baber/WOPTO huggingface dataset:
Patent SI-1154987-T1 (SI)
Title: Phenylalaninol derivatives
Inventor: SIDDURI ACHYTHARAO
IPC: C07C317/44
Filed: 2000-02-12
Abstract: New Phenylalaninol derivatives (I). Phenylalaninol derivatives of formula (I) are new: [Image] X : a benzamide group of formula (i), a heterocyclyl-amide group of formula (ii) or an imidazolin-3-yl-4-one group of formula (iii): [Image] R 15halo, NO 2, CN, lower alkylsulfonyl, lower alkyl, lower alkoxy, lower alkoxycarbonyl, carboxy, lower alkylaminosulfonyl, lower perfluoroalkyl, lower alkylthio, lower hydroxyalkyl, alkoxy-lower alkyl, alkylthio-lower alkyl, alkylsulfinyl-lower alkyl, alkylsulfonyl-lower alkyl, lower alkylsulfinyl, lower alkanoyl, aroyl, aryl or aryloxy; R 16H, halo, NO 2, CN, lower alkyl, OH lower perfluoroalkyl or lower alkylthio; Het : 5-6 membered heteroaryl containing 1-2 N, O or S; or 9-10 membered bicyclic heteroaryl containing 1-4 O, S or N; R 30H or lower alkyl; p : 0-1; R 18aryl or heteroaryl; R 19optionally substituted lower alkyl, aryl, heteroaryl, aralkyl or heteroaralkyl; R 20lower alkanoyl or aroyl; Y : a group of formula (iv) or (v) or a 5-6 membered heteroaryl, bonded via C and containing 1-3 O, N or S and optionally substituted by 1-2 lower alkyl, cycloalkyl, halo, CN, perfluoroalkyl or aryl, provided that at least one of the substituents is adjacent to the bonding C; [Image] a : an optional double bond; R 22, R 23H, lower alkyl, lower alkoxy, lower cycloalkyl, aryl aralkyl, NO 2, CN, lower alkylthio, lower alkylsulfinyl, lower alkylsulfonyl, lower alkanoyl, halo or perfluoro lower alkyl; provided that at least one is not H; R 24H, lower alkyl, lower alkoxy, aryl, NO 2, CN, lower alkylsulfony or halo; R 25lower alkyl, lower alkenyl (optionally fluorinated) or R 26(CH 2) e; R 26aryl, heteroaryl, N 3, CN, OH, lower alkoxy. lower alkoxycarbonyl, lower alkanoyl, lower alkylthio, lower alkylsulfonyl, lower alkylsulfinyl, perfluoro-lower alkanoyl, NO 2 or NR 28R 29; R 28H or lower alkyl; R 29H, lower alkyl, lower alkoxycarbonyl, lower alkanoyl, aroyl, perfluoro lower alkanoylamino, lower alkylsulfonyl, lower alkylaminocarbonyl or arylaminocarbonyl; or R 28 + R 294-6 membered carbocyclic ring optionally containing 1 O, N or S and optionally substituted on C by lower alkyl or halo; Q : (CH 2) fO, (CH 2) fS, (CH 2) fN(R 27), (CH 2) f or a bond; R 27H, lower alkyl, aryl, lower alkanoyl, aroyl or lower alkoxycarbonyl; e : 0-4; and f : 1-3. An independent claim is included for preparation of (I). ACTIVITY : Antirheumatic; antiarthritic; antiasthmatic; antiinflammatory; neuroprotective. MECHANISM OF ACTION : (I) inhibit the binding of vascular cell adhesion molecule-1 (VCAM1) and fibronectin to the integrin VLA-4 (not defined) on circulating lymphocytes, eosinophils, basophils and monocytes.
Patent SI-1470385-T1 (SI)
Title: A method for suppressing ejection of fragments and shrapnel during destruction of shrapnel munitions
Inventor: DONOVAN JOHN L
IPC: F42B33/06
Filed: 2002-12-30
Abstract: A method of suppressing shrapnel ejection inherent with fragmentary and shrapnel munition destruction. The present invention utilizes a method of imploding an initiating explosive onto the munition device whereby the munition device is exploded. The method has the counterbalancing effect between the explosion and the implosion, thus controlling and drastically decreasing the quantity, velocity, and kinetic energy of the resultant shrapnel ejection. An alternate embodiment of the present invention utilizes a combination of a cylindrical container with the wrapped munition device. The munition device to be destroyed is wrapped with flexible explosive material and placed into the cylindrical container and the resultant void space between the container walls and the munition is filled with pourable or fluid explosive material. Upon detonation of the flexible explosive material and fluid explosive material, an implosion and simultaneous chain reaction occurs whereby detonating the munition device itself. The resultant implosion substantially destroys the munition device and negates the need for any further manual dismantling.
Patent SI-1587821-T1 (SI)
Title: Compositions and methods for stabilizing transthyretin and inhibiting transthyretin misfolding
Inventor: KELLY JEFFREY W
IPC: G01N33/53
Filed: 2003-12-19
Abstract: Kinetic stabilization of the native state of transthyretin is an effective mechanism for preventing protein misfolding. Because transthyretin misfolding plays an important role in transthyretin amyloid diseases, inhibiting such misfolding can be used as an effective treatment or prophylaxis for such diseases. Treatment methods, screening methods, as well as specific transthyretin stabilizing compounds are disclosed.
Patent SI-1975183-T1 (SI)
Title: Tumour-specific recognition molecules
Inventor: GOLETZ STEFFEN
IPC: A61K47/48
Filed: 2003-12-01
Abstract: Recognition molecules (RM), especially antibodies (A) that bind specifically to the Core-1 (C1) antigen, comprising defined amino acids sequences (1-6) given in the specification and below, are new. Recognition molecules (RM), especially antibodies (A) that bind specifically to the Core-1 (C1) antigen, comprising defined amino acids sequences (1-6): (a) AsnTyrTrpLeuGly (1); (b) AspIleTyrPro(Gly) 3TyrThrAsnTyrAsnGluLysPheLysGly (2); (c) AspIleTyrPro(Gly) 2SerTyrThrAsnTyrAsnGluLysPheLysGly (3); (d) TyrAspAlaAlaGlyProTrpPheAlaTyr (4); (e) TyrAspAlaAlaGlyProGlyPheAlaTyr (5); or (f) TyrAspAsnHisTyrPheAspTyr (6). Independent claims are also included for: (1) construct (B) consisting of (A) fused, chemically coupled or non-covalently associated with additional sequences and/or structures; (2) isolated nucleic acid (NA) containing sequences that encode at least one (A) or (B); (3) expression cassette or vector (X) comprising NA and functionally linked promoter; (4) virus or host cell that contains at least one (X); (5) organism that contains at least one host cell of (4); (6) method for preparing (A); and (7) kit containing (A) and/or (B). ACTIVITY : Cytostatic. A multibody (104; sequence of about 200 amino acids reproduced) was coupled to a chelating group then loaded with yttrium99. It was injected (dose 100 MicroCi) into the tail vein of a mouse, subcutaneously implanted with ZA-75-1 (Core-1 positive) tumor cells. A second dose was given after 3 weeks and this treatment produced a significant reduction in tumor growth (no figures given). MECHANISM OF ACTION : Neutralization of Core-1 antigen; Vaccine.
Patent SI-1630336-T1 (SI)
Title: Door with a device for improving the opening behaviour of the door, in particular of a sectional overhead door
Inventor: GROSSE DIETMAR
IPC: E05D15/00
Filed: 2004-08-27
Abstract: The door has a door blade with top and bottom segments, in which each segment has two ends facing opening and closing directions of the blade, respectively. The bottom segment with three rollers shifts its middle roller (16) in the opening direction between its ends, where the middle roller is not adjacent to the end facing the closing direction. The shifted roller is placed in a curved rail section when the blade is opened widely. The curved section is connected to horizontal and vertical sections of the rail. The rollers of each segment slide together in the opening direction of the door.
Patent SI-2805712-T1 (SI)
Title: Heat sterilization of glucocorticoidsteriods
Inventor: ASHLEY ADRIAN
IPC: A61K9/00
Filed: 2005-05-17
Abstract: The present invention provides a method for the sterilization of a labile glucocorticosteroid, which method comprises heat-treating by moist heat the labile glucocorticosteroid in the form of a suspension for a sterilizing-effective time. The methods and compositions according to the invention are useful as therapeutic tools to prevent, reverse, and/or reduce the symptoms of allergic and/or inflammatory conditions in a mammalian patient. The invention also provides methods and compositions, which may be manipulated and fine-tuned to fit the condition(s) to be treated while producing fewer side effects.
Patent SI-1981346-T1 (SI)
Title: Cooling apparatus for cooling dough products and method for cooling dough products
Inventor: VAN CAPELLEVEEN PIETER
IPC: A21C15/00
Filed: 2007-01-24
Abstract: A cooling apparatus (1) and a method for cooling dough products (B), for instance loaves of bread, provided with a cooling space (2) with at least one carrier cabinet (3, 4, 5, 6), wherein the cooling apparatus (1) is provided with a conveying system (T) with carriers (7) so that the carriers are conveyable through the cooling apparatus, while cooling means (9) are present in the cooling space (2) for cooling air, the conveying system (T) comprising a forward path (H) which carries dough products (B) through the at least one carrier cabinet (3, 4, 5, 6), wherein the conveying system (T) comprises a return path (R), wherein the carriers (7) are conveyable through the cooling apparatus (1) in a closed circuit.
Patent SI-2461297-T1 (SI)
Title: Personal identification number distribution device and method
Inventor: AAGE PETER K
IPC: G07F7/00
Filed: 2008-11-12
Abstract: The method of distributing a personal identification number to a user of a card associated with said personal identification number comprises: 
- a step of sending to the user, via a first channel, a request code (260) associated with said card, 
- a step of receiving said request code (260) via a second channel, 
- a step of searching for a record (200) matching the received request code (260), 
- a step of retrieving, from the matching record, the personal identification number (210) associated with said received request code (260) and 
- a step of sending the retrieved personal identification number (210) via a third channel to said user.
Patent SI-2643437-T1 (SI)
Title: Use of a methanol containing fuel composition and prozess for powering a compression ignition engine
Inventor: MORRIS GREG
IPC: F02B51/00
Filed: 2011-11-25
Abstract: A diesel engine fuel composition comprising methanol at a level of at least 20% by weight of the fuel; water at a level at least 20% by weight of the fuel; a ratio of water to methanol of between 20:80 to 80:20; a total amount of water and methanol of at least 60% by weight of the fuel composition, and one or more additives, in a total amount of at least 0.1% by weight of the fuel, wherein the level of sodium chloride, if present as an additive, is between 0 to 0.5% by weight of the fuel, and the level of flavorant, if present as an additive, is between 0 to 1.5% of the composition is provided. Also provided is a process for powering a compression ignition engine using a fuel comprising methanol and water, including inlet air pre-heating, and associated systems and uses of the fuel composition.
Patent TR-201810664-T1 (TR)
Title: Kaynaşık fenil halkaya sahip C-glikozid türevleri veya bunların farmasötik olarak kabul edilebilen tuzları, bunları hazırlamak için usul ve bunları içeren farmasötik bileşim.
Inventor: JOON WOO NAM
IPC: C07H15/203
Filed: 2017-01-03
Abstract: Mevcut tarifname, bir kaynaşık fenil halkaya sahip C-glikozid türevleri veya bunların farmasötik kabul edilebilen tuzlarına, bunları hazırlamak için bir usule, bunları içeren farmasötik bir bileşime, bunların bir kullanımına ve bunu kullanarak SGLT1 ve SGLT2?nin ikili inhibisyonu için bir usule ilişkindir. Mevcut tarifnamenin yeni bir bileşiği, SGLT1 ve SGLT2?ye karşı bir ikili inhibitör aktivitesine sahiptir, dolayısıyla bir diyabet terapötik madde olarak değerli şekilde kullanılır.
Patent DE-3587172-T2 (DE)
Inventor: GUIRE E
IPC: C12Q1/54
Filed: 1985-09-30
Granted: 1993-06-17
Abstract: Apparatuses and methods are disclosed which can be used in the field (i.e., outside the laboratory environment) to determine qualitatively and at least semiquantitatively the presence or absence of minute quantities of ligand. The apparatus can be in the form of a strip comprising a support means provided with a groove intermediate its ends forming a crease line upon which the strip can be folded upon itself with bibulous elements and spaced from the crease line and arranged so that when the strip is folded upon itself the bibulous elements become aligned with each other and come into liquid contact.
Patent DE-3780009-T2 (DE)
Inventor: ALBECK MICHAEL
IPC: A21D2/36
Filed: 1987-11-16
Granted: 1993-01-07
Abstract: Antioxidant compositions and methods are disclosed that are prepared by the extraction of natural antioxidants from plant substrates.
Patent DE-3788861-T2 (DE)
Inventor: ROBSON MICHAEL JOHN
IPC: A01N53/00
Filed: 1987-11-17
Granted: 1994-05-19
Abstract: The invention provides novel insecticidally and acaricidally active compounds of formula (I) : <CHEM> wherein X represents the residue of any carboxylic acid X-COOH which forms an insecticidally active ester with a 3-phenoxybenzyl alcohol, and R, R<6> and R<7> are each selected from hydrogen, halogen, and alkyl of up to four carbon atoms, provided that at least one of R, R<6> and R<7> represents halogen, and further provided that R and R<6> are not both bromine when R<7> is hydrogen. The invention also provides processes for the preparation of compounds of formula (I), compositions comprising them, and methods of combating insect and acarine pests therewith. The invention provides intermediates for the preparation of the compounds of formula (I), those intermediates having the formula : <CHEM> and processes for their preparation. t
Patent DE-3855845-T2 (DE)
Inventor: ENGSTROEM CARL-OTTO
IPC: G09F15/00
Filed: 1988-04-08
Granted: 1997-07-03
Abstract: PCT No. PCT/SE88/00171 Sec. 371 Date Sep. 13, 1989 Sec. 102(e) Date Sep. 13, 1989 PCT Filed Apr. 8, 1988 PCT Pub. No. WO88/08186 PCT Pub. Date Oct. 20, 1988.The present invention relates to a device for receiving essentially planar products, preferably graphic products, which includes two or several frames. Each frame can receive two such products and is formed by four frame members with a longitudinal first flange and a second flange located at one longitudinal narrow side of the first flange. A product inserted into the frame engages the first flanges of the four frame members with its one side and abuts the other flanges with its side edges. The frames are sidewardly hingedly interconnected by means of band-shaped hinges, these band-shaped hinges being designed with two ends and provided with a resilient folding or bending at each end, which is arranged to be received and/or restrained between two opposing walls defining a space in a respective frame member.
Patent DE-3873724-T2 (DE)
Inventor: SPENCER JAMES R
IPC: C22C1/04
Filed: 1988-12-27
Granted: 1993-01-28
Abstract: A consolidated tungsten heavy alloy body consisting essentially of from about 88% to about 98% by weight of nickel, from about 0.25% to about 1.5% by weight of a grain size reducing additive selected from the group consisting of ruthenium, rhenium and mixtures thereof, balance iron and nickel in a weight ratio of nickel to iron of from about 1:1 to about 9:1 wherein the consolidated body has greater than about 2500 grains per square millimeter as determined from the microstructure of the body. A process for producing the consolidated body comprises forming a relative uniform blend of the described metal powders, compacting the powders to form a green body then solid state sintering to remove binders followed by liquid phase sintering the green body to full density.
Patent DE-3874973-T2 (DE)
Inventor: DATTA SUDHIN
IPC: C08F210/00
Filed: 1988-06-08
Granted: 1993-02-18
Abstract: Polymers of olefin monomers and a substantially uniform concentration of carboxyl, hydroxyl, thio, amino, cabonyl and imino functional group-containing monomers. Polymers of olefin monomers and carboxyl, hydroxyl, thio, amino, carbonyl and imino functional group-containing monomers substantially devoid of halogen. Method for preparing polymers by reacting carboxyl, hydroxyl, thio, amino, carbonyl and imino functional group-containing monomers with non-halogenated organometallic compounds to form masked, functional group-containing monomers and polymerizing polymer chain monomers with the masked, functional group-containing monomers to produce a polymer chain. Method for forming masked, functional group-containing monomers by reacting carboxyl, hydroxyl, thio, amino, carbonyl and imino functional group-containing monomers with non-halogenated organometallic compounds. Masked, carboxyl, hydroxyl, thio, amino, carbonyl and imino functional group-containing monomers.
Patent DE-3877440-T2 (DE)
Inventor: STEADLY HARVEY
IPC: B01D69/10
Filed: 1988-01-29
Granted: 1993-05-13
Abstract: Integral gradient, skinned, submicroscopically porous, anisotropic, hydrophilic, asymmetric polyamide membranes comprising: (a) a first porous polyamide zone obtained from a polyamide solution formulated to give coagulated film with pores of a given size, (b) a fabric support imbedded in the first porous polyamide layer, and (c) a second porous polyamide zone having a skinned outer surface, obtained from a polyamide solution having the same constituents as the solution used to form the first porous polyamide zone but solution post-treated to give pores substantially smaller than those in the first porous polyamide zone, as well as a process for producing such membranes, are disclosed.
Patent DE-3889191-T2 (DE)
Inventor: CRONIN DAVID V
IPC: G11B5/596
Filed: 1988-09-30
Granted: 1994-08-04
Abstract: A magnetic data storage system for use with a double sided disk in which a prerecorded pattern of opaque optical lines is used to define the tracks in which magnetic data is to be stored. A separate optical system including an illumination source and a photosensitive detector is provided on a read/write assembly for each side of the disk. Each detector is designed also to serve as a reference grating. The illumination source is designed to image the prerecorded pattern of optical lines on the reference grating as an indication of the alignment of the read/write head of the assembly and a desired data track and any misalignment of the head and track generates a servo signal. The detector uses four separate photocells interleaved in a prescribed fashion to form a quadrature detector that is adjustable to compensate for various non-uniformities. One form of illumination source uses a surface-emitting light emitting diode and optics for forming a multiple beam source.
Patent TR-199800718-T2 (TR)
Inventor: ADAMS EDWARD JOHN
IPC: A01N41/06
Filed: 1996-10-08
Abstract: Istenmeyen bitkilerin kontrol edilmesi için kullanima yönelik (1) formülünün bilesikleri, ve N-oksitleri ve tarimsal açidan müsait tuzlari anlatilmistir. Bahsedilen (1) formülünde, J, J-^, J-19'dur. R2, C1-C6 alkoksi, C1-C6 haloalkoksi, C1-C6 haloalkil, C3-C6 sikloalkil, C3-C6 halosikloalkil, C2-C6 alkoksialkil, C2-C6 haloalkoksialkil, C2-C6 alkenil, C2-C6 haloalkenil, C3-C6 alkoksialkenil, C2C6 alkinil; C2-C6 haloalkinil, C2-C6 siyanoalkil, C1-C6 nitroalkil, (CH2)p-OR6, CH=CH(CH2)q-OR6, C=C(CH2)q-OR6, C2-C6 alkiltioalkil, C2-C6 alkilsülfinilalkil, C2-C6 alkilsülfonilalkil, C3-C8 alkoksikarbonilalkil, C3-C8 alkilkarboniloksialkil ya da istege göre C1-C6 alkil ile ikame edilmis oksiranildir; ayni zamanda (I)formülünün bilesiklerini ihtiva eden bilesimler ve istenmeyen bitkilerin kontrol edilmesi için bir yöntemde anlatilmistir. Bu yöntem, bitkiler ya da ortamlarinin (I) formülünün bir bilesiginin etkili bir miktari ile temasa getirilmesini içermektedir.
Patent TR-199901910-T2 (TR)
Inventor: JENSEN JORGEN KORSGAARD
IPC: G06F3/0354
Filed: 1998-02-11
Abstract: The present invention provides an input device for positioning a cursor on a computer screen by movement of a ball whose rotary movements are transformed into electronic signals, which is unique in that the angular rotations of the ball can be detected by an optical detection means by use of substantively coherent light in such a manner that the rotation of the ball is converted into data values with respect to an x-axis and a y-axis, said axes being preferably perpendicular to each other. This provides a compact detecting device which is suitable for the construction of a computer mouse with the shape of a ball-point pen.
Patent TR-199902575-T2 (TR)
Inventor: ROEDEL WOLFGANG
IPC: A61K9/19
Filed: 1998-04-11
Abstract: Bulus biomoleküllerin depolamada stabil liyofilize farmasötik preparasyonlarina iliskindir; biomoleküller proteinler, peptitler, nükleik asitler ve karbonhidratlar arasindan seçilir ve ayrica bir veya birkaç bazik D veya L-amino asit, buna ek olarak bir veya birkaç aminodikarboksilik asit, hidroksikarboksilik asit veya dikarboksilik asit veya fizyolojik olarak uyumlu tuzlarini içerir. Yardimci maddeler liyofilizatta tamamen veya kismen amorf bir formda bulunur.
Patent TR-199902699-T2 (TR)
Title: Yeni disazo boyarmaddeler.
Inventor: KALWEIT DETLEF
IPC: C07D239/42
Filed: 1998-05-22
Abstract: Bulus formül (I) bilesikler ve bunlarin tuzlarina uygun bilesiklere iliskindir, burada X hidrojen veya kloroyu temsil etmekte, R1 ve R3 hidrojen veya metili temsil etmekte, R2 ve R4 hidrojen, metil veya metoksiyi temsil etmekte ve R5 hidrojen veya C1-4 alkili temsil etmektedir ve bunlar hidroksi grubu ihtiva eden ve ayrica azot ihtiva eden organik substratlarin boyanmasi ve basilmasinda ve mürekkep fiskirtma islemine uygun baski mürekkeplerinin hazirlanmasinda lif tepkin boyarmaddelerdir.
Patent TR-199903189-T2 (TR)
Inventor: DOSENBACH CORNELIA
IPC: A61K31/695
Filed: 1998-06-26
Abstract: Kristalin formdaki Formül (I) 33-epikloro-33-desoksiaskomisini        Formül I        ve A ve B formlari gibi çesitli totomerik veya solvat formlari. Bunlarin hazirlanmasi, amorf bir formül (I) bilesiginin veya A formundan farkli bir formül (I) bilesiginin veya B formundan farkli bir formül (I) bilesiginin, sirasiyla bunlarin bir solüsyonundan kristalinizasyon saglayici sartlar altinda veya sirasiyla A veya B formunun kristalinizasyonunu tercihe bagli olarak saglayan sartlar altinda uygun sekilde dönüstürülmesini kapsar. Böyle kristalinler, özellikle krem, emülsiyon ve merhem gibi farmasötik biçimlerde kullanilmak amaciyla bilesigin topikal galenik formlarinin hazirlanmasinda kullanilmak üzere ortaya konmaktadir.
Patent DE-60004164-T2 (DE)
Inventor: DARSHAN EZRA
IPC: B28D1/14
Filed: 2000-05-16
Granted: 2004-05-27
Abstract: Apparatus for processing a data stream (110) comprises a data stream receiver (150) operative to receive a transport stream (TS), TS storage apparatus (170) operative to store at least a portion of the TS having a beginning and comprising a plurality of TS packets. The apparatus comprises candidate determining apparatus (190) operative to determine, from among the plurality of TS packets, at least one TS packet comprising a candidate access point, candidate offset storage apparatus (170) operative to store in an index store a byte offset of the candidate access point, and arrival time storage apparatus (170) operative to store in the index store a plurality of indications of byte offset, each byte offset being associated with an arrival time of a received TS packet. The TS comprises a partially scrambled TS having a scrambled data portion (130) and an unscrambled data portion (140), and the data stream receiver (150) also comprises analyzing apparatus (160). The analyzing apparatus is operative to distinguish between the scrambled data portion (130) and the unscrambled data portion (140) and to provide the unscrambled data portion (140) for analysis by the candidate determining apparatus (190). The candidate determining apparatus (190) is operative to determine said at least one TS packet comprising a candidate access point based on examination of at least part of the unscrambled data portion (140) provided by the analyzing apparatus (160). <IMAGE>