baber/WOPTO huggingface dataset:
Patent ZA-83774-B (ZA)
Title: Substituted debenzodiazepinones,process for the preparation thereof and pharmaceutical compositions containing these compounds
Inventor: TRUMMLITZ GUENTER DR
IPC: C07F9/40
Filed: 1983-02-04
Abstract: The specification describes new substituted dibenzodiazepinones of formula    <IMAGE>  (I)  wherein R1 is hydrogen or chlorine atom and R is (1-methyl-4-piperidinyl)methyl, (1-methyl-1,2,5,6-tetrahydro-4-pyridinyl)methyl,1-methyl-1,2,5,6-tetra hydro-4-pyridinyl, (1-methyl-4-piperidinylidene)methyl,(2,3-dehydro-8-methyl-8-aza-bicycl o[3,2,1]oct-3-yl)-methyl, (8-methyl-8-aza-bicyclo[3,2,1]oct-3-ylidene)-methyl or an endo-or exo-(8-methyl-8-azabicyclo[3,2,1]oct-3-yl)methyl each being optionally substituted by one or two methyls on the heterocyclic ring, and the nontoxic, pharmaceutically acceptable acid addition salts thereof, processes for preparing them and pharmaceutical compositions containing these compounds. The compounds of formula I have an antiulcerative effect and an inhibitory effect on the secretion of gastric substances having anticholinergic activity, such as dryness of the mouth and mydriasis.
Patent ZA-93984-B (ZA)
Title: 3,5-substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic and medicament containing them.
Inventor: LANG FLORIAN
IPC: A61P15/00
Filed: 1993-02-12
Abstract: There are described benzoylguanidines of the formula I <IMAGE> where R(1) is equal to R(4)-SOm or R(5)R(6)N-SO2-, where R(4) and R(5) are equal to alk(en)yl, -CnH2n-R(7), and where R(7) is equal to cycloalkyl or phenyl, where R(5) also denotes H, R(6) is equal to H or C1-C4-alkyl, R(2) is hydrogen, halogen, alkyl, -O-(CH2)mCpF2p+1, -X-R(10), where X is equal to O, S, NR(11), R(10) is equal to H, (cyclo)alkyl(methyl), -CnH2n-R(12) where R(12) is equal to phenyl, R(3), inter alia, is defined as R(1),  and their pharmaceutically tolerable salts. The compounds I are prepared by reaction of compounds of the formula II <IMAGE> in which L represents a leaving group which can be easily substituted nucleophilically, with guanidine. Compounds I are outstandingly suitable as antiarrhythmic medicaments having a cardioprotective component for infarct prophylaxis and infract treatment and for the treatment of angina pectoris, where they also preventively inhibit or strongly decrease the pathophysiological processes during the formation of ischaemically induced damage. They are moreover distinguished by a strong inhibitory action on cell proliferation. They can therefore be used as antiatherosclerotics, agents against diabetic late complications, cancers, fibrotic disorders such as pulmonary fibrosis, fibrosis of the liver or fibrosis of the kidneys. They are effective inhibitors of the cellular sodium/protons antiporter (Na<+>/H<+> exchanger).
Patent ZA-95756-B (ZA)
Title: Macrocyclic difluorostatone derivatives useful as antiviral agents
Inventor: FARR ROBERT A
IPC: C07K5/03
Filed: 1995-01-31
Abstract: PCT No. PCT/US94/13711 Sec. 371 Date Sep. 9, 1996 Sec. 102(e) Date Sep. 9, 1996 PCT Filed Nov. 28, 1994 PCT Pub. No. WO95/21186 PCT Pub. Date Aug. 10, 1995The present invention provides novel macrocyclic difluorostatone derivatives which are useful as antiviral agents. More specifically, these novel compounds are useful as inhibitors of retroviral proteases required for replication, particularly the HIV-1 and HIV-2 viral proteases, in the prevention or treatment of infection by the human immunodeficiency virus (HIV), and in the treatment of consequent pathological conditions such as the acquired immunodeficiency syndrome (AIDS) in mammals capable of being infected with HIV virus.
Patent AT-398859-B (AT)
Inventor: ZEITSCHEK RUDOLF DIPL ING
IPC: G08B29/02
Filed: 1990-05-11
Granted: 1995-02-27
Abstract: A method and a circuit are described for indicating different input signal states, in which a signalling device is activated or de-activated continuously or intermittently. This happens in such a way that levels (U2, U3) are provided for intermittent operation which differ from the levels for continuous activation (U4) or de-activation (U1). <IMAGE>
Patent AT-401560-B (AT)
Title: Method for the production of a burner arrangement
IPC: F23D14/10
Filed: 1993-06-25
Granted: 1996-10-25
Abstract: Method for the production of a burner arrangement with a plurality of burner bars 1, with an over-ignition burner 3 and with a burner plate 20, the over-ignition burner 3 and the burner bars 1 being produced from sheet-metal blanks, of which the edges running in the longitudinal direction are connected to one another via an essentially radially projecting seam 11, and the seams 11 being inserted into slots 12 of the burner plate 20. <IMAGE>
Patent AT-408123-B (AT)
Title: Frame for a sliding door for dry interior work
IPC: E06B1/12
Filed: 1999-09-29
Granted: 2001-09-25
Abstract: The invention relates to a frame for a sliding door for dry interior work, in the case of which the door leaf can be displaced into a pocket between gypsum plasterboards. The invention is characterized in that the associated frame, as is known per se, comprises individual profile parts 11, 20, in that the lintel 20 and at least the pocket-side vertical frame part 11 are of two-part configuration in each case, and in that the pocket-side vertical frame parts 11 are fastened on the finished wall by means of link plates 14, which are pushed into or between the gypsum plasterboards 12, 13 and screwed thereto. <IMAGE>
Patent AT-396040-B (AT)
Title: Clock (time piece) with an electronic movement
IPC: G04G99/00
Filed: 1989-12-18
Granted: 1993-05-25
Abstract: The clock is connected to an optical display unit 2 and an acoustic unit 3 for reproducing visual or acoustic information which can be called up from a memory. The electronic movement is formed by a separate computer 7; 12 with an associated register array 13 for time program storage. The computer has 7;12 an interface for networking or for connection to a public data network 11, and also outputs for driving the optical display unit 2 and the acoustic unit 3. <IMAGE>
Patent DK-155793-B (DK)
Inventor: ARVIDSSON FOLKE LARS-ERIK
IPC: C07D207/08
Filed: 1981-07-31
Abstract: Compounds of the formula <CHEM> wherein Z<3> is R or R<6>CO, wherein R is an alkyl group having 1-5 carbon atoms, a hydroxyalkyl, dimethylaminoalkyl or methylthioalkyl group having 2-6 carbon atoms in the alkyl part and having the heteroatom bound in a position other than 1-position, an alkenyl group having 3-5 carbon atoms other than an 1-alkenyl group, and R<6> is an alkyl or alkoxy group containing 1-4 carbon atoms or an alkenyl group with 2-4 carbon atoms, R<7> is an alkyl group with 1-5 carbon atoms, an allyl or benzyl group, and n is 1 or 2 provided that Z<3> is other than methyl and ethyl when n is 2 and R<7> is CH3 or an acid addition salt thereof. The compounds are useful as intermediates or starting materials for preparation of therapeutically useful substituted phenyl-azacycloalkanes.
Patent FI-52051-B (FI)
Inventor: BOURGEOIS MICHEL
IPC: F17C3/02
Filed: 1971-09-02
Granted: 1977-02-28
Abstract: Methane tanker comprises two heat insulating barriers and two fluid-tight barriers, positioned alternately with a fluid-tight barrier innermost and the outermost insulating barrier attached to the hull of the ship. The other fluid-tight barrier is positioned between the two insulating barriers and comprises vertical plates joined together by welding to horizontal metallic strips. One edge of each strip is slidably connected to the outer insulating barrier and the other edge is resiliently connected to the inner insulating barrier.
Patent FI-75220-B (FI)
Inventor: OLSSON KARL BOERJE
IPC: F23R7/00
Filed: 1984-08-28
Granted: 1988-01-29
Abstract: The non-return valve in the air inlet of a pulsating burner includes a flat circular ring of elastic steel. The outer edge of the ring is provided between annular abutment surfaces with a predetermined play. The inner edge of the ring is movable from a closed position to a fully open position in which it has the shape of a truncated cone. The angle between the conical surface of the frustrum and its base is small in the fully open position, on the order of 3 DEG , and resistance to opening is extremely small to permit rapid changes between the open and closed positions.
Patent FI-83091-B (FI)
Inventor: BUSCHFELD ADOLF
IPC: C08G8/28
Filed: 1984-12-20
Granted: 1991-02-15
Abstract: 1. Process for producing modified phenolic resin bonding agents characterized by preparing as known per se phenol-formaldehyde resins with a viscosity of higher than 300 mPa.s (at 20 degrees C) with a solids content of 20 to 55% and adding to the viscous phenolic resin solutions 2 to 30 wt.-% urea, relative to the phenolic resin solution, the phenol-formaldehyde resins being prepared with as much alkali as is required to ensure that the modified resin solution resulting therefrom contains 2 to 12 wt.-% alkali (titrated, calculated as NaOH).
Patent FI-78800-B (FI)
Inventor: DANIELSEN GEIR
IPC: H05K9/00
Filed: 1985-05-23
Granted: 1989-05-31
Abstract: The invention relates to a flat pack or housing for a radio apparatus having a rectangular cross-section comprising an opening at the front side and an opening at the back side which are respectively closable with a cover and also relates to a support mount for the radio apparatus. Such a radio apparatus provides the user with the possibility of versatile use at various use locations and is securable in a receptacle. To this end, the housing is divided into two tub-shaped main chambers by a bottom plate oriented parallel to the plane of the openings. The individual assemblies of the radio apparatus are disposed RF-shielded in the main chambers and the main chambers being closed by the covers by means of a central screw. Outside guide rails for acceptance into the support mount are disposed at opposite lateral faces of the housing. The support mount is composed of a sheet metal panel bent at three sides. The lower, bent part of the panel forms a chamber with a further bent sheet metal part which carries contacting elements and further assemblies for additional functions of the radio apparatus are accommodated in said latter chamber. A carrying shackle pivotable by 90 DEG  is attached at the upper side of the radio apparatus. This carrying shackle provides a latching function when the radio apparatus is inserted in the support mount.
Patent FI-84783-B (FI)
Inventor: HARRISON PAUL JONATHAN
IPC: A61K9/52
Filed: 1985-06-04
Granted: 1991-10-15
Abstract: A pharmaceutical composition comprising a plurality of, beads constituting a unit dose of a solid steroid medicament enclosed in a gastric-juice soluble material, for example gelatin capsules. Each bead comprises finely divided discrete solid steroidal particles bound onto a particulate core by a binder soluble in water.
Patent FI-83989-B (FI)
Title: Arrangement for air control
Inventor: ANDERSSON THOMAS
IPC: B65G69/00
Filed: 1987-11-06
Granted: 1991-06-14
Abstract: The invention, the object of which is to provide a simple, reliable and inexpensively manufactured arrangement for air control, intended primarily for use in conjunction with inflatable sealing elements for loading bay openings and similar, is characterized essentially in that their discharges into an air chamber, such as that formed by the internal cavity in the sealing element in question, a large-section channel containing a damper (8) so arranged as to bring the inside of the air chamber into open communication with an inlet channel containing a fan (4), preferably of the low-pressure type, for the purpose of inflating the air chamber, and alternately with the atmosphere for the purpose of evacuating the air chamber, for which purpose the damper is controlled in such a way by the air flow of the fan that it is caused to change over to the position which interrupts the open communication between the inside of the air chamber and the atmosphere as the fan approaches its operating speed, in this way opening the communication via the fan for the purpose of inflating the air chamber, and vice versa, i.e. to change over to the position which opens up the communication between the air chamber and the atmosphere as the speed of the fan decreases.
Patent FI-85454-B (FI)
Inventor: KAERKKAEINEN AULIS
IPC: B63B35/73
Filed: 1991-01-14
Granted: 1992-01-15
Abstract: The object of the invention is a transportation device which consists of a cover (1, 2) made of an elastic fabric material with filling material placed inside it. The presently available devices, especially those intended for downhill sliding i.e. sledges, toboggans, sliders and so on are usually rigid and when sliding downhill one has to endure bumps etc. as the device goes over uneven ground. In the transportation device, according to the invention, the filling material is a granular-like material which at least partially is free to move around inside the transportation device and moulds to the shape of the user.
Patent FI-108428-B (FI)
Inventor: MANN HORST
IPC: B65D21/00
Filed: 1993-02-10
Granted: 2002-01-31
Abstract: A container, consisting of a hollow shaped body (1), in particular of plastic material,   - having an upper part (2) and a lower part (3) which can be separated to receive objects, - having end faces (7) which are arranged perpendicular to the longitudinal axis of said body, and of which in each case one has a projection (5) and the other has a cutout (15) in which the projection (5) of the one end face can be inserted to produce a releasable connection, and - having connecting means (4) on the circumference of at least one of the parts (2, 3) of the shaped body (1), is constructed for the purpose of bringing about sliding or plug-in connection possibilities in virtually any directions and for use as a plug-in module for a plurality of dimensions, in such a way   - that a projection (5) is provided in one of the end faces (7) which contains the cutout (15) to receive the projection (5) of the other one of the end faces (7), and - that recesses (4) and elevations (8) which alternate with one another are provided on the circumference of the at least one part (3) of the shaped body (1), by means of which recesses and elevations a sliding or plug-in connection can be produced, by engagement of at least one elevation (8) in at least one recess (4), on the circumference of different shaped bodies (1) in each case.   <IMAGE>
Patent FI-98388-B (FI)
Inventor: KINNUNEN JORMA
IPC: D21H23/70
Filed: 1993-11-29
Granted: 1997-02-28
Abstract: An apparatus to facilitate tail threading of a paper web and a method of threading the tail of a paper web (1) to be coated through a coating line during startup or web break, in which an edge strip is slit from the web to act as the tail of the web which is first threaded through the line and then widened to the normal width of the web by moving the edge strip slitter. Said edge strip is first guided to a movable support element (12) located after the edge strip slitting point in the travel direction of the web (1) and the strip is supported against said movable support element (12) and is passed supported by said movable support element (12) to the next support element (14). A guiding/auxiliary support element (31) is brought to the discontinuity points of web support path and the edge strip is passed with the help of said auxiliary support element over the discontinuity and the edge strip is passed through the entire coating line supported by said sequential support elements (2, 12, 14, 18, 19, 22, 25) and said guiding/auxiliary support elements (31).
Patent FI-113184-B (FI)
Inventor: ZABEAU MARC
IPC: C12Q1/6858
Filed: 1994-03-24
Granted: 2004-03-15
Abstract: The invention relates to a process for the controlled amplification of at least one part of a starting DNA containing a plurality of restriction sites for a determined specific restriction endonuclease, and of which at least part of its nucleic acid is unknown. Application of this process to human, animal or plant DNA fingerprinting, to identification of restriction fragment length polymorphisms. Kit for the application of the process.
Patent FI-108862-B (FI)
Inventor: FOGUET RAFAEL
IPC: A61K31/443
Filed: 1995-11-08
Granted: 2002-04-15
Abstract: PCT No. PCT/EP95/01007 Sec. 371 Date Feb. 20, 1996 Sec. 102(e) Date Feb. 20, 1996 PCT Filed Mar. 17, 1995 PCT Pub. No. WO95/25732 PCT Pub. Date Sep. 28, 1995The invention relates to new N-benzoylmethyl-piperidines of the general formula (I):    <IMAGE>  (I)  wherein X is a halogen atom, as well as their pharmaceutically acceptable addition salts. The compounds are potentially useful to treat depressions.
Patent FI-106417-B (FI)
Inventor: RUUTU JUSSI
IPC: H04L12/56
Filed: 1998-12-08
Granted: 2001-01-31
Abstract: The invention is related to optimization of data transmission in TCP/IP networks, particularly to problems created by transmission of encrypted traffic. According to the invention, an indication of a TCP ACK being carried in the encrypted payload of a IP datagram is added in the IP header of the datagram. The indication may simply be a flag indicating the presence of a TCP acknowledgment. The indication may also contain the acknowledgment number, which allows processing of the encrypted traffic based on the acknowledgment number. In IPv4 datagrams, the indication may be inserted as an extra option field. In IPv6 datagrams, the indication may be inserted as an extension header.
Patent HU-189449-B (HU)
Title: Device for melting and controlled feeding thermoplastic glues
Inventor: LEIBHARD ERICH
IPC: B05C5/04
Filed: 1980-04-24
Abstract: In a device for the melting and measured discharge of a thermoplastic adhesive, a sealing sleeve conveys the solid thermoplastic adhesive into the inlet end of a melting chamber. The sealing sleeve is formed of a temperature resistant, poor heat conductive material with good sliding properties, such as polytetrafluoroethylene. Further, the sealing sleeve is provided with slots extending in the axial direction of the sleeve from the end more remote from the melting chamber toward the melting chamber.
Patent HU-185379-B (HU)
Title: Process for the production of the nonapeptide and decapeptide derivatives of the luteotrope releasing factor
Inventor: NESTOR JOHN J
IPC: C07K14/00
Filed: 1980-06-10
Abstract: Nonapeptide and decapeptide analogs of LH-RH of the formula (pyro)Glu-His-V-Ser-W-X-Y-Arg-Pro-Z (I) and the pharmaceutically acceptable salts thereof wherein: V is tryptophyl, phenylalanyl or 3-(1-naphthyl)-L-alanyl; W is tyrosyl, phenylalanyl or 3-(1-pentafluorophenyl)-L-alanyl; X is a D-amino acid residue <IMAGE>   wherein R is (a) a carbocyclic aryl-containing radical selected from the group consisting of naphthyl, anthryl, fluorenyl, phenanthryl, biphenylyl, benzhydryl and phenyl substituted with three or more straight chain lower alkyl groups; or (b) a saturated carbocyclic radical selected from the group consisting of cyclohexyl substituted with three or more straight chain lower alkyl groups, perhydronaphthyl, perhydrobiphenylyl, perhydro-2,2-diphenylmethyl and adamantyl; Y is leucyl, isoleucyl, nor-leucyl or N-methyl-leucyl; Z is glycinamide or -NH-R1, wherein R1 is lower alkyl, cycloalkyl, fluoro lower alkyl or   <IMAGE>  wherein R2 is hydrogen or lower alkyl, are disclosed. These compounds exhibit potent LH-RH agonist properties.
Patent HU-195489-B (HU)
Inventor: BESZEDICS GYULA
IPC: C07D231/36
Filed: 1986-04-14
Abstract: A találmány tárgya eljárás 1,2-difenil-4-[(2-fenil-szu]finil)-etiI]-3,5-pirazolidindion előállítására 1,2-difenil-4-[(2-fenil-tio)-etil]-3,5-pirazoIidindionnak ecetsav jelenlétében végrehajtott hidrogén-peroxidos oxidáció- ja útján, amely abban áll, hogy az oxidációt katalizátorként használt, pK = 0-3 értékű sav jelenlétében alifás alkoholban, klórozott vagy aromás szénhidrogénben 0 °C és 20 °C közötti hőmérsékleten végzik. Az eljárással kapott termék, a szulfinpirazon értékes gyógyszerkészítmények hatóanyaga -1-
Patent HU-206643-B (HU)
Title: Method for gas-circulating regenerating zone of movable-bed catalyzer
Inventor: GREENWOOD ARTHUR RAYMOND
IPC: B01J38/12
Filed: 1986-04-24
Abstract: Particulate catalyst which has been used in a hydrocarbon conversion process such as catalytic reforming is regenerated in a moving bed regeneration zone (12). The catalyst being regenerated is passed into the top of the zone (12) and slowly moves downward as a dense bed (14, 19, 20) which is contacted successively with an oxygen-containing gas stream (31), a temperature-adjusting gas stream (30) and either a drying gas stream (37) or a chlorination gas stream (39) or both at different elevations within the regeneration zone (12). A key feature involves employing a portion of relatively hot combustion gas (26) withdrawn from one portion of the zone (12) as the temperature-adjusting gas stream (30) in a different portion of the zone after compression, with the remainder of the compressed combustion gas (27) being cooled (32) and recycled to the combustion zone as the gas stream (31). This eliminates the need to employ a heater to provide a suitable heating gas stream.
Patent HU-187719-B (HU)
Title: Method for making positive acivated material of the lead accumulatotrs
Inventor: HORVATH PAL
IPC: H01M4/56
Filed: 1982-06-02
Abstract: Method for the production of positive active material for lead storage batteries, this active material consists of PbO and PbOx - where x is a number between 1 and 2 - and some powder being composed of not more than 30 to 35% lead in optional rate and some water. The basis of the invention is mixing glycerine and polytetrafluorethylene, as addition, to the active material.
Patent HU-188046-B (HU)
Title: Method for disinfecting and curing raw hides
Inventor: MARGOLD FRANZ
IPC: C14C1/02
Filed: 1981-06-17
Abstract: Hides and skins are disinfected and preserved by contacting them with a mixture of an inorganic zinc salt and an acid amide and subsequently with common salt and an acid having a disinfectant and preservative action. The mixture of zinc salt and acid amide is used in general in an amount of at most 2 weight %. The efficiency of the mixture may be improved by using additionally a further organic preservative. Carboxylic acids are especially suitable for the aftertreatment using a salt-acid pickle. The process is particularly appropriate for preserving hides and skins as well as furskins of different kinds and provenance.
Patent HU-195349-B (HU)
Inventor: KOVACS KALMAN
IPC: G06F3/00
Filed: 1986-06-04
Abstract: A találmány kapcsolási elrendezés kétállapotú érzékelő és/vagy működtető elemek digitális számítógéphez való illesztésére, amely kapcsolási elrendezésnek az elemek érintkezőihez csatlakoztatható kontaktus figyelői (31 A, 31B) és a digitális számítógéphez csatlakoztatható állapotjelző kimenetei (29A, 29B) vannak. A találmány szerint egy-egy állapotjelző kimenet (29A, 29B) vagy egy kontaktus figyelő (31A, 31B) kimenetére,vagy annak egyik bemenetére (27A, 27B) van csatlakoztatva, továbbá az állapotjelző kimenetek (29A, 29B) első változás érzékelőkön (33A, 33B) keresztül logikai vagy-kapcsolatot megvalósító kapuáramkör (37) bemenetelhez vannak csatlakoztatva, amely kapuáramkör (37) kimenete a digitáüs számítógéphez csatlakoztató változásjelző kimenethez (41) van csatlakoztatva. 1*1 M* ΜβΟ, GOtFlffi  -1-
Patent HU-192232-B (HU)
Title: Process for producing 9-alpha,11-alpha epoxy-steroides and pharmaceutical compositions containing them
Inventor: BIOLLAZ MICHAEL
IPC: C07J71/00
Filed: 1985-06-20
Abstract: 7α-Acylthio-9α,11α-epoxy-20-spirox-4-en-3,21-dione der Formel I
     worin R ein Niederalkanoyl und -A-A- die Ethylen- oder Cyclopropylene-Gruppe ist, weisen eine hohe Aldosteron-antagonisierende Wirksamkeit ohne nennenswerte sexual-spezifische nebenwirkungen auf und sind als Kalium-sparende Dieuretika in der Therapie verschiedener Formen von Hyperaldosteronismus anwendbar. Die Verbindungen sind gemäss konventioneller Verfahren der Steroid-chemie erhältlich.