baber/WOPTO huggingface dataset:
Patent FI-882369-A0 (FI)
Inventor: SUGIMOTO HACHIRO
IPC: C07D211/70
Filed: 1988-05-19
Abstract: Heterocyclic amines of formula (I) and their salts are new: where A is (opt. substd.) phenyl or naphthyl, pyridyl, thienyl, tetralyl, quinolinyl, benzofuranyl, quinazolinyl, benzothienyl, 1,2,3,4-tetrahydro-2-quinolinyl or 1-oxo-1,2,3,4-tetrahydro -2-naphthyl; X is -CH2, -CO-, -CHOH-, -CHMe- or -CH(CH2NEt2)-; m is 1-3; n is 0-4; Y is C or N; Z is -CH2-, -CO-, -CHOR1-, -CHHal-, -CH=, or a group of formula (II), (III) or (IV); R1 is H, lower alkyl, acyl, aralkyl or heteroaralkyl, Hal is halogen; B is phenyl or naphthyl opt. substd. by one or two groups chosen from halogen, lower alkyl or lower alkoxy; Z-B may be bound at either of the positions starred on the ring.
Patent FI-895363-A0 (FI)
Inventor: LINDQUIST BJOERN KARL VALTER
IPC: B01D53/34
Filed: 1989-11-10
Abstract: The invention relates to a method for extracting dioxins and like highly toxic, organic contaminants from a gas. The invention is characterized by contacting the gas with a liquid aerosol over a pre-determined period of time, and by electrically charging the particles present in the aerosol, both solid and liquid particles, and subsequently separating the particles from the gas, preferably with the aid of a wet electrostatic precipitator.
Patent FI-903820-A0 (FI)
Inventor: EFFLAND RICHARD CHARLES
IPC: C07D401/14
Filed: 1990-07-31
Abstract: This invention relates to 2,3-dihydro-1-(pyridinylamino)-indoles of the formula <CHEM> wherein R1 is hydrogen, loweralkyl, aryl, arylloweralkyl, alkenyl, alkynyl or heteroarylloweralkyl selected from the group consisting of pyridinylmethyl, pyridinylethyl, thienylmethyl, thienylethyl; R2 and R3 are independently hydrogen, loweralkyl, aryl, arylloweralkyl or heteroarylloweralkyl selected from the group consisting of pyridinylmethyl, pyridinylethyl, thienylmethyl, thienylethyl; or R2 and R3 together form a cycloalkane ring of 4 to 6 carbons or a spiro-fused aryl or heteroaryl cycloalkane; X and Y are independently hydrogen, halogen, hydroxy, loweralkyl, loweralkoxy, nitro, amino or trifluoromethyl; m and n are independently integers of 1 to 3, the pharmaceutically acceptable acid addition salts thereof and where appropriate, the optical, geometrical and stereoisomers and racemic mixtures thereof. The compounds of this invention are useful as analgesics, anticonvulsants, for enhancing memory and for the treatment of Alzheimer's disease.
Patent FI-905743-A0 (FI)
Inventor: M LARRECQ MICHEL
IPC: B22D11/06
Filed: 1990-11-21
Abstract: Device for continuous casting of thin metal strips (6) between two parallel rotating rolls (2), comprising lateral faces at the ends of the rolls defining, with the rolls, the casting space for the molten metal (1), characterised in that it comprises a flat cover (7), arranged above the molten metal (1) and in the immediate vicinity of its meniscus in order to form a thermal screen which is of a size so as to cover over the entire surface of the molten metal, this cover (7) being provided with a refractory coating (8) on its face which is turned towards the molten metal and bearing on the two rolls (2). This cover forms a thermal shield or screen preventing any incipient surface solidification of the bath of molten metal (1). Advantageously, an inert gas may be injected between the meniscus (4) and the cover (7) through the latter. 
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Patent FI-911245-A0 (FI)
Inventor: KLUSER REMO
IPC: F16D37/02
Filed: 1991-03-13
Abstract: PCT No. PCT/EP90/00853 Sec. 371 Date May 13, 1991 Sec. 102(e) Date May 13, 1991 PCT Filed May 28, 1990 PCT Pub. No. WO91/01420 PCT Pub. Date Feb. 7, 1991.Fastening element for mounting insulating strips or plates on a solid structure includes a large-surface washer, a tubular extension and a locking member which is mounted to an end portion of the fastener and protrudes into the extension so that the fastener and the tubular extension form two telescopic elements movable relative to each other. The two telescopic elements can be adjusted and locked relative to each other in a desired position due to the provision of interengaging ribs, grooves or corrugations formed on the telescopic elements.
Patent FI-913254-A0 (FI)
Inventor: WIESCHOLLEK RAPHAEL
IPC: A01N25/14
Filed: 1991-07-04
Abstract: The invention relates to novel ready-for-use formulations of the known herbicidal active substances metamitron (I) + ethofumesate (II) +  (A) phenmedipham (III) or  (B) phenmedipham (III) and desmedipham (IV) or  (C) desmidipham (IV), preferably solid formulations such as water-dispersible powders (WP) or water-dispersible granules (WG), the ratio by weight of the active substances (I):(II):(III) or (IV) being (1):(0.05 to 1):(0.05 to 1), that of the active substances (I):(II):(III):(IV) being (1):(0.05 to 1):(0.05 to 1):(0.05 to 1), and the total active substance content in each case being between 20 and 75% by weight, and to their use as herbicides, in particular as selective herbicides in beet.
Patent FI-931644-A0 (FI)
Inventor: BAECKERUD STIG LENNART
IPC: G01N33/20
Filed: 1993-04-13
Abstract: PCT No. PCT/SE91/00686 Sec. 371 Date Apr. 15, 1993 Sec. 102(e) Date Apr. 15, 1993 PCT Filed Oct. 11, 1991 PCT Pub. No. WO92/06810 PCT Pub. Date Apr. 30, 1992.During production of ductile cast iron, controlling and correcting the composition of the cast iron melt, including extracting a sample from the melt, the mother melt, and adding an amount of an oxide, a sulphite or an oxy-sulphide with the ability to oxidize an amount of the modifying agent present in the sample and corresponding to the fading rate expected to occur during the casting process as a whole. The sample is permitted to solidify in a sample vessel equipped with two thermocouples, one in the center of the sample vessel and the other in the vicinity of the sample vessel wall. The temperature and time are recorded during the process of solidification in a manner known per se and nodularity is calculated. If the amount of modifying agent is too low to secure a fully nodular graphite throughout the whole casting period, an appropriate amount of modifying agent is added.
Patent FI-943262-A0 (FI)
Inventor: HUMM SIEGFRIED
IPC: G09F15/00
Filed: 1994-07-08
Abstract: A device for holding a sign or the like on a motor vehicle contains a plate-shaped support, which can be fastened to the motor vehicle, and has a space for the sign to be held. Attached to the frame is at least one frame element which has a release position making it possible to insert and/or remove the sign and, in cooperation with the support, has a locking position which prevents the insertion and/or removal of the sign. <IMAGE>
Patent FI-943721-A0 (FI)
Inventor: KIRJAVAINEN KARI
IPC: B29C71/00
Filed: 1994-08-12
Abstract: Film of dielectric material, self-adhesive by virtue of an electrostatic force, which film contains gas blisters preferably of a flat shape. To achieve an adhesive quality of the film, the film is given a large internal unipolar charge, which is created by charging the film by means of an electric field intensive enough to produce partial discharges in the gas blisters and to cause the charges to move into the dielectric material of the film.
Patent FI-951134-A0 (FI)
Inventor: DORAN THOMAS I
IPC: A61K31/593
Filed: 1995-03-10
Abstract: This invention is for 1α-fluoro-25-hydroxy-16-ene-23-yne-cholecalciferol, which can be further characterized by the formula:and which is useful as an agent for the treatment of sebaceous gland diseases such as acne and sebhorreic dermatitis. It can be prepared by removing the silyl protecting groups from a corresponding compound with silyl protected hydroxy groups.
Patent FI-956330-A0 (FI)
Inventor: PERRAUD ERIC
IPC: C09D5/03
Filed: 1995-12-29
Abstract: PCT No. PCT/FR94/00804 Sec. 371 Date May 31, 1996 Sec. 102(e) Date May 31, 1996 PCT Filed Jun. 30, 1994 PCT Pub. No. WO95/01403 PCT Pub. Date Jan. 12, 1995The invention relates to a mixture in powder form and comprising (i) at least one polyamide and (ii) at least one polymer (A) containing hydroxyl functional groups and compatible with the polyamide. The polymer (A) may be an ethylene/vinyl alcohol copolymer. The mixture may be used to coat metal substrates.
Patent FI-956360-A0 (FI)
Inventor: PIIRAINEN OLLI
IPC: H04J3/00
Filed: 1995-12-29
Abstract: PCT No. PCT/FI96/00697 Sec. 371 Date Jun. 26, 1998 Sec. 102(e) Date Jun. 26, 1998 PCT Filed Dec. 23, 1996 PCT Pub. No. WO97/24819 PCT Pub. Date Jul. 10, 1997A method of detecting a call set-up burst, and a receiver, in a digital radio system, the receiver comprising a converter (304) for sampling a signal received in a given time slot, means (400) for correlating digitalized samples with a known training sequence, and means (402) for computing the energy of the correlation results obtained, means (404) for looking for the maximum values of a string of samples of a given order from the computed energies, and means (408) for averaging the maximum values found per one sample. To improve reliability of detecting a call set-up burst, the receiver comprises means (410) for averaging the energy of the other samples of the time slot per one sample, and means (412) for comparing the averaged maximum energy values with the energy values of the other samples.
Patent FI-972628-A0 (FI)
Inventor: BREU VOLKER
IPC: C07D239/46
Filed: 1997-06-18
Abstract: PCT No. PCT/EP95/04843 Sec. 371 Date Aug. 15, 1997 Sec. 102(e) Date Aug. 15, 1997 PCT Filed Dec. 8, 1995 PCT Pub. No. WO96/19459 PCT Pub. Date Jun. 27, 1996Compounds of the formula: where A, B, R1-R8 are as described herein are endothelin inhibitors that can be used in treating diseases associated with endothelin, such as high blood pressure. Chemical synthesis of these compounds and pharmaceutical compositions containing these compounds are also useful.
Patent FI-972856-A0 (FI)
Inventor: JUNTTILA JAAKKO
IPC: F16K31/50
Filed: 1997-07-04
Abstract: A control device, e.g. for a door closer provided with a body part (10) and whose operation is controlled by a pressure medium, comprising a screw-threaded adjustment member (1) screw-threadedly engageable in an opening in the body part (10) and a separate substantially hollow control member (2) which in use is arranged to restrict when necessary the flow of the pressure medium. Turning of the adjustment member (1) with respect to the body part (10), brings about movement of the control member (2) in the axial direction of the control device for providing the desired control. The control member (2) is arranged to be attachable to and detachable from the adjustment member (1) in the radial direction and movement of the control member (2) with respect to the adjustment member (1) in the axial direction is prevented. <IMAGE>
Patent FI-974387-A0 (FI)
Inventor: ENWALD PETRI
IPC: B65H19/22
Filed: 1997-12-01
Abstract: A change device of a reel-up in placed in the reel-up of a paper web in connection with the reel spool (2) forming the core of a new roll and located against the web (W) running onto the old roll (R). The change device comprises a guiding device (3) which is provided with nozzles or the like which are positioned and directed with respect to the reel spool (2) in such a way that they direct air jets (S) to the new end of the web following the cut-off point of the web (W) substantially over the full width of the web, to guide the web around the reel spool (2).
Patent FI-990113-A0 (FI)
Inventor: KINNI JOUNI
IPC: F23C10/20
Filed: 1999-01-21
Abstract: A method for adjusting a supply of gaseous medium to a fluidized bed boiler performing a combustion process and including a pipe grate comprising a plurality of pipes. An active area of the pipe grate is adjusted to form at least one inactive bed area that is out of use by shutting off the supply of gaseous medium to some of the pipes of the pipe grate utilizing pipe-specific control means included in at least some of the pipes of the pipe grate. Cooling medium is conducted through cooling channels located in the pipes in the at least one inactive bed area at least during the combustion process.
Patent IL-65166-A0 (IL)
Title: Triazolylalkyl-thioethers,their preparation and their use as plant growth regulators and fungicides
IPC: A01N43/653
Filed: 1982-03-04
Abstract: Triazolylalkyl-thioether plant growth regulators and fungicides of the formula   <IMAGE>   in which A represents the keto group or the CH(OH) group, R1 represents alkyl, alkenyl, alkynyl, optionally substituted cycloalkyl, alkylaminoalkyl, alkoxycarbonylalkyl, optionally substituted phenyl or optionally substituted phenylalkyl, R2 represents alkyl, R3 represents alkyl or halogenoalkyl, R4 represents alkyl, halogenoalkyl, alkoxy, alkoxymethyl, alkylthio, alkylthiomethyl, optionally substituted phenyl, optionally substituted benzyl, optionally substituted phenoxy, optionally substituted phenoxymethyl, optionally substituted phenylthio, optionally substituted phenylthiomethyl, alkenyl, alkoxycarbonyl or cyano, or R3 and R4, conjointly with the carbon atom to which they are bonded, represent optionally substituted cycloalkyl and X1, X2, X3, X4 and X5 are selected independently and each represent hydrogen, hologen, alkyl, halogenoalkyl, halogenoalkoxy, alkoxy, alkylthio, halogenoalkylthio, alkylamino, dialkylamino, nitro, cyano, hydroxyl, alkoxycarbonyl, optionally substituted phenyl, optionally substituted phenoxy or optionally substituted benzyloxy, or an acid addition salt or metal salt complex thereof.
Patent IL-66596-A0 (IL)
Title: Antihypertensive substituted n-alkanoylheterocyclic carboxylic acid derivatives,compositions containing them and methods for their use
IPC: C07K5/02
Filed: 1982-08-20
Abstract: Novel inhibitors of angiotensin converting enzyme are disclosed which have the general formula <CHEM> wherein R1 and/or R3 form complex amides and imides thereof, X = S, O or NR9, R4 and R5 form with -N-C- a 4-6 membered ring structure as described and the other R substituents are selected from a variety of disclosed groups.
Patent IL-90172-A0 (IL)
Title: 2,3-dihydro-imidazo(1,2-a)furo and-thieno pyridine derivatives,their preparation and pharmaceutical compositions containing them
IPC: A61P7/02
Filed: 1989-05-03
Abstract: The intention discloses compounds of formula I <CHEM>  wherein  T is <CHEM>   They can be prepared by dehydration. They are indicated for use as inhibitors of platelet activating factor (PAF) and as anti-tumor agents.
Patent IL-106359-A0 (IL)
Title: Antiinflammatory indolinyl n-hydroxyurea and n-hydroxamic acid derivatives
IPC: A61P7/02
Filed: 1993-07-15
Abstract: Certain novel indoline derivatives having the ability to inhibit the 5-lipoxygenase enzyme and having formula (I) wherein R1 is C1-C4 alkyl or -NR2R3; R2 and R3 are each, independently, hydrogen or C1-C4 alkyl; R4 is C3-C6 cycloalkyl, C4-C7 cycloalkylalkyl, aryloxy C2-C4 alkyl,  arylthio C2-C4 alkyl, arylamino C2-C4 alkyl, arylsulfinyl C2-C4 alkyl, aryl, aryl C1-C6 alkyl, aryloxyaryl C1-C6 alkyl or arylthioaryl C1-C6 alkyl, and the aryl groups in the said aryloxyalkyl, arylthioalkyl, arylaminoalkyl, arylsulfinylalkyl, aryl, arylalkyl, aryloxyarylalkyl and arylthioarylalkyl may be substituted up to the maximal number of substituents and the substituents are each independently, selected from the group consisting of halo, cyano, C1-C5 alkyl, C2-C6 alkenyl, C1-C5 alkoxy, C2-C6 alkenyloxy, C2-C6 alkoxyalkyl, halosubstituted C1-C4 alkyl, halosubstituted C1-C4 alkoxy, C2-C5 alkoxycarbonyl, aminocarbonyl and C1-C4 alkylthio; A is C1-C6 alkylene, C3-C6 alkenylene or -O-(CH2)m-; Y is each independently, halogen, halosubstituted C1-C6 alkyl, C1-C6 alkyl, C2-C6 alkenyl, C1-C6 alkoxy or C3-C8 alkenyloxy;  m is 2, 3 or 4; n is 0, 1, 2 or 3; and provided that the substituent Y, if present, and the linking group A are attached to the aromatic ring. These compounds are useful in the treatment of alleviation of inflammatory diseases, allergic conditions and cardiovascular diseases in mammals and as the active ingredient in pharmaceutical compositions for treating such conditions.
Patent IL-107522-A0 (IL)
Title: Device for automatically feeding curtain hooks to a sewing machine
IPC: D05B3/18
Filed: 1993-11-07
Abstract: For feeding curtain hooks, each consisting of a strip (1) and the hook (5) connected thereto, to a sewing machine which can sew the strip of an infed curtain hook onto a curtain pleat, use is made of a device comprising a storage holder (12) for the curtain hooks, and a device (9) for moving one curtain hook at a time from the storage holder (12) to a desired position for sewing on the strip of that curtain hook. According to the invention, the device (9) move the curtain hooks only in one straight line, the storage holder (12) is in the form of a vertical tube in which the curtain hooks can be stored stacked on top of one another, the bottom end of the storage holder (12) lies in or just above the straight movement path of the moving part (25) of the device (9), so that the moving part (25) can pick up the bottom hook in the storage holder (12), and the moving part (25) of the device ( 9) can return to the initial position during sewing on of the strip of the curtain hook held in position by the pressure foot of the sewing machine.
Patent IL-107891-A0 (IL)
Title: Benzocycloheptenes, benzoxepines and benzothiepines
IPC: C07D213/24
Filed: 1993-12-06
Abstract: PCT No. PCT/EP93/03445 Sec. 371 Date Aug. 5, 1994 Sec. 102(e) Date Aug. 5, 1994 PCT Filed Dec. 7, 1993 PCT Pub. No. WO94/13658 PCT Pub. Date Jun. 23, 1994The subject of the invention is compounds of general formula:    <IMAGE>  I  in which: X represents O or CHR, R1, R2, R3 and R4, which are identical or different, represent a hydrogen atom or a C1-C7 alkyl group, it being possible for R1 to additionally form a bond with R; R5 represents a hydrogen atom, a hydroxyl group or R5, taken together with R7, forms a bond or a >O; group; R6 represents a group of formula:   <IMAGE>    in which R10 and R11, taken together with the carbon atom to which they are attached, form a nitrogenous heterocyclic group, and their N-oxides and pharmaceutically acceptable salts. These compounds are powerful activators of potassium channels.
Patent IL-110389-A0 (IL)
Title: Aspirating plunger for power injector cartridges
Inventor: LIEBERT RICHARD T
IPC: A61M5/31
Filed: 1994-07-20
Abstract: A self-aspirating hypodermic cartridge (1) which contains an injectable fluid therein comprising a generally cylindrical barrel (3) having a wall, and a plunger (10,50,44) reciprocable in said barrel (3) to aspirate the cartridge (1) and to expel said injectable fluid therefrom said plunger (10,50,44) comprising: a female ring component (10), with a vertically oriented cylindrical hole (36), having a cylindrical flat bottom portion (20), a cylindrical flat top portion (30) spaced from said cylindrical flat bottom portion (20), and a side portion (40) connecting said cylindrical bottom and top portions (20,30) and integral therewith, said side portion (40) having a degree of incline with respect to a horizontal plane of from about 1° to about 89°; a mushroom-shaped male component (50) having a cylindrical plunger shaft (52) slideably positioned into said female ring component (10), and a cone-shaped head (56) at one end of the shaft (52) and integral therewith having a degree of incline with respect to a horizontal plane of from about 1° to about 89°; and an elastomeric diaphragm-shell (44) having a cylindrical bottom portion (42) and a generally cone-shaped side portion (48) integral therewith covering said male and female components (50,10), said cylindrical bottom portion (42) being adapted to form a slideable seal between the female ring component (10) and the wall of the cylindrical barrel (3), and said cone-shaped side portion (48) being adapted to serve as a diaphragm whereby upon alternate exertion of pressure upon said plunger shaft (52) and release thereof the deformation of the diaphragm reduces head space in the cylindrical barrel (3) thereby expelling head space gas and upon release of pressure the diaphragm returns to its original shape resulting in aspiration, is described herein.
Patent IL-114641-A0 (IL)
Title: Pharmaceutical compositions containing fluoxetine
IPC: A61K47/38
Filed: 1995-07-18
Abstract: Pharmaceutical formulations of fluoxetine or an acid addition salt thereof, suitable for manufacturing dispersible tablets by direct compression and comprising, in addition to the active ingredient, the appropriate excipients and coadjuvants, selected from among disintegrants, diluents, lubricants, anti-adherents, sweeteners, flavorings and, optionally, colorants.Said formulations are suitable for manufacturing dispersible tablets which disintegrate in less than three minutes in water at 19•C - 21•C, and are appropriate for treatment of depression.
Patent IL-128462-A0 (IL)
Title: Process for the preparation of an optically active indoline-2-carboxylic acid or derivative thereof
IPC: C07B57/00
Filed: 1999-02-10
Abstract: Process for the preparation of an optically active N-acyl-indoline-2-carboxylic acid in which a mixture of enantiomers of N-acyl-indoline-2-carboxylic acid is contacted with an optically active resolving agent and the optically active N-acyl-indoline-2-carboxylic acid is liberated from the resulting diastereomeric salt, as resolving agent use being made of a compound of formula 1, where R1 represents an alkyl group and R2 a (hetero) aryl group or where R1 and R2 together with the C atoms to which they are bound form a cycloalkyl group with 5-8 C atoms, fused with a (hetero) aryl group. Preferably, a mixture of enantiomers of an N-acyl-indoline-2-carboxylic acid is prepared in a process comprising the steps of Fischer indole cyclization of a 2-phenylhydrazone propionic acid or a derivative thereof in the presence of an acid catalyst, if necessary hydrolysis of the derivative to the corresponding acid, acylation at the N-position and reduction of the indole compound to the corresponding indoline compound, after which the resulting N-acyl-indoline-2-carboxylic acid is subjected to the resolution. The 2-phenylhydrazonopropionic acid or a derivative thereof is preferably obtained from phenylhydrazine and pyruvic acid or the corresponding derivative thereof.
Patent IL-139129-A0 (IL)
Title: Diagnosis and treatment of hepatic disorders
IPC: A61P1/16
Filed: 1999-05-12
Abstract: The present invention encompasses methods and compositions useful in diagnosing and treating hepatic disorders, especially those characterized by inflammation. The method comprises administration of an agent which prevents the interaction of MAdCAM with a MAdCAM binding partner or ligand. These compositions are useful in treating diseases or disorders involving  alpha 4 beta 7/MAdCAM blockade, as well as inhibiting a primary event in the inflammatory response such as blocking interactions between intercellular adhesion molecules and their ligands. Disorders treatable using the methods disclosed herein include infections, especially viral infections, iatrogenic disorders, cholestatic disorders, hereditary disorders, sarcoidosis, organ transplant, and the like. The diagnostic methods of the invention can be employed to detect the presence of a disorder or to monitor the course of therapy used to treat the disorder.