baber/WOPTO huggingface dataset:
Patent CO-5700719-A2 (CO)
Title: Derivados de alcanos azaespiro como inhibidores de las metaloproteasas
Inventor: WENQING YAO
IPC: C07D401/02
Filed: 2005-10-19
Abstract: 1.- Un compuesto de Fórmula I o II: o un enantiómero, diaestereoisómero, prodroga, solvato, metabolito o sal farmacéuticamente aceptable del mismo, donde:A es CWOH, CWNHOH, CWNHOR5, N(OH)CHO, N(OH)CWR6, SH, SR7 o hidantoinilo;B es (CH2)n, (CH2)nC=W, (CRdRf)nNR8, NR8(CRdRf)n, (CRdRf)nO(CRdRf)r, (CRdRf)nS(CRdRf)r, O(C=W)NR8, O, N, NR8, S(O)m, S, C(O)NR8(CRdRf)n, C(O)(CRdRf)n o combinaciones de los mismos;G es (CH2)n, (CH2)nC=W, (CRdRf)nNR8, NR8(CRdRf)n, (CRdRf)nO(CRdRf)r, (CRdRf)nS(CRdRf)r, O(C=W)NR8, O, N, NR8, S(O)m, S, C(O)NR8(CRdRf)n, C(O)(CRdRf)n, o combinaciones de los mismos;D es oxígeno o azufre;X está ausente o es (CH2)j, alquileno C1-10 sustituido con 0 a 3 Ra, alquenileno C2-10 sustituido con 0 a 2 Ra, N, O, NRb, S(O)m, C=O, NRbC(O), NRbC(O)O, NRbC(O)NRb, C(O)O, OC(O), S(O)mNRb, NRbS(O)m, NRbS(O)mNRb, (CRdRf)jNRb, NRb(CRdRf)j o combinaciones de los mismos;Y está ausente o es (CH2)j, alquileno C1-10 sustituido con 0 a 3 Ra, alquenileno C2-10 sustituido, con 0 a 2 Ra, N, O, NRb, S(O)m, C=O, NRbC(O), NRbC(O)O, NRbC(O)NRb, C(O)O, OC(O), S(O)mNRb, NRbS(O)m, NRbS(O)mNRb, (CRdRf)jNRb, NRb(CRdRf)j o combinaciones de los mismos;M es CO o S(O)¡;U está ausente o es alquileno C1-10 sustituido con 0 a 5 Ra, alquenileno C2-10 sustituido con 0 a 2 Ra, N, O, NRb, NRbC(O), NRbC(O)O, NRbC(O)NRb, NRbS(O)m, NRbS(O)NRb o combinaciones de los mismos;V está ausente o es H, carbociclilo C3-13 sustituido con 0-5 Re o heterociclilo sustituido con 0-5 Re;U' está ausente o es alquileno C1-10 sustituido con 0 a 5 Ra, alquenileno C2-10 sustituido con 0 a 2 Ra, N, O, NRbS(O)m, C=O, NRbC(O), NRbC(O)O, NRbC(O)NRb, C(O)O, OC(O), S(O)mNRb, NRbS(O)m, NRbS(O)NRb o combinaciones de los mismos; ...
Patent CO-6270325-A2 (CO)
Title: Formas solidas de (s)-etil-2-amino-3-(4-(2-amino-6((r)-1-(4-cloro-2-(3-metil-1h-pirazol-1-yl)fenil)-2,2,2,2-trifluoroetoxi)-pirimidina-4-il)fenil)propanoato y metodos de uso
Inventor: BEDNARZ MARK STEPHEN
IPC: C07D403/12
Filed: 2010-04-28
Abstract: Formas solidas de (S)-etil-2-amino-3-(4-(2-amino-6-((R)-1-(4-cloro-2-(3-metil-1H-pirazol-1-il)fenil) -2,2,2-trifluoroetoxi) pirimidin-4-il) fenil) propanoato y sus sales son descubiertas por esta aplicacion de patente. 1.- (S)-etil-2-amino-3-(4 -(2-amino-6-((R) -1- (4-cloro-2-)3-metil-1H-pirazol-1-il) fenil) -2,2,2-trifluoroetoxi) pirimidin-4-il)fenil) propanoato cristalino o una sal farmacéuticamente aceptable del mismo.2.- Un compuesto, que (S)-etil-2-amino-3-(4-(2-amino-6-((R) -1- (4-cloro-2-(3-metil-1H-pirazol-1-iI)fenil) -2,2,2- trifluoroetoxi) pirimidin-4-il) fenil) propanoato cristalino.3.- El compuesto de la reivindicacion 2, que tiene un punto de fusion de 104°C.4.- El compuesto de la reivindicacion 2, que tiene una patron de difraccion de rayos X en polvo, con picos en uno o mas de cerca de 10,7, 12,2, 12,8, 17,7 y/o 22,0 grados 2?. 5.- El compuesto de la reivindicacion 2, que tiene un patron de difraccion de rayos X en polvo que es sustancialmente la misma que la que se muestra en la Figura 1.6.- Una sal cristalina de (S)-etil 2-amino-3-(4-(2-amino-6-((R)-1-(4-cloro-2-(3-metil-1H-pirazol-1-il) fenil) -2,2,2-trifluoroetoxi) pirimidin-4-il) fenil) propanoato.7.- La sal cristalina de la reivindicacion 6, la cual es una sal de hipurato. 8.- La sal cristalina de la reivindicacion 7, la cual tiene un punto de fusion de 145°C.9.- La sal cristalina de la reivindicacion 7, que tiene una patron de difraccion de rayos X en polvo integrado por picos en uno o mas de alrededor de 8,2, 9,5, 12,6, 16,9, 21,8, 22,0, 22,7, 24,3 o 29,1 grados 2?.
Patent CO-6491086-A2 (CO)
Title: Compuesto alimenticion de grasa vegetal, proceso de preparacion del compuesto alimenticion de rasa vegetal y uso del compuesto alimenticio de grasa vegetal en la preparacion de rellenos
Inventor: GRIMALDI RENATO
IPC: A23D7/00
Filed: 2012-01-26
Abstract: Esta invención se refiere a un compuesto alimenticio de grasa vegetal, que incluye i) una base interesterificada formada de aceite de semilla de algodón liquido en una mayor proporción y aceite de semilla de algodón completamente hidrogenado; ii) aceite de palma completamente hidrogenado, y iii) un antioxidante, tal compuesto contiene un límite máximo de 2% de ácidos grasos trans y un contenido de ácidos grasos saturados inferior a 48% en peso en relación con el peso total del compuesto. Esta invención también se refiere a un proceso de preparación de un compuesto alimenticio graso que contiene un máximo de 2% de ácidos grasos trans, que comprende las fases de hidrogenación completa del aceite vegetal, interesterificación de aceite hidrogenado, y desodorización del aceite. La invención también incluye el uso de la composición alimenticia de grasa vegetal de la invención en la preparación de un relleno para aplicaciones alimenticias.
Patent CO-7230338-A2 (CO)
Title: Pilar protésico definitivo adaptable y respectivo método de dobla
Inventor: MITTELSTÄDT FRIEDRICH GEORG
IPC: A61C13/12
Filed: 2014-12-23
Abstract: La presente invención se refiere a un pilar protésico definitivo adaptable yrespectivo método de dobla, perteneciente al campo de la implantodoncia dental,siendo que dicho método se define especialmente por un proceso de doblapersonalizado, que le auxilia al cirujano dentista y/o técnico en prótesis dental, aorientar la parte aérea del pilar hacia una inclinación favorable a la instalación de lafutura corona protésica. Particularmente y de forma constructiva , un modelo de pilarprotésico definitivo, está formado por un segmento de apoyo y anclaje (1), seguidode una región de conexión (2) a un implante, comprendiendo una zona de sacrificio yanclaje (3), seguida de una región de estrechamiento (4) en el tercio inferior paraadaptación angular; y con origen en esta; una porción de asentamiento y fijación (5)de una prótesis (no ilustrada). De forma específica, la operación de dobla de un pilarprotésico definitivo, consiste de un método que armoniza un dispositivo angulador(D); un pilar de referencia (R) de material plástico de fácil maleabilidad, y degeometría similar a un pilar protésico definitivo; y un tapón protector (31 o 32) queserá acoplado a la porción de asentamiento y fljación(5) de la prótesis (no ilustrado)de un pilar definitivo.
Patent EP-1072472-A2 (EP)
Inventor: FABBRI CORSARINI LUCIANO
IPC: B60R9/12
Filed: 2000-01-07
Abstract: A ski-rack applicable to motor vehicles, fixed structures and the like,
comprising a bracket-like element (1) which can be fixed to a supporting
structure (3) and supports, on one arm thereof (5), at least one locking
element (12) which is mounted so that it can oscillate in order to engage at
least one ski arranged between the arms (5) of the bracket-like element (1).
Patent EP-1048448-A2 (EP)
Title: Hydromechanischer Pressenantrieb
Inventor: HARSCH ERICH
IPC: B30B1/16
Filed: 2000-03-09
Abstract: Die Erfindung betrifft ein hydromechanisches Antriebssystem
für mindestens einen Pressenstößel (3) einer Schneid- und/oder
Umformpresse, wobei mindestens ein Antriebszylinder (4) mit einer
nachfolgenden kinematischen Kette (9,10,12) verbunden ist. Diese
kinematische Kette (9,10,12) ist so gestaltet, daß bei einem einfachen
Kolbenhub in nur eine Richtung ein kompletter Stößelhub, d.h.
eine abwärts- und aufwärtsgerichtete Bewegung erfolgt. Das
vorgeschlagene Antriebssystem ist zusätzlich mechanisch
zwangssynchronisiert.
Patent EP-1039496-A2 (EP)
Inventor: KYRTSOS CHRISTOS
IPC: H01H35/14
Filed: 2000-03-22
Abstract: A vibration sensor includes a housing having an opening, and a movable
trigger retained within the housing by a resilient member. The moveable trigger
includes a projection of a dimension to fit at least partially through the opening. The
resilient member retains the movable trigger within the housing until overcome by a
predetermined acceleration. Whereas the moveable trigger is maintained within the
housing the vibration sensor is minimally affected by radial acceleration while
providing a calibrated resistance which must be overcome by an acceleration of
predetermined severity along the measured direction. When the sensor experiences a
predetermined acceleration, the trigger slides within the housing until the projection
encounters the opening. The projection then "pops" through the opening such that the
projection encounters a switch which awakes and activates a transmitter to send a
signal to a warning device.
Patent EP-1036633-A2 (EP)
Inventor: HAGIWARA KOICHI
IPC: B24C5/04
Filed: 2000-03-16
Abstract: A water pump (2) is connected to a mixer (4) so as to blast high
pressure water at a high speed in the mixer (4). The air and powder
are supplied to the blast flow of the high pressure water through
an air supply pipe (9) and a powder supply pipe (14) respectively so that
a mixture flow composed of the gas, the droplet-like fluid, and
powder is formed. The mixture flow is blasted from a nozzle (15)
at a high speed so as to be sprayed onto a surface to be treated.
Thus, impact actions held by the powder and the droplet-like
fluid as cleansing/scraping media are given to the surface to
be treated. Thus, a cleansing/scraping operation is achieved.
Then, if the fluid, gas or the like supplied to the mixer (4) is
heated, the cleansing/scraping operation can be further
accelerated.
Patent EP-1054289-A2 (EP)
Inventor: SCHWAB ARMIN DR-ING
IPC: E06B9/24
Filed: 2000-05-15
Abstract: A preset mounting arrangement has one or more backing layers (2) for transmitting light. Two or more layers (3,4) consist of material with variable transmission properties for visible light and/or heat radiation. The layers are stretched flat and set at distance apart, each having strips (3',3,4',4) parallel to each other made from a material with variable transmission properties
Patent EP-1063385-A2 (EP)
Inventor: WEICKER MARIO
IPC: E06B9/17
Filed: 2000-06-21
Abstract: A hollow chamber (10) open on the outside along the length of the end-rod contains a holder (6,20) on which is fixed the edge part of the curtain inserted into the hollow chamber. The position of the holder in relation to the end rod is adjusted by a positioning piece (30). The holder has protuberances (22) fitting into matching holes on the edge of the curtain.
Patent EP-1044838-A2 (EP)
Inventor: FARLAND DAVID MARC DIPL-ING
IPC: E05B51/02
Filed: 1998-06-16
Abstract: The locking device has a first connecting unit for fixing of the top (9) on the vehicle and at least one second connecting u (5) at a distance away from the first. The second connecting unit has a spigot-form component (7) fitted to the top, and a guide component (17) to accommodate the spigot. The second locking unit has a locking component (21) for occasional locking of the spi in the guide component and is connected to the locking mechanism in such a way that with fixing of the first locking mechanism i its locking position the locking of the spigot takes place simultaneously.
Patent EP-1102028-A2 (EP)
Inventor: LEUPOLZ ANDREAS
IPC: F41H3/00
Filed: 2000-08-26
Abstract: An infra-red camouflage system comprises a thermorefractive layer system or a thermorefractive material. The material has a negative temp coefft.
Patent EP-1069756-A2 (EP)
Inventor: NO YOUNG
IPC: H04N5/765
Filed: 2000-07-03
Abstract: A method of operating an electronic imaging system (20) as a
distributed processor network is provided for a system that includes multiple
imaging components such as digital cameras (22), printers (34), etc., wherein each
component is connected to an intelligence module (24-36) having a
microcontroller (58) and memory (62). In the method, the intelligence modules
(24-36) are interconnected by way of a data interface (28-37) to form a system
network. Next, different image processing steps are assigned to different ones of
the intelligence modules (24-36). Image data entered and stored within the
imaging system (20) is divided into a plurality of data groups, each of which
preferably corresponds to a portion of an image. Finally, the data groups are
serially entered through each of the intelligence modules (24-36) such that a
specific sequence of image processing steps are conducted on each data group
until the processing of a specific image is completed. The method efficiently
utilizes all the microcontroller capability present in the network intelligence
modules (24-36), thereby minimizing the processing time required to render
images.
Patent EP-1028256-A2 (EP)
Inventor: YU DEQUAN
IPC: F04D5/00
Filed: 2000-01-17
Abstract: A fuel pump has a motor (14) with a shaft (18)
extending therefrom and an impeller (20) fitted thereon for
pumping fuel from a fuel tank to an internal combustion
engine. A pumping chamber (36), which encases the impeller
(20), is comprised of a cover channel (38) and a bottom
channel (40) formed in a pump cover (24) and a pump bottom
(22), respectively. The impeller (20) has a plurality of
radially extending vanes (50) on an outer circumference
separated by partitions (56) of shorter radial length. The
partitions are comprised of substantially quarter-circle
shaped arcuate portions (60) extending from the outer
circumference of the impeller (20) to a diverging portion,
preferably to a substantially flat top (66) with rounded
corners (67). Fluid active vane grooves thus formed
circumferentially between the vanes (50) and axially between
the partitions (60) which reduce fuel vortices angular
acceleration within the pumping chamber (36) thus increasing
pump efficiency.
Patent EP-1064892-A2 (EP)
Inventor: TAKAI HISASHI
IPC: B32B27/00
Filed: 2000-06-22
Abstract: A flexible sheet 1 includes a plastic sheet 2 and a fibrous
assembly 3 bonded to the lower surface of the sheet 2. The sheet
2 is formed with projections 20, ribbon-shaped regions 8, fine
slits 9 defined between each pair of adjacent ribbon-shaped
regions 8, 8, bridge-like regions 10, 10A, 10B connecting each
pair of adjacent ribbon-shaped regions 8 and rising regions 12,
12A, 12B extending upward from edges of the ribbon-shaped
regions 8. The fibrous assembly 3 are partially exposed within
the respective fine slits 9.
Patent EP-1065583-A2 (EP)
Inventor: MUSTAFA MAZIN
IPC: G06F3/023
Filed: 2000-07-03
Abstract: A computer system includes a status register tor receiving events which cause the
computer system to change to a low power mode or back to a normal power mode. The
status register is selectively coupled to a keyboard controller to receive an interrupt from
the keyboard controller when a sleep/wake key is actuated on a keyboard. When the
computer system is normally powered, the keyboard interrupt is not routed to the status
register. If the computer system is powered down, the keyboard interrupt is routed so that
actuation of the sleep/wake key will awake the computer system.
Patent EP-1077547-A2 (EP)
Inventor: NEWELL JASON
IPC: H04H60/27
Filed: 2000-08-08
Abstract: The invention provides a television system including a broadcast
data receiver. The broadcast data receiver includes a data storage
means into which can be sent viewer selected portions of data which
are received, having been broadcast from a remote location. In one
embodiment the data which is broadcast and received is in addition
to the video and/or audio data broadcast to allow scheduled
programmes to be generated and it is from this additional data that
the viewer can select to store portions of the same which relates to
specified subject matter or themes. The portions of data can then be
subsequently selected for display via display screens and/or
speakers such as those of a television set.
Patent EP-1083175-A2 (EP)
Inventor: KONOSU TOSHIYUKI
IPC: A61P31/00
Filed: 2000-09-08
Abstract: Compounds of the following formula (I) and pharmaceutically acceptable salts
and ester derivatives thereof:
 
wherein Ar is a phenyl group which may optionally be substituted by from 1 to 3
substituents selected from the group consisting of halogen atoms and trifluoromethyl
groups have excellent antifungal activity.
Patent EP-1111498-A2 (EP)
Inventor: MATSUSHIMA JUN
IPC: G06F13/38
Filed: 2000-12-01
Abstract: Connected to a CD-RW drive (30) having an IDE apparatus interface
(31), a speech apparatus output terminal (32), and a power supply apparatus
input terminal (33), a converting unit (20) has an IDE unit interface (21), a
speech unit input terminal (22), a power supply unit output terminal (23), a USB
unit interface (24), a speech unit output terminal (25), and a power supply unit
input terminal (26). The converting unit (20) comprises an IDE/USB converting
circuit (27) connected between the IDE unit interface (21) and the USB unit
interface (24). The IDE/USB converting circuit (27) carries out an interface
conversion between an IDE interface and a USB interface. The converting unit
(20) further comprises a noise filter (28) connected between the power supply
unit input terminal (26) and the power supply unit output terminal (23). The
speech unit input terminal (22) is directly connected to the speech unit output
terminal (25).
Patent EP-1072884-A2 (EP)
Inventor: KELLY WILLIAM M
IPC: G01N21/88
Filed: 2000-07-28
Abstract: An illuminator (1) has a printed circuit board (5) supporting a ring of light emitting
diodes (LEDs) (6). An annular Fresnel lens (7) and the board (5) are both mounted
in a housing (2) having a central through-hole (3) for a camera field of view. The
lens (7) mixes light from the LEDs (6) in the tangential direction and it also controls
spread in the radial direction so there is uniform illumination over a target plane (4).
Any individual point on the target plane (4) receives illumination from over 25% of
the light sources (6). The illuminator is thus particularly effective, compact, and
suitable for a wide range of industrial applications. Choice of lens and of the spatial
arrangement allows versatility. The illuminator design is easily scaleable by
changing the size and spacing between the light sources.
Patent EP-1061103-A2 (EP)
Inventor: KAUL BANSI LAL
IPC: C09D11/00
Filed: 2000-06-16
Abstract: Compounds of the formula:
 
where R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , R 7 , R 8 , R' 5 , R' 6 , R' 7 , R' 8  are hydrogen, halogen, hydroxy, -NO 2 ,
-CN, -CF 3 , -CONH 2 , C 1-12 alkyl, phenyl, naphthyl, phenanthryl, anthryl, R 9 R 10 N-, R 9 -O- or
R 9 -S-, -CONHR 10 , -CONR 9 R 10  in which R 9  and R 10  are C 1 -C 6 -alkyl, C 6 -C 10 -aryl, (C 6 -C 10 )-aryl-(C 1 -C 6 )-alkyl
or (C 1 -C 6 )-alkyl-(C 6 -C 10 )-aryl, in which the alkyl and/or aryl radicals can
optionally be substituted by hydroxyl, C 1 -C 6 -alkoxy, C 6 -C 10 -aryloxy or halogen; and optionally
two adjacent groups can form an isocyclic or heterocyclic group; 
are eminently suitable for the mass coloring of polymers, in particular polar polymers, for
coloring toners, powders and powder coating materials as well as for coloring ink-jet inks.
Patent EP-1165604-A2 (EP)
Inventor: ST GEORGE-HYSLOP PETER H
IPC: C12Q1/68
Filed: 2000-02-11
Abstract: L'invention concerne un procédé de stimulation de la croissance nerveuse, notamment de régénération nerveuse, consistant à mettre en contact des cellules nerveuses avec la protéine humaine neuronale Armadillo (hNPRAP), apparentée à la Plakophiline. Dans un mode de réalisation spécifique, la protéine hNPRAP provoque le développement de nombreuses extensions cellulaires, longiformes, similaires à un bourgeonnement axonal observé lors de la régénération neuronale et de la formation de synapses. L'invention concerne encore des compositions pharmaceutiques comprenant la protéine hNPRAP, ou bien un vecteur de thérapie génique exprimant la protéine hNPRAP, de même que des procédés d'identification de substances modulant l'expression de la protéine hNPRAP.
Patent EP-1177081-A2 (EP)
Inventor: NAAMANKA JANNE SAMULI
IPC: B28B7/38
Filed: 2000-02-17
Abstract: A method for creating a patterned concrete surface with the aid of a concrete surface retarding agent. According to the invention, printing technique or an output technique is used to transfer the surface retarding agent forming the desired pattern to the surface coming into direct contact with the concrete to be cast. The printing or output technique can also be used to transfer a release agent or other substance affecting the surface of the concrete to the surface coming into contact with the concrete to be cast, in the same or in a separate transfer stage.
Patent EP-1075638-A2 (EP)
Inventor: MOSSBERG JONATHAN E
IPC: F41A17/06
Filed: 2000-01-20
Abstract: A firearm safety enhancement system is provided for enabling use of a firearm only by an authorized individual. At least one electrically activated preventer is provided having a first position for preventing use of firearm and having a second position for enabling use of the firearm. An electrical activation circuit is operatively connected to the preventer to move the preventer between the first and second positions. A portable power supply is carried in said firearm and is coupled to the activation circuit for providing power. A power signal transmitter is operatively connected to the power supply for transmitting an electromagnetic power signal at a regular frequency. A passive identification tag is mounted to a personal adornment to be carried or worn by an individual and is preprogrammed with an authorized identification code preselected from a large number of available identification codes. The passive identification tag is responsive to the power signal to impose a coded return signal on the power signal. The return coded signal is representative of the preprogrammed authorized identification code so that the power signal acts as a carrier of the imposed coded return signal. A reader circuit is connected to the power signal transmitter and to the electrical activation circuit. The reader circuit is responsive only to an authorized identification code to activate the electrical activation circuit to provide power from the portable power supply to move the at least one preventer between the first preventing position and the second unblocked position for enabling use of the firearm.
Patent EP-1196440-A2 (EP)
Inventor: LITTLE ROGER G
IPC: A61P19/02
Filed: 2000-06-23
Abstract: The present invention relates generally to small peptide-based constructs, including derivatized constructs, and their therapeutic uses. The sequences of these constructs are based on a reverse subsequence derived from Domain II of bactericidal/permeability-increasing protein (BPI).
Patent EP-1208373-A2 (EP)
Inventor: VOLKE FRANK
IPC: G01N29/28
Filed: 2000-08-22
Abstract: A coupling medium of a thin layer of a homogenized mixture of at least one polysaccharide or disaccharide such as trehalose; a surface-active substance such as sodium dioctylsulfosuccinate; and water acts as a coupling medium for transverse ultrasonic waves, when the homogenized mixture is applied to surfaces of a transmitting, respectively receiving, transducer for transverse ultrasonic waves; and a surface of a probe.
Patent EP-1230604-A2 (EP)
Title: Robustness and notifications in travel planning system
Inventor: GALPERIN GREGORY R
IPC: G06Q10/00
Filed: 2000-11-01
Abstract: A method includes determining a travel itinerary that includes a first segment that is scheduled to arrive at a location at an arrival time and a second segment that is scheduled to depart from the location at a departure time. The method also includes deriving a probability distribution of delays in the arrival time based on an arrival statistical model of the first segment, retrieving  a minimum connection time required by a traveler traveling in the first segment to connect to the second segment, and computing a likelihood that the traveler will fail to connect to the second segment based on the probability distribution of delays in the arrival time. Annotations are derived from the computed likelihood and added to the travel itinerary.