baber/WOPTO huggingface dataset:
Patent EA-008631-B1 (EA)
Title: Method of squeezing foundry sand, match plate, and upper and lower flasks
Inventor: HIRATA MINORU
IPC: B22C15/02
Filed: 2005-04-27
Abstract: In a conventional apparatus for molding molds, foundry sand is filled in an upper and a lower molding space defined by a match plate, an upper and a lower flask, and an upper and a lower squeeze plate, and then the foundry sand is squeezed by causing the upper and the lower squeeze plate to further approach each other. However, the hardness and strength near the inner surface that corresponds to the match plate, of an upper and a lower mold made by the conventional apparatus, are not high enough.To solve this problem, in this invention the following method is applied: a method for squeezing foundry sand filled in an upper and a lower molding space, comprising: a step to squeeze the foundry sand by causing the upper and the lower squeeze plate to further approach each other, and a step to squeeze it by causing the pattern portions of the match plate to move to each of the upper and the lower squeeze plate.
Patent EA-012589-B1 (EA)
Title: Derivatives of 4-(benzyl)piperazine carboxylic acid phenylamide and associated compounds as fatty acid amide hydrolase inhibitors for the treatment of anxiety, pain and other disorders
Inventor: APODACA RICHARD
IPC: A61P25/04
Filed: 2005-12-29
Abstract: Compounds of formula (I) : wherein, Z is -N-or>CH; Ris -H or –Calkyl; Aris 2-thiazolyl, 2-pyridyl, 3-pyridyl, 4-pyridyl, 2-pyrimidinyl, 4-primidinyl, 5-pyrimidinyl, each unsubstituted or substituted at a carbon ring member with one or two Rmoieties; where each Rmoiety is independently selected from the group consisting of –Calkyl, -Calkenyl, -OH, -OCalkyl, halo, -CF, -OCF, -SCF, -SH, -S(O)Calkyl, -OSOCalkyl, -COCalkyl, -COH, -COCalkyl, -N(R)R, -SONRR, -NRSOR, -C(=O)NRR, -NO, and -CN, wherein Rand Rare each independently -H or –Calkyl; and Aris defined in the claims are useful as FAAH inhibitors. Such compounds may be used in pharmaceutical compositions and methods for the treatment of disease states, disorders, and conditions mediated by fatty acid amide hydrolase (FAAH) activity. Thus, the compounds may be administered to treat, e.g., anxiety, pain, inflammation, sleep disorders, eating disorders, or movement disorders (such as multiple sclerosis).
Patent EA-014504-B1 (EA)
Title: Patch and uses thereof
Inventor: DUPONT CHRISTOPHE
IPC: B05D1/04
Filed: 2007-04-24
Abstract: A patch comprising a support having electrostatic properties is provided wherein a periphery of the support is coated with an adhesive material, and all or part of the non-adhesive surface of the support is covered with at least one biologically active substance in the form of particles that is adhered to the non-adhesive part of the support by electrostatic forces.
Patent EA-014959-B1 (EA)
Title: Glycine transporter-1 inhibitors
Inventor: HITCHCOCK STEPHEN
IPC: C07D333/20
Filed: 2007-06-26
Abstract: The present invention provides compounds of formula (I)wherein: n is an integer from 1 to 3; Rand Rare independently selected from hydrogen or (C-C)alkyl; Rand Rare independently hydrogen; Ris hydrogen or (C-C)alkyl; Aris optionally substituted aryl, heteroaryl or cycloalkyl; and Aris optionally substituted aryl. Such compounds are glycine transporter 1 (GlytT-1) useful for the treatment of diseases treatable by inhibition of GlyT1 such as is Schizophrenia, cognitive disorder associated with Schizophrenia, anxiety, or depression. Also provided are pharmaceutical compositions containing such compounds and processes for preparing such compounds.
Patent EA-016913-B1 (EA)
Title: Process for preparing triazolones
Inventor: ARZENO HUMBERTO BARTOLOME
IPC: C07C205/11
Filed: 2008-05-20
Abstract: The present process provides a improved method for the preparation of alkylsulfanyl substituted triazoles 2 which are useful intermediates in a new process for the preparation of triazolones 20.
Patent EA-016211-B1 (EA)
Title: Method and strand sintering equipment for continuous sintering and pre-reduction of pelletized mineral material
Inventor: OLLILA JANNE
IPC: C22B1/16
Filed: 2008-09-01
Abstract: A method and strand sintering equipment for continuous sintering and pre-reducing of pelletized mineral material. The equipment includes a strand sintering furnace (1). The equipment includes a connecting channel (14, 15), which provides flow communication from a lower exhaust gas duct (8, 9) to an inlet gas duct (12, 13) to conduct at least part of the gas exiting a heating/sintering zone (II, II) to a cooling zone (V, VI), a gas sensor (16, 17), which is arranged in the connecting channel (14, 15) to detect the gas composition, a leakage air channel (18, 19), which provides flow communication between the lower exhaust gas duct (8, 9) and the atmosphere, and a leakage air valve (20, 21), which is in the leakage air channel (18, 19) to open and close the flow communication. To render the gas composition reductive, a control device (22) is arranged to monitor the gas compositions detected by the gas sensor (16, 17) and, on the basis of that, to control the leakage air valve (20, 21) for controlling the access of air from the atmosphere to the exhaust gas duct (8, 9) to adjust the oxygen content of the gas, and/or to adjust the combustion air coefficient of a burner (7) for adjusting the carbon monoxide content of the gas.
Patent EA-017842-B1 (EA)
Title: Azetidine derivatives and use thereof
Inventor: ROUGHLEY STEPHEN
IPC: C07D205/04
Filed: 2009-02-27
Abstract: Compounds of formula (I) are inhibitors of fatty acid amide hydrolase, (FAAH), and which are useful in the treatment of diseases or medical conditions which benefit from inhibition of FAAH activity, such as anxiety, depression pain, inflammation, and eating, sleep, neurodegenerative and movement disorders:wherein Aris phenyl; Ais phenyl, pyridyl, pyrimidinyl, pyrazinyl or pyridazinyl or oxadiazolyl, any of which being optionally substituted; and Aris an optionally substituted divalent phenylene or a pyridinylene radical.
Patent EA-019536-B1 (EA)
Title: Peptide synthesis using enzymatic activation and coupling
Inventor: QUAEDFLIEG PETER JAN LEONARD MARIO
IPC: C07K14/435
Filed: 2009-11-19
Abstract: Method for enzymatically synthesising a peptide, comprising enzymatically preparing an ester or a thioester from: (i) an N-terminal protected amino acid, an N-terminal protected amino acid C-terminal ester, an N-terminal protected peptide, or an N-terminal protected peptide C-terminal ester; and (ii) an alcohol represented by the formula HO-CX-Z respectively a thiol represented by the formula HS-CX-Z, each X independently representing a halogen atom or a hydrogen atom; and Z being selected from the group of sp-hybridised carbons comprising at least two substituents comprising a heteroatom directly attached to the sp-hybridised carbon and sp-hybridised carbons comprising one or two substituents comprising a heteroatom directly attached to the sp-hybridised carbon, the preparation of the ester or thioester being carried out in a reaction medium comprising 2 wt.% water or less based on the weight of liquids in the reaction medium; and enzymatically coupling the prepared ester or thioester with an, optionally C-terminal protected, amino acid or with an, optionally C-terminal protected, peptide, thereby synthesising the peptide in a reaction medium comprising 2 wt.% water or less based on the total weight of the reaction medium.
Patent EA-027074-B1 (EA)
Title: Method of detecting genetic material chlamydia trachomatis, nucleic acid probe (embodiments), forward (embodiments) and reverse (embodiments) pcr primers, pcr component comprising same, kit comprising said component and method of detecting genetic material pectobacterium atrosepticium
Inventor: PEARCE DAVID
IPC: C12Q1/68
Filed: 2010-12-17
Abstract: A method of detecting genetic material deriving from Chlamydia trachomatis comprising detection of a specified nucleic acid sequence, optionally using specific primers and sounds (probes) and optionally in combination with the detection of genetic material deriving from Pectobacterium atrosepticum as an internal control; and related products and kits.
Patent EA-031660-B1 (EA)
Title: Inhalator
Inventor: KNUDSEN CARSTEN LEONHARD
IPC: A61M15/06
Filed: 2011-03-04
Abstract: An inhalator (1) comprising a housing with at least a first compartment (30) and a second compartment (40), and including one or more substances, said second compartment (40) including at least one air entry port (50), said inhalator (1) having a first end (21) proximal to said first compartment (30) and a second end (22) proximal to said second compartment (40), an inhalation part (27) being at said second end (22), said first compartment (30) being for storing at least one substance and including in an inoperative state of said inhalator (1) a plurality of sealing bodies (60) arranged in a neighboring relationship, each pair of neighboring bodies (60) defining at least in part a sealed chamber (62) for containing a substance, said bodies (60) being movable together with said at least one substance from said first compartment (30) into said second compartment (40) to define an operative state of said inhalator (1) wherein said one or more substances are contained in said second compartment (40), whereby air entering through said air entry port (50) and taking up, such as by evaporation, said at least one substance when contained in said second compartment (40) may be inhaled through said inhalation part (27), characterized in a release device in said first compartment (30), said release device being for moving said bodies (60) into said second compartment and allowing said air to flow to said air entry port (50) in said operative state.
Patent EA-029580-B1 (EA)
Title: Container for liquids
Inventor: JAKOBSEN JAN BOERGE
IPC: G21F5/12
Filed: 2012-07-12
Abstract: The present invention relates to a container for liquids, a method of filling it and the use of the container according to the invention for holding and storing radioactive substances. The container for a liquid comprises a cavity for holding the liquid, the cavity being bounded by walls (1) at the sides and at the bottom, an opening for filling the cavity with the liquid, a closure for closing off the cavity, the closure having a piercing region for inserting a cannula into the cavity, a bottom casing (20) which surrounds the walls of the cavity in the standing area, a top casing (10) which surrounds the pierceable closure with the exception of the piercing region, and a film (30) which extends from the top casing to the bottom casing and surrounds those areas of the walls of the cavity which are not already surrounded by the top casing or bottom casing.
Patent EA-027946-B1 (EA)
Title: System for monitoring electric supply lines
Inventor: KNOOP KJELL
IPC: G01K1/14
Filed: 2012-08-31
Abstract: A sensor system for monitoring temperature loads and other impacts on electrical supply installations comprises at least two sensor devices arranged in series at positions in the electrical supply installation to be monitored, one or more signal transmitters connected to each of the sensor devices, one or more signal receivers adapted to communicate with and receive signals from the signal transmitters, and a processing unit connected to at least one of the signal receivers for processing the signals and providing an indication signal.
Patent EA-026892-B1 (EA)
Title: TRIAZOLONE COMPOUNDS AS mPGES-1 INHIBITORS
Inventor: GHARAT LAXMIKANT ATMARAM
IPC: C07D417/12
Filed: 2013-06-10
Abstract: The present disclosure is directed to compounds of formulas (II) and (III) and pharmaceutically acceptable salts thereof as inhibitors of the microsomal prostaglandin E synthase-1 (mPGES-1) enzyme. These compounds are useful in the treatment of a disease, disorder or syndrome mediated by the microsomal prostaglandin E synthase-1.
Patent EA-032004-B1 (EA)
Inventor: ZARIPOV AZAT GUMEROVICH
IPC: A01K15/02
Filed: 2015-03-23
Abstract: Изобретение относится к способам обнаружения взрывчатых и других целевых веществ с помощью собак-детекторов и может быть использовано в аэропортах, вокзалах и других местах скопления людей. Технический результат, на достижение которого направлено изобретение, заключается в повышении достоверности обнаружения взрывчатых и других целевых веществ с помощью собак-детекторов и снижении затрат времени на проведения досмотра. Указанный технический результат достигается в способе обнаружения взрывчатых и других целевых веществ с помощью собак-детекторов, при котором выполняют досмотр объекта собакой-детектором в сопровождении кинолога, визуально отслеживают изменение поведения собаки-детектора и при изменении поведения собаки-детектора определяют присутствие взрывчатых и/или других целевых веществ. Указанный технический результат достигается тем, что до проведения досмотра объекта определяют комплексную психофизиологическую реакцию собаки-детектора на обнаружение запаха взрывчатого и/или другого целевого вещества заданной концентрации, а при изменении поведения собаки-детектора во время досмотра объекта определяют текущую комплексную психофизиологическую реакцию собаки-детектора, сравнивают ее с ранее определенной реакцией на обнаружение запаха и по результатам сравнения делают вывод об обнаружении собакой-детектором взрывчатых и/или других целевых веществ.
Patent EA-025504-B1 (EA)
Title: Sapo-34 molecular sieve and method for preparation thereof
Inventor: TIAN PENG
IPC: C01B37/08
Filed: 2012-09-26
Abstract: The present invention concerns a SAPO-34 molecular sieve and method for preparing the same, whose chemical composition in the anhydrous state is expressed as mSDA·(SiAlP)O, wherein m is from 0.08 to 0.3, and x is from 0.01 to 0.60, and y is from 0.2 to 0.60, and z is from 0.2 to 0.60, and x+y+z=1. There is the template agent SDA in micropores of the molecular sieve. SDA is organic amine with the structural formula as (CH)NRN(CH), wherein R is saturated straight-chain or branch-chain alkylene group with the number of carbon atoms at a range from 2 to 5. There is a slight Si enrichment phenomenon on the crystal surface of the molecular sieve crystal, and the ratio of the surface Si content to the bulk Si content of the crystal ranges from 1.50 to 1.01. Said SAPO-34 molecular sieve after calcined at a temperature range from 400 to 700°C in air can be used as a gas adsorbent and catalysts for acid-catalyzed reaction or oxygenate to olefin reaction.
Patent EA-029495-B1 (EA)
Title: Process for producing fine, morphologically optimized particles using jet mill
Inventor: HANDL WERNER
IPC: B02C19/06
Filed: 2014-03-11
Abstract: The present invention relates to a process for producing fine particles with a high aspect ratio and/or a low specific surface area by means of jet mills, wherein an alkaline grinding aid is added to the grinding gas before it is fed into the grinding chamber of the jet mill. The invention relates to the micronisation of particles of layered structure material having an interplanar distance ranging from 0.30 to 0.40 nm as measured by X-ray diffraction method.
Patent EA-031289-B1 (EA)
Title: Method for storage and discharge of loose materials, primarily grain, from containers and stores
Inventor: TULESHOV AMANDYK KUATOVICH
IPC: B65G65/42
Filed: 2016-03-16
Abstract: The invention is related to containers and stores for grain, in particular, to a grain storage and discharge method. The technical result of the invention is efficiency of grain storage in a store, selective (sectional), along the conveyor length, discharge of grain in case of detection of local (point-like) heating of grain mass. Said technical result is attained by provision of a grain storage method including grain discharge from containers and stores, grain feed toward a conveyor, grain feed onto the conveyor through longitudinal openings in a selective manner, skipping one or several sections along the conveyor length, conveyance of grain on the conveyor, wherein a closed box is used having side walls and a lid and mounted horizontally or obliquely in respect of the horizon, grain is fed onto the conveyor through longitudinal openings in side walls of the box equipped with sectional shutting devices, and grain feeding toward the conveyor is performed by gravity over two surfaces inclined relative to the horizon and installed so that their bottom edges are located at the bottom edges of the longitudinal openings in the side walls of the box. For implementing the proposed grain storage method and for monitoring grain storage, an automated system is used in the store that monitors temperature of grain mass and, in case of local overheating, shuts the longitudinal discharge openings in the sections where there is no overheating. After selective shutting of the longitudinal discharge openings, grain is discharged only from the section(s) where local overheating of grain mass is detected.
Patent EA-035171-B1 (EA)
Title: Conjugates based on psma binding ligands or psma inhibitors for positron emission tomography
Inventor: VLAHOV IONTCHO R
IPC: G01N33/82
Filed: 2014-11-13
Abstract: Described herein are compounds, compositions and methods for diagnosing and/or monitoring a pathogenic disease using positron emission tomography. Furthermore, described are conjugates of the formula B-L-P, wherein B is a radical of a targeting agent selected from PSMA binding ligands or PSMA inhibitors; L is a divalent linker comprising aspartic acid, lysine or arginine, and P is a radical of an imaging agent or radiotherapy agent, such as a radionuclide or radionuclide containing group, or a radical of a compound capable of binding a radionuclide, such as a metal chelating group.
Patent EA-033758-B1 (EA)
Title: 1,2-substituted cyclopentanes as orexin receptor antagonists
Inventor: FIELDHOUSE CHARLOTTE
IPC: A61K31/44
Filed: 2015-02-19
Abstract: The present invention provides compounds of formula (I) and pharmaceutically acceptable salts thereof:wherein L, X, R, R, R, Rand Rare as defined in the specification, processes for their preparation, pharmaceutical compositions containing them and their use in therapy, particularly in the treatment or prevention of conditions having an association with the orexin sub-type 1 receptor.
Patent EA-039000-B1 (EA)
Title: Composition having antiviral effect
Inventor: AMMER RICHARD
Filed: 2016-09-16
Abstract: The invention relates to a pharmaceutical composition which comprises tyrothricine, benzalkonium chloride, and/or benzocaine for use in antiviral therapy or in the treatment of a viral infection.
Patent EA-037719-B1 (EA)
Title: Window assembly with a transparent layer and an antenna element
Inventor: SHIMO KENICHIRO
IPC: H01Q9/40
Filed: 2016-05-11
Abstract: The invention relates to a window assembly having a transparent layer and an antenna element. The technical result consists in increasing efficient antenna performance and in simplifying manufacture and installation of the window assembly with the antenna. The window assembly includes a substrate with an electrically conductive light transparent layer that is performed to reduce transmission of infrared radiation through the window assembly, an area of the transparent layer having a periphery. The substrate further comprises an outer region devoid of the transparent layer and defined adjacent to and along the periphery. An elongated antenna element is disposed in the outer region on the substrate, the element defining a first end and an opposing second end. A feeding element is coupled to the elongated antenna element for energizing the elongated antenna element, such that the elongated antenna element is performed to transmit or receive radio frequency signals. Said area of the transparent layer defines at least two protrusions being spaced apart from one another and extending integrally from the area and into the outer region. The elongated antenna element abuts and is in direct electrical contact with said at least two protrusions. The feeding element couples to the elongated antenna element at a location between said at least two protrusions or at one of said least two protrusions.
Patent EA-036718-B1 (EA)
Title: Self-contained heat meter and method of its implementation
Inventor: TEPLYSHEV VYACHESLAV YURIEVICH
IPC: G01K17/10
Filed: 2019-07-10
Abstract: The invention can be used to determine flow rate in a pipeline completely filled with electroconductive liquid medium, at objects remote from industrial power supply. A heat meter is supplied from autonomous power supply comprising two batteries. EFM (electromagnetic flow meter) supply is carried out by current of rectangular shape. To select the optimum power supply determined are thermal noise voltages in the EFM circuit, in a wide range of change of active resistance, frequency and temperature. Current consumption is defined. Dependences of EFM thermal noise on the temperature higher than 20°C are determined at different resistances of EFM winding and frequency band. In quiescent mode, initial value of thermal noise voltage is determined, in working mode - current one, depending on change of frequency band, active resistances, noise temperature coefficient. Operator monitors working mode of the self-contained heat meter. Under control of a microcontroller, after amplification, matched digitized signals bearing information on flow rate of fluids and temperature are stored and registered in computer unit memory. Significant reduction of electric energy consumption is provided, signal/noise ratio is improved by three orders.
Patent ES-2170669-B1 (ES)
Title: Procedimiento para la encuadernacion de las hojas de un album o libro.
Inventor: ROMERO VENEGAS SALVADOR
IPC: B42B5/06
Filed: 2000-06-15
Granted: 2003-12-16
Abstract: Procedimiento para la encuadernación de las hojas de un álbum o libro; comprende utilizar una pieza prismática con un rehundido longitudinal central de fondo curvo-cóncavo. En el rehundido se dispone en sentido vertical el conjunto de hojas del álbum o libro que se alinean con la ayuda de una pieza plana extrema dispuesta en sentido transversal al rehundido y a tope con uno de los extremos de la pieza prismática. En esta posición las hojas se relacionan por el extremo superior por medio de una pinza. El conjunto de hojas así formado se pone sobre una superficie horizontal presentando el extremo libre de las hojas la forma convexa del lomo que se conforma al depositar cada hoja, empezando por la que se encuentra sobre la superficie y en su cara superior una tira de adhesivo en la parte extrema central, y posteriormente pegar por este procedimiento el resto de las hojas.
Patent ES-2180398-B1 (ES)
Title: Sistema para el control del caudal a traves de una conduccion.
Inventor: MARTINEZ ALMELA JESUS
IPC: G05D7/03
Filed: 2000-12-11
Granted: 2004-03-01
Abstract: Sistema para el control del caudal a través de una conducción que comprende un caudalímetro magnético instalado en un punto de la conducción (1), una válvula de paso servocontrolada (4) instalada en la conducción en un punto situado aguas abajo respecto de la posición del caudalímetro magnético (3) y un equipo de control electrónico (9) a través del que se actúa la válvula de paso (4), en función de las señales proporcionadas por el caudalímetro (3).