baber/WOPTO huggingface dataset:
Patent AP-2000001961-A0 (AP)
Title: Pharmaceutical aerosol formulation.
Inventor: CAVAILLON PASCAL
IPC: A61K47/12
Filed: 1999-04-15
Abstract: The present invention relates to novel pharmaceutical aerosol formulations comprising: (a)a therapeutic agent in the form of particles coated by at least one coating excipient and at least one surfactant, in suspension in (b)a liquefied propellant gas for the administration of therapeutic agents particularly by the pulmonary route and to a process for preparing these formulation. It also related to novel particles suitable for use in such formulations.
Patent AP-2002002420-A0 (AP)
Title: Fused pyrrolecarboxamides: gaba brain receptor ligands.
Inventor: ALBAUGH PAMELA
IPC: A61P43/00
Filed: 2000-08-30
Abstract: Substituted pyrrolecarboxamides compounds are disclosed. These compounds are highly selective agonists, antagonists or inverse agonists for gabaa brain receptors or prodrugs of agonists, antagonists or inverse agonists for gabaa brain receptors and are therefore useful in the diagnosis and treatment of anxiety, depression, alzheimer's dementia, sleep and seizure disorders, overdose with benzodiazepine drugs and or enhancement of memory. Pharmaceutcal compositions, including packaged pharmaceutical compositions, are further provided. Compounds of the invention are also useful as probes for the localization of gabaa receptors in tissue samplets.
Patent MC-1443-A1 (MC)
Inventor: GRIMBERG GEORGES SERGE
IPC: C01F11/30
Filed: 1982-02-11
Abstract: 1. Process for preparing a stable powder of a crystallized hygroscopic mineral salt containing in its molecule a large number of water molecules making it deliquescent and impossible to be distributed in hard capsules or in bags, characterized by crushing the crystallized hygroscopic mineral salt in the presence of dry yeast having a very fine particle size and within the range of 7.7 to 25% in weight with respect to the saft, up to obtaining a finely pulverulent homogeneous mixture which is stable and able to be easily put in hard capsule or in bags.
Patent ZW-7384-A1 (ZW)
Title: Electrical outlet system
Inventor: COOKE ALAN JOHN
IPC: H02G3/20
Filed: 1984-05-07
Abstract: A mains electrical connection system has male (100) and female (110) coupler fittings that make electrical connections after entry of contacts (31) from one fitting into the other and relative linear movement of the fittings. Those electrical connections are displaced from entries (27, 28) for the contacts (31) and thus safe from finger access. Further intercouplings are also shown (55, 56) with same taking at least most of mechanical loading from attempts to separate. One projection (55) for the latter purpose is used for earth connections. Cased socket units and plugs units are disclosed for incorporation into electrical outlet/connection accessories as desired.
Patent IE-910597-A1 (IE)
Title: Peptides which inhibit blood coagulation, processes for the preparation thereof and the use thereof
Inventor: STUEBER WERNER
IPC: A61K38/00
Filed: 1991-02-21
Abstract: Peptides of the formula I  A1-A2-A3-A4-A5-A6-A7-A8-A9-A10-A11-A12-A13-A14-A15  in which   A1 is hydrogen, cysteine, acetylcysteine, one or two alkyl groups with 1-4 C atoms, an acyl group with 2-10 C atoms, an acyl group with 2-10 C atoms and another carboxyl group, or a protective group customary in peptide chemistry,   A2 is a bond, Asn, Asp, Gln or Glu,   A3 is a bond, Gly or Ala,   A4 is Glu or Asp,   A5 is Phe, Tyr, Trp, Pgl (phenylglycine) or Nal (naphthylalanine),   A6 is Glu or Asp,   A7 is Glu, Asp, Pro or Ala,   A8 is Ile, Leu, Val, Nle or Phe,   A9 is Pro or Hyp,   A10 is Glu or Asp,   A11 is Glu or Asp, A12 is Phe(SO3H) or Phe(PO3H2) (preferably in the p position) or Pgl(SO3H) or Pgl(PO3H2) (preferably in the p position),   A13 is a bond, Leu, Ile, Val or Ala,   A14 is a bond, Gln, Asn, Glu, Asp or Cys and A15 is Cys, Cys-amide, an OH group of the alpha-carboxyl group, free or esterified with a lower alcohol with up to 4 C atoms, which can also be in the form of the carboxamide functionality whose hydrogens can optionally be replaced by alkyl groups with up to 4 C atoms, and a process for the preparation thereof are described. These peptides inhibit blood coagulation and can be used as anticoagulants.
Patent LU-87145-A1 (LU)
Inventor: GRIAT JACQUELINE
IPC: A61K31/355
Filed: 1988-02-26
Abstract: Method for improving the aesthetic aspect of the skin comprises applying daily to the skin a cosmetic compsn contg a mixt of vitamins in a vehicle suitable for a topical applicn and administering orally and daily a prepn also contg a mixt of vehicles in a vehicle suitable for such administration, the method being continued until the desired result is reached. Pref. the method is effected: for 3-5 weeks and pref the compsn. contains a mixt of vitamins E A, B2, B5 and H, and pref. it also contains Vitamins F, D, B6 and/or folic acid.
Patent MA-38983-A1 (MA)
Title: Disque pourvu d'au moins deux éléments de connexion électrique et d'un conducteur de liaison
Inventor: SCHMALBUCH KLAUS
IPC: H05B3/84
Filed: 2016-04-22
Abstract: L'invention concerne un disque pourvu d'au moins deux éléments de connexion (4) et d'un conducteur de liaison (6). Ce disque comprend au moins - un substrat (1) présentant une structure électroconductrice (3) sur au moins une partie du substrat (1), - au moins deux éléments de connexion électrique (4) sur au moins une partie de la structure électroconductrice (3), - au moins une surface de contact (9) sur la face inférieure de chaque élément de connexion (4), - une masse de soudure (8) permettant de relier les surfaces de contact (9) des éléments de connexion électrique (4), dans au moins une certaine zone, à la structure électroconductrice (3) et - un conducteur de liaison (6), lequel relie de manière électroconductrice les éléments de connexion (4) les uns aux autres, les surfaces de contact (9) les plus proches les unes des autres d'éléments de connexion (4) voisins présentant entre elles un écart x d'au moins 70 mm.
Patent MA-39235-A1 (MA)
Title: Dispositif électronique intelligent de régulation de tension de charge des batteries plomb acide automobile
Inventor: ZAZI MALIKA
IPC: H02J7/04
Filed: 2016-07-27
Abstract: L'invention est relative à un nouveau dispositif électronique de régulation de tension de charge des batteries plomb acide automobile, basé sur un microcontrôleur, des entrées/ sorties pour le diagnostic ainsi que des capteurs de tension, de courant et de température. Ce régulateur intelligent, en plus de sa fonction de régulation de tension, il maintient la batterie dans des conditions optimales. En effet la charge de la batterie est calculée en fonction de son état de charge (soc), son état de vie (soh) et de sa température afin de profiter de sa capacité maximale et d'éviter la sulfatation. Le régulateur intelligent est équipé d'un bus can (controller area network) afin de transmettre toutes les données utiles à l'ordinateur de bord de la voiture.
Patent UY-26461-A1 (UY)
Title: Procedimiento para la preparación de hidrocloruro de epinastina en la modificación cristalina de alto punto de fusión.
Inventor: DACH ROLF DR
IPC: A61P37/08
Filed: 2000-11-29
Abstract: La invención se refiere a un procedimiento para la preparación de hidrocloruro de epinastina en la modificación cristalina de alto punto de fusión.
Patent UY-26712-A1 (UY)
Title: Máscara para administrar fármacos a animales
Inventor: BARNEY BRIAN
Filed: 2001-05-16
Abstract: Una máscara de animal para sujetarla de manera que se pueda retirar de la porción adecuada de la cabeza de un animal como el frente de la cabeza o sobre una fosa nasal para la administración efectiva de fármacos o medicamentos, para absorción pulmonar o nasal. Los anillos de la máscara encajan entre sí, formando una sucesión de anillos de tamano monótono decreciente que se extienden de manera telescópica, desde el anillo más grande hasta el anillo más pequeno para formar un borde relativamente flexible. Un adaptador de interfase de animal se extiende desde el anillo más grande y se adapta para establecer un sello sustancial entre el adaptador de interfase de animal y la cara de un animal. La máscara para animal se puede plegar para permitir su uso en condición total o parcialmente abierta y para permitir el transporte fácil y cómodo en una condición plegada o cerrada
Patent UY-30502-A1 (UY)
Title: " azolilmetiloxiranos, su uso para combatir hongos fitopatógenos, así como productos que los contienen (vi) "
Inventor: KLASS LOHMANN JAN
IPC: A01N43/653
Filed: 2007-07-24
Abstract: Azolilmetiloxiranos de la fórmula I donde A o B significa fenilo, que está sustituido con un CN y, opcionalmente, por uno a tres de los siguientes sustituyentes halógeno, NO2, amino, C1-C4-aquilo, C1-C4-alcoxi, C1-C4-halógenoalquilo, C1-C4-halógenoalcoxi, C1-C4-alquilamino, C1-C4-dialquilamino, tio o C1-C4-alquilito, y el respectivo otro sustituyente A o B significa fenilo o heteroarilo de cinco o seis miembros, estando estos sustituyentes, opcionalmente, sustituidos según se indica en la descripción de la solicitud, asi como sus sales de adición ácidas o sales metálicos fitocompatibles, el uso de los compuestos de la fórmula I para combatir hongos fitopatógenos y productos que los contienen.
Patent AT-524761-A1 (AT)
Title: Schnallenbauteil
IPC: A44B11/10
Filed: 2021-02-15
Abstract: Schnallenbauteil (1, 2) mit einem Grundkörper (3) und einem Klemmsteg (4) , wobei der Grundkörper (3) eine Gurtaufnahmeöffnung (5) aufweist und der Klemmsteg (4) in der Gurtaufnahmeöffnung (5) zum Festklemmen eines um den 5 Klemmsteg (4) herum geführten Gurtes (6) zwischen dem Klemmsteg (4) und einem, die Gurtaufnahmeöffnung (5) begrenzenden Rand (7) des Grundkörpers (3) verschiebbar am Grundkörper (3) gelagert ist, wobei das Schnallenbauteil (1, 2) zusätzlich eine Klappe (8) aufweist, welche mittels eines io Schwenkgelenks (9) verschwenkbar am Grundkörper (3) gelagert ist, wobei die Klappe (8) eine Klemmfläche (10) zum Festklemmen des Gurtes (6) zwischen der Klemmfläche (10) der Klappe (8) und dem Klemmsteg (4) in einer Klemmstellung der Klappe (8) aufweist. (Fig. 5)
Patent AT-524831-A1 (AT)
Title: DYNA-FLEX: Skischuhe mit dynamischem und einstellbarem Flexverhalten
Inventor: FRANZ BRACHNER ING
IPC: A43B5/04
Filed: 2021-02-23
Abstract: Es wird Schutz begehrt für die Anbringung einer Zugfeder an der Skischuh-Rückseite, zur flexiblen Verbindung von Ober- und Unterteil des Skischuhs. Diese Zugfeder, die ausgeklinkt und vorgespannt werden kann, ermöglicht das stufenlose und individuelle Einstellen das Widerstands bei Vorwärtsbewegung, sowie dynamisches Entlasten bei Rückwärtsbewegung.
Patent AT-509403-A1 (AT)
Title: Fliessfähiger verfüllwerkstoff für künetten
IPC: C04B24/32
Filed: 2010-01-20
Abstract: Fließfähiger Verfüllwerkstoff für Künetten, enthaltend zumindest eine natürliche Gesteinskörnung und/oder rezyklierte Gesteinskörnung und/oder rezyklierte Hochbau-Restmassen und Wasser, zu dem ein Fließmittel und/oder ein Stabilisierungsmittel und/oder ein Mittel zur Herabsetzung des Reibungswiderstands beigemischt ist bzw. sind.
Patent DZ-1765-A1 (DZ)
IPC: C07D/
Filed: 1994-03-30
Granted: 2002-02-17
Abstract: (S)- alpha -phenyl-2-pyridineethanamine (S)-malate is useful in the treatment of neurodegenerative disorders. It is an anticonvulsant and a neuroprotective agent.
Patent ES-173603-A1 (ES)
Title: PERFECCIONAMIENTOS EN DISPOSITIVOS PARA TURBINAS DE VAPOR CON UN MiNIMO DE EMPAQUETADURAS LABERiNTICAS, CERRANDO HERMÉTICAMENTE CONTRA DIFERENTES PRESIONES
Filed: 1946-05-17
Abstract: Perfeccionamientos en dispositivos para turbinas de vapor con un mínimo de dos empaquetaduras de laberinto cerrando herméticamente contra diferentes altas presiones en las que se montan anillos fijos de carbón o de un material físicamente equivalente cuyo dispositivo comprende una tubería que comunica por lo menos dos cámaras intermedias de las empaquetaduras de laberinto y una segunda tubería que sirve apra la llegada de vapor vivo que actúa como vapor de obturación en las empaquetaduras de laberinto caracterizados por el hecho de que se equipa la conducción que une las cámaras intermedias con un dispositivo de desagüe y porque se preven en unión con este dispositivo medios que permiten la entrada al vapor de obturación en la tubería de unión citada impidiendo en cambio tal entrada a toda agua de condensación que llegue a las tuberías de vapor vivo y de desagüe.
Patent ES-184125-A1 (ES)
Title: UN SISTEMA DE SENALAMIENTO Y ENCLAVAMIENTO PARA EL MANDO DEL TRáFICO FERROVIARIO
Filed: 1948-06-15
Abstract: Establecimiento de un itinerario que se efectúa por medio de un solo dispositivo de contacto como botón palanca o análogo y en una sola maniobre el itinerario así establecido se anula automáticamente paso a paso después del paso del convoy que recorre la ruta correspondiente al itinerario.
Patent ES-185934-A1 (ES)
Title: Un sistema de comunicaciones
Filed: 1948-10-27
Abstract: Sistema de comunicaciones que comprende un primer grupo de terminales o bornes un segundo grupo de bornes y un equipo conmutador múltiple ( 110 109 150 170 179) entre los dos grupos de bornes para conectar selectivamente cualquier borne del primer grupo con cualquier otro del segundo grupo; caracterizado por medios ( 140 185) para poner en situación de marcar a uno de los bornes de uno de los grupos; medios ( 104 107 109) para prolongar el circuito en situación de marcar por todos los trayectos libres del equipo conmutador múltiple desde el borne marcado hasta los bornes del otro grupo y medios ( 174 177) para seleccionar uno de los trayectos marcados a fin de conectar el borne del primer grupo con uno de los del segundo grupo.
Patent ES-256220-A1 (ES)
Title: New steroid compounds
IPC: C07J75/00
Filed: 1960-02-25
Abstract: The invention comprises 19-nortestosterones of the general formula <FORM:0888665/IV (b)/1> wherein R represents hydrogen or an acyl group derived from an aliphatic, cyclic or partly cyclic carboxylic acid containing not more than 9 carbon atoms, and the preparation of the above 4-hydroxy substituted compound by dehydrating 17a - methyl - 19 - nor - andros - tone-4,5,17b -triol-3-one in alkaline solution at room temperature, e.g. by means of a methanolic solution of potassium hydroxide and, if necessary, neutralising the solution, e.g. with acetic acid, and, when required, esterifying the 4-hydroxy compound with the required acid chloride or anhydride to form a 4-ester of the above general formula, e.g. in the presence of a tertiary amine such as pyridine. Esters mentioned are the 4-acetate, propionate, b -cyclopentylpropionate, benzoate and b -phenylpropionate. Detailed examples are given. Reference has been directed by the Comptroller to Specification 864,610.ALSO:A therapeutic composition comprises at least one 19-nortestosterone of the general formula <FORM:0888665/VI/1> wherein R represents hydrogen or an acyl group derived from an aliphatic, cyclic or partly cyclic carboxylic acid containing not more than 9 carbon atoms, and a pharmaceutically acceptable carrier therefor. Reference has been directed by the Comptroller to Specification 864,610.
Patent ES-336811-A1 (ES)
Title: Polyamide-Acids and Polyimides Derived Therefrom
IPC: C08G73/14
Filed: 1967-02-14
Abstract: Polyimides and the precursor polyamide acids are derived from N,N1.di-(aminophenyl) ureas and dianhydrides. In examples, polyamideacids are prepared from 3,31- or 4,41-diaminophenyl urea and 3,31,4,41-benzophenone tetracarboxylic dianhydride, pyromellitic dianhydride or a dianhydride of the formula in solution in N-methyl-2-pyrrolidone or cresol and polyimide films are cast from the solutions. Other dianhydrides, solvents and diluents are mentioned.
Patent ES-346308-A1 (ES)
Title: Production of cyclodextrin
IPC: C12P19/18
Filed: 1967-10-21
Abstract: Cyclodextrins are prepared from a starch hydrolysate (as defined below) having a dextrose equivalent in the range 0À5-20, by conversion with cyclodextrin transglycosylase in an aqueous medium. The starch hydrolysate is obtained by enzymatic or acid hydrolysis of gelatinized starch, and may be converted at 40-60 C., at pH 5À5-7À5 using 100-1000 Tilden-Hudson units of enzyme per 100 g. of starch. The product may be separated by recrystallization or by complex formation with one of the following: p-cymene, tetra- or trichloroethylene benzene, carbon disulphide, toluene, hexane, cyclohexane, naphthalene, chloroform, carbon tetrachloride, bromobenzene, anthracene or thymol, whereby a precipitate forms. The complexing agent may be added during conversion to increase the product yield. Many starches are specified, including amylose and amylopectin.
Patent ES-352752-A1 (ES)
Title: Production of Aminobenzimidazoles
IPC: A61K31/415
Filed: 1968-04-15
Abstract: Compounds of formula wherein R is a 5-membered ring containing 1-3 hetero (N, O and/or S) atoms, and R 1 is H, OH, C 1-5 alkyl or C 1 _ 5 alkoxy, are prepared by reducing the corresponding 5-nitrobenzimidazoles the latter are prepared by reacting the unnitrated compounds with conc. HNO 3 in an acidic solvent medium.
Patent ES-361648-A1 (ES)
Title: Process for dealkylating hydrocarbons
IPC: B01J21/16
Filed: 1968-12-19
Abstract: Alkyl-aromatics are hydrodealkylated over a catalyst comprising compounds of at least one metal from each of Groups I A and VIA of the Mendeleev Periodic Table deposited on an alumina having the following characteristics: (a) specific surface: 40-120 m2/gm. (b) porous volume: 0À4-0À8 c.c./gm. (c) more than 75% of the porous volume corresponds to pores of 100-2000 diameter and (d) an acidity below 0.07 calory/sq. metre measured at 400 C. under a reduced pressure of 300 mm. Hg. The catalyst may additionally contain an iron group metal, e.g. Co or Ni, and inert gaseous diluents may be present. Toluene, xylenes, ethylbenzene and isopropylbenzene may be dealkylated, and the products may be desulphurized by hydrogen treatment over a Co/Mo catalyst.
Patent ES-366712-A1 (ES)
Title: Process and device for producing extinguishing foam
IPC: B01F5/04
Filed: 1969-05-02
Abstract: A jet of high expansion fire-extinguishing foam is ejected above a jet of foam of lower expansion so that it may be carried over a longer distance by the latter. The jets are produced by inducing air into streams of foamproducing liquid ejected through nozzles 16, 11 into tubes 1, 2. The degree of expansion of the foams may be governed by the shapes of the nozzles. Tube 1 may be longer than tube 2.
Patent ES-369926-A1 (ES)
Title: IMPROVEMENTS IN OR RELATING TO COMPOUNDS CONTAINING A PLURALITY OF BIS-(p-HALOPHENOXY) ACETOXY FUNCTIONS
IPC: C07D213/30
Filed: 1969-07-26
Abstract: Novel compounds containing a plurality of bis-(p-halophenoxy)acetoxy functions of the general formula wherein n is a whole number of from 2 to 6, X 1 and X 2 , which are the same, are each a chlorine or bromine atom, A is either a saturated C 2-6 aliphatic hydrocarbon moiety having 2-6 units of valency, the number of units of valency of A being equal to n, and no carbon atom having more than one unit of valency or, when n is 2, A is (i) a divalent group of the formula in which X1 1 and X1 2 , which are the same, are each a chlorine or bromine atom, or (ii) a divalent group of the formula are prepared (a) by reaction of a bis-(p-halophenoxy)-acetic acid or derivative thereof of the general formula wherein Y is a chlorine, bromine or iodine atom, a hydroxy group or a group of the formula with an alcohol or derivative thereof of the general formula A-(OM)n, wherein M is a hydrogen or alkali metal atom, with the proviso that when Y is a hydroxy group, M is a hydrogen atom, or (b) by reaction of an alcohol of the general formula A-(OH) n with a bis-(p-halophenoxy)-acetic acid ester or malonic acid ester of the general formula wherein Z 1 is a R-O-CO- group, in which R is a C 1-6 alkyl group, and Z 2 is as Z 1 or a hydrogen atom, with the proviso that when Z 2 is as Z 1 , the reaction is carried out at a temperature sufficiently high for partial decarboxylation to occur. Alcohols or derivatives thereof of the fourth general formula above wherein A is (i) above are prepared by reduction of a bis-(p-halophenoxy)-malonic acid ester of the fifth general formula above. Bis - (p - halophenoxy) - acetic acid esters or malonic acid esters of the fifth general formula above are prepared by reaction of a p-halophenol of the general formula with a dihalo-acetic acid ester or malonic acid ester of the general formula (X 1 ) 2 CZ 1 Z 2 , the p-halophenol being in the form of an alkali metal phenolate or the reaction being carried out in the presence of an acid-binding agent. Pharmaceutical compositions having hypocholesteremic/hypolipemic activity comprise, as active ingredient, a compound containing a plurality of bis-(p-halophenoxy)acetoxy functions of the first general formula above, in combination with a pharmaceutically acceptable diluent or carrier, and may be administered orally.
Patent ES-386175-A1 (ES)
Title: Oscillator with electrodynamic drive and electromagnetic detection, especially for use in an electronic clock
IPC: G04C3/00
Filed: 1970-12-04
Abstract: An oscillator of the swinging-mass type, especially for use in an electronic clockwork wherein an amplifier feedback circuit is provided between a pickup coil and a drive coil electromagnetically coupled with the swinging mass. The swinging mass is formed with a pair of oppositely poled permanent magnets spaced apart by a distance less than the magnetic cross-section of the coil means constituting the pickup and drive coils.
Patent ES-390680-A1 (ES)
Title: Antipollution exhaust system for an internal combustion engine
IPC: F01N3/30
Filed: 1971-04-28
Abstract: A system for reducing the back pressure on the exhaust valves of an internal combustion engine which includes, for instance, a source of compressed air, which may be powered by the internal combustion engine, and, in particular, a unique momentum transfer pump device which utilizes the high pressure compressed air output to create a suction or lower pressure at the exhaust manifold. A diffuser may be connected at the output end of the momentum pump to further increase the efficiency of the momentum pump.
Patent ES-393742-A1 (ES)
Title: Bag machine
IPC: B31B37/26
Filed: 1971-07-29
Abstract: The bag machine of the present disclosure is of the type which can produce bags made of various thermoplastic sheet material and can be adapted to make side weld or bottom weld bags. The following description will, however, be confined to the production of side weld bags.
Patent ES-396143-A1 (ES)
Title: 4-(2-hydroxy-3-isopropylamino-propoxy)-indole/isosorbitol - dinitrate compsn - for treatment of angina pectoris
IPC: A61K31/40
Filed: 1971-10-19
Abstract: The indole deriv. may be present as the free base or as a salt e.g. citrate or hydrogen maleate. The wt. ratio of the indole isosorbitol dinitrate is 1:1 to 1:5.