baber/WOPTO huggingface dataset:
Patent SK-5802002-A3 (SK)
Title: Pharmaceutically active sulfonamide derivatives
Inventor: ARKINSTALL STEPHEN
IPC: A61K31/4525
Filed: 2000-09-28
Abstract: The present invention is related to sulfonamide derivatives of formula I notably for use as pharmaceutically active compounds, as well as to pharmaceutical formulations containing such sulfonamide derivatives. Said sulfonamide derivatives are efficient modulators of the JNK pathway, they are in particular efficient and selective inhibitors of JNK 2 and 3. The present invention is furthermore related to novel sulfonamide derivatives as well as to methods of their preparation. <CHEM> The compounds of formula I according to the present invention being suitable pharmaceutical agents are those wherein   Ar<1> and Ar<2> are independently from each other substituted or unsubstituted aryl or heteroaryl groups,   X is O or S, preferably O; R<1> is hydrogen or a C1-C6-alkyl group, preferably H, or R<1> forms a substituted or unsubstituted 5-6-membered saturated or non-saturated ring with Ar<1>; n is an integer from 0 to 5, preferably between 1-3 and most preferred 1.   Y within formula I is an unsubstituted or a substituted 4-12-membered saturated cyclic or bicyclic alkyl containing at least one nitrogen atom, whereby one nitrogen atom within said ring is forming a bond with the sulfonyl group of formula I thus providing the sulfonamide.
Patent SU-843787-A3 (SU)
Inventor: PRAJSER UILBER DEVID
IPC: G11C5/02
Filed: 1977-03-30
Granted: 1981-06-30
Abstract: A semiconductor memory produced in a unipolar technology includes a cell which has an inversion capacitor with one terminal connected to a bit/sense line, the other terminal is coupled to a source of charges by a pulse from a word line. To provide a word organized array of these cells, each word includes a source of charges produced at the surface of a semiconductor substrate and plurality of inversion capacitors are formed also at the surface of the semiconductor in spaced apart relationship from the charge source. Information is written into the capacitors by applying voltages of two different magnitudes, representing 1 and 0 bits of information, to one terminal of the capacitors while a word pulse produces inversion layers at the surface of the substrate between the capacitors to interconnect serially the charge source with each of the capacitors. The capacitors having the larger voltage store the greater amount of charge. This charge can then be detected by measuring the voltage across the storage capacitors when a work pulse again connects the charge source with each of the capacitors.
Patent SU-1093240-A3 (SU)
Inventor: KOLINDZHER KENNET DZH
IPC: B60R21/13
Filed: 1978-01-06
Granted: 1984-05-15
Abstract: 1497765 Tractor cab mountings INTERNATIONAL HARVESTER CO 24 May 1976 [24 Oct 1975] 21413/76 Heading B7B A cab 24 and rollover protective structure (ROPS) 38 are secured to a platform assembly 36 which is resiliently and releasably hinged at opposite sides by respective pairs of isolators 154, 156 to two cross beams 108 of a platform support 14 on the tractor chassis 12 so that components beneath the platform assembly 36 are accessible. The cab, platform assembly and platform support are offset from the longitudinal axis of the tractor and extend beyond the chassis 12 at one side. The axes of hinge pins 180 of the isolators 154, 156 are parallel to the longitudinal axis. Each hinge pin 180 is secured in an apertured knuckle portion 130 of the respective cross beam 108 and the ends are resiliently mounted in polyurethane bushings 182 carried by a knuckle device 134, itself secured by bolts 166 to a seat platform 168. Bolts 166 also secure a foot 162 of an upright member 90 of the ROPS 38 to the platform 168 and the ROPS is connected to the roof of the cab 24. When the tractor overturns, for example by turning anticlockwise in Fig. 4, the energy of initial ground impact is absorbed by clockwise movement of the ROPS member 90 to 90a until surfaces 132 and 136 facing each other across the gap 6 in the isolator interengage and thereby lock the joint.
Patent SU-810088-A3 (SU)
Inventor: KYUSTERS EDUARD
IPC: D06B11/00
Filed: 1978-09-28
Granted: 1981-02-28
Abstract: In a device for applying designs to advancing webs, particularly textile and similar webs, in which the design liquid is present, prior to application to the web, in the form of a film extending over the web in the width direction an air nozzle in the form of a tube extending across the web close to the film, the tube supported for rotation and for movement back and forth across the web, the tube having a plurality air outlet openings distributed over its surface, and supplied compressed air feed line is used to irregularize the film.
Patent SU-795523-A3 (SU)
Inventor: ZOMMER RYUDIGER
IPC: H04N1/40
Filed: 1978-11-16
Granted: 1981-01-07
Abstract: A method and apparatus for recording graphic or image information by means of punctiform recording spots which are arranged line-by-line according to a recording grid, or multi-lined within a matrix, whereby at the beginning of a contour proceeding obliquely to the recording direction, the first recording spot is displaced in the direction of the contour when its edge does not coincide with the contour and, in order to improve the end edge of such a contour proceeding obliquely to the recording direction, the recording of the last recording spot may be additionally displaced relative to the preceding recording spot by a retarding in time of the recording of said last spot.
Patent SU-818499-A3 (SU)
Inventor: MYULLER EKART
IPC: F02M61/10
Filed: 1979-04-06
Granted: 1981-03-30
Abstract: A fuel injector, for internal combustion engines, having a nozzle needle supported in a nozzle body so as to be axially displaceable therein. The nozzle needle, which can be lifted off its valve seat by the pressure of fuel, has a throttling pin which, at least during part of its lift, projects below the valve seat into a bore centrally arranged in the nozzle body. The throttling pin has at least one control edge or flat portion which is shaped and oriented in such a way that the fuel spray direction and/or the fuel spray characteristic or pattern vary with the nozzle needle lift.
Patent SU-902657-A3 (SU)
Inventor: KAJUKE ZHAN-FRANSUA
IPC: B24B13/02
Filed: 1979-04-16
Granted: 1982-01-30
Abstract: Apparatus for machining, polishing and/or smoothing workpieces having curved surfaces such as optical or ophthalmic lenses. A bearing head maintains a tool against a workpiece. Pressure is applied by a pneumatic piston and cylinder unit for establishing contact pressure between the workpiece and the tool. An eccentric drive mechanism including a compound table generates relative displacement between the workpiece and the tool. The pneumatic piston and cylinder unit actually forms part of the tool holder spindle. The cylinder or piston rod of the unit is provided with a tool holder block mounting the tool and the other of the piston rod or cylinder is attached to the drive mechanism. The bearing head has a freely rotating position and a locked position preventing rotation.
Patent SU-1215609-A3 (SU)
Inventor: OKHTA RIOUO
IPC: B29C57/04
Filed: 1979-10-02
Granted: 1986-02-28
Abstract: PURPOSE:To form a fancet excellent in the inside shape and dimensional accuracy, by slidably fitting the segments of a split cylindrical metal mold whose diameter is reduced by displacing moving members back, on the tapered surfaces of the finger parts of the moving members. CONSTITUTION:A hydraulic cylinder 11 is driven to displace a flange 9 on the rear end of the second moving member 5b back to an end plate 61 on a sleeve 6. The second metal mold segment 12b falls toward the axis of a support bar 1 due to the backward displacement of the second moving member 5b. When the fall has ended, the projection m of the second metal mold segment 12b is located inside the diameter of a fancet W shown by a dotted line. A piston rod 8 is thereafter retracted by a hydraulic cylinder so that the finger part 52b of the second moving member 5b and the finger part 52a of the first moving member 5a are simultaneously displaced back.
Patent SU-1272987-A3 (SU)
Title: Непрерывный способ получени эпихлоргидрина
Inventor: BUKALA YUZEF
IPC: C07D303/02
Filed: 1984-03-07
Granted: 1986-11-23
Abstract: Изобретение касаетс  эпоксидных  соединений, в частйости производства  эпихлоргидрина, примен емого дл  получени  эпоксидньЕХ смол и глицерина.  Дл  снижени  расхода пара в процессе  дегидрохлорировани  (ДГХ) дихлорпропанолов  (ДХП) и уменьшени  образовани  побочных продуктов ДГХ провод т  в других услови х. Процесс ведут в  следующей последовательности: а) ДГХ  ведут в предреакторе в водной суспензии  Са(ОН)2 вз той в 4-20%-ном мол рном  избытке при Т  313-343 К в  течение 20-1000 с до степени ДГХ   20-70 мол.%; б) реакционную смесь  подают в верхнюю часть реакционноотгонной  колонны под давлением 0,030 ,08 МПа, а в нижнюю - вод ной пар,  причем сверху направл ют струю полученного  после реакции раствора,  смешанного с водным слоем дистилл та,  § поступающего с верхней части колонны  и содержащего ЭПХ и HjO; в) отход СО  щий дистилл т раздел ют на водный  слой, возвращаемьй в колонну, и органический , содержащий 92-98% ЭХГ.  Окончание ДХГ проходит в верхней части  реакционно-отгонной колонны. В услови х  неполного превращени  ДХП  снижаетс  до 2-8 мае.% образование  побочных продуктов против 13,4 мае.2  в известном случае; расход пара 5 7  кг, против 9 кг на кг ЭХГ. 3 ил.
Patent SU-1637662-A3 (SU)
Inventor: PERRONE DIEGO
IPC: B01J2/24
Filed: 1985-10-15
Granted: 1991-03-23
Abstract: A new anhydrous sodium dichromate in flakes, Na2Cr2O7, m.p. 356 DEG C. (dec. 400 DEG  C.) is described, characterized in that it comes in flakes with an area of approx. 1 cm2, thickness 0.5 mm and apparent specific gravity 1.10 (absolute 2.748) at 25 DEG  C.; it is not deliquescent, nor does it become powdery. It is prepared from dihydrate sodium dichromate or aqueous solutions thereof using a new process in two stages, namely (a) evaporation-melting of the dihydrate salt or concentrated aqueous solution at a strictly controlled temperature of around 380 DEG  C. and no higher, and (b) flaking of the melted mass obtained thereby, as it is being rapidly cooled to 150 DEG -160 DEG  C. The apparatus for carrying out the process is also claimed; said apparatus consisting essentially of a dehydrator-melter oven, a flaker rotating at 10-20 revs per minute and a heat recovery system. The thermic contribution, respectively positive and negative in the two stages, is provided by means of a particular eutectic mixture of melted salts, which melts at 139 DEG C. Said mixture is composed of KNO3 52.2%, NaNO3  7.0%, NaNO2 39.4%, K2Cr2O7 1.4%.
Patent WO-0045163-A3 (WO)
Title: Boitier de microcapteur
Inventor: BONNE ULRICH
IPC: G01N25/18
Filed: 2000-01-27
Abstract: L'invention concerne une structure de boîtier de microcapteur comprenant au moins une entrée au niveau de l'une de ses extrémités et un capteur de propriétés thermiques au niveau de l'autre extrémité. Un écran de convection est placé entre l'entrée et le capteur. Un échantillon de fluide est prélevé au niveau de l'entrée dans un canal véhiculant le fluide à échantillonner. Les lignes d'écoulement par convection du fluide sont barrées par l'écran de convection. Le fluide diffuse dans une cavité située entre l'écran et le capteur. Le capteur détecte une propriété thermique du fluide diffusé. Un écran préféré est pourvu d'orifices sur son périmètre, une partie centrale solide de l'écran couvrant le capteur à une certaine distance. Le canal véhiculant le fluide peut être équipé de déflecteurs destinés à atténuer le bruit de turbulence et à faciliter le transport du fluide vers le boîtier du capteur ou hors de celui-ci.
Patent WO-0054152-A3 (WO)
Title: System and method for determining cluster membership in a heterogeneous distributed system
Inventor: MODIRI RAMIN
IPC: G06F11/00
Filed: 2000-03-06
Abstract: A distributed computer system and method for determining cluster membership in a distributed computer system. A plurality of computers configurable as cluster nodes are coupled through one or more public and/or private communications networks. Cluster management software running on the plurality of computers is configured to group various ones of the computers into a cluster. Weighting values are assigned to each node, such as by relative processing power. Each fully connected subset of nodes are grouped into a possible cluster configuration. The weighting value of each subset is calculated. The membership in the cluster is chosen based on the subset with the optimum weighting value among all the possible cluster configurations. The maximum weighting value may be adjusted if the maximum weighting value is greater than or equal to the sum of all other weighting values for all other nodes in the current cluster configuration. The maximum weighting factor may be adjusted to a value below the sum of all other weighting values for all other nodes in the current cluster configuration.
Patent WO-0073155-A3 (WO)
Inventor: GIAMPAVOLO PAUL
IPC: B65D19/38
Filed: 2000-05-17
Abstract: A pallet guard (40) includes a plurality of modular pallet guard sections (38). Each pallet guard section (38) comprises a connecting piece (44) and a wall (42). The connecting pieces are adjustable. The walls (42) are matable with another pallet guard section (38) so that the pallet guard is adjustable to accommodate varying size pallets and/or spill-over merchandise on the pallet. Each connecting piece (44) may be moveable between a first position, wherein the connecting piece is straight, and a second angled position where the pallet connecting piece forms a corner.
Patent WO-0129774-A3 (WO)
Title: Systeme destine a distribuer et a recharger rapidement des cartes de transport
Inventor: NEWSOME MATTHEW J
IPC: G07F17/42
Filed: 2000-10-20
Abstract: L'invention concerne un terminal de recharge se présentant sous la forme d'un dispositif compact d'utilisation et d'installation faciles destiné à un environnement d'encaissement automatique. Ce dispositif permet de recharger et de distribuer des cartes de transport exclusivement au moyen de fonctions de crédit et de débit. Ce terminal de recharge permet de réduire les longues files d'attente généralement associées aux distributeurs automatiques nécessitant des billets ou de la monnaie. Ledit terminal de recharge permet également la vente de billets en dehors des gares ou des stations, notamment dans des centres commerciaux, des épiceries, des bureaux de poste et des aéroports.
Patent WO-0178087-A3 (WO)
Title: Magnetically-responsive microspheres
Inventor: CHANDLER DONALD J
IPC: H01F1/11
Filed: 2001-04-06
Abstract: Microspheres are constructed using magnetic particles. Hybrid microspheres are constructed using fluorescent or luminescent microspheres and magnetic nanoparticles. Reactive moieties on the surface of the resultant particles can be used for attachment of biologically active molecules, thus allowing selective separations and analytical assays to be performed. Distinguishable subsets of microspheres can be constructed based on fluorescent intensities, and separations can be affected based on variable degree of magnetic content.
Patent WO-0178683-A3 (WO)
Title: Formulations a liberation lente
Inventor: OKUMU FRANKLIN
IPC: A61K9/00
Filed: 2001-04-19
Abstract: L'invention concerne une préparation à libération lente d'une hormone de croissance, notamment de l'hormone de croissance humaine.
Patent WO-0192918-A3 (WO)
Title: Systeme de deploiement de capteurs sismiques marins
Inventor: AMBS LORAN
IPC: G01V1/38
Filed: 2001-05-24
Abstract: La présente invention concerne un système permettant de recueillir des données en provenance de formations géologiques sous l'eau.  Une pluralité de boîtiers hydrodynamiques peuvent être déployés dans l'eau et descendre à grande vitesse à travers l'eau jusqu'à ce que les boîtiers entrent en contact avec les formations géologiques.  Un contrôleur couplé à chaque boîtier reconfigure le boîtier afin d'améliorer le contact entre celui-ci et les formations géologiques, et de réduire l'impact des courants océaniques s'exerçant contre le boîtier.  Un capteur sismique marin est couplé à chaque boîtier afin de détecter des données sismiques et de capter son orientation.  Chaque boîtier peut être déconnecté du capteur sismique marin associé afin de faciliter le retrait des capteurs sismiques et leur remontée jusqu'à la surface de l'eau.
Patent WO-0203645-A3 (WO)
Title: Procede et appareil de synchronisation de la presentation de donnees audio et d'applications visuelles
Inventor: MARKS BENNETT
IPC: A63F13/12
Filed: 2001-06-27
Abstract: L'invention porte sur un serveur (100) pouvant recevoir des communications comportant à la fois des données audio et des données d'application, ces dernières pouvant illustrer des progrès dans des conversations ou des jeux. A cet effet, le serveur filtre lesdites données en fonction d'une application (109) et transmet chaque communication à des clients participant  ayant rejoint la conversation ou le jeu, sans excepter celui qui est à l'origine de la communication.
Patent WO-0228962-A3 (WO)
Inventor: BEKELE SOLOMON
IPC: B32B27/30
Filed: 2001-09-19
Abstract: A composition includes greater than 50 % by weight such as between 51 % and 99 % by weight, of a first PVdC copolymer having a weight average molecular weight of between 80,000 and 125,000, and less than 50 % by weight, such as between 1 % and 49 %, by weight of a second PVdC copolymer having a weight average molecular weight of between 126,000 and 180,000, the weight percent of each of the first and second polymers based on the combined weight of the first and second polymers. A film includes at least one layer having the above composition. A film can have at least one layer including a blend of a first vinylidene chloride polymer and a second vinylidene chloride polymer, the film having a free shrink ratio of between 0.6 and 2.2 at a shrink temperature of 180 °F., or a free shrink ratio of between 0.8 and 1.4 at a shrink temperature of 200 °F. Methods of making the film of the invention are also disclosed.
Patent WO-0236734-A3 (WO)
Title: Aza- et polyaza-naphtalenyl cetones utiles en tant qu'inhibiteurs de l'integrase du vih
Inventor: ZHUANG LINGHANG
IPC: A61P31/18
Filed: 2001-10-09
Abstract: L'invention concerne certains aza- et polyaza-naphtalényl cétones, dont certains quinolinyl et naphthyridinyl cétones utilisés en tant qu'inhibiteurs de l'intégrase du VIH et en tant qu'inhibiteurs de la réplication du VIH. Ces composés sont utiles dans la prévention ou le traitement de l'infection par le VIH et le traitement du SIDA ou le retardement de son apparition, en tant que composés ou sels pharmaceutiquement acceptables, ou en tant qu'ingrédients dans les compositions pharmaceutiques, éventuellement en combinaison avec d'autres anti-viraux, immunomodulateurs, antibiotiques ou vaccins. L'invention concerne également des méthodes de traitement du SIDA ou des méthodes permettant de retarder son apparition, ainsi que des méthodes de prévention ou de traitement d'une infection par le HIV.
Patent WO-0240122-A3 (WO)
Title: Distributeur de liquide a flacon rigide et a vessie interieure souple
Inventor: PY DANIEL
IPC: B67D7/58
Filed: 2001-10-23
Abstract: La présente invention concerne un distributeur destiné à distribuer un liquide, qui comprend un flacon rigide possédant une chambre à liquide principale contenant un liquide, et un ensemble pompe qui est en communication fluidique avec cette chambre à liquide principale et qui est agencé de façon à distribuer une quantité prédéterminée de liquide en provenance de la chambre à liquide principale. Une vessie souple située dans la chambre à liquide principale est agencée de façon à se dilater pour remplir le creux créé dans cette chambre à liquide principale pendant la distribution du liquide par l'ensemble pompe. La vessie souple à tendance à forcer vers l'extérieur en direction du flacon rigide et, à son tour, elle augmente la pression dans la chambre à liquide principale par rapport à l'intérieur de la vessie de façon à empêcher ainsi l'intrusion d'air ou de vapeurs dans cette vessie ou dans la chambre à liquide principale.
Patent WO-02052763-A3 (WO)
Title: Multiple format secure voice apparatus for communication handsets
Inventor: BLANCHARD SCOTT D
IPC: H04W88/02
Filed: 2001-12-10
Abstract: Multiple format secure voice apparatus for communication handsets includes a core unit (12) with a speaker (15), a microphone (16), a keypad (17), and a display (18). The core unit also includes an audio circuit (20) coupled to the speaker and the microphone, an encryption/decryption element (25) coupled to the audio circuit, a coder/decoder element (27) coupled to the audio circuit and the encryption/decryption element, and a control element (30) coupled to the keypad, the display, the audio circuit, the encryption/decryption element, and the coder/decoder element. A standard interface coupling (35) is connected to an audio I/O terminal (21), a data I/O terminal (28) of the coder/decoder element, and a control I/O terminal (32) of the control element. A mating standard interface coupling (40) mates with the standard interface coupling of the core unit and is coupled to the mating standard interface coupling.
Patent WO-02057741-A3 (WO)
Title: Anticorps monoclonaux et antigenes de surface pour la detection et le traitement du cancer a petites cellules (sclc)
Inventor: GELBER COHAVA
IPC: C12N5/10
Filed: 2001-11-01
Abstract: L'invention concerne des nouveaux anticorps monoclonaux et des fragments de liaison de ceux-ci, qui reconnaissent les antigènes de surface que l'on trouve dans les cellules du cancer à petites cellules (SCLC), et qui sont immunoréactifs avec ceux-ci. Les anticorps de l'invention sont spécifiques de certaines tumeurs et sont utiles pour la thérapie, le diagnostic, le contrôle, la détection et l'imagerie de maladies du type SCLC et de patients souffrant de SCLC. Les antigènes de surface spécifiques de SCLC reconnus par les anticorps peuvent servir de cibles pour la détection, le diagnostic, l'inhibition ou l'élimination des cellules de SCLC.
Patent WO-02059313-A3 (WO)
Title: Nouvelles proteines, et acides nucleiques codant pour elles
Inventor: LI LI
IPC: C12N15/12
Filed: 2001-12-18
Abstract: L'invention porte sur des séquences d'acides nucléiques codant pour de nouveaux polypeptides, sur les polypeptides codés par lesdites séquences, sur les anticorps se fixant immunospécifiquement auxdits polypeptides, ainsi que sur des dérivés, des variantes, des mutants, ou des fragments desdits polypeptides, polynucléotides et anticorps. L'invention porte également sur des procédés thérapeutiques, diagnostiques et de recherche, en vue du diagnostic, du traitement et de la prévention de troubles liés à ces nouveaux acides nucléiques humains et à ces nouvelles protéines humaines.
Patent WO-02058628-A3 (WO)
Title: Methodes immunotherapeutiques permettant la modulation extracorporelle du recepteur cd36 et de ses ligands
Inventor: SRIVASTAVA PRAMOD K
IPC: A61M1/36
Filed: 2001-12-21
Abstract: La présente invention concerne des méthodes permettant de moduler une réponse immunitaire chez un patient par modulation des niveaux de circulation des ligands du CD36. Plus particulièrement, l'invention concerne une méthode d'aphérèse extracorporelle, pouvant être utilisée pour moduler les niveaux des ligands du CD36 dans la circulation sanguine chez un patient nécessitant une immunothérapie.