baber/WOPTO huggingface dataset:
Patent RU-2734256-C2 (RU)
Title: Novel compounds
Inventor: KEMP Mark Ien
IPC: A61P25/28
Filed: 2016-12-16
Granted: 2020-10-13
Abstract: FIELD: pharmaceuticals. 
     SUBSTANCE: invention relates to a compound of formula (I) or a pharmaceutically acceptable salt thereof, having inhibitory activity on ubiquitin-C-terminal hydrolase 30. In formula (I), each of R 1a , R 1b , R 1c , R 1d , R 1e  and R 1g  is hydrogen; R 1f  is hydrogen, or R 1f  together with R 2  forms a pyrrolidine ring substituted with an oxo group; R 2  is hydrogen or C 1 -C 6 alkyl, or R 2  together with R 1f  forms a pyrrolidine ring substituted with an oxo group; X is C(R 3 )(R 4 ), where each of R 3  and R 4  independently represents hydrogen, cyano or C 1 -C 6 alkyl; L is a covalent bond, -SO 2 -, -C(O)-, -CONR 5 -, -C(O)-C 1 -C 6 alkylene, -C(O)-C 2 -C 6 alkenylene or -C 2 -C 6 alkenylene; A is substituted 5–6 membered monocyclic heteroaryl or phenyl ring or substituted 8–12-membered bicyclic heteroaryl or naphthyl ring, wherein said heteroaryl rings contain from 1 to 4 heteroatoms independently selected from nitrogen, oxygen and sulfur; R 5  is hydrogen, where ring A is substituted with one group -Q 1 -(R 6 ) n , where n is 1; and additionally optionally substituted with one, two or three groups -Q 1 -(R 6 ) n , where n equals 0; n is 0 or 1; when n is equal to 0, Q 1  is halogen, cyano, oxo, -CONR 7 R 8 , -C 1 -C 6 alkyl or -C 1 -C 6 alkoxy, wherein said C 1 -C 6 alkyl is optionally substituted with one or more halogens; when n is 1, Q 1  is a covalent bond, an oxygen atom, -C 1 -C 6 alkylene or -SO 2 NR 7 -; R 6  denotes a phenyl ring, 3–6 membered cycloalkyl ring, 5–6 membered heterocyclyl ring containing one nitrogen atom, or 5–6 membered heteroaryl ring containing 1 or 2 heteroatoms independently selected from nitrogen, oxygen and sulfur; each of R 7  and R 8  independently represents hydrogen or C 1 -C 6 alkyl, where R 6  is optionally substituted with one or more substitutes, each of which is independently selected from halogen, cyano, -C 1 -C 6 alkyl and -C 1 -C 6 alkoxy, wherein said C 1 -C 6 alkyl is optionally substituted with one or more halogens. Invention also relates to compounds selected from a group consisting of 3-((quinolin-2-ylamino)methyl)pyrrolidine-1-carbonitrile, 3-(((6-fluorobenzo[d]thiazol-2-yl)amino)methyl)pyrrolidine-1-carbonitrile, 3-((isoquinolin-1-ylamino)methyl)pyrrolidine-1-carbonitrile, etc., and to a pharmaceutical composition containing said compounds together with one or more pharmaceutically acceptable excipients and having the activity of inhibitors of ubiquitin-C-terminal hydrolase.  
     
       
     
     EFFECT: novel compounds are disclosed. 
     19 cl, 1 dwg, 4 tbl, 54 ex
Patent RU-2738862-C2 (RU)
Inventor: FATENKOV OLEG VENIAMINOVICH
IPC: A61B5/00
Filed: 2018-08-13
Granted: 2020-12-17
Abstract: FIELD: medical diagnostics. 
     SUBSTANCE: invention refers to methods of diagnosing the state of the cardiovascular system. Method involves collecting anamnesis, physical examination and instrumental examination. After collecting medical history and physical examination, the doctor enters the obtained information into personal computer (1) with the corresponding software (SW). Computer (1) has communication with cloud processing and data processing system (3). Further, the patient lies on the couch, upper and lower extremities are covered with air pressure gauges, sphygmograms, apexcardiograms and ankle-brachial index (ABI) measurements. Electrodes are installed for rheogram removal (place is determined by type of examination) and ECG in the II lead. Parameters recording unit (2) measures arterial pressure, records an apexcardiogram, a sphygmogram with a given iteration step and measures the ABI. Rheogram is recorded simultaneously. Simultaneously ECG is removed in the II lead. Obtained information from unit (2) is transmitted to PC (1), where it is carried out together with data of cloud system (3), processing the obtained information and displaying the primary diagnosis with the treatment recommendations. 
     EFFECT: invention provides higher rate of diagnosing, as well as improved quality of examination of cardiovascular system. 
     1 cl, 2 dwg
Patent RU-2748889-C2 (RU)
Title: Support of frequency overlapping carriers
Inventor: BALDEMAIR ROBERT
IPC: H04W16/14
Filed: 2018-03-29
Granted: 2021-06-01
Abstract: FIELD: wireless communication.SUBSTANCE: invention relates to wireless communication and can be used to support frequency-overlapping carriers among the first radio access technology (RAT) and the second RAT, with the first RAT being New Radio (NR), and the second RAT being Long Term Evolution (LTE). The information of the second RAT is determined to be signaled to the wireless device of the first RAT. The second RAT information is configured to allow the wireless device of the first RAT to determine, at the resource element level, the resources reserved for transmissions of the second RAT, where the second RAT information also includes physical downlink shared channel bitmap templates for the second RAT, wherein the bitmap indicates radio resources to the wireless device to exclude NRs from the reserved resources. The second RAT is transmitted to the wireless device of the first RAT.EFFECT: invention is aimed at improving efficiency in configuring reserved NR resources to support coexistence of coincident NR carriers with LTE.17 cl, 12 dwg
Patent RU-2756560-C2 (RU)
Title: Reloading device for collecting and transferring harvested material to vehicle
Inventor: FLIEGL SEN JOSEF
IPC: A01D90/10
Filed: 2017-09-25
Granted: 2021-10-01
Abstract: FIELD: agriculture.SUBSTANCE: reloading device (4) for collecting and transferring harvested material to vehicle (6) includes collecting unit (8) for collecting harvested material from the ground, cutting unit (9) for grinding collected harvested material, storage unit (10) for receiving ground harvested material, a transporting device for transporting ground harvested material from storage unit (10) to reloading unit (11) of reloading device (4). Ground harvested material is transported relatively to the vertical direction and the lateral direction of reloading device (4) obliquely upwards and thereby into a cargo compartment of vehicle (6), located laterally adjacent to reloading device (4), above a wall of the cargo compartment.EFFECT: invention provides for the collection and transfer of stem-type biomass to the vehicle.14 cl, 13 dwg
Patent UA-40389-C2 (UA)
Title: Method for production of sorbent of spherical titanium phosphate based granulation
Inventor: STRELKO VOLODYMYR VASYLIOVYCH
Filed: 2000-12-27
Abstract: Invention concerns the synthesis of inorganic sorbents. The method for production of sorbent of spherical titanium phosphate based granulation consists in mixing of aqueous solution of titanyl sulfate, which contains compounds of iron with phosphoric acid, dispersion of reaction mixture in the medium of organic liquid immiscible with water with formation of granules of hydrogel, their washing with water and desiccation. Invention ensures narrow size distribution, high value of the sorption volume of pores and sorption capacity.
Patent UA-74779-C2 (UA)
Title: Dietary compositions to reduce weight gain in domestic animals and a method to reduce weight gain in domestic animals
IPC: A23L19/10
Filed: 2000-02-24
Abstract: Dietary compositions and methods employ a mammal food base and a component comprising estrogen, androgen or a mixture thereof in an amount sufficient to reduce weight gain normally incurred in the mammal type subsequent to neutering, castration, spaying, ovariectomy or ovariohysterectomy, or post menopause. Preferably, the component comprises phytoestrogen, phytoandrogen or a mixture thereof. The compositions are adapted for administration to the mammal on a regular, preferably daily, basis.
Patent UA-52515-C2 (UA)
Title: Electrode rod for electric arc welding
Inventor: KOLOTYI VALENTYN PETROVYCH
IPC: B23K35/02
Filed: 2002-08-06
Abstract: Invention relates to the field of the technology of construction materials and it can be used for production of iron rods of electrodes for manual electric arc welding. The rod of electrode for electric arc welding contains cylindrical and end surfaces. On the faces suitable components of mechanical lock are performed for guaranteeing the sequential interconnection of the rods. It allows to reduce the consumption of electrodes during welding due to the exclusion of cinders.
Patent UA-76418-C2 (UA)
Title: Antitumour derivatives of ecteinascidin , pharmaceutical composition on their basis and a method for the treatment of diseases
IPC: A61K31/498
Filed: 2001-04-12
Abstract: Compounds having a fused ecteinascidin five ring system with a 1,4 bridge and compounds in which the -NH2 or -OH of the 1,4 bridge is derivatised are disclosed. Such compounds are useful in the treatment of tumours.
Patent UA-58364-C2 (UA)
Inventor: BAIRACHNYI BORYS IVANOVYCH
Filed: 2002-12-05
Abstract: Винахід відноситься до області гальваностегії, зокрема до способів приготування борфтористоводневого електроліту для осадження покриттів сплавом олово-свинець. У розчин борфтористоводневої кислоти вводять борну кислоту і гідрохінон, розчиняють вуглекислий свинець і в отриманому електроліті здійснюють електрохімічне розчинення металів шляхом електролізу. Використовують бездіафрагмовий електролізер, а після електролізу вводять добавки поверхнево-активних речовин. Винахід запобігає окисленню двовалентного олова, забезпечує зниження витрат та спрощення технологічного процесу.
Patent UA-64497-C2 (UA)
Title: Method for producing near-beer
Inventor: PERETIATKO PETRO VASYLIOVYCH
IPC: C12H3/00
Filed: 2003-06-12
Abstract: A method for producing near-bear comprises dealcholisation of beer, which contains alcohol, on dialysis module, carbonization, cooling and bottling. In dialysation dialysate is delivered at the pressure of 1.5-2.0 bar at quantitative ratio of beer and dilysate of 1:(46).
Patent UA-76156-C2 (UA)
Title: Multipurpose chair
Inventor: PETRUSHEVSKYI IVAN IVANOVYCH
IPC: A61F5/00
Filed: 2004-01-08
Abstract: The multipurpose chair contains the adjustable hinged seat and back with the supports for the arms designed as the armrests and the supports for the designed as the footstep connected with the means for stimulation. The supports also comprise the adjustable demountable pelots for the neck, the back, and the legs as well as the belt, the head holder, and axillary suspension supports. The armrests are connected with the demountable table containingthe optical displaying device. The footstep has the fastening belts for the legs. The means for stimulation is designed as the electric stimulator with the electrodes.
Patent UA-74313-C2 (UA)
Title: Suspension of seat of transportation means
Inventor: PYLYPENKO VIKTOR VASYLIOVYCH
Filed: 2005-04-12
Abstract: Suspension of seat of transportation means contains a guiding linkwork, a mechanism of suspension height adjusting, a pneumatic elastic element with air supplying line, a damper, a supporting platform for seat and supporting base of the transportation means. The pneumatic elastic element and the damper interact with the supporting platform and base about pair of corresponding hinges and are executed as single pneumo-elastic-damping mechanism which has two chambers of constant and changeable volume. The changeable volume chamber is formed by a housing and a piston which are tightly jointed on close circuit by a rubber-cord sleeve. The chambers of constant and changeable volume are connected by a pneumo-throttle with a back valve, an axial channel of the piston is connected with the air supplying line of the transportation means by a three-position pneumo-valve.
Patent UA-78131-C2 (UA)
Title: A polymeric composition
Inventor: DREBEZOVA LIUDMYLA PETRIVNA
IPC: C01F7/02
Filed: 2005-06-09
Abstract: A polymeric composition contains chloroprene rubber, zinc oxide, magnesium oxide, stearic acid, low molecular polyethylene, naphtam, wax, antimony trioxide, chloroparaffin, aluminium hydroxide and chemically oxidized graphite. The composition is used in rubber industry for making thermally expanded material, which is used for increasing fire resistance of different surfaces and structures such as profiles, plates and other.
Patent UA-94023-C2 (UA)
Title: Use of an agent produced from a parasite for control of diseases
Inventor: WEINSTOCK JOEL
IPC: A61K35/62
Filed: 2004-10-22
Abstract: The invention relates to a method of screening a heminthic parasite preparation that affects a regulatory T cell function and a method of treating a disease by altering a regulatory T cell activity through the administration of a parasite preparation.
Patent UA-84800-C2 (UA)
Title: Heating saturator
Inventor: PUSHANKO MYKOLA MYKOLAIOVYCH
IPC: C13B20/04
Filed: 2007-04-13
Abstract: A heating saturator has a vertical cylindrical housing with side pipes for juice supply and discharge, devices for supply of saturation gas and providing its long-term contact with juice. According to the invention, over the upper part of the vertical cylindrical housing a device is installed as a cyclone with double walls, between which water is circulated by screwd path, with two tangentially located pipes for supply of a mix of vapor, gases and juice drops into the device, and central pipe for discharge of gas mix. The construction of the heating saturator allows full operation of apparatus functions for saturation process, providing of use of the heat of formed gas-vapor mixture and decreasing of emissions into athmosphere of saturation juice drops, which provides heat saving and decreasing of environment pollution.
Patent UA-84499-C2 (UA)
Title: Method for growing maize and soybean for silage in south-eastern forest-steppe of ukraine
Inventor: SOBKO MYKOLA HENNADIIOVYCH
IPC: A01B79/02
Filed: 2007-05-16
Abstract: The invention relates to a method for growing maize and soybean for silage in the North-Eastern Forest-Steppe of Ukraine that includes joint simultaneous sowing of the soybean variety Podilska an amount of 200 thousand seeds/ha and maize variety Dniprovskyi 310 in an amount of 50 thousand seeds/ha. The use of the method contributes to increasing the yield and the protein content in a preserved feed.
Patent UA-87002-C2 (UA)
Title: Deployable solar concentrator (embodiments)
Inventor: RUEL VINCENT
IPC: H02S30/20
Filed: 2005-10-11
Abstract: A space solar concentrator based on deployable reflectors attached to a panel base is described. Each of the reflectors includes sides coated with reflective coating on surfaces facing away from the base. In one embodiment, the sides of the reflector have thicker portion to provide stiffness for deployment absent compressive force, and thinner portion to reduce weight and storage energy. In another embodiment, both reflective sides are unfolded when the reflectors are in stowed position. During deployment, a stop side will limit the deployment of both reflective sides and ensure the proper reflecting position. In addition, these embodiments reduce the storage energy.
Patent UA-91034-C2 (UA)
Title: Cone crusher provided with system for adjusting interjaw space
Inventor: DELILLE JEAN-PIERRE
IPC: B02C2/00
Filed: 2005-07-12
Abstract: The inventive cone crusher comprises a tapered crushing vessel whose wall bears a fixed jaw (1) and a cynical head (2) mounted on a shaft which is coaxially arranged with respect to the vessel and is provided with an eccentric. Said eccentric bears a mobile jaw (2), The space between the jaws (1, 3) including a total wear compensation is set in a stationary condition prior to operation by means enabling the fixed jaw (1) to move vertically with respect to a body (11), while adjustment, safety and daily wear compensation paths are adjustable during the crusher operation by means of at least one jack (7) which is arranged under the mobile jaw (2) enables said jaw to be vertically movable.
Patent UA-85776-C2 (UA)
Title: Torque convertor
Inventor: PRYMA ANATOLII MYKOLAIOVYCH
IPC: F16K17/00
Filed: 2007-07-11
Abstract: A torque convertor has a body with nozzle, cover with discharge channel, membrane drive, gate with seal and shutoff ring. The design of the torque convertor provides stable support of water pressure in broad range of inlet and outlet water pressure.
Patent UA-95446-C2 (UA)
Title: Mutations in oas1 genes
Inventor: IADONATO SHON P
IPC: C12N9/12
Filed: 2006-03-05
Abstract: Modified amino acid sequence of OAS1 protein and genes related thereto, are provided.
Patent UA-99706-C2 (UA)
Title: Test bench for verification of instruments for measurement of gas flow rate
Inventor: KUZMIN SERHII VIKTOROVYCH
IPC: G01F25/00
Filed: 2008-07-11
Abstract: A test bench for the verification of instruments for measurement of gas flow rate relates to measurement technique, in particular to metrology. The test bench comprises connected in sequence functional blocks such as block for gas heating, block for reduction of gas pressure, at least one verification line and block of standard gages. As standard gages one uses nozzles of critical flow, block of standard gages comprises a mobile block of nozzles of critical flow. In parallel to the block for reduction of gas pressure a bypass is connected, on the verification line the tested meter or flow rate meter is installed. Input of the test bench is a connected to the block for gas heating unit for connection to main gas pipeline of natural gas, and the output of the test bench is a connected to the block of nozzles of critical flow unit for connection to gas pipelines with smaller gas pressure. The test bench provides increase of accuracy and quality of verification.
Patent UA-94600-C2 (UA)
Title: Indole sulfonamide modulators of progesterone receptors
Inventor: BLEISCH THOMAS JOHN
IPC: C07D209/12
Filed: 2007-01-17
Abstract: Compounds of Formula (I), wherein n is 1 or 2, and R1, R2, R3, R4, RS, R6, R7, and R8 are as defined herein, their preparation, pharmaceutical compositions, and methods of use are disclosed., (I)
Patent UA-97814-C2 (UA)
Title: Method for production of lead -acid accumulators with electrolyte pumping
Inventor: DZENZERSKYI VIKTOR OLEKSANDROVYCH
IPC: H01M10/44
Filed: 2009-04-29
Abstract: A method for forming lead-acid accumulators using water cooling consists of the following stages: accumulators or accumulator batteries are collected into groups, poured with electrolyte, after settling it is formed using direct and/or pulse current during four stages. At the first stage through the accumulators DC is passed during 5-20 min, which does not exceed 0.02 of Caccumulator nominal capacity; than current value is increased to 0.3-0.7 C;at the second stage DC of 0.3-0.7 Cis passed through the accumulators during 0.5-3 hours; at the third stage current value is decreased to 0.1-0.2 Cduring 0.5-2 hours; at the fourth stage additionally 0.1-0.2 Ccurrent is passed through the accumulators during 5-10 hours. During process of the accumulator formation, through every accumulator and a common tank with electrolyte a forming electrolyte of 1.05-1.20 g/cmdensity is pumped at 96-2400 ml/min circulation rate, which for 0.5-2.0 hours before end of formation procedure is substituted with the electrolyte with operating density of 1.26-1.31 g/cm. The electrolyte of operating density is pumped in the same manner – at the same rate, all pumped electrolyte is cooled in the tank, and in the end of the formation procedure the electrolyte of operating density is left. The technical result is the increase of manufacturing rate of positive electrolytes and the decrease of dispersion of electrolyte density and accumulators electric characteristics. Utility quality: accumulator capacity increase, standardization of technical characteristics thereof.
Patent UA-95673-C2 (UA)
Title: Test system for control of parameters set which relate to operation of device for opto-electronic information display
Inventor: GERMAIN AURELIE
IPC: H04N17/04
Filed: 2008-03-21
Abstract: According to the invention, the test system uses a digital photography device (4) that can be remotely controlled from a computer system including a processor (20) coupled to a man/machine interface (21) and to the presentation device to be tested by a remote transmission means. A means is further provided for centring the photographic apparatus (4) opposite the presentation device (5) to be tested. The processor (20) is programmed so as to carry out a self-positioning phase of the photographic apparatus, an automatic focalisation phase of the lens, and a test phase of the information presentation device.
Patent UA-99496-C2 (UA)
Title: Complex filter for a smoking article, a cigarette which comprises the complex filter and a method for making this filter
Inventor: YANG SZU-SUNG
IPC: A24D3/02
Filed: 2008-12-22
Abstract: Provided is a cigarette filter (10) and method of making the filter. The filter (10) comprises an adsorbent (12) dispersed within the filter (10) and a downstream plug (16) of randomly-oriented fibers (14). The randomly-oriented fibers (14) mechanically capture adsorbent particles entrained in tobacco smoke. One or more plugs (25) of axially-oriented fibers (30) may also be located upstream or downstream or both of the adsorbent (12), and are included in an amount sufficient to adjust the length of the filter (10).
Patent UA-106055-C2 (UA)
Title: Roller of an agricultural machine
IPC: A01B29/00
Filed: 2011-05-30
Abstract: The applied roller (1; 1A) comprises a cylindrical core (2; 2A), made in such a manner as to allow rotating around the longitudinal axis (3) and is equipped with equidistant crowns (4; 4A), between which cleaners (5; 5A) are arranged. Each of the cleaners (5; 5A) comprises a plate (6; 6A) and a support (7; 7A), at the lower end of which the plate (6; 6A) is mounted, the upper end thereof is fixed on a carrying structure (8), passing in parallel to the longitudinal axis (3). The carrying structure (8) comprises an area (10) of fixing the supports (7; 7A), limited by the back half of the carrying structure (8), if one looks transversely to the working direction (A). In the stated area (10) of fixing the carrying structure (8) comprises two grooves (11, 12) forming a guide.
Patent UA-100786-C2 (UA)
Title: Signaling device of locomotive brake line status
Inventor: MARKOVSKYI VOLODYMYR KINDRATOVYCH
IPC: B60T17/22
Filed: 2011-06-14
Abstract: The invention relates to the railway transport and improves quality of control of brake line condition and its reliability in operation. A signaling device has a split body with internal partition separated by movable partitions made in the form of diaphragms. On a spring-loaded diaphragm forming a chamber with a body connected by a pipe to the locomotive brake line a valve rod is secured which is passed through a center hole of the inner partition of the body. On the check valve electrical contacts of a signaling device are mounted and between the intermediate part of the signaling device and its lid the diaphragm is mounted forming two chambers, one chamber is connected by the pipe to the brake line and the second chamber is connected by the pipe to a compensation tank of locomotive. A rod is mounted on the diaphragm and cinematically connected to an indicator of air output.