Patent IL-131865-A (IL)
Title: Substituted salicyclic acid amides, processes for their production and bactericides and fungicides containing them
IPC: C07D285/08
Filed: 1998-03-02
Abstract: Compounds of the formula wherein: X represents NO2, NH2 or R1-(C=O)-NH-; R1 represents hydrogen, methyl or methoxy; R represents hydrogen or benzyl; Y1, Y2, Y3, Y4 and Y5 are identical or different and each represents hydrogen, fluorine, chlorine, bromine, cyano, methyl, ethyl, methoxy, trifluoromethyl or 2259 י" ד באלול התשס" ד - August 31, 2004 difluoromethoxy, and either Y2 or Y3 represents -G-Z, in which G represents -A-Ar1- or -T-Ar1-O-, in which Ar1 represents 1,2,4-thiadiazolediyl, 1,3,4-thiadiazolediyl, 1,2,4-oxadiazolediyl, 1,3,4-oxadiazolediyl or represents pyridinediyl, pyrimidinediyl or 1,3,5-triazinediyl, each of which is optionally mono- or disubstituted by identical or different substituents selected from the group consisting of fluorine, chlorine, cyano, methyl, cyclopropyl, methoxy, methylthio, trifluromethyl, difluoromethoxy, trifluoromethoxy, difluorochloromethoxy, T represents a single bond, represents oxygen, sulphur, -CH2-O-, CH2-S-, methylene, ethylene or propylene and Z represents methyl, ethyl, n- or i-propyl, n-, i-, s- or t-butyl, which is optionally mono- to trisubstituted by identical or different substituents selected from the group consisting of fluorine, chlorine, cyano or methoxy; represents in each case optionally fluorine- or chlorine-substituted vinyl, allyl or propargyl; represents cyclopropyl, cyclobutyl, cyclopentyl or cyclohexyl, each of which is optionally mono- to trisubstituted by identical or different substituents selected from the group consisting of fluorine, chlorine, cyano, methoxy, phenyl, methyl or ethyl; or Z represents phenyl, pyridyl, pyrimidyl or thienyl, each of which is optionally mono- to trisubstituted by identical or different substituents, where the possible substituents are selected from the list below: fluorine, chlorine, bromine, cyano, methyl, ethyl, n- or i-propyl, n-, i-, s- or t-butyl, methoxy, ethoxy, n- or i-propoxy, methylthio, ethylthio, n- or i-propylthio, methylsulphinyl, ethylsulphinyl, methylsulponyl or ethylsulphonyl, trifluoromethyl, trifluoroethyl, difluoromethoxy, trifluoromethoxy, difluorochloromethoxy, trifluoroethoxy, difluoromethylthio, trifluoromethylthio, difluorochloromethylthio, trifluoromethylsulphinyl, trifluoromethylsulphonyl, methoxycarbonyl, ethoxycarbonyl or phenoxy; in each case doubly attached methylenedioxy, ethylenedioxy, each of which is optionally mono- to tetrasubstituted by identical or different substituents selected from the group consisting of fluorine, chlorine, methyl, trifluoromethyl and ethyl, cyclopropyl, cyclobutyl, cyclopentyl, cyclohexyl, phenyl, phenoxy, or a grouping in which A1 represents methyl, ethyl, n- or i-propyl, n-, i-, s- or t-butyl, cyclopropyl or cyclobutyl, A2 represents methyl, ethyl, n- or i-propyl, n-, i-, s- or t-butyl, allyl, propargyl, but- 2-en-l-yl, 2-methyl-prop-1-en-3-yl, cyanomethyl, methoxymethyl, ethoxymethyl, methoxyethyl, ethoxyethyl, methylthiomethyl, ethylthiomethyl, methythioethyl, ethylthioethyl, dimethylaminomethyl, dimethylaminoethyl, methylaminomethyl, methylaminoethyl or benzyl, or a grouping 2260 י" ד באלול התשס" ד - August 31, 2004 in which A3 represents methyl or ethyl and A4, A5, A6 and A7 are identical or different and independently of one another each represents hydrogen, methyl, ethyl, n- or i-propyl, n-, i-, s- or t-butyl, hydroxymethyl, trifluoromethyl or trifluoroethyl, or A4 and A5 or A4 and A6 or A6 and A7 together with the respective carbon atoms to which they are attached form a cycloaliphatic ring having five, six or seven carbon atoms.