baber/WOPTO huggingface dataset:
Patent PT-1462442-E (PT)
Title: Crystals of bicalutamide and process for their production
Inventor: SHINTAKU TETSUYA
IPC: C07C317/26
Filed: 2002-12-13
Abstract: The present invention relates to a crystal of bicalutamide having a defined form, as well as economical and industrially practical production methods of bicalutamide and a crystal thereof, which are superior in environmental benignity and safety. <??>Accordingly, the present invention provides a production method of bicalutamide represented by the formula (I): <CHEM> which includes at least a step of reacting a compound represented by the formula (3): <CHEM> with an oxidizing agent, a production method of a crystal of bicalutamide, as well as a crystal form of bicalutamide as defined by X-ray diffraction (XRD) or solid <13>C NMR measurement. <IMAGE>
Patent PT-1599468-E (PT)
Title: 1,2,3-trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto such as diabetes and hyperglycemia
Inventor: SEMPLE GRAEME
IPC: C07D417/14
Filed: 2004-01-14
Abstract: The present invention relates to certain 1,2,3-trisubstituted aryl and heteroaryl derivatives of Formula (Ia) that are modulators of metabolism. Accordingly, compounds of the present invention are useful in the prophylaxis or treatment of metabolic disorders and complications thereof, such as, diabetes and obesity.
Patent PT-1730920-E (PT)
Title: Set of equipment for secure direct information transfer over the internet
Inventor: JOBBAGY MIKLOS
IPC: H04L29/06
Filed: 2004-11-02
Abstract: A set of equipment for secure direct information transfer over the Internet contains information transmitting terminal devices for collaborating with an information forwarding network, taking part in the information traffic. The individual information transmitting terminal devices are equipped with a sender partial unit, a receiver partial unit and a storage partial unit comprising an ID-register containing a device identification signal, a C-register for storing a coding key and a D-register for storing a decoding key. The C-register containing the coding key is connected to the sender partial unit, and a coding key and a collaborating decoding key are allocated to each individual information transmitting terminal device.
Patent PT-1570964-E (PT)
Title: Planer & thicknesser
Inventor: BETTACCHINI MARCELLO
IPC: B27C1/06
Filed: 2005-01-28
Abstract: A planer and thicknesser comprising a frame having a passage way which extends through the frame from one aperture in a wall of the frame to another aperture in a wall of the frame; an upper table having a front and rear sections (14,16) mounted on the frame in such a manner in order to form a slot between the front and rear sections of the upper table; a cutting drum (24) rotatably mounted within the frame such that an upper lengthwise section of the periphery of the cutting drum projects upwardly through the slot and a lower lengthwise section of the periphery of the cutting drum projects downwardly into the passage way; a lower table, substantially parallel to the upper table, mounted either within the passageway or forms the base of the passageway, below the cutting drum; and a dust extractor (250,254,256);  characterised in that  the dust extractor is capable of being connected to the underside of the upper table when the upper table is being used ( Fig. 20 ) and being connected to top of the upper table when the lower table is being used ( Fig. 19 ).
Patent PT-1637098-E (PT)
Title: Lower leg orthosis
Inventor: GUENTHER NORBERT G
IPC: A61F5/01
Filed: 2002-04-23
Abstract: The lower leg (4) is enclosed in a sleeve (2) which, together with a support spring (22) is linked to a foot-sleeve (6). The flexure of the support spring towards the foot-sleeve is restricted by a wedge-shaped thrust piece (32) which is detachably fixed to the rear end side of the foot-sleeve or to the support spring. No contact is made between a heel part or lower-leg side part of the support spring and the rear end side of the foot-sleeve in a resting position.
Patent PT-1776091-E (PT)
Title: Ocular implant made by a double extrusion process
Inventor: SHIAH JANE GUO
IPC: A61K9/20
Filed: 2005-07-25
Abstract: A bioerodible implant for treating an ocular condition comprises an active agent dispersed within a biodegradable polymer matrix, wherein at least about 75% of the particles of the active agent have a diameter of less than about 10 µm.
Patent PT-640587-E (PT)
Inventor: KLEEMANN HEINZ-WERNER
IPC: A61K31/185
Filed: 1994-08-18
Abstract: Benzoyl-guanidine derivatives (III) are new. (III) are of formula X2-CO-N=C(NH2)2 X2 = R101 = hydrogen, fluoro, chloro, hydroxy, amino or trifluoromethyl; R102 = hydrogen, fluoro, chloro, bromo, cyano, CqF2qCF3, R13SO2, R14R15NCO, R16CO or R17R18NSO2; R13, R14, R16 and R17 = 1-8C alkyl, 3-4C alkenyl, CnH2n-R20, trifluoromethyl or, except for R13, hydrogen; n = 0 or 1; q = 1-5; R20 = 3-6C cycloalkyl or phenyl, optionally substituted by 1-2 of fluoro, chloro, trifluoromethyl, methyl, methoxy or NR21R22; R21 and R22 = hydrogen or methyl; R104 = 1-8C alkyl, CnH2nR20, trifluoromethyl, (iso)quinolyl, pyrrolyl, pyridyl or imidazolyl (all these rings bonded via carbon or nitrogen and optionally substituted by 1 or 2 fluoro, chloro, trifluoromethyl, methoxy, hydroxy or amino (optionally substituted by 1 or 2 methyl)), R87SO2, R88R89NSO2, or R93-ethynyl; R87 = 1-4C alkyl or trifluoromethyl; R88 = hydrogen, 1-4C alkyl, trifluoromethyl, or (CH2)anR90; an = 0 or 1; R90 and R93 = phenyl, optionally substituted as in R20; R103 = any of a wide range of substituents . The full definitions are given in the DEFINITIONS (Full Definitions) Field.
Patent PT-687291-E (PT)
Inventor: VOGEL ALICE MARIE
IPC: C11D1/62
Filed: 1994-02-23
Abstract: The present invention relates to softening compounds; stable, homogeneous, preferably concentrated, aqueous liquid and solid textile treatment compositions; and intermediate compositions and/or processes for making said compositions. The compositions of the present invention contain diester quaternary ammonium compounds wherein the fatty acyl groups have an Iodine Value of from greater than about 5 to less than about 100, a cis/trans isomer weight ratio of greater than about 30/70 when the Iodine Value is less than about 25, the level of unsaturation being less than about 65% by weight, wherein said compounds are capable of forming concentrated aqueous compositions with concentrations greater than about 13% by weight at an Iodine Value of greater than about 10 without viscosity modifiers other than normal polar organic solvents present in the raw material of the compound or added electrolyte.
Patent PT-705255-E (PT)
Inventor: SZEJTLI JOSZEF
IPC: C07D295/30
Filed: 1995-04-25
Abstract: PCT No. PCT/HU95/00011 Sec. 371 Date Apr. 16, 1996 Sec. 102(e) Date Apr. 16, 1996 PCT Filed Apr. 25, 1995 PCT Pub. No. WO95/29172 PCT Pub. Date Nov. 2, 1995New inclusion complexes which are stable in their so-lid state formed of SIN-1A and cyclodextrins or cyclodextrin derivatives and optionally also containing ions as catalyst or stabilizer. The complexes release nitric oxide at room temperature upon dissolving in water or aqueous systems. The ions are preferably carboxylic acid anions such as acetate, formiate, propionate, ascorbinate, tartarate and/or lactate and/or inorganic acid anions such as phosphate, phosphite, borate, carbonate, hydrocarbonate, sulfate, sulfite and/or cations such as alkali and/or ammonium. Pharmaceutical compositions as well as kits containing the complexes. The kits are to be used as NO-liberating standards to release NO in a predictable amount and rate on dissolving in aqueous media. Processes for the preparation of the complexes by subjecting at a suitable pH SIN-1 to the catalytic action of ions to shift the equilibrium towards formation of SIN-1A in the presence of cyclodextrins or cyclodextrin derivatives capable to form inclusion complexes, whereby the SIN-1A formed is immediately complexed and stabilized and isolating in the solid state the obtained new complexes optionally containing ions. A preferred process includes reacting SIN-1 and a cyclodextrin or cyclodextrin derivative in the solid state in the presence of a salt as a catalyst by thoroughly admixing or milling the components together or by freeze drying an aqueous, oxygen-free solution containing the components, followed preferably by "second drying" in vacuo.
Patent PT-805796-E (PT)
Inventor: ADAMS STEVEN P
IPC: A61K31/00
Filed: 1996-01-18
Abstract: The present invention relates to novel compounds that are useful for inhibition and prevention of cell adhesion and cell adhesion-mediated pathologies. This invention also relates to pharmaceutical formulations comprising these compounds and methods of using them for inhibition and prevention of cell adhesion and cell adhesion-mediated pathologies. The compounds and pharmaceutical compositions of this invention can be used as therapeutic or prophylactic agents. They are particularly well-suited for treatment of many inflammatory and autoimmune diseases.
Patent PT-861228-E (PT)
Inventor: BYK GERARDO
IPC: C12N15/87
Filed: 1996-11-08
Abstract: Lipopolyamines useful for the transfection of nucleic acid and methods of preparation thereof are disclosed. The lipopolyamines are of general formula I, in which R4 comprises at least one C10-C22 aliphatic radical.
Patent PT-818270-E (PT)
Inventor: OBRIST BASIL
IPC: B23Q3/06
Filed: 1997-06-02
Abstract: The tension device has a coupling element (1) facing the item being clamped and a locally fixed tension element. The coupling element has grooves (13) which for fine-centring and determining the position in the X and/or Y direction interact with centring pins on the tension element. The tension bolt required for mutual fixing of the two elements is mounted on the tension element. The coupling element has a support member (11) projecting over the fine centring parts in order to protect these parts. The inside of the support member corresponds to the outer contour of the locally fixed coupling element.
Patent PT-951374-E (PT)
Inventor: BISHOP IAN H
IPC: B22F3/10
Filed: 1998-01-06
Abstract: The invention relates to a method of removing water-insoluble binder from a porous article formed from pressed particulate material, such as tantalum powder. The invention provides a method capable of removing substantially all of the binder from the article for high purity applications, such as capacitor manufacture. The method comprises contacting the article with an aqueous solution of an agent which reacts with said binder to produce a water soluble derivative thereof whereby said binder derivative may be substantially dissolved in said solution. In a particular embodiment, the derivative is produced by hydrolysis of a fatty acid binder.
Patent PT-1036192-E (PT)
Inventor: EPPS DENNIS E
IPC: G01N33/68
Filed: 1998-12-02
Abstract: The invention relates to novel fluorescence-based assays for protein kinases and phosphatases which can be used in high throughput screening. The methods of the invention utilize a competitive immunoassay to determine the amount of substrate that is phosphorylated or dephosphorylated during the course of a kinase or phosphatase reaction to yield a product, as well as the phosphorylating or dephosphorylating activity of a kinase or phosphatase.
Patent PT-945430-E (PT)
Inventor: BERNARD BALMER DR
IPC: C07C235/80
Filed: 1999-03-11
Abstract: Solid melts of acetoacetic acid aryl amide derivatives (I) are new. The melts contain 5-15 wt. % water. Solid melts of acetoacetic acid aryl amide derivatives of formula (I) are new. The melts are ready to use industrially and contain 5-15 wt. % water. R = H or one or more substituents selected from alkyl, alkoxy or halo. An Independent claim is also included for preparation of (I).
Patent PT-1086912-E (PT)
Inventor: PIRENEI ALESSANDRO
IPC: B65G47/82
Filed: 1999-09-22
Abstract: Herein described is a method for the planar transfer of groups of products in general, from a first (S) to a substantially coplanar second (A) position, without altering the original configuration-arrangement of the said groups, where the formation of a rigid cast for each group G present in the first position (S) takes place, followed by planar transfer of this rigid cast to the other position (A), where the products are then released. <IMAGE>
Patent PT-1060353-E (PT)
Inventor: RYLEWSKI EUGENIUSZ
IPC: F24J2/40
Filed: 1999-02-26
Abstract: A device for transferring heat between a panel heated by solar radiation and a wall surface, including an insulating plate mounted parallel between the panel and the wall surface, to define a closed external space between the panel and the insulating plate, and a closed internal space between the insulating plate and the wall. An air circulator is interposed between the external space and the internal space and can be put selectively in an open state allowing circulation of air between the external space and the internal space, and thus allowing thermal transfer between the panel and the wall, and a closed state preventing circulation of air between the external space and the internal space, and thus preventing thermal transfer between the panel and the wall.
Patent PT-1137595-E (PT)
Title: Novel rheology regulators such as ground natural calcium carbonates optionally treated with a fatty acid or salt and their use
Inventor: LOMAN HENNY DI
IPC: C08K3/00
Filed: 1999-10-01
Abstract: The invention relates to the selection of a natural calcium carbonate crushed to a high degree of fineness, possibly treated with one or more fatty acids or one or more of their salts or mixtures thereof, and its use as a rheology regulator for polymeric compositions. The specific surface area is 14 to 30 m2/g measured according to the BET method to ISO 4652, and the oil absorption is greater than 16 measured according to ISO 787-V (Rub-out method). The conditions of mixing of the constituents and manufacture are improved, as well as the properties of the final product.
Patent PT-1046147-E (PT)
Inventor: RUTTER NICHOLAS ALEXANDER
IPC: G01N27/00
Filed: 1999-10-07
Abstract: Provided is an alarm for detecting radiation, smoke and/or other air pollutants and includes detection means, first means for connection to a light fitting, and second means for connection to a light source. Electrical connection means connects the first means and the second means to enable the light source to be powered from the light fitting. In addition, a battery powers the alarm during periods of non-use of the light source, and isolating means thermally isolates the detection means from at least one of the electrical connection means, the light fitting and the light source.
Patent PT-1117636-E (PT)
Inventor: KEIL MICHAEL
IPC: C07D317/28
Filed: 1999-09-16
Abstract: The present invention relates to a method for the production of trion-bis(oxime ether) derivatives of formula (I), wherein the substituents have the following meaning: R1, R3 represent unsubstituted, partially or totally halogenated C1-C6-alkyl or C3-C6-cycloalkyl; R2, R4 represent C1-C4-alkyl or a methyl substituted by C2-C4-alkenyl, C2-C4-alkinyl or phenyl and X represents oxygen or N-OH. The invention also relates to the intermediate products obtained with said method.
Patent PT-1128894-E (PT)
Inventor: HUMBLOT CEDRIC
IPC: B01D53/64
Filed: 1999-10-21
Abstract: The invention concerns a combined method for purifying fume contaminated by hydrogen chloride and heavy metals, rendering inert the heavy metals and upgrading the hydrogen chloride, which consists in: subjecting the fume (6) to a treatment, by dry or semi-humid process, with a basic reagent (8) comprising a soda compound; collecting from said treatment a solid residue (13) containing the heavy metals; dispersing the solid residue and a hydraulic binder (18) in water (20) to form an aqueous broth (21); and extracting from the broth the solid mass (28) which is eliminated, and an aqueous solution (29).
Patent IE-780082-L (IE)
Title: Connecting a flowline to a subsea station
IPC: F16L37/00
Filed: 1978-01-13
Abstract: An apparatus and method of connecting a flowline to a subsea station in which such a connection may be remotely controlled and the method employed is independent of water depth. A flowline connector apparatus which includes a receptacle connector supported by a subsea station and has its axis directed toward the approach of the flowline, an elongated connector mandrel on a proximate end of the flowline, a pulling means releasably connected to the subsea station adjacent the connector receptacle, and lock means on the receptacle for interlocking engagement with the mandrel to retain the mandrel in selected longitudinal position relative to the receptacle and with a connector end of the mandrel exposed inboardly thereof. A method of securing a flowline to a subsea station.
[US4133182A]
Patent IE-870218-L (IE)
Title: Stackable container
IPC: G11B23/02
Filed: 1987-01-28
Abstract: A stackable cassette container 11 including a sliding drawer 15 has a base with two side walls and a rear wall joining the side walls. A pair of guides are provided inwardly of the upper marginal edge of the side walls to fit a removeable lid with complementary guides to the container. A further pair of guides are provided on the underside of the base to facilitate stacking of containers by engagement of these guides with the guides on the upper marginal edge of the side walls of a like container after removal of the lid. Complementary snap locking lugs are provided on the underside of the base and on the upper marginal edge of the rearwall to releasably lock two engaged containers together. The snap locking lugs can be formed so that disengagement is prevented whilst the drawer of the uppermost container is in the closed position. <IMAGE>
[GB2185965A]
Patent IE-820246-L (IE)
Title: Electric fuse
IPC: H01H85/18
Filed: 1982-02-04
Abstract: The electric fuse comprises a porous filler and a combination of a pair of terminals mutually insulated except for one or more metallic fuse conductors. These conductors comprise two kinds of metal so arranged that the current from one terminal to the other will pass successively and alternately through the two kinds of metal, beginning and ending in the first kind of metal. The second metal has pronounced reductions in cross-section defining one or more fuse elements, and is particularly suited to withstand for a long time a temperature at a fuse element near the melting point without significant deterioration. The first metal is selected to provide favorable conditions for current interruption with the arc burning between foot-points on parts of said first metal. The electric fuse may be used under marginal conditions both in respect of the steady state operating current and of the operating voltage and provides with an extremely fast action and current limiting operation. Such operating conditions are generally associated with fuses used for the protection of semi-conductor devices.
[EP0059334A2]
Patent IE-32682-L (IE)
Title: Central heating boiler
IPC: F24H1/32
Filed: 1969-03-28
Abstract: 1,246,816. Sectional boilers. STREBELWERK G.m.b.H. 19 Dec., 1968 [15 Nov., 1968], No. 60460/68. Heading F4A. In a sectional fluid fuel fired central heating boiler having an axial combustion chamber 2, the return heating gas passages 14 . . . 20, communicating with the combustion chamber, and the forward heating gas passages 22 and 24, communicating with the flue gas collector 10, are bounded in the central boiler sections by inner and outer circumferentially extending water chambers 30 and 28 and connecting radial water channels 32. The two return passages 14 and 16 adjacent the water outlet connection bosses 34 and the two return passages 18 and 20 adjacent the water inlet connection bosses 26 are connected to the two forward passages 22 and 24 therebetween in the front section 6 of the boiler through the flow reversing chambers 13. Cleaning apertures 50, 52 and 56 are provided for the heating gas passages. Finned plates 42 may be mounted in the heating gas passages.
[GB1246816A]
Patent IE-820515-L (IE)
Title: Clamp
IPC: F16L33/10
Filed: 1982-03-08
Abstract: A clamp has a split ring with projections extending outwardly from shoulders on the ring. The projections converge towards each other outwardly of the ring and have grooves onto which a nut is threaded. This causes the projections to be moved towards each other thereby closing the gap in the ring, and tightening the clamp. The inward movement of the projections is facilitated by grooves in the shoulders. A rib and projections are provided on the radially inner surface of the ring to facilitate the gripping of a body clamped by the clamp. A strengthening rib and handles are provided on the radially outer surface of the ring. The clamp is simple and secure and can be manufactured cheaply from a plastics material.
[US4446605A]
Patent IE-34138-L (IE)
Title: Lumilysergic acid
IPC: C07D457/04
Filed: 1970-05-08
Abstract: 1,244,145. Lumilisergic acid derivatives. SOC. FARMACEUTICI ITALIA. 11 May, 1970 [13 May, 1969], No. 22631/70. Heading C2C. ' Lumilisergic acid derivative of formula wherein R is C 1-4 alkyl, are prepared by treating lysergic acid with an alcohol ROH in the presence of an inorganic acid and irradiating with light.
[GB1244145A]
Patent IE-42977-L (IE)
Title: Triaryl-piperidine methanols.
IPC: C07D211/52
Filed: 1976-04-15
Abstract: Novel compounds of the general formula (I)  and their acid addition salts, in which the substituents have the meaning given in Patent Claim 1, are prepared by reducing the corresponding acid amide compounds of the formula (II)  The novel compounds of the formula (I) and their salts are valuable anti-diarrhoea agents. They have only slight, if any, analgesic side-effects. (From US3998832 A) [FR2307530A1]
Patent IE-35400-L (IE)
Title: Tyres, tread pattern
IPC: B60C11/03
Filed: 1971-06-24
Abstract: 1360203 Pneumatic tyres DUNLOP HOLDINGS Ltd 28 June 1971 [3 July 1970] 32304/70 Heading B7C A pneumatic tyre, e.g. for a heavy vehicle, has a tread comprising tortuous, e.g. zig-zag, axial grooves 11 extending for a distance of between “ and ¢ of the total tread width T from each tread edge to define axial bars 18, and a pair of circumferential grooves 17, e.g. of zig-zag form as shown, of lesser depth than the grooves 11 and disposed one one each side of the tyre equator X-X, for each groove 17 the circumferential plane lying midway between the axially innermost and outermost extremities of the groove being located at a distance of between T/10 and T/4 from the nearer tread edge such that the grooves 17 divide the bars 18 and intersect each groove 11 between its ends, both the grooves 11 and 17 being 'wide', i.e. of sufficient width to remain open in the tread/ground contact patch in use. The tread may, as shown, also have axial zig-zag grooves 16 which are 'narrow', i.e. of such width as to close in the tread/ground contact patch in use, and there may be other 'wide' grooves in the tread in addition to those 11, 17. The grooves 17 may have a lesser depth adjacent their intersections with the grooves 11 than at points away from these intersections. Each zig-zag groove 11 may, as shown, have four limbs 12-15 whose respective inclinations to the tyre axis are' 10, 20, 25 and 55 degrees. The tyre may have a cross-ply carcass.
[GB1360203A]