baber/WOPTO huggingface dataset:
Patent DE-60002472-T2 (DE)
Inventor: GOENCZI CSABA
IPC: C07B61/00
Filed: 2000-07-13
Granted: 2004-02-26
Abstract: The invention relates to a process for the preparation of spiro[(4-cyclohexanone)-[3H]indol]-2'[1'H]-one derivatives of the general formula I wherein R<SUP>1 </SUP>and R<SUP>2 </SUP>independently stand for hydrogen, C<SUB>1-4</SUB>alkyl, C<SUB>1-4</SUB>alkoxy, C<SUB>1-4</SUB>alkylthio, C<SUB>1-4</SUB>polyfluoroalkyl, C<SUB>1-4</SUB>polyfluoroalkoxy, C<SUB>3-7</SUB>cycloalkyloxy, C<SUB>3-7</SUB>cycloalkylthio, phenoxy, benzyloxy or nitro group-, characterized by reacting an indolin-2-one derivative of the general formula II wherein R<SUP>1 </SUP>and R<SUP>2 </SUP>are as defined above-with a compound capable for introducing a protective group, selected from 2-tetrahydropyranyl, 1-diethoxy-methylene or C<SUB>1-4</SUB>alkoxycarbonylethyl group, coupling the compound of general formula III, thus obtained-wherein R<SUP>1 </SUP>and R<SUP>2 </SUP>are as defined above and A stands for a protective group, selected from 2-tetrahydropyranyl, 1-diethoxy-methylene or C<SUB>1-4</SUB>alkoxycarbonylethyl group-with an acrylic acid C<SUB>1-4</SUB>ester, cyclizing the resulting compound of the general formula IV wherein R<SUP>1</SUP>, R<SUP>2 </SUP>and A are as defined above, R<SUP>3 </SUP>stands for C<SUB>1-4 </SUB>alkyl group-, eliminating the -COOR<SUP>3 </SUP>group and the A protective group of the keto-ester of general formula V wherein R<SUP>1</SUP>, R<SUP>2</SUP>, R<SUP>3 </SUP>and A are as defined above, optionally without isolation of the compounds of the general formulae IV
Patent DE-60002474-T2 (DE)
Inventor: DOUTRE ALLEN
IPC: H04M1/72445
Filed: 2000-07-26
Granted: 2004-02-19
Abstract: A metallic alloy having a semi-solid range between the liquidus temperature and the solidus temperature of the metallic alloy is processed by cooling the metallic alloy from an initial metallic alloy elevated temperature to a semi-solid temperature of less than the liquidus temperature and more than the solidus temperature, and maintaining the metallic alloy at the semi-solid temperature for a sufficient time to produce a semi-solid structure in the metallic alloy of a globular solid phase dispersed in a liquid phase. The cooling may be accomplished by providing a crucible at a crucible initial temperature below the solidus temperature, pouring the metallic alloy into the crucible, and allowing the metallic alloy and the crucible to reach a thermal equilibrium between the liquidus temperature and the solidus temperature of the metallic alloy. The method further includes removing at least some, but not all, of the liquid phase present in the semi-solid structure of the metallic alloy to form a solid-enriched semi-solid structure of the metallic alloy, and forming the metallic alloy having the solid-enriched semi-solid structure into a shape.
Patent DE-60003132-T2 (DE)
Inventor: MICHIYA HAJIME
IPC: H01R12/58
Filed: 2000-08-22
Granted: 2004-04-08
Abstract: Disclosed is an efficient method for electrically connecting two sets of electrode terminals in array on the respective electronic board units such as a combination of a liquid crystal display panel (LCD panel) and a circuit board therefor in assemblage of a display unit by interposing a press-contact connector therebetween. Instead of simply interposing the connector between arrays of electrode terminals, the connector is conjoined with a clip member of a metal by which the connector is secured to the LCD panel or circuit board by clipping a periphery thereof with the clipping parts having resilience at both end portions of the clip member so that the efficiency and reliability of the assemblage works of a LCD panel and circuit board can be greatly improved.  <IMAGE>
Patent DE-60008478-T2 (DE)
Inventor: HOKE JR
IPC: F23D14/22
Filed: 2000-10-16
Granted: 2004-11-25
Abstract: An air-fuel burner (42) is used to maintain an operating temperature in a furnace normally heated with an oxy-fuel burner when the supply of oxygen is temporally reduced or stopped. Preferably, both the oxy-fuel burner and the air-fuel burner mount to a common pre-combustor (14) having a first passage (26) and a separate second passage (32) disposed beneath and coextensive with the first passage (26). When using the oxy-fuel burner, the oxy-fuel flame is directed through the first passage (26) and additional oxygen is directed through the second passage. When using the air-fuel burner, air or oxygen-enriched air is directed through the first passage (26) and fuel is separately directed through the second passage (32). Water cooling of the furnace gases can be used to reduce the volume of exhaust gases when operating with the air-fuel burner. <IMAGE>
Patent DE-60010204-T2 (DE)
Inventor: AGOSTINI ISABELLE
IPC: A61Q1/12
Filed: 2000-06-20
Granted: 2005-04-21
Abstract: Topically applicable cosmetic/dermatological compositions suited for improvedly UV-photoprotecting human skin and/or hair against the deleterious effects of ultraviolet irradiation, advantageously oil-in-water emulsions, contain SPF-synergistically enhancing amounts of (a) at least one UV-screening benzotriazole-substituted silicon compound and (b) at least one UV-screening cinnamic acid derivative, formulated into (c) a topically applicable, cosmetically/dermatologically acceptable vehicle, diluent or carrier therefor.
Patent DE-60013225-T2 (DE)
Inventor: MOGI KINICHI
IPC: C07D211/52
Filed: 2000-11-07
Granted: 2005-09-01
Abstract: Described is a 4-hydroxy-4-phenylpiperidine derivative represented by the following formula (1): <CHEM> Äwherein, R<1> and R<2> are the same or different and each independently represents a hydrogen atom, a lower alkyl, or the like, R<3> represents a hydrogen atom or a group -(CR<4>R<5>)n-Y (in which, R<4> and R<5> each represents a hydrogen atom or a lower alkyl group, Y represents a group -COOR<6>, -CONR<7>R<8>, -OR<9> or -OCOR<10> (in which R<6>, R<9> and R<10> each independently represents a hydrogen atom, a lower alkyl group, or the like, R<7> and R<8> are the same or different and each independently represents a hydrogen atom, a lower alkyl group, or the like), and n stands for 1 to 6)Ü, or salt thereof. The compound exhibits excellent peripheral analgesic action.
Patent DE-60015508-T2 (DE)
Inventor: DELONG ANTHONY
IPC: C07C405/00
Filed: 2000-02-29
Granted: 2005-04-21
Abstract: Compounds having the general structure: which are useful for the treatment of a variety of diseases and conditions, such as bone disorders.
Patent DE-60017537-T2 (DE)
Inventor: HITOMI YASUHIRO
IPC: A01K89/01
Filed: 2000-11-29
Granted: 2006-01-12
Abstract: A spinning reel spool made lightweight while maintaining the strength of the bobbin trunk. The spinning reel spool (4) includes a spool main section (7), a front flange section (8), and a front-flange fixing member (9). The spool main section (7) has a bobbin trunk (7a), a tubular skirt portion (7b) with a larger diameter that is formed unitarily with the rear end of the bobbin trunk (7a), and an inner barrel member (7c) made of a synthetic resin polymer, which is fitted to the inner circumference of the bobbin trunk (7a). The front flange section (8) has a larger diameter and is attached to the front end of the bobbin trunk (7a). The front-flange fixing member (9) fastens the front flange section (8) to the spool main section (7). The bobbin trunk (7a) and the skirt portion (7b) constitute dual larger-smaller stage tubular element that is formed unitarily by press-working a sheet of an aluminum alloy. The inner barrel member (7c) is made of a synthetic resin polymer and is fitted into the bobbin trunk (7a). <IMAGE>
Patent DE-60018211-T2 (DE)
Inventor: HAVENS R
IPC: B29K33/00
Filed: 2000-12-12
Granted: 2005-12-29
Abstract: Microreaction molds and methods of molding very thin films onto substrate surfaces are provided. The molds and molding methods allow for consistency and uniformity in the thicknesses of the films that are applied to the substrate surfaces. The molds may be single composite, such as etched silica, or multicomposite, such as quartz/metal. The molds may further comprise an adjustable molding cavity. The molds of this invention are particularly applicable to generating thin polymeric films onto microchip substrates.
Patent DE-60020112-T2 (DE)
Inventor: FERREE BRET A
IPC: A61B17/56
Filed: 2000-05-30
Granted: 2006-02-02
Abstract: Methods and apparatus for treating disc herniation provide a conformable device which assumes a first shape associated with insertion and a second shape or expanded shape to occlude the defect which typically follows partial discectomy. The device may take different forms including patches size to cover the defect or plugs adapted to fill the defect. In a preferred embodiment, however, the device is a gel or other liquid or semi-liquid which solidifies to occlude the defect from within the body of the disc itself. In another preferred embodiment, a mesh screen is collapsed into an elongated form for the purposes of insertion, thereby minimizing the size of the requisite incision while avoiding delicate surrounding nerves. Such a configuration also permits the use of instrumentation to install the device, including, for example, a hollow tube or sheath adapted to hold the collapsed screen, and a push rod to expel the collapsed device out of the sheath for use in occluding the disc defect. A device may further include one or more anchors to assist in permanently affixing the device with respect to the defect.
Patent DE-60028125-T2 (DE)
Inventor: SUDER TIMOTHY ANDREW
IPC: F02M45/08
Filed: 2000-03-08
Granted: 2007-05-03
Abstract: A method and apparatus for rate shaping a fuel injection profile in a diesel engine. The system includes a fuel injector having a pump chamber, a fuel injecting plunger, a supply line, and a discharge nozzle. A rotation of a camshaft causes reciprocation of the plunger and movement of fuel from the supply line through the chamber to the corresponding cylinder. A spill valve is positioned between the chamber and the nozzle, the valve having a first position providing a maximum fuel injection rate, a second position providing a substantially zero fuel injection rate, and at least one intermediate position providing an intermediate fuel injection rate. The method includes the steps of pressurizing fuel fed to a fuel injector nozzle, partially opening a spill valve communicating with the fuel injector nozzle so that the fuel injector injects fuel into a corresponding engine cylinder at a first fuel injection rate for a predetermined first period of time during an engine fuel injection cycle, and fully opening the spill valve so that the fuel injector injects fuel into the corresponding engine cylinder at a second fuel injection rate for a remainder of the engine fuel injection cycle, wherein the first injection rate and the second injection rate shape a fuel flow rate of injected fuel. <IMAGE>
Patent DE-60032082-T2 (DE)
Inventor: ROSENBERG ZEIL B
IPC: A61M37/00
Filed: 2000-08-07
Granted: 2007-06-21
Abstract: A transdermal delivery device includes a plurality of microneedles for injecting a substance such as a pharmaceutical agent into or below the stratum corneum of the skin. The device has housing formed from a top and bottom wall to define a chamber for containing a pharmaceutical agent. An inlet port is provided in the top wall of the housing for supplying the pharmaceutical agent to the chamber and directing the agent to the microneedles. The housing can have a Luer lock type fitting for coupling with a syringe having a Luer lock collar to inject the pharmaceutical agent into the housing. The housing can be divided into a plurality of chambers by an internal wall for supplying different agents simultaneously or sequentially to a patient. The microneedles have a length of about 5-250 microns and generally about 50-100 microns. <IMAGE>
Patent DE-60037019-T2 (DE)
Inventor: PETTERSSON OLA
IPC: H01L21/8238
Filed: 2000-02-09
Granted: 2008-08-14
Abstract: Electrical connection pads for integrated semiconductor circuits have a protective diode formed by a doped region located in a well of opposite doping and another protective diode formed by a well which surrounds another doped region of the same doping type as a contact area and is surrounded by another well of oppositive doping. The doped regions are connected to the pad and are continuous. Narrow strips extend at or along a portion of the periphery of the pad. Also, the well for which the other doped region serves as a contact, has a strip-shape and is located at the periphery of the pad. The other doped region is also used as a contact for forming an electrical resistor connected to an input/output path of the integrated circuit. The resistor is formed in the well surrounding the other doped region. Another contact of the resistor is formed by a further doped region of the same doping type, also having a strip-shape and located in the same well at the periphery of the pad and beneath a marginal portion of the pad. The resistor thereby does not require any extra space.
Patent DE-60102945-T2 (DE)
Inventor: TANIGUCHI MITSUNORI
IPC: C05F17/02
Filed: 2001-01-31
Granted: 2004-09-02
Abstract: A composting container permitting a compost even with bridges contained therewithin to be discharged. The composting container includes a tubular barrel portion (1) fabricated of an air permeable material, and an openable top lid (6) and an openable bottom lid (4) respectively arranged at the top and bottom thereof, wherein the tubular barrel (1) on the lower half thereof has at least one longitudinally openable port. <IMAGE>
Patent DE-60106292-T2 (DE)
Inventor: SPATAFORA MARIO
IPC: B65B57/12
Filed: 2001-11-12
Granted: 2005-11-10
Abstract: A cigarette packer ( 1 ) incorporates a station at which cigarettes ( 2 ) are formed into groups ( 12 ) and from which the groups ( 12 ) are advanced by a first conveyor ( 13 ) along a first feed path (P) toward a wrapping station ( 16 ). A first inspection device ( 24 ) located along the first feed path (P) detects initially whether or not there are any defective cigarettes ( 2 ) in each group ( 12 ), and a second inspection device ( 45 ) located along a second conveyor ( 30 ) then identifies the single defective cigarettes ( 2 ) detected by the first device ( 24 ); the second inspection device ( 45 ) operates in conjunction with a rejection unit ( 46 ) by which defective cigarettes ( 2 ) are removed from the second conveyor ( 30 ).
Patent DE-60111840-T2 (DE)
Inventor: MARTIN E
IPC: G01F23/26
Filed: 2001-04-13
Granted: 2006-08-03
Abstract: A capacitance measurement circuit and probe includes a drive circuit couplable to a constant-current source, a threshold detector, a probe capacitor, and a reference capacitor. The circuit includes a plurality of switches being actuatable to alternately couple the current source to the probe capacitor and to the reference capacitor. The drive circuit is configured to alternately generate a signal of linear ramp waveform having a slope that is proportional to the magnitude of capacitance of the probe capacitor and of the reference capacitor. The voltage differential between the probe capacitor and reference capacitor are actively nulled to nominally eliminate a parasitic capacitance therebetween.
Patent DE-60112274-T2 (DE)
Inventor: SCHUURMAN ARJAN
IPC: B29C67/00
Filed: 2001-05-14
Granted: 2006-04-20
Abstract: In a method for applying a layer containing at least polymer material to a substrate, there is applied to the substrate a film of polymer particles dispersed in a non-reactive liquid. By subjecting these at least polymer material-containing particles to an energy flow, which is locally at least substantially converted into heat, the particles will fuse with each other as a result of such a heat treatment. In particular, the heat treatment is done with the aid of a laser device operative in the UV region, or a laser device operative outside this region, though then in combination with a heat transferring agent in the film.
Patent DE-60113392-T2 (DE)
Inventor: MENSITIERI GIUSEPPE
IPC: C09K3/00
Filed: 2001-03-09
Granted: 2006-04-27
Abstract: A superabsorbent polysaccharide can be obtained by crosslinking a polysaccharide or derivative thereof with at least 1 % by weight of a flexible spacer having a chain length of at least 9 chain atoms and having terminal activated coupling groups. The flexible spacer may comprise a polyalkyleneglycol with a molecular weight from about 400 to 10,000. The coupling groups may be provided by divinyl sulphone units.
Patent DE-60115946-T2 (DE)
Inventor: LANT JOSEPH
IPC: C11D17/00
Filed: 2001-10-23
Granted: 2006-09-07
Abstract: The present invention relates to a shaped detergent composition comprising: (a) a surfactant; and (b) at least one particle comprising benefit agent wherein the particle floats in deionized water at 20° C. In the compositions of the present invention the particle(s) comprising the benefit agent survive well in the wash liquor and, therefore, it is easier to control the release of the active. In addition, the present shaped compositions can be effectively dosed via the dispensing drawer of standard washing machines.
Patent DE-60118793-T2 (DE)
Inventor: QUIBELL MARTIN
IPC: A61P29/00
Filed: 2001-11-16
Granted: 2007-04-26
Abstract: In formula (IV) R1 = R'C(O), R'SO2, R' = a bicyclic, saturated or unsaturated, 8-12 membered ring system containing 0-4 hetero atoms selected from S, O and N, which is optionally substituted with up to four substituents independently selected from groups a), b), and c) below; or R'= a monocyclic, saturated or unsaturated, 5-7 membered ring containing 0-3 hetero atoms selected from S, O and N, which monocyclic ring bears at least one substituent selected from group a) and/or c) and which may optionally bear one or two further substituents selected from group b); R4 = H, C1-7-alkyl, Ar-C1-7-alkyl, Ar, C3-7-cycloalkyl; C2-7-alkenyl; R3 = C1-7-alkyl, C2-C7 alkenyl, C2-C7 alkenyl, C3-7-cycloalkyl, Ar-C1-7-alkyl, Ar; R5 = C1-7-alkyl, halogen, Ar-C1-7-alkyl, C0-3-alkyl-CONR3R4 or a bulky amine, R6 is H, C1-7-alkyl, Ar-C1-7-alkyl, C1-3-alkyl-SO2-R<ix>, C1-3-alkyl-C(O)-NHR<ix> or CH2XAr, q is 0 or 1, have utility as inhibitors of cysteine proteases such as cathepsin K and falcipain.
Patent DE-60118877-T2 (DE)
Inventor: CATTANEO GIANANGELO
IPC: A61F13/15
Filed: 2001-06-18
Granted: 2006-11-30
Abstract: This envelope, indicatively of polyethylene film, for containing absorbent articles with adhesive, such as sanitary towels for women, pantie protectors, incontinence products, has its inner surface provided with non-stick material, indicatively of silicone nature, distributed in dotted manner, so that those surface regions which do not contain it offer a removal and retention action on excess adhesive or generally a reduction in the adherence of the usual adhesives applied to the sanitary towel, the action being adaptable to the type of use by choosing the type of dotting. <IMAGE>
Patent DE-60130274-T2 (DE)
Inventor: CHEADLE BRIAN
IPC: F28D9/00
Filed: 2001-06-22
Granted: 2008-05-21
Abstract: A heat exchanger is disclosed using a plurality of stacked plate pairs (216) consisting of face-to-face, mating plates, each plate having edge flanges (220,222) extending along edges thereof, first and second spaced-apart primary ridges (224,226) each having a portion thereof located in a common first plane with at least one of said edge flanges, a secondary ridge (228) having a portion thereof located in a second plane spaced from said first plane and substantially parallel thereto; said secondary ridge being provided between an adjacent one of said edge flanges (220,222) and said first primary ridge of the respective plate; said secondary ridges being arranged such that in back-to-back plate pairs, said secondary ridges are joined; said primary ridges having openings (238) formed therein for the passage of the first heat exchanging fluid. <??>The primary and secondary ridges are elongate, intermediate areas (232) are located between said first and second primary ridges, and the intermediate areas of each plate pair have spaced-apart portions to form an inner flow passage (236) between the plates. <??>The secondary ridges have openings (240) formed therein for the passage of said second heat exchanging fluid and said openings (240) communicate to define a manifold for the flow of said second heat exchanging fuid, said intermediate areas of back-to-back plate pairs have spaced-apart portions defining outer flow passages (256) therebetween, and the primary ridges (224,226) of at least one plate of each pair include ribs (260) extending across the width of least one primary ridge of the at least one plate and distributed along the length of the primary ridge, said ribs (260) being located between and separated from said openings (238) formed in the primary ridge and forming crossover passages so that the crossover passages of each plate pair permit said secondary heat exchanging fluid to flow transversely across its respective primary ridges (224,226) and through its respective inner flow passage (236). <IMAGE>
Patent DE-60130693-T2 (DE)
Inventor: OLIVEIRA GARY A
IPC: B60W30/18
Filed: 2001-01-16
Granted: 2008-07-31
Abstract: A transfer case includes an input shaft (50), an output shaft (40), and a gear set (48) selectively operable to translate torque between the input and output shafts at reduced speeds. A clutch (84) is operable to translate torque between the input and output shafts either directly or through the gear set. An actuator (100), having a rotational output, is operatively coupled to the clutch for moving the clutch between predetermined positions. A control unit is employed in connection with the transfer case to effect the method of synchronizing low to high shifts in the transfer case. To this end, the control unit calculates the speed of the actuator as it moves the clutch to a neutral position. The control unit further determines the additional time until the clutch will reach a predetermined synchronization point using the speed of the actuator and the remaining rotational distance through which the actuator must move for the clutch to reach the predetermined synchronization point. The control unit is further operable to stop the actuator when the clutch has reached the synchronization point for no longer than a predetermined time. The control unit then senses and compares the rotational speeds of the input and output shafts and signals the actuator to complete the shift from low to high by moving the clutch to provide direct torque translation between the input and output shafts when the difference in the rotational speeds of the input and output shafts is less than a predetermined value. <IMAGE>
Patent DE-60202853-T2 (DE)
Inventor: OGILVIE W
IPC: C07D471/14
Filed: 2002-03-21
Granted: 2006-02-09
Abstract: A compound of formula I: wherein A is a connecting chain of (C1-3) alkyl; B is O or S; R<1 >is H, (C1-6) alkyl, halo, CF3, or OR<1a >wherein R<1a >is H or (C1-6)alkyl; R<2 >is H or Me; R<3 >is H or Me; R<4 >is H, (C1-4) alkyl, (C3-4) cycloalkyl and (C1-4)alkyl(C3-7)cycloalkyl; W is selected from wherein, a) one of Y is SO2 and the other Y is NR<5>, provided that both are not the same, wherein R<5 >is H, (C1-6)alkyl,(C3-6) cycloalkyl, the alkyl being substituted, COR<5o>, COOR<5p >or CONR<5q>PR<5q>; and each R<8 >is H, (C1-4) alkyl, (C3-6) cycloalkyl, or (C1-4) alkyl-(C3-6) cycloalkyl; or b) E is CR<8a>R<8b >wherein R<8a >and R<8b >is H, or alkyl and J is CH2; or J is CR<8a>R<8b >and E is CH2, and the dotted line represents a single bond; or c) E is C(O) and J is CR<8a>R<8b >or J is C(O) and E is CR<8a>R<8b >and the dotted line represents a single bond; or d) E and J are CR<8a>R<8b >and the dotted line represents a double bond. Compounds of formula I have activity against HIV WT and double mutant strains.
Patent DE-60205873-T2 (DE)
Inventor: LANGE DIETMAR
IPC: A01K23/00
Filed: 2002-02-28
Granted: 2006-02-23
Abstract: A cat lavatory with a lower part and a container holding an absorbent material that can be inserted into the lower part, characterised in that the container comprises a lining layer of non-woven material.