baber/WOPTO huggingface dataset:
Patent ZA-911980-B (ZA)
Title: Tenidap as an inhibitor of the release of elastage by neutrophils
Inventor: LOOSE LELAND DAVID
IPC: C07D409/06
Filed: 1991-03-18
Abstract: This invention relates to the use of tenidap, 5-chloro-2,3-dihydro-2-oxo-3-(2-thienylcarbonyl)-indole-1-carboxamide, and the pharmaceutically-acceptable base salts thereof to inhibit the release of elastase by neutrophils in a mammal. This invention also relates to the use of tenidap and its salts for treating elastase-mediated diseases and dysfunctions such as arteritis, proteinuria and pulmonary emphysema in mammals. The methods of this invention comprise administering an effective amount of tenidap or salts thereof to a mammal.
Patent ZA-926618-B (ZA)
Title: Process for the drying and granulation of aspartame.
Inventor: SLANGEN HUBERTUS JOZEF MARIA
IPC: B01J2/16
Filed: 1992-09-01
Abstract: The invention relates to a process for the drying and granulation of aspartame through the thermal treatment of a wet mass of aspartame crystals using a hot carrier gas, characterised in that a wet mass of aspartame crystals is supplied, in a continuous process, to a high-speed paddle dryer fitted with a jacket heated to a temperature of 80-190 DEG C and with paddles, mounted on a central shaft with a controllable speed of rotation, at an adjustable distance from and angle to the jacket, which are positioned so that the required particle size of the granules is realized, the speed of rotation being chosen so that the Froude number is higher than 1, and the supplied product is treated in the paddle dryer for 15-600 seconds, with the simultaneous presence of a carrier gas having an inlet temperature of 100-200 DEG C, and the granular product obtained is discharged from the paddle dryer and, if necessary, dried further - in a manner known per se - in one or more drying steps in other drying equipment. With the use of high-speed paddle dryer aspartame with good microbiological properties is very easily obtained. <IMAGE>
Patent ZA-928513-B (ZA)
Title: Articulated structures for dolls or puppet bodies.
Inventor: RODRIGUEZ FERRE JOSE MANUEL
IPC: A63H33/10
Filed: 1992-11-04
Abstract: The articulated structure for dolls or puppet bodies of the invention consists of a structure or skeleton-like framework in which the various elements and members which comprise it are connected with one another at their ends by means of link connections (8,9) which in combination with the structure of the referenced ends constitute ball and socket articulations. The link connections are formed by two spheres 8a connected by a radial appendix 8b, over which is injected the integrating material making up the semispherical catches 9, constructed in the ends of the elements or members of the skeleton-like framework. The improvements are applicable in the manfuacture of articulated structures for dolls which permit stable and voluntary positioning of their members or connecting parts. <IMAGE>
Patent ZA-933900-B (ZA)
Title: Lining for a block-shaped container and transport pack for said lining
Inventor: GIEZEN MAURICE GERARDUS MARIA
IPC: B65D77/06
Filed: 1993-06-03
Abstract: A lining (1) for a block-shaped container, which lining is made of flexible material and can be placed folded in the container, and can then be brought to the desired shape in the container through filling. The lining is folded up or rolled up to the form of an elongated strip, which can be placed in the container in a position in which it extends with its lengthwise direction at least between the top edge and the bottom wall thereof, in such a way that during filling the lining can unfold relative to said lengthwise direction towards the two opposite sides.
Patent ZA-938574-B (ZA)
Title: Substituted amidino compounds their manufacture and methods of treatment
Inventor: MORISSEY MICHAEL MARTIN
IPC: C07C271/64
Filed: 1993-11-17
Abstract: PCT No. PCT/US93/10876 Sec. 371 Date Jul. 25, 1995 Sec. 102(e) Date Jul. 25, 1995 PCT Filed Nov. 12, 1993 PCT Pub. No. WO94/11341 PCT Pub. Date May 26, 1994   <IMAGE>  (I)  The invention relates to the compounds of formula (I) wherein the C(=NH)-NHR3 group may be in tautomeric or isomeric form, and pharmaceutically acceptable salts thereof, in which: R1 is amino which is mono- or disubstituted by a substituent selected from an aliphatic hydrocarbon radical, an araliphatic hydrocarbon radical, an aromatic radical, and a cycloaliphatic hydrocarbon radical or is amino which is disubstituted by a divalent aliphatic hydrocarbon radical or a said radical interrupted by oxygen; R2 is hydroxy which is etherified by an aliphatic alcohol which is substituted by carboxy, by esterified carboxy or by amidated carboxy; R3 is hydrogen or an acyl radical which is derived from an organic carbonic acid, an organic carboxylic acid, a sulfonic acid, or a carbamic acid; X1 and X3, independently of one another, are oxygen (-O-) or sulphur (-S-); and X2 is a divalent aliphatic hydrocarbon radical which may be interrupted by an aromatic radical. The compounds are useful as selective LTB4 receptor antagonists in the treatment of conditions or syndromes in mammals which are responsive to LTB4 receptor antagonism.
Patent ZA-942728-B (ZA)
Title: Substituted phenoxyisobutryric acids and esters
Inventor: REGNIER GILBERT
IPC: C07C59/90
Filed: 1994-04-20
Abstract: The substituted phenoxyisobutyric acids and their esters of formula I: <IMAGE>  in which:     - X represents an oxygen atom, a sulphur atom or a single bond; - A represents a single bond or a hydrocarbon radical containing from 1 to 9 carbon atoms in a straight or branched chain optionally containing a double bond, a cyclopropyl radical, an oxygen atom or a carbonyl radical, or optionally substituted by a halogen atom or a hydroxyl radical; - R represents a hydrogen atom or an alkyl radical containing from 1 to 6 carbon atoms in a straight or branched chain optionally substituted by one or two hydroxyl radicals;   - R1 and R3:     . each simultaneously represent a hydrogen atom, or . together form a bridge (CH2)n in which n takes the values 1 or 2, or   . R1 represents:     . a methyl radical, or . a single bond which forms a double bond with the group A when the latter is a hydrocarbon radical, and   . in each of these cases, R3 simultaneously represents a hydrogen atom;   - R2 and R6, which are identical or different, each represent a hydrogen atom or a methyl radical; - R4 and R5, which are identical or different, each represent an alkyl radical containing from 1 to 6 carbon atoms in a straight or branched chain; - R7 represents a hydrogen atom or a labile protective group such as, for example, a CH3CO-, C2H5O-CH2- or benzyl radical; and - Z represents a hydrogen or halogen atom or an alkyl or alkoxy radical each containing from 1 to 5 carbon atoms in a straight or branched chain; and, when they exist, the corresponding enantiomers and diastereoisomers, as well as the physiologically tolerable salts of the compounds I with appropriate bases, can be used in therapeutics.d
Patent ZA-944933-B (ZA)
Title: A novel compound form
Inventor: KAELLSTROEM LARS AEKE
IPC: A61K/
Filed: 1994-07-07
Abstract: A novel compound form of magnesium omeprazole, i.e. with a degree of crystallinity which is higher than 70% as determined by x-ray powder diffraction, useful in the manufacture of pharmaceutical formulations, the use of the product and the process for its production are described.
Patent ZA-951049-B (ZA)
Title: Holl w con ainer havi g a v ry thin inert or impermeable inner surface layer by coating the inside surface of the preform
Inventor: PLESTER GEORGE
IPC: B29B11/08
Filed: 1995-02-09
Abstract: A very thin inner layer composed of a polymer chosen for its barrier and/or inertness properties is fabricated within a container preform constructed mainly from another polymer, or a structure of polymers. The inner layer on the preform is produced either by a controlled coating method involving coating of the injection mold core rod prior to injection molding or by a coating applied directly to the preform after injection molding. This enables both inner and main layers to be brought together at a time when the interface between them is molten. A tie layer can be employed, when desirable, to enable the layers to be combined without melting the layer interface.
Patent ZA-954815-B (ZA)
Title: Mold separation method and apparatus
Inventor: KINDT-LARSEN TURE
IPC: B29L11/00
Filed: 1995-06-09
Abstract: The present invention provides an apparatus for separating individual contact lens mold assemblies using a steam and demolding means.
Patent ZA-962932-B (ZA)
Title: Device for keeping and delivering a homogeneous cellulose suspension
Inventor: ZIKELI STEFAN
IPC: C08B1/00
Filed: 1996-04-12
Abstract: A method for keeping and delivering a homogeneous suspension of shredded cellulose in an aqueous amine oxide is provided using a horizontal cylindrical vessel including a conveyor screw which is parallel to and partially coextensive with the stirring elements in the vessel.
Patent ZA-968047-B (ZA)
Title: Apparatus for descaling semi-finished products
Inventor: GAYDOUL JUERGEN
IPC: B21B45/08
Filed: 1996-09-25
Abstract: PCT No. PCT/EP96/04126 Sec. 371 Date May 20, 1998 Sec. 102(e) Date May 20, 1998 PCT Filed Sep. 20, 1996 PCT Pub. No. WO97/11797 PCT Pub. Date Apr. 3, 1997An apparatus for descaling semi-finished products, such as thin slabs or steel strips in rolling mills by highly pressurized water that is sprayed through a nozzle device onto the surface of the semi-finished product is characterized in that the nozzle device is movable with a vertical component above the surface of the semi-finished product by means of a drive. The drive can be controlled by a control device that receives a target distance as input value and an actual distance between the nozzle device and the surface of the semi-finished product detected by means of a distance sensor. The control device supplies an output signal via a signal line to the drive for resetting any deviation to zero. Hence, the nozzle device is always kept at a desired target distance even if humps such as bulgings occur on the surface of the semi-finished product.
Patent GB-2370998-B (GB)
Title: Device for assisting therapeutic lower leg,calf-muscle,ankle,foot and toe exercise for reducing the risk of deep vein thrombosis (DVT)
Inventor: FLYNN MICHAEL RICHARD
IPC: A61H1/02
Filed: 2002-03-28
Granted: 2002-11-27
Abstract: A lower leg exercise device (1) has an upper panel (2) and a lower panel (3) which are hingedly attached together along opposing longitudinal sides. A pair of elliptical forming panels (8) are hingedly attached to the lower panel (3) and are each foldable between a first position in which they lie substantially flat against the lower panel, whereby the upper panel may be collapsed flat against the lower panel for compact storage, and a second position in which they engage between the first and second panels in an upstanding manner so as to maintain the panels in spaced apart relationship. In said second position, the loading applied by the convexly curved upper and lower edges of the forming panels (8) to the upper and lower panels (2,3) results in said panels each adopting a convexly curved shape. In use, the device is placed an the floor in its erect configuration, the user placing their feet on the upper panel and rocking the device back and forth on the curved lower panel.
Patent GB-2400463-B (GB)
Title: Data processing apparatus and method for distributing and authenticating electronic documents
Inventor: SHEVADE RAVINDRA WAMAN
IPC: H04L9/32
Filed: 2003-04-11
Granted: 2005-05-25
Abstract: A data processing system for distributing and authenticating documents from a plurality of parties to a recipient data processing apparatus is disclosed. The system comprises a plurality of document distribution devices each configured to generate an original hash value from the content of a file containing a document to be distributed. A recipient data processing apparatus is configured to generate an original super hash value from the plurality of the original hash values, and to distribute the original super hash value to each of the document distribution devices. The system provides assurance that distributed documents have not been tampered with during communication, by an unscrupulous distributing party, or by an unscrupulous recipient by only submitting a hash value of the document to be distributed. The hash value provides for assurance at the eventual recipient of the document that no changes to the document have been made.
Patent GB-2449335-B (GB)
Title: An irrigation device
Inventor: WILLIAMS DAVID
IPC: A01G25/02
Filed: 2008-04-24
Granted: 2009-05-27
Abstract: A device for irrigating soil or other substrates is provided. The device is at least in part biodegradable, minimising its impact on the environment and also provides focused irrigation towards desired areas. The device includes a connector end for connection with a liquid supply, and a biodegradable body adapted to receive liquid from the connector end, wherein the outer surface of the body is substantially water resistant with the exception of one or more feeder areas.
Patent GB-2083330-B (GB)
Title: Heat transfer elements
IPC: H05B3/14
Filed: 1980-06-13
Granted: 1983-11-23
Abstract: A heating element comprises a body provided by fibrous tubes of an electrically conductive material, a voidage between the tubes providing a path for a fluid to be heated. The material may be silicon, silicon carbide, or silicon rich-silicon nitride. The heating element is manufactured by coating a fibrous carbon precursor with the material, and heating the coated precursor in an oxidizing environment so as to remove the carbon precursor by oxidation. The heating element has one application for a heat transfer system for controlling the temperature of a hot working device. The system comprises a fluid circuit including the hot working device, the heating element through which the fluid is driven by a pump, and a temperature controller for sensing the temperature of the device and controlling the temperature of the heating element as a function of the device temperature.
Patent GB-2100290-B (GB)
Title: Corrosion protection system
IPC: C23F13/02
Filed: 1982-06-11
Granted: 1984-02-08
Abstract: Methods of preventing corrosion in which current flows between the to-be-protected substrate and a distributed electrode whose electrochemically active surface provided by an element which is composed of a conductive polymer and which is at least 500 microns thick. In one embodiment, the electrode is a flexible strip comprising a highly conductive core, eg. of copper, and a conductive polymer element surrounding the core. In another embodiment, the electrode is a conductive polymer layer which conforms to the surface of the substrate but is separated from it by a layer of insulation.
Patent GB-2194989-B (GB)
Title: Rod advancing mechanisms
Inventor: COX JOHN PATRICK ANTHONY
IPC: F04B9/14
Filed: 1986-09-15
Granted: 1990-08-08
Abstract: A dispenser gun having a rod-advancing mechanism of the tilting gripper kind employs a hardened steel rod (4) of circular cross-section and a sintered metal gripper (12) having a circular hole (21) through which the rod slides. The gripper has, on at least one side, an indentation (25,28; 31,32) having a generally arcuate base and running into the hole (21). The gripper when tilted grips the rod firmly without marking the rod.
Patent GB-2200046-B (GB)
Title: Pharmaceutical compositions for treating gastric disorders
Inventor: TYERS MICHAEL BRIAN
IPC: A61P1/00
Filed: 1987-11-27
Granted: 1990-09-26
Abstract: The invention relates to the use of compounds of the general formula (I)whereinR' represents a hydrogen atom or a C<sub>1-10</sub> alkyl, C<sub>3-7</sub> cycloalkyl, C<sub>3-7</sub> cycloalkyl-(C<sub>1-4</sub>) alkyl, C<sub>3</sub>-<sub>6</sub> alkenyl, C<sub>3-10</sub> alkynyl, phenyl or phenyl-C<sub>1-3</sub> alkyl group; and one of the groups represented byR<sup>2</sup>, R<sup>3</sup> and R<sup>4</sup> is a hydrogen atom or a C<sub>1-3</sub> alkyl, C<sub>3-7</sub>cycloalkyl, C<sub>2-6</sub> alkenyl or phenyl - C<sub>1-3</sub> alkyl group and each of the other two groups, which may be the same or different, represents a hydrogen atom or a C<sub>1-6</sub> alkyl group; and physiologically acceptable salts and solvates thereof, for the relief of nausea and vomiting and/or the promotion of gastric emptying and for the manufacture of a medicament for this purpose. Promotion of gastric emptying may be for the relief of gastro-intestinal disorders associated with gastric stasis or may be of advantage in radiological examination procedures.The invention also relates to a product containing a therapeutic agent liable to induce nausea and vomiting, e.g. a cytostatic agent such as a cyclophosphamide, an alkylating agent or a platinum complex, and a compound of the general formula (1) as a combined preparation for simultaneous separate or sequential use in therapy.
Patent GB-2209939-B (GB)
Title: The use of 13,14-dihydro-15-keto-prostaglandins as ocular hypotensive agents
Inventor: UENO RYUZO
IPC: A61P27/02
Filed: 1988-09-08
Granted: 1992-01-02
Abstract: The present invention relates to ocular hypotensive agents which contain 13,14-dihydro-15-keto-prostaglandins, which show no transient ocular hypertensive response that PGs usually show.
Patent GB-2299998-B (GB)
Title: Compositions for inhibiting thrombogenesis
Inventor: WEITZ JEFFREY I
IPC: C08B37/00
Filed: 1996-04-01
Granted: 1997-03-26
Abstract: The present invention provides compositions for inactivating thrombin bound to fibrin within a thrombus or clot, whereby the ability of clot-bound thrombin to catalytically promote further clot accretion is substantially diminished or eliminated. The compositions of the present invention are particularly useful for preventing thrombosis in the circuit of cardiac bypass apparatus and in patients undergoing renal dialysis, and for treating patients suffering from or at risk of suffering from thrombus-related cardiovascular conditions, such as unstable angina, acute myocardial infarction (heart attack), cerebrovascular accidents (stroke), pulmonary embolism, deep vein thrombosis, arterial thrombosis, etc. The compositions comprise agents which activate heparin cofactor II mediated inhibition of thrombin and having minimal affinity for antitrhombin III. Preferred agents are low molecular weight heparin preparations (MW of 3,000-8,000) prepared by depolymerising heparin using nitrous acid, oxidising the resultant product with periodate and reducing it with borohydride. The product has its non-sulphated uronic acid residues in open ring form and it substantially free of aldehyde groups.
Patent HU-212517-B (HU)
Inventor: HOLDEN RONALD
IPC: A01H5/10
Filed: 1992-03-24
Abstract: (57) KIVONAT
A beltenyésztett kukoricavonalra az jellemző, hogy első
levélhüvelye antociános elszíneződést mutat, a nővirág
megjelenési ideje késői, a kalászkapelyvák gyenge
antociános elszíneződést mutatnak, a szár ízesülések
antociános elszíneződéstől mentesek, a növény középmagas,
a címer oldalelágazásai közbenső állásúak, a
főcímerág hosszú, szemtermésének hátoldala sárgaszínű,
a csutka antociános elszíneződéssel rendelkezik.
Patent HU-216172-B (HU)
Title: Self-propelled combine-harvester with tiltable cutting range
IPC: A01D41/14
Filed: 1992-10-16
Abstract: The present invention describes a self-propelled combine harvester with a horizontally foldable cutting unit consisting of two cutting-unit halves (14, 15) so that the cutting unit, after being used for work, can be pivoted from the working position into a transport position, so that the permissible maximum width for road transport is not exceeded. To make it possible by simple means to obtain the pivoting movement of the two cutting-unit halves (14, 15), there are provided two very simply constructed drives, of which the first performs the introductory pivoting movement from the working position into the transport position and the second drive is switched on only when the two cutting-unit halves (14, 15) are at a point just before they reach their end position for road transport. The two drives can be designed as follow-up drives. It is also possible, however, to switch on the second drive in addition to the first, that is to say both drives remain switched on to the end. <IMAGE>
Patent HU-217840-B (HU)
Inventor: BOES MICHAEL
IPC: C07D209/96
Filed: 1994-10-17
Abstract: A találmány szerinti (I) általános képletű triciklikuspirrolszármazékok (mely képletben R1–R4 jelentése hidrogénatom,halogénatom, 1–7 szénatomos alkil-, fenil-, 3–6 szénatomos cikloalkil-vagy 1– 7 szénatomos alkoxicsoport, és R2 2–7 szénatomos alkanoil-oxi-, mezil-oxi- vagy (1–7 szénatomos alkoxi)-- karbonil-csoportot isképviselhet; R5–R7 jelentése hidrogénatom vagy 1–7 szénatomosalkilcsoport; X jelentése –CH2–CH(C6H5)–, –YCH2–, –CH=CH– vagy–(CR11R12)n– csoport, ahol R11 és R12 jelentése hidrogénatom vagy 1–7szénatomos alkilcsoport, vagy R11 és R12 közül az egyik hidrogénatomotés a másik fenilcsoportot képvisel; n értéke 1 vagy 2; és Y jelentése–O– vagy –S–) és a bázikus (I) általános képletű vegyületekgyógyászatilag alkalmas sói gyógyászati tulajdonságokkal rendelkező újvegyületek. A találmány szerinti új vegyületek különösen központiidegrendszeri zavarok, kardiovaszkuláris zavarok ésgasztrointesztinális zavarok kezelésére vagy megelőzésére alkalmasgyógyászati készítmények előállítására alkalmazhatók. ŕ
Patent HU-219870-B (HU)
Title: Apparatus for creating a branch point in a pipeline
Inventor: STRINGHETTA SANDRINE
IPC: F16L41/00
Filed: 1996-09-11
Abstract: The apparatus to put in place from ground level a branch connection (10) onto a main underground distribution pipe (1). It consists of a frame (100) containing a vertical support (110) provided with guide slides (112a,112b,113a,113b,114a,114b) and a support (130) placed on the lower part of the frame and designed to position itself under the main pipe (1). There is a connector positioner (200) attached too the frame and containing a hollow sleeve (201) with a temporary holder (239) of the connector (10) and a jack (220 to 226) for pressing the connector (10) onto the main pipe (1). Sealing is provided between the sleeve (201) and the connector (10) to allow the insertion of the drilling tools (270) the fixing piece (280) between the branch connector (10) and the main pipe (1), a blocking piece (300) of the connector (10) and the seal (310) so that no fluid circulating in the main pipe leaks out externally.
Patent IT-1239382-B (IT)
Title: Template for cassettes of magnetic tape
IPC: G11B/
Filed: 1990-03-12
Granted: 1993-10-20
Abstract: The invention concerns a template for cassettes of magnetic tape which includes a sheet-type component which can be inserted between the axial ends of the spools of magnetic tape and the internal walls of the box-shaped case of the cassette and which defines a pair of through holes to correspond with the hubs of the said spools. The sheet-type component has, in at least one of its sections, at least an area in relief for the centring of the magnetic tape and/or of the hubs. The invention is characterised by the fact that it includes, in the external areas of the axes of the said pair of holes in relation to the median transverse axis of the said sheet-type component, at least awindow which belongs at least partially to the said area in relief to reduce the elastic rigidity of the sheet-type component in the area affected by the running of the magnetic tape during its winding and/or unwinding.