baber/WOPTO huggingface dataset:
Patent IL-148482-A (IL)
Title: Methods of preparing substituted tetracyclines with transition metal-based chemistries, some such novel compounds and use thereof in the preparation of medicaments
IPC: A61K31/65
Filed: 2002-03-04
Abstract: The present invention relates to novel chemistries which allow for heretofore unobtainable substituted tetracycline compounds which exhibit significant antibacterial activity. The methods disclosed herein utilize reactive tetracycline-based precursor compounds, reactive organic substituent precursors and transition metal catalysts under conditions such that a tetracycline compound substituted with the desired organic substituent is formed. In one embodiment of the invention, a substituted tetracycline compound may be prepared by combining a reactive tetracycline-based precursor compound such as an arene tetracycline diazonium salt, and a reactive organic substituent precursor, e.g., alkenes, substituted alkenes, vinyl monomers, aromatics and heteroaromatics, in the presence of a transition metal catalyst, such as palladium chloride, under conditions such that a tetracycline compound substituted with the organic substituent is formed. Such compounds may optionally act as intermediates for making other compounds, e.g., hydrogenation of unsaturated groups on the substituent.
Patent IL-148947-A (IL)
Title: Batch sludge dehydrator
IPC: F26B/
Filed: 1999-10-05
Abstract: A dehydrating apparatus (10) includes a chamber (12) for receiving wet material to be dehydrated. A rotatably-mounted agitator (26) is provided with the chamber (12). The agitator (26) is adapted to agitate material in the chamber when the agitator rotates in a first direction (28) and convey the material out of the chamber when the agitator rotates in the other, second direction (30).
Patent IL-173441-A (IL)
Title: Injectable composition for the extended release of aripiprazole and use of a mixture of aripiprazole in an injection vehicle
IPC: A61K47/38
Filed: 2006-01-30
Abstract: The present invention relates, in part, to the discovery that a pharmaceutical composition comprising aripiprazole and a carrier administered in a bolus injection resulted in an extended release profile similar to that obtained by the injection of a polylactide-co-glycolide microsphere formulation containing the active agent. This surprising result provides pharmacologically beneficial extended release formulations without the complexities and expense associated with the manufacture of microspheres.
Patent IL-189290-A (IL)
Title: Argatroban formulation
Filed: 2008-02-05
Abstract: An aqueous, stable, sterile pharmaceutical composition of the thrombin inhibitor argatroban in a solution containing an acid to solubilize the argatroban, substantially free from dehydrated alcohol is described, as well as a method for its preparation.
Patent IL-193170-A (IL)
Title: Chimeric flavivirus vaccines
IPC: C12N/
Filed: 2008-07-31
Abstract: A chimeric live, infectious, attenuated virus, containing a yellow fever virus, in which the nucleotide sequence for a prM-E protein is either deleted, truncated, or mutated, so that functional prM-E protein is not expressed, and integrated into the genome of the yellow fever virus, a nucleotide sequence encoding a prM-E protein of a second, different flavivirus, so that the prM-E protein of the second flavivirus is expressed.
Patent IL-195808-A (IL)
Title: Genes encoding flavone synthase proteins
IPC: C12N9/02
Filed: 2008-12-09
Abstract: DNA obtained, for example, from snapdragon or torenia, encoding an enzyme that can convert flavanones directly to flavones, and its uses; the DNA and amino acid sequences for enzymes encoded thereby are listed as SEQ.ID. No. 1 & 2 and 3 & 4, for example. Introduction of the genes into plants can, for example, alter the flower colors of the plants.
Patent IL-206114-A (IL)
Title: Orally adminstered peptides to ameliorate atherosclerosis
IPC: A61P37/02
Filed: 2010-05-31
Abstract: This invention provides novel peptides that ameliorate one or more symptoms of atherosclerosis (see Figure 23). The peptides comprise at least one class A amphipathic helix and at least one D amino acid The peptides are highly stable and readily administered via an oral route.
Patent JP-H0646119-A (JP)
Title: Recall dial number storage system for telephone set
Inventor: KISHIMOTO KAZUNORI
IPC: H04M1/27
Filed: 1992-04-21
Abstract: PURPOSE:To effectively utilize a memory by preventing the same dial number from being superposed in an area storing the dial number of a dial number memory part. CONSTITUTION:A memory control part 3 receives a transmission dial number from a dial button dipressing part 1, temporarily stores it, investigates the storage areas (1) to (3) of the dial number memory part 2 and investigates the presence/absence of the storage of the same number first. When the same number is present thereon, the same number in the storage areas (1) to (3) is erased, the remaining numbers are moved to the storage area of the old number and the number being temporarily-stored is moved to the stoage area of the young number so as to be stored. A memory calling part 4 temporarily stores the dial number received from the memory control part 3 to store it in a display part 5 and, on the other hand, sends the storing dial number to an automatic transmission part 6 at the time of being driven by the automatic transmission part 6, which automatically transmits the dial number received by requiring to the memory calling part 4 to a communication channel.
Patent JP-2000293922-A (JP)
Title: Autochanger type magnetic recording/reproducing device for digital data storage(dds) cartridge
Inventor: WATABE KOJI
IPC: G11B17/26
Filed: 1999-04-07
Abstract: PROBLEM TO BE SOLVED: To provide an autochanger type magnetic recording/reproducing device for a DDS cartridge, capable of preventing the damaging of the DDS and a drive by cutting off the incursion of dust into a casing provided in the autochanger type magnetic recording/reproducing device for the digital data storage(DDS) cartridge, preventing recording/reproducing errors, and reducing a temperature increase in the casing. SOLUTION: This device D is provided with a DDS cartridge 12, a DDS drive 1, a magazine 8, an autochanger mechanism 2 for selecting one DDS cartridge 12 from the magazine 8, and a control circuit board 10 having a control circuit for controlling the autochanger mechanism 2. At least the autochanger mechanism 2 is housed in a casing 20 having a top cover 3, a bottom cover 4, a bezel 5 and cutoff elastic members 7 provided at respective intervals, and the control circuit board 10 is provided outside the casing 20.
Patent JP-S5625708-A (JP)
Title: Connecting method for optical fiber
Inventor: GOTOU AKIYA
IPC: G02B6/24
Filed: 1979-08-08
Abstract: PURPOSE:To perform adhesion easily and efficiently by inserting 2 optical fibers to be connected, from both the ends of a pipe whose inside diameter is a little larger than the outside diameter of the former, placing an ultraviolet ray hardening adhesive agent which has been inserted beforehand, between them, pressing them, and hardening the adhesive by transmitting ultraviolet rays from the other end. CONSTITUTION:A quartz fiber 2 of the outside diameter which is a little thinner than the inside diameter of a pipe is inserted from both the sides of a stainless steel pipe or a synthetic resin pipe 1 whose hardness is large. An ultraviolet ray hardening adhesive is inserted beforehand in the center of the pipe 1. The adhesive is applied between the two fibers, they are pressed, and they are hardened by transmitting ultraviolet rays or N2 laser rays and applying them to the adhesive part. In this case, a remaining adhesive in case the quartz fibers 2 have been press-contacted is made to overflow from the discharge port 3. In this regard, loss of rays is decreased by using synthetic resin or glass for the pipe 1, and making its refractive index smaller than the refractive index of the adhesive. In this way, the adhering work can be performed easily and efficiently.
Patent JP-H0684452-A (JP)
Title: Thermoelectric field emission cathode
Inventor: IDE MASARU
IPC: H01J1/30
Filed: 1992-03-27
Abstract: PURPOSE:To provide a thermoelectric field cathode which can be started to operate with a practical, efficient schedule without causing a discharge phenomenon by providing a cover layer of Zr and O over the surface of a specific W single crystal acicular electrode, and limiting the size of the tip of the electrode. CONSTITUTION:In a thermoelectric field emission cathode comprising an acicular electrode 1 of tungsten single crystal of <100> orientation, having a cover layer of zirconium and oxygen provided on the surface thereof, and a suppressor electrode 2, the tip of the acicular electrode 1 is projected from the outer surface of the suppressor electrode 2 by 0.15 to 0.35mm. As the causes of emission of an electron beam from the thermoelectric field emission cathode, the temperature, the degree of vacuum, the shape and the surface configuration of the thermoelectric field emission cathode (electrode portion), and the field intensity of that portion are mentioned. At startup via which the thermoelectric field emission cathode is led to its operating state, evaporation of oxides or the like attaching to the electrode surface occurs and the electrode surface is purified.
Patent JP-H08268865-A (JP)
Title: Cosmetic
Inventor: NISHIO HIROYUKI
IPC: C09K23/02
Filed: 1995-03-30
Abstract: PURPOSE: To prepare a cosmetic which comprises an ionic surfactant bearing an amide group of a specific structure and has high skin safety, excellent storage stability and physical functions. CONSTITUTION: This cosmetic contains an anionic surfactant bearing 2 hydrophobic and 2 hydrophilic groups and containing an amide group represented by the formula (the number of carbon atoms of RCO; 20, 18, 14, 12, 10 or 8; (n) is 2-4; X is H, an alkali metal ion, ammonium ion, an organic ammonium ion) as an active ingredient in an amount of 0.01-5wt.%. In addition, another surfactant, an emulsifier, a perfume, a colorant, a preservative and a pigment are appropriately incorporated therewith to give base cosmetic, make-up cosmetic, hair cosmetic and the like. The compound of the formula is obtained by reaction of an alkylenediamine with a 2-halogenoethanol, diacylating the product, introducing sulfate group thereinto and neutralizing the obtained product with a base.
Patent JP-H11278582-A (JP)
Title: Transparent conductive cover tape
Inventor: NISHIZAWA MASUMI
IPC: C08L23/08
Filed: 1998-03-27
Abstract: PROBLEM TO BE SOLVED: To manufacture a cover tape of superior bonding properties when a polystyrene carrying tape is heat sealed and also provided with superior antistatic properties and transparency. SOLUTION: A cover tape is formed of at least a biaxially oriented resin film layer 5, a heat sealant layer 4, and an antistatic layer 3 laminated successively, and the heat sealant layer 4 is composed of ethylene copolymerized resin, and the antistatic layer 3 is formed of a layer in which an antimony dope oxide tin having the 0.2-2.0 μm long axial direction particles and the 0.01-0.02 μm axial direction particles and also having the 20-30 particle diameter ratio between the long axis and the short taxis is dispersed in the ethylene copolymerized resin.
Patent JP-S61261515-A (JP)
Title: Apparatus and method for rising and falling guide leader in ground improvement machine
Inventor: NOGATA HIROSHI
IPC: E02D3/12
Filed: 1985-05-14
Abstract: PURPOSE:To simply secure the rising and falling of a guide leader by a method in which the guide leader is tilted and turned to the direction of rising by controlling the height of its top to low levels and by pulling up its intermediate portion, and is then again restored to the upright position. CONSTITUTION:A ship base 1, a guide leader 2, and a bracket 3 projected from the end of the base 1 are provided, and they are rotatably connected with the basal portion of the leader 2 and a shaft 4. A treating machine 5 is hung down from the side face of the leader 2 by a wire (c) through a sheave pivotally supported on the top of the leader 2. The integrally collected tops 7 of frames 6 of a tripod supporting structure are positioned in the face of the intermediate portion of the leader 2. The long and great guide leader can thus be very simply raised or made to fall down with good efficiency even in regions where heights are limited according to areas, time periods, etc., like air ports and its neighboring areas.
Patent JP-S60241613-A (JP)
Inventor: NISHIKAWA SEIICHI
IPC: H01B13/00
Filed: 1985-05-14
Abstract: (57)【要約】本公報は電子出願前の出願データであるた め要約のデータは記録されません。
Patent JP-S5527925-A (JP)
Title: Method of manufacturing senser
Inventor: OGAWA KUNI
IPC: G01N27/12
Filed: 1978-08-17
Abstract: PURPOSE: To make possible detection of density of gas and vapor contained in a material at a high sensitivity by changing mere measuring temperatures used if ultrafine grain film of Sn oxide as a sensitive material is sticked onto a supporting substrate in a special atmosphere.  
     CONSTITUTION: Sn, SnO or SnO 2  are evaporized in the atmosphere of O 2  gas pressure of 0.1W1 Tor and on the substrate 3 on which electrodes 9, 10 are previously mounted by vacuum evaporation, etc. is formed ultrafine grain film 11 of Sn oxide. This senser can selectively detect isobutane if measured at 200°C or vapor if measured at room temperature. 
     COPYRIGHT: (C)1980,JPO&Japio
Patent JP-S62257639-A (JP)
Title: Information processor
Inventor: ANDO HIDEO
IPC: G11B7/09
Filed: 1986-04-30
Abstract: PURPOSE:To simplify the magnetic circuit and to obtain a small-sized, light weight titled processor with low cost by using the 1st coil so as to move at elast an objective lens in an optical head in the 1st direction, and using the 2nd coil to move the lens in the 2nd direction orthogonal to the 1st direction. CONSTITUTION:The objective lens 18 is provided in the optical head 5, the objective lens 18 is moved in the optical head 5 vertically, that is, unidirectionally in approaching/parting to/from the information storage medium 1 and moved by an objective lens drive circuit 20 in response to a signal from an out-of-focus detection circuit 19. Further, a head support is moved laterally with the objective lens 18 and moved within the range of recording area of the medium 1 for accessing. As to the track deviation caused by the eccentricity of the medium 1, the optical head 5 is moved for correction.
Patent JP-H02279962-A (JP)
Title: Air conditioner
Inventor: SEKIGAMI KUNIMORI
IPC: F25B29/00
Filed: 1989-04-20
Abstract: PURPOSE:To make it possible to select freely a simultaneous cooling operation and a simultaneous heating operating for a plurality of user side units and cooling and heating simultaneous operations based on an arbitrary user side unit by constituting a unit-to-unit pipe which connects a heat source side unit with a plurality of user side unit of three refrigerant pipes of a high pressure gas pipe, a low pressure gas pipe, and a liquid pipe. CONSTITUTION:A unit interspace which connects a heat source side unit 1 with user side unit 5a, 5b, 5c, and 5d comprises a high pressure gas pipe 12 which branches a pipeline 11 from a refrigerant discharge pipeline 7, a low pressure gas pipeline 15 branched from a refrigerant suction pipeline 8, and liquid pipeline 14 connected with heat source side heat exchangers 3a and 3b. One end of a specific user side heat exchanger 6d is connected with the high pressure gas pipeline 12 by way of an on/off valve 18 while the other end is connected with the liquid pipe 14. On the other hand, other user side heat exchangers 6a, 6b, and 6c are branched and connected with the high pressure gas pipeline 14 and the low pressure gas pipeline 13 by way of change over valves 15a, 16a, 15b, 15b, 15c and 16c respectively, and connected with the liquid pipeline 14 by way of refrigerant decompression devices 17a, 17b, and 17c, such as motor-driven expansion valves. The heat source side heat exchanger 3a, the user side heat exchanger 6a, and the specific user side heat exchanger 6d are a double pipe type water service heat exchanger.
Patent JP-S583619-A (JP)
Title: Production of honeycomb type filter
Inventor: NISHIO SHINJI
IPC: F01N3/02
Filed: 1981-06-29
Abstract: PURPOSE:To easily produce a honeycomb structure in which the ends of every other passage are closed, by a method wherein the second ends of tubular passages having the first ends closed are stopped up with an organic binder, and the second end part is immersed into a casting slip containing an inorganic powder, followed by firing. CONSTITUTION:A honeycomb structure is molded from body prepared by kneading an inorganic  powder of cordierite or the like and a binder. Then, only the first end face of the structure is immersed into a casting slip prepared by adding acetone to said body, and after taking out the  structure from the casting slip, the casting slip is blown off for every other tubular passage by blowing compressed air from the second end face of the structure, and the casting slip remaining in the passages is dried. Next, the second end face of the structure is immersed into a casting slip consisting solely of an organic binder such as vinyl acetate to stop up the entire part of the second end face, and the slurry is blown off by compressed air blown from the first  end face so that the binder is left only at the second ends of the passages which are closed at the first ends. After drying the binder left in the structure, the second end face of the structure is immersed in the same casting slip as that used for immersing the first end face, whereby only the second ends of the passages closed at the first ends are stopped up with the casting slip containing the inorganic powder. The structure thus obtained is dried and is fired at a temperature at which only the organic binder is pyrolyzed.
Patent JP-S5325310-A (JP)
Title: Vertical deflection unit
Inventor: SHIOTANI YUUICHI
IPC: H04N3/223
Filed: 1976-08-23
Abstract: PURPOSE:To adjust the vertical amplitude without deteriorating the vertical lineaaity by forming the vertical deflection position using a saw-tooth wave circuit, comparison circuit, driving circuit, output circuit and feedback circuit respectively.
Patent JP-S5529631-A (JP)
Title: Icebreaker
Inventor: URABE NAMIO
IPC: B63B35/08
Filed: 1978-08-21
Abstract: PURPOSE: To prevent the reduction of propulsive force by constituting an icebreaker so that small pieces of ice plates after ice-breaking fall down on non-broken ice plates on both sides of the ship by means of a spade body and evading the effect of small pieces of broken ice to the screw of the icebreaker.  
     CONSTITUTION: A bow protruded part 3 is formed which has a knife-edge part 2 at the front surface of the bow lower than a draft line 1 (in ice-breaking), and a spade body 4 is installed on the outer surface of the ship side from the upper part to the rear part. The spade body 4 is installed so as to form rising gradient towards rear part for the outer surface of the ship side and to form falling grandient towards  the outside of the ship body more at the rear part. At the bottom of the ship at the  bow, a ballast tank 7 is arranged, which helps the change from the average draft  line 8 in the navigation in no-ice water area to the average draft line in performing ice-breaking operation through navigation in frozen water area. If desired, a  number of opening parts are formed on the upper side along the spade body 4, and  from said opened parts, discharge water in high temperature is discharged. 
     COPYRIGHT: (C)1980,JPO&Japio
Patent JP-S583997-A (JP)
Title: Regulating method for deposition of electrodeposition paint film
Inventor: ASAI HISASHI
IPC: C25D13/00
Filed: 1981-06-29
Abstract: PURPOSE:To deposit paint films of a uniform desired thickness on a substrate in the stage of moving the substrate along the conveyance line in a coating cell and painting the same by electrodeposition by regulating the size of insulation members covering the stationary electrodes facing the side parts of the substrate. CONSTITUTION:The water soluble paint 16 in an electrodeposition cell 15 is maintained at prescribed pH, temp. and concn. A positive voltage is applied to bare electrodes 23, and diaphragm electrodes 25 and a negative voltage to an electrode bar 20, that is, the car body 2 of a substrate. In this state, the body 2 is moved, and paint components are allowed to deposit over the entire surface of the body only for a constant time when the body moves in a conveyance line 17. Here, the field intensities around the respective  surfaces in the bottom part 11 and upper part 14 of the body are kept approximately equal to the field intensities around the surfaces in both side parts 12 of the body. More specifically, the side parts 12 are nearest the electrodes 25, but the field intensities in these parts are so regulated by insulation members 26 of a prescribed longitudinal width L that they are weakened by a prescribed rate. The paint films of a uniform thickness are deposited on the respective parts of the body 2 by this.
Patent JP-H09278346-A (JP)
Title: Bedding base and bedding base lifting equipment
Inventor: HAMADA FUSAO
IPC: B66F9/06
Filed: 1996-04-23
Abstract: PROBLEM TO BE SOLVED: To provide a bedding base and bedding base lifting equipment that simplifies bedding laying and storage work while being simple in constitution and easy to manufacture. SOLUTION: A bedding base A is formed of a rectangular frame body, a cloth body 11 supported on the frame body, and belts 12, 12 locked to the frame body so as to longitudinally hold bedding B laid on the cloth body 11. It is so constituted that the frame body can be lifted while holding the bedding B by the belts 12, 12. The frame body is formed by connecting two partial frame bodies 13, 14 symmetrically formed in almost the same U-shape from the top view. These two partial frame bodies 13, 14 are connected in a relative distance changeable state, and the bedding B as it is integrated with the bedding base A is raised and lowered by bedding base lifting equipment.
Patent JP-H06293740-A (JP)
Title: Azole compound, its production and use thereof
Inventor: ITO KATSUMI
IPC: A61P31/10
Filed: 1993-04-27
Abstract: PURPOSE:To obtain a new azole compound usable for preventing and treating mammal mycotic infection, having low toxicity and strongly antifungal activity against fungus and a board antifungal spectrum. CONSTITUTION:A compound of formula I (Ar is substituted phenyl; R<1> and R<2> are H, lower alkyl to together bonded to form lower alkylene; R<3> is group to be bonded through C atom; R<4> is H or acyl; X is N or CH; Y and Z are N, [CH which may be replaced with lower alkyl) or its salt such as 2-[(1R,2 R)-2-(2,4-difluorophenyl)-2-hydroxy-1-methy1-3-(1H-1,2,4-triazol-1-yl) propyl]-4-(4- trifluoromethoxyphenyl)-3 (2H,4H)-1,2,4-triazolone. This compound is obtained by reacting a compound of formula 11 with a compound of formula III or its salt. The compound can be used as an agricultural antifungal agent.
Patent JP-S58218533-A (JP)
Inventor: MURAI KUNIHIKO
IPC: E04H15/20
Filed: 1982-06-12
Abstract: (57)【要約】本公報は電子出願前の出願データであるた め要約のデータは記録されません。
Patent JP-S61254832-A (JP)
Inventor: BUORUFUGANGU ZAMUHAABAA
IPC: C12M1/26
Filed: 1986-05-02
Abstract: (57)【要約】本公報は電子出願前の出願データであるた め要約のデータは記録されません。