baber/WOPTO huggingface dataset:
Patent AU-5700990-A (AU)
Title: Diphenylurea derivatives
Inventor: SEKIYA TETSUO
IPC: A61P3/06
Filed: 1990-06-13
Abstract: Novel diphenylurea derivatives represented by the following formula (I): <CHEM> wherein R1 is an alkyl group of 5 to 18 carbon atoms, each of R2 and R3 is independently an alkyl group of 1 to 5 carbon atoms, an alkoxy group of 1 to 5 carbon atoms or a halogen atom, R4 is hydrogen atom, an alkyl group of 1 to 5 carbon atoms, an alkoxy group of 1 to 5 carbon atoms or a halogen atom, and X is oxygen atom or sulfur atom, are provided. The compounds are potent in reducing the cholesterol level in serum, and useful for treating hyperlipemia and atherosclerosis.
Patent AU-5756298-A (AU)
Title: Attenuated salmonella strain used as a vehicle for oral immunization
Inventor: DARJI AYUB
IPC: C12R1/42
Filed: 1997-12-11
Abstract: The present invention is directed to an attenuated Salmonella comprising a eukaryotic expression vector for delivery of the eukaryotic expression vector to a eukaryotic cell. Delivery may be to eukaryotic cells cultured in vitro or to cells in vivo, such as by oral administration of the attenuated Salmonella comprising the eukaryotic expression vector.
Patent AU-5762994-A (AU)
Title: A filler for a thermoplastic composition
Inventor: HIGGS ROBERT PHILIP
IPC: C09C3/10
Filed: 1994-03-07
Abstract: There is disclosed a thermoplastics composition comprising a thermoplastic polymer having incorporated therein a coated particulate inorganic material. The coating on the particles of the inorganic material comprises a combination of a natural or synthetic polymeric material and a wax having a melting point not higher than the melting point of the thermoplastics polymer, and the polymeric material is present in the coating in an amount of from 1% to 10% by weight, based on the weight of dry inorganic material. The improved thermoplastic composition of the invention may be used in making moulded components for automobiles.
Patent AU-5824586-A (AU)
Title: New process for the production of 7-ACA derivatives
Inventor: PRAGER BERNHARD CHRISTIAN
IPC: C07D501/18
Filed: 1986-06-02
Abstract: The invention provides an improved process for the production of 7-amino-3-alkoxymethylcephem-4-carboxyl acid derivatives.
Patent AU-5829800-A (AU)
Title: Process for making high density and large particle size cobalt hydroxide or cobalt mixed hydroxides and a product made by this process
Inventor: MARTIKAINEN MIKA
IPC: C01G51/00
Filed: 2000-06-28
Abstract: The invention relates to a method for preparing a cobaltous hydroxide with a high density and a large particle size or an alloy hydroxide of cobalt and some other metal, in which a complexing agent and hydroxide ion is added to an aqueous cobalt brine or an aqueous brine of cobalt and some other metal under alkaline conditions in order to form a metal hydroxide. In this method, the complexing agent is selected so as to form an ammonium complex with the metal ion. The molar ratio of complexing agent to metal is about 0.5-3, and the pH is regulated in the range 10-13.
Patent AU-5852996-A (AU)
Title: Serum preparations for inhibiting retroviruses and tumor growth
Inventor: HOWARD MARK E
IPC: A61K39/395
Filed: 1996-05-03
Abstract: Serum and immunoglobulin preparations obtained from sharks are used to prepare compositions, including pharmaceutical compositions, for inhibiting retrovirus replication in susceptible cells. Thus, the serum preparations are useful for inhibiting diseases associated with retroviral infection, such as acquired immunodeficiency syndrome. The serum concentrates and immunoglobulins therefrom are also used to inhibit growth of tumor cells, especially sarcomas and leukemias.
Patent AU-5957998-A (AU)
Title: High melt flow propylene polymer produced by gas-phase polymerization
Inventor: LIN CHI-HUNG
IPC: C08F4/646
Filed: 1998-01-08
Abstract: A process to produce high melt flow propylene polymer comprises polymerizing propylene in the presence of a titanium-containing, magnesium-containing, high activity catalyst and an aluminum alkyl cocatalyst in a gas phase system which uses condensed liquid to control temperature wherein the external catalyst modifier is a tetraalkylorthosilicate, preferably tetraethylorthosilicate, at process conditions of temperature, hydrogen concentration, and Si/Mg, Al/Mg and Al/Si atomic ratios, to produce a high melt flow propylene polymer at high yield.
Patent AU-5994299-A (AU)
Title: Pyridinium derivatives for the management of aging-related and diabetic vascular complications, process for their preparation and therapeutic uses thereof
Inventor: SANKARANARAYANAN ALANGUDI
IPC: A61K31/4436
Filed: 1999-10-15
Abstract: Pyridinium derivatives (I) and their salts are new. Pyridinium derivatives of formula (I) and their salts are new: [Image] R 1R 4R 5 or N(R 7)N(R 7)R 9; R 4N(R 7)R 6O, N(R 7)R 6N(R 7), OR 6O, or OR 6N(R 7); R 6alkyl; R 5alkyl, aryl, heteroaryl, COR 7, SO 2R 7, C(S)NHR 7, C(NH)NHR 7, C(O)R 1 0, C(O)NHR 7, or N(R 7)N=C(R 7)R 1 0; R 7,R 1 0H, alkyl, aryl or heteroaryl (provided that the N of the heteroaryl, when present, of R 1 0 is optionally quarternized with compounds such as X-CH 2C(O)R 3; R 2F, Cl, Br, I, OR 7, NO 2, alkyl, aryl, heteroaryl, formyl, acyl, C(O)NR 7R 1 0, CO 2R 7, NR 7R 1 0, N=C(R 7)R 1 0, SR 7, SO 2NH 2, SO 2-alkyl or SO 2-aryl; m : 0-2; R 3R 7, OR 7, NR 7R 1 0, N=C(R 7)R 1 0, N(R 7)NR 7R 1 0, N(R 7)N=C(R 7)R 1 0 or CH(R 7)C(O)R 8; R 8R 7, OR 7 or NR 7R 1 0; R 9H, alkyl, aryl, heteroaryl, C(O)R 1 0, SO 2R 1 0, C(S)NHR 1 0, C(NH)NHR 1 0, or C(O)NHR 1 0; and X : halide, acetate, perchlorate, sulfate, oxalate, citrate, tosylate, maleate, mesylate, carbonate, sulfite, phosphoric hydrogen, phosphonate, phosphate, BF 4 -> or PF 6 -> (provided that when 2 alkyl groups are present on the same C or N, they may link together to form a cycloalkyl group). Independent claims are also included for: (a) a process for the preparation of (I) comprising preparing the properly substituted pyridine derivative followed by quarternization; (b) the use of (I) in the manufacture of a medicament for diabetic complications and aging-related diseases including kidney disease, nerve damage, retinopathy, artherosclerosis, microangiopathy, endothelial dysfunctions, dermatological conditions, discoloration of teeth and other organ dysfunctions; (c) a method for treating a diabetic patient by breaking preformed advanced glycation end products (AGE) comprising administration of (I) either singly or in combination with another drug. ACTIVITY : Antidiabetic; nephrotropic; neuroprotective; ophthalmological; antiarteriosclerotic; dermatological; dental. Tests were performed to study the efficacy of (I) in the inhibition of advanced glycation end products (AGE) breaker activity. Bovine serum albumin (160 mg/ml) and glucose sugar (1.6 M) were dissolved in phosphate buffered saline. Sodium azide was added at 0.2 % concentration. The solution was filtered and kept for aging at 37 [deg] C for 16 weeks. After 16 weeks the solution was dialyzed against PBS, aliquoted and stored at -20 [deg] C. The AGE breaking activity of N,N'-bis[3-carbonyl-1-(2-phenyl-2-oxoethyl)pyridinium]hydrazine dibromide (Ia) at 5 mM was tested, and found to be 13 %. MECHANISM OF ACTION : None given.
Patent AU-6186299-A (AU)
Title: Formulations and methods for isolating nucleic acids from any complex starting material and subsequent complex genetic analysis
Inventor: HILLEBRAND TIMO
IPC: C12N15/10
Filed: 1999-07-23
Abstract: The subject of the invention are formulations not containing chaotropic components for isolating nucleic acids with binding to a solid phase, in particular of DNA, from optional complex starting materials and quantities containing a lysis/binding buffer system which comprises at least one antichaotropic salt component, a solid phase and wash and elution buffers known as such. The lysis/binding buffer system may be an aqueous solution or a solid formulation in reaction vessels ready for use. All carriers used for isolation by means of chaotropic reagents, preferably glass fiber mats, glass membranes, silica carriers, ceramics, zeolites or materials showing negatively functionalised surfaces or chemically modified surfaces which may be converted to a negative charge potential may serve as a solid phase.Furthermore, the subject of the invention is a method for isolating nucleic acids, in particular DNA, from optional complex starting materials with using the formulations according to the invention which is characterized by the lysis of the starting material, binding of nucleic acids to a carrier, washing of the nucleic acids bound to the carrier and elution of nucleic acids.
Patent AU-6314980-A (AU)
Title: Make ethylidene diacetate from co and hydrogen and methyl acetate or di methyl ether
Inventor: KUBBELER H K
IPC: C07C69/16
Filed: 1980-10-10
Abstract: The invention relates to an improved process for making 1,1-diacetoxyethane by reacting methyl acetate and/or dimethylether with carbon monoxide and hydrogen under practically anhydrous conditions, at temperatures of 350 DEG  to 575 DEG  K., under pressures of 1 to 300 bars, and in the presence of a catalyst system containing noble metals belonging to group VIII of the periodic system of the elements, or compounds thereof, and iodine and/or its compounds. The improved process is effected in the presence of a catalyst system containing, as additional ingredients, an aliphatic carboxylic acid having 1 to 8 carbon atoms, a heterocyclic aromatic compound, in which at least one hetero atom is a quaternary nitrogen atom, and a manganese or rhenium compound.
Patent AU-6375190-A (AU)
Title: Dietary supplement and method of minimizing effects of infection through diet
Inventor: MASCIOLI EDWARD A
IPC: A23L33/00
Filed: 1990-10-03
Abstract: Disclosed is a method of minimizing infection and minimizing the risks of infection in at risk animals and patients. A dietary supplement to accomplish this objective is also disclosed. The method includes the step of administering a diet rich in  omega 3 fatty acids, for example by adding a substantial proportion of fish oils to the diet. The dietary supplement is particularly well suited to patients receiving total parenteral nutrition. A parenteral diet or diet supplement containing a mixture of oils, one rich in  omega 3 fatty acids and the other rich in  omega 6 fatty acids is disclosed.
Patent AU-6427286-A (AU)
Title: Vehicle brakelights activating device
Inventor: ECKSTEIN MORDECHAI
IPC: B60Q/
Filed: 1986-10-22
Abstract: A device is provided, associated with the accelerator pedal of motor cars adapted to cause the lighting of the brake lights shortly before the brake pedal is applied in case of braking in an emergency. In one disclosed version of the device, it comprises a bellows mounted on the accelerator pedal. During normal driving, the bellows is pressed down to minimum volume thereof. When abruptly released, a sub-pressure is developed which is used to momentarily lift a metal flap which closes the brakelights circuit. The lights remain on until the light circuit is taken over by the brake pedal switching circuit. According to another version, the operation is based on the relative abrupt movement of a magnetic core surrounded by an induction coil. The electromotive force will generate a current effective to close the brakelights circuit.
Patent AU-6429300-A (AU)
Title: Mono and multifunctional alkoxyamines for the preparation of functionalized macromers
Inventor: KRAMER ANDREAS DR
IPC: C07F7/18
Filed: 2000-06-26
Abstract: The invention pertains to a compound of formula (I), (II) or (III)wherein R1 and R2 are independently of each other hydrogen, C1-C18alkyl, C3-C18alkenyl, C3-C18alkinyl or phenyl which are unsubstituted or substituted by NO2, halogen, amino, hydroxy, cyano, carboxy, C1-C4alkoxy, C1-C4alkylthio, C1-C4alkylamino or di(C1-C4alkyl)amino; A is a group capable of forming a stable free nitroxyl radical A*, which is bound via its oxygen atom to the carbon atom; Y is O, NR3 or CHR3-Xa, wherein Xa is O, S or NR3; R3 is hydrogen, C1-C18alkyl, C3-C18alkenyl, C3-C18alkinyl or phenyl which are unsubstituted or substituted by NO2, halogen, amino, hydroxy, cyano, carboxy, C1-C4alkoxy, C1-C4alkylthio, C1-C4alkylamino or di(C1-C4alkyl)amino; Q1 is an organic or inorganic radical, derived from a compound having at least one functional group being capable of reacting with a hydroxy group; Q2 is an organic radical derived from a mono or polyfunctional alcohol, mono or polyfunctional aminoalcohol, mono or polyfunctional amine mono or polyfunctional mercaptane, mono or polyfunctional phenol or mono or polyfunctional thiophenol; and n is a number from 1 to 20; with the proviso, that in formula (I) if n is 1, Q1 is notor if n is 2, R1 is H and R2 is -CH2-O-tert-butyl, A is not 2,2,6,6-tetramethylpiperidine or 2,2,6,6-tetramethylpiperidine-4-carboxylic acid. Further subjects of the invention are a composition comprising above compounds and at least one ethylenically unsaturated monomer, process for polymerization and the (co)polymers obtained therefrom.
Patent AU-6444694-A (AU)
Title: Polypeptide bombesin antagonists
Inventor: SCHALLY ANDREW VICTOR
IPC: A61K38/08
Filed: 1994-03-07
Abstract: Pseudopeptides comprising a peptide of formula I: X-A1-A2-Trp-Ala-Val-Gly-His-Leu-psi-A9-Q wherein X is hydrogen, a single bond linking the alpha amino group of A1 to the gamma carboxyl moiety on the 3-priopionyl moiety of A2 when A2 is Glu, or a group of formula R1CO- wherein R1 is selected from the groups consisting of a) hydrogen, C1-10alkyl, phenyl or phenyl-C1-10-alkyl, p-HI-phenyl, p-HI-phenyl-C1-10-alkyl, naphthyl, naphthyl-C1-10-alkyl, indolyl, indolyl-C1-10-alkyl, pyridyl, pyridyl-C1-10-alkyl, thienyl, thienyl-C1-10-alkyl, cyclohexyl or cyclohexyl-C1-10-alkyl, where HI=F, Cl, Br, OH, CH3 or OCH3; b) N(R2)(R3)-, wherein R2 is hydrogen, C1-10alkyl, phenyl or phenyl-C1-10-alkyl, R3 is hydrogen or C1-10alkyl; c) R4O-, wherein R4 is C1-10alkyl, phenyl or phenyl-1-10-alkyl; A1 is a D- or L- amino acid residue selected from the group consisting of Phe, p-HI-Phe, pGlu, Nal, Pal, Tpi, unsubstituted Trp or Trp substituted in the benzene ring by one or more members selected from the group consisting of F, Cl, Br, NH2 or C1-3alkyl; or A1 is a peptide bond linking the acyl moiety of R1CO- to the alpha amino moiety of A2; A2 is Gln, Glu[-], Glu(Y) or His, wherein [-] is a single bond linking the gamma carboxyl group of A2 when A2 is Glu with the alpha amino group of A1 where X is a single bond, Y is -OR5 or -N(R5)(R6) wherein R5 is hydrogen, C1-3 alkyl or phenyl; R6 is hydrogen or C1-3alkyl; and R7 is hydrogen, C1-3alkyl or -NHCONH2; Leu-ypsi- is a reduced form of Leu wherein the C=O moiety of Leu is instead -CH2- such that the bond of this -CH2- moiety with the alpha amino moiety of the adjacent A9 residue is a pseudopeptide bond; A9 is Tac, MTac, or DMTac; and Q is NH2 or OQ1 where Q1 is hydrogen, C1-10alkyl, phenyl or phenyl-C1-10-alkyl; and the pharmaceutically acceptable acids or salts thereof.
Patent AU-6469700-A (AU)
Title: Anti-deflagrating operating actuator
Inventor: MARTINO BERNARDINO DE
IPC: H02K5/136
Filed: 2000-07-27
Abstract: An anti-deflagrating actuator adapted to operate in an explosion risk environment includes an external power source and internal components such as a gear reducer, and one of a motion transmission mechanism and a mechanism for transforming rotary motion into linear motion. The internal components are integrally protected within an external housing having a uniform area of free volume that is formed in a shape that outlines the internal components. The actuator further includes a plurality of outlets for connecting electrical power and other control connections received from external sources. These outlets are positioned on the external housing so that they prevent, among other things, kinking of the wiring, which can impair wiring resistance.
Patent AU-6472996-A (AU)
Title: Apparatus for working floor surfaces
Inventor: BERGSTRAND CLAES-GORAN
IPC: E04F21/24
Filed: 1996-06-07
Abstract: An apparatus for working floor surfaces, for example when laying a floor with a thermosetting plastic surface. The apparatus comprises a handle (10) which is designed as an extension arm which is connected to a tool carrier (18) having at least one working tool (19). They are brought to sweep the floor surface by rotation of the tool carrier around an axis of rotation (17) which is substantially vertical in use. The handle enables movement of the apparatus along the floor surface and is connected to the tool carrier via a pivot shaft (15) which is substantially horizontal in use. The pivot connection (15) of the handle (10) to the tool carrier (18) is located at a distance from the axis (17) of rotation of the tool carrier. A support means (21) for the handle is located at the opposite side of the axis (17) of rotation, relative to the pivot connection of the handle.
Patent AU-6563500-A (AU)
Title: Conduits and conduit elements for transporting flowable media
Inventor: KELLER HERMANN
IPC: F16L9/12
Filed: 2000-07-12
Abstract: The invention relates to conduits (1) which are used to transport flowable media. The inside of the conduit (2) which comes into contact with the flowable medium has a structured surface which enables a turbulent or quasi-turbulent boundary layer to be formed between the wall of the conduit and the main flow of said medium. The specially structured surface which is formed by high (4) and low (3) macroscopic and/or microscopic areas can increase the speed of the transported medium and the capacity to entrain particles which are contained in the transported medium or disposed on the wall of the conduit.
Patent AU-6616690-A (AU)
Title: Interactive audio visual work
Inventor: BILLINGS ZEB
IPC: G09B5/06
Filed: 1990-10-11
Abstract: An audio-visual book includes a plurality of pages and a text portion on the plurality of pages. The text portion includes, on each of at least two of the pages, both a plurality of lines of text and a plurality of different predetermined graphic depictions related in concept to the subject matter of the text and interposed within the lines of text. A switching mechanism is disposed in predetermined relationship to the text portion and includes a plurality of individually actuable elements, each of the switches being associated with one of the graphic depictions. A digital sound generator, responsive to actuation of one of the switches, is provided for selectively effecting generation of a sound associated with the subject of the depiction associated with the one switch.
Patent AU-6860396-A (AU)
Title: Purified coprinus laccases and nucleic acids encoding same
Inventor: YAVER DEBBIE SUE
IPC: C07K14/37
Filed: 1996-08-20
Abstract: The present invention relates to polypeptides having laccase activity and isolated nucleic acid sequences encoding the polypeptides. The invention also relates to nucleic acid constructs, vectors, and host cells comprising the nucleic acid sequences as well as methods for producing the polypeptides.
Patent AU-6878496-A (AU)
Title: Packaging for a drink based on anethole
Inventor: NOBLE PHILIPPE
IPC: A23L2/00
Filed: 1996-08-21
Abstract: The invention relates to a packaging made up of at least one inner, containing an alcoholic or nonalcoholic beverage based on anethole, in which the inner foil of said packaging is made up of a film of polyamide including aromatic units. The packaging is preferably intended to contain weakly alcoholic beverages and the polyamide results from the polycondensation of meta-xylylenediamine with adipic acid.
Patent AU-6879287-A (AU)
Title: Method for the preservation of wood
Inventor: COOKE THEODORE F JR
IPC: B27K3/38
Filed: 1987-02-13
Abstract: A method for the preservation of wood is disclosed : whereby the wood is treated with an aqueous, alkaline solution of an alkylol group containing phenol.
Patent AU-7070098-A (AU)
Title: Resistance marker for monocotyledons
Inventor: FREEMAN JUDY PATRICIA
IPC: C12N15/82
Filed: 1998-04-24
Abstract: The use of sulphonamide resistance genes as selectable markers in wheat is provided.
Patent AU-7115887-A (AU)
Title: 5H-1,3,4-thiadiazolo(3,2-a)pyrimidin-5-one derivatives and agricultural-horticultural fungicide composition containing the same
Inventor: TOKUNAGA YUKIO
IPC: A01N43/90
Filed: 1987-04-07
Abstract: A new class of 5H-1,3,4-thiadiazolo[3,2-a]pyrimidin-5-one derivatives of formula <CHEM> wherein X is hydrogen, halogen, alkyl, alkoxy, phenyl, phenoxy, cyano or nitro group; and Y is hydrogen, halogen, haloalkyl, alkoxy, alkynyl which may be substituted with a phenyl or a cyano, and an agricultural-horticultural fungicidal composition containing said derivative.
Patent AU-7215300-A (AU)
Title: Optical disc and optical disc apparatus
Inventor: SHISHIDO YUKIO
IPC: G11B7/007
Filed: 2000-12-11
Abstract: The present invention facilitates identification of whether or not an optical disc is a optical disc of which recording capacity is enlarged. A synchronization pattern of ATIP information embedded into guide grooves irradiated with a light spot is made to be different between a high density optical disc and a standard density optical disc of which recording capacity is not enlarged. Specifically, while the synchronization pattern of the standard density optical disc is preferably made into "3T+1T+1T+3T" (where "T" represents a minimum channel bit of a signal obtained by reading a positional information), the synchronization pattern of the high density optical disc is preferably made into "3T+3T+1T+1T" for example. By reading the ATIP information and recognizing the synchronization pattern thereof, it can be easily and quickly identified whether the optical disc has a standard density or a high density. <IMAGE>
Patent AU-7385294-A (AU)
Title: High concentrated, solid mepiquat chloride and chlormequat chloride products
Inventor: JAGER KARL-FRIEDRICH
IPC: A01N25/08
Filed: 1994-07-09
Abstract: The present invention provides hygroscopic plant growth regulator formulations in solid forms and associated methods of making the powders and tablets. The most preferred formulation uses an effective amount of an N,N-dimethyl-piperidinium salt.
Patent AU-7590591-A (AU)
Title: Process for the synthesis of N-3(-1H-imidazol-1-yl)phenyl-4-(substituted)-2- pyrimidinamines
Inventor: DEAN WILLIAM DENNIS
IPC: C07D405/14
Filed: 1991-04-24
Abstract: The invention provides a novel process for producing N-[3-(1H-imidazol-1-yl-4-(substituted-2-pyrimidinamine compounds in which the substituent is a 2-pyridinyl, 3-pyrindinyl, 4-pyridinyl, 2-furanyl or 2-thienyl group. The process includes the steps of (1) reacting a 3-(1H-imidazol-1-yl)benzamine with cyanamide and a halogen acid while controlling the pH of the reaction between pH about 2 to about 3.5 and recovering a [3-(1H-imidazol-1-yl)phenyl] guanidine dihydrohalide and (2) reacting the [3-(1H-imidazol-1-yl)phenyl] quanidine dihydrohalide so recovered with an appropriately substituted 3-dimethylamino-1-(substituted)-2-propen-1-one and a base at a pH of from about 10.5 to about 11.5 and recovering the N-[3-(1H-imidazol-1-yl)phenyl-4-(substituted)-2-pyrimidamine compound so produced. The novel process provides improved yield and purity by adhering to the stated crucial pH ranges.
Patent AU-7753298-A (AU)
Title: Bandpass reactive collison cell
Inventor: TANNER SCOTT D
IPC: H01J49/42
Filed: 1998-06-02
Abstract: A method of reducing isobaric interferences by transmitting ions from an ion source through an ion transmission device, typically a quadrupole collision cell, and then into an analyzing mass spectrometer, in which the collision cell is operated with a pass band which rejects intermediate ions which would otherwise tend to react to form isobaric interferences. Preferably ammonia is used as a reaction gas in the collision cell. Depending on the chemistry involved, the collision cell may be operated to set the low mass cutoff at an appropriate level, or more usually, the pass band will have both high and low mass cutoffs determined by applying both RF and DC to the collision cell. The collision cell may also be operated with a pass band to transmit ions into a time-of-flight (TOF) mass spectrometer, thus limiting the mass range of ions entering the TOF and thereby improving the duty cycle of the TOF.