baber/WOPTO huggingface dataset:
Patent MA-23018-A1 (MA)
IPC: A61P31/04
Filed: 1993-11-02
Abstract: The subject of the invention is the compounds of formula (I): <IMAGE>  in which,   . either R represents a radical (CH2)nAr1, n representing an integer between 1 and 6, Ar1 representing: - either a substituted carbocyclic aryl radical, or an optionally substituted heterocyclic aryl radical, . or R represents a radical XAr2, in which X is an alkyl radical interrupted by O, S, SO, SO2, <IMAGE> -C-NH, Ar2 being an optionally substituted aryl or heteroaryl radical,  Z representing a hydrogen atom or the residue of an acid.   The compounds of formula (I) have valuable antibiotic properties.
Patent MA-28175-A1 (MA)
Title: Composes organiques
Inventor: BAESCHLIN DANIEL KASPAR
IPC: A61K31/165
Filed: 2006-05-24
Abstract: La présente invention concerne des composés amides d'acide -amino- -hydroxy- -aryl-alkanoïque représentés par la formule (I) et les sels de ceux-ci, présentant des propriétés d'inhibition de la rénine. Cette invention concerne également des compositions pharmaceutiques comprenant ces composés, ainsi que des méthodes consistant à les administrer pour traiter l'hypertension, l'athérosclérose, un syndrome coronarien instable, une insuffisance cardiaque congestive, une hypertrophie cardiaque, une librose cardiaque, un post-infarctus en cas de cardiomyopathie, un dysfonctionnement diastoiique, une maladie rénale chronique, une flbrose hépatique, des complications entraînées par des diabètes, telles qu'une néphropathie, une vasculopathie, et une neuropahtie, des maladies des vaisseaux coronariens, une resténose après une angioplastie, une augmentation de la pression intra-occulaire, un glaucome, une croissance vasculaire anormale, un hyperaldosteronisme, une déficience cognitive, la maladie d'Alzheimer, la démence, les états d'anxiété et les troubles cognilifs.
Patent MA-37418-A1 (MA)
Title: Covoiturage dynamique integré à un système de transport public
Inventor: YOUNES MOUMEN
IPC: G06Q50/00
Filed: 2014-10-10
Abstract: Un système de covoiturage dynamique intégré à un système d’accès au transport public. Le système a comme objectif le contournement des difficultés relevées pour lancer un covoiturage dynamique efficace. Il propose dynamiquement, grâce à l’utilisation d’un appareil mobile, l’ensemble des options de déplacement d’un endroit a à un endroit b. Il s’agit d’une application informatique embarquée sur un appareil mobile caractérise par une connectivité internet et des équipements de géolocalisation. Application embarquée interagit avec des serveurs déployés sur le réseau internet assurant la communication avec les services d’opérateur de télécommunication, les services de transport public, ainsi que la gestion du covoiturage.
Patent MA-37776-A1 (MA)
Title: Prédiction de la réponse à un traitement par un inhibiteur de jak/stat
Inventor: CAO ALEXANDER
IPC: C12Q1/68
Filed: 2013-07-24
Abstract: L'invention concerne, en partie, une méthode de sélection d'un sujet ayant un cancer pour le traitement par un inhibiteur de jak/stat et un procédé de détermination si une dose thérapeutiquement efficace d'un inhibiteur de jak/stat a été administrée.
Patent MA-39369-A1 (MA)
Title: Prise isolante
Inventor: ANIS KIRAMA
IPC: H02H5/12
Filed: 2016-10-04
Abstract: Dispositif sous forme une multiprise électrique isolante caractérisé en ce qu'il comporte un système permettant de faire la différence entre l'être humain et les équipements électriques et un système sécurisant chargement des smartphones. Ce dispositif permet aussi la communication à distance avec l'utilisateur à travers une application mobile qui permet d'indiquer la consommation instantanée par prise, la commande à distance des prises électriques connectés, cette application permet aussi de générer un bilan énergétique de l'installation vers la fin du mois.
Patent UY-23570-A1 (UY)
Inventor: LOHMANN HELMUT
IPC: C08G77/38
Filed: 1993-04-21
Abstract: PCT No. PCT/EP93/00983 Sec. 371 Date Feb. 8, 1995 Sec. 102(e) Date Feb. 8, 1995 PCT Filed Apr. 23, 1993 PCT Pub. No. WO93/22464 PCT Pub. Date Nov. 11, 1993A process is disclosed for waterproofing materials having a fibrous structure, such as leather, persian leather or leather replacement materials, by using waterproofing agents containing sulfosuccinic acid esters. Also disclosed are waterproofing agents used to carry out this process. The sulfosuccinic acid esters are prepared by reacting maleic anhydride with monohydric or polyhydric alcohols, then by sulfitizing them. Reactive siloxanes may also be used as polyhydric alcohols.
Patent UY-24006-A1 (UY)
Inventor: JOHN NESTOR
IPC: A61P43/00
Filed: 1995-07-27
Abstract: The L-monovaline ester derived from 2-(2-amino-1,6-dihydro-6-oxo-purin-9-yl)methoxy-1,3-propanediol and its pharmaceutically acceptable salts are disclosed which are of value as antiviral agents with improved absorption.
Patent UY-24989-A1 (UY)
Title: Carprofeno, un inhibidor de cox-2, útil en el tratamiento del dolor e inflamación en perros
Inventor: PAUL RICKETTS ANTHONY
IPC: A61K31/403
Filed: 1998-05-04
Abstract: Tratamiento o prevención de procesos y enfermedades inflamatorias en perros asociadas con la actividad de la ciclo-oxigenasa-2 (COX-2) inducible, mientras que al mismo tiempo se reducen o eliminan los efectos secundarios indeseables asociados con la inhibición simultánea de la actividad de la ciclo-oxigenasa-1 (COX-1) constitutiva, mediante la inhibición selectiva de la actividad de COX-2 con respecto a la actividad de la COX-1, donde la relación de selectividad de COX-2:COX-1 es de al menos 3:1 basándose en los niveles de inhibición ex vivo medidos en sangre entera; el inhibidor es un miembro seleccionado entre el grupo de AINEs (anti-inflamatorios no esteroideos). En particular, el inhibidor de COX-2 que se reinvidica es el carprofeno [(+)-(S) ácido 6-cloro-alfa-metil-9H-carbazol-2-acético].
Patent UY-27941-A1 (UY)
Title: Derivados de indol o derivados de bencimidazol para modular ikb quinasa
Inventor: RITZELER DR OLAF
IPC: A61K31/4439
Filed: 2003-08-15
Abstract: Derivados de indol o derivados de bencimidazol para modular IKB quinasa. Compuestos de la fórmula I son adecuados para preparar productos farmacéuticos para la profilaxia y terapia de enfermedades cuyo curso implica una actividad incrementada de IKB quinasa.
Patent UY-28231-A1 (UY)
Title: Metodos y composiciones farmacéuticas para la obtención confiable de niveles aceptables de testosterona en suero.
Inventor: HUBLER DORIS
IPC: A61K47/44
Filed: 2004-03-12
Abstract: Composiciones farmacéuticas, formuladas para administración por inyección, que comprenden un éster de tertosterona, en particular undecanoato de testosterona, en un vehículo que comprende aceite de ricino y un co-solvente. Al inyectar las composiciones de acuerdo con un esquema de administración particular, se obtienen niveles confiables de testosterona en suero, dentro del rango fisiológico normal, por un período prolongado. Esto permite el uso de las composiciones en terapias de reemplazo hormonal y en la anticoncepción masculina, sin el monitoreo concomitante de los niveles de testosterona en suero a cargo de un médico.
Patent UY-29343-A1 (UY)
Title: Pirazolopiridinas y sales de las mismas, una composición farmacéutica que comprende dichos compuestos, un método para prepararlos y su uso.
Inventor: THIERAUCH KARL-HEINZ
IPC: C07D231/54
Filed: 2006-01-23
Abstract: Pirazolopiridinas de acuerdo con la fórmula general (I): y sales de las mismas, composiciones farmacéuticas que comprenden dichas pirazolopiridinas y un método para preparar dichas pirzolopiridinas así como el uso de las mismas para fabricar una composición farmacéutica para el tratamiento de enfermedades de crecimiento vascular desregulado o de enfermedades acompanadas con crecimiento vascular desregulado, donde los compuestos interfiere efectivamente con la angiopoyetina y por lo tanto influyen en la senalización de Tie2.
Patent AT-500119-A1 (AT)
IPC: A61K31/216
Filed: 1999-04-09
Abstract: Tilidine Mesylate has high stability, an improved taste and a suitable pH range in aqueous solution in comparison to known Tilidine salts. It may be presented in liquid or solid formulations, particularly with a retard profile. The novel salt is prepared by reacting Tilidine Base with Mesylic Acid in a solvent such as Ethyl Acetate, MIBK or Acetone at a reaction temperature of from 0 to 40  DEG C.
Patent CS-923387-A1 (CS)
Title: Lubricant oil for stomatologic instruments and responsive apparatus
Inventor: KLUCHO PAVOL RNDR
IPC: C10M161/00
Filed: 1987-12-15
Abstract: A lubricating oil for stomatological instruments comprises (a) 70-99.8 wt% of highly refined medicinal vaseline oil with kinematic viscosity 32-65 square mm/sec. at 20 deg.C and solidification point not above -50 deg.C, (b) 0-28% of vegetable or animal oil, and/or (c) 0-10% of esters of monocarboxylic acids and mono-alcohols and/or polyols and/or aliphatic dicarboxylic acids, citric, isocitric, phthalic or terephthalic acid and (un)branched aliphatic mono-alcohols, with mol.wt. 80-800, (d) 0.1-1.5% of polymers with mol.wt. 3,000-120,000, (e) 0.0001-0.1% of a phenolic antioxidant, and (f) 0.0001-0.002% of polysiloxane oils with varying mol.wt., as anti-foam.
Patent ES-160376-A1 (ES)
Title: PERFECCIONAMIENTOS INTRODUCIDOS EN LOS PROCEDIMIENTOS DE FABRICACIoN DEL CAUCHO
Filed: 1943-02-17
Abstract: Procedimiento para la fabricación de caucho caracterizado por el hecho de que se somete la primera materia constituida por lo menos en parte por caucho sintético a la acción de por lo menos un líquido susceptible de incorporarse a dicha materia en proporciones adecuadas entre 5 y 50% y de mantenerse en la misma aún después de tratamientos ulteriores tales como la vulcanización.
Patent ES-182494-A1 (ES)
Title: Un sistema de bloqueo para receptores
IPC: H04J3/04
Filed: 1948-02-20
Abstract: Sistema de bloqueo para receptores de impulsos de señal, caracterizado por un sistema que bloquea el funcionamiento del receptor, por lo menos, durante la mayor parte de cada intervalo de tiempo que existe entre impulsos de señal sucesivos de un tren dado de tales impulsos, comprendiendo un paso mezclador para recibir el tren de impulsos de señal, medios que respondan a cada impulso de señal para producir un impulso de bloqueo de una duración igual, por lo menos, a la mayor parte del intervalo entre al impulso y el impulso inmediato siguiente de dicho tren, y medios para aplicar dicho impulso de bloqueo a dicho paso mezclador que bloquee su funcionamiento durante el tiempo de tal impulso de bloqueo.
Patent ES-187659-A1 (ES)
Title: PERFECCIONAMIENTOS EN SISTEMAS TRANSMISORES DE ENERGiA
IPC: F16D37/02
Filed: 1949-03-31
Abstract: Perfeccionamientos en sistemas transmisores de energía caracterizados por el hecho de constar tales sistemas medios de potencia absorbida o trabajo medios de potencia generada o disponible medios transmisores de potencia medios conectantes entre los citados medios de potencia absorbida y de potencia generada medios de control controlando a dichos medios transmisores de potencial a las conexiones hechas entre los referidos medios de potencia absorbida y generada respondiendo los citados medios el control a la acción combinada de ambos medios de potencia absorbida y generada antes citados.
Patent ES-196315-A1 (ES)
Title: UNA INSTALACIoN DE HOGAR
Filed: 1951-01-27
Abstract: Una instalación de hogar enfriada por agua con una cámara de combustión vertida dentro de la cual es introducido el combustible por la parte superior o desde la cual las cenizas y pavesas son descargadas cerca del fondo mientras que al menos parte del aire de combustión es alimentado por aberturas de la pared delantera y los gases de combustión son atraídos por aberturas de la pared trasera caracterizada porque cada una de las paredes provistas de aberturas es de construcción tubular que comprende una fila de tubos verticales espaciados a través de los cuales está destinada a pasar el agua de enfriamiento de un sistema de circulación de agua por ejemplo disponiendo los extremos para que se abran en una cámara colectora y/o en la camisa de agua de la instalación de hogar.
Patent ES-275012-A1 (ES)
Title: Process for the preparation of 10 -methyl steroids
IPC: C07J75/00
Filed: 1962-02-28
Abstract: The invention comprises 10b -methyl-13b -n-propyl-gona-4,9(11)-dien-3-one derivatives of the general formula <FORM:1003085/C2/1> in which R represents the oxygen atom of a keto group, or a hydrogen atom and either a hydroxy group or an ester group derived from either a mineral acid or an organic carboxylic acid, and a process in which a 17b -acyloxy-13b -alkyl - 4,5 - seco - gon - 9 - ene - 3,5 - dione is protected at the 3-position, the 3-protected compound is subjected to methylation in the presence of an enolizing agent to effect methylation at the 10b -position and migration of the 9(10)-double bond to the 9(11)-position, the 3-protected keto group is liberated and the thus-freed ketonic compound is cyclized by alkali metal hydroxide into the corresponding 13b -alkyl - 17b - hydroxy - 10b - methyl - gona - 4,9(11)-dien-3-one. Protection of the 3-keto group may be effected by ketalization, e.g. with methyl-ethyl-dioxolan. Methylation may be effected with methyl iodide in the presence of potassium t.-amylate. Cyclization may be effected with potassium hydroxide in methanol. The 17b -hydroxy group in the so-obtained product may be oxidized to obtain the corresponding 17-keto compound with chromic anhydride in acetic acid, or esterified by an esterifying agent derived from either a mineral acid or an organic carboxylic acid. Specifications 979,892, 979,898 and 1,003,086 are referred to.
Patent ES-296736-A1 (ES)
Title: Carbon black product
IPC: C09C1/58
Filed: 1964-02-22
Abstract: A pelletized carbon black, suitable for compounding in elastomers, consists of a fluffy (i.e. non-pelletized) carbon black and an oleaginous pellet-binding material of low volatility which is compatible with and soluble in an elastomer mix. The individual kinetic particle units of the carbon black are separately coated with a film of the oleaginous material which is present in a quantity of from 1 to 90% of the oil absorption value (defined in the Specification) of the carbon black. The pelletized carbon black preferably contains from 1 to 15% by weight of oleaginous material. The oleaginous material may be an aromatic rubber compounding oil, for example obtained by solvent extraction from crude petroleum hydrocarbon fractions, a cycloparaffinic rubber compounding oil obtained by solvent extraction from hydrocarbon fractions, a thermoplastic resin, for example rosin, rosin derivatives, phenolic, terpene, coumarone-indene, urea-formaldehyde and melamine resins and lower molecular polystyrenes, used as such, in solution in other oleaginous materials or in a volatile solvent, or a fatty acid, for example oleic, lauric or stearic acid mixtures of oleaginous materials may be used. The carbon black may be pelletized in a dry pelletizing process using, for example, a solution of wood rosin in a naphthenic rubber compounding oil alternatively, the oleaginous material may be added in the form of an emulsion or a water-soluble derivative, for example the ammonium salt of lauric acid, to a water-wetted paste of the carbon black, the mixture being pelletized in a wet pelletizing process and dried at elevated temperature.
Patent ES-302223-A1 (ES)
Title: Improvements in fuel injection pumps for reciprocating internal combustion engines
IPC: F02M59/44
Filed: 1964-07-17
Abstract: In a fuel injection pump of the type in which the piston has a helical control edge 3 co-operating with a low pressure part 4 and is rotatably adjustable to vary the delivery, the piston has a leakage collecting groove 7 connected by an internal passage 8 to a part 9 extended by a groove 10 in the surface of the piston and arranged to communicate during at least part of the piston stroke with a further low pressure part 5.
Patent ES-304602-A1 (ES)
Title: New esters of secondary amino-alcohols
IPC: C07D295/088
Filed: 1964-10-02
Abstract: Novel compounds of the Formula I wherein X represents a hydrogen or halogen atom or an alkyl or alkoxy radical, y represents a hydrogen atom or an alkyl radical, Z and Z1, the same or different, represent hydrogen atoms or C1- 4 alkyl radicals or together with the nitrogen atom form a heterocyclic radical which may contain other hetero-atoms, and n represents 1, 2, 3 or 4, and acid addition salts thereof, are prepared by reacting an alcohol of the Formula II with an acid chloride of the Formula III. <FORM:1060005/C2/1> <FORM:1060005/C2/2> <FORM:1060005/C2/3> Carboxylic acid chlorides of the Formula III may be prepared by chlorination of the corresponding carboxylic acids which latter may be prepared by hydrolysis of the corresponding 4-cyano-4-(X-phenyl)-tetrahydropyrans. 4 - Cyano - 4 - (X - phenyl) tetrahydropyrans may be prepared by reacting the corresponding phenylacetonitriles with bis - (2 - chloroethyl) ether in the presence of sodamide.
Patent ES-337002-A1 (ES)
Title: Process and apparatus for the determination of water in an organic liquid
IPC: G01N25/48
Filed: 1967-02-18
Abstract: In a process for the determination of water contained in liquid organic material, the water containing liquid organic material is fed through a cell 4 together with the organic material in anhydrous form to which has been added one or more halogen derivatives of metalloids and acid halides, and the change in temperature caused by reacting the two liquids is determined by thermistors 5 as a measure of the water content. Both liquid streams pass through coils 8 in the water tank 2, and then through tank 3 before entering the cell 4.
Patent ES-337164-A1 (ES)
Title: Luminaire
IPC: F21V29/15
Filed: 1967-02-22
Abstract: A luminaire having a sealed optical system consisting of a reflector and a transparent closure sealed thereto has an air filter arranged to remove solid or gaseous impurities, inserted into the system, heat from a lamp inside the system causing expulsion of air while it is in operation, cool air being drawn into the interior through the filter when the lamp is not operating. In the form shown for use as a street lamp, a reflector 2 is enclosed in a housing 1, the mouth of the reflector being closed by a globe or refractor with the interposition of a sealing gasket. A cup-shaped housing is mounted in an opening in the reflector and carries a holder 11 for the lamp 12, a sealing gasket being provided around the junction of the housing and reflector. A filter 15 consisting of a tube of resilient material in which is a mass of, for example, activated charcoal is mounted in the side of the housing. In a modification, the luminaire consists of a reflector closed at the bottom by a window and secured at the top to a housing having a series of openings behind which is an annular window. The housing is secured to a supporting member containing the control gear for the lamp. The filter is mounted in an aperture in the reflector.
Patent ES-341889-A1 (ES)
Title: Pumps and reversible pump turbines
IPC: F03B15/00
Filed: 1967-06-16
Abstract: A clutch 26, 28 between a starter turbine runner 18 and a pump-turbine runner 4, 6 (see Division F1), is engaged by supplying pressure water through pipe 32 into a sealed chamber 30, and is disengaged by supplying pressure water to an annular space 52, or by supplying pressure fluid through pipes 40 to jacks 38 the space 52 then being permanently connected to a low pressure. When the clutch is disengaged by pressurizing the space 52, the space is thereafter connected to a low pressure via a valved passage 54 and the clutch is maintained in its disengaged position by the jacks 38. Movement of the jacks 38 is co-ordinated by switches 48. The clutch may alternatively comprise one or a number of pairs of engageable flat annular surfaces, or a dog coupling. The clutch may be engaged automatically when the runner 4, 6 overspeeds.
Patent ES-346681-A1 (ES)
Title: A Pressure Modifying Device for a Hydraulic Braking System
IPC: B60T8/18
Filed: 1967-11-02
Abstract: A hydraulic brake pressure modifying device comprises a tipping valve 36 interposed between a port 32, connectible to a master cylinder and a further port 24 feeding slave cylinders, the tipping valve 36 being engaged by an annular shoulder on a piston 26 so that the valve 36 is open when no brake application is required. When the hydraulic pressure at the outlet 24, acting on the piston 26 is sufficient to overcome the force F, valve 36 closes, so as to limit the pressure or rate of increase of pressure at the outlet. As shown, a differential piston 26 is employed, so that valve 36 is in lapping condition during braking so as to meter a given flow towards the outlet to pressure balance the piston 26. A stop 62 may be adjusted so as to vary the outlet pressure at which valve 36 becomes effective. In Fig. 2 (not shown) valve 36 is spring- biased in a downward direction, port 24 being used as inlet and the outlet port replacing stop 62. In Fig. 1 (not shown) the passage 50 is omitted. The force F may be responsive to load on one axle.
Patent ES-347580-A1 (ES)
Title: Fungicidal and fungistatic n-(dialkylaminoalkyl) - carbamic acid and thiocarbamic acid esters
IPC: C07C271/20
Filed: 1967-11-24
Abstract: Seeds are fungicidally treated with a compound_of the general formula wherein R represents an aliphatic hydrocarbon group, X represents an oxygen or sulphur atom, and n represents an integer within the range of from 1 to 5. The compound may be in admixture with (a) a liquid carrier together with a wetting, emulsifying, or dispersing agent or an adhesive, or (b) a solid carrier or mixture of liquid and solid carriers. Suitable carriers are water, xylene, chlorobenzene, cyclohexanol, cyclohexanone, dioxan, aceto nitrile, ethyl acetate, dimethyl formamide, dimethyl sulphoxide, lime, kaolin, chalk, talcum, attaclay, and silicic acid. Suitable surfactants are salts of ligninsulphonic acid and alkylated benzenesulphonic acids, sulphonated acid amides and their salts, polyethoxylated amines, and alcohols. A dyestuff, such as New Fuchsine, may be added.
Patent ES-348781-A1 (ES)
Title: New Phenothiazine Derivatives and Process for their Production
IPC: A61K31/00
Filed: 1967-12-29
Abstract: The invention comprises 10-[3-(N-formyl-N- methylamino) - propyl] - phenothiazine and the corresponding 3-chloro-compound and their preparation by reacting an N-alkali metal derivative of phenothiazine or 3-chlorophenothiazine with a reactive derivative of 3-hydroxy- 1 - (N - formyl - N - methylamino) - propane or by formylating a 10-(3-methylaminopropyl)- phenothiazine or 10-(3-methylaminopropyl)-3- chlorophenothiazine. Therapeutic compositions for oral or parenteral administration and having CNS depressant and analgesic properties comprise the compounds of the invention with a carrier.
Patent ES-358151-A1 (ES)
Title: Neutron-generating targets
IPC: H05H3/06
Filed: 1968-09-14
Abstract: A target, for neutron production by deuterium or tritium bombardment, is formed of a mixture of metal hydrides. A mixture of required metal powders is heated in an atmosphere of deuterium or tritium to form the hydrides. The proportions of the metals are selected so as to cause a zero volume charge during hydriding in the mixture and thus to preserve a high mechanical stability.