baber/WOPTO huggingface dataset:
Patent JP-2002503356-A (JP)
Title: リソグラフィック投影装置を走査する鏡像投影系及びこのような系を具えるリソグラフィック装置
IPC: G02B17/06
Filed: 1998-10-19
Abstract: (57)【要約】
ステップ及び走査リソグラフィック装置で使用される鏡像投影系であって、マスクパターン（１５）は、円弧形断面を有するＥＵＶ照射のビーム（ｂ）によって基板（２０）の複数の領域上で繰り返しスキャンされて結像される。６個以上の結像ミラーを有する投影系よりも廉価に製造しやすいこの系は、５個の結像ミラー（５〜９）しか有しないが、良好な開口数及び許容し得る像の環状領域幅を有する。新規の投影系を設けたＥＵＶリソグラフィック投影装置は、６個のミラーの投影系を設けた装置のウェファスループットより約５０％高いウェファスループットを有する。さらに、それはコンパクトな構造を有する。
Patent JP-H09512559-A (JP)
IPC: C07D491/22
Filed: 1995-05-02
Abstract: The present invention relates to a method for preparing intermediates useful in the preparation of camptothecin and camptothecin-like compounds and to the intermediates used in this preparation. In particular, the invention provides a process for the preparation of a compound of formula II' <CHEM> wherein X is halogen, which comprises reacting a compound of formula III <CHEM>  with a compound of formula IX' <CHEM>
Patent JP-H10510337-A (JP)
IPC: E04B1/86
Filed: 1996-03-27
Abstract: The invention relates to vibration damping wall material or wall covering material. The material is comprised of a laminate which includes two thin metal sheets and a solid rubber layer sandwiched therebetween. The rubber layer has the form of a rubber foil or rubber film having a thickness of 0.08-0.30 mm and produced by carrier calendaring and is vulcanized to each metal sheet. The metal sheets suitably have a thickness of 0.2-0.7 mm. The rubber layer is conveniently formed from an electrically conductive rubber mixture. When the wall material is intended for use with structures that delimit rooms or like locations in which a high standard of hygiene is demanded, the metal sheets may consist of stainless steel.
Patent JP-H10500232-A (JP)
Title: 収納携帯型オーバーヘッドプロジェクター
IPC: G03B21/30
Filed: 1995-05-04
Abstract: (57)【要約】
その上面にフレネルレンズ（１６）を収容するステージ本体（１２）を有する収納型オーバヘッドプロジェクター（１０）である。該ステージ本体は、ランプ包囲体（１４）を形成し得るように一側部の厚みを厚くしてある。ヒンジ式ミラーも該本体内に設けられて、また、ヒンジ式ランプソケットがランプ包囲体内に設けられている。二対の収納型脚部（２４、２６）が、本体に及びランプ包囲体にヒンジ式に結合して、且つ展開してミラー及びランプを下降させ、収納可能な基部を形成する。該脚部はランプ及びミラーを傾動させ、光がミラーによりフレネルレンズを通じて上方に反射される。更なる対の収納型脚部が釣合わせ機能を果たす。収縮可能なベローズ（４７）、光バッフル（２５）及びミラーがランプ及びミラーに対する光遮蔽性で且つ気密の包囲体を提供する。
Patent JP-2001502263-A (JP)
Title: 鉄道車両用車載発電機システム
IPC: B61D43/00
Filed: 1997-03-04
Abstract: (57)【要約】
発明は、貨車、有蓋貨車、等の現行の鉄道車両に取付けられる車載発電機システムに関し、車両の軸の回転によりシステムに動力が供給される。車両の電気的に制御されたブレーキ用のバッテリーに充電する手段として使用することが望ましい。このような車両は、典型的には複数の軸を取り付け、軸に略平行に整列された突起を有するジャーナルボックス、即ちアダプタブロックを有するシャシーを含む。各軸は、軸端から内側に軸に対し回転可能に取付けられた１対のホイールを有する。発電機は静止したステータ（２９）に対し回転運動する様固定されたロータ（２８）を含み、このような回転運動により回転しないハウジング（３２）内の発電機を含むステータに電流を生じる。特徴はロータを取付ける為に中空シャフト（３０）を設けることであり、シャフトは対応する軸端（２６）に摺動可能に受容され、且つ軸端にキー止めされる。最後に、ハウジングを回転しない様に固定する好適な手段は、突起（２２）にキー止めされた軸方向に延びるアーム（９２）である。
Patent JP-2001511714-A (JP)
Title: 化学的機械的研磨のための一体型パッド・ベルト構造
IPC: B24B21/00
Filed: 1998-02-11
Abstract: (57)【要約】
表面を研磨するための一体型パッド・ベルト構造であり、研磨パッドと一体化したベルトを包含し、この研摩パッドが継ぎ目無し研磨面を形成する。
Patent JP-2001513317-A (JP)
Title: モータ逆転回路
IPC: H02P7/00
Filed: 1998-02-05
Abstract: (57)【要約】
双方向ＤＣモータを作動させるために逆転回路が設けられる。この回路はＨブリッジ回路リレーを備えており、Ｈブリッジ回路リレーは第１と第２のリレーを有する。第１のリレーは第１の接点を第１の期間で接続し、モータの第１の接続を電力源に接続して第１のモードで作動させる。第２のリレーは第２の接点を第２の期間で接続し、モータの第２の接続を電力源に接続して第２のモードで作動させる。リレー回路はさらにスイッチを有し、このスイッチは少なくとも１つの接点を有し、この接点は第１または第２のリレー２をそれぞれ第１または第２の接続にもたらす。第３乗れイーがスイッチと動作的に関連して設けられており、モータの第３の接点を、少なくとも１つの接点が第１または第２のリレーを作動させるときに電力源に接続する。第３の接続は、少なくとも１つの接点が第１または第２のリレーを不活性化するとき第１または第２の接続の解除に先行して接続解除される。
Patent JP-2000508672-A (JP)
Title: 置換ベンジルアミン及びうつ病の治療のためのその使用
IPC: A61P25/22
Filed: 1997-04-15
Abstract: (57)【要約】
本発明は、式（Ｉ）［式中、Ｒ 1 及びＲ 2 は、同じか又は異なっていてよく、それぞれ、Ｃ 6-12 アリール、Ｃ 2-14 ヘテロアリール、Ｃ 6-12 アリールＣ 1-6 アルキル、Ｃ 2-14 ヘテロアリールＣ 1-6 アルキル（但し、アルキル、アリール又はヘテロアリール部は、Ｃ 1-6 アルコキシ、Ｃ 1-6 アルキル、Ｃ 3-6 シクロアルキル、Ｃ 4-6 シクロアルケニル、Ｃ 6-12 アリール、Ｃ 2-14 ヘテロアリール、ハロゲン、アミノ、ヒドロキシ、ハロＣ 1-6 アルキル、ニトロ、Ｃ 1-6 アルキルチオ、スルホンアミド、Ｃ 1-6 アルキルスルホニル、ヒドロキシＣ 1-6 アルキル、Ｃ 1-6 アルコキシカルボニル、カルボキシル、カルボキシＣ 1-6 アルキル、カルボキサミド及びＣ 1-6 アルキルカルボキサミドから選択された１個又はそれ以上の置換基により任意に置換されていてよい）、水素、Ｃ 1-6 アルキル、Ｃ 3-6 シクロアルキル、Ｃ 4-6 シクロアルケニル、Ｃ 2-6 アルケニル、Ｃ 2-6 アルキニル及びＣ 1-6 アルコキシＣ 1-6 アルキル（但し、アルキル、シクロアルキル、シクロアルケニル、アルケニル、アルキニル又はアルコキシアルキル部は、アミノ、ハロゲン、ヒドロキシ、Ｃ 1-6 アルキルカルボキサミド、カルボキサミド、カルボキシ、Ｃ 1-6 アルコキシカルボニル、Ｃ 1-6 アルキルカルボキシ及びカルボキシＣ 1-6 アルキルから選択された１個又はそれ以上の置換基により任意に置換されていてよい）から選択されるか又はＲ 1 及びＲ 2 の１個は上記定義した通りであり且つ１個はヒドロキシであり、Ｒ 3 及びＲ 4 は、同じか又は異なっていてよく、それぞれ、Ｃ 6-12 アリール、Ｃ 2-14 ヘテロアリール、Ｃ 6-12 アリールＣ 1-6 アルキル、Ｃ 2-14 ヘテロアリールＣ 1-6 アルキル（但し、アルキル、アリール又はヘテロアリール部は、Ｃ 1-6 アルコキシ、Ｃ 1-6 アルキル、Ｃ 3-6 シクロアルキル、Ｃ 4-6 シクロアルケニル、Ｃ 6-12 アリール、Ｃ 2-14 ヘテロアリール、ハロゲン、アミノ、ヒドロキシ、ハロＣ 1-6 アルキル、ニトロ、Ｃ 1-6 アルキルチオ、スルホンアミド、Ｃ 1-6 アルキルスルホニル、ヒドロキシＣ 1-6 アルキル、Ｃ 1-6 アルコキシカルボニル、カルボキシル、カルボキシＣ 1-6 アルキル、Ｃ 1-6 アルキルカルボキサミド及びカルボキサミドから選択された１個又はそれ以上の置換基により任意に置換されていてよい）、水素、Ｃ 1-6 アルキル、Ｃ 3-6 シクロアルキル、Ｃ 3-6 シクロアルキルＣ 1-6 アルキル、Ｃ 4-6 シクロアルケニル、Ｃ 2-6 アルケニル、Ｃ 2-6 アルキニル、Ｃ 1-6 アルコキシＣ 1-6 アルキル、ハロＣ 1-6 アルキル、ハロＣ 2-6 アルケニル、ハロＣ 2-6 アルキニル、シアノ、カルボキシル、Ｃ 1-6 アルキルカルボキシ及びカルボキシＣ 1-6 アルキル（但し、アルキル、シクロアルキル、シクロアルケニル、アルケニル、アルキニル又はアルコキシアルキル部は、アミノ、ヒドロキシ、Ｃ 1-6 アルキルカルボキサミド、カルボキサミド、カルボキシ、Ｃ 1-6 アルコキシカルボニル、Ｃ 1-6 アルキルカルボキシ及びカルボキシＣ 1-6 アルキルから選択された１個又はそれ以上の置換基により任意に置換されていてよい）から選択されるか又はＲ 3 若しくはＲ 4 の１個は、Ｒ 1 若しくはＲ 2 の１個及びそれが結合しているＮ原子と一緒に、５−又は６−員の複素環式環を形成し、Ｒ 5 は、ハロゲン、水素、Ｃ 1-6 アルキル及びＣ 1-6 アルコキシから選択された１個又はそれ以上の環置換基を表わし、そしてＲ 6 は、式（Ａ）（式中、点線は任意に存在する結合を表わし、Ｙは酸素又は−ＮＲ 8 （Ｒ 8 は水素又はＣ 1-6 アルキルである）であり、そしてＲ 7 は、水素、ハロゲン、ハロＣ 1-6 アルキル、Ｃ 1-6 アルキル及びＣ 1-6 アルコキシから選択された１個又はそれ以上の置換基を表わす）の単一の環置換基を表わす］のある種の新規なベンジルアミン誘導体又はその薬物的に許容される塩若しくは溶媒和物に関する。本発明はまた、その調製方法、それを含有する薬剤組成物及び医学療法、特にうつ病の治療に於けるその使用に関する。
Patent JP-2000508706-A (JP)
IPC: B01J20/22
Filed: 1997-04-23
Abstract: PCT No. PCT/EP97/02062 Sec. 371 Date Oct. 22, 1998 Sec. 102(e) Date Oct. 22, 1998 PCT Filed Apr. 23, 1997 PCT Pub. No. WO97/40088 PCT Pub. Date Oct. 30, 1997Process for preparing fine-particle, water-insoluble polymers of aziridines by polymerizing aziridines, preferably ethylenimine, in the presence of crosslinkers which contain at least two functional groups, and in at least one ether, and also modified, water-insoluble polymers of aziridines which can be obtained by reacting fine-particle, water-insoluble, crosslinked polymers of aziridines, in aqueous medium, with carbon disulfide or formaldehyde and a nucleophilic agent from the group consisting of alkali metal cyanides, primary amines, secondary amines, alkali metal sulfites and alkali metal phosphites, and use of the modified and non-modified fine-particle, water-insoluble polymers for immobilizing active compounds, as absorbents for aldehydes, ketones and acids, and also for removing heavy metal ions from wastewaters.
Patent JP-2000509296-A (JP)
IPC: A61B19/00
Filed: 1997-04-18
Abstract: The invention provides a method for magnetic resonance imaging and spectroscopic analysis of a specimen which includes positioning the specimen within a main magnetic field and introducing an antenna having a loopless antenna portion in close proximity to the specimen. Radio frequency pulses are provided to the region of interest to excite magnetic resonance signals, gradient magnetic pulses are applied to the region of interest with the antenna receiving magnetic resonance signals and emitting responsive output signals. A processor processes the responsive output signals to provide image information for display in a desired manner. The method in a preferred form involves employing a flexible antenna. The method in another preferred form involves employing an impedance matching circuit electrically interposed between the loopless antenna and the processor to enhance radio frequency power transfer and magnetic resonance signal-to-noise ratio from the loopless antenna to the processor. The method may be used on a wide variety of specimens and in a preferred use is introduced into small blood vessels of a patient to facilitate determination of atherosclerotic plaque. Medical intervention procedures, such as plaque removal, may be employed generally simultaneously with the imaging of the present invention. Corresponding apparatus and magnetic resonance antenna assembly are provided.
Patent JP-2000509715-A (JP)
Title: 炎症を処置するための方法
IPC: A61P29/00
Filed: 1997-04-29
Abstract: (57)【要約】
炎症性疾患、特に敗血症性ショック、ならびに炎症性腸疾患、慢性関節リウマチ、多発性硬化症、ブドウ膜炎、および乾癬のような自己免疫疾患によって起こる炎症性状態の処置または予防のための薬物の製造のためのIL-10とステロイドとの組合せの使用が提供される。IL-10および少なくとも１つのステロイド（例えば、ベタメタゾンまたはその誘導体）を含む、薬学的組成物およびキットもまた、提供される。
Patent JP-2001522234-A (JP)
Title: β−カテニン、ＴＣＦ−４およびＡＰＣは相互作用して癌を防ぐ
IPC: C12Q1/68
Filed: 1998-03-20
Abstract: (57)【要約】
APC癌抑制タンパタ質は、Tcf/Lef転写因子と相互作用することが最近示されたタンパク質である、β-カテニンに結合する。ここに、大腸上皮に発現している、Tcfファミリーの一員をコードする遺伝子（hTcf-4）をクローン化し、特徴付けた。hTcf-4は、β-カテニンと結合したときにのみ転写をトランス活性化する。APC -/- 大腸癌細胞の核に、Tcfレポーター遺伝子の転写によって測定されるように、構成的に活性な、安定なβ-カテニンhTCF-4複合体が含まれていることを見出した。APCを再び導入するとhTcf4からβ-カテニンが除かれ、転写のトランス活性化が失われた。APC機能の喪失に起因するTCF標的遺伝子の構成的な転写は、大腸癌の初期の悪性形質転換における決定的な出来事であり得る。大腸癌に見出される変異体APC遺伝子の産物はβ-カテニン/Tcf-4転写活性化の調節ができないことも、ここに示す。さらに、無傷のAPC遺伝子を持つ大腸癌が、機能的重要なリン酸化部位を変えるような、β-カテニンの微妙な活性化変異を含むことを示した。これらの結果は、β-カテニンの調節がAPCの腫瘍抑制効果に決定的であること、およびこの調節をAPCあるいはβ-カテニンのいずれかの変異によって回避し得ることを示している。
Patent JP-2001519802-A (JP)
Title: ハロフラボノイド及び／又はニトロ置換フラボノイドの抗不安薬としての使用
IPC: A61P25/22
Filed: 1998-03-25
Abstract: (57)【要約】
式（Ｉ）のフラボノイド化合物及びそのダイマーを用いて不安を治療する方法と、式（Ｉ）の化合物とそのダイマーと、式（Ｉ）の化合物の使用と、式（Ｉ）のフラボノイド化合物及びそのダイマーから成る薬学的製剤。
Patent JP-2002501489-A (JP)
Title: コード付きケミカルライブラリーの調製方法
IPC: C07B61/00
Filed: 1998-04-14
Abstract: (57)【要約】
コード付きケミカルライブラリーの調製方法であって、複数の合成用粒子上におけるケミカルライブラリーを合成し、ライブラリー合成中にこれら合成用粒子上に高エネルギー放射線を用いてコードを書き込み、これにより複数のコード付き合成用粒子上におけるケミカルライブラリーを調製し、そのコードを参照して、合成用粒子に結合したライブラリー化合物の識別を行う方法。
Patent MD-20050045-A (MD)
Inventor: BICICOV VLADIMIR
IPC: A63H3/26
Filed: 2005-02-15
Abstract: Inventia se refera la fabricarea jucariilor. Ecenta inventiei consta in aceea ca jucaria contine undispozitiv pentru eruptia lichidului, executat informa de membrana 2 cu volum variabil pentru umplere cu lichid cu o presiune mai mare decat cea atmosferica. Membrana 2 este dotata cu cel putin un tub capilar 11, iar in orificiul lui de intrare este instalata o supapa de retinere 10. Dispozitivul pentru schimbarea directiei si dinamicii eruptiei lichidului contine o placa mobila 14 cu orificii, in care sunt amplasate capetele tuburilor capilare11 cu posibilitatea abaterii lor. Jucaria continesuplimentar un dispozitiv pentru intreruperea eruptiei, executat ca o placa 16 cu orificiu, care este amplasata cu posibilitatea inchiderii tuturor tuburilor capilare 11 sau deschiderii lor selective. Pe suprafata corpului 1 jucariei poate fi aplicata o acoperire termosensibila.
Patent MX-163297-A (MX)
Inventor: LAURITZEN NELS JENS
IPC: A61F13/02
Filed: 1983-11-11
Abstract: Adhesive bandages comprising a pad area and adjacent adhesive-coated areas are prepared from a single sheet of heat-fusible bandage material, preferably a nonwoven batt material, by overlapping the center portion of the material in a Z-fold to form a triple thickness pad area, and heat calendaring the material adjacent the desired pad area to provide a surface suitable for coating with adhesive. The integrity of the pad is preserved by heat fusing the material along the folded edges of the pad.
Patent MX-160959-A (MX)
Inventor: KING PATRICK DANA
IPC: F27D3/15
Filed: 1984-03-23
Abstract: A sliding gate valve assembly employed on the side of a furnace as a furnace valve is so structured that the shut off of metal flow from the furnace occurs by directing the slide gate (21) to the up position rather than the down position. In addition, to facilitate a reduction in space at the slide gate, the slide gate is desirably configured to be asymmetrical, with the short end extending upwardly from the pour opening (29) in the nozzle. A refractory lined heat shield (26) protects the sliding gate carrier (22) and also serves to mount a collector extension (30) when used. The slide gate (21) is provided with a metallic frame (60) which retains a monolithic refractory (80) into which erosion resistant refractory inserts or performed members (29,70) are cast. Means are desirably provided to remove the spent refractory for remanufacture thereby reclaiming the casting. Similarly in the stationary plate (20), means are provided for remanufacture and for facilitating proper orientation of erosion-resistant refractory inserts in the manufacture of the stationary plate. The stationary plate is symmetrical to provide full travel pressure face relationship with the sliding gate (21). Both the stationary plate (20) and slide gate (21) casting have spring pad back up reinforcements. The statutory plate desirably has means for securing a well nozzle (19) to it.
Patent NZ-202143-A (NZ)
Title: Triorganotin-isocyanuric compounds and pesticidal compositions
Inventor: WEHNER W
IPC: A01N55/04
Filed: 1982-10-12
Abstract: There are described triorganotin-isocyanuric compounds of the formula <IMAGE>  (I)  wherein R is C1-C6-alkyl, phenyl, C5-C8-cycloalkyl or <IMAGE>  X is oxygen or sulfur, and Y1 and Y2 are each hydrogen or -Sn-R)3, as well as a process for producing this compound, and the use thereof for combating pests.
Patent NZ-202324-A (NZ)
Title: Cow milk increasing supplement with hydroxybutyric acid derivatives
Inventor: CUMMINS E W
IPC: A23K1/18
Filed: 1982-10-29
Abstract: The milk production of dairy cows is increased by incorporating as part of their diet a feed supplement containing an effective amount of  gamma -methylmercapto- alpha -hydroxybutyric acid and its oligomers. One may, for example, employ the supplement at a rate of from 1 to 2.5 kg per tonne of feed.
Patent NZ-210649-A (NZ)
Title: Shrouded electrical isolator
Inventor: MENNELL T W
IPC: H01H9/20
Filed: 1984-12-20
Abstract: An electrical isolator has an insulated housing with input and output conductors (1, 2) therein. A spring contact (6) is mounted within the housing for movement between open and closed positions. An insulating shroud (15) fully shields that part of the bridging contact accessible through an access opening of the housing. Manually operable pressure applying means may be operated when the bridging contact is in the closed position to control that contact between a tightened condition applying pressure between the bridging contact and the conductors without the use of springs, and a free condition wherein the contact pressure is reduced.
Patent NZ-222779-A (NZ)
Title: Loading and verifying program data
Inventor: NIBBY CHESTER M
IPC: G06F9/24
Filed: 1987-12-02
Abstract: A central subsystem of a data processing system includes a writable control store which is loaded with firmware to control the central subsystem operations. The central subsystem logic is responsive to a sequence of commands from a system management facility to load the control store and verify that the control store firmware is loaded correctly.
Patent NZ-239075-A (NZ)
Title: A cosmetic water-in-oil emulsion lipstick
Inventor: DUNPHY PATRICK JOSEPH
IPC: C09K23/14
Filed: 1991-07-22
Abstract: A cosmetic emulsion suitable for topical application to the lips comprises in addition to oil and water, an emulsifier system comprising:     i) as a first emulsifier, a phospholipid, and ii) a second emulsifier having a melting point of from -20 DEG C to 80 DEG C.   Preferred emulsions are lipsticks and lip gloss product which can additionally comprise wax.
Patent NZ-247904-A (NZ)
Title: Fungicidal and herbicidal 1,2,4-triazoles (where q is 1- or 4-(1,2,4-triazole))
Inventor: SHABER STEVEN HOWARD
IPC: C07D521/00
Filed: 1993-06-16
Abstract: Fungicidal and herbicidal compounds are disclosed having the formula   <CHEM>  wherein X is (C6-C10)aryl optionally substituted with up to three substituents which are independently hydroxy, halo, nitro, trihalomethyl, cyano, (C1-C4)alkyl, (C1-C4)alkoxy, (C1-C4)alkylthio, (C1-C4)alkylsulfinyl, (C1-C4)alkylsulfonyl, (C1-C4)alkoxy(C1-C4)alkoxy, (C1-C4)alkylcarbonyl, (C2-C8)alkenyl, (C2-C4)alkenyloxy, (C2-C8)alkynyl, (C2-C8)alkynyloxy, phenyl, phenyl monosubstituted with halo, alkyl or alkoxy, phenoxy or phenoxy monosubstituted with halo, alkyl or alkoxy; or a 5 or 6 membered heterocyclic ring having up to three different hetero atoms selected from nitrogen, oxygen and sulphur and optionally substituted with up to two substituents which are independently (C6-C10)aryl or halo; or X is substituted with -O- at the 2-position to complete a lactone with W; Q is 1-(1,2,4-triazolyl) or 4-(1,2,4-triazolyl) optionally substituted with up to two substituents which are independently halo, (C1-C4)alkyl, nitro, cyano, mercapto or (C1-C5)alkylmercapto; Z is cyano, alkoxycarbonyl, (C1-C12)alkyl, halo(C1-C12)alkyl, (C2-C8)alkenyl, halo(C2-C8)alkenyl, (C2-C8)alkynyl, (C3-C8)cycloalkyl, (C5-C8)cycloalkenyl, (C3-C8)cycloalkylalkyl, (C6-C10)aryl, (C7-C11)aralkyl, heterocyclyl or heterocyclyl(C1-C4)alkyl, provided X and Z are not heterocyclyl at the same time; W is -OK, -OR, -OR'OR'', -OR'Y, -OR'COOR'', -OR'OCOR'', -NB2, morpholinyl, piperidinyl, piperidinyl substituted with (C1-C4)alkyl, or an oxygen completing a lactone when joined with X; B is hydrogen, (C1-C12)alkyl, hydroxy(C3-C5)alkyl or (C2-C6)alkenyl; R is (C1-C12)alkyl, X, (C3-C8)alkenyl, (C3-C8)alkynyl, (C3-C8)cycloalkyl(C1-C5)alkyl, cyano(C1-C5)alkyl, hydroxy(C2-C4)alkyl or epoxy(C1-C5)alkyl, all of which are optionally halogenated, or is hydrogen; provided that when Z is phenyl, W is not NB2 and when Z is methyl, W is not methoxy;     R' is (-CH(CH3)-)p(-CH2-)n or (-CH2-)qCH=CH(-CH2-)m;     n is an integer from 0 to 6;     p is 0 or 1, provided n and p are not both 0;     q and m are each independently integers from 0 to 3; R'' is (C1-C6)alkyl, X, Y-(C1-C4)alkyl or (C1-C2)trialkylsilyl(C1-C4)alkyl, all optionally halogenated, or hydrogen; and Y is phenyl, naphthyl, piperidinyl, triazolyl, pyrazinyl, phthalimido, morpholinyl, pyridyl, thienyl, furyl or (C3-C8)cycloalkyl, all of which may be optionally substituted with the substituents defined for X; and the agronomically acceptable enantiomorphs, acid addition salts and metal salt complexes thereof. Processes for making the compounds are also disclosed.
Patent NZ-258116-A (NZ)
Title: 5-amino-3-aminomethyl-indan, -benzofuran, and -benzothiophene derivatives; pharmaceutical compositions
Inventor: PERREGAARD JENS KRISTIAN
IPC: C07C233/43
Filed: 1993-12-08
Abstract: Compounds of formula I    <IMAGE>  I  wherein R1=(cyclo)alk(en)yl, aralkyl, alkyl(oxy)carbonyl, CONH2, etc.; R2=H, (cyclo)alk(en)yl, aralkyl, etc.; R3-R5=H, halo, alkyl, alkoxy, etc.; R6,R7=H, alkyl; R6R7=atoms to complete a ring; R8,R9=groups cited for R2, 2-oxoimidazolidinoalkyl, etc.; NR8R9=heterocyclyl; 1 of X,Y=CH2 and the other=CH2, O, S were prepd. Thus, 1-indancarboxylic acid was converted in 5 steps to 1-(N,N-dipropylaminomethyl)-6-formylaminoindane oxalate which had ED50 of 0.0055.mu.M/kg s.c. in the 8-OH DPAT cue agonism test in rats.
Patent NZ-272208-A (NZ)
Title: Composition comprising an active substance occluded within a dendrimer which has terminal groups containing blocking groups
Inventor: JANSEN JOHAN FRANZ GRADUS ANTO
IPC: A61K47/48
Filed: 1995-05-25
Abstract: The invention relates to a composition consisting of a dendrimer provided with blocking agents and an active substance occluded in the dendrimer. According to the invention a blocking agent is a compound which is sterically of sufficient size, which readily enters into a chemical bond with the terminal groups of a dendrimer and which can also be split off from the dendrimer or be modified without thereby affecting the chemical structure of the dendrimer and the active substance. The blocking agent can be provided with protective groups. Such conjugates have the advantage that the time at which the releasing of the active substance starts, can be controlled. The invention also relates to a process for the preparation of such a composition and to a process for the controlled release of the active substance.
Patent NZ-330475-A (NZ)
Title: Antibodies, and use thereof in measuring lipid peroxidation in biological samples and method for inducing inflammation
Inventor: PARTHASARATHY SAMPATH
IPC: C07K17/02
Filed: 1997-09-19
Abstract: A method and kit for the diagnosis and quantification of the state of oxidation, and more specifically, the level of lipid peroxidation, of a host is provided that includes contacting a host biological sample with an antibody to an antigen formed by the reaction of a lipid hydroperoxide with a primary amine.  This method assesses the risk of, or existence of, oxidative damage in the host.  The invention also includes monoclonal and polyclonal antibodies, as well as antibody fragments, optionally in purified or isolated form.
Patent NZ-334957-A (NZ)
Title: Bracket with flanged base and cantilever beam
Inventor: MCDONALD RODERICK RAYMOND
IPC: A47B96/06
Filed: 1999-03-31
Abstract: A cantilever bracket includes a mounting plate 11 which has flanges extending from each side.  These flanges contact the surface to which the bracket is attached.  A cavity 19 is formed in plate 11 by pressing the material inwards so that it projects in the same direction as the flanges.  The cavity contains a hole 20 for a fastener.  A cantilever beam 13 extends outwards from the mounting plate.  The cantilever beam is U-shaped with the sides 14 bent inwards to form a U-shape as at 15.
Patent NZ-501402-A (NZ)
Title: Toilet system with vacuum suction
Inventor: HABERZETTL MICHAEL
IPC: E03F1/00
Filed: 1998-06-03
Abstract: A toilet system with vacuum suction, in which an insert (1) is placed in a toilet bowl (10).  The insert has a stench trap (6) at the bottom end, and is connected at the top edge to a flushing pipe with flushing nozzles (7), which can be connected to a pressurized water pipe (2).  The stench trap (6) is connected via a suction conduit (3) to a suction unit, which can be emptied via a floor drain into a collecting basin or into the sewerage system.
Patent NZ-502795-A (NZ)
Title: Method of identifying molecular interactions employing counterselection and at least two hybrid molecules or two hybrid systems
Inventor: VIDAL MARC
IPC: C12Q1/68
Filed: 1996-04-11
Abstract: A method for determining whether a first test protein is capable of interacting with a second test protein comprises: (a)  providing in a cell: (i) one or two different reporter genes each operably linked to a different  DNA-binding-protein recognition site and (ii) a first fusion gene which expresses a first hybrid protein, the first hybrid protein comprising a test protein covalently bonded to a DNA-binding moiety which is capable of specifically binding to the DNA-binding-protein recognition site; (iii) a second fusion gene which express a second hybrid protein, the second hybrid protein comprising a test protein covalently bonded to a gene activating moiety and (b) detecting expression of the reporter gene as a measure of the ability of the first test protein to interact with the second test protein. A method for determining whether a first and second test protein is capable of interacting with a third test protein comprises: (a) providing in a cell: (i) at two different  reporter genes each operably linked to a different  DNA-binding-protein recognition site; (iv) a first fusion gene which expresses a first hybrid protein, the first hybrid protein comprising the first test protein covalently bonded covalently bonded to a DNA-binding moiety which is capable of specifically binding to the DNA-binding-protein recognition site; (ii) a second fusion gene which expresses a second hybrid protein, the second hybrid protein comprising the second test protein covalently bonded covalently bonded to a DNA-binding moiety which is capable of specifically binding to the DNA-binding-protein recognition site (iii) a third fusion gene which expresses a third hybrid protein, the third hybrid protein comprising a third test protein covalently bonded to a gene activating moiety and (b) detecting expression of the reporter gene as a measure of the ability of the first test protein to interact with the second test protein. Also disclosed is the cell as described above.