baber/WOPTO huggingface dataset:
Patent AU-2003217936-A1 (AU)
Title: Piperazine substituted aryl benzodiazepines and their use as dopamine receptor antagonists for the treatment of psychotic disorders
Inventor: ROCCO VINCENT PATRICK
IPC: C07D498/02
Filed: 2003-03-17
Abstract: Described herein are antipyschotic compounds of formula (I) wherein, A is an optionally benzo-fused five or six member aromatic ring having zero to three hetero atoms independently selected from N, O, and S; Alk is (C<SUB>1-4</SUB>) alkylene optionally substituted with OH, methoxy, ethoxy, or F; Ar is optionally substituted phenyl, naphthyl, monocyclic heteroaromatic, or bicyclic heteroaromatic; R<SUP>1 </SUP>is hydrogen or (C<SUB>1-4</SUB>) alkyl optionally substituted with OH, OR<SUP>3</SUP>, or OCH<SUB>2</SUB>CH<SUB>2</SUB>OH, wherein R<SUP>3 </SUP>is (C<SUB>1-2</SUB>) alkyl; R<SUP>2 </SUP>is H, (C<SUB>1-6</SUB>) alkyl, halogen, fluorinated (C<SUB>1-6</SUB>) alkyl, OR<SUP>4</SUP>, SR<SUP>4</SUP>, NO<SUB>2</SUB>, CN, COR<SUP>4</SUP>, CONR<SUP>5</SUP>R<SUP>6</SUP>, SO<SUB>2</SUB>NR<SUP>5</SUP>R<SUP>6</SUP>, NR<SUP>5</SUP>R<SUP>6</SUP>, NR<SUP>5</SUP>COR<SUP>4</SUP>, NR<SUP>5</SUP>SO<SUB>2</SUB>R<SUP>4</SUP>, or optionally substituted phenyl, wherein R<SUP>4 </SUP>is hydrogen, (C<SUB>1-6</SUB>) alkyl, fluorinated (C<SUB>1-6</SUB>) alkyl, or optionally substituted phenyl, R<SUP>5 </SUP>and R<SUP>6 </SUP>are independently hydrogen, (C<SUB>1-6</SUB>) alkyl, or optionally substituted phenyl; Z is one or two substituents independently selected from hydrogen, halogen, (C<SUB>1-6</SUB>) alkyl, fluorinated (C<SUB>1-6</SUB>) alkyl, OR<SUP>7</SUP>, SR<SUP>7</SUP>, NO<SUB>2</SUB>, CN, COR<SUP>7</SUP>, CONR<SUP>8</SUP>R<SUP>9</SUP>, SO<SUB>2</SUB>NR<SUP>8</SUP>R<SUP>9</SUP>, NR<SUP>8</SUP>SO<SUB>2</SUB>R<SUP>7</SUP>, NR<SUP>8</SUP>R<SUP>9</SUP>, or optionally substituted phenyl, wherein R<SUP>7 </SUP>is hydrogen, (C<SUB>1-6</SUB>) alkyl, fluorinated alkyl, or optionally substituted phenyl, R<SUP>8 </SUP>and R<SUP>9 </SUP>are independently hydrogen, (C<SUB>1-6</SUB>) alkyl, or optionally substituted phenyl; and salts, solvates, and crystal forms thereof. Also described are the use of the compounds of formula (I) as antagonists of the dopamine D<SUB>2 </SUB>receptor and as agents for the treatment of psychosis and bipolar disorder, and pharmaceutical formulations of the compounds of formula (I).
Patent AU-2003229019-A1 (AU)
Title: Land grid array fabrication using elastomer core and conducting metal shell or mesh
Inventor: HOUGHAM GARETH G
IPC: H01R43/00
Filed: 2003-05-13
Abstract: Methods for fabricating Land Grid Array (LGA) interposer contacts that are both conducting and elastic. Also provided are LGA interposer contacts as produced by the inventive methods. Provided is LGA type which utilizes a pure unfilled elastomer button core that is covered with an electrically-conductive material that is continuous from the top surface to the bottom surface of the button structure. In order to obviate the disadvantages and drawbacks which are presently encountered in the technology pertaining to the fabrication and structure of land grid arrays using electrically-conductive interposer contacts, there is provided both methods and structure for molding elastomer buttons into premetallized LGA carrier sheets, and wherein the non-conductive elastomer buttons are surface-metallized in order to convert them into conductive electrical contacts.
Patent AU-2003230055-A1 (AU)
Title: Method and device for entering words in a user interface of an electronic device
Inventor: JOERESSEN OLAF
IPC: G06F3/023
Filed: 2003-05-07
Abstract: A device, comprising: a display, having a display area, for displaying information content; a user input device; and a processor, for controlling the display, arranged to incrementally change the size of the display area while displaying the information content, in response to successive inputs from the user input device.
Patent AU-2003239776-A1 (AU)
Title: A transducer for bioacoustic signals
Inventor: ANDERSEN KNUD BJORN
IPC: H04R1/46
Filed: 2003-06-23
Abstract: In well-known electronic stethoscopic transducers the sensitive element is influenced by signals transmitted via the skin, and the rear side is enclosed in a housing to prevent airborne noise from reaching the sensitive element. According to the invention, an improved signal-to-noise ratio is obtained by letting the transducer be a piezoelectric transflexural diaphragm in contact with the skin, the rear side of the diaphragm communicating with the surrounding air via an acoustical network, thereby receiving airborne noise which acts to counteract the influence of noise coming from the skin.
Patent AU-2003244152-A1 (AU)
Title: Biocompatible polymer and filter for selectively eliminating leucocytes using the same
Inventor: KUNO SUSUMU
IPC: A61K35/14
Filed: 2003-06-17
Abstract: A polymer having an extremely low elution property, excelling in biocompatibility, and useful for selective leukocyte removal filter is provided. A filter material for selective removal of leukocytes, a filter apparatus for selective removal of leukocytes, and a system for selective removal of leukocytes using the above polymer are also provided. The above polymer comprises 8-45 mol% of a unit originating from a polymerizable monomer having a polyalkylene oxide chain, 30-90 mol% of a unit originating from a polymerizable monomer having a hydrophobic group, and 2-50 mol% of a unit originating from a polymerizable monomer having a hydroxyl group.
Patent AU-2003246056-A1 (AU)
Title: High-gradient recursive locating system
Inventor: GOVARI ASSAF
IPC: A61B1/00
Filed: 2003-09-12
Abstract: A system for tracking a probe within an area of operations such as a patient's body comprises a set of primary radiators disposed at known locations. The primary radiators are driven by a control unit to track the positions of a plurality of secondary radiators with respect to the primary radiators. The secondary radiators are optionally movable, and are driven to track the position of the probe with respect to the secondary radiators. A calculation is performed to determine the corresponding position of the probe with respect to the fixed locations. Radiators at each level of the hierarchy generate fields that are locally optimized for detection by the next level of the hierarchy and for the minimization of interference by nearby metallic objects. The system is also capable of determining the angular alignment of the probe with respect to a known coordinate system. <IMAGE>
Patent AU-2003246639-A1 (AU)
Title: Hair treatment compositions comprising hydroxy compounds
Inventor: CORNWELL PAUL ALFRED
IPC: A61K8/34
Filed: 2003-06-26
Abstract: The invention provides a hair treatment composition such as a shampoo or conditioner suitable for topical application to hair for the repair and prevention of damage comprising a hydroxy compound having the following parameters: i) electrotopological state indice of OH S_sOH<9.26 (ii) multigraph information content indice BIC>0.8 (iii) electrotopological state indice of CH3 S_sCH3<6.26 and (iv) a molecular weight greater than 90 wherein the composition does not dye the hair. Preferred hydroxy compounds are 2-methyl-2-hexanol, 2-methyl-2-heptanol, 2-methyl-3-heptanol, 2-methyl-2-pentanol, 2-methyl-3-hexanol, 3-methyl-2-pentanol, 2-methyl-1-pentanol.
Patent AU-2003252791-A1 (AU)
Title: Shaping pulley assembly for belt notching machine
Inventor: CAPORUSSO ALESSANDRO
IPC: B24B21/00
Filed: 2003-10-02
Abstract: The assembly has a stationary center (7) and a removable counter-center (8) both being live centers housed in respective housings (10, 11) of stationary center and removable counter-center. An idle shaping pulley (4) in the form of a cylindrical roller has center holes opposite to each other for the fixed center and the removable counter-center on the respective bases of the shaping pulley.
Patent AU-2003254224-A1 (AU)
Title: Tissue and fluid sampling device
Inventor: BROWN STUART B
IPC: A61B10/00
Filed: 2003-07-28
Abstract: An instrument for removing a tissue sample from a subject comprises a plurality of tissue sampling devices having respective chambers, the tissue sampling devices being radially disposed along a length of the instrument such that upon insertion of the instrument into the subject one or more samples are extracted and isolated in the respective chambers of the sampling devices at the site at which removal occurs.
Patent AU-2003272766-A1 (AU)
Title: Color changing tape, label, card and game intermediates
Inventor: DRONZEK PETER J JR
IPC: B32B27/08
Filed: 2003-09-29
Abstract: This invention relates to color changing tape, label, card and game intermediates for evidence of use, concealing proprietary information or gaming or promotional information until the intermediate is separated. The intermediate includes a substrate of clear or transparent or colored translucent polymeric film or translucent paper combined with judiciously selected cleanly separable translucent colored coatings in intimate contact to form one translucent color that leave no residue when separated.
Patent AU-2003283551-A1 (AU)
Title: Radiotherapy apparatus and operating method
Inventor: BROWN KEVIN JOHN
IPC: A61B6/03
Filed: 2003-11-13
Abstract: A radiotherapy apparatus comprises a source of therapeutic radiation, a source of imaging radiation and a two-dimensional imager for the imaging radiation, a computing means for preparing tomography data from the output of the imager, the therapeutic source being controllable on the basis of feedback from the tomography data, wherein the computing means is arranged to prepare a plurality of intersecting sectional views from the output of the imager, akin to a portal image but with better contrast and the detail of a section rather than that of a projection. This is easier to interpret and visualise a series of sectional than a three dimensional view. Pixels of the images are the result of averaging a plurality of voxels arranged transverse to the section, typically orthogonal and linear. Typically, good results can be achieved using between 5 and 20 voxels. About 10 is suitable, ie between 7 and 15. There is a ideally a display means for showing the sectional views to an operator. The therapeutic source can then be controlled on the basis of instructions from the operator, given via an input means such as a mouse or other pointer, which is preferably correlated to the display. This correlation can be via a superimposed image on the display which is moveable in response to operation of the input means. The superimposed image can derived from one of a previous investigation and a treatment of the patient, so that it corresponds in shape to the area or the image which is being sought. The superimposed image is preferably an outline so that the underlying image is clear.
Patent AU-2003296424-A1 (AU)
Title: Neurotoxic amino acid or neurotoxic derivative thereof associated with neurological disorders
Inventor: BANACK SANDRA
IPC: G01N33/567
Filed: 2003-12-08
Abstract: The invention relates to a method for screening an environmental sample to determine if the environmental sample is associated with exposure of a subject to a neurotoxic amino acid or neurotoxic derivative thereof associated with a neurological disorder, comprising, obtaining a keratinous tissue sample from the subject and analyzing the sample to determine the amount of ²-N-methylamino-L-alanine (BMAA) or a BMAA derivative, and obtaining an environmental sample from material that may be ingested by the subject and analyzing the environmental sample to determine the presence of BMAA or a BMAA derivative, wherein the presence of BMAA or a BMAA derivative in the environmental sample indicates exposure of the subject to at least one neurotoxic amino acid or neurotoxic derivative thereof associated with a neurological disorder. Furthermore, the invention relates to a method for screening a food chain for a neurotoxic amino acid or neurotoxic derivative thereof associated with a neurological disorder comprising, obtaining environmental samples from at least two trophic levels of the food chain and analyzing each environmental sample to determine the presence of BMAA or a BMAA derivative, wherein the presence of BMAA of a BMAA derivative in at least one sample indicates at least one neurotoxic amino acid associated with a neurological disorder is found in the food chain. Finally, a kit for screening an environmental sample to determine if the environmental sample is associated with exposure of a subject to a neurotoxic amino acid associated with a neurological disorder, comprising means for identifying material that may be ingested by the subject and obtaining an environmental sample from the material, and assay means for analyzing the environmental sample to determine the presence of BMAA or a BMAA derivative is envisaged.
Patent WO-2004110570-A1 (WO)
Title: Appareil buccal
Inventor: FARRELL CHRISTOPHER JOHN
IPC: A63B71/08
Filed: 2004-06-11
Abstract: La présente invention concerne un système de protection (1) utilisé dans le domaine sportif, qui doit être placé dans la bouche de l'utilisateur. Ce système de protection (1) comprend généralement un élément de base (2) qui présente habituellement une forme de U correspondant au contour de la mâchoire d'un utilisateur et qui définit un canal supérieur (10) dans lequel une rangée supérieure de dents d'un utilisateur peut être reçue. Le système de protection comprend également un élément d'engagement de dents (3) associé au canal (10) qui est constitué d'une matière pouvant se conformer à la bouche de l'utilisateur ou être moulée à la forme de la bouche de l'utilisateur. Le système de protection comprend également un système d'absorption de choc qui est associé à l'élément de base (2), afin d'absorber un choc d'impact. Ce système d'absorption de choc comprend des canaux ouverts dans l'élément de base (2), qui fonctionnement comme des ressorts pneumatiques. Il est avantageux que l'élément de base comprenne du polyéthylène mélangé à 10 % maximum d'éthylène-acétate de vinyle (EVA). L'ajout d'EVA offre plus de souplesse au système de protection selon cette invention. L'élément d'engagement de dents est constitué d'EVA.
Patent WO-2005047525-A1 (WO)
Title: Procedes pour valider une cible afin de moduler l'action de l'insuline et cribler des modulateurs de l'action de l'insuline et utilisations therapeutiques de ceux-ci
Inventor: JAMES DAVID
IPC: C12Q1/25
Filed: 2004-11-15
Abstract: La présente invention concerne plusieurs formats de dosage pour déterminer l'effet de composés sur un ou plusieurs phénotypes associés à un métabolisme dans une cellule, un tissu ou un animal. Ces formats de dosage sont basés sur la découverte que Cbl (par ex. le c-Cbl protooncogène) est un régulateur en amont de l'activité de AMPK et de l'activité de ACC dans le muscle et que cette voie de régulation modifie toute la dépense énergétique du corps et toute la sensibilité à l'insuline du corps.
Patent WO-2005058444-A1 (WO)
Title: Machine de jeu a ligne de paiement etendue et a elements a n faces
Inventor: QUAYLE JASON
IPC: G07F17/34
Filed: 2004-12-17
Abstract: L'invention concerne une machine de jeu pour un jeu de hasard selon laquelle un gain dudit jeu de hasard est déterminé par un motif de ligne de paiement prédéfini faisant partie d'une pluralité de motifs de ligne de paiement comprenant des inscriptions affichés sur un moyen d'affichage par un module de commande de jeu ; lesdits motifs de ligne de paiement étant formés par une sélection d'éléments d'une matrice de colonnes et de rangées, et le nombre d'éléments formant un quelconque motif de ligne de paiement étant supérieur au nombre de colonnes de ladite matrice.
Patent AU-2004203096-A1 (AU)
Title: Support assembly for output shaft of reciprocating power tool
Inventor: MILLION PHIL
IPC: B23D51/02
Filed: 2004-07-08
Abstract: A support assembly (62) for an output shaft (20) of a jigsaw is disclosed. The support assembly (62) comprises a support housing (64), a lower bearing (102) arranged in the support housing and adapted to support an output shaft (20) of the jigsaw for reciprocating movement of the output shaft along a first axis relative to the lower bearing and to substantially prevent movement of the output shaft (20) relative to the lower bearing (102) in a direction transverse to the first axis, and a blade support roller (110) adapted to abut a jigsaw blade (18). A support arm 108 supporting the blade support roller (110) is adapted to pivot to a limited extent relative to the lower bearing (102) about at least one second axis transverse to the first axis to minimise the extent to which a force applied by the jigsaw blade (18) to the blade support roller (110) during cutting action causes the lower bearing (102) to apply a turning moment to the output shaft (20) about an axis transverse to the first axis. <IMAGE>
Patent AU-2004239252-A1 (AU)
Title: Excess flow shutoff
Inventor: DWIGHT N JOHNSON
IPC: F16K17/34
Filed: 2004-05-05
Abstract: A flexible connector incorporates an excess flow shutoff at its inlet to prevent uncontrolled flow in the event of a failure such as rupture or separation of the connector. A shutoff sleeve moves in a body between an upstream, open position and a downstream, closed position. A spring biases the shutoff sleeve toward the open position. The sleeve includes a flow metering passage, and a pressure drop resulting from excess flow through the passage moves the sleeve to the closed position against a shutoff seat. A time delay is provided by a damping system including a variable volume damper chamber defined in part by a flexible bladder. Upstream pressure is communicated to the damper chamber by a restricted flow passage provided by metal to metal contact of a washer against a body surface.
Patent WO-2005119462-A1 (WO)
Title: Dispositif multiniveau de transfert securise d'informations
Inventor: DREWER PETER
IPC: G06F13/00
Filed: 2005-05-31
Abstract: La présente invention se rapporte à un système de diffusion d'informations permettant de diffuser sélectivement des informations depuis un réseau informatique vers au moins un autre réseau informatique de classification inférieure. Ce système possède un certain nombre de configurations possibles dont l'une inclut un dispositif de diffusion d'informations connecté audit réseau informatique, ce dispositif de diffusion d'informations comportant une unité de traitement pouvant répondre à une commande utilisateur pour sélectionner les informations à diffuser; au moins une entrée pour informations pouvant être commandée par l'unité de traitement de manière à recevoir les informations provenant d'un ordinateur et/ou d'un dispositif d'entrée d'ordinateur commandé par un usager; au moins une sortie d'informations pouvant être commandée par l'unité de traitement pour délivrer en sortie des informations à afficher à l'intérieur dudit réseau informatique; au moins une autre sortie pour informations pouvant être commandée par l'unité de traitement de manière à délivrer en sortie des informations, lesdites informations à délivrer en sortie devant au moins être communiquées à l'intérieur dudit réseau informatique aux fins d'un traitement ultérieur et renvoyées pour affichage; ou devant être diffusées directement à partir dudit réseau informatique à l'intérieur duquel le dispositif de diffusion est situé et à destination d'un autre réseau informatique; ou devant être communiquées à l'intérieur du réseau informatique aux fins d'un traitement ultérieur et diffusées vers l'autre réseau; dans ce système, les actions sont déterminées par l'unité de traitement et des actions prédéterminées sont possibles si et seulement si un utilisateur du dispositif de diffusion d'informations commande à l'unité de traitement de diffuser sélectivement des informations à l'autre réseau. Ce système implique également l'utilisation de sentinelles de diffusion d'informations permettant de diffuser des informations à d'autres réseaux et d'autres dispositifs du type serveurs de quarantaine permettant de traiter les informations et de délivrer des versions mieux adaptées à la diffusion, des serveurs d'audit permettant d'enregistrer les opérations du système et des serveurs de stadification permettant de délivrer à partir dudit réseau des informations qui peuvent être demandées par les autres réseaux.
Patent AU-2005246538-A1 (AU)
Title: Supporting a switch between audio coder modes
Inventor: OJALA PASI
IPC: G10L19/14
Filed: 2005-04-15
Abstract: The invention relates to a method for supporting an encoding of an audio signal, wherein a first coder mode and a second coder mode are available for encoding a respective section of an audio signal. The second coder mode enables a coding of a respective section based on a first coding model, which requires for an encoding of a respective section only information from the section itself, and based on a second coding model, which requires for an encoding of a respective section in addition an overlap signal with information from a preceding section. After a switch from the first coder mode to the second coder mode, always the first coding model is used for encoding a first section of the audio signal. This section can then be employed to generate an artificial overlap signal for a subsequent section, which is possibly to be encoded with the second coding model.
Patent AU-2005260057-A1 (AU)
Title: Nonwoven-elastomeric laminate with improved bonding between elastomer and nonwoven web
Inventor: HUANG ZHISONG
IPC: B32B27/04
Filed: 2005-06-28
Abstract: In one embodiment, the present invention relates to an extrusion bonded laminate including an elastomeric film directly bonded to at least one nonwoven web layer substantially continuously over at least a major portion of the laminate, in which the laminate is extensible in at least one direction, and in which the elastomeric film includes a vinyl arene-containing block copolymer, and in which the elastomeric film is substantially free of a tackifying amount of a tackifier, and to a process for producing an extrusion bonded laminate. In one embodiment, the total vinyl arene content of the elastomeric film is about 30% or less. The extrusion bonded laminate is useful, for example, in a diaper tab.
Patent AU-2005281513-A1 (AU)
Title: Container cover and dispenser therefor
Inventor: EDMUNDS MELISSA
IPC: B65D41/22
Filed: 2005-09-08
Abstract: A container cover prevents spillage of contents. In one embodiment, the container cover includes a flexible body having a first portion that can be stretched over a mouth of a container. The container cover also includes a second portion providing a periphery around the first portion that can contract against the sides of a container on which the container cover is placed to hold the cover in position. The first portion when stretched over the mouth of the container has an extension forming an area of slack for the container cover to allow the container cover to expand as a result of increased pressure within the container. The container cover further includes the first portion also including an aperture to receive a tube for withdrawing contents from the container. The first portion of the container cover includes a venting system. The venting system is provided by a valve.
Patent AU-2005293821-A1 (AU)
Title: N,N'-dithenylurea derivatives used in the form of kinase inhibitors
Inventor: STAEHLE WOLFGANG
IPC: A61P35/00
Filed: 2005-10-04
Abstract: Compounds of the formula (I), in which R1a-R1e, R2a, R2b, R3 and R5 have the meanings indicated in claim 1, are inhibitors of tyrosine kinases, in particular TIE-2, and Raf kinases and can be employed, inter alia, for the treatment of tumors.
Patent AU-2005307902-A1 (AU)
Title: Training apparatus
Inventor: PLANKE TORE
IPC: A61H1/02
Filed: 2005-11-24
Abstract: A device for use with an exercise apparatus consisting of at least one hanging, length-adjustable and lockable rope (10, 11) which at its lower end has a gripping means (13, 14), e.g., a gripping loop. A vibration means (12; 16) is designed, when attached via a rope engaging member (8, 9) to a portion of such rope, to impart to the rope and thus its gripping means (13, 14) a vibratory motion.