baber/WOPTO huggingface dataset:
Patent CZ-286753-B6 (CZ)
Title: Derivative of piperidine-4-carboxylic acid, pharmaceutical preparation containing thereof, process of its preparation and use
Inventor: ASK ANNA-LENA
IPC: C07D211/32
Filed: 1995-02-03
Abstract: In the present invention there are described derivatives of piperidine-4-carboxylic acid of the general formula A, in which Z represents the group of the general formula (i) or a carbonyl group, Ri1 represents hydrogen or Ri2, Ri2 represents an alkyl group containing 1 to 3 carbon atoms or Ri1 and Ri2 together form a chain {-(CHi2)in-}, wherein n is3, 4 or 5 or a chain {-(CHi2)O(CHi2)i2-}, m is 0 or 1, p is 1 or 2, Ri3 represents hydrogen or {-COCHi3} and Ri4 represents hydrogen, {-CHi3}, {-OH} or {-OCHi3} with the proviso that when Z represents the carbonyl group then p is 2, further pharmaceutically acceptable salts of those derivatives, several processes of their preparation as well as their use for preparing pharmaceutical preparations. The invented derivatives exhibit both local anaesthetic and analgesic activities.
Patent CZ-282334-B6 (CZ)
Title: High-production strain of penicillium chrysogenum ccm 8196 micro-organism
Inventor: BUCKO MICHAL ING DRSC
IPC: C12R1/82
Filed: 1995-09-18
Abstract: A high-production strain of the microorganism Penicillium chrysogenum CCM 8196 (NMG FOK 15). The strain was obtained by selecting mutants produced by exposure of the spores to chemical mutagens and an increased concentration of phenylacetic acid during submerged cultivation. The  subsequent passive selection resulted in the strain of Penicillium chrysogenum CCM 8196 (NMG FOK 15) producing more than 35,000 IU PEN G/ml in168 hours of cultivation in aerated flasks at 25 degrees C.
Patent CZ-295205-B6 (CZ)
Title: Boronizing preparation
Inventor: BAUDIS ULRICH DR
IPC: C23C8/70
Filed: 1999-07-08
Abstract: In the present invention, there is disclosed a boronizing agent in the form of a paste for the production of boride layers on metallic components. The boronizing agent contains boron-releasing substances, activating substances and inert, refractory extenders together with water and optionally auxiliaries required for paste formulation. It contains a combination of 1 to 5 percent by weight of potassium tetrafluoroborate and 5 to 40 percent by weight of calcium fluoride, in each case relative to the boronizing agent total weight, as the activating substance. Using this boronizing agent, single-phase Fei2B-containing boride layers on iron material-based components can be produced.
Patent CZ-295568-B6 (CZ)
Title: Process for preparing cyclodextrin
Inventor: GRULL DIETMAR DR
IPC: C12P19/04
Filed: 1999-08-11
Abstract: In the present invention, there is disclosed a process for preparing cyclodextrin from amylopectin potato starch by treating thereof with cyclodextrin glycosyl transferase wherein the preparation process is characterized in that amylopectin potato starch is used as a starting starch material. Said amylopectin potato starch is obtained from potatoes being inhibited with respect to formation of amylose by breeding or genetic, optionally another molecular-biology process. This starting starch material associates positive effects of a natural amylopectin starch with these of potato starch, and exhibits among other a low content of lipids and proteins, thus higher purity.
Patent CZ-288393-B6 (CZ)
Title: Use of phenyl substituted 1,4-dihydropyridines for preparing medicaments, phenyl substituted 1,4-dihydropyridines per se, and process of their preparation as well as medicaments in which said substances are comprised
Inventor: MEIER HEINRICH DR
IPC: A61K31/44
Filed: 1994-12-09
Abstract: The present invention relates to the use of phenyl substituted 1,4-dihydropyridines of the general formula I, in which the substituents have specific meanings, further novel phenyl substituted 1,4-dihydropyridines per se and process of their preparation by reacting halophenyl-aldehydes with {beta}-keto esters, optionally under isolation of ylidene compounds and with enamines as well as medicaments in which these substances are comprised, particularly cerebrally active preparations.
Patent CZ-287637-B6 (CZ)
Title: Process and apparatus for attaching half-finished products of glass articles
Inventor: DAEA BRUNO ING
IPC: B24B41/00
Filed: 1999-10-06
Abstract: The invented Process for attaching half-finished products of glass articles is carried out in such a manner that the half-finished product is put in a bed (2) of a clamping device that is filled under normal temperature with a liquid clamping substance. After the half-finished product (3) is positioned the clamping substance is cooled down to temperature being lower than melting point thereof. After cooling of the clamping substance the half-finished products (3) are machined by grinding or polishing at continuous removal of heat. Release of the half-finished products (3) after machining is made by warming up the clamping substance. The apparatus for making the above-described process is provided with a plate (1) of good thermal conductivity. In this plate (1) there is performed a bed (2) being negative relief of a half-finished product (3). The plate (1) is provided on both its sides with heat insulation (4) and a system of internal channels (5). In order to enable positioning of the half-finished product (3) during machining there is mounted by means of a joint (8) in a supporting plate (6) a clamp (7) whose end part (9) is provided with the bed (2) and encircled by a pipe (11) with flexible supply (12) and discharge (13) of a heat-carrying medium.
Patent CZ-286083-B6 (CZ)
Title: Machining center
Inventor: GRUENER MAGNUS
IPC: B23Q7/14
Filed: 1995-06-20
Abstract: A gripping mechanism is formed by a clamping mechanism (25) and a workpiece (26) driver (15) is arranged together with the clamping mechanism in exchangeable manner on a positioning mechanism (16), whereby place (37) of workpiece (26) preparation is identical with the workpiece (26) stowing place (37). A workpiece (26) transport mechanism (45, 45') serves for feeding and/or withdrawal of workpieces (26) to be machined or already machined workpieces (26) into, optionally from a workpiece (26) exchange station (35), whereby the workpiece (26) driver (15) is provided with a faceplate (47) on the bottom side (48) of which there is arranged the clamping mechanism (25).
Patent CZ-298637-B6 (CZ)
Title: Rotary drum supporting device
Inventor: METTAVANT PIERRE
IPC: F26B11/02
Filed: 1998-04-14
Abstract: The present invention concerns support device (1) for a cylindrical drum (2) intended particularly for ovens, driers, cooling plants or the like devices, designed for thermal and/or chemical treatment of materials, wherein the support device (1) comprises at least a track roller (3), co-operating with said cylindrical rotary drum (2), and at least two bearings (5, 5') for enabling said roller (3) to rotate about its rotation axis (4). The invention is characterized in that the device further comprises: a frame (7), whereto said bearings (5, 5') are secured, mounted articulated about a pivoting axis (11) substantially perpendicular to the plane passing through said roller (3) rotation axis (4) and perpendicular to a block (6) on which said device (1) is placed, called articulating plane; linking means (8), flexible along a predetermined direction (9, 9'), called flexibility direction, and rigid in the directions orthogonal to said flexibility direction (9, 9'), to maintain said bearings (5, 5') on said block (6) while allowing the frame (7) to move freely in articulation, such that the roller (3) is aligned with the drum (2) when the latter is pivoting.
Patent CZ-305018-B6 (CZ)
Title: Waste aluminium recycling process and apparatus for making the same
Inventor: Trávníček Ivan
IPC: C22B7/00
Filed: 2013-09-30
Abstract: In the present invention, there is disclosed a process for recycling waste aluminium wherein the process is characterized in that waste aluminium is crushed to small particles, the particles are cleaned from pollutants by chemical process and then they are dissolved in sulfuric acid. During this process, hydrogen is liberated and aluminium sulfate produced. The invention also discloses apparatus for making the above-described process, which apparatus comprises waste aluminium preparation room, a reactor for carrying out dissolution of the waste aluminium, a gas circuit for distribution of hydrogen and withdrawal of odors, a water circuit for the distribution of new water or treatment of used water, a thermal circuit for the production and distribution of heat, and a chemicals preparation room for the preparation and separation of chemicals.
Patent CZ-305540-B6 (CZ)
Title: Heat treatment process of high-alloy steel
Inventor: Mašek Bohuslav
IPC: C22C38/00
Filed: 2014-05-21
Abstract: The present invention relates to a process for heat treatment of high-alloy steel having the resulting structure of undissolved metal carbides in the form of globulitic particles, austenitic and martensitic structure. The heat treatment process consists in heating a metal blank to a temperature in the range of 1270 to 1280 degC, at a heating rate within the range of 40 to 45 degC/s. Subsequently the metal blank is subjected to pressure in thixotropic process and then it is let to cool down to ambient temperature.
Patent CZ-306937-B6 (CZ)
Title: A method of producing a venting insert
Inventor: ROZKOŠNÝ LUBOŠ
IPC: B22D17/20
Filed: 2015-10-05
Abstract: It is described a vent plug for molds , especially molds for cast of metals under pressure, which is formed by body ( 7 ) with a part ( 1 ) to take out of the heat and a flow part ( 2 ) which is provided with flow path ( 5 ) , the which follows from the vent channel formed by shaped space ( 4 ) . The part ( 1 ) is preferably formed from a copper or its alloys and the flow part ( 2 ) is made of a metal with a higher hardness than is the part ( 1 ) , and is usually made of tool steel. The flow part ( 2 ) is on the part ( 1 ) to take out the heat applied by 3D printing.
Patent CZ-307796-B6 (CZ)
Title: Arylbenzothiazolylurea derivatives, preparing and using them
Inventor: Musílek Kamil
IPC: C07D277/82
Filed: 2018-03-27
Abstract: The invention provides new general formula I arylbenzothiazolylurea derivatives and pharmaceutically acceptable alkali metal salts, ammonia or their amines, or acid addition salts where Ris selected from -COOH, -COO (C 1 -C 4 alkyl), -CONH, -CONH (C 1 -C 4 alkyl), -CON (C 1 -C 4 alkyl), -NH, -NH (C 1 -C 4 alkyl), -N (C 1 -C 4 alkyl), -NHCO (C 1 -C 4 alkyl), -N (C 1 -C 2 alkyl) CO (C 1 -C 4 alkyl). These new aryl benzothiazolyl urea derivatives are inhibitors of betaamyloid alcohol dehydrogenase (ABAD) enzymatic activity. The invention also includes a method of preparing them and their therapeutic use in treating Alzheimer's disease and / or dementia.
Patent CZ-308897-B6 (CZ)
Title: Process for preparing submicron and / or micron crystalline tungsten oxide tubes, and submicron and / or micron crystalline tungsten oxide tubes prepared in this way
Inventor: Macák Jan
IPC: C01G41/02
Filed: 2020-11-03
Abstract: Process for preparing submicron and / or micron crystalline tungsten oxide tubes with an outer diameter of 400 to 1,600 nm consists of preparing an aqueous or aqueous-ethanol precursor solution which contains 5 to 25% by weight of ammonium metatungstate as a precursor of WO3 and 5 to 25 by weight of polyvinylpyrrolidone polymer with a molar mass of 40,000 to 1,300,000 g / mol, polyvinyl alcohol with a molar mass of 31,000 to 19,000 g / mol, polyethylene glycol with a molar mass of 200,000 to 1,000,000 g / mol, or mixtures of at least two of them, the weight ratio of ammonium metatungstate and the polymer / polymer mixture is 1:5 to 2:1. This precursor solution is then converted by centrifugal spinning into precursor submicron and / or micron fibres, which are then calcined for 4 to 13 hours at 300 to 500 °C, gradually burning the organic material and initiating WO3 crystallization on the outer surface of the precursor fibres, towards the centre of the precursor fibres. This produces a volume contraction of the material inside the fibres which, together with the escape of gases which are formed during the combustion of the organic part of the precursor fibre, forms a hollow structure of the final micron and / or submicron WO3 tubes.The solution also relates to submicron and / or micron crystalline tungsten oxide tubes prepared in this way.
Patent CZ-302157-B6 (CZ)
Title: Coated tablet with cyclophosphamide, process for preparing thereof and process for preparing tablet core
Inventor: ENGEL JUERGEN
IPC: A61P35/00
Filed: 1999-06-08
Abstract: In the present invention, there is disclosed a coated tablet, which contains cyclophosphamide as an active substance, one or more fillers being selected from the group consisting of lactose monohydrate, D-mannitol and calcium monohydrogen orthophosphate, one or more dry binders being selected from the group consisting of non pre-swollen cornstarch and microfine cellulose, highly disperse silica as a flow regulator, and a lubricant being selected from the group consisting of magnesium stearate, stearic acid, glycerol palmitostearate, polyethylene glycol, talc and glycerol monobeherate, whereas the core can contain adjuvants either individually or alternatively in any desired mixture. There is also disclosed a process for preparing the above-described tablet core by sieving and homogenization of all ingredients excluding magnesium stearate, adding and mixing magnesium stearate and pressing the tablet core mixture. Further disclosed is a process for preparing the coated tablet by spraying said core with suspension prepared by dissolving 11.83 g of polyethylene glycol and 2.37 g of polysorbate 80 in water, further by dissolving 1.9 g of carboxymethylcellulose sodium in 80.0 g of water, proceeded further with bringing both solutions together, adding 23.67 g of talc, 23.67 g of titanium dioxide and 0.24 g of simethicone, homogenization and then adding 17.73 g of a 30% strength ethyl acrylate/methyl methacrylate copolymer dispersion.
Patent CZ-296359-B6 (CZ)
Title: L-arabino-disaccharides of anthracyclines, processes for their preparation, and pharmaceutical mixtures containing them
Inventor: ANIMATI FABIO
IPC: C07H15/252
Filed: 2000-03-08
Abstract: In the present invention, there are disclosed compounds of the general formula I, pharmaceutically acceptable salts thereof, processes of their preparation and pharmaceutical mixtures in which these compounds are comprised. The compounds according to the present invention exhibit anticancer activity.
Patent CZ-301257-B6 (CZ)
Title: Metal billet for use in hot dilation forming, bottomed container manufactured from this metal billet, radioactive substance container comprising the bottomed container, apparatus for producing the bottomed container, process for producing the bottome
Inventor: FUNAKOSHI YOSHIHIKO
IPC: G21F5/008
Filed: 2001-03-26
Abstract: In the present invention, there is disclosed a metal billet (200) serving as a blank for the manufacture of a bottomed container (1) forming a part of a radioactive substance container (100) of a cylinder, to be used for hot dilation forming, wherein said metal billet (200) has a backward side (200b) with respect to the pressing direction, said backward side (200a) having rear cross section perpendicular to the metal billet (200) longitudinal direction, wherein said metal billet (200) has a forward side (200b) with respect to the pressing direction, said forward side (200b) having front cross section perpendicular to the metal billet (200) longitudinal direction, wherein the invention is characterized in that said rear cross section comprises the projection of said front cross section. There is also disclosed a bottomed container (1) produced by hot dilating from a metal billet (200), a radioactive substance container (100) comprising the bottomed container (1), an apparatus for producing the bottomed container (1), a process for producing the bottomed container (1) from the metal billet (200) by hot dilating inside c container (300) for forming using a die (410).
Patent CZ-302265-B6 (CZ)
Title: Control of glass forming I. S. machine with respect to feasible schedule in an unwrapped bottle forming process
Inventor: SIMON JONATHAN S
IPC: C03B9/41
Filed: 2002-04-05
Abstract: A control for defining data for setting the times for controlled events in a glass forming machine which is controlled by a programmable sequencer which defines the time of a machine cycle. A computerized model of a mathematical representation of a network constraint diagram of the unwrapped bottle forming process is provided with computer analysis for analyzing the computerized model as a constrained optimization problem for determining, with inputs including the following:; 1. the motion durations of each of the mechanisms from the retracted position to the advanced position and from the advanced position to the retracted position, 2. the submotion durations of the mechanisms, 3. the machine cycle time, and 4. the time in an unwrapped bottle forming process for each displacement to begin and for each valve to be turned "on" and "off", and 5. the target time for an optimized machine cycle, the machine cycle time and the event times for an optimized process wherein an alternate machine cycle time for a feasible schedule in an unwrapped bottle forming process and the event time in the feasible schedule for each displacement to begin and for each valve to be turned "on" and "off" can be used for establishing a control instruction for efficient production process of the glass forming I. S. machine.
Patent SK-285865-B6 (SK)
Title: Pharmaceutical formulation with masked taste and method for the production thereof
Inventor: BECOURT PHILIPPE
IPC: A61K31/00
Filed: 2002-06-21
Abstract: A pharmaceutical formulation with masked taste, the masking of which persists during the administration of the formulation, especially in the form of a suspension in aqueous vehicle, contains at least a cellulose-based polymer that is soluble in organic solvents but virtually insoluble in water irrespective of the pH, a methacrylic polymer that is soluble in acidic medium and virtually insoluble at neutral or alkaline pH, an active principle uniformly distributed and in molecular form in the mixture, which is in the form of an atomized matrix, a basic agent of organic nature or a basic salt which are pharmaceutically acceptable and an adsorbent. A method for the production of the pharmaceutical formulation is also described and a method for masking the taste of pharmaceutical products.
Patent DE-10124336-B8 (DE)
Inventor: DINGERT UWE
IPC: A47L1/08
Filed: 2001-05-18
Granted: 2009-07-09
Abstract: The bearer (1) forms a latent heat storage with fitted temperature sensor made of plastics with inbuilt thermochrome material so plastics casing acts as cleaning fluid tank. Part of the tank wall forms a heat guide, being here of reduced thickness and reinforcibly ribbed. The bearer is made of polymer material and fitted with a handle (2) hinged to the bearer base through a universal joint (6) in the center of the bearer top. The wiper (3) is a removable fleece, knitted etc or woven cloth and is fastened to the bearer. The tank has a stoppable opening for the cleaning fluid to be pumped out.
Patent EP-1183390-B8 (EP)
Inventor: O'CONNOR JOHN
IPC: C12N15/02
Filed: 2000-05-12
Granted: 2006-05-03
Abstract: The present invention provides a method of predicting pregnancy outcome in a subject by determining the amount of an early pregnancy associated molecular isoform of hCG in a sample. The present invention further provides a method for determining the amount of early pregnancy associated molecular isoforms of human chorionic gonadotropin (hCG) in a sample. The present invention also provides a diagnostic kit for determining the amount of early pregnancy associated hCG in a sample. The present invention additionally provides an antibody which specifically binds to an early pregnancy associated molecular isoform of human chorionic gonadotropin. Finally, the present invention provides methods for detecting trophoblast or non-trophoblast malignancy in a sample.
Patent EP-1268347-B8 (EP)
Inventor: GONZALEZ JOSE
IPC: C07C209/68
Filed: 2001-04-05
Granted: 2005-09-21
Abstract: A novel complex salt off palladium sulfate and ethylenediamine contains 31 to 41% by weight of palladium and has a molar ratio [SO4]:[Pd] of between 0.9 and 1.15 and a ratio [ethylenediamine ]:[Pd] of between 0.8 and 1.2. The invention further relates to a process for the preparation of this complex salt, and to the use of this complex salt for introducing palladium into an aqueous electrolysis bath of acidic pH for the electrochemical deposition of palladium or one of its alloys, or for adjusting the palladium concentration of such a bath.
Patent EP-1546545-B8 (EP)
Inventor: KRONBERGER MAXIMILIAN
IPC: F02M59/44
Filed: 2003-09-12
Granted: 2007-08-01
Abstract: The invention relates to a pump/nozzle unit for delivering fuel (10) into a combustion chamber (12) of an internal combustion engine, comprising a fuel pump (14-22), which can be controlled and/or regulated and which has a control valve (22) with a valve needle (48) that is displaced by a piezo actuator (76). The comparatively short travel of the piezo actuator (76) is increased by a mechanical multiplication device (56, 58) to the extent necessary for displacing the valve needle (48). In order to avoid jeopardizing the pressure resistance of the control valve housing while yet providing the comparatively wear-resistant contact areas (80, 82) coming into contact with the mechanical multiplication device (56, 58), the invention provides that the control valve housing is made of a material having a comparatively lower basic hardness, for example, Ovako 677, and the contact areas (80, 82) of the control valve (22) are subsequently hardened by laser.
Patent EP-2129821-B8 (EP)
Inventor: MUENSTERMANN ULLRICH
IPC: D04H1/46
Filed: 2008-02-21
Granted: 2012-02-29
Abstract: The invention relates to a device for processing nonwoven fabrics made of fibers and/or filaments, or other web material, comprising a hollow distributor device (2) having a plurality of nozzle openings (2.2), wherein a gaseous medium can be applied to the nonwoven fabric or web material by means of the distributor device. According to the invention, the nozzle openings (2.2) are located in a housing wall (2.1) of a distributor device (2), said housing wall facing the nonwoven fabric or web material.
Patent BR-PI0514831-B8 (BR)
Title: assento de veículo automotivo
Inventor: AUMOND JEAN CLAUDE
IPC: B60N2/30
Filed: 2005-07-20
Abstract: assento de veículo automotivo. o assento de veículo automotivo compreende o encosto do assento (3), o assento em si (2), conectado ao encosto (3) por uma conexão com pivô (p1) e ao assoalho do veículo por um suporte frontal (p2). o inventivo assento acondicionável também compreende um braço móvel (7) conectado ao encosto e ao assoalho por duas juntas-pivô (p4, p5), tornando o assento móvel entre uma condição de estendido, na qual o assento em si (2) está substancialmente paralelo ao assoalho, o encosto (3) está em posição substancialmente vertical e cada braço móvel (7) está posicionado na extensão do encosto (3), possibilitando assim que possa ser movido para cima, e uma condição de recolhido quando o encosto (3) está inclinado por sobre o assento (2) durante a transição entres as condições de recolhido para estendido, cada pivô de braço móvel (7) está em uma direção oposta á direção do pivô do encosto (2), de modo que fica posicionado ao longo do mesmo.