baber/WOPTO huggingface dataset:
Patent IL-91556-A0 (IL)
Title: Substituted 2-aminopyrimidine derivatives,their preparation and their use as pesticides
IPC: C07D401/12
Filed: 1989-09-07
Abstract: Compounds of the formula <IMAGE>  in which: R1 denotes phenyl or phenyl which is monosubstituted to trisubstituted by R4; R2 denotes hydrogen, C1-C5-alkyl, C1-C5-alkyl substituted by the radicals OR5 or SR5, C3-C6-cycloalkyl, C3-C6-cycloalkyl monosubstituted to trisubstituted by C1-C4-alkyl or halogen, C2-C5-alkenyl, C2-C5-alkynyl or the formyl radical; R3 denotes hydrogen, C1-C4-alkyl, C1-C4-alkyl which is substituted by halogen, cyano or the radicals OR5 or SR5, C3-C6-cycloalkyl or C3-C6-cycloalkyl which is monosubstituted to trisubstituted by C1-C4-alkyl or halogen; R4 denotes halogen, C1-C3-alkyl, C1-C2-haloalkyl, C1-C3-alkoxy or C1-C3-haloalkoxy; R5 denotes hydrogen, C1-C5-alkyl, C3-C5-alkenyl, C3-C5-alkynyl or the radical (CH2)n-X-C1-C3-alkyl;  R7 denotes the group -NH2, <IMAGE> or <IMAGE>;  R8 denotes hydrogen, C1-C3-alkyl or C1-C3-haloalkyl; R9 denotes hydrogen, C1-C8-alkyl, C1-C3-alkyl substituted by hydroxyl, OR12, SR12 or N(R12)2, C3-C6-cycloalkyl, cyclopropyl substituted by SR12, C3-C10-alkenyl, C1-C3-haloalkyl, phenyl, phenyl which is monosubstituted to trisubstituted by halogen, C1-C3-alkyl, C1-C3-alkoxy, C1-C3-haloalkoxy, C1-C2-haloalkyl, hydroxyl, nitro, cyano, amino or dimethylamino, 1- or 2-naphthyl, 1-, 2- or 3-pyridyl,   <IMAGE> or <IMAGE>; R8 and R9, together with the carbon atom in the radical R7, form a saturated or unsaturated ring consisting of 4 to 7 carbon atoms; R10 denotes CH(R8)R9, phenyl, C3-C5-alkenyl, C3-C5-alkynyl or cyanoalkyl having 2 or 3 carbon atoms in the alkyl radical; R11 denotes hydrogen, C1-C5-alkyl, C3-C5-alkenyl, C3-C5-alkynyl or cyanoalkyl having 2 or 3 carbon atoms in the alkyl radical;  R12 denotes CH3 or C2H5;  X denotes oxygen or sulphur;  Z denotes O, S, NH or NCH3; and  n denotes 1 to 3; including their acid addition salts and metal salt complexes, have useful microbicidal properties. The novel active compounds can be employed in plant protection for preventing the attack of crop plants by phytopathogenic microorganisms or by harmful insects and for controlling these pests.
Patent IL-91945-A0 (IL)
Title: Digital modulator
IPC: H04L27/12
Filed: 1989-10-11
Abstract: A modulation circuit is used in a GMSK modulation system. The system includes I-channel (210) and Q-channel (212) ROM look-up tables, each preprogrammed for generating a representative digital waveform based on an input data stream (250) and a clock signal (252). Each digital waveform is converted to an analog signal for subsequent radio frequency (RF) modulation. Each ROM is addressed by an interpolation counter (224) controlled by the clock signal (252), by a data shift register (226) receiving the input data (250) at a rate corresponding to the clock signal, and by a quadrant register (230), also receiving the input data for specifying the phase of the data signal with respect to the clock signal. Additionally, a signal (242) indicating the arrival of a non-integer bit interval is provided. In response to this signal, ROM addressing is updated in order to provide control of the modulated carrier's phase angle.
Patent AU-PR406701-A0 (AU)
Title: Crown wheel forging method and apparatus
IPC: B21J13/14
Filed: 2001-03-29
Abstract: A method of producing a bevel gear, particularly a bevel ring gear, the bevel gear comprising mounting surfaces. The method comprising the steps of flashless warm forging a blank, preferably an annular blank, in a forging die to produce the bevel gear with precision forged teeth; performing a hardening operation on the teeth; and then, without machining, finishing the teeth by lapping the teeth with a mating bevel gear. A die apparatus for use in a press for forging the bevel ring gear from the annular blank is also disclosed.
Patent FI-20050507-A0 (FI)
Inventor: SEPPAE HEIKKI
IPC: H01Q7/00
Filed: 2005-05-12
Abstract: The invention relates to an antenna construction for a double-ended antenna circuit 4. The antenna construction comprises a conductive ground place (6) on a first surface, a transmission line (3) on at least one second surface, connected to the ground plane (6) through a fold (1) in the edge of the antenna construction, so that the fold acts as a primary source of a magnetic field, an insulation layer (7) arranged between the first and the second surfaces, and an electronic component (4), in which there is a double-ended antenna connector, connected to the antenna construction. According to the invention, the electronic component (4) is attached to the second surface of the antenna construction and connected from the first antenna terminal to the transmission line (3) and from the second terminal to either a second transmission line (3) or the fold (1).
Patent FI-20085817-A0 (FI)
Inventor: AUVINEN RISTO
IPC: F01C/
Filed: 2008-09-02
Abstract: The invention relates to a planetary-motion rotary piston engine which includes a polygonal piston (I)5 a motion space of the piston where the motions of the piston (1) are arranged rotating around two polar axes by alternate strokes and, when moving the piston (1) at a smooth velocity of rotation, the successive striking motions of the piston angle are equal of their angular velocity on successive paths which are symmetrical with each other in relation to a symmetry plane halving the distance between the polar axes, and a power transmission device. According to the invention, in connection with a centre shaft (3) of the piston (1) of the planetary-motion rotary piston engine moved by alternate strokes around two different polar axes (P, Pl) in the rotation space there is a planetary shaft (P3) being the rotation axis of rotation, moving planetarily rotating along a path. When an extreme end of an eccentric structure of the moving piston (1) is at relatively long distances from the planetary shaft (P3) and the rotation support shaft (P or Pl), the planetary-motion rotary piston engine has a large rotational volume in relation to the size of the piston, whereby large volume changes required for enlarging and compressing are created and the piston can better utilise the expansion and compression of medium.
Patent IL-100772-A0 (IL)
Title: Optical fiber connector
IPC: G02B6/00
Filed: 1992-01-27
Abstract: A prior optical fiber connector (20) includes an elongated mandrel (21) of substantially uniformly elliptical cross section that is encompassed by a resiliently deformable housing (26) which, in its relatively undeformed state, can optically interconnect two optical fibers by urging their ends against a straight longitudinal groove in the surface of the mandrel (21). The interconnection can be made more easily when there is, either integral with or around the housing, an envelope (27) incorporating a pair of second-class levers (28) which, when squeezed together by ones fingers, deform the housing. The extremities of the levers can be formed to permit the connector to be releasably attached to a patch panel or to an optical fiber distribution module. <IMAGE>
Patent IL-110956-A0 (IL)
Title: Hydroxy-substituted azetidinone compounds useful as hypocholesterolemic agents
IPC: A61P7/00
Filed: 1994-09-13
Abstract: Hydroxy-substd. azetidinone derivs. of formula (I) and their salts are new. Ar1,Ar2 = aryl (opt. substd. by 1-5 gps. R4); Ar3 = aryl (opt. substd. by 1-5 gps. R5); X, Y, Z = CH2, CH(1-6C alkyl) or C(di(1-6C alkyl); R, R2 = OR6, OCOR6, OCOOR9 or OCONR6R7; R1, R3 = H, 1-6C alkyl or aryl; q, r = 0 or 1; m, n, p = 0-4, provided that i) at least one of q and r is 1, and the sum of m, n q and r is 1-6, and ii) when p is 0 and r is 1, the sum of m, q and n is 1-5; R4 = 1-6C alkyl, OR6, OCOR6, OCOR9, O(CH2)sOR6, OCONR6R7, NR6R7, NR6COR7, NR6COOR9, NR9, NR6CONR7R8, NR6CONR7R8, NR6SO2R9, COOR6, CONR6R7, COR6, SO2NR6R7, S(O)tR9, O(CH2)uCOOR6, O(CH2)uCONR6R7, lower alkylCOOR6, CH=CH-COOR6, CF3, CN, NO2 or halogen; R5 = OR6, OCOR6, O(CO)R9, O(CH2)vOR6, -O(CO)NR6R7, NR6R7, NR6COR7, NR6COOR9, NR6COOR9, NR6CONR7R8, NR6SO2R9, COOR6, CONR6R7, COR6, SO2NR6R7, S(O)tR9, -O(CH2)uCOOR6, O(CH2)uCONR6R7, lower alkylCOOR6 or -CH=CH-COOR6; s = 1-5; t = 0-2; u = 1-10; v = 1-5; R6, R7, R8 = H, 1-6C alkyl (opt.substd. with aryl) or aryl; and R9 = 1-6C alkyl (opt. substd. with aryl) or aryl.
Patent IL-112099-A0 (IL)
Title: N-oxides of 4-arylpiperazines and 4-arylpiperidines and pharmaceutical compositions containing them
IPC: C07D295/24
Filed: 1994-12-21
Abstract: Compounds of general formula (I) are disclosed as novel antipsychotic agents.
Patent IL-117684-A0 (IL)
Title: Novel intermediates and process for the manufacture of camptothecin derivatives (CPT-11) and related compounds
IPC: C07D471/14
Filed: 1996-03-27
Abstract: PCT No. PCT/US96/04163 Sec. 371 Date Oct. 2, 1997 Sec. 102(e) Date Oct. 2, 1997 PCT Filed Apr. 1, 1996 PCT Pub. No. WO96/31513 PCT Pub. Date Oct. 10, 1996This invention relates to intermediates and processes for the synthesis of camtothecin derivatives, such as irinotecan. Related procedures and compounds are disclosed, such as a method of making mappicine.
Patent IL-128568-A0 (IL)
Title: Use of cyclooxygenase-2 inhibitors for the manufacture of a medicament for the treatment and prevention of neoplasia
IPC: C07D417/04
Filed: 1997-10-14
Abstract: The present invention relates to a pharmaceutical composition for the treatment of a neoplasia, which comprises a compound of formula II and an anti-neoplastic agent
Patent IL-133663-A0 (IL)
Title: Method for production of hydroxylamine sulfate in the conventional process for the synthesis of caprolactam
IPC: C07D201/06
Filed: 1999-12-22
Abstract: An improvement in the conventional process for the production of caprolactam. The process involves:   (a) reacting air with ammonia gas in an ammonia conversion zone to produce nitric oxide; (b) oxidizing a portion of the nitric oxide to nitrogen dioxide to produce an NOx-rich process gas stream; (c) reacting the NOx-rich stream with ammonium carbonate in a nitriting zone to produce ammonium nitrite; (d) reducing the ammonium nitrite to hydroxylamine diammonium sulfate; (e) hydrolyzing the hydroxylamine diammonium sulfate to hydroxylamine sulfate; (f) oximating the hydroxylamine sulfate with cyclohexanone to produce cyclohexanone oxime; and   (g) converting the cyclohexanone oxime to caprolactam. The process is improved by adding supplemental oxygen downstream of the ammonia conversion zone to increase the quantity and rate of formation of nitrogen dioxide in the NOx-rich process gas stream. <IMAGE>
Patent IL-136735-A0 (IL)
Title: Substituted 2-benzylamino-2-phenyl-acetamide compounds
IPC: A61P25/00
Filed: 1998-12-12
Abstract: Compounds which are substituted 2-benzylamino-2-phenyl-acetamide compounds of formula (I)wherein:n is zero, 1, 2 or 3;X is -O-, -S-, -CH2- or -NH-;each of R, R1, R2 and R3, independently, is hydrogen, C1-C6 alkyl, halogen, hydroxy, C1-C6 alkoxy or trifluoromethyl;each of R4 and R5, independently, is hydrogen, C1-C6 alkyl or C3-C7 cycloalkyl; or pharmaceutically acceptable salts thereof, are useful in treating conditions such as chronic or neuropathic pain.
Patent IL-137255-A0 (IL)
Title: Frozen food product
IPC: A23G9/32
Filed: 1998-12-23
Abstract: A process for the manufacture of a frozen food product comprising antifreeze peptides, wherein the process comprises one or more of the following steps; (i) a (pre-) freezing) step which is a nucleation dominated freezing process; (ii) a (post-) compaction step using a screw extruder or a (piston) compactor; The invention aims at providing the food manufacturer with a greater flexibility for using antifreeze peptide material in frozen food products when aiming to obtain a product with improved recrystallization properties in combination with a good texture. In particular it has been found that the texture of frozen food products containing antifreeze peptides can markedly be improved by carefully controlling its production method.
Patent IL-138345-A0 (IL)
Title: Novel compositions of epropsartan
IPC: A61K9/14
Filed: 1999-03-11
Abstract: This invention relates to a novel composition comprising eprosartan, or a salt, solvate, or hydrate thereof, in particulate form, a process for its production and methods of using the composition to block angiotensin II receptors and to treat hypertension, congestive heart failure and renal failure.
Patent IL-141392-A0 (IL)
Title: Orientation-directed construction of plasmids
IPC: C12N15/66
Filed: 2001-02-12
Abstract: A method for orientation-directed construction of a construct including at least two nucleic acid segments of interest. Products are provided having phosphorylated blunt ends derived from the nucleic acid segments of interest. Separate ligation reactions are performed wherein in each reaction the phosphorylated blunt-ended products of two different segments obtained in the previous step are ligated to create a combined ligated sequence. PCR amplification reaction is performed using the combined ligated sequence obtained in the previous step as a template and specific enrichment primers direct the PCR amplification towards the desired orientation. Each combined ligated sequence is amplified in a separate reaction creating a combined product having phosphorylated blunt ends. The combined product is isolated and purified to have the enriched desired orientation. Self-ligation of the isolated purified combined product is performed to create a circular double-stranded DNA construct containing the desired segments properly aligned and operably linked.
Patent IL-146882-A0 (IL)
Title: Robust autofocus system for a microscope
IPC: G02B7/36
Filed: 2000-05-30
Abstract: The present invention provides a method and apparatus for autofocusing of an optical instrument, especially a microscope (10). The autofocus scheme includes a digital gradient filter for generating a focus score from each captured image. Images may be captured at various positions and the focus scores analysed to determine a focus score maximum. The position corresponding to this maximum is then taken as the focus position. The spatial extent of the filter is preferably settable so that the digital filter settably selects elements of the image depending on their size in the image. Thus, the filtering process is controllable so that it is influenced by elements of the image whose size may be specified by the operator indirectly by way of the spatial extent of the filter. This allows the exclusion of small or large elements of the image from the autofocusing procedure which the filter should preferably ignore. The autofocus scheme is particularly useful for autofocusing biological specimens.
Patent IL-154778-A0 (IL)
Title: RECEPTOR IN THE EDb FIBRONECTIN DOMAIN
IPC: G01N33/50
Filed: 2001-08-30
Abstract: The invention relates to a protein that binds specifically to the ED<SUB>b</SUB>-fibronectin domains, process for screening compounds that bind to a receptor of the ED<SUB>b</SUB>-fibronectin domains or to ED<SUB>b</SUB>-fibronectin domains themselves, as well as the uses of protein.
Patent IL-156514-A0 (IL)
Title: Improved vascular prosthesis and method for production thereof
IPC: B29C67/20
Filed: 2001-12-17
Abstract: An apparatus for forming a tubular structure from a liquefied polymer, the apparatus comprising: (a) a dispenser for dispensing the liquefied polymer; (b) a precipitation electrode being at a first potential relative to the dispenser, the precipitation electrode being designed and constructed for generating a polymeric shell thereupon; and (c) a mechanism for increasing a local density of the polymeric shell in a plurality of predetermined sub-regions of the polymeric shell, thereby to provide a tubular structure having an alternating density in a longitudinal direction.
Patent IL-156860-A0 (IL)
Title: Cutting head for machine tool
IPC: B23B29/03
Filed: 2002-01-15
Abstract: The invention concerns a cutting head ( 13 ) to be secured in an adapter ( 9 ) in a machine tool for chip removing machining. The cutting head ( 13 ) comprises a flange with a first side creating a coupling surface ( 4 ) adapted for being secured to the adapter ( 9 ). On the opposite of the flange, it is situated an other side creating at least one surface ( 1 A) with an outwards extending protrusion ( 8 ), with securing means adapted for securing a cutting insert ( 5 ) with at least one cutting edge. The weight of the cutting head ( 13 ) is reduced as compared to the strength of the cutting head ( 13 ), and the natural frequency of the cutting head ( 13 ) is thereby increased when this is secured to the adapter ( 9 ).
Patent IL-172134-A0 (IL)
Title: Use of 2,2,3,3, tetramethylcyclopropane carboxylic acid derivatives for treating psychiatric disorders
IPC: A61K31/16
Filed: 2005-11-23
Abstract: The invention relates to the use of 2,2,3,3 tetramethylcyclopropane carboxylic acid derivative compounds for the preparation of a medicament for treating a psychiatric disorder preferably a bipolar disorder. The invention additionally relates to the use of the compounds for the preparation of an inhibitor of MIP synthase and to a pharmaceutical composition comprising the compounds for treating a psychiatric disorder. A method for treating a psychiatric disorder preferably a bipolar disorder and a method for inhibiting an enzyme having MIP synthase activity is provided.
Patent IL-176263-A0 (IL)
Title: Flame retardant compositions and their use
IPC: C08L25/02
Filed: 2006-06-12
Abstract: Disclosed are flame retardant compositions comprised of (a) brominated anionic styrenic polymer, and (b) at least one polybrominated alpha-omega diphenylalkane having a total of at least 6 bromine atoms directly bonded to the phenyl rings and in the range of 1 to 6 carbon atoms in the alkylene group disposed between the phenyl groups, and specified flame retarded polymer compositions with which have been blended (a) and (b) individually or in combination.
Patent IL-188257-A0 (IL)
Title: Bovine abcg2 gene missense mutations and uses thereof
Filed: 2007-12-19
Abstract: A quantitative trait locus (QTL) affecting milk fat and protein concentration was localized to a 4cM confidence interval on chromosome 6 centered on the microsatellite BM143. The genes and sequence variation in this region were characterized, and common haplotypes spanning five polymorphic sites in the genes IBSP, SPP1, PKD2, and ABCG2 for two sires heterozygous for this QTL were localized. Expression of SPP1 and ABCG2 in the bovine mammary gland increased from parturition through lactation. SPP1 was sequenced, and all the coding exons of ABCG2 and PKD2 were sequenced for these two sires. The single nucleotide change capable of encoding a substitution of tyrosine-581 to serine (Y581S) in the ABCG2 transporter was the only polymorphism corresponding to the segregation status of all three heterozygous and 15 homozygous sires for the QTL in the Israeli and US Holstein populations.
Patent IL-200778-A0 (IL)
Title: Unitary accommodating intraocular lenses (aiols) and discrete base members for use therewith
Filed: 2009-09-06
Abstract: Unitary accommodating intraocular lenses (AIOLs) including a haptics system for self-anchoring in a human eye's ciliary sulcus and a resiliently elastically compressible shape memory optical element having a continuously variable Diopter strength between a first Diopter strength in a non-compressed state and a second Diopter strength different than its first Diopter strength in a compressed state. The unitary AIOLS include an optical element with an exposed trailing surface and are intended to be used with a discrete base member for applying an axial compression force against the exposed trailing surface from a posterior direction. Some unitary AIOLs are intended to be used with either a purpose designed base member or a previously implanted standard in-the-bag IOL. Other unitary AIOLs are intended to be solely used with a purpose designed base member.
Patent IL-211777-A0 (IL)
Title: System for electrically connecting batteries to electric vehicles
IPC: H01M50/249
Filed: 2011-03-17
Abstract: A method of exchanging a battery in an at least partially electric vehicle comprises removing a first battery from a cavity in an underside of an at least partially electric vehicle, inserting the second battery into the cavity in the underside of the at least partially electric vehicle, temporarily storing at least one of said first and second batteries in a standby location (1308) during said exchange process to thereby reduce a time duration required for said exchange process.
Patent RO-125648-A0 (RO)
Title: Seeder for hoeing plants
Inventor: CIUBUCCIU GHERASIM
IPC: A01C7/04
Filed: 2010-04-19
Abstract: The invention relates to a seeder with electro-vacuumetric distribution for hoeing plants. According to the invention, the seeder consists of a feeding chamber (1) inside which there is mounted, coaxially with the axis thereof, an axle (2) having in cross section a square form which has mounted, at an end, a stirrer (3) and a distributing disk (4), and, at the other end, there is provided a driving channel (a), inside thereof there is a driving pin (5) mounted on the shaft of an electric motor (6) of variable speed mounted on some fastening supports (7), which, in their turn, are positioned on a supporting cover (8) by means of some fixing screws (9), the electric motor (6) having the role of rotating the distributing disk (4) depending on a distance (d) between some grains (22), in order to obtain the vacuum needed for driving the grains (22) on the disk (4), there being used an electro-ventilator (16) or a mini-exhauster (31).
Patent RO-126938-A0 (RO)
Title: Nano-nickel core, process for preparing the same and installation for producing heat energy, equipped with such a core
Inventor: IONESCU CAZEMIR BENEDICT
IPC: B22F9/02
Filed: 2011-06-27
Abstract: The invention relates to a nano-nickel core, to a process for preparing the same, and to an installation equipped with such a core which produces thermal energy. According to the invention, the core consists of a support sponge with high thermal conductivity such as copper, nickel, iron, stainless steel, graphitic carbon, titanium carbide and similar, whereon there is applied a matrix of graphitic carbon with open pores, having a pore diameter in the range of 3...50 nm, which contains in the open meso-pores nickel nano-crystals, inside the open pores of the support sponge there being an alkaline metal such as sodium, potassium or an alloy thereof together with a catalyst system. The claimed process consists in the synthesis of a matrix made of graphitic carbon on the walls of cells with open porosity using as matrix with controlled architecture, a silicate or an aluminosilicate, the formed pores will be useful as matrix wherein there are deposited the nickel nano-crystals, and finally the open pores of the support sponge are filled with alkaline metal and with other components of the catalytic system. The installation equipped with one or several nano-nickel cores, as claimed by the invention, comprises a system for producing thermal energy, a system for preheating and triggering the reactions, a heat exchange system of thermal syphon type, whose evaporation-boiling area comprises a metal cylinder () made of copper or aluminium wherein there are dug some boiling channels (), with a heating resistor () of the heat producing vessel () closed with a cap (), a pipe () for hydrogen supply provided with a tap () a condensing-cooling area comprising a cupola () fixed on the cylinder () through the flange () a conduit () with a tap () and a worm () wherethrough the secondary cooling fluid circulates, and the system for thermal insulation and a shield for protection against radiation.