baber/WOPTO huggingface dataset:
Patent SK-16599-A3 (SK)
Title: 2-saccharinyl methyl heterocyclic carboxylates, compositions them containing, and their use as proteolytic enzyme inhibitors
Inventor: DUNLAP RICHARD P
IPC: A61K9/20
Filed: 1999-02-08
Abstract: 4-R<4>-R<5>-2-Saccharinylmethyl heterocyclic carboxylates, having the formula: <CHEM>  wherein: Het is a 5- or 6-membered monocyclic heterocycle or a 9- or 10-membered bicyclic heterocycle containing from 1 to 2 heteroatoms selected from oxygen, nitrogen and sulfur or said heterocycles substituted by from one to three, the same or different, members of the group consisting of lower-alkyl, perfluorolower-alkyl, lower-alkoxy, oxo, phenyl, halogen, and -O-(C2-C10 alkylene)-N=B where N=B is dilower-alkylamino, 1-pyrrolidinyl, 1-piperidinyl, 4-morpholinyl, 1-piperazinyl, or 4-lower-alkyl-1-piperazinyl; R<4> is hydrogen, halogen , lower-alkyl, perfluorolower-alkyl, perchlorolower-alkyl, lower-alkenyl, lower-alkynyl, cyano, carboxamido, amino, lower-alkylamino, dilower-alkylamino, lower-alkoxy, benzyloxy, lower-alkoxycarbonyl, hydroxy or phenyl; and R<5> is hydrogen or from one to two substituents in any of the 5-, 6- or 7-positions. The compounds of the present invention inhibit the activity of serine proteases, specifically human leukocyte elastase and the chymotrypsin-like enzymes, and are thus useful in the treatment of degenerative disease conditions such as emohysema, rheumatoid arthritis, pancreatitis, cystic fibrosis, chronic bronchitis, adult respiratory distress syndrome, inflammatory bowel disease, psoriasis, bullous pemphigoid and alpha-1-antitrypsin deficiency.
Patent SK-48798-A3 (SK)
Title: Method and apparatus for controlling the temperature of the bed of a bubbling bed boiler
Inventor: RAIKO MARKKU
IPC: F23C10/20
Filed: 1996-10-18
Abstract: The present invention relates to a method and assembly for controlling the bed temperature in a fluidized-bed boiler, particularly in boilers fired with coal or other fuels of high heat value but difficult to gasify. Above the fluidized bed (6), but below the freeboard (8), is arranged a cooling zone (19) and the fluidizing gas is injected into a portion of the bed at an excess rate per unit area, whereby over the area of increased fluidizing gas injection, the bed is expanded upward into the cooling zone, wherefrom unburned combustible material and the particulate matter of the bed can fall back in the bed. The gas injection (9) with the higher flow rate is arranged to the center of the fluidized bed, whereby the return circulation can occur past the waterwall portions enclosing the cooling zone, thus facilitating efficient heat transfer from the refluxed bed material in the form of radiation absorbed by the heat transfer surfaces of the cooling zone waterwalls.
Patent SK-57093-A3 (SK)
Title: Method of coal flotation
Inventor: MACHO VENDELIN
IPC: B03D1/02
Filed: 1993-06-07
Abstract: Coal flotation, coal for coking purposes especially is provdided in water sludge, after having grinded and air blowing together with flotation agent is applied, while this flotation agent is prepared based on hydrocarbons and / or plant oils and oxygen organic compounds. However, 100 weight parts of coal is treated by 0,1 up to 1,1 weigh part of flotation agent, while this agent consits of foamer and skimmer. Foamer in a quantity of 15 up to 85 weight percent of flotation agent is saponified partially and or partially hydrolysed triglyceride of plant oil and a synthetic mixture consisting of 55 up to 99 weight percent, at least three aliphatic and / or acyclic alcohol, and / or ketons with 3 up to 18 carbon atoms in a molecule, while the rest up to 100 percent is created by ethers and esters especially, aldehydes, carboxyl acids, hydroxyacids. Skimmer is created based on the hydrocarbon fraction and / or oil or methylester related to at least one unsaturated carboxyl acid C14 up to C22.
Patent CH-631047G-A3 (CH)
IPC: H03F3/34
Filed: 1979-07-13
Abstract: An amplifier includes an inverter with two transistors of complementary types. The first transistor is biased through a third transistor of the same type of conductivity by a first reference voltage, the third transistor being biased by a third voltage of reference. The second transistor is biased through a fourth transistor of the same type of conductivity by a second voltage of reference, the fourth transistor being biased by a fourth voltage of reference. The first and second voltages of reference are determined so that without any alternating input signal the current in the first and second transistors of the inverter is minimum. The third and fourth voltages of reference are determined so that the equivalent resistances of the third and fourth transistors are very high.
Patent CZ-138592-A3 (CZ)
Title: Acetic acid derivative, process of its preparation and a pharmaceutical composition in which said derivative is comprised
Inventor: GUTHRIE ROBERT WILLIAM
IPC: C07C49/825
Filed: 1992-05-07
Abstract: The invention relates to compounds of the formula Q and n are as described herein. Their pharmaceutically acceptable salts, and when appropriate, enantiomers, racemates, diastereomers or mixtures thereof or geometric isomer or mixtures thereof, and pharmaceutically acceptable salts thereof. The compounds of formula I inhibit enzyme carnitine acyltransferase 1 (CAT-1) and are therefore useful in the prevention of injury to ischemic tissue, and can limit infarct size, improve cardiac function and prevent arrhythmias during and following a myocardial infarction.
Patent CZ-306592-A3 (CZ)
Title: 3-phenylpyrazole derivatives, process of their preparation and fungicidal compositions in which said derivatives are comprised
Inventor: CHENE ALAIN
IPC: C07D231/38
Filed: 1992-10-08
Abstract: The new fungicidal phenylpyrazoles are of formula I or Ib: <IMAGE>  in which:   X = H, hal, NO2, CN, SCN, (C1-C4)alkyl, (C1-C4)alkenyl, (C1-C4)alkynyl, (C1-C4)alkoxy, (C1-C4)alkylthio, phenyl, phenoxy, monoalkyl- or dialkyl- or phenylamino, alkylcarbonyl, carbamoyl, carboxyl, benzoyl, alkylsulphinyl or alkylsulphonyl; Y, Z = H, hal, OH, NO2, NO, CN, SCN, (C1-C4)alkyl, (C1-C4)alkenyl, (C1-C4)alkynyl, (C1-C4)alkoxy, (C1-C4)alkylthio, phenyl, phenoxy, monoalkyl- or dialkyl- or phenylamino, alkylcarbonyl, carbamoyl, carboxyl, benzoyl, alkylsulphinyl or alkylsulphonyl, and the like; Y, Z can also form a bridge containing 1 to 4 atoms, one at least of which may be an optionally substituted heteroatom; R is H, Hal, NO2, (halo)alkyl, phenyl, S(O)mR1, CH2NR3, (CH2)m R4, CH(R5)XR6, CHR7R8, C(X)R10, COXR19, and the like.   Products which can be used as fungicides in agriculture.
Patent CS-358791-A3 (CS)
Title: Use of a combination of an angiotensin-creating enzyme inhibitor and calcium antagonist for application at albuminuria
Inventor: BECKER REINHARD DR
IPC: A61K31/41
Filed: 1991-11-26
Abstract: An angiotensin converting enzyme inhibitor (I) can be used in combination with Ca antagonists (III) in the prevention and therapy of proteinuria. Pref. (A) Ramipril and felodipine; (B) Ramipril and 4-(2,3-dichlorophenyl) -2,6-dimethyl-3- (1,2,4-oxadiazol-5-yl) -S-isopropoxy carbonyl-1,4-dihydropyridine (IIb), (c) Trandolapril and felodipine; (D) Trandolapril and (IIb), (E) Trandolapril and Verapamil; (F) Quinapril and felodipine; (G) Quinapril and (IIIb) or the physiologically acceptable salts of these components.
Patent CZ-632190-A3 (CZ)
Inventor: HUDEC FRANTISEK ING
IPC: F23N5/08
Filed: 1990-12-18
Abstract: Zapojení k sledování kvality plamene hoření, hlavně pro
automatizované řídicí systémy, zejména v energetice obsahuje
vyhodnocovací obvod pro hlídání plamene, zvláště
olejových a plynových hořáků. Podstatou je zapojení se
vstupní částí, kde jsou vytvářeny impulzy z proudu tekoucího
fotonkou při ionizaci, s tvarovačem (20), převodníkem
(30) kmitočet-proud, komparátorem (40), výkonovým členem
(50), referenčním zdrojem (60) a obvodem (70) testování.
Zapojení může být využito hlavně v průmyslových
technologiích, zejména pak v energetických blocích a
teplárnách s automatickými řídicími systémy.
Patent CZ-107799-A3 (CZ)
Inventor: SAINTS KEITH W
IPC: H04B7/00
Filed: 1997-09-23
Abstract: Při způsobu se měří hodnoty energie v pásmu a poté se
vypočítává hodnota neinterferující energie. Hodnota
neinterefující energie se odečítá od uvedené hodnoty energie v
pásmu, čímž se získá hodnota interferenčního šumu. Měř! se
energie bitu přijímaného signálu a na základě hodnoty
interferenčního šumu a uvedená energie bitu se vypočítává se
poměr signálu k šumu. Podobně jsou generovány povely pro
řízení výkonu akumulováním předem určeného celočíselného
nn/Mii r-----y- ■, ■ vzorlni -------------------- ---- ---- dpmnduínvan^hn sionáln wnni*ítáváním . jr v
hodnoty šumu pro demodulovaný signál na základě uvedených
vzorků, měřením energie bitu pro demodulovaný signál, načež
se vypočítá hodnota poměru signálu k šumu pro
demodulovaný signál na základě hodnoty šumu a hodnoty
energie bitu.
Patent CZ-126893-A3 (CZ)
Title: Capacitor
Inventor: ROTH ZDENEK ING CSC
IPC: F28B1/02
Filed: 1993-06-25
Abstract: The device is formed by several tubular clusters of heat transfer pipes (2), through which the cooling water flows. The steam-air mixture enters the condenser from the side. In each tubular cluster of heat transfer pipes (2), on the side reverse from the steam-air mixture input, there is a cooling space (30) linked to the central hollow (3). Fitted in the cooling space (30) are the heat transfer pipes of the steam-air mixture cooler (4). The tubular cluster and steam-air mixture cooler (4) are terminated by the side wall (50) and upper wall (51) of the cover (5), fitted in contact with them and hermetically joined to them is a collection channel (8) with metering holes (80). Another part of the cover (5) forms a perpendicular shield (52), connected to the upper wall (51) of the cover (5) and inserted into the perpendicular fin between the steam-air cooler (4) of steam-air mixture and adjacent part of the tubular cluster.<IMAGE>
Patent CZ-9901655-A3 (CZ)
Title: Circuit arrangement of entry into protected areas
Inventor: PROCHAZKA ZDENEK ING
IPC: G07C9/27
Filed: 1999-05-10
Abstract: In a protected area (1), equipped by an electronic lock (2) and by a reading device (3) of chip cards (4), connected to a discriminating unit (5), a user terminal (7) is located, which is connected to an evaluation centre (6). The evaluation centre (6) is connected with an access events memory (9), with a discriminating unit (5) and with a monitoring terminal (8), while the access events memory (9) is also connected to the discriminating unit (5). This arrangement enables entrance into the protected area (1) only to authorized users, equipped by the pertinent chip card (4). This arrangement further enables the user, who ascertains damages, to transmit the report about discovered status via user terminal (7) into the evaluation centre (6), which compares time of change of the status in the protected area (1) with time of access events, stored in the access events memory (9), assigns responsibility for ascertained damages and eventually abolishes the right of access for the responsible persons by means of discriminating unit (5) and that all can occur without personal presence or performance of supervising staff.
Patent CZ-182297-A3 (CZ)
Title: Therapeutic preparation for inhalation containing parathyroid hormone, pth
Inventor: BACKSTROM KJELL
IPC: A61K9/00
Filed: 1995-12-08
Abstract: The present invention relates to compositions and methods for pulmonary administration of full-length parathyroid hormone to mammalian hosts for the treatment of osteoporosis. Thus there is provided a therapeutic, dry powder preparation suitable for inhalation comprising (i) as an active substance, a parathyroid hormone having an amino acid sequence which is at least 90% homologous to the sequence shown as SEQ ID NO: 1 in the Sequence Listing having the biological activities of the full-length parathyroid hormone; (ii) a pharmaceutically acceptable carrier consisting of coarse particles; and, optionally, (iii) as an active substance, a substance which enhances the absorption of parathyroid hormone in the lower respiratory tract; wherein an ordered mixture is formed between said active compound(s) and the carrier; in which at least 50% of the total mass of the active substance parathyroid hormone consists of (a) particles having a diameter of up to 10 microns; or (b) agglomerates of such particles. <IMAGE>
Patent CZ-200794-A3 (CZ)
Title: Process for producing toothed wheels from steel plate by cold forming
Inventor: HIMMEROEDER HELGE
IPC: B21D53/28
Filed: 1993-02-19
Abstract: A method of forming a toothed wheel comprising the steps of cold-forming a circular piece of sheet metal of predetermined thickness into a preform, rotating (1) a rotary holding unit with the preform secured thereto about the preform axis and with a control surface of the holding unit underlying at least a portion of an annular section of the preform and (2) a tooth-forming tool unit in a predetermined rotational relation wherein the axes of rotation are parallel and the rotational speeds are synchronized, and while in the predetermined rotational relation affecting a relative movement between the units and the axes thereof in a direction toward one another to engage a tooth-forming periphery of the tooth-forming tool unit in cooperating metal-deforming relation with the annular section inwardly of the exterior periphery thereof until the sheet metal of the annular section is cold-formed into the series of teeth, the peripheries of which are cold-formed by rolling contact with the tooth-forming periphery of the tooth-forming tool unit and portions of the sides of which are smooth and cold-formed by contact with smooth tooth-side forming surfaces so that an amount of sheet metal which would otherwise uncontrollably flow axially outwardly of the smooth tooth-side forming surfaces is concentrated within the teeth and/or the radially inward back-up therefor and the toothed wheel made thereby.
Patent CZ-256693-A3 (CZ)
Title: Method of measuring spectropolarimetric properties of optically active substances and a dichrograph for making the same
Inventor: ROKOS JIRI ING
IPC: G01N21/21
Filed: 1993-11-26
Abstract: The dichrograph and accompanying method are usable for parallel measurement of circular dichroism according to the first harmonic of photoelectric current of the detector, optical rotation acccording to the second harmonic and transparency according to the null harmonic. It contains the switch (3) of ray, from which alternatively exit two parallel rays - measurement ray (4) and reference ray (5), going through one mutual modulator of elipticity (6), achromatic phase element (9) which is during calibration of circular unit situated in the reference ray (5). Moreover it contains two analyzers - the measurement analyzer (8) in the measurement ray (4) behind the couvette (7) and the reference analyzer (10) in the reference ray (5). The measurement analyzer (8) has the optical axis turned for 45 DEG  same as the modulator (6). The reference analyzer (10) is during measurement turned for unit angle, e.g. for 1 DEG , to the measurement analyzer (8).
Patent CZ-273096-A3 (CZ)
Title: Re-constitution method of lyophilized drug and apparatus for making the same
Inventor: HARRIS DALE C
IPC: A61J1/06
Filed: 1994-03-14
Abstract: A cartridge assembly (90) for holding a lyophilized product, forming a disposable portion of a pen injector (104), includes a cylindrical glass cartridge (58) adapted to receive the product, a closure cap (20), a cartridge case (76), and a plunger mechanism. The closure cap (20) is adapted to retain an elastomeric disc seal (52) during lyophilization and includes diametrically opposed ledges (38, 40). The closure cap (20) and seal (52) are adapted to cover a neck portion of the ampule (58), the neck portion having on its end a radially extending circumferential flange (62). The ledges (38, 40) of the closure cap (20) and the flange (62) of the neck portion allow the closure cap (20) to remain open during lyophilization, oxygen purge and nitrogen overlay. An oval-shaped indentation formed on the inside of the closure cap (20) aids in snapping the closure cap (20) about the flange (62) without crimping to retain the closure cap (20) underneath the flange (62). Reconstitution of the lyophilized drug is accomplished without foaming by use of an obliquely angled connector (30) which causes the diluent to indirectly impinge on the drug. The injection pen (104) and cartridge assembly (90) cooperate such that the length of travel of the plunger rod (108) during retraction is less than the axial length of a recess (107) in the rod tip (73).
Patent CZ-281697-A3 (CZ)
Title: Material for coating wires
Inventor: RICHARDSON PETER JAMES
IPC: C09D123/04
Filed: 1996-03-06
Abstract: A wire coating composition comprises 100 php (parts per hundred parts of polypropylene) polypropylene polymer or copolymer, 1 to 20 php of polyethylene wax and 100 to 200 php of magnesium hydroxide which is provided with a hydrophobic coating. The wire coating composition does not contain any halogen and is essentially free of phosphorous and phosphorous salts.
Patent CZ-292696-A3 (CZ)
Title: Position correction method of aiming elements, particularly of weapon dial sight relative to the axis of a barrel bore and apparatus for making the same
Inventor: BASCHWITZ RUBIO JAVIER
IPC: F41G3/32
Filed: 1996-02-02
Abstract: Device and method for correcting the position of aiming elements of an arm, specially a sight, with respect to the bore axis of said arm, comprised of a hollow tube having an appropriate length so that it can be introduced in the arm, in place of the bolt of the latter, the tube presenting a truncated end so as to be adapted to the calibre in the mouth of the chamber, and provided externally with a bush having an outside diameter corresponding to the entrance point of the bolt, so that it is centred. Said device is provided internally with a laser beam emitting system with supplying and switching means, said beams going through the truncated area appropriately bored as well as optionally, another stepped surface adapted to the firing mouth and also axially bored so that the beam materialises, on a target placed according to adequate distance tables, the impact point by means of a light point and, with respect to the latter, correcting the sight by acting on the corresponding sight adjusting mechanisms. <IMAGE>
Patent CZ-307296-A3 (CZ)
Title: Synergetic herbicidal composition and method of its application
Inventor: LAKE BYRON HARVEY
IPC: A01N57/12
Filed: 1995-03-30
Abstract: A synergistic herbicidal composition comprising atrazine and either NMSC (i.e., 2-(2'-nitro-4'-methylsulfonylbenzoyl)-1,3-cyclohexanedione), or NMSOC (i.e., 2-(2'-nitro-4'-methylsulfonyloxybenzoyl)-1,3-cyclohexanedione):   <IMAGE>    <IMAGE>   Also disclosed is a method of controlling undesirable vegetation by applying an effective amount of such composition to the locus of the vegetation to be controlled.
Patent CZ-346297-A3 (CZ)
Title: Process for preparing aqueous solution of sodium hydroxide
Inventor: POSAR FRANCESCO
IPC: C01D1/04
Filed: 1997-10-31
Abstract: Production of an aqueous solution of sodium hydroxide from electrodialysis of sodium carbonate in an electrodialysis cell with three compartments is claimed. A solution of sodium carbonate is introduced in one compartment of the cell delimited between two cationic membranes. An acid is added to one compartment delimited between one of the cationic membranes and a cationic side of a bipolar membrane. An aqueous solution of sodium hydroxide of a compartment adjacent to the anionic side of the bipolar membrane is then extracted.
Patent ES-188284-A3 (ES)
Title: PERFECCIONAMIENTOS EN LAS MáQUINAS PARA PREPARAR CAFÉ EXPRÉS
Filed: 1949-05-14
Abstract: Perfeccionamientos en las máquinas para preparar café exprés caracterizados por disponer una o mas aspitas constituidas por un cilindro en el que se desliza un émbolo que da paso al interior de dicho cilindro al agua procedente de la caldera y la impide luego a través de la capa de café molido contenido en el filtro dispuesto en la parte inferior del cilindro.
Patent SK-167199-A3 (SK)
Title: Fungicide mixtures
Inventor: SCHELBERGER KLAUS
IPC: A01N37/50
Filed: 1998-06-05
Abstract: The invention relates to a fungicide mixture, containing at least one active agent chosen from a1) carbamates of formula (Ia), wherein T means CH or N, n stands for 0, 1 or 2 and R is halogen, C1-C4 alkyl or C1-C4alkyl halide and the radicals R can be different when n is 2; and a2) oximether carboxylic acid ester of formula (Ib), a3) oximether carboxylic acid amide of formula (Ic), and b) at least one active agent of formulae (II.1) to (II.5), in a synergetically effective quantity. The invention also relates to a method for using the inventive mixtures as fungicides.
Patent SK-192000-A3 (SK)
Title: MICROORGANISMS OF GENUS AMYCOLATOPSIS OR ACTINOMADURA, ENZYMESì (54) OBTAINED THEREFROM AND PROCESS FOR PREPARING AMIDES
Inventor: ROBINS KAREN TRACEY
IPC: C12N9/88
Filed: 1998-07-22
Abstract: Microorganisms of species Amycolatopsis or Actinomadura able to convert nitriles into amides and provide enzyme extracts, are new. Also claimed are: (1) microorganisms of the species Rhodococcus GF270 (DSM 12211) and GF376 (DSM 12175), their variants and their mutants and their enzyme extracts, capable of converting nitriles into amides; (2) an enzyme with nitrile hydratase-activity obtained from the microorganisms above.
Patent SK-361892-A3 (SK)
Title: High-frequency msv mixing
Inventor: HYBEN PETER
IPC: H03C1/02
Filed: 1992-12-10
Abstract: The basic principle of the high frequency MSV mixer, consisting of a dielectric substrate, on which the micro band exciting converter, closed to magnetostatic wave is created of one side, is based on that, on the dielectric substrate (1) along the exciting converter (2), there is crated a modulation micro band line (4) and this line is symmetric in the shape of the simple meander and it is connected over the exciting converter, and on the area closed to parallel converters, there is located ferromagnetic layer (5) pre-magnetized in the perpendicular direction. The output of the modulation line (4) can be connected to the conductive layer (3).
Patent SK-582016-A3 (SK)
Inventor: LUKAC PETER
IPC: E06B5/11
Filed: 2013-12-16
Abstract: Dvere, najmä bezpečnostné, sú z bočných strán a z hornej strany vybavené dvojfalcovou obrubovou kovovou lištou (1), ktorá je svojimi kotviacimi elementmi votknutá do obvodového dreveného rámu (2). Drevený rám (2) je z vnútornej strany vybavený kovovou výstužou (3). V kovovej výstuži (3) je závitovým spojom pomocou tyče (6) upevnené teleso (7) zámku. Kovovou výstužou (3) je L profil alebo pásovina. Dvere sú vybavené závesom dverí, ktorý pozostáva z dvojfalcového dverového krídla (8) s otvormi (9). Výplň (5) dverí je protipožiarna a/alebo protihluková.
Patent AT-519180-A3 (AT)
Title: Mal- und Zeichen-Board
Inventor: JOSEF FEUERER
IPC: B43L5/00
Filed: 2016-10-14
Abstract: Mal- und Zeichenboard, wobei ein Basiselement (1) Leisten (1b, 1c) sowie Grifflöcher (1a) und Einschubschlitze (1v, 1v1, 1v2, 1w, 1w1, 1w2) zur Handhabung bzw. zur Aufnahme von Stützelementen (2, 4, 5, 6) aufweist, welche ebenfalls Grifflöcher und Einschubschlitze umfassen, wobei ein Einschubfach (3) vorgesehen ist, welches dem Verstauen der Teile beim Transport am Basiselement (1) dient.
Patent WO-9952514-A3 (WO)
Inventor: MARGREITER RAIMUND
IPC: A61P35/00
Filed: 1999-04-14
Abstract: The invention relates to the use of a compound of formula (I), wherein R1 is a base defined by one of the formulae (a), (b), (c) and (d), and R2 is hydrogen, C1-C4 alkyl, bromine, fluorine, chlorine or iodine, or a pharmaceutically acceptable salt thereof, for producing a medicament for immunosuppressive therapy of the human or animal body. The invention also relates to combination preparations with cyclosporine A, tacrolismus, mycophenolatemofetil, daclizumab, rapamycin and/or one or more corticosteroids.