceutical compositions comprising them and methods of using such compounds as antifungal agents.
Patent IE-910523-A1 (IE)
Title: Substituted urea compounds and their preparation and use
IPC: A61K31/46
Filed: 1991-02-15
Abstract: New substituted urea compounds of formula I, or a pharmaceutically acceptable salt thereof:  (* CHEMICAL STRUCTURE *) I wherein A is  (* CHEMICAL STRUCTURE *)  wherein R3 is an oxadiazol, substituted with C1-8-alkyl, C2-8-alkenyl, C2-8 alkynyl, C3-7 cycloalkyl, benzyl, phenyl, C1-6-alkoxy, C1-6-alkylthio, amino or alkylamino; R2 is -H or lower alkyl; X is O or S; and R1 is a group of formula II, III, IV or V  (* CHEMICAL STRUCTURE *) II  (* CHEMICAL STRUCTURE *) III  (* CHEMICAL STRUCTURE *) IV  where n is 2 or 3, P is 1 or 2, q is 1 to 3, r is 1-3 and R4 and R5 are H,C1-7 alkyl or C3-6 cycloalkyl; and N-oxides thereof. The compounds are useful in pharmaceutical preparations for treating psychotic disorders, nausea and vomiting.
Patent IE-910945-A1 (IE)
Title: Smoking substitute
Inventor: CARLSSON THOMMY
IPC: A61K31/715
Filed: 1991-03-21
Abstract: The invention relates to a smoking substitute containing nicotine in the form of an inclusion complex with a cyclodextrin compound. The composition also comprises excipients accepted for food or pharmaceutical use. For sublingual or buccal administration, the excipient is a directly compressible water-soluble substance, more specifically, selected from lactose, cyclodextrin, sorbitol and mannitol. A preferable composition is 0.1- 10% w/w nicotine in the form of a cyclodextrin complex, 0.05-0.3% lubricant, with the remainder excipient as above .
Patent MA-41884-A1 (MA)
Title: Système de dessalement avec compression mécanique de vapeur couplée à un système photovoltaïque
Inventor: EL KHATTABI EL MEHDI
IPC: C02F1/04
Filed: 2018-01-22
Abstract: Les trois problèmes critiquent face à la vie humaine, la crise de l’eau, l’énergie et la pollution, aussi bien qu'il existe un manque d’eau qui menace 40% de la population mondiale. Ce prototype permet d’alléger ces problématiques, c’est un mécanisme innovant reflété dans une combinaison d'unité de dessalement de l’eau de mer par la compression de vapeur mécanique (mvc) et une machine frigorifique par absorption (arm), alimentée par des collecteurs solaires photovoltaïques-thermiques (pvt). C’est un système autonome permet de fournir l'eau potable froide sans besoin de réseaux électriques ni des ressources d'énergies fossiles cette innovation présente une grande compatibilité entre les besoins de consommateurs et la source d’énergie solaire, c’est-à-dire, l’existence de grand potentiel du gisement solaire mener à l’augmentation du coefficient de performance de ce système, d’où il existe un grand besoin en matière de froid et de l’eau.
Patent MA-53520-A1 (MA)
Title: Méthode et plateforme de vidéosurveillance distribuée autonome de détection et suivi des événements en temps réel à travers des caméras intelligentes interconnectées à bas coût
Inventor: AZZAKHNINI MOHAMMED
IPC: H04N7/18
Filed: 2021-06-11
Abstract: La présente invention décrit une méthode et plateforme de vidéosurveillance distribuée autonome pour détecter et suivre les évènements qui se déroulent dans une zone surveillée par une collection dispersée de caméras intelligentes peu coûteuses et faiblement couplées. L'idée est de faire interconnecter un ensemble de caméras qui sont connectées à des systèmes de traitements dotés d’un espace de stockage qui sert de base de données locale pour chaque caméra. Cet ensemble représente notre caméra intelligente dans ce brevet. Notre méthode et plateforme proposée s’appuie sur des algorithmes de vision par ordinateur appropriés afin d’effectuer les taches de détection, de suivi et d’identification des objets en mouvements. Par la suite, chaque objet détecté sera représenté par une signature en trois dimensions qui l’identifie de manière unique. Cette signature est construite en combinant les aspects visuels de l’objet pris de différents angles de vue. De cette façon, chaque objet suivi sera reconnu par les autres caméras intelligentes et cela à partir de n’importe quel angle par lequel il a été détecté. Les différentes signatures, qui sont stockées dans la base de données locale à chaque caméra, sont utilisées pour rechercher des objets d’intérêts ou pour constituer la trajectoire complète parcourue par un objet dans la zone surveillée
Patent UY-24819-A1 (UY)
Title: Nuevos compuestos
Inventor: BROMIDGE STEVEN MARK KING FRANCIS DAVID
IPC: A61P43/00
Filed: 1997-12-18
Abstract: Nuevos derivados sulfonamidas, con actividad sobre el snc, procedimiento. Los ejemplos demuestran una estructura sulfonamida repetitiva cuyo nitrógeno está sustituido por fenilo sustituido: en posición 3 por 4. Metil piperozina y en posición 4 por metoxilo, los sustituyentes unidos al s de la sulfonamida son: benceno, benceno sustituido, benzofurano, tiofeno, isoxazol, que a su vez pueden estar sustituidos también.
Patent UY-29068-A1 (UY)
Title: Inhibidores de la arn polimerasa dependiente de arn del virus de la hepatitis c y composiciones y tratamientos que los usan
Inventor: JEWELL TANYA MICHELLE
IPC: A61K31/33
Filed: 2005-08-15
Abstract: La presente invención proporciona compuestos de fórmula (4) y sus sales farmacéuticamente aceptables y solvatos, que son útiles como inhibidores de la enzima polimerasa del virus de la Hepatitis C (HCV) y también son útiles para el tratamiento de infecciones por HCV en mamíferos infectados por HCV. La presente invención también proporciona composiciones farmacéuticas que comprenden compuestos de fórmula (4), sus sales farmacéuticamente aceptables y solvatos. Además, la presente invención proporciona compuestos intermedios y métodos útiles en la preparación de compuestos de fórmula (4).
Patent UY-31908-A1 (UY)
Title: Composiciones liquidas de limpieza ligera y métodos de elaboracion y uso de las mismas
Inventor: WISNIEWSKI KAREN
IPC: C11D1/00
Filed: 2009-06-17
Abstract: La invencion comprende composiciones líquidas de limpieza, como por ejemplo, los lavaplatos líquidos, y métodos de su elaboracion y uso, que poseen una habilidad de limpieza incrementada. Las composiciones de limpieza de la invencion incluyen composiciones líquidas de limpieza ligera de acidez liviana con baja toxicidad y eficacia anti bacterial sobre las superfiecies, como por ejemplo, superficies duras.
Patent ES-178046-A1 (ES)
Title: Un procedimiento de hacer objetos anulares de fundicion gris
IPC: B22D13/00
Filed: 1947-05-14
Abstract: Un procedimiento de hacer objetos de hierro fundido gris anulares caracterizado porque se introduce en un molde de metal no aislado hierro fundido capaz de transformarse en hierro gris en enfriamiento hacer girar el molde sobre un eje longitudinal para distribuir rápidamente al hierro en una capa delgada alrededor de la periferia del molde para la solidificación virtualmente instantánea y simultánea en todo el molde y quitar la pieza fundida del molde virtualmente en el momento en que el hierro se ha solidificado lo bastante para conservar su forma y producir al enfriarse lentamente una pieza de fundición que tiene virtualmente todo el carbono en forma de perlita y grafito.
Patent ES-178648-A1 (ES)
Title: Perfeccionamientos en la construccion de cierres para canones
Filed: 1947-06-26
Abstract: Perfeccionamientos en la construcción de cierres para cañones, que incluyen un cierre para cañón, que comprende un anillo de cierre que lleva el mecanismo de cerrojo y que está montado en un anillo de cañón para rotación excéntrica con respecto al cañón de la pieza; el anillo de cierre está dispuesto de modo tal que, por su rotación, puede abrirse y cerrarse el cerrojo; el grado de rotación activa de abertura y de cierre está limitado por medio de un fiador de retención pivotadamente montado en el anillo de cierre y preparado para apoyarse contra topes del anillo de cañón, montados respectivamente, junto a las posiciones activas completamente abierta y enteramente cerrada del cerrojo; el fiador de retención citado está preparado de modo tal que puede separarse del tope adyacente a la posición activa completamente abierta del cerrojo para que éste pueda girar interiormente y separarse del anillo de cañón.
Patent ES-180596-A1 (ES)
Title: Mejoras introducidas en la construccion de baterias del tipo de capas
Filed: 1947-11-22
Abstract: Mejoras introducidas en la construcción de baterías del tipo de capas según las cuales los electrodos negativos encajan en otro formando receptáculos para los restantes componentes de las pilas y según las cuales las partes encajadas de los electrodos negativos se separan entre sí por los bordes impermeables de una hoja porosa que forra el electrodo.
Patent ES-180722-A1 (ES)
Title: PERFECCIONAMIENTOS INTRODUCIDOS EN LOS MÉTODOS FOTOGRáFICOS DE ESTAMPACIoN
Filed: 1947-12-01
Abstract: Perfeccionamientos introducidos en los métodos fotográficos de estampación sobre cualquier clase de soporte, caracterizados por la combinación de las operaciones siguientes: a) Preparación preliminar del soporte en la región a estampar mediante una solución resinosa que lleva incorporada una sal de cadmio (por ejemplo, cloruro de cadmio en la proporción de 2 - 5%, referida al total de dicha solución); b) sensibilización local mediante la utilización de una solución de una sal fotosensible (por ejemplo, nitrato de plata); c) exposición a un foco de rayos actínicos; d) viraje y fijado combinados, en un baño único que además del ingrediente fijador usual contiene cloruro de oro y nitrato de plata; e) lavado y secado finales.
Patent ES-264384-A1 (ES)
Title: A method for removing stresses in cables made from synthetic, linear polyamides, and cables thus treated
IPC: H01B3/30
Filed: 1961-01-27
Abstract: Stresses in cables made from synthetic linear polyamides are removed by treating the cables with hot, acid-free mineral oil. The temperature of treatment is preferably between 100 DEG C. and 10 DEG C. below the melting-point of the polyamide from which the cable is made. The oil may contain an antioxidant. The treatment may be applied in a continuous or a discontinuous manner to cable which may be relaxed or under tension. In an example, a cable of poly-S -caprolactam is treated with Tellus No. 41 oil at 140 DEG C. The tensile strength after treatment is compared with that of similar cable treated with hot water. The treated cable contains 12% by weight of oil.ALSO:Stresses in cables made from synthetic linear polyamides are removed by treating the cables with hot, acid-free mineral oil. The temperature of treatment is preferably between 100 DEG C. and 10 DEG C. below the melting-point of the polyamide from which the cable is made. The oil may contain an anti-oxidant. The treatment may be applied in a discontinuous or a continuous manner to cable which may be relaxed or under tension. In an example, a cable of poly-e -caprolactum, is treated with Tellus No. 41 oil at 140 DEG C. The tensile strength after treatment is compared with that of similar cable treated with hot water. The oil-treated cable contains 12% by weight of oil.
Patent ES-264827-A1 (ES)
Title: Novel sulphonamides and a process for the manufacture thereof
IPC: C07D239/42
Filed: 1961-02-11
Abstract: The invention comprises 4-sulphanilamido-6-halogeno-pyrimidines such as 4-sulphanilamido-6-chloro-pyrimidine, and salts thereof and comprises also the preparation of these compounds by reacting a 4,6-dihalo-pyrimidine, e.g. 4,6-dichloro-, dibromo- or diiodopyrimidine, with the sodium salt of sulphanilamide. Pharmaceutical preparations having antibacterial activity comprise the above compounds of the invention in association with an organic or inorganic, solid or liquid carrier suitable for enteral or parenteral administration. The preparations suitably take the form of tablets, dragees, suppositories, capsules, solutions, emulsions or suspensions and may contain emulsifying, preserving, stabilizing or wetting agents, salts for varying the osmolic pressure or buffers, and other therapeutically useful substances.
Patent ES-274100-A1 (ES)
Title: Improvements relating to brewing
IPC: C12C3/04
Filed: 1962-01-27
Abstract: In treating hops to improve their brewing qualities, e.g immediately before they are added to a mash, loose hops are introduced, in the presence of an ordinary atmosphere, into a gas-tight vessel, which is then evacuated, by suction, to a reduced pressure between 15 and 5, e.g. 10, mm. of mercury, maintained for 15 to 60 minutes by introducing pure air or a neutral gas, such as carbon dioxide, into the vessel whilst the remaining ordinary atmosphere and unwanted odours and vapours are sucked out. The hops may be ground before being treated. The air-tight vessel may be connected to the source of pure air or neutral gas through a valve, which is set to open when the desired reduced pressure is reached, and remain open for as long as that pressure is maintained.
Patent ES-307739-A1 (ES)
Title: Control circuits for electric motors
IPC: H02P1/44
Filed: 1964-12-31
Abstract: A single-phase induction motor drive the compressor of a refrigerator and has main and auxiliary stator windings 58a, 58b. The auxiliary winding poles are at 45 degrees with the main winding poles, the auxiliary windings having the higher impedance. Initially, both stator windings are energized directly through contacts 106, 108. After a short period, however, resistance-wire 100 expands to break contact 108 whereby capacitor 110 is connected in series with winding 58b. If there is an overload, contact 106 opens to disconnect the motor. A timer motor 90 periodically opens contact 92a to de-energize fan motor 96 and the compressor motor, and energize heating-coil 95 associated with the evaporator. The operation of the heating-coil continues until defrost thermostat 97 opens the circuit. Afterwards, the timer motor restores the circuit to its initial condition. The fan motor 96 circulates air over the evaporator provided that the timer contacts 92a are closed, the refrigerator door is closed, and the cabinet-temperature is not too low. The compressor motor has a fan with radial flow vanes which are cast as part of the rotor, and axial flow vanes which are formed from a sheet metal disc attached to the ends of the radial flow vanes.
Patent ES-333486-A1 (ES)
Title: Novel urea derivatives and their production
IPC: C07D493/08
Filed: 1966-11-17
Abstract: Novel compounds of Formula I wherein X represents a methylene, ethylene' imino or C 1-2 alkylimino or alkanoylimino group, or oxygen, Y represents oxygen or sulphur, R 1 , R 2 and R5 represent hydrogen or a C 1-4 alkyl group, R 3 and R 4 represent hydrogen, halogen up to the atomic number 35, trifluoromethyl, or C 1-4 low alkyl or alkoxy or C 1-2 alkanoyl groups, and n represents 0 or 1, are prepared (1) by reacting an amine of Formula II wherein X1 has the meaning given for X above with the exception of the imino group, with a suitable phenyl isocyanate or isothiocyanate or with a reactive functional derivative of a suitable carbanilic acid or thiocarbanilic acid, and, if desired, splitting off any low alkanoyl radical in X1 by hydrolysis, (2) by reacting an isocyanate or isothiocyanate of Formula VI or a reactive functional derivative of a carbamic acid or thiocarbamic acid of Formula VII with a suitable aniline, and, if desired, splitting off any low alkanoyl radical in X1 by hydrolysis, (3) by reacting a compound of Formula VIII with a compound of formula H 2 Y, and, if desired, splitting off any low alkanoyl radical in X1 by hydrolysis, or (4) by converting a thiourea obtained as described above into the corresponding urea. 2-Oxa - adamantane - 1 - amine may be prepared by reacting bicyclo[3,3,1]nonan-3,7-dione with benzylamine, reducing the 3-benzylamino- 2 - oxaadamantan - 1 - ol obtained with lithium aluminium hydride, and debenzylating the N - benzyl - 2 - oxaadamantane - 1 - amine thus formed. 1 - (1 - Adamantyl) - 3 - (3,4 - dichlorophenyl)- carbodiimide may be obtained by treating 1-(1- adamantyl) - 3 - (3,4 - dichlorophenyl) - thiourea with anhydrous magnesium sulphate and lead oxide. Therapeutic compositions having anti-bacterial activity, which may be administered locally, parenterally or orally, contain as active ingredient a compound of Formula I above.