baber/WOPTO huggingface dataset:
Patent DE-60313634-T2 (DE)
Inventor: AICHER THOMAS DANIEL
IPC: C07D403/04
Filed: 2003-07-28
Granted: 2008-01-31
Abstract: Described herein are compounds of formula (I) wherein: is an optionally benzo-fused five or six member aromatic ring having zero to three hetero atoms independently selected from N, S, and O; Alk is (C<SUB>1-4</SUB>) alkylene or hydroxy substituted (C<SUB>1-4</SUB>) alkylene; X is oxygen or sulfur; R<SUP>1 </SUP>is hydrogen, (C<SUB>1-6</SUB>) fluroalkyl, (C<SUB>3-6</SUB>) cycloalkyl, or (C<SUB>1-4</SUB>) alkyl, wherein the (C<SUB>1-4</SUB>) alkyl is unsubstituted or substituted with hydroxy, methoxy, ethoxy, OCH<SUB>2</SUB>CH<SUB>2</SUB>OH, or -CN; R<SUP>2 </SUP>is H, halogen, (C<SUB>1-6</SUB>) fluoroalkyl, (C<SUB>1-6</SUB>) cycloalkyl, OR<SUP>4</SUP>, SR<SUP>4</SUP>, NO<SUB>2</SUB>, CN, COR<SUP>4</SUP>, C(O)OR<SUP>4</SUP>, CONR<SUP>5</SUP>R<SUP>6</SUP>, NR<SUP>5</SUP>R<SUP>6</SUP>, SO<SUB>2</SUB>NR<SUP>5</SUP>R<SUP>6</SUP>, NR<SUP>5</SUP>COR<SUP>4</SUP>, NR<SUP>5</SUP>SO<SUB>2</SUB>R<SUP>4</SUP>, optionally substituted aromatic, or (C<SUB>1-6</SUB>) alkyl, wherein (C<SUB>1-6</SUB>) alkyl is unsubstituted or substituted with a hydroxy group; R<SUP>3 </SUP>is hydrogen (C<SUB>1-6</SUB>) fluoroalkyl, (C<SUB>2-6</SUB>) alkenyl, Ar, (C<SUB>1-4</SUB>)alkyl-Ar, or (C<SUB>1-4</SUB>) alkyl wherein (C<SUB>1-4</SUB>) alkyly is unsubstituted or substituted with a phenyl; R<SUP>4 </SUP>is hydrogen, (C<SUB>1-6</SUB>) alkyl, (C<SUB>1-6</SUB>) fluoroalkyl, or optionally substituted aromatic; R<SUP>5 </SUP>and R<SUP>6 </SUP>are independently hydrogen, (C<SUB>1-6</SUB>) alkyl, or optionally substituted aromatic, R<SUP>7 </SUP>is hydrogen, (C<SUB>1-6</SUB>) alkyl, (C<SUB>1-6</SUB>) fluoroalkyl, or optionally substituted aromatic; R<SUP>8 </SUP>and R<SUP>9 </SUP>are independently hydrogen, (C<SUB>1-6</SUB>) alkyl, or optionally substituted aromatic; Ar is optionally substituted phenyl, napthyl, monocyclic heteroaromatic or bicyclic heteroaromatic; Z<SUP>1 </SUP>and Z<SUP>2 </SUP>are independently selected from hydrogen, halogen, (C<SUB>1-6</SUB>) alkyl, (C<SUB>1-6</SUB>) fluoroalkyl, OR<SUP>7</SUP>, SR<SUP>7</SUP>, NO<SUP>2</SUP>, CN, COR<SUP>7</SUP>, CONR<SUP>8</SUP>R<SUP>9</SUP>, NR<SUP>8</SUP>R<SUP>9</SUP>, and optionally substituted aromatic; and all salts, solvates, optical and geometric isomers, and crystalline forms thereof. Also, described are the use of the compounds of formula (I) as antagonists of the dopamine D2 receptor and as agents for the treatment of psychosis and bipolar disorders, and pharmaceutical formulations of the compounds of formula (I)
Patent DE-60315012-T2 (DE)
Inventor: FORSTER IAN J
IPC: B60C23/04
Filed: 2003-04-24
Granted: 2008-04-03
Abstract: An antenna coupled to a wireless communication device is comprised of a conductive component, such as a series of conductive elements, that forms a conductor if placed under a threshold force. The conductor is coupled to the wireless communication device so that the wireless communication device is capable of communicating at an operating frequency defined by the length and construction of the conductor. By communicating using the conductor as an antenna, the wireless communication device may provide an indication of force to an interrogation reader. Furthermore, a conductive support element, such as a tuning ring, may be used for communication as well as coupling the conductive component to the wireless communication device. Multiple conductive components may be coupled to the wireless communication device for communicating at multiple frequencies if placed under multiple threshold forces.
Patent DE-60318312-T2 (DE)
Inventor: COUREAU LAURENT
IPC: G06F21/10
Filed: 2003-05-12
Granted: 2008-12-11
Abstract: A technique for managing access to protected digital content stored in a content broadcasting server ( 11 ) and transmitted to a mobile terminal ( 10 ) connected to a cellular mobile network ( 20 ). A copy of a right of use being stored in a right-of-use management server ( 12 ), said management system is adapted to transmit to said mobile terminal ( 10 ) a message updating said right to use the digital content without any request for a connection from said mobile terminal ( 10 ) to said right-of-use management server ( 12 ).
Patent DE-60319617-T2 (DE)
Inventor: DOLBY JEREMY
IPC: D04H3/02
Filed: 2003-03-07
Granted: 2009-04-02
Abstract: A preform moulding material (12) comprising at least two individual layers (14,16) of fibrous reinforcement material and a matrix resin material between adjacent fibrous reinforcement layers (14,16) to form a prepreg, wherein the matrix resin material impregnates and conjoins the fibrous reinforcement layers (14,16) thereby obviating the need for an additional bonding means to join the individual fibrous reinforcement layers (14,16), wherein the orientation of the fibres of one of the reinforcement layers (14,16) differs from the orientation of the fibres of another reinforcement layer (14,16) whereby said preform moulding material (12) is a multi-axial prepreg.
Patent DE-68902252-T2 (DE)
Inventor: MORANE BRUNO
IPC: A45D40/26
Filed: 1989-02-17
Granted: 1993-03-25
Abstract: Recipient for nail vanish comprising a cap (1) to which is fixed a brush (4) and a bottle (2). This recipient has an elongated shape similar to that of a pen and the bottle (2) is divided into two compartments (5, 6) by a valve (7), in particular a ball valve. The valve (7) is open when the cap (1) of the recipient is in the low position with respect to the bottle (2). 
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Patent DE-68915466-T2 (DE)
Inventor: PARKER DAVID HIRAM
IPC: G01M17/02
Filed: 1989-01-05
Granted: 1994-09-08
Abstract: A method is disclosed for evaluating the level of objectionable noise associated with the operation of a tire by virtue of its tread contacting a road surface, which comprises digitizing the tread design on a coordinate system so as to define load-supporting portions of the tread in contact with the pavement, and distinguish them in binary form from those portions of the tread which are not in contact, as multiple matrix elements; defining a generally arcuate profile of a leading or trailing edge of a footprint of the tread by fitting an equation to the edge; sequentially performing the time ensemble summation, of the noise produced by each matrix element, over every matrix element on the entire circumferential surface; converting the sequence of summation to a periodic analog signal; converting the analog signal to a sound; and aurally evaluating the sound. In a simplified case 0's and 1's along at least one footprint edge are sequentially summed around the circumference of the tire. The system requires only a means for digitizing the tread pattern, a computer to perform the necessary manipulations of data, and a means to convert a digital signal to an analog signal. Having subjectively chosen a tread pattern deemed to have an acceptable noise level, ribs are then relatively rotated one with respect to another to obtain an improved level of tread noise.
Patent DE-68918789-T2 (DE)
Inventor: BURDICK CHARLES LEE
IPC: C08L39/00
Filed: 1989-08-03
Granted: 1995-02-09
Abstract: A suspension of an anionic or nonionic water-soluble polymer in an aqueous solution of an inorganic ammonium salt is characterized in that the polymer comprises at least 15% of the total weight of the suspension, the ammonium salt has a multivalent anion, and the weight ratio of the ammonium salt to the water is at least 0.15.
Patent DE-68920305-T2 (DE)
Inventor: THOMAS BRUCE
IPC: C12N1/00
Filed: 1989-08-07
Granted: 1995-07-20
Abstract: Plant species having enhanced superoxide dismutase activity as a result of transformation with a DNA expression cassette comprising an E. coli MnSOD gene are provided. Transportation of the expression product of the gene may be targeted to a specific cell organelle, such as the chloroplast.
Patent DE-69002154-T2 (DE)
Inventor: LILLA STEFANIA
IPC: F24D19/06
Filed: 1990-12-14
Granted: 1993-11-25
Abstract: A shelf (1) supported on a structure (2) presenting a row of equally spaced, parallel columns (3), and having an object-holder member (5) and at least one element (4) by which it is fastened to the structure (2). The fastening element (4) comprises two bodies (6, 13), the first (6) of which supports the object-holder member (5) and presents at least a first edge (6c) on which is formed a surface (12) mating with the column (3), and the second (13) of which presents a first portion (14) hinged to a second edge (6a) of the first body (6), a second portion (15) diametrically opposed to the aforementioned mating surface (12) so that the column (3) mates with its inside edge, and a cross section smaller than the distance between two adjacent columns (3), so as to enable insertion, during assembly, inside the structure (2) and between the aforementioned adjacent columns (3). <IMAGE>
Patent DE-69002666-T2 (DE)
Inventor: SANSEVERO FRANK M
IPC: B66B21/06
Filed: 1990-03-14
Granted: 1994-03-10
Abstract: An escalator is provided with a curved path of travel from its entry to its exit landings. The path of travel of the escalator steps as seen in plan is a curve having a fixed center and a constant radius from landing to landing. In elevation, each landing portion will be disposed in vertically spaced horizontal planes, and there will be a medial constant slope ascending or descending portion. Interconnecting each landing portion with the constant slope portion will be entry and exit transitional curved portions of varying slope as seen in the elevational view. To enable the steps to traverse the curved path successfully, the effective length of the outer of the step chains is varied at different points along the path of travel of the escalator.
Patent DE-69003431-T2 (DE)
Inventor: GRANELLI RENATO
IPC: D03D47/30
Filed: 1990-04-09
Granted: 1994-01-20
Abstract: The invention concerns a manufacturing method of a secondary nozzle to produce secondary jets in air looms, of the type consisting of a tubular element open at one end and having a gauged hole in correspondence of the opposite end. According to the invention, said method comprises the following steps: - cutting to size a steel rod and finishing its outer surface with centesimal tolerance; - drilling said steel rod with an axial dead hole of gauged dimensions with centesimal tolerance; and - permanently deforming on a die said drilled steel rod, with flattening of at least one part thereof near its closed end and shaping of this end according to an inclined plane, and subsequently forming a gauged hole on said inclined end surface.
Patent DE-69007801-T2 (DE)
Inventor: OHE TATSUYA MITSUI PETROCHEMIC
IPC: B23K26/00
Filed: 1990-01-08
Granted: 1994-07-28
Abstract: A tube having holes formed at precise positions is obtained by preparing a tube in which a substantially black synthetic resin film portion (1) and a synthetic resin film portion (2) having a color other than substantially balck are formed alternately in its circumferential direction and then drilling the black synthetic resin film portion (1) by a laser beam (3).
Patent DE-69017331-T2 (DE)
Inventor: FOTHERINGHAM IAN GRAHAM
IPC: C12N15/60
Filed: 1990-09-19
Granted: 1995-09-21
Abstract: Disclosed are DNA sequences encoding deletion, substitution and/or addition analogs of the E. coli enzyme, chorismate mutase/prephenate dehydratase (CMPD). Preferred expression products include [des-Gln<3><0><7>, des-Ala<3><0><8>, des-Gly<3><0><9>, des-Ala<3><1><0>]CMPD; [Leu<3><0><6>]CMPD; [des-Thr<3><0><4>, Lys<3><0><5>, des-Gln<3><0><6>]CMPD; and [Cys<3><0><9>]CMPD display enzymatic activity of the wild type enzyme but are more resistant to inhibition in the presence of phenylalanine.
Patent DE-69018478-T2 (DE)
Inventor: KLEEMOLA PERTTI
IPC: B65D77/20
Filed: 1990-11-16
Granted: 1995-08-24
Abstract: PCT No. PCT/FI90/00277 Sec. 371 Date Apr. 22, 1992 Sec. 102(e) Date Apr. 22, 1992 PCT Filed Nov. 16, 1990 PCT Pub. No. WO92/04187 PCT Pub. Date Mar. 19, 1992.The invention relates to a container including a container body made of a paperboard-based material and having a top opening at one end, a bottom opening at an other end, a bottom closing the bottom opening, and a lid for closing the top opening. An edge area around the top opening of the container body includes a continuous body section having substantially the shape of a truncated cone, and which extends around, and tapers towards, the top opening so that the generatrix of the continuous body section is at an angle with the generatrix of the container body. The lid is detachably attached to the continuous body section and includes a section having the shape of a truncated cone and the angle of taper of which substantially corresponds to the shape of the continuous body section.
Patent DE-69023687-T2 (DE)
Inventor: SENDELWECK GENE KARL
IPC: H04N9/64
Filed: 1990-04-18
Granted: 1996-06-27
Abstract: An auxiliary video input terminal (S-terminal) couples luminance amd chrominance input signals to respective inputs of peaking circuits (52, 58) in the display processor (40) of a receiver. The chrominance input signal is subjected to pre-distortion (de-peaking) (80) to correct for sideband amplitude distortion in the chrominance peaking filter of the receiver thereby preventing color distortion in displayed images. The luminance signal is subjected to additional peaking (52) at a frequency greater than the characteristic peaking frequency of the luminance peaking filter thereby enhancing the sharpness of wideband luminance input signals displayed by the receiver. <IMAGE>
Patent DE-69025209-T2 (DE)
Inventor: KENTATSU KUNIHIRO
IPC: G11B7/125
Filed: 1990-02-12
Granted: 1996-11-14
Abstract: The apparatus records/reproduces information onto/from an optical card (1) by relatively moving the optical card to the optical head. The optical head has an optical system for producing focusing and tracking control signals. The optical system includes a light emitting diode having a narrow slit-like light emitting surface as a light source. The optical system has photo sensitive elements for focusing control, a photo sensitive element for tracking control, and a recorded information reproducing photo sensitive element which are used to detect the reflected lights from the optical card of a slit light which is emitted from the light emitting diode.
Patent DE-69025336-T2 (DE)
Inventor: KEEFER LARRY KAY
IPC: A61P9/08
Filed: 1990-10-15
Granted: 1996-09-05
Abstract: This invention concerns antihypertensive compositions and a method of lowering blood pressure in mammals. The active component of the compositions is a compound of the formula:   <IMAGE> I  wherein J is an organic or inorganic moiety, M+x is a pharmaceutically acceptable cation and the compound decomposes under physiological conditions to release nitric oxide (NO).
Patent DE-69032840-T2 (DE)
Inventor: HOPPENSTEIN REUBEN
IPC: H04N13/189
Filed: 1990-09-24
Granted: 1999-07-29
Abstract: A method and apparatus for the creation of multi-dimensional images are provided. A plurality of image capture devices are arranged in a predetermined pattern about a target image. A lenticular device divides the target image into a plurality of separate and equally sized strip images with the device being located between the target image and the image capture devices. A screening device may be further located between the lenticular device and the image capture devices to create a composite image for storage and/or transmission over standard transmission and display equipment.
Patent DE-69102211-T2 (DE)
Inventor: NODA KAZUO
IPC: A61K9/54
Filed: 1991-06-27
Granted: 1994-09-15
Abstract: A controlled release pharmaceutical preparation comprising a core containing a medicinal compound and a coating layer containing a water-repellent salt and a water-insoluble and slightly water-permeable acrylic polymer having trimethylammoniumethyl group. Said preparation releases a medicinal compound in a sigmoid type dissolution pattern irrespective of the PH of a dissolution medium.
Patent DE-69109660-T2 (DE)
Inventor: NEMOTO ISAO
IPC: B62M19/00
Filed: 1991-12-30
Granted: 1996-01-11
Abstract: A pneumatic type auxiliary driving apparatus in a bicycle comprising a rotor (13) connected to a wheel (11) of the bicycle, a pneumatic compressing means (20) which compresses air in accordance with the rotation of the rotor (13), an accumulating means (30) which accumulates the air compressed by the pneumatic compressing mechanism (20), and a pneumatic power releasing means which transmits rotational power to the rotor by means of the compressed pneumatic air accumulated in the accumulating means (30). <IMAGE>
Patent DE-69112716-T2 (DE)
Inventor: TAKEDA KOJI
IPC: C12P7/02
Filed: 1991-06-14
Granted: 1996-02-01
Abstract: A method for introducing hydroxyl groups into vitamin D compound at the 1 alpha - and/or 25-positions in the presence of a cyclodextrin compound is effected by the use of a reaction mixture containing a microorganism capable of hydroxylating vitamin D compound or an enzyme produced from the microorganism.
Patent DE-69119990-T2 (DE)
Inventor: GRIFFIOEN WILLEM
IPC: H02G1/08
Filed: 1991-07-12
Granted: 1996-11-07
Abstract: The invention relates to a method, a device and a method for installing a cable in a tubular cable duct. In the method, the foremost end (3) of the cable (1) in the duct (10) and subsequent portions of the cable are first accelerated in a short time with continuous supply of further portions of cable from a torsion-free store. Then, from the instant a certain speed v is reached, the cable is maintained at a tension such that, at said speed and tension, centrifugal forces in bends and inwardly pulling components of tensioning forces in the cable compensate for one another at the position of said bends, the further portions of the cable being supplied at a supply speed such that the part of the cable already fed into the duct can continue to slide on the basis of its mass moment of inertia. The acceleration can be achieved by causing propelling forces to act on the cable upstream of the inlet end (10a) of the duct in conjunction with pulling forces which act at least on the foremost end (3) of the cable (1) in the duct. The magnitude of at least the propelling forces is controlled by adjusting to zero the net transverse force on the cable, in a bend (8; 51) in the cable located beyond the position where the propelling forces act upon the cable in the direction of movement of the cable. Advantages are that much higher installation speeds and/or greater installation lengths in one go are possible. <IMAGE>
Patent DE-69126879-T2 (DE)
Inventor: MAO MARK
IPC: C11D1/52
Filed: 1991-09-25
Granted: 1998-02-19
Abstract: Disclosed is an improved detergent composition comprising one or more anionic surfactants, nonionic surfactants, or mixtures thereof, and detersive enzymes, the improvement which comprises incorporating into said composition an enzyme performance-enhancing amount of a polyhydroxy fatty acid amide material of formula (I), wherein R<1> is H1, C1-C4 hydrocarbyl, 2-hydroxy ethyl, 2-hydroxy propyl, or a mixture thereof, R2 is C5-C31 hydrocarbyl, and Z is a polyhydroxyhydrocarbyl having a linear hydrocarbyl chain with at least three hydroxyls directly connected to said chain, or an alkoxylated derivative thereof.
Patent DE-69211374-T2 (DE)
Inventor: BALSELLS PETER J
IPC: F16L37/084
Filed: 1992-01-21
Granted: 1997-02-06
Abstract: A locking mechanism (10) is disclosed which includes a garter-type canted-coil spring (16) having elliptical coils with a coil height (CH) and a coil width (CW) measured, respectively, along a minor (20) and a major axis (18) of the elliptical coils for holding and locking a first (12) and second member (14) to one another. The first member (12) includes a first groove (24) for retaining the spring (16) with the first groove (24) having a depth (D1) less than the coil width (CW) in order that a portion of each coil extends outwardly from the first groove (24). The second member (14) includes a second groove (34) for accepting the extended portion (30) of each coil (16) and for loading the coils (16) generally along the major axis (18) thereof, said first (12) and second members (14) being locked to one another when the coils (16) are disposed within and loaded by the first (24) and second (34) grooves. <IMAGE>
Patent DE-69211478-T2 (DE)
Inventor: SHEA EDWARD M
IPC: B01D24/46
Filed: 1992-10-23
Granted: 1996-10-24
Abstract: A self-supporting modular underdrain member for use in a liquid filtration system comprises a main body or housing including a pair of longitudinally extending inclined walls which may have a pair of generally triangular transverse walls connecting the inclined walls to one another, the inclined walls each being provided with a pair of longitudinally extending recesses and a plurality of orifices communicating with each of the recesses. A pair of flanges are connected to the inclined walls for attaching the underdrain body to a floor surface so that the inclined walls, any transverse walls and the floor surface define a cross-sectionally triangular underdrain chamber. Two pairs of elongate cover plates are attached to the inclined walls over the recesses to form in each of the inclined walls a pair of longitudinally extending plenums for the equalization of backwash air and water flow. Each of the cover plates being provided with a plurality of spaced slots. <IMAGE>
Patent DE-69213680-T2 (DE)
Inventor: BUENDIA JEAN
IPC: C07J41/00
Filed: 1992-11-05
Granted: 1997-03-06
Abstract: A process for the preparation of a compound of the formula    <IMAGE>  I  wherein R1 is selected from the group consisting of hydrogen, alkyl of 1 to 4 carbon atoms optionally substituted by halogen or a nitrogen or oxygen function and alkenyl and alkynyl of 2 to 4 carbon atoms, R2 is alkyl of 1 to 4 carbon atoms and the A, B, C and D rings are optionally substituted by at least one member of the group consisting of optionally protected -OH or =0, halogen, alkyl and alkoxy of 1 to 4 carbon atoms and alkenyl and alkynyl of 2 to 4 carbon atoms comprising reacting a compound of the formula    <IMAGE>  II  wherein R1 and R2 and the A, B, C and D rings are defined as above with an oxidizing agent in the presence of water and an at least partially water-miscible solvent to obtain a compound of the formula    <IMAGE>  III  wherein R1 and R2 and the A, B, C and D rings are defined as above, subjecting the latter to a solvolysis in a basic or acidic media and optionally subjecting the product to a deprotection reaction of any protected -OH or =0 groups to obtain the compound of formula I and novel intermediates.
Patent DE-69216016-T2 (DE)
Inventor: TAKAHASHI YOSHIKAZU
IPC: H01L23/433
Filed: 1992-09-04
Granted: 1997-04-03
Abstract: To solve the problem that very little heat is dissipated from the surface, the capacity is restricted, and the inductance is high when electrodes on the surface of many semiconductor elements contained in one container with the terminal conductors are connected by wire bonding, the invention provides a semiconductor device (1) wherein a current flowing and heat-dissipating path is formed by contacting bodies (2,5) that make contact with the electrodes (11,12) on the surface of the semiconductor elements and the spring via a spring (6) that makes contact with the inner face of the terminal body (7), which has one face exposed to the outside, or a heat dissipating path is formed by contacting bodies, the pressurising body being coupled with the contacting body via the electrically conductive plate, and the spring, and a current flowing path is formed by connecting an electrically conductive plate with the terminal body. This construction allows the module to be cooled from both sides of the container, and allows the inductance to be reduced. <IMAGE>
Patent DE-69230379-T2 (DE)
Inventor: HOLTON ROBERT A
IPC: C07D409/12
Filed: 1992-09-22
Granted: 2000-05-25
Abstract: 10-Desacetoxytaxol and its derivs. of formula (I) are new, where R2 = H or opt. protected OH; R3, R4 = H, opt. protected OH, Me, -SH, -NH2 or -NR8R9; R5 = R10 or -OR10; R6, R7 = H, alkyl or aryl; R8, R9 = H, alkyl, alkenyl, alkynyl or aryl; R10 = alkoxy, alkyl, alkenyl, alkynyl or aryl; provided that when R2 = H then R3 and R4 are not opt. protected OH. 10-Desacetoxytaxol and 10- desoxytaxotere, are specifically claimed.