baber/WOPTO huggingface dataset:
Patent BR-PI0924543-B1 (BR)
Title: composição farmacêutica de liberação controlada, e seu processo de preparação
Inventor: GERHARD RENNER
IPC: A61K9/50
Filed: 2009-03-18
Abstract: COMPOSIÇÃO FARMACÊUTICADE LIBERAÇÃO CONTROLADA COM RESISTÊNCIA CONTRA A INFLUÊNCIA DE ETANOL EMPREGANDO UM REVESTIMENTO COMPREENDENDO POLÍMERO VINÍLICOS NEUTROS E EXCIPIENTES. A presente invenção refere-se a uma composição farmacêutica de liberação controlada compreendendo um núcleo, compreendendo um principio farmaceuticamente ativo, onde o núcleo é revestido com uma camada de revestimento que confere resistência ao etanol que tem o efeito de conferir o perfil de liberação do princípio farmaceuticamente ativo para ser resistente contra a influência de etanol, onde a camada de revestimento que confere resistência ao etanol compreende pelo menos 70% em peso de uma mistura de uma porção polimérica a ) e uma porção de excipiente b), o nde a porção polimêrica a) consite em um poliméro vinilico ou copolímero vinilico essencialmente neutro e insóluvel em água e a porção de excipiente b) consite nos excipientes b1 100 a 250% em peso de um lubrificante inerte não poroso, b2) 1 a 35% em peso de um composto celulísico; b3) 0,1 a 25% em peso de um emulsificante e adicionalmente ou como alternativa para b3): b4) 0,1 a 30% em peso de um plastificante onde os excipientes de porção de excipientes b) são cada um deles, calculados com base no peso seco da porção polimérica a).
Patent BR-PI0924660-B1 (BR)
Title: método de paging, método de atualização de localização, enodeb, retransmissora, sistema de comunicação e meio legível por computador não transitório
Inventor: BO LIN
IPC: H04W68/02
Filed: 2009-04-28
Abstract: MÉTODO DE ENVIO DE RADIOCHAMADA, ENODEB, RETRANSMISSORA, SISTEMA DE COMUNICAÇÃO COMPREENDO A RETRANSMISSORA E PRODUTO DE PROGRAMA DE COMPUTADOR. A presente invenção refere-se a um método de envio de radiochamada que pode reduzir o tempo de processamento de sinalização de um envio de radiochamada de sistema e poupar recursos de envio de radiochamada. O método inclui: o recebimento, por um eNodeB, de uma mensagem de envio de radiochamada, em que a mensagem de envio de radiochamada porta uma identidade de área de rastreamento; o envio de radiochamada para um equipamento de usuário se a identidade de área de rastreamento na mensagem de envio de radio chamada for a identidade de área de rastreamento do eNodeB; e a instrução de uma retransmissora para enviar uma radiochamada. Um método de atualização de localização também é descrito, o qual reduz a carga de sinalização produzida pela atualização de localização. O método inclui: a geração, por uma retransmissora, de uma mensagem de sistema, em que a mensagem de sistema inclui uma identidade de área de rastreamento da retransmissora; e a difusão da mensagem de sistema, e o disparo de um equipamento de usuário em uma célula da retransmissora para iniciar uma requisição de (...).
Patent BR-PI1000651-B1 (BR)
Title: dispositivo de freio para uma motocicleta
Inventor: KAZUHIKO TANI
IPC: B60T8/17
Filed: 2010-03-10
Abstract: DISPOSITIVO DE FREIO PARA UMA MOTOCICLETA. A presente invenção refere-se a um dispositivo de freio para uma motocicleta que é capaz de realizar uma operação de frenagem que não cause desconforto mesmo para motocicletas providas com um sistema de freio combinado. Um dispositivo de freio (10) para uma motocicleta é capaz de realizar eletricamente o acionamento de modo a controlar uma pinça de freio de roda dianteira (16) e uma pinça de freio de roda traseira (18) em resposta a cada operação de uma alavanca de freio (12) e um pedal de freio (14) e é configurado de modo que a pinça de freio de roda traseira (18) e a pinça de freio da roda dianteira (16) possam ser combinadas com base na operação do pedal de freio (14). O dispositivo de freio (10) realiza correções de uma pressão hidráulica alvo que atua na pinça de freio de roda dianteira (16) usando uma função pré-ajustada prescrita de tal maneira a dar uma força de frenagem menor do que uma força de frenagem correspondente à uma operação adicional da alavanca de freio (12), quando a alavanca de freio (12) é adicionalmente operada no estado em que o pedal de freio (14) é operado e a pinça de freio da roda dianteira (16) está (...).
Patent BR-PI1004062-B1 (BR)
Title: válvula de coluna de perfuração e método para preparar uma válvula de coluna de perfuração
Inventor: DERRYL SCHROEDER
IPC: E21B21/10
Filed: 2010-10-25
Abstract: VÁLVULA DE COLUNA DE PERFURAÇÃO CONFIGURADA PARA SER AFIXADA A UM REVESTIMENTO PARA CONECTAR A PERFURAÇÃO A UMA SONDA, MÉTODO PARA PREPARAR UMA VÁLVULA DE COLUNA DE PERFURAÇÃO PARA SER CONECTADA A UM REVESTIMENTO PARA CONECTAR UMA PERFURAÇÃO A UMA SONDA, VÁLVULA DE COLUNA DE PERFURAÇÃO CONFIGURADA PARA SER AFIXADA A UM REVESTIMENTO PARA CONECTAR UMA PERFURAÇÃO A UMA SONDA E MÉTODO PARA CONTROLAR UMA VÁLVULA DE COLUNA DE PERFURAÇÃO. Trata-se de um método e uma válvula de coluna de perfuração (70, 160) para fechar um conduto através do qual um fluido de pressão alta flui. A válvula de coluna de perfuração (70, 160) inclui um alojamento alongado (162) que tem uma cavidade interna (79), um elemento de vedação (56) afixado a uma primeira extremidade (74) do alojamento alongado (162), sendo que o elemento de vedação (56) fica disposto dentro da cavidade interna (79) para que um fluxo de liquido (80) através da cavidade interna (79) a partir da primeira extremidade (74) para uma segunda extremidade (76) seja permitido,uma válvula de deslizamento (50) configurada para deslizar para e partir do elemento de vedação (56) para que quando a válvula de deslizamento (50) entrar em contato com o elemento de vedação (56) o fluxo de liquido seja suprimido, um cartucho de propensão (90) configurado para aplicar uma primeira força (...).
Patent BR-PI1105321-B1 (BR)
Title: Dispositivo de segurança intra-cassete de equipamentos bancários
Inventor: NELSON TAVARES DE PINHO
IPC: E05G1/14
Filed: 2011-12-19
Abstract: 'dispositivo de segurança intra-cassete de equipamentos bancários', sendo o dispositivo (1) montado sob a tampa (t) de um cassete (c) que armazenam cédulas (a); o dispositivo (1) compreende um bloco principal (2) dotado com cavidades (3) preenchidas com material pirotécnico (5), o qual pode ser incendiado por um pavio (9) que é ativado por um filamento metálico (11) que é alimentado eletricamente pelo circuito do cassete (c).
Patent EA-002926-B1 (EA)
Title: Aqueous suspensions of submicron 9-hydroxyrisperidone fatty acid esters
Inventor: FRANCOIS MARC KAREL JOSEF
IPC: A61P25/24
Filed: 1998-11-10
Abstract: 1. A pharmaceutical composition suitable as a depot formulation for administration by intramuscular or subcutaneous injection, comprising a dispersion of particles consisting essentially of a therapeutically effective amount of a crystalline 9-hydroxyrisperidone fatty acid ester having the formula   or a salt, or a stereoisomer or a stereoisomeric mixture thereof, wherein R represents a straight C9-C19alkyl radical; having a surfactant adsorbed to the surface thereof in an amount effective in maintaining a specific surface area > 4 m2/g (corresponding to an effective average particle size of less than 2,000 nm) in a pharmaceutically acceptable carrier comprising water. 2. A composition according to Claim 1 wherein R represents a straight C15 (penta-decyl) chain and the active ingredient is 9-hydroxyrisperidone-palmitate ester. 3. A composition according to Claim 1 wherein the composition further comprises a suspending agent, and optionally one or more preservatives, buffers and isotonizing agents. 4. A composition according to Claim 3 wherein the suspending agent is sodium carboxymethyl cellulose and the surfactant is polysorbate 20. 5. A composition according to Claim 4 wherein the preservative is benzyl alcohol and the isotonizing agent is mannitol or a phosphate buffer. 6. A composition according to Claim 1 having a viscosity of less than 75 mPaxs. 7. A composition according to Claim 3 comprising by weight based on the total volume of the composition: (a) from 3 to 20 % (w/v) of the prodrug; (b) from 0.5 to 2 % (w/v) of a wetting agent; (c) one or more buffering agents sufficient to render the composition neutral to very slightly basic (up to pH 8.5); (d) from 0.5 to 2 % (w/v) of a suspending agent; (e) up to 2 % (w/v) preservatives; and (f) water up to 100%. 8. A pharmaceutical composition as claimed in any one of Claims 1 to 7 for use as a medicament in the treatment of psychosis, schizophrenia, schizoaffective disorders, non-schizophrenic psychoses, behavioural disturbances associated with neurodegenerative disorders, e.g. in dementia, behavioural disturbances in mental retardation and autism, Tourette's syndrome, bipolar mania, depression, anxiety. 9. The use of a composition as claimed in any one of Claims 1 to 7 for the preparation of a medicament for treating psychosis, schizophrenia, schizoaffective disorders, non-schizophrenic psychoses, behavioural disturbances associated with neurodegenerative disorders, e.g. in dementia, behavioural disturbances in mental retardation and autism, Tourette's syndrome, bipolar mania, depression, anxiety.
Patent EA-005734-B1 (EA)
Title: Method of treating rheumatoid arthritis
Inventor: BROWNING JEFFREY L
IPC: A61P21/00
Filed: 1996-07-19
Abstract: This invention relates to a methods of treating rheumatoid arthritis in a human by administering an effective amount of a lymphotoxin- beta receptor (LT-beta-R) blocking agent, in particular, soluble LT-beta-R, fused with Fc domain of human Ig.
Patent EA-007817-B1 (EA)
Title: Trailed reaper
Inventor: WALLACE DONALD JAMES STEERLING
IPC: A01D34/03
Filed: 2004-06-17
Abstract: The invention relates to agricultural engineering, in particular to reapers attached to a mechanical power source.Maintaining the right angle between a tractor movement direction and a reaper's load-carrying beam axis during run operation, elimination of bending moment in the carrier frame in operation and transport positions, a quick transfer of the reaper from transport state to operational and vise verse without wheel's rotation, smooth adaptation to relief and elimination of unexpected loads at sudden relief changes is attained in the trailed reaper which comprises a chassis, with the reaper carrier and left and right supporting wheels, an attachment device the chassis and a platform with a cutting apparatus and, according to the invention, is further provided with a turnable wheel mounted on a cantilever arm and protruded forward relative to the cutting apparatus, the supporting wheels are adapted to turn and change wheel leaning angle relative to the vertical axis, wherein the right wheel is adapted to change the angle towards the reaper movement, the chassis is connected with the platform by a rod arranged parallel to the load-carrying beam, and the cantilever arm is connected to the load-carrying beam by a hinge and a spring.
Patent EA-009456-B1 (EA)
Title: PYRIMIDONE DERIVATIVES AS INTERMEDIATES FOR PREPARING GSK3β OR GSK3β AND cdk5/p25 INHIBITORS
Inventor: GALLET THIERRY
IPC: A61P25/34
Filed: 2002-09-19
Abstract: The invention relates to a pyrimidone derivative represented by formula (I)wherein R1 represents a pyrimidine ring optionally substituted by a Ccycloalkyl group, Calkyl group, a Calkoxy group, a benzyl group or a halogen atom; R3 and R4 represents each independently a hydrogen atom, Calkyl group, a hydroxy group, a Calkoxy group or a halogen atom; R5 represents a hydrogen atom, a Calkyl group or a halogen atom; when m equals 0, p equals 1,2 or 3, when m equals 1, p equals 0,1 or 2, when m equals 2, p equals 0 or 1; acceptable as an intermediate for preparing compounds having inhibiting activity towards GSK3 beta 3 or GSK3 beta 3 and cdk5/p25 and useful as an active ingredient for preventive and/or therapeutic treatment of a neurodegenerative disease caused by abnormal activity of GSK3 beta 3 or GSK3 beta 3 and cdk5/p25, such as Alzheimer disease.
Patent EA-009276-B1 (EA)
Title: Configurations and methods for power generation with integrated lng regasification
Inventor: MAK JOHN
IPC: F01K25/08
Filed: 2005-07-14
Abstract: LNG cold is used in a plurality of cycles in a combined power plant to increase power output. Especially preferred plant configurations integrate a combined cycle power plant with a regasification operation in which in a first stage LNG cold provides cooling in an open or closed power cycle. Most preferably, a significant portion of the LNG is vaporized in the first stage. In a second stage LNG cold provides cooling for a heat transfer medium that is used to provide refrigeration for the cooling water to a steam power turbine and for an air intake chiller of a combustion turbine in the power plant.
Patent EA-014197-B1 (EA)
Title: Main section and auxiliary section type dual-countershaft twelve-speed transmission for vehicle
Inventor: YANG LIN
IPC: B60K17/08
Filed: 2006-10-25
Abstract: A main section and auxiliary section type dual-countershaft twelve-speed transmission for vehicle is comprised of a main section and an auxiliary section. The main section includes a first shaft (1), a second shaft (10) and several countershafts (14) provided on both sides of the second shaft (10). There is gear drive provided between the second shaft and the countershaft. There are six gears on the second shaft, each of which is positioned independently. There are three synchronizers (4) on the second shaft. A shifting fork (5) of the synchronizer is connected to the control mechanism and gear lever by a fork shaft (16). A main shaft (20) and a countershaft (22) are provided in the auxiliary section. The gear (29) engages with the gear (28), and the gear (25) engages with the gear (30). A synchronizer (9), the shifting fork (15) and the fork shaft (31) are provided between the gear (25) and the gear (29). The synchronizer is self-locked by the reverse taper teeth. The fork shaft is self-locked by the mechanism composed of a spring (18) and a steel ball (19).
Patent EA-015129-B1 (EA)
Title: Piperidine gpcr agonists
Inventor: FYFE MATTHEW COLIN THOR
IPC: A61P3/04
Filed: 2008-01-04
Abstract: Compounds of formula (I): or pharmaceutically acceptable salts thereof, are GPCR agonists and are useful as for the treatment of obesity and diabetes.
Patent EA-022377-B1 (EA)
Title: Umami active fraction and method to prepare the same
Inventor: DUBBELMAN SANDER
IPC: A23L19/00
Filed: 2008-12-19
Abstract: The present invention relates to a food industry, in particular, to a taste enhancing umami-active fraction of a plant extract which a) is capable of passing ultra filtration membranes having a molecular weight cut off of 250 kDa, b) comprises at least 1, but not less than 50 wt.% of glutamic acid, by dry weight of the fraction, c) is substantially free from lycopene, d) has a w/w ratio of glucose to glutamic acid of less than 7, but more than 0.01, and e) has a w/w ratio of citric acid to glutamic acid of at most 0.7. Preferably, an umami-active fraction is derived from a tomato fraction. Also proposed are embodiments of a method of preparing an umami-active fraction of a plant extract, food products containing said fraction and a method of preparing such food products.
Patent EA-018694-B1 (EA)
Title: Antiaircraft guided missile
Inventor: ZVONOV ALEXANDER ALEXANDROVICH
IPC: F02K9/42
Filed: 2011-01-18
Abstract: An antiaircraft guided missile (AAGM) comprise a missile body 1 incorporating a main propulsive jet 2, fuel source 3 for the get propulsion motor, a warhead 4 for air assault weapon destruction, an autopilot system 5, internal electric power supply 6, and an on-board computer 7 for airborne equipment and the missile flight control. In this case, the main propulsive jet is equipped with a jet nozzle 8 and is connected, through a supply inlet, with the rocket fuel source 3 and, through a combustion products outlet, with the missile jet nozzle. The main propulsive jet 2 is made as a plasma-jet burst-type motor. The plasma-jet motor comprises an electric detonation chamber 11 for fuel combustion which is of a material, transparent or non-transparent for electromagnetic waves. The chamber 11 is equipped with a rocket fuel pre-ionizer 12 and an ionizer 13. A magneto hydrodynamic (MHD) generator installed at the missile jet nozzle 8 serves as the internal electric power supply 6, and the fuel source 3 is made as a tank 9 with compressed air and an impulse gas supply dozer 10 or as a tank 9 with liquefied fuel. AAGM features decreased weight and dimensional characteristics and increased operational range due to reduction of consumed fuel.
Patent EA-019765-B1 (EA)
Title: Live trap for trapping rodents
Inventor: CINK JAMES H
IPC: A01M23/08
Filed: 2009-09-21
Abstract: A live trap is provided for trapping rodents. The live trap includes a housing having an interior space and at least one opening through which rodents enter the interior space of the housing. A first trap mechanism is provided that is positionable in the live trap for trapping rodents within the live trap. A second trap mechanism is provided that is different from the first trap mechanism and positionable in the live trap for trapping rodents within the live trap. The live trap and trap mechanisms are configured for selective releasable securement of each of the respective first and second trap mechanisms in the live trap to permit interchangeable use of the first and second trap mechanisms in the live trap.
Patent EA-024150-B1 (EA)
Title: Notification method for cases where establishing call is impossible, and system for implementing such method in cellular communication networks
Inventor: GUMIROV VITALIY SHAMILOVICH
IPC: H04W4/12
Filed: 2012-03-07
Abstract: The invention is related to methods and systems for providing services to communication network subscribers, in particular, to notification of calling subscribers in cases where it is impossible to establish telephone connection to the called subscriber. In the notification method according to the invention, in case of impossibility to establish the call, a signal message re-addressed from the cellular communication network received over ISUP or SIP protocol, the code of the cause of re-addressing, and telephone numbers of the called and calling subscribers are used; immediately upon receiving the signal message, a signal for release of the telephone connection is formed and sent to the cellular communication network, a notifying message formation algorithm is selected, at least one notifying message is formed with or without participation of the user, and at least one notifying message is transmitted in the form of SMS message, or USSD message, or MMS message, or HTTP protocol packet, or e-mail message. The invented system for notification in case of impossibility to establish a call in cellular communication networks comprises the following components interacting with each other: a central business logic unit that selects a formation algorithm and forms at least one notifying message according to the selected algorithm with or without participation of the user; an accounts control unit that allows saving in the account the user's instructions for formation of a notifying message without participation of the user; an interface unit including a controller interacting with C7 signal network; and a request processing unit that interacts with cellular communication networks and the central business logic unit and is designed so that it receives a signal message and, immediately upon receipt of the signal message, shapes and sends to the cellular communication network a signal for release of the telephone connection. The technical result of the method and system according to the invention is a higher efficiency of utilisation of voice channels and a lower load on signal and voice channels.
Patent EA-022116-B1 (EA)
Title: Pesticidal mixtures containing isoxazoline derivatives and insecticide
Inventor: HOEGGER PATRIK
IPC: A01P9/00
Filed: 2011-02-03
Abstract: The present invention relates to pesticidal mixtures comprising a component A and a component B, wherein the component A is a compound of formula (I)wherein one of Yand Yis S, SO or SOand the other is CH; L is a direct bond or methylene; Aand Aare C-H; Ris hydrogen or methyl; Ris chlorodifluoromethyl or trifluoromethyl; Ris 3,5-dibromophenyl, 3,5-dichlorophenyl, 3,4-dichlorophenyl, or 3,4,5-trichlorophenyl; Ris methyl; Ris hydrogen; or Rand Rtogether form a bridging 1,3-butadiene group; and component B is a compound selected from the group consisting of abamectin, chlorpyrifos, cyantraniliprole, emamectin, lambda-cyhalothrin, pymetrozine, spirotetramat, thiamethoxam, clothianidin, imidacloprid and flonicamid. The present invention also relates to methods of controlling insects, acarines, nematodes or molluscs by applying said mixtures, seeds, treated by said mixtures and to methods of coating seeds with said mixtures.
Patent EA-024699-B1 (EA)
Title: Pharmaceutical immediate release tablet comprising sevelamer carbonate
Inventor: OSINGA NIELS JAAP
IPC: A61K31/785
Filed: 2009-10-22
Abstract: The invention relates to a pharmaceutical immediate release tablet comprising a core comprising 70-85 wt.% of sevelamer carbonate, calculated as an anhydrous compound, and 10-25 wt.% of lactose monohydrate and a water soluble film coat surrounding the core; and also to a process of making such tablet and to the use thereof for the control and/or adjustment of the level of serum phosphorus.
Patent EA-026375-B1 (EA)
Title: Antigen binding proteins specific for serum amyloid p component
Inventor: BHINDER TEJINDER KAUR
IPC: C07K16/18
Filed: 2011-03-01
Abstract: The present invention relates to antigen binding proteins, such as antibodies, which bind to serum amyloid P component (SAP), polynucleotides encoding such antigen binding proteins, pharmaceutical compositions comprising said antigen binding proteins and methods of manufacture. The present invention also concerns the use of such antigen binding proteins in the treatment or prophylaxis of diseases associated with amyloid deposition including systemic amyloidosis, local amyloidosis, Alzheimer's disease, and type 2 diabetes.
Patent EA-023134-B1 (EA)
Title: Assembly formed of at least two wall elements
Inventor: EBERLEIN MARTIN
IPC: B62B3/14
Filed: 2011-09-09
Abstract: The invention relates to an assembly (1) formed of at least two wall elements (2, 6), in which the wall elements (2, 6) comprise vertically and horizontally arranged reinforcing elements (10, 11) and the wall elements (2, 6) are either movably connected to one another or are present separately and can be transposed into a space-saving arrangement within a common region (14), wherein, in this arrangement, and according to a first embodiment, either the vertical reinforcing elements (10) of the wall element (6) are located in at least one interspace (12) which is formed by vertical reinforcing elements (10) of the wall element (2), or wherein, according to a second embodiment, the horizontal reinforcing elements (11) of the wall element (6) are located in at least one interspace (13) which is formed by horizontal reinforcing elements (11) of the wall element (2). The invention is distinguished in that, in the space-saving arrangement and within the common region (14) according to the first embodiment, the horizontally extending reinforcing elements (11) of the at least one wall element (6) are at the same time also completely or partially located in interspaces (13) which are formed on the wall element (2) by horizontal reinforcing elements (11), or in that, according to the second embodiment, the vertically arranged reinforcing elements (10) of the at least one wall element (6) are at the same time also completely or partially located in interspaces (12) which are formed on the wall element (2) by vertical reinforcing elements (10), and in that, in both embodiments, the interspaces (12, 13), when viewed across the thickness thereof, are arranged with an offset.