baber/WOPTO huggingface dataset:
Patent LV-10606-A (LV)
Inventor: EMONDS-ALT XAVIER
IPC: C07D211/22
Filed: 1993-02-25
Abstract: Arylalkylamines of formula: 
<IMAGE>
 in which: 
 
  - Y denotes 
  - either a group Cy-N in which: 
 
  Cy denotes an optionally substituted phenyl, a C3-C7 cycloalkyl, a pyrimidinyl or a pyridyl, 
 
  - or a group 
<IMAGE>
 in which 
 
  Ar denotes an optionally substituted phenyl, a pyridyl or a thienyl, 
  x is zero or one, 
  X denotes especially a hydroxyl, a C1-C4 alkoxy, a C1-C4 acyloxy, a carboxyl, a C1-C4 carbalkoxy, a cyano, a group -N-(X1)2 in which the groups X1 independently denote hydrogen or a C1-C4 alkyl, a group -S-X2 in which X2 denotes hydrogen or a C1-C4 alkyl group, a group 
<IMAGE>
 in which Alk is a C1-C6 alkyl, or else X forms a double bond with the carbon atom to which it is bonded and with the neighbouring carbon atom in the heterocyclic ring, 
 
  - m is 2 or 3, 
  - Ar' denotes an optionally substituted phenyl, a thienyl, a benzothienyl, a naphthyl or an indolyl, 
  - R denotes hydrogen or a C1-C6 alkyl, 
  - T denotes a group chosen from -CO- and -CW-NH-, W being an oxygen or sulphur atom, and 
  - Z denotes either hydrogen or M or OM when T denotes the group -CO-, or M when T denotes the group -CW-NH-, M denotes a C1-C6 alkyl, a phenylalkyl, a pyridylalkyl, a naphthylalkyl, a pyridylthioalkyl, a styryl or an optionally substituted mono-, di- or tricyclic aromatic or heteroaromatic group, 
  or one of its salts with inorganic or organic acids. 
 
<??>Application: antagonists of neurokinin receptors.
Patent LV-11019-A (LV)
Inventor: AHLBORN GUENTER
IPC: B61F5/16
Filed: 1993-06-29
Abstract: The invention relates to the linkage of the running gear 2 and 3 and the frame 1 of a railway vehicle with wheel sets clamped securely via axle bearings in a running gear frame 4 and 5, the frame 1 being linked to the running gear frame 4 and 5 via leaf carrying springs 6 and open link suspension 7 without a bogie pin and a frictional rotation restrictor 8 being arranged between the running gear frames 4 and 5 and frame 1. The object of the invention consists in designing the link between the running gear 2 and 3 and frame 1 in such a way that, even when the axle is partially or completely relieved of load or the axle suspension loads, the leaf carrying springs 6 of the running gear 2 and 3 and thus the suspension of the open links 7 are stressed to such an extent that a sufficient restoring effect and a sufficiently large rotational restriction of the running gear 2 and 3 are maintained. This object is achieved in that, between running gear frames 4 and 5 and frame 1, a spring 10 is arranged which clamps said frames to one another and is acted upon inversely proportional to the stress of the leaf carrying springs 6 of the running gear 2 and 3. <IMAGE>
Patent LV-10625-A (LV)
Inventor: ARASAKI MOTOHIRO
IPC: C07D239/00
Filed: 1993-12-17
Abstract: Compounds represented by the general formula (I), <CHEM> wherein R<1> is a saturated or unsaturated, straight or branched hydrocarbon radical [wherein the number of carbon atoms in the longest straight chain of this hydrocarbon radical ranges from three to seven], or a radical of the formula -(CH2)n-Y [in which n is an integer from 0 to 4, when Y is a cyclohexyl radical, or n is an integer from 2 to 4, when Y is a lower alkoxy radical having 1 to 4 carbon atom(s) or a phenyl radical], and R<2> is a hydrogen atom or a radical easily hydrolyzable under physiological conditions, as well as hydrates or solvates of the compounds of the general formula (I), can be utilized in the treatment of tumors, They can be prepared by reacting a compound of formula R<1>-OCOCl with a N<4>-unsubstituted 5'-deoxy-5-fluorocytidine of the above formula I, wherein R<2> would stand for protecting groups, and if necessary removing the protecting groups. <IMAGE>
Patent LV-12085-A (LV)
Inventor: BRASEL KENNETH
IPC: A01N1/00
Filed: 1998-04-02
Abstract: Flt3-ligand can be used to generate large numbers of dendritic cells from hematopoietic progenitor and stem cells. Flt3-ligand can be used to augment immune responses in vivo, and expand dendritic cells ex vivo. Such dendritic cells can then be used to present tumor, viral or other antigens to naive T cells, can be useful as vaccine adjuvants.
Patent ME-P11408-A (ME)
Inventor: CAMUS PHILIPPE
IPC: A61P25/28
Filed: 2000-01-28
Abstract: Pronalazak se odnosi na N-piperidino-5-(4-bromofenil)-1-(2,4-dihlorofenil)-4-etilpirazol-3-karboksamid, njegove soli i solvate, koji su snažni antagonisti kanabinoid CB1 receptorima. Postupak za njihovu pripremu sastoji se od dovođenja u reakciju funkcionalnih derivata 5-(4-bromofenil)-1-(2,4-dihlorofenil)-4-etilpirazol-3-karboksilne kisjeline sa 1-aminopiperidinom sa, po želji, salifikacijom poslije toga.
Patent ME-P36008-A (ME)
Title: Pharmaceutical combination of ethinylestradiol and drospirenone for use as a contraceptive
Inventor: HEIL WOLFGANG
IPC: A61K31/58
Filed: 2000-08-31
Abstract: The present invention relates to a multiple-phase pharmaceutical preparation consisting of a number of separately packaged and individually removable daily dosage units placed in a packaging unit and intended for oral administration for a period of at least 21 consecutive days, wherein said daily dosage unit comprises a natural estrogen, such as estradiol in an amount of from 0.5 mg to 4 mg, and 2 to 4 mg of drospirenone, and wherein at least 70% of said drospirenone is dissolved from said dosage unit within 30 minutes, as determined by USP XXIII Paddle Method II using water at 37°C as the dissolution media and 50 rpm as the stirring rate.
Patent YU-107286-A (YU)
Title: Process for preparation of bis-(piperazinyl)-(or homopiperazinyl)-alkanes
Inventor: DEVLIN J P
IPC: C07D295/084
Filed: 1986-06-19
Abstract: 1. Bis-(piperazinyl- or homopiperazinyl) alkanes of the general formula I  see diagramm : EP0122488,P21,F1  wherein R1 , R2 , R3 and R4 which may be identical to or different from each other, are each hydrogen, alkyl having 1 to 4 carbon atoms, hydroxyl, alkoxy having 1 to 4 carbon atoms, alkanoyloxy having up to 4 carbon atoms, halogen, trihalomethyl, di-C1-4 alkylamino, C1-4 alkoxycarbonyl, nitro, cyano or acyl having 1 to 3 carbon atoms ; R5 and R6 , which may be identical to or different from each other, are each hydrogen, methyl, hydroxyl, carboxyl, C1-4 alkoxycarbonyl, hydroxymethyl, phenyl or p-chlorophenyl, R7 and R8 are each hydrogen or methyl ; j and k are integers from 0 to 3, their sum being no more than 4 ; m and n are integers from 0 to 3, their sum being no more than 4 ; A is -CH2 - or -CH2 CH2 - ; or R5 and R7 together or R6 and R8 together are oxo, provided k or m is other than O ; or R5 and R7 together and R6 and R8 together are oxo, provided k or m are other than O ; R9 and R10 , which may be the same or different, represent hydrogen or from one to four methyl substituents on the carbon atoms of the piperazine ring (A = -CH2 -) ; R11 , R12 , R13 and R14 , which may be identical to or different from each other, are each hydrogen or methyl ; or R11 and R12 together and/or R13 and R14 together are oxo ; and X is alkylene of 1 to 2 carbon atoms, optionally hydroxy-substituted with the proviso that when A = -CH2 -, R1 to R14 are hydrogen and j, k, m and n are each zero, then X cannot be 1,2-ethylenediol, and physiologically acceptable acid addition salts thereof.
Patent YU-37304-A (YU)
Title: Specific binding agents of human angiopoietin-2
Inventor: OLINER JONATHAN
IPC: A61K38/08
Filed: 2002-10-11
Abstract: The present invention relates to specific peptides that recognize and bind to Angiopoietin-2, peptibodies comprising the peptides, methods of making such peptides and peptibodies, and methods of diagnosis and treatment using the peptides and peptibodies.
Patent AU-1084497-A (AU)
Title: Telecommunications switch having a universal applications program interface for stantardized interactive call processing communications
Inventor: HEBERT MARK P
IPC: H04Q3/545
Filed: 1996-11-27
Abstract: The present invention is a universal host-to-switch application program interface (API) utilizing a generic message format for performing call control processing and capable of being customized to meet telecommunications application and network signalling protocol requirements. The generic message formats have programmable fields for transmitting commands, status, and data between the host application and the switch. The present invention further comprises a programmable telecommunication switch that provides a user with the ability to define a desired signalling protocol, either "standard" or custom in nature, for performing any desired switching functions. The present invention includes a protocol development environment which enables a user to define a separate finite state machine for each port provided by the switch. Each finite state machine may be independently defined by combining a series of elementary processing steps, called atomic functions, into primitives, which are in turn combined with states and events to define the desired state machine. Such state machines may include atomic functions configured to generate predetermined messages under predetermined conditions and containing predetermined information. Such state machines may further include the ability to respond to state events that include the receipt of generic API messages configured to provide the state machine with information from the host application.
Patent AU-1155295-A (AU)
Title: Assay for the determination of protein in a biological sample
Inventor: ALBARELLA JAMES
IPC: G01N33/493
Filed: 1995-02-03
Abstract: The detection of protein is accomplished by using a test element containing a phenolsulfonephthalein protein error indicator a buffer and an aliphatic ether-polycarbonate present in an amount equal to or less than ten percent by weight.
Patent AU-1160795-A (AU)
Title: Decorating method and products
Inventor: KAMEN MELVIN E
IPC: C09D11/10
Filed: 1995-02-07
Abstract: d) Radiation-curable polymer composition, for use in a method for decorating substrates with hot-stamping foil, which composition comprises 10 90% (preferably 35 - 90%) of a radiation-curable cycloaliphatic epoxide, 1 - 20% (preferably 3 - 15%) of an ester-containing polyol, preferably with a molecular weight less than 850 and viscosity less than 60 Pa.s, e.g. a polycaprolactone polyol, and 1 - 20% (preferably 3 - 15%) of a defoaming agent e.g. polyvinylbutylether. The composition preferably contains an adhesion-promoter, e.g. 1 - 10% of a silane; and/or when the composition is to be cured by actinic radiation it also desirably comprises a photoinitiator, e.g. 0.5 - 20% (preferably 3 to 15%) of a carbonyl compound and/or a photosensitive onium salt. It may comprise 1 - 50% of pigment.
Patent AU-1270492-A (AU)
Title: Improved blood substitute
Inventor: FEOLA MARIO
IPC: C07K1/30
Filed: 1991-12-13
Abstract: An improved blood substitute comprises purified hemoglobin, preferably bovine, cross-linked intramolecularly with periodate-oxydized ATP (o-ATP) and intermolecularly with periodate-oxidized adenosine (o-adenosine), combined with reduced glutathione (GSH), and optionally enriched with mannitol, non-electrolytes, and/or electrolytes. The blood substitute has prolonged intravascular persistence, can sustain plasma volume, has low oxygen affinity, can work as a physiological oxygen carrier, has vasodilator activity and can reduce the vasoconstriction that follows hemorrhage. A method of treating a human afflicted with acute blood loss and/or a sickling crisis of sickle cell anemia comprises intravenously administrating to the human an effective volume of the blood substitute.
Patent AU-1342000-A (AU)
Title: Plasma fuel processing for nox control of lean burn engines
Inventor: BALKO EDWARD N
IPC: F01N13/02
Filed: 1999-11-04
Abstract: A highly reactive reducing gas mixture is produced from vehicle fuel and introduced into the exhaust gas of an internal combustion engine (10) operated at lean burn conditions and passed over a reducing catalyst (15) to covert NOx emissions to benign emissions. The reducing means for producing from fuel used by said engine a reactive mixture substantially in gaseous form comprises a cracking unit (19) and an oxidation catalyst (22). Air (18,20) can be introduced to the cracked fuel prior to passage over the oxidation catalyst. <IMAGE>
Patent AU-1590797-A (AU)
Title: Method and device for measuring the height of the cutting table
Inventor: LANGKJAER CARSTEN
IPC: A01D41/14
Filed: 1997-01-29
Abstract: A method for measuring the height of the cutting table of an earth-processing implement or an agricultural implement, such as, for example, a combine harvester, relative to a surface of a ground having crops by means of an acoustic transducer arrangement. The method includes forming the sound signal emitted by the transducer arrangement by a pseudonoise signal covering a predetermined frequency band. Comparing the sound signal with the reflected signal. Mutually delaying the sound signal and the reflected signal until the comparison has reached its optimum. Whereafter, the delay represents a measurement of the distance to the surface of the ground.
Patent AU-1733783-A (AU)
Title: Electrophotographic microform system
Inventor: PLUMADORE JOHN D
IPC: G03G15/26
Filed: 1983-07-27
Abstract: Apparatus for imaging and developing electrophotographic elements includes a single module (16) within which there is housed three processing stations (18, 20, 22) equidistantly spaced apart at distances corresponding to the distance separating the image frames of an electrophotographic element microformat. The first station (18) charges and exposes a first image frame of the element (12), the second station (20) tones and preliminarily dries the first image frame while a second image frame is located at the first station (18) for charging and exposure, and the third station (22) completes the drying and fuses the first image frame while the second image frame is now toned and partially dried, a new third image frame being presented to the first station (18) for charging and exposure. An intermittent film transport system, not shown, conveys the film element (12) in a unidirectional mode throughout the processing as indicated by the directional arrow (24). The aforenoted inter-station spacing is facilitated by the compact arrangement of the components at the station with the toning components at the second station (20) partially overlapping the charging/exposure components at the first station (18) and the final dry/fuse components at the third station (22). Processing of any particular single image frame of the film element (12) is thus completed in a minimum amount of time as is the processing of a multiplicity of image frames of the element (12) due to the simultaneous processing of the image frames at the three stations (18, 20, 22) in a time-staggered mode.
Patent AU-1737092-A (AU)
Title: Improvements in or relating to organic compounds
IPC: A01N25/32
Filed: 1992-06-03
Abstract: Microencapsulated agrochemicals based on crosslinked polyester polymers particularly suited to rapidly leaching herbicides.
Patent AU-1882301-A (AU)
Title: Method for scaling fresh fish and removing its internal organs and device for implementation of the offered method
Inventor: PURETZ AVROHOM
IPC: A22C25/02
Filed: 2000-12-17
Abstract: A fish is scaled, and its internal organs removed, by continuously advancing the fish along a treatment path while simultaneously exposing the fish body to high-pressure water jets. During treatment the fish is positioned vertically, with the belly downwards. The forces required for holding and transporting the fish are applied laterally to the upper part of the fish body, which is harder, without touching the belly area, which is soft and therefore is left free. The descaled fish proceeds to a position for cutting the belly area and removing the internal organs. The treatment is carried out in the same devices efficiently and without deterioration of the gustatory properties.
Patent AU-1929099-A (AU)
Title: Identifying the items most relevant to a current query based on items selected in connection with similar queries
Inventor: BOWMAN DWAYNE
IPC: G06Q30/02
Filed: 1998-12-18
Abstract: The present invention provides a software facility for identifying the items most relevant to a current query based on items selected in connection with similar queries. In preferred embodiments of the invention, the facility receives a query specifying one or more query terms. In response, the facility generates a query result identifying a plurality of items that satisfy the query. The facility then produces a ranking value for at least a portion of the items identified in the query result by combining the relative frequencies with which users selected that item from the query results generated from queries specifying each of the terms specified by the query. The facility identifies as most relevant those items having the highest ranking values.
Patent AU-2066201-A (AU)
Title: Mirroring in a stacked network switch configuration
Inventor: KALKUNTE MOHAN
IPC: H04L12/56
Filed: 2000-12-07
Abstract: A method of mirroring data to a mirrored to port in a plurality of switches. The method has the steps of determining if data was sent to all of said plurality of switches; determining if said data was sent to a mirrored to port (MTP); and resending said data to all of said plurality of switches if mirroring is enabled and said data was not sent to said MTP.
Patent AU-2127599-A (AU)
Title: Support material with low pit level
Inventor: RAABE GUNTER
IPC: B29C48/08
Filed: 1999-03-18
Abstract: The surface of a polyolefin-coated substrate material is formed with a cooling cylinder, which has an electrolytically structurized surface with a standard deviation,  sigma Rz, of the roughness Rz of 0.050-0.120 mu m. An Independent claim is also included for the production of the coated substrate.
Patent AU-2150392-A (AU)
Title: Cable length adjustment device
IPC: F16C1/14
Filed: 1992-05-21
Abstract: A cable length adjustment device comprising an elongated member, a locking member formed to prevent translatory movement of the elongated member when in a first locked position, and allow for translatory movement of the elongated member in a second unlocked position, and a housing substantially encasing the locking member.
Patent AU-2169499-A (AU)
Title: Protein humaine beta-trcp
Inventor: BENAROUS RICHARD
IPC: C12N15/00
Filed: 1999-01-29
Abstract: The present invention relates to the human betaTrCP protein for the targeting of proteins towards proteasome degradation pathways, which is capable of interacting with the Vpu protein of HIV-1 virus, with the cell proteins IkappaB and beta-catenin and with the cell protein Skp1p, to its peptide fragments and to the nucleic acid sequences coding for said protein and its fragments.It further relates to the use of the human beta-TrCP protein or its peptide fragments for the screening of anti-HIV-1 antiviral agents, antitumoral agents and anti-inflammatory agents, to the antiviral agents, antitumoral agents and anti-inflammatory agents, and to the antibodies directed against said protein and its peptide fragments.
Patent AU-2346595-A (AU)
Title: Call forwarding method and arrangement for a mobile terminating call
Inventor: PALVIAINEN KEIJO
IPC: H04W4/16
Filed: 1995-05-02
Abstract: PCT No. PCT/FI95/00236 Sec. 371 Date Jan. 4, 1996 Sec. 102(e) Date Jan. 4, 1996 PCT Filed May 2, 1995 PCT Pub. No. WO95/31076 PCT Pub. Date Nov. 16, 1995A call forwarding method and arrangement for a mobile terminating call, for preventing the taped intermediate announcements that are often made during call forwarding, and which can cause a delay in the call set-up, from possibly causing the time-out of the calling modem or telefax terminal and thus the failure of the call. Information concerning the type of call is transmitted to the mobile exchange handling the call included, for instance, in a message where the subscriber database notifies the carrying-out of call forwarding, and provides a call forwarding number. The mobile exchange implementing the call forwarding checks the type data of the call and omits possible intermediate announcements associated with the call forwarding in case of a data call, but allows intermediate announcements in case of speech calls.
Patent AU-2399499-A (AU)
Title: Internet subscriber profile
Inventor: BLEUSE PATRICE
IPC: H04M3/42
Filed: 1999-04-23
Abstract: The internet access unit allows the internet services required by the user to be accessed whilst other services are not available to that user.
Patent AU-2420692-A (AU)
Title: Reagents and methods for the quantification of total doxepins in biological fluids
IPC: G01N33/94
Filed: 1992-07-29
Abstract: Immunoassay methods and reagents for the quantification of total doxepins (i.e., E-doxepin, Z-doxepin, E-desmethyldoxepin, and Z-desmethyldoxepin) in a test sample are disclosed. The quantification of total doxepins is accomplished in an immunoassay employing antibodies and labeled reagents prepared with doxepin derivatives of the Formula II:    <IMAGE>  II  wherein Y-Z can be C=CH or N-CH2, R1 is a linking group, R2 can be H or CH3, and Q can be a detectable moiety or an immunogenic carrier material. The antibody reagent comprises antibodies which are capable of binding to total doxepins and which are produced with one or more immunogens prepared from the doxepin derivative of Formula II, and the labeled reagent is also prepared from the doxepin derivative of Formula II.
Patent AU-2592684-A (AU)
Title: E-shaped resilient metal spring seal resistent to high temperature and high pressure conditions
Inventor: KARR MICHAEL ANDREW
IPC: F16L23/02
Filed: 1984-03-20
Abstract: A metallic spring member 30 cooperates with grooves 32, 34 disposed in pressure containing members 10, 12. The spring member 30 has an E-shaped cross section and is compressed both horizontally and vertically when the members 10, 12 are fully engaged. The seal is self-energizing under normal operating conditions and able to accommodate small, but significant relative motion between the pressure containing members 10, 12 during conditions of abnormally high and unevenly distributed temperature.
Patent AU-2623197-A (AU)
Title: Method for the detection of telomerase activity
Inventor: EMRICH THOMAS
IPC: C12Q1/68
Filed: 1996-11-27
Abstract: The invention concerns a method for the detection of telomerase activity wherein(a) a sample to be tested is provided,(b) a first primer suitable as a telomerase substrate and nucleoside triphosphates are added and the reaction mixture is incubated under conditions under which a primer extension by the telomerase can take place,(c) an amplification of the extension product produced by the telomerase is carried out,(d) the amplification product produced in step (c) is immobilized on a solid phase and(e) the immobilized amplification product is detected qualitatively or/and quantitatively. Furthermore the invention concerns a suitable reagent kit for carrying out the method.