baber/WOPTO huggingface dataset:
Patent IL-109161-A0 (IL)
Title: Amino alcohol derivatives, methods for the preparation thereof, and pharmaceutical compositions containing the same
IPC: C07D207/408
Filed: 1994-03-29
Abstract: The invention provides a group of compounds that are effective agents to inhibit specific cellular signaling events often induced by inflammatory stimuli, to act as anti-inflammatory or immunosuppressive agents, to act as cytotoxic agents for treatment of cancers, or to be directly or indirectly antimicrobial to yeast or fungal infections. More specifically, the inventive compounds have at least one amino alcohol (or derivative thereof) functional group on a side chain attached to a core moiety. The inventive compounds are useful antagonists to control intracellular levels of specific sn-2 unsaturated phosphatidic acids and corresponding phosphatidic acid-derived diacylglycerols, intracellular cell signaling messengers which occur in response to pro-inflammatory and selectively proliferative stimuli.
Patent IL-110820-A0 (IL)
Title: N-substituted heterocyclic derivatives and their preparation
IPC: A61K31/513
Filed: 1994-08-30
Abstract: Heterocyclic N-substituted derivatives of formula (I) and their salts are new. R1, R2 = H, 1-6C alkyl, 1-4C alkoxy, NH2, NH2CH2-, COOH, (1-4C alkoxy)carbonyl, CN, tetrazolyl, methyltetrazolyl, methylsulphonylamino, trifluoromethyl sulphonylamino(methyl), N-cyanoacetamide, N-hydroxy- acetamide, N-((4-carboxy)-1, 3-thiazol-2-yl) acetamido, ureido, 2-cyanoguanidinocarbonyl, 2-cyano-guanidino-methyl, imidazol-1-yl-carbonyl, 3-cyano-2-methyl isothioureidomethyl, with the proviso that R1 and R2 are not both H. R3 = H, 1-6C alkyl (optionally substituted by one or more halogen, 2-6C alkenyl, 3-7C cycloalkyl, Ph, phenyl-(1-3C alkyl) or (2-3C alkenyl)phenyl; the Ph groups are optionally substituted by at least 1 halogen, 1-4C alkyl, halogen-(1-4C alkyl), polyhalogeno-(1-4C alkyl), OH or 1-4C alkoxy. R4, R5 = 1-6C alkyl, Ph, phenyl-(1-3C alkyl), the alkyl, phenyl and phenylalkyl groups being optionally substituted by one or more halogen, perfluoro-(1-4C alkyl), OH or 1-4C alkoxy. Or R4 and R5 together form =CR7R8, (CH2)n or (CH2)pY(CH2)q. R7 = H, 1-4C alkyl or Ph; R8 = 1-4C alkyl or Ph. Y = O, S, C (substituted by 1-4C alkyl, Ph or phenyl-(1-3C alkyl) or NR6. R6 = H, 1-4C alkyl, phenyl-(1-3C alkyl), 1-4C alkylcarbonyl, halogeno-(1-4C(alkyl)carbonyl, polyhalo-(1-4C alkyl)carbonyl, -COPh, alpha-aminoacyl or an N-protecting group. Or R4 and R5 together form indane or adamantane. p + q = m; n = 2-11; m = 2-5; X = O or S. z and t = 0 or one is 0 and the other is 1. Specifically claimed is 2-n-butyl-4- spirocyclopentane -1-((2'-(5-tetrazolyl) biphenyl-4-yl)methyl) -2-imidazolin-5-one.
Patent IL-115535-A0 (IL)
Title: High solids copolymer dispersion from a latex and its use in sealants
IPC: C08F265/04
Filed: 1995-10-06
Abstract: A method for polymerizing predominantly one or more acrylate and/or vinyl acetate monomers in the presence of a latex results in high solids dispersions of polymer particles with lower viscosities than traditionally observed. A significant wt. % of added monomers can be present in large particles, having nonspherical shapes. Some of the original latex particles are retained during the polymerization and these increase the solids content and lower the viscosity by packing in the interstices between large particles. The total polymer solids content can easily be varied from 70 to 92 or more wt. % which are higher than achieved in any previously reported aqueous polymerizations. The viscosities at very high solids contents become paste-like but the materials still are stable to storage and further handling without breaking the dispersion into an agglomerated polymer portion and released water. The dispersions are useful to form sealants, membranes, etc., either with or without other additives. A preferred use is as an acrylate water-based caulking compound where the high solids and thixotropy of the dispersion allows for formation of a water-based caulk with low shrinkage.
Patent IL-130327-A0 (IL)
Title: A process for inhibiting stem elongation in bulbous plants
IPC: A01G5/06
Filed: 1997-12-12
Abstract: A process of inhibiting stem elongation in ornamental bulbous plants or in cut flowers from such plants, involving treating such plants or flowers with an effective amount of ACC synthase inhibitor, such as aminoethoxyvinylglycine and aminooxyacetic acid to inhibit stem elongation, by administration of a solid, semi-solid or a solution of such ACC synthase inhibitor.
Patent IL-130725-A0 (IL)
Title: Field transplanter
IPC: A01C11/02
Filed: 1997-12-31
Abstract: The present specification discloses apparatus for transplanting seedlings (24) from a tray (6) that has a plurality of seedling retaining cells (34), into a prepared ground planting position, the apparatus having tray holding means (1), seedling eject means (15, 16, 17) for removing one or more seedlings (24) from the seedling retaining cells (34), seedling delivery means (26, 27, 29) for receiving a seedling (24) ejected from the tray (6) and delivering same via a travel path to a ground planting preparation device (78) arranged to at least partly prepare said ground planting position, seedling holding means (100) associated with the ground planting preparation device arranged to hold a seedling delivered by said seedling delivery means (26, 27, 29), plant plug removal means (82, 83, 85) arranged between said seedling eject means (15, 16, 17) and said seedling holding means (100) to remove any plant plug (84) not containing a seedling viable for planting from said travel path prior to reaching said seedling holding means (100), and seedling planting means (89) to move a said seedling from said seedling holding means (100) to the prepared ground planting position in response to said apparatus having travelled a predetermined distance over the ground.
Patent IL-142852-A0 (IL)
Title: A COMPLEX OF A CHAPERONE WITH β-AMYLOID AND METHODS EMPLOYING THIS COMPLEX
IPC: A61K38/00
Filed: 1999-10-29
Abstract: A chaperone protein Q2 and β-amyloid can form a complex. This complex can be detected in a biological sample, such as, for example, tissues or fluids from a mammal. Q2 levels can also be detected in a biological sample. A method for determining the Q2 level in a biological sample and comparing that level to a normal Q2 level can be used to detect, screen, diagnose, or otherwise determine a person's susceptibility to Alzheimer's disease such as, for example, the presence or absence of Alzheimer's disease, of symptoms of this disease, of factors leading to or associated with this disease, of likelihood of developing this disease, and the like. In one embodiment, a decline in Q2 level correlates to an increased likelihood of developing Alzheimer's disease. In another embodiment, a decline in Q2 level correlates to an increase in β-amyloid aggregation. The method may further include screening for an apolipoprotein E genotype, which is associated with Alzheimer's disease.
Patent IL-146248-A0 (IL)
Title: A method and apparatus for automatically producing tubular knitwear items provided with at least a brace, shoulder strap, loop and the like, and products obtained thereby
IPC: D04B9/20
Filed: 2000-05-19
Abstract: The invention relates to tubular knitwear items complete with shoulder straps (20, 21), braces and various openings for legs or arms, manufactured without the usual cutting and sewing operations. Through the appropriate selection of needles, in accordance with the jaquard design and to the operating cycle of the knitting machine, the invention allows the separation and automatic programmed resumption of knitted courses for defined areas or zones, thereby obtaining at least a complete opening or brace, formed by at least a simple or double welt, or even multiple, edges, depending on circumstances. Lastly, the invention eliminates the current necessary cut and sew operations and the consequent, usual and costly fabric scrap.
Patent IL-149213-A0 (IL)
Title: Oxime o-ether compounds and fungicides for agricultural and horticultural use
IPC: A01N43/40
Filed: 2000-11-02
Abstract: The present invention relates to novel oxime O-ether compounds represented by a general formula ÄIÜ; <CHEM> wherein R<1> represents C1-6 alkyl, C3-6 cycloalkyl, C1-6 alkoxy, etc., m represents an integer of 1 to 4, R<2> represents hydrogen atom, C1-6 alkyl, etc., R<3> and R<4> each independently represents hydrogen atom or C1-6 alkyl, etc., R<5> represents hydrogen atom, C1-6 alkyl, etc., R<6> represents C1-6 alkyl, C2-6 alkenyl, C2-6 alkynyl, C1-6 alkoxy, Halogeno atom atom atom, etc. and n represents an integer of 1 to 4, and a fungicide for agricultural and horticultural use comprising the compound as the active ingredient.
Patent IL-169894-A0 (IL)
Title: Aircraft with forward opening inlay spoilers for yaw control
IPC: B64D7/00
Filed: 2005-07-26
Abstract: An aircraft comprises first and second wings positioned on opposite sides of a longitudinal axis with each of the first and second wings including an upper surface and a lower surface, wherein no control surfaces are attached to the lower surface of the wings. A first forward opening control surface is attached by a first hinge to an upper surface of the first wing and a second forward opening control surface being attached by a second hinge to an upper surface of the second wing. Each of the first and second hinges is canted with respect to a direction perpendicular to the longitudinal axis. A method of yaw control performed by the aircraft is also included.
Patent IL-190075-A0 (IL)
Title: Two-component systems for producing flexible coatings
Filed: 2008-03-11
Abstract: Two-component coating systems containing (A) a polyisocyanate prepolymer with allophanate-linked polyether groups and (B) an amino-functional polyaspartate ester. Two-component coating systems containing (at least) (A) a polyisocyanate prepolymer with allophanate-linked polyether groups and (B) an amino-functional polyaspartate ester of formula (I). X : n-valent organic residue of an n-functional polyamine; R 1>, R 2>organic groups which are inert towards isocyanate groups under reaction conditions; n : at least 2. Independent claims are included for (1) coatings obtained from the systems described above (2) substrates coated with these coatings. [Image].
Patent IL-204030-A0 (IL)
Title: Modulators of p-selectin glycoprotein ligand 1
IPC: C07K16/28
Filed: 2010-02-18
Abstract: Compounds that bind to P-Selectin Glycoprotein 1 (PSGL-1) on the surface of T cells or natural killer (NK) cells can be used to induce T cell or NK cell depletion and/or to induce T cell or NK cell apoptosis. The compounds and methods of the invention can be used to control unwanted T cell- or NK cell-mediated immune responses in conditions such as autoimmune diseases, transplant rejection, and allergic diseases.
Patent IL-216418-A0 (IL)
Title: New therapeutical uses of inecalcitol
Filed: 2011-11-17
Abstract: The present invention thus concerns a method for treating and/or preventing rickets, osteoporosis, osteomalacia, psoriasis, autoimmune diseases such as multiple sclerosis or type I diabetes, hyperparathyroidism, benign prostate hyperplasia, any type of cancer or any vitamin D relevant disease comprising administering inecalcitol at doses comprised between 1 mg/day and 100 mg/day to a human patient in need thereof.
Patent RO-126109-A0 (RO)
Title: Method for preventing skidding and blocking of the driving wheels of the urban passenger transportation vehicles driven by chopper and direct current motor
Inventor: DUMITRESCU CAMIL
IPC: G05B19/00
Filed: 2009-11-13
Abstract: The invention relates to a method for preventing skidding and blocking of the driving wheel of a vehicle driven by chopper and direct current motor. According to the invention, the method is based on processing by means of a software the voltage and current through the vehicle traction motor, acting for lowering the start up torque when the driving wheel skids, or in braking conditions when the wheel is blocked, and comprises a first step (A) of introducing the values of some normal operation parameters of a vehicle, a second step (B) of detecting an abnormal operation condition based on a first stage (B1) for taking over the operating parameters and a second stage (B2) of comparing with a view to detecting an abnormal operation condition, a third step (C) when a decision is made whether the abnormal operation condition is due to the occurrence of a skidding or blocking phenomenon or to other causes and a fourth step (D) in which corrections are made to the torque developed by the motor so as to eliminate skidding or locking of the driving wheel.
Patent AU-2002953115-A0 (AU)
Title: Glue line use of synthetic pyrethroids for wood products
IPC: C09J9/00
Filed: 2002-12-05
Abstract: The invention provides glue, glue line resin systems and wood products incorporating glues with bifenthrin. Methods are disclosed for the application of such glue and resin systems with bifenthrin. The glues with bifenthrin are effective for preserving wood including engineered wood products, with or without additional surface sprays.
Patent ZW-1387-A1 (ZW)
Title: New dihydrobenzofuran-and chroman-carboxamide derivatives,processes for the preparation thereof and use thereof as neuroleptics
Inventor: JACQUELINE FRANCESCHINE
IPC: C07D311/04
Filed: 1987-01-23
Abstract: The invention relates to new dihydrobenzofuran- and chroman-carboxamide derivatives of the general formula:   <IMAGE> (I) in which R and R' are each hydrogen or methyl; n is 1 or 2; m is 1 or 2; Z is either   <IMAGE> (a)   wherein R1 and R2 are lower alkyl, or <IMAGE> (b)  wherein R3 is alkyl, alkenyl, cycloalkyl-alkyl, cycloalkenyl-alkyl, X is H, NH2, methoxy, or methyl and Y is H, Cl, cycloalkylmethylsulfonyl, alkylsulfamoyl or alkylsulfonyl and to their pharmacologically acceptable acid addition salts and their optical isomers, to the processes for the preparation thereof and to the use thereof as medicaments, especially as neuroleptics.
Patent IT-9000309-A1 (IT)
Inventor: MASSOCCO GIORGIO
IPC: B02C18/02
Filed: 1990-06-12
Abstract: PCT No. PCT/IT91/00048 Sec. 371 Date Apr. 3, 1992 Sec. 102(e) Date Apr. 3, 1992 PCT Filed Jun. 10, 1991 PCT Pub. No. WO91/19568 PCT Pub. Date Dec. 26, 1991.The invention concerns equipment for continuous chopping of municipal refuse and other solid wastes in general, consisting of: Section I: refuse collection subsystem, first compaction and conveyance to chopping section; Section II: subsystem for final compaction and chopping ribbon of refuse; Section III: subsystem for collection of chopped refuse and conveyance to landfill sites; Section IV: subsystem for collection and disposal of wastewaters. The equipment permits a ten-to fifteen-fold reduction in the initial volume of the refuse, together with a chopping operation which allows this volume to be maintained and to obtain refuse of a sufficiently uniform size prior to transportation or to disposal in landfill sites.
Patent MA-20150361-A1 (MA)
Title: Acier lamine a chaud ou a froid a faible densite, son procede de mise en oeuvre et son utilisation
Inventor: ZUAZO RODRIGUEZ IAN ALBERTO
IPC: C22C38/06
Filed: 2013-05-27
Abstract: L'invention concerne une tôle d'acier laminée dont la résistance mécanique est supérieure ou égale à 600 mpa et l'allongement à rupture est supérieur ou égale à 20% ainsi que son procédé de fabrication. La composition chimique de la tôle de l'invention comprend : 0,10 = c = 0,30 %, 6,0 = mn = 15,0 %, 6,0 = al = 15,0 %, et à titre optionnel, un ou plusieurs éléments choisis parmi: si = 2,0%, ti = 0,2%, v = 0,6% et nb = 0,3% le reste de la composition étant composé de fer et d'impuretés inévitables résultant de l'élaboration. Le rapport du poids du manganèse sur celui d'aluminium est tel que :
Patent MA-38982-A1 (MA)
Title: Nouvel octahydro-cyclobuta [1,2-c; 3,4-c'] dipyrrol-2-yl
Inventor: MATTEI PATRIZIO
IPC: C07D487/04
Filed: 2014-11-24
Abstract: The invention provides novel compounds having the general formula (i) wherein r1, y and r2 are as described herein, compositions including the compounds and methods of using the compounds.
Patent MA-52675-A1 (MA)
Title: Anticorps anti-staphylococcus et leurs utilisations
Inventor: KYRATSOUS CHRISTOS
IPC: C07K16/12
Filed: 2019-11-20
Abstract: L'invention concerne des anticorps spécifiques ou des fragments de liaison à l'antigène qui se lient à des antigènes staphylococciques, les anticorps et les fragments de liaison à l'antigène présentant une liaison fc atténuée à la protéine a ou à une protéine homologue. L'invention concerne également des compositions comprenant les anticorps et des procédés d'utilisation. Les anticorps et les compositions sont utiles pour traiter une infection staphylococcique, réduire des titres bactériens sériques ou rénaux, et traiter des symptômes associés à une infection staphylococcique. Les anticorps peuvent également prévenir la gravité et/ou la durée de la maladie primaire.
Patent UY-29270-A1 (UY)
Title: Compuestos quimicos
Inventor: BUTLIN ROGER JOHN
IPC: C07D215/02
Filed: 2005-12-20
Abstract: Se describen compuestos de fórmula (I), y sales y profármacos de los mismos: en donde, por ejemplo, R1 está opcionalmente sustituidos arilo o heteroarilo; Y es un grupo de enlace seleccionado de, por ejemplo, un enlace directo, y una cadena de alquilo (sustituido); R2 es un grupo arilo opcionalmente sustituido, un cicloalquilo opcionalmente sustituido o un grupo heterocíclico opcionalmente sustituido. También se descirben procesos para preparar dichos compuestos y su uso como inhibidores de DGAT, por ejemplo en el tratamiento de la obesidad.
Patent UY-30650-A1 (UY)
Title: Sal de acido p-toluensulfonico de 5-amino-3-(2??-o-acetil-3??-desoxi-b-d-ribofuranosil)-3h-tiazol[4,5-d]pirimidin-2-ona y métodos de preparacion
Inventor: WANG TINGMAN
IPC: A61P31/00
Filed: 2007-10-17
Abstract: La presente descripcion se refiere a sal de ácido p-toluensulfonico de 5-amino-3-(2??-0-acetil-3??-desoxi-beta-D-ribofuranosil)-3H-tiazolo[4,5-d]pirimidin-2-ona y a su uso para tratar condiciones patologicas tales como infecciones virales, tumores y cáncer.
Patent UY-30961-A1 (UY)
Title: Comprimido famacéutico, capa de comprimido comprendiendo ingrediente activo telmisartan, un agente basico y sorbitol, proceso de preparacion y aplicaciones,
Inventor: MAERZ FRIEDER
IPC: A61K9/20
Filed: 2008-03-13
Abstract: Un comprimido o capa de comprimido farmacéutico que comprende el antagonista del receptor de angiotensina II telmisartán en forma amorfa, un agente básico y sorbitol, caracterizado porque el sorbitol tiene un área de superficie específica de entre 0,73-3,5 m2/g.
Patent CS-812288-A1 (CS)
Title: Rolling down device
Inventor: PLESINGER PETR
IPC: C03B9/00
Filed: 1988-12-08
Abstract: The mechanised prodn. of parisons for hollow glass articles uses two planishing tools on a spring-loaded holder, pivoted to a swivelling arm. The arm terminates in a positioner. A first tool planisher the round bottom and another the side walls of the parison.
Patent ES-148276-A1 (ES)
Title: RECIPIENTE COLECTOR PARA BASURAS Y ANáLOGAS
IPC: B65F3/22
Filed: 1940-03-30
Abstract: Un recipiente colector para basura o análogapreferentemente montado en un vehículoprovisto de un tornillo transportador rotativo montado en una caja en forma de tubo para cargar basura bajo presión en el recipientecaracterizado porque a lo largo de alo menos parte de la circunferencia de la cajael espacio entre la superficie del tornilloo su prolongación anterior y la cajaes menor en una extremidad o en ambas extremidades de la superficie del tornillorespectivamente la parte anterior de la cajaque en un plano perpendicular al eje del tornillo a través de la parte anterior de una abertura de carga practicada en la caja.
Patent ES-169323-A1 (ES)
Title: Un procedimiento para el alamacenaje y transporte de gases licuados en disolventes.
Filed: 1945-03-23
Abstract: Un procedimiento para el almacenaje y para el transporte de gases licuados disolventes especialmente de acetileno caracterizado porque el gas se incorpora a una masa de relleno que a su vez se carga en botellas poliglobulares de acero ligero de espesor de pared muy reducido.
Patent ES-179841-A1 (ES)
Title: Un procedimiento de localizar senales sonoras en portadores de registros sonoros
Filed: 1947-09-22
Abstract: Un procedimiento de localizar señales sonoras invisibles en portadores de registros sonoros, caracterizado porque muestra las señales sonoras en un aparato indicador en circuito con una cabeza reproductora.
Patent ES-182228-A1 (ES)
Title: Un sistema de suministro de energia eléctrica de alta frecuencia
Filed: 1948-02-10
Abstract: Sistema para suministrar energía de alta frecuencia, a voltaje constante, a una carga que comprende una fuente para proveer energía a una alta frecuencia dada incluyendo un circuito de válvula que tiene una salida de corriente constante, un circuito que conecta las citadas fuente y carga incluyendo los elementos de capacidad e inductivos de un valor tal que provean una condición de resonancia a la citada frecuencia dada.
Patent ES-189336-A1 (ES)
Title: SISTEMA IMPULSOR DE NEGOCIOS MEDIANTE TiTULOS DE INTERCAMBIO DE VALOR GARANTIZADO
Filed: 1949-08-05
Abstract: Sistema impulsor de negocios mediante títulos de intercambio de calor garantizado en que se reivindica la póliza cuyo texto se expone en los anexos I y II cuyo desarrollo es objeto del cuerpo de esta memoria que igualmente queda reivindicado por constituir ambos una misma cosa con carácter de imposible separación.
Patent ES-198970-A1 (ES)
Title: PERFECCIONAMIENTOS EN LA CONSTRUCCIoN DE LOS TERMoMETROS DE MERCURIO A CONTACTO GRADUABLE
Filed: 1951-07-27
Abstract: Perfeccionamientos en la construcción de los termómetros de mercurio a contacto graduable caracterizado por disponerse en el interior del tubo capilar de los termómetros un hilo de resistencia graduable y por el instrumento indicador que estará dispuesto a cualquier distancia del termómetro propiamente dicho.