baber/WOPTO huggingface dataset:
Patent SI-3000808-T1 (SI)
Title: 5-((halophenyl)-3-hydroxy-pyridin-2-yl)-carboxylic acid derivatives as intermediates for the preparation of carbonylamino alkanoic acids, esters and amides thereof
Inventor: LANTHIER CHRISTOPHER M
IPC: C07D213/00
Filed: 2012-06-05
Abstract: Disclosed are processes for preparing [(3-hydroxypyridine-2-carbonyl)amino]-alkanoic acids, derivatives, inter alia, 5-aryl substituted and 5-heteroaryl substituted [(3-hydroxypyridine-2-carbonyl]amino}acetic acids. Further disclosed are methods for making prodrugs of [(3-hydroxypyridine-2-carbonyl)-amino]acetic acids, for example, [(3-hydroxypyridine-2-carbonyl]amino}acetic acid esters and {[3-hydroxypyridine-2-carbonyl]amino}acetic acid amides. The disclosed compounds are useful as prolyl hydroxylase inhibitors or for treating conditions wherein prolyl hydroxylase inhibition is desired.
Patent SI-2944633-T1 (SI)
Title: Pyridine derivative
Inventor: MARUYAMA AKINOBU
IPC: C07D409/00
Filed: 2013-11-13
Abstract: Provided is a pyridine derivative represented by formula (I), a prodrug thereof, a pharmaceutically acceptable salt of the pyridine derivative or the prodrug, or a solvate of the pyridine derivative, the prodrug or the pharmaceutically acceptable salt, which is useful for treatment or prophylaxis of diseases associated with URAT1 such as gout, hyperuricemia, hypertension, kidney diseases such as interstitial nephritis, diabetes, arteriosclerosis and Lesch-Nyhan syndrome.
Patent TR-200701771-T1 (TR)
Title: Bir pişirici cihaz.
Inventor: KAYIHAN S ASLI
IPC: F24C15/12
Filed: 2005-10-06
Abstract: Bu buluş, estetik bir görünüm oluşturan ve temizlik şartlarını sağlayan, üst kapağın (3) açılıp kapanmasıyla ileriye ve geriye doğru hareket edebilen bir bek tablası (4) içeren bir pişirici cihaz (1) ile ilgilidir.
Patent DE-3688418-T2 (DE)
Inventor: KUSHNER PETER
IPC: C07K14/61
Filed: 1986-02-11
Granted: 1993-08-26
Abstract: An expression system for recombinant production of a desired protein comprises CHO cells transformed with a DNA sequence having the desired protein coding sequence under control of the human metallothionein-II promoter. The cells can be maintained on serum-free medium and induced in the presence of an induction mediator. In addition, the system may include an enhancer element and/or a resistance-conferring gene to provide increased levels of expression. The system can process genomic as well as intronless DNA, and is capable of producing proteins which have the same characteristics as those obtained from native sources. Human growth hormone which is indistinguishable from that produced by the pituitary has been thus produced.
Patent DE-3751148-T2 (DE)
Inventor: STUBER ISTVAN
IPC: G02B21/00
Filed: 1987-12-10
Granted: 1995-07-06
Abstract: The depth sharpness increasing device has an image forming layer (6) inserted between a primary (5) and secondary magnifier (7) of the composite magnifying system, in respect to the travel of the beam after the object (4) in the image plane of the primary magnifier. The layer is formed by independent particles dispersed in a medium, the index of refraction which differs from that of the particles. The image forming layer is displaceable in the image plane so that miages coincide with the object plane of the secondary magnifier. - The primary magnifier may consist of a primary objective and primary ocular or projector, while the secondary magnifier comprises a secondary objective and a secondary ocular or projector.
Patent DE-3788404-T2 (DE)
Inventor: LINKSY CARY BRUCE
IPC: A61L15/00
Filed: 1987-09-28
Granted: 1994-05-05
Abstract: An improved adhesion-preventative barrier fabric comprising an oxidized regenerated cellulose (ORC) fabric (or matrix having equivalent properties) which is drapable, conformable, adherent to body organs, and substantially absorbable within thirty (30) days in the body, which fabric has heparin absorbed thereon, said heparin being present in a non-toxic, adhesion-preventative, effective amount and potency; and, the process of using said improved barrier fabric or matrix to administer heparin to prevent surgical adhesions.
Patent TR-199801780-T2 (TR)
Title: Silindir seklindeki yükleri araç üstüne tespit etmek için sökülüp takilabilir tertibat.
Inventor: THIRIET DANIEL
IPC: B60P7/12
Filed: 1997-03-12
Abstract: Bobin gibi silindir seklindeki yüklerin, yükleme tabanli bir araç üstüne tesbiti için sökülüp-takilabilir bir tertibat. Tesbit tertibatinda en az bir çerçeve sirasi (A,B) olusturacak sekilde ard arda sirasiyla yükleme tabaninin üstüne yerlestirilen birçok kati çerçeve (1) vardir, bu kati çerçevelerin (1) her birinde, çerçevenin (1) üstüne sökülüp-takilabilir sekilde tutturulmus iki egik kama (3) bulunur .
Patent TR-199802788-T2 (TR)
Inventor: TSAMOURGELIS ILIAS
IPC: B65D5/00
Filed: 1997-06-30
Abstract: Bu bulus, her defasinda ve her kenar için kagit dalgalarinin düzenlenmesinin ayri ayri belirlenmesini gerektiren birçok sert kagit veya kivrilmis levhadan olusabilen, ürünlerin paketlenmesi ve tasinmasi için ekonomik bir karton kutu ile ilgilidir. Böyle  bir ekonomik karton kutuda kenarlarin (A1,A2,A3) uzantilari (F1,F2,...,F6)90  içe dogru dönerler ve böylece küçük kenarlarin (A4,A5)dis kisimlari ile uygun olarak ve F2 ve F8 ile tabana (A2) yapistirilabilir. Uzantilar (N1,N2) dönerek disaridan kenarlara (A4 ve A5) yapisirken küçük kenarlarda sütunlar (K1,K2,K3.K4) olusturulur. Kenarlarin (A1,A3) yüksekligi, karton kutunun yüksekligine denk olunca, uzantilar (N1,N2) karton kutunun kapagini teskil ederler. Kenarlarin (A4 ve A5) çikintilari (P1,P2,P3,P4), kutularin üst üste yerlestirilmesi esnasinda araliklara (E1,E2, E3,E4) uygun olarak girer.
Patent TR-199901839-T2 (TR)
Inventor: SKOWRONSKI RICHARD
IPC: H02G11/02
Filed: 1998-01-16
Abstract: Gizlenebilir bir çikrik tertibati; arka tarafta bulunan iki adet damla sekilli mafhaza ile mahfaza içine yerlestirilmis olan ve bir eksen etrafinda dönmek üzere mile oturtulmus olanbir makaradan meydana gelir. Makara ve mahfaza, eksen etrafindaki  mahfaza içerisinde ok sayida göz bulundugunu gösterir. Makara ve mahfaza; ayni zamanda, gizlenebilir bir sekilde içlerine saklanan ikinci uzunluktaki bir kablodan ibaret bir kablo saklama gözü ile yine içlerine saklanan belli uzunluktaki bir kablodan ibaret bir kablo uzatma gözü, yani biryay gözü ile bir de kilitgözü vazifesi görürler. Mahfazanin ayrica ikinci bir paralel eksen üzerinde bulunan yay germe bölmesi ile kablo ayarlama bölmesi mevcuttur. Sabit güçlü bir yay; makaranin kablo gizleme yönünde dönmesini saglamak üzere yay saklama gözünden yay germe bölgesine kadar uzanir.
Patent TR-199902197-T2 (TR)
Inventor: WOLFF HANS-PETER
IPC: C07D277/00
Filed: 1998-03-17
Abstract: Formül (III)'e uygun bilesiklerin eldesi için olup FORMÜL (III).burada: A;CH=CH vya S;W,O;X,S,O veya NR2; buradaki R2 kismi hidrojen veya C1-C6 alkildir; Y, CH veya N; R, ihtiyari olarak C1-C3 alkil, CF3, C1-C3 alkoksi, F,CI veya brom ile mono veya di-sübstitüe olmus naftil, tiyenil veya fenil; R1, hidrojen veya C1-C6 alkil ve; n, 1-3 demektir, özelligi,A,W,X,Y,R,R1 ve n'nin yukaridaki gibi tanimlandigi Formül (IV) 'e uygun bir bilesigin, protik bir çözücü madde içinde metalik alüminyum ile indirgenmesidir. FORMÜL (IV).
Patent DE-60005001-T2 (DE)
Inventor: KENCHAMMANA-HOSEKOTE R
IPC: H04L12/56
Filed: 2000-03-28
Granted: 2004-07-08
Abstract: A network scheduler for real time applications is described. The network scheduler supports scheduling of network packets in a multi-threaded operating system to insure correct scheduling order and to preclude kernel preemption of active threads. The network scheduler resides between a kernel (and device drivers) and multiple sessions at the user-level. The network scheduler uses input/output control primitives such as HOLD and RELEASE to control servicing of the queues of packets at the kernel or network device driver. The control primitives serve as a middleware interface to the underlying kernel or network device driver. The network scheduler functions as a proxy scheduler to manage the queues of packets at the kernel or network device driver.
Patent DE-60015729-T2 (DE)
Inventor: SERBAN BOGDAN
IPC: B60R21/015
Filed: 2000-02-28
Granted: 2005-12-29
Abstract: A system for stopping the deployment of an airbag in a vehicle includes a detector for detecting a position of the airbag with respect to an occupant of the vehicle and an airbag operating device. The detector is located on the airbag in an area which, upon deployment of the airbag, is facing the occupant of the vehicle. The detector generates a position signal which is sent to the airbag operating device such that the airbag operating device stops the deployment of the airbag when the position signal indicates a predetermined position of the airbag in relation to the occupant.
Patent DE-60019011-T2 (DE)
Inventor: SPATAFORA MARIO
IPC: B65B11/28
Filed: 2000-04-06
Granted: 2006-04-27
Abstract: The invention relates to a method and device for continuously wrapping products (3), according to which, during the continuous feed of the products (3) and respective intermediate wrappers (2a) which have four flaps (26, 27, 28, 29) to be folded, projecting in such a way that they are offset from the lower surface (30) of the product (3), along a path (P) with an instantaneous tangent (T) extending in a first direction (D1) which may vary from point to point on the path (P), two opposite flaps (28, 26) make contact with respective first and second folding tools (36, 37), located on opposite sides of an intermediate folding portion (100) of the path (P). During their movement along respective closed paths (01, 02), the first and second folding tools (36, 37) are subject to a first movement in a second direction (D'2, D''2) transversal to the first direction (D1), a second movement in the first direction (D1), and a third movement, consisting of an oscillation about a relative longitudinal axis (97, 98), so that each folding tool (36, 37) pursues and folds each flap (28, 26), whilst remaining parallel with the instantaneous tangent (T) and, therefore, with the surface (30) of each product (3). <IMAGE>
Patent DE-60019088-T2 (DE)
Inventor: BEUDON DIDIER
IPC: F24F13/068
Filed: 2000-01-25
Granted: 2006-02-02
Abstract: An installation includes a worktop, a first wall and a device for the close protection of products arranged on the worktop, whereby the products are sensitive to contamination from the ambient environment. The products are protected by diffusion of a sterile air stream in a direction substantially perpendicular or parallel to the worktop. The device extends along the worktop and has a least one end adjoining the first wall so that there is an air gap between the end and the first wall. The end is formed by a porous second wall made of perforated material, extending substantially perpendicular to a longitudinal axis of the device, in such a way as to create in the gap a sterile air leakage directed outward away from the worktop, whereby the sterile air leakage counters any ambient air induction into the gap toward the worktop.
Patent DE-60021039-T2 (DE)
Inventor: ROOM THIERRY
IPC: A47C31/11
Filed: 2000-10-04
Granted: 2006-06-29
Abstract: Seat cover comprises envelope (1) with two sections (2, 2') attached to each other by seam (3). Envelope has opening means (7) allowing seam to give way under predetermined stress, but ensuring resistance for smaller stress, so that gap (8) can appear or not between two sections depending on stress applied. Opening means includes reinforcement element (9) placed parallel to seam and comprising braid (10).
Patent DE-60029141-T2 (DE)
Inventor: AHLGREN JONNI
IPC: D21H23/14
Filed: 2000-12-04
Granted: 2007-01-11
Abstract: The invention relates to a method for the production of paper or board, wherein retention aids are added to the stream of stock. Improved retention and more effective dewatering are achieved by adding to the stream of stock a cationic polymer solution and a suspension-form microparticle mixture composed of a swellable clay of the smectite group and a colloidal synthetic metal silicate in which the prevalent cation is magnesium.
Patent DE-60029588-T2 (DE)
Inventor: MAUBLANT JEAN
IPC: G01T1/164
Filed: 2000-06-22
Granted: 2007-08-09
Abstract: This invention concerns a device for detecting and locating a radioactive source emitting gamma rays, characterized in that it comprises: first means for determining the direction of the gamma radiation emitting source relative to the centre of the detector comprising: gamma radiation sensing means; a plurality of means for evaluating the gamma radiation flux; means analyzing the gamma radiation flux for determining the direction of-the radiation source; second means for directing the radioactive emitting source comprising mechanical means for causing the device to move, so as to bring its centerline nearer the gamma radiation emitting source; means physically representing the device centerline.
Patent DE-60033932-T2 (DE)
Inventor: COOKE JOHN P
IPC: A61K38/08
Filed: 2000-06-05
Granted: 2007-12-06
Abstract: Cardiovascular cell proliferation in a blood vessel subjected to trauma, such as angioplasty, vascular graft, anastomosis, or organ transplant, can be inhibited by contacting the vessel with a polymer consisting of from 6 to about 30 amino acid subunits, where at least 50% of the subunits are arginine, and the polymer contains at least six contiguous arginine subunits. Exemplary polymers for this purpose include arginine homopolymers 7 to 15 subunits in length.
Patent DE-60034158-T2 (DE)
Inventor: FUJIWARA TAKAYUKI
IPC: B65H19/22
Filed: 2000-06-21
Granted: 2007-12-13
Abstract: A film winding apparatus has a film winding mechanism (50) for rotating a roll core (28) to wind an elongate film (24) around the roll core (28) thereby to produce a film roll (30), a product receiving mechanism (52) for gripping the film roll (30) while tensioning the elongate film (24), the product receiving mechanism (52) being displaceable away from the film winding mechanism (50), and a cutting mechanism (54) for transversely cutting off the elongate film (24) while the elongate film (24) is being tensioned by the product receiving mechanism (52). The elongate film (24) can be wound highly accurately around the roll core (28) with a simple process and arrangement.
Patent DE-60105154-T2 (DE)
Inventor: COLDREN A
IPC: H01S5/20
Filed: 2001-06-01
Granted: 2005-09-08
Abstract: A tunable laser is disclosed including a gain section for creating a light beam over a bandwidth, a phase section for controlling the light beam around a center frequency of the bandwidth, a waveguide for guiding and reflecting the light beam in a cavity including a relatively low energy bandgap separate-confinement-heterostructure (SCH), a front mirror bounding an end of the cavity and a back mirror bounding an opposite end of the cavity wherein gain is provided by at least one of the group comprising the phase section, the front mirror and the back mirror.
Patent DE-60115054-T2 (DE)
Inventor: ALLEN SHELLEY JANE
IPC: A61K38/17
Filed: 2001-08-17
Granted: 2006-07-27
Abstract: This invention relates to the treatment of cancer and is particularly, though not exclusively concerned with the treatment of pancreatic cancer. In particular the invention related to the use of TrkAIg2 in the preparation of a medicament for the treatment and/or prevention of cancer in a patient.
Patent DE-60115176-T2 (DE)
Inventor: PRINCE JONATHAN WILLIAM
IPC: A47C1/03
Filed: 2001-09-26
Granted: 2006-07-13
Abstract: An arm assembly (24) is provided for a chair (12). The chair (12) has a forward direction and a rearward direction. The arm assembly (24) comprises an armrest (26) and a support structure (28). A mounting device movably mounts the armrest to the support structure. The mounting device constrains the movement of the armrest (26) relative to the support structure to movement in a substantially horizontal plane having two degrees of freedom defined by first and second transversely arranged axes lying within the substantially horizontal plane. The armrest (26) thus move in a substantially planar fashion without changing the orientation of the armrest (26).
Patent DE-60116270-T2 (DE)
Inventor: CARLSSON LEIF
IPC: B21D5/01
Filed: 2001-02-22
Granted: 2006-08-24
Abstract: Workpiece controlled shaping of metal, preferably in the form of plates or bands of high tensile limit, preferably above 1000N per square mm, comprises heat treating the workpiece in planar form along notches or zones to reduce locally the tensile limit. The workpiece is then bent, folded or shaped along the heat-treated notches or zones, either directly or after cooling.
Patent DE-60119124-T2 (DE)
Inventor: CAI HUI
IPC: A61K31/275
Filed: 2001-08-10
Granted: 2006-11-30
Abstract: Substituted pyrazoles of general formula methods of manufacturing them, compositions containing them, and methods of using them to, for example, treat autoimmune diseases mediated by cathepsin S, and inhibit cathepsin S activity, are described.
Patent DE-60122575-T2 (DE)
Inventor: SUI ZHIHUA
IPC: A61P15/08
Filed: 2001-12-11
Granted: 2007-09-13
Abstract: The present invention is directed to novel 7-heterocyclyl quinoline and thienoÄ2,3-bÜpyridine derivatives of the general formula (I) or (II), wherein all variables are as herein defined, pharmaceutical compositions containing them and their use in the treatment of disorders and conditions associated with gonadotropin releasing hormone (GnRH). The compounds of the invention are antagonists of GnRH, useful in the treatment of the infertility, prostate cancer, benign prostate hyperplasia (BPH) and as contraceptives.
Patent DE-60124460-T2 (DE)
Inventor: WHITSON ROBERT C
IPC: G01N33/49
Filed: 2001-07-02
Granted: 2007-09-20
Abstract: A test sensor (360) for use in the determination of the concentration of a chemical in blood, the test sensor comprising: a housing having a disposable end cap (350) at a test end, the removable end cap including an aperture at the test end; a test chamber (202) disposed within the end cap, the test chamber having an inset (208) disposed adjacent to the aperture in the test end, the test chamber being adapted to collect blood through the inlet; and a lance (203) disposed within the end cap of the housing and coupled to the test sensor, an actuation of the lance causing the lance to extend through the aperture of the end cap, the lance being disposable with the disposable end cap. The lance comprises a spring (212) having a first end (218) and a second end (220) disposed between a needle (206) and a base (204) wherein the first end of spring is coupled to the base and the second end of the spring is coupled to the needle.
Patent DE-60124545-T2 (DE)
Inventor: BUELOW MARTIN
IPC: B01J20/34
Filed: 2001-09-13
Granted: 2007-08-09
Abstract: An adsorbent composition, which is comprised by both an active adsorbent component and an active thinner component, is disclosed. The active thinner component will range in weight from about 5 % to about 80 % of the composition. The adsorbent composition is useful in separating a gas component from a gas mixture such as in cyclic adsorption processes.
Patent DE-60127166-T2 (DE)
Inventor: GROVER RAYMOND J
IPC: H01L27/04
Filed: 2001-11-16
Granted: 2008-01-10
Abstract: Trench-gate field-effect transistors, for example power MOSFETs, are disclosed having trenched electrode configurations (11,23) that permit fast switching of the transistor, while also providing over-voltage protection for the gate dielectric (21) and facilitating manufacture. The gate electrode (11) comprising a semiconductor material of one conductivity type (n) is present in an upper part of a deeper insulated trench (20,21) that extends into a drain region (14,14a) of the transistor. A lower electrode (23) connected to a source (13,33) of the transistor is present in the lower part of the trench. This lower electrode (23) comprises a semiconductor material of opposite conductivity type (p) that adjoins the semiconductor material of the gate electrode (11) to form a p-n junction (31) between the gate electrode (11) and the lower electrode (23). The p-n junction (31) provides a protection diode (D) between the gate electrode (11) and the source (13,33). The gate electrode (11) is shielded from most of the drain region by the lower electrode (23), so reducing the gate-drain capacitance and improving the switching speed of the transistor.
Patent DE-60129242-T2 (DE)
Inventor: FOX ALYSON
IPC: A61P19/08
Filed: 2001-11-27
Granted: 2008-03-13
Abstract: A method for the treatment of pain, in particular antinociceptive or anti-allodynic treatment of pain, in a patient in need of such treatment, e.g. a patient with osteoporosis or osteopenia, a tumour patient or a patient suffering from an inflammatory disease, which comprises administering an effective amount of a bisphosphonate, e.g. zoledronic acid or salts or hydrates thereof, to the patient
Patent DE-60130640-T2 (DE)
Inventor: DELUCA HECTOR F
IPC: C07F7/18
Filed: 2001-03-29
Granted: 2008-07-17
Abstract: This invention provides a novel class of vitamin D related compounds, namely, the 2-alkylidene-19-nor-vitamin D derivatives, as well as a general method for their chemical synthesis. The compounds have the formula: where Y1 and Y2, which may be the same or different, are each selected from the group consisting of hydrogen and a hydroxy-protecting group, R6 and R8, which may be the same or different, are each selected from hydrogen, alkyl, hydroxyalkyl and fluoroalkyl, or when taken together represent the group -(CH2)X- where X is an integer from 2 to 5, and where the group R represents any of the typical side chains known for vitamin D type compounds. These 2-substituted compounds are characterized by relatively high intestinal calcium transport activity and relatively high bone calcium mobilization activity resulting in novel therapeutic agents for the treatment of diseases where bone formation is desired, particularly low bone turnover osteoporosis. These compounds also exhibit pronounced activity in arresting the proliferation of undifferentiated cells and inducing their differentiation to the monocyte thus evidencing use as anti-cancer agents and for the treatment of diseases such as psoriasis.
Patent DE-60131765-T2 (DE)
Inventor: PERROT SEBASTIEN
IPC: H04L12/56
Filed: 2001-10-18
Granted: 2008-11-20
Abstract: Method for linking a first and a second communication bus through a wireless link, comprising a first portal connected to the first bus and a second portal connected to the second bus, said first and second portal communicating over a wireless connection. The method comprises the steps of: associating the two portals to the wireless network; exchanging, between the two portals of self identification packets of nodes connected to their respective local busses, including the self identification packets of the portals themselves; generating a reset on each bus; carrying out a self identification procedure on each bus, where each portal generates self identification packets for itself and for nodes of the respective remote bus, using the self identification packets received following the association step.
Patent DE-60201263-T2 (DE)
Inventor: PHILLIPS JEFFREY
IPC: F16D65/06
Filed: 2002-03-08
Granted: 2005-09-29
Abstract: A disc brake friction pad (10, Fig 1(a)) has a back plate (12) and friction material mounted thereon as an array of discrete friction elements (20). The elements are each resiliently mounted on an end region (58) of an individually associated support spring finger (52, Fig 2(a)) and the other end region (56) of the finger is secured against to the back plate. The end regions are substantially parallel and separated by a central region (60) inclined with respect thereto at an angle of about 30 DEG  to displace the second end region and its friction element from the back plate. The support spring finger is stiff but has resilience, at least in the central region adjoining the end regions, permitting the friction element to be resiliently displaced towards the back plate against the restoring bias of the finger. The shape of the finger permits the friction element to displace with little rotation. The support spring fingers may alternatively be formed as tongues (752, Fig 8) cut from, and deflected out of, the back plate.