baber/WOPTO huggingface dataset:
Patent AU-660359-B2 (AU)
Title: Hydroxylated metabolites and derivatives of doxazosin as anti-atherosclerosis agents
Inventor: WONG SAMUEL SIU-MING
IPC: A61K31/505
Filed: 1993-03-31
Granted: 1995-06-22
Abstract: This invention relates to the use of certain hydroxylated metabolites and derivatives of doxazosin and their pharmaceutically acceptable acid addition salts for retarding the development of atherosclerosis in a mammal. Such compounds are useful for reducing atherosclerotic plaque involvement and for retarding and reducing both lipid deposition fibrosis in the development of atherosclerotic plaques.
Patent AU-693608-B2 (AU)
Title: Harmonic ultrasound imaging with microbubbles
Inventor: SCHUTT ERNEST G
IPC: A61K49/22
Filed: 1995-09-26
Granted: 1998-07-02
Abstract: A method for ultrasonic harmonic imaging is disclosed, which uses microbubbles particularly selected for their properties of reradiating ultrasound energy at frequencies other than the exciting frequency.
Patent AU-573681-B2 (AU)
Title: Infinitely variable transmission
Inventor: CADEE THEODORUS PETRUS MARIA
IPC: F16H61/662
Filed: 1985-01-18
Granted: 1988-06-16
Abstract: An infinitely variable transmission for a device with an internal combustion engine, provided with an endless transmission member (14) which has been looped over two pulleys, (2,3;8,9) each having a groove situated between conical sheaves, (2,3;8,9) at least one of which in each pulley is axially displaceable through an associated hydraulic cylinder, (4, 12) and also provided with a first control valve (40) for regulation of the fluid pressure in the cylinder of the driven pulley (8,9) and in the supply line to a second control valve (20), the latter valve being intended for adjustment of the transmission ratio by regulation of the amount of fluid supplied to and discharged from the cylinder (4) of the driving pulley, (2,3) wherein means (71) have been provided for the operation of the first control valve (40) which depend on the pressure of the gas drawn in by the internal- combustion engine inasmuch as upon an increase of this pressure (a lower vacuum), the fluid pressure in the cylinder (12) of the driven pulley (8,9) rises.
Patent AU-700404-B2 (AU)
Title: Monomers and composition which can be crosslinked and croslinked polymers
Inventor: MUHLEBACH ANDREAS
IPC: C07C13/28
Filed: 1995-11-06
Granted: 1999-01-07
Abstract: PCT No. PCT/EP95/04359 Sec. 371 Date May 14, 1997 Sec. 102(e) Date May 14, 1997 PCT Filed Nov. 6, 1995 PCT Pub. No. WO96/16008 PCT Pub. Date May 30, 1996Compounds of the formula I(A)n-B(I)in which A is the radical of a strained cycloolefin, B is a direct bond or an n-valent bridging group and n is an integer from 2 to 8, with the exception of 1,2-bisnorbornenyl-ethane and norbornenecarboxylic acid norbornenemethyl ester. The compounds of the formula I can be polymerized with one-component catalysts (ring-opening metathesis polymerization).
Patent AU-602117-B2 (AU)
Title: Graft polymers which are water-soluble or dispersible in water, their preparation and use
Inventor: BERENDT HANS-ULRICH
IPC: C08F283/06
Filed: 1989-09-29
Granted: 1990-09-27
Abstract: Graft polymers which are obtainable from (A) 2%-30% by weight of an addition product from alkylene oxide onto an aliphatic alcohol which is at least trihydric having 3 to 10 carbon atoms and (B) 70%-98% by weight of a grafted-on monomer mixture of (1) 20% to 50% by weight of an N-substituted or N-unsubstituted acrylamide or methacrylamide and (2) 50% to 80% by weight of an N-vinyl-substituted amide or of a vinyl ester, derived in each case from a saturated aliphatic monocarboxylic acid, where the sums of (A) and (B), and (1) and (2) in each case add up to 100%. These novel graft polymer are suitable as dyeing assistants, particularly as padding assistants or liquor binders when dyeing cellulose fibre materials.
Patent AU-628414-B2 (AU)
Title: Bone cement
Inventor: KINDT-LARSEN TURE
IPC: A61L24/06
Filed: 1989-09-26
Granted: 1992-09-17
Abstract: An acrylate based bone cement with well balanced low exotherm, low residual monomer, and high strength properties formulated from (1) a liquid component containing at least three different monomeric (meth)acrylates, e.g. a C1-C2 alkyl methacrylate, a straight or branched long chain (meth)acrylate having a molecular weight of at least 168, and a cyclic (meth)acrylate having a molecular weight of at least 168, and (2) a polymer powder component containing (meth)acrylate polymers or copolymers. The final bone cement may also contain conventional additives such as polymerization inhibitors, activators, crosslinkers, X-ray contrast material, polymerization initiators, antibiotics, antiseptics, and the like.
Patent AU-716973-B2 (AU)
Title: New substituted 7,12-dioxabenz(a)anthracene compounds, process for preparing them and pharmaceutical compositions containing them
Inventor: COUDERT GERARD
IPC: C07D319/24
Filed: 1997-11-07
Granted: 2000-03-09
Abstract: 7,12-Dioxabenz(a)anthracene derivatives of formula (I) and their isomers and addition salts are new: R1 = H or OR; R = H or 1-6C alkyl (optionally substituted by aryl or heteroaryl); R2 = H, halo, OH, 1-6C alkoxy, CHO, CF3SO3, CN, 2-7C alkyloxycarbonyl, aryloxycarbonyl, NRa'Rb' or BNRa''Rb''; Ra', Ra'' = di(1-6C alkyl)amino(1-6C alkyl); or Ra'' = 1-6C alkyl optionally substituted by OH; Rb', Rb'' = H or 1-6C alkyl; B = CO or CH2; X = N (optionally substituted by Rc') or X'; X' = CR3; Rc' = 1-6C alkyl; R3 = H, 2-7C alkoxycarbonyl or BNRa''Rb'' or CX'R2 = a group of formula (a): Y = N or CR4; R4 = H or OR''; R'' = H, 1-6C alkyl (optionally substituted by OH), aryl or heteroaryl; aryl = Ph or naphthyl (optionally substituted by halo, 1-6C alkyl, OH, 1-6C alkoxy or trihalomethyl); heteroaryl = mono- or bicyclic aromatic group containing 1-2 heteroatoms comprising O, S and/or N (optionally substituted by halo, 1-6C alkyl, OH, 1-6C alkoxy or trihalomethyl); provided that when X = N and Y = CH, or when X = CH and Y = N, or when X=Y = CH, then R1 and R2 are not both H. N2-(7,12-dioxa-3-hydroxybenzo(a)anthracene-5,6-maleimido)-N1,N1-dimeth ylethylenediamine hydrochloride is specifically claimed.
Patent AU-624443-B2 (AU)
Title: Siloxane-based refrigerating oil
Inventor: ENDRES ROBERT
IPC: C09K5/04
Filed: 1989-11-17
Granted: 1992-06-11
Abstract: The present invention relates to cooling oils which are free of salt, alcohol, halohydrocarbons and halocarbons and have a low viscosity at low temperatures and which consist of mixtures of hexamethyldisiloxane and/or octamethyltrisiloxane and/or linear decamethyltetrasiloxane and/or octamethylcyclotetrasiloxane and/or decamethylcyclopentasiloxane.
Patent AU-582377-B2 (AU)
Title: Imidazo``1,5-a``pyrimidine derivatives and process for their preparation
Inventor: IRIKURA TSUTOMU
IPC: C07D401/12
Filed: 1985-07-30
Granted: 1989-03-23
Abstract: This invention relates to novel imidazo (1, 5-a) pyrimidines, with antifungal activities having the formulawherein R, is halogen, R<sub>2</sub> is hydrogen or halogen, X is a sulfur, a sulfinyl group, a sulfonyl group or an oxygen atom, m and n are each independently 0 or 1, A is a phenyl group which may be substituted, a cycloalkyl group or an aromatic heterocyclic group which may be substituted.
Patent AU-695920-B2 (AU)
Title: Thrombin inhibitors based on the amino acid sequence of hirudin
Inventor: DIMAIO JOHN
IPC: C07K14/815
Filed: 1996-03-18
Granted: 1998-08-27
Abstract: A thrombin inhibitor comprising a first bulky hydrophobic portion interacting with the catalytic site of thrombin responsible for proteolysis and a second portion at least maintaining the hydrophobic and acidic character of amino acids 55 to 60 of native hirudin at the C-terminal non-catalytic region of N-acetyl-hirudin45-65. Between the first and second portions is a divalent linker moiety having a chain length of at least 10 carbon atoms. Connecting the first bulky hydrophobic portion and the linker is a peptidomimetic bond. Preferably, the bulky hydrophobic portion comprises at least one amino acid of D-configuration. The compounds are useful in the treatment of thrombotic disorders.
Patent AU-534090-B2 (AU)
Title: Prostacyclins
Inventor: SKUBALLA WERNER
IPC: A61K31/557
Filed: 1979-10-19
Granted: 1984-01-05
Abstract: Compounds of the formula   <IMAGE>   wherein R1 is (a) hydrogen, (b) C1-10 alkyl, (c) C1-10 alkyl substituted by halogen; C1-4 alkoxy; C6-10 aryl; C6-10 aryl substituted by 1-3 halogen atoms, a phenyl group, 1-3 C1-4 alkyl groups or a chloromethyl, fluoromethyl, trifluoromethyl, carboxy, hydroxy or C1-4 alkoxy group; di-C1-4-alkylamino; or tri-C1-4-alkylammonium, (d) C4-10 cycloalkyl, (e) C4-10 cycloalkyl substituted by C1-4 alkyl, (f) C6-10 aryl, (g) C6-10 aryl substituted by 1-3 halogen atoms, a phenyl group 1-3 C1-4 alkyl groups or a chloromethyl, fluoromethyl, trifluoromethyl, carboxy, hydroxy or C1-4 alkoxy group, or (h) an aromatic heterocycle of 5 or 6 ring atoms one of which is O, N or S; A is -CH2-CH2-, trans-CH=CH- or -C 3BOND C-; W is hydroxymethylene, RO-methylene, CH3 or CH3,   <IMAGE>   wherein OH or OR is in the  alpha - or  beta -position and R is an in vivo hydrolyzable and physiologically acceptable ether or acyl group which is conventional for modifying OH groups in prostaglandins; D and E together are a direct bond, or D is C1-10 alkylene, C1-10 alkenylene or C1-10 alkynylene or one of these groups substituted by fluorine, and E is oxygen, -C 3BOND C- or a direct bond; R2 is (a) a C1-10 hydrocarbon aliphatic radical, (b) a C6-10 hydrocarbon aliphatic radical substituted by C6-10 aryl or by C6-10 aryl substituted by 1-3 halogen atoms, a phenyl group, 1-3 C1-4 alkyl groups or a chloromethyl, fluoromethyl, trifluoromethyl, carboxy, hydroxy or C1-4 alkoxy group; (c) C4-10 cycloalkyl, (d) C4-10 cycloalkyl substituted by C1-4 alkyl, (e) C6-10 aryl, (f) C6-10 aryl substituted by 1-3 halogen atoms, a phenyl group, 1-3 C1-4 alkyl groups or a chloromethyl, fluoromethyl, trifluoromethyl, carboxy, hydroxy or C1-4 alkoxy group; or (h) an aromatic heterocycle of 5 or 6 ring atoms one of which is O, N or S; and R3 is OH or OR; and, when R1 is hydrogen, the salts thereof with physiologically compatible bases, are effective as antihypertensive, bronchiodilators, thrombocyte aggregation inhibitors, inter alia.
Patent AU-571767-B2 (AU)
Title: Fabric conditioning composition
Inventor: DUFFIN BRYAN
IPC: D06M15/248
Filed: 1986-01-09
Granted: 1988-04-21
Abstract: A fabric conditioning composition contains a fabric softening agent, which may be a cationic or nonionic material, and a polymeric drape-imparting agent, such as a vlnyl acetate-vinyl chloride copolymer, in the form of positively charged thermoplastic particles having a softening point of 25-200°C, especially above 50°C. When treated fabrics are ironed above this softening temperature, the particles coalesce to form a drape imparting film on the fabric. Non-ironed fabrics exhibit a softening benefit.
Patent AU-633082-B2 (AU)
Title: Pyranyl cyanoguanidine derivatives
IPC: A61K/
Filed: 1990-04-30
Granted: 1993-01-21
Abstract: Novel compounds having the formula <CHEM>  wherein <CHEM> are disclosed. These compounds have potassium channel activating activity and are useful, for example, as cardiovascular agents, especially as antiischemic agents.
Patent AU-757606-B2 (AU)
Title: Decorated pearl with integrated ornamental element
Inventor: WEINMANN GABRIELE
IPC: A44C17/00
Filed: 1999-09-03
Granted: 2003-02-27
Abstract: The invention relates to natural or artificial pearl in which one or more ornamental elements (4) are inserted in form of an inlay with or without a mount, wherein the outer visible top or ornamental side opposite the pearl of each inlay has a horizontal projection with a random contour and dimensions confined by the limits of the spherical surface and wherein the inner bottom side facing the pearl of each inlay is fitted with locking or anchoring means (20). Each inlay is lodged with positive-fit or at least substantially with positive-fit in an appropriately matching groove (6) (slot, cavity), locking and/or anchoring means being formed in the bottom and/or wall of said groove which interact with the corresponding inlay, preferably by positive locking according to the key-lock principle, and in or on which the inlay inserted into the groove is fixed in or on the pearl.
Patent AU-535021-B2 (AU)
Title: Separation of gas mixtures
Inventor: ROHDE WILHELM
IPC: F25J3/04
Filed: 1980-05-22
Granted: 1984-03-01
Abstract: In the fractionation of a gaseous mixture, e.g., air, by rectification, wherein liquid in the sump of a rectifying column is heated and thereby partially vaporized; and simultaneously sump liquid is withdrawn from a lower zone of the sump liquid bath, and is recycled into the bath above the point of withdrawal, the improvement, prior to the recycle step, of passing the withdrawn sump liquid from the lower zone into a heat exchanger disposed in the sump, said heat exchanger having a substantially sealed bottom end at a level below the liquid level of the sump, and an open top end at a level higher than the liquid level of the sump; said withdrawn sump liquid being passed into the bottom end of said heat exchanger and partially vaporized therein, and removing resultant liquid-vapor mixture from the heat exchanger at the top end above the level of the liquid bath. This system provides pump-free circulation of the sump liquid and the use incorporates an on-line adsorber to remove deleterious impurities from the sump liquid, e.g., hydrocarbons from oxygen.
Patent AU-629012-B2 (AU)
Title: Novel 3-methoximinopropionic esters and fungicides containing them
Inventor: WENDEROTH BERND
IPC: C07C255/64
Filed: 1990-07-12
Granted: 1992-09-24
Abstract: 3-Methoximinopropionic esters of the formula   <IMAGE> (I)  where the radicals R (m=1 to 5) are each hydrogen, halogen, cyano, nitro, alkyl, cycloalkyl, alkenyl, alkoxy, haloalkyl, haloalkoxy, unsubstituted or substituted phenyl, unsubstituted or substituted phenoxy, unsubstituted or substituted benzyl or unsubstituted or substituted benzyloxy, or the group  <IMAGE>  is naphthyl, and X is methyleneoxy, oxymethylene, ethylene, ethenylene, thiomethylene or oxygen, and fungicides containing these compounds.
Patent AU-697656-B2 (AU)
Title: Bicyclolactam compounds, use thereof and intermediates for preparing thereof
Inventor: OGAWA KAZUO
IPC: A61K31/473
Filed: 1996-06-07
Granted: 1998-10-15
Abstract: Bicyclolactam compounds represented by general formula (1) are useful as the active ingredient of medicines having an excellent anxiolytic effect and a high safety with little side effects such as a hypnotic effect, a muscle relaxing effect, a sedative effect, etc. In said formula, R represents oxo or -OR<1> (wherein R<1> represents hydrogen or acyl); A represents one of the following groups (2) and (3); Q represents hydrogen or lower alkyl; l is 1 or 2, m is 0 or 1; and n is 0, 1 or 2, provided that m and n are not 0 at the same time; R<2> represents optionally substituted benzoyl.
Patent AU-686517-B2 (AU)
Title: Alarm-triggered locking device for the catch and/or hinge region of a door or window to be protected
Inventor: MATOUSCHEK ERICH
IPC: E05B15/02
Filed: 1996-08-28
Granted: 1998-02-05
Abstract: PCT No. PCT/EP94/03796 Sec. 371 Date Aug. 13, 1996 Sec. 102(e) Date Aug. 12, 1996 PCT Filed Nov. 16, 1994 PCT Pub. No. WO95/21980 PCT Pub. Date Aug. 17, 1995An alarm-triggering locking mechanism for the lock and/or hinge area of a door to be secured or a window to be secured is proposed, which is embodied as a locking plate (23) which can be attached to a door or window frame by means of holding screws (27) embodied as the first blocking device. A second blocking device, which is harder to overcome by the effect of force, is embodied as at least one striker element (25) rigidly connected with the locking plate (23) and which, following the limited movement of the locking plate (23) in the opening direction, comes to rest against a counter-striker element (26) anchored on the door or window frame. An alarm, in particular a silent alarm, is triggered via radio or the telephone net after the first blocking device has been overcome. The burglar is thereafter delayed by the second blocking device, which makes it possible for security forces to reach the location of the break-in and to arrest the burglar while the break-in is still in progress.
Patent AU-732739-B2 (AU)
Title: Floor mat system
Inventor: KESSLER RONALD N
IPC: A47G27/04
Filed: 1998-03-13
Granted: 2001-04-26
Abstract: A floor mat system and clip for use therewith can be installed to any floor and includes a floor mat formed from a series of first and second cris-crossed ribs which form rectangular-shaped openings therebetween, and clip having a rectangular-shape base and four outwardly extending raised projections. Certain of the second ribs have an enlarged bottom which forms a latching shoulder on each side thereof. The projections of the clip have a generally triangular-shaped end which snap-fits with the latching shoulder of the certain second ribs and which aligns with certain of the openings of the floor mat. A pair of holes are formed in the clip which align with other of the openings of the floor mat when attached thereto.
Patent AU-641437-B2 (AU)
Title: Non-toxic corrosion inhibitive compositions and methods therefor
Inventor: SHARABY AHMED
IPC: B05D7/14
Filed: 1990-10-22
Granted: 1993-09-23
Abstract: Corrosion and/or crack growth of metals exposed to a salt water environment is inhibited by applying to a metal surface cerous molybdate and/or at least one water soluble ammonium salt of a phosphorus acid. Sealant compositions for such purpose are produced by blending the inhibitor substance(s) with a curable liquid polymer which is preferably curable to an elastomer.
Patent AU-733163-B2 (AU)
Title: Apparatus and method for forming cereal food products
Inventor: CAPODIECI ROBERTO A
IPC: A23L5/30
Filed: 1998-04-29
Granted: 2001-05-10
Abstract: A apparatus and method for infusing flavors into cereal grains and agglomerating the grains into a unitary food product. Grains of cereal, powdered soluble flavors and a moisturizing liquid are supplied to a mixer. The flavors, liquid and cereal grains are thoroughly mixed and the grains surface moisturized and then discharged into a product-forming chamber which is ultrasonically energized for a sufficient period of time so that the flavors are infused within the interiors of the grains which are agglomerated into a unitary product.
Patent AU-634054-B2 (AU)
Title: Process for control of pitch deposition from pulps in papermarking systems
IPC: D21H17/45
Filed: 1991-04-23
Granted: 1993-02-11
Abstract: An improved process for controlling natural pitch deposition in pulp and papermaking aqueous systems involves the use of ampholytic polymers containing diallyl dimethyl ammonium quaternary salts and also containing (meth) acrylic acid salts and optionally containing (alkyl) acrylic acid esters or hydroxy esters. These ampholytic polymers give improved results in terms of control of natural pitch in the manufacture of pulp and paper.
Patent AU-764362-B2 (AU)
Title: Method of the diagnosis of renal disorder, hemolytic-uremic syndrome and intestinal hemorrhagic escherichia coli infection
Inventor: MIWA MASAO
IPC: G01N33/569
Filed: 2000-10-06
Granted: 2003-08-14
Abstract: Methods for diagnosing renal disorder, hemolytic uremic syndrome and enterohemorrhagic E. coli infectious disease at an early stage, and for diagnosing the severity of these diseases are provided. Detection of excretion of AQP2 and/or molecules derived therefrom into urine of a subject, or determination of the amount of excretion of the same is conducted to diagnose the morbidity or the severity of renal disorder, hemolytic uremic syndrome and enterohemorrhagic E. coli infectious disease of the subject. For the detection and determination of AQP2, an immunochemical process may be suitably employed in which an antibody that specifically recognizes AQP2. <IMAGE>
Patent AU-645812-B2 (AU)
Title: Inhibition of viral infection
Inventor: COLLINS MARY KATHARINE LEVINGE
IPC: A61K31/455
Filed: 1991-05-24
Granted: 1994-01-27
Abstract: The use of a poly(ADP-ribose) polymerase inhibitor, preferably 3-N-formylamino benzamide for the treatment of a subject against infection by a virus, in which the viral or proviral DNA integrates into the chromosome or chromosomes during its replication cycle.
Patent AU-648802-B2 (AU)
Title: Parathyroid hypertensive factor
Inventor: PANG PETER K T
IPC: G01N33/50
Filed: 1991-06-27
Granted: 1994-05-05
Abstract: Hypertensive mammals may be treated to lower mean blood pressure by administering a calcium channel blocking agent together with a calcium supplement. The hypotensive effect of this combination is synergistic and the dose response is more predictable than the administration of either of these agents singly. <IMAGE>
Patent AU-736757-B2 (AU)
Title: Device for a materials handling vehicle
Inventor: DUNLAP DANNY L
IPC: B66F17/00
Filed: 1998-07-14
Granted: 2001-08-02
Abstract: A materials handling vehicle is provided with a frame including an operator's compartment having an entrance, a drive mechanism supported on the frame, a material handling unit coupled to the frame, and a device including an actuator located across the threshold of the entrance of the operator's compartment. The device generates an alert signal when a portion of an operator's body engages the actuator.
Patent AU-657105-B2 (AU)
Title: Holder for objects inside a rotating drum
Inventor: ROUMAGNAC JEAN-PATRICK
IPC: A61L2/26
Filed: 1991-10-28
Granted: 1995-03-02
Abstract: PCT No. PCT/FR91/00848 Sec. 371 Date May 7, 1993 Sec. 102(e) Date May 7, 1993 PCT Filed Oct. 28, 1991 PCT Pub. No. WO92/08498 PCT Pub. Date May 29, 1992.A holder for objects inside a rotating drum, particularly that of a sterilizer. The holder includes a pressure plate which can be brought into position for holding the objects by a motor-driven mechanism. This mechanism has a rod with threaded portions interacting with sleeves. These sleeves control the movement of pairs of link arms which are rigidly fixed to the pressure plate and are in contact with the drum wall.
Patent AU-729461-B2 (AU)
Title: Process for releasing an active principle contained in a multiple emulsion
Inventor: BIBETTE JEROME
IPC: B01J13/00
Filed: 1998-08-05
Granted: 2001-02-01
Abstract: A method for the controlled release of an active principle contained in a multiple water-in-oil-in-water emulsion characterized in that the multiple emulsion comprises an invert emulsion Ei with an aqueous phase A1 containing at least a hydrophilic active principle. The emulsion Ei is dispersed in the form of direct emulsion droplets Ed, in a continuous aqueous phase A2, with the two emulsions Ed and Ei stabilized by at least a surfactant, present in their respective continuous phases. The multiple emulsion is brought in the presence of an effective amount of an agent for transforming it into a direct emulsion and induce the release of the active principle, contained in the aqueous phase A1 of emulsion Ei, in the aqueous phase A2.
Patent AU-651414-B2 (AU)
Title: Binding of recognizing substances to liposomes
Inventor: MARGALIT RIMONA
IPC: A61K9/127
Filed: 1991-10-30
Granted: 1994-07-21
Abstract: Methodologies have been developed and certain recognizing substances and crosslinking reagents have been identified to modify liposomes. Crosslinking reagents link residues on the liposomal surface to the residues offered by certain recognizing substances. The crosslinking reagents include glutaraldehyde (GAD) and a water soluble carbodiimide, preferably, 1-ethyl-3-(3-dimethylaminopropyl) carbodiimide (EDC). The recognizing substances include gelatin, collagen, and hyaluronic acid (HA). Following these methodologies, recognizing substances can be utilized as an adhesive or glue to attach the liposomes onto a target area. These "bioadhesive" liposomes offer potential advantages as a microscopic drug delivery system.