baber/WOPTO huggingface dataset:
Patent ME-P22508-A (ME)
Inventor: BADORC ALAIN
IPC: C07D221/00
Filed: 2003-04-02
Abstract: Predmetni pronalazak se odnosi na derivate formule I: gdje: R1 predstavlja -OH, (C1-C5)alkoksi, karboksil, (C2-C6)-alkoksikarbonil, -NR5R6, -NH-S02-Alk; -NH-S02-Ph, -NH-CO-Ph, -N(Alk)-CO-Ph; -NH-CO-NH-Ph, -NH-CO-Alk, -NHC02-Alk, -0-(CH2)n-cAlk, -O-Alk-COOR7, -O-Alk-0-Rx, -O-Alk-OH, -0-Alk-C(NH2)NOH, -0-Alk-NR5R6, -O-Alk-CN, -0-(CH2)n-Ph, -0-Alk-CO-NR5R6, -CO-NH-(CH2)m-COOR7, CO-NH-Alk; R2 predstavlja H, (C1-C5)alil, (C1-C5)alkil halogenid, (C3-C6)cikloalkil ili fenil koji je po potrebi susptituisan; A predstavlja radikal -CO-, -SO- ili -S02-,; R3 i R4, isti ili različiti, svaki predstavlja H, (C1-C5)alkoksi, amino, karboksil, (C2-C6)-allkoksikarbonil, -OH, nitro, hidroksiamino, -Alk-COOR7, -NR5R6, -NH-Alk-COOR7. -NH-COO-Alk, -N(R11)-SO2-Alk-NR9R10, -N(R11)-S02-Alk, -N(R11)-S02-Alk-NR5R6, -N(R11)-CO-Alk-NR9R10, -N(R11)-CO-Alk, -N(R11)-CO-CF3, -NH-Alk-HetN, -0-Alk-NR9R10, -0-Alk-CO--NR5R6, -O-Alk-HetN; ili R3 i R4 zajedno obrazuju 5- ili 6-člani nezasićen heterocikl, po potrebi u vidu jedne od farmaceutski prihvatljivih soli.
Patent YU-17404-A (YU)
Title: Novel pyrroles having hypolipidemic hypocholesteremic activities, process for the preparation and pharmaceutical compositions containing them and their use in medicine
Inventor: LOHRAY BRAJ BHUSHAN
IPC: G06F3/14
Filed: 2002-07-25
Abstract: The present invention relates to novel substituted pyrrole compounds, their derivatives, their analogs, their tautomeric forms, their stereoisomers, their polymorphs, their pharmaceutically acceptable salts, their pharmaceutically acceptable solvates and pharmaceutically acceptable compositions containing them. This invention particularly relates to novel substituted pyrrole compounds of the general formula (I), their analogs, their derivatives, their polymorphs, their tautomeric forms, their pharmaceutically acceptable salts, their pharmaceutically acceptable solvates and their pharmaceutical compositions containing them. The invention also relates to the process for preparing such compounds, a composition containing such a compound and the use of such a compound and composition in medicine. The compounds lower triglyceride levels in blood and may be useful in the treatment of obesity, hyperlipidaemia, hypercholesteremia, syndrome X and diabetes.
Patent AU-1074201-A (AU)
Title: Surgical instrument for ablation and aspiration
Inventor: SHARKEY HUGH R
IPC: A61B17/00
Filed: 2000-10-05
Abstract: An electrosurgical aspiration instrument that permits aspiration of an area being treated by the instrument. The instrument is coupled at a proximal end to a power source and includes an energy application surface area at a distal end. The power source supplied energy to the energy application surface area such that the distal end of the instrument may apply energy to the treatment area to modify the characteristics of biological material, such as biological tissue in the area. An aspiration lumen is formed through the instrument with an opening through the energy application surface area. The energy application surface area is configured to reduce blockage of the opening. Accordingly, aspiration may be performed simultaneously with electrosurgical treatment whereby unwanted matter such as by-products, biological debris and excess fluid is removed from the treatment area. The electrosurgical aspiration instrument also permits both functions to be performed at different times, with the advantage of not requiring instruments to be switched on during the treatment procedure or removed from the treatment site.
Patent AU-1161300-A (AU)
Title: Treatment set containing lungsurfactant compositions
Inventor: GERMANN PAUL-GEORG
IPC: A61P11/00
Filed: 1999-11-09
Abstract: The invention describes a set for the treatment of IRDS, ALI or ARDS, comprising a first container which has a volume of 50 to 500 ml and contains a pulverulent pulmonary surfactant preparation, the amount of phospholipids in the container being 50 to 500 mg, and a second container which has a volume of 50 to 500 ml and contains a pulverulent pulmonary surfactant preparation, where the amount of phospholipids in the second container is 1 to 10 g.
Patent AU-1182595-A (AU)
Title: Fluxless soldering pretreating system and method using fluorine-containing plasma
Inventor: BOBBIO STEPHEN M
IPC: B23K1/20
Filed: 1994-11-16
Abstract: A fluxless soldering sample pretreating system includes a sample chamber having an opening therein and a sample holder. A sample chamber extension extends outwardly from the opening to define a passageway from the sample chamber extension, through the opening, and into the sample chamber. A fluorine-containing gas is supplied into the sample chamber extension. Am energy source such as a microwave oven surrounds the sample chamber extension. The microwave oven produces microwave energy in the sample chamber extension to form a plasma therein and dissociate the fluorine-containing gas into atomic fluorine. A perforated aluminum plate extends transversely across the passageway and blocks the plasma from traversing the passageway from the sample chamber extension into the sample chamber, while allowing the atomic fluorine to traverse the passageway from the sample chamber extension into the sample holder. A second chamber extension, gas supply and microwave oven may be added to improve uniformity for large samples.
Patent AU-1284697-A (AU)
Title: Method for treating excessive aggression
Inventor: BEASLEY CHARLES M JR
IPC: A61K31/5513
Filed: 1996-12-04
Abstract: The invention provides a method for treating extreme aggression comprising administering an effective amount of olanzapine to a patient in need thereof.
Patent AU-1400799-A (AU)
Title: Spring interior and method of making same
Inventor: GRUENINGER SIEGFRIED
IPC: A47C27/06
Filed: 1998-11-12
Abstract: The spring interior (10) comprises springs (12) with different spring constants (hardness). The variation of the spring constant is effected by changing the average radius of the windings (13) between the central winding (15) and the two end rings (14) of each individual spring. With a spring winding machine (21) whose bending tools can be set and adjusted by software during the production, in this manner spring interiors (10) may be manufactured which comprise any amount of zones of differing hardness. With this, all springs (12) consist of wire with the same diameter, the same end ring (14) diameter and the same height, and the automatic manufacture may be effected without conversion of the spring interior assembly automatic machines.
Patent AU-1432888-A (AU)
Title: Double bellows purge valve
Inventor: CORNIEA DONALD G
IPC: B65B39/04
Filed: 1988-04-07
Abstract: The unit (10) includes a first valve element (24) that is held within a liquid passageway by a first spring mechanism (40). This spring mechanism is designed to yield under pressure to allow the first valve element to move off a valve seat (26) in the opening to allow liquid to pass through. In order to allow air that is trapped on the downstream side of the valve element to escape, air vents (42) are provided in the first valve element. A second valve element (44) is held under compressive force by a second spring (46) over air vents located in the first valve element.
Patent AU-1505895-A (AU)
Title: Biphenyl derivatives
Inventor: AKASAKA KOZO
IPC: C07D295/096
Filed: 1995-03-24
Abstract: A biphenyl derivative represented by the following formula (I) or a pharmacologically acceptable salt thereof: <CHEM> wherein R<1> represents a hydrogen atom, a halogen atom, a hydroxyl group, an amino group, a lower alkyl group, a halogenated lower alkyl group, a lower alkoxy group, a halogenated lower alkoxy group, a lower alkoxyalkyl group, a lower alkoxyalkoxy group, an aryl group, an aralkyl group, a heteroaryl group, a heteroarylalkyl group, a halogenated heteroarylalkyl group, a cyano lower alkyl group, a hydroxy lower alkyl group, an amino lower alkyl group, a lower alkoxycarbonyl group, an aryloxycarbonyl group, a cyano group, a formyl group, a lower acyl group, an aralkylcarbonyl group, a cycloether group, an alkenyl group, an alkynyl group, a lower alkylsulfinyl group, a lower alkylsulfonyl group, a lower alkylaminosulfonyl group, an arylaminosulfonyl group, a lower alkylsulfonylamino group, a halogenated lower alkylsulfonylamino group or an arylsulfonylamino group; R<2> and R<3> may be the same or different from each other and each represents a hydrogen atom, a halogen atom, a lower alkyl group, a halogenated lower alkyl group, a lower alkoxy group, a halogenated lower alkoxy group or a cyano group; R<4> represents a hydrogen atom or a halogen atom; R<5> represents a hydrogen atom, a lower alkyl group, a halogenated lower alkyl group, a hydroxy lower alkyl group, a lower alkoxycarbonyl group or an aryloxycarbonyl group; and n is 0 or an integer of 1 to 3, which exhibits dopamine 2 receptor antagonism and/or serotonin 2 receptor antagonism, is clinically useful for treating and ameliorating mental disorders such as cerebrovascular disorder, aggressive behavior due to senile dementia, mental excitation, poriomania, delirium, hallucination, hyperkinesia, schizophrenia, emotional disturbance, depression, neurosis, psychophysiologic disorder and anxiety neurosis.
Patent AU-1600892-A (AU)
Title: Reduction products of rapamycin as immunosuppressants, antiinflammatory or antifungal agents
IPC: A61P29/00
Filed: 1992-05-05
Abstract: Products of formula (I) obtained from the chemical reduction of one or more of the ketone groups at positions 15, 27 and 33 of Rapamycin with diisobutylaluminum hydride or sodium triacetoxyborohydride have been shown to have pharmacological properties which would make them useful in the treatment of transplantation rejection, autoimmune diseases, diseases of inflammation and Candida albicans infections. <CHEM> u
Patent AU-1802695-A (AU)
Title: Euphausiid harvesting and processing method and apparatus
Inventor: SAXBY DAVID J
IPC: A01K61/00
Filed: 1995-02-28
Abstract: Method and apparatus for harvesting and processing zooplankton and, in particular, for harvesting and processing euphausiids for subsequent use as a feed product for early stage juvenile or larvae feed or for a food product as an additive. The euphausiids are continuously harvested from coastal waters and dewatered. The dewatered product is passed to a heat exchanger (50) to increase its temperature and, thence, to a digester (51) where a desired level of enzymatic activity is obtained. The product is then held by a surge tank (80) for subsequent transfer to a ball dryer (81) where the product is dried at a relatively low temperature without destroying the stabilized enzymes created in the digester. The digesting step may be deleted in the event the use of the product is for a food product. <IMAGE>
Patent AU-1812795-A (AU)
Title: Novel amino acid derivatives, method of producing them and pharmaceutical compositions containing these compounds
Inventor: ESSER FRANZ
IPC: C07K5/02
Filed: 1995-03-02
Abstract: The invention relates to new amino acid derivatives of general formula I    <IMAGE>  (I)  and the pharmaceutically acceptable salts thereof, wherein the group R2 is   <IMAGE>   and R1, A, G, Y, Z and m have the meanings given in the specification, and the preparation and use thereof. The new compounds are valuable neurokinin (tachykinin)-antagonists.
Patent AU-1841300-A (AU)
Title: Carboxylic acids and carboxylic acid isosteres of n-heterocyclic compounds
Inventor: HAMILTON GREGORY S
IPC: A61K31/401
Filed: 1999-12-03
Abstract: This invention relates to novel N-heterocyclic carboxylic acids and carboxylic acid isosteres, their preparation and use for treating neurological disorders including physically damaged nerves and neurodegenerative diseases, for treating alopecia and promoting hair growth, for treating vision disorders and/or improving vision, and for treating memory impairment and/or enhancing memory performance by administering such compounds.
Patent AU-2056695-A (AU)
Title: Mold separation method and apparatus
Inventor: KINDT-LARSEN TURE
IPC: B29C33/00
Filed: 1995-06-09
Abstract: The present invention provides an apparatus for separating individual contact lens mold assemblies using a steam and demolding means.
Patent AU-2102899-A (AU)
Title: Graphic layout controller for television environment
Inventor: WUGOFSKI THEODORE D
IPC: G06F9/44
Filed: 1999-01-05
Abstract: The present invention utilizes a graphics layout language that is defined by the broadcaster or the studio to control the layout of graphic overlays in relation to corresponding images presented on a display. Each user interface component is divided into objects that define their individual behaviors and presentations. Data files using the hypertext markup language, HTML, layout these objects on the screen. By varying the HTML data files, control is provided to the broadcaster over what objects are displayed on the screen, where they are placed on the screen, and to a limited effect, their behavior. This can be accomplished without re-writing the executables as would be necessary in other television type user interface implementations.
Patent AU-2537092-A (AU)
Title: N-alkyl-3-phenyl-3-(2-alkylthiophenoxy)propylamines
IPC: C07C217/48
Filed: 1992-09-25
Abstract: This invention provides N-alkyl-3-phenyl-3-(2-substituted phenoxy)propylamines which are useful to treat neurological disorders associated with norepinephrine imbalance.
Patent AU-2683484-A (AU)
Title: Composition for treating atrophic rhinitis
Inventor: MAGYAR KAROLY
IPC: A23K20/195
Filed: 1984-04-13
Abstract: 1. Claims for the Contracting States : BE, CH, DE, FR, GB, IT, LI, NL, SE Medicaments and/or feed concentrates having an antibacterial activity and a content of a) 2-[(methoxycarbonylhydrazono)-methylene]-quinoxaline-1,4- dioxide, characterized in that it contains b) 2-(methyl)-5,7-di-(chloro)-8-(hydroxy)-quinoline as another (other) active ingredient(s). 1. Claims for the Contracting State : AT A process for preparing medicaments and/or feed concentrates having an antibacterial activity and a content of a) 2-[(methoxycarbonylhydrazono)-methylene]-quinoxaline-1,4- dioxide and b) 2-(methyl)-5,7-di-(chloro)-8-(hydroxy)-quinoline as additional ingredient, characterized in that they are prepared by mixing these active ingredients and optionally 1 or more solid and/or liquid carrier(s) which is (are) conventional in medicaments and/or feed concentrates.
Patent AU-2763397-A (AU)
Title: Method and apparatus for grading fish according to size
Inventor: PEDERSEN OLE ENGGAARD
IPC: A01K61/90
Filed: 1997-05-05
Abstract: Fish (17) of different sizes are graded by means of gently sloping grilles (2, 3, 4, 5) consisting of smooth rounded rods or tubes extending in directions parallel to the plane of the drawing, preferably being kept wet by water sprayed from nozzles (18). In this manner, rapid grading can be achieved without damage to the fish and using relatively light equipment, as dictinct from water-filled tanks previously used for this purpose.
Patent AU-3106489-A (AU)
Title: Preparation of aqueous polyalkyl methacrylate dispersions by an emulsion polymerization in two stages and their use in wood finishes
Inventor: DEHNE HEINRICH
IPC: C08F220/14
Filed: 1989-03-07
Abstract: A process for the preparation of aqueous dispersions of alkyl methacrylate copolymers with mono- and/or dicarboxylic acids containing from 3 to 6 carbon atoms by stepwise emulsion copolymerisation in the presence of conventional water-soluble, free radical-forming polymerisation initiators and in the presence of conventional emulsifiers at conventional polymerisation temperatures is characterised in that  85.25-37.5% by weight of methyl methacrylate, 14.75-62.5% by weight of n-butyl methacrylate and/or isobutyl methacrylate, 1-5% by weight of  alpha , beta -monoolefinically unsaturated mono- and/or dicarboxylic acids containing 3-6 carbon atoms, and 0-5% by weight of amides of  alpha , beta -monoolefinically unsaturated mono- and/or dicarboxylic acids containing 3-5 carbon atoms, are polymerised in aqueous emulsion in two steps in such a manner that the dispersion has a minimum film-forming temperature of 65-110 DEG C and a light transparency of at least 85%. This dispersion is used together with a further polyalkyl methacrylate dispersion, but one which has a minimum film-forming temperature of from 20 to 60 DEG C, as a binder in wood paints.
Patent AU-3166497-A (AU)
Title: 1,2,4-benzothiadiazine derivatives, their preparation and use
Inventor: PIROTTE BERNARD
IPC: C07D453/06
Filed: 1997-06-19
Abstract: 1,2,4-Benzothiadiazine derivatives represented by formulawherein D, R1, R2, R3, R4, R5, R12, R13, R14, R15 are defined in the description, composition thereof and methods for preparing the compounds are described.The compounds are useful in the treatment of diseases of the central nervous system, the cardiovascular system, the pulmonary system, the gastrointestinal system and the endocrinological system.
Patent AU-3174293-A (AU)
Title: Ventilation device
Inventor: NILSEN TROND
IPC: F24F7/08
Filed: 1992-12-23
Abstract: PCT No. PCT/NO92/00205 Sec. 371 Date Sep. 30, 1993 Sec. 102(e) Date Sep. 30, 1993 PCT Filed Dec. 23, 1992 PCT Pub. No. WO93/13364 PCT Pub. Date Jul. 8, 1993.Ventilation device with a heat exchange element, preferably for arrangement in an outer wall (13) of premises which are to be ventilated with balanced volumes of ambient air (15). The ventilation device comprises a pair of air flow passages (23A,23B) each including two separate ventilation tubes (16,19) aligned in the direction of air flow, with generally identical heat exchange elements (18,22) at the ends thereof. A fan (24A,24B) is located centrally between the two heat exchange elements in each passage.
Patent AU-3179795-A (AU)
Title: Impedance feedback monitor for electrosurgical instrument
Inventor: YATES DAVID C
IPC: A61B17/32
Filed: 1995-09-21
Abstract: An impedance monitoring device is provided for monitoring the electrical impedance of tissue as it is treated with electrosurgical energy. Based on a predicted model of tissue impedance and a number of initial impedance readings, the impedance at which tissue treatment is completed is predicted. More particularly, a minimum impedance level is measured and a function of the minimum impedance is used to determine impedance at which coagulation is completed. A control device is provided for bringing the output of the generator within an optimum range based on a system load curve. In one embodiment the impedance monitoring device is used in conjunction with a bipolar electrosurgical instrument. Preferably, the instrument comprises electrically opposite electrodes located on one or more tissue engaging surfaces for engaging tissue to be treated. <IMAGE>
Patent AU-3211184-A (AU)
Title: Novel 1-piperazinecarboxamide derivatives
Inventor: KONRAD BJORK ANDERS KARL
IPC: C07D295/18
Filed: 1984-08-02
Abstract: 1-piparazinecarboxamide derivatives are described which have the formula (I) 
<CHEM>
 wherein R1 is a member selected from hydrogen, halogen or trifluoromethyl;
 wherein X is selected from:
 > CO (Ia)
 > CHOH (Ib) > CHOR8 (Ib min ) > CHOCOR8 (Ib sec )
 > CH2 (Ic)
 > C = CR6R7 (Id)
 > CH - CHR6R7 (Ie) 
<CHEM>
 wherein R2 and R3 are the same or different and selected from hydrogen or lower alkyl;
 wherein Z ist either oxygen or sulfur;
 wherein Y is -NR4R5, where R4 and R5 are the same or different and selected from hydrogen, alkyl, alkenyl, cycloalkyl, aryl, aryl-(lower alkyl), or R4 and R5 may together with the N-atom form a 5- or 6- or 7-membered satin red ring, where one of the carbon atoms may be exchanged for O, NR8 or NCOR8;
 wherein R6 and R7 are the same or different and selected from hydrogen or lower alkyl;
 wherein R8 is lower alkyl or lower alkenyl;
 with the proviso that when X is > CO, then R4 is hydrogen and R5 is different from hydrogen. 
<??>Pharmaceutical compositions containing said 1-piperazinecarboxamide derivates are also described. 
<??>The derivatives are useful in treating mental disorders and/or aggression in man and in treating aggression in animals and for calming animals. 
<??>Different processes for preparing the derivatives are also described.
Patent AU-3282784-A (AU)
Title: Thread rolling dies and method
Inventor: TAUBERT HUBERT
IPC: B21H3/06
Filed: 1984-09-07
Abstract: Method and dies for threading a screw comprises providing a screw blank with a portion of its length of lobular cross section and an adjacent portion of the blank of circular cross section. The blank is rolled between roll dies so as to roll the thread on the circular portion and simultaneously roll the thread at the lobes only on the lobular portion. Thereafter, the blank is rolled to additional regions of the dies wherein the thread is rolled to form on the lobular section, while the cylindrical section passes through regions of clearance or relief on the dies.
Patent AU-3340999-A (AU)
Title: Zymogenic nucleic acid detection methods, and related molecules and kits
Inventor: TODD ALISON
IPC: C12Q1/68
Filed: 1999-02-22
Abstract: This application provides methods of detecting and quantitatively determining a target nucleic acid sequence in a sample, which comprise contacting the sample with a primer and a zymogene which encodes, but which itself is the anti-sense sequence of, a catalytic nucleic acid sequence, so that when the target is present, a single amplified nucleic acid molecule is produced which comprises the sequences of both the target and catalytic molecules. This invention further provides a method of simultaneously detecting the presence of a plurality of target nucleic acid sequences in a sample. Finally, this invention provides molecules and kits for practicing the instant methods.
Patent AU-3540889-A (AU)
Title: Video telecommunication system and method for compressing and decompressing digital color video data
Inventor: MUSIC JOHN
IPC: H04N9/808
Filed: 1989-03-23
Abstract: The method and system of compressing and decompressing digital color video data in a video communication system utilizes a digital color video signal having three video color components, and involves the determination of a predetermined number of the most visually significant combinations of color components in a picture frame, and the encoding of the color components as compressed color codes in a series of run length and compressed color code combinations. Line-to-line differences and movement of edges and segments of the picture frames are determined, and frame-to-frame differences are also encoded to reduce the amount of information to a minimum. Further statistical encoding of at least a portion of the run length and color code combinations is also provided. The digitally compressed color component codes are decoded according to a look up table to form a table of the three digital color components for each run length, and the run lengths and corresponding color components are stored in an array in a buffer memory to represent the scan lines in a video picture frame.
Patent AU-3568400-A (AU)
Title: Cover assembly
Inventor: ELSE ROBERT ARTHUR
IPC: A63C19/12
Filed: 2000-03-30
Abstract: A cover assembly for temporarily covering areas such as an ice rink, to support people or other items thereon. The assembly comprises a number of components (10) which can be engaged with other such components (10) placed adjacent thereto-on the surface to be covered. The components include upper and lower parts (12, 16) with a gap (20) being provided between such parts to provide insulation from the underlying area. Adjacent components (10) are retained together by locking means (22) which are provided on two adjacent sides of each component (10). and are selectively engageable in recesses (32) on adjacent components (10).