baber/WOPTO huggingface dataset:
Patent EP-0584191-A1 (EP)
Inventor: CHARPENTIER BRUNO
IPC: C07C69/007
Filed: 1992-05-04
Abstract: Composés bicycliques aromatiques, caractérisés par le fait qu'ils répondent à la formule générale (I) dans laquelle: R1 représente notamment -H, -CH3, -CH2OH, -OH, -CHO, -CONH2, -COOH, -COOalkyle, -SH, -S-alkyle, etc..., R2 est H; R3 est H, aryle, aralkyle ou alkyle inférieur éventuellement substitué par un hydroxyle, un alcoxy inférieur ou un radical -CO-R12, R12 est notamment H, alkyle inférieur, hydroxyle, alcoxy inférieur, ou R2 et R3 pris ensemble forment avec le noyau benzénique un cycle naphtalénique; R4 est un alkyle linéaire ou ramifié ou non ayant de 1 à 15 atomes de carbone ou un radical cycloaliphatique, R5 représente notamment -(CH2)n-R13, -CH=CH-(CH2)n-R13, n étant 0 ou 1 à 6, R13 représentant -COR15, monohydroxyalkyle, polyhydroxyalkyle, alkyle inférieur époxydé ou -O-CO-R16, R15 représente notamment -OH, -Oalkyle, -Oaryle, R16 est notamment H, alkyle inférieur, aryle, ou aralkyle. R6 et R7 sont H, un halogène, alkyle inférieur ou -OR16, ainsi que les sels des composés de formule (I) pour lesquels R1 représente un groupement acide carboxylique, et les analogues chiraux desdits composés de formule (I).
Patent EP-0547229-A1 (EP)
Inventor: KOMIYA KATSUO
IPC: A61K47/02
Filed: 1992-06-22
Abstract: Préparation à usage externe contenant de la cyclosporine comme principe actif, et caractérisée par le fait qu'elle contient a) de la cyclosporine, b) un solvant organique servant à dissoudre celle-ci, c) un ester d'acide gras d'un alcool monovalent qui se liquéfie à 25 °C et présente en tout au moins 8 atomes de carbone, et/ou une alcanolamine liquide à 25 °C, d) une substance oléagineuse solide à 25 °C, et e) un agent tensioactif. La teneur en cyclosporine est comprise entre 0,1 et 10 % en poids, et la teneur en ester et/ou alcanolamine est comprise entre 1 et 15 % en poids. La préparation présente une excellente efficacité en ce qui concerne le traitement d'eczémas atopiques, de psoriasis, d'eczémas allergiques et ainsi de suite.
Patent EP-0678158-A1 (EP)
Inventor: WUNNING JOHN J
IPC: F01L9/20
Filed: 1992-05-18
Abstract: L'invention se rapporte à un système de régulation (14) pour un moteur à combustion interne (100) possédant une pluralité de cylindres (C1-Cn) et un vilebrequin rotatif (110). Chaque cylindre (C1-Cn) possède une soupape d'admission, une soupape d'échappement (120, 125) et un injecteur de carburant (130) à commande électronique. Le système de régulation comporte un détecteur (155) qui contrôle la rotation du vilebrequin (110) et produit en réaction un train d'impulsions concernant le vilebrequin. Un ordinateur (216) génère des signaux de paramètres de fonctionnement incluant l'un parmi plusieurs modes de fonctionnement du moteur (100). Un premier microprocesseur (226) reçoit le train d'impulsions concernant le vilebrequin, détermine en réaction la vitesse du moteur (100) et génère un signal représentatif de la vitesse déterminée du moteur. Un second microprocesseur (222) reçoit les signaux de paramètres de fonctionnement et le signal de vitesse du moteur, détermine en réaction les événements de l'injecteur de la soupape pour chaque cylindre (C1-Cn) pour exécuter en réaction le mode de fonctionnement du moteur choisi. Le second microprocesseur (222) génère des signaux représentatifs des événements déterminés de l'injecteur et de la soupape.
Patent EP-0539574-A1 (EP)
Title: Boite a surfaces inclinees
Inventor: EGGUM SHAWN D
IPC: H01L21/673
Filed: 1992-04-07
Abstract: Récipient servant à ranger et à transporter un boîtier de tranches de silicium rempli de tranches, le récipient se composant d'une boîte pourvue d'un couvercle pouvant être ouvert, la base de la boîte comprenant une partie en forme de panneau inférieur incliné et une partie en forme de panneau latéral incliné soutenant la base du boîtier et la paroi terminale à barre en H.
Patent EP-0598750-A1 (EP)
Inventor: BLAGG JULIAN C O PFIZER CENTRA
IPC: A61P3/06
Filed: 1992-07-20
Abstract: Composés répondant à la formule (I), et leurs sels pharmaceutiquement acceptables, dans laquelle Y représente alkylène C1-C6 éventuellement substitué par alkyle C1-C6; R représente H, OH, halo, alkyle C1-C4 ou alcoxy C1-C4 R1, R2, R3 et R4, indépendamment les uns des autres, sont sélectionnés parmi H , alkyle C1-C4, alcoxy C1-C4, OH, halo et CF3; l'un de R6, R7 et R8 représente un groupe de la formule (a) ou (b), les autres, conjointement avec R5 et R9, et indépendamment les uns des autres, étant sélectionnés parmi H, alkyle C1-C4 alcoxy C1-4, halo et haloalkyle(C1-C4); R10 représente COOH, COOR11 ou CONR12R13; R11 représente un groupe biolabile à formation d'esters; R12 et R13, indépendamment l'un de l'autre, sont sélectionnés parmi H et alkyle C1-C4; R14 représente H, alkyle C1-C6, cycloalkyle C3-C7 ou aryle; et le terme ''aryle'', tel qu'il est employé dans les notations de R6, R7, R8 et R14, signifie phényle éventuellement substitué par alkyle C1-C6, alcoxy C1-C6, alcényle C2-C6, OH, halo, CF3, halo(alkyle C1-C6), nitro, amino, alcanamido C2-C6, alcanoyle C2-C6, ou phényle; compositions pharmaceutiques les contenant; leurs procédés de préparation; et leurs utilisations.
Patent EP-0650596-A1 (EP)
Inventor: SCHMIDT GEOFFREY J
IPC: A61K47/48
Filed: 1992-03-30
Abstract: L'invention concerne un procédé de régulation du processus métabolique de l'inositol dans une cellule. Ce procédé consiste à introduire dans ladite cellule une molécule qui peut ensuite coupler un récepteur lié à une membrane, pouvant être activé par un signal externe, à une phosphodiestérase intracellulaire du genre sensible à générer une seconde substance messagère IP3. Cette molécule est sélectionnée dans le groupe se composant d'une protéine A purifiée, de fragments actifs, d'analogues actifs, et de produits de fusion actifs de ceux-ci. L'invention concerne également des procédés de détection d'une protéine A et des procédés d'inhibition de la croissance et de la prolifération des cellules cancéreuses à l'aide d'anticorps anti-protéine A.
Patent EP-0612349-A1 (EP)
Title: NOVEL THROMBIN INHIBITOR PROTEIN FROM -i(REDUVII).
Inventor: FRIEDRICH THOMAS
IPC: C07K14/00
Filed: 1992-10-27
Abstract: PCT No. PCT/EP92/02450 Sec. 371 Date Apr. 26, 1994 Sec. 102(e) Date Apr. 26, 1994 PCT Filed Oct. 27, 1992 PCT Pub. No. WO93/09232 PCT Pub. Date May 13, 1993.A novel thrombin-inhibitory protein from assassin bugs with a molecular weight of about 12,000 dalton and the N terminus Glu-Gly-Gly-Glu-Pro-Cys-Ala-Cys-Pro-His-Ala-Leu-His-Arg-Val-Cys-Gly-Ser-Asp is described. The protein is suitable for controlling diseases.
Patent EP-0609387-A1 (EP)
Inventor: NASH BRIAN
IPC: C08K3/36
Filed: 1992-10-23
Abstract: Sont décrites de nouvelles dispersions siliconées en une et en deux parties, qui conviennent pour appliquer une surface siliconée texturée durable sur des articles siliconés et non siliconés. La surface non bloquante est obtenue par enduction au trempé d'un article avec une couche finale. La dispersion utilisée pour les couches finales comprend une charge de silice hydrophile unique présentant une surface spécifique d'environ 75-200 m2 par gramme, au moins un polysiloxane réticulable et un agent de réticulation. Les particules de silice, noyées de manière fiable à l'intérieur de la couche finale de silicone de manière à ce que certaines parties s'étendent vers l'extérieur au-delà de la nouvelle surface siliconée extérieure de l'article, présentent une surface texturée non bloquante et non allergénique.
Patent EP-0614411-A1 (EP)
Inventor: NIELSEN JENS
IPC: B26F3/00
Filed: 1992-11-27
Abstract: Vanne de commande du découpage par jet de liquide, notamment des produits alimentaires tels que les filets de poisson. Elle comporte une plaque (1) à laquelle est relié un arbre moteur (3). Un moteur (2) peut positionner la plaque de manière qu'elle se trouve dans la trajectoire du jet de liquide (4) utilisé dans l'opération de découpage, ou la retirer.
Patent EP-0553682-A1 (EP)
Title: Imidazo  4,5-b pyridine derivatives as Angiotensin II antagonists
Inventor: OKU TERUO
IPC: A61P9/00
Filed: 1993-01-19
Abstract: A compound of the formula :
       
 wherein
     R¹   is hydrogen, halogen, nitro, lower alkyl, lower alkoxy, amino or acylamino,   R², R³ and R⁴   are each hydrogen, halogen, nitro, cyano, lower alkyl, lower alkenyl, lower alkylthio, mono or di or trihalo(lower)alkyl, oxo(lower)alkyl, hydroxy(lower)alkyl or optionally esterified carboxy; or   R² and R³   are linked together to form 1,3-butadienylene,   R⁵   is hydrogen or imino-protective group,   R⁶ and R⁷   are each hydrogen or lower alkyl,   R⁸   is hydrogen or lower alkyl which may have a substituent selected from the group consisting of halogen and lower alkoxy,   A   is lower alkylene,   Q   is CH or N,   X   is N or CH,   Y   is NH, O or S, and   Z   is NH, S, SO₂ or O.    and pharmaceutically acceptable salt thereof, processes for their preparation and pharmaceutical compositions comprising them as an active ingredient.
Patent EP-0559181-A1 (EP)
Inventor: MASSENZANA FABRIZIO
IPC: B31F1/28
Filed: 1993-03-03
Abstract: A process for coupling component elements of a multi-layered corrugated board consists in disposing the component elements previously coated with an adhesive material on a heating surface, and effecting an air suction close to the heating surface. A machine is provided which comprises heating members (6) forming a heating surface (5) and adapted to supply heat to a web of corrugated board, and a suction apparatus (10) adapted to create vacuum areas (12) contiguous to the heating surface (5).
Patent EP-0562470-A1 (EP)
Inventor: SCHLUMPF FLORIAN MASCH ING HTL
IPC: B62M11/14
Filed: 1993-03-19
Abstract: A variable bottom bracket ball bearing gear change for a bicycle or the like is proposed, which gear change comprises essentially a bottom bracket ball bearing housing (15), a transmission case (40) with associated chain wheel (35) and a drive shaft (20) which is operatively connected to peddle cranks (1, 2). 
<??>In the drive shaft (20) which is constructed as a hollow body a switch axle is arranged which can be actuated from the outside by means of switching elements (50, 50') operatively connected thereto in such a way that a clutch element which is operatively connected to the drive shaft (20) can be engaged with the chain wheel (35) which is provided with corresponding recesses or with a disc which is constructed for example as a sun wheel and is also provided with recesses. 
<??>The recesses which are provided in the chain wheel (35) and in the sun wheel are constructed offset in a stepped manner in such a way that the clutch element which can be connected to the chain wheel (35) or the disc can be engaged in a first phase with play and in a second phase without play in a locking fashion. 
<IMAGE>
Patent EP-0570892-A1 (EP)
Inventor: SAKAI MASANORI C O CANON KABUS
IPC: H04N1/32
Filed: 1993-05-17
Abstract: An information processing system comprises a core, a sub-unit (for example, a facsimile unit, a file unit, and a computer interface unit, a formater or an image memory) connected to the core, and the core and the sub-unit are connected by two types of buses, synchronous type and asynchronous type. Where the data transfer between the core and the sub-unit is to be effected through the asynchronous bus, the core may simultaneously transfer data to other sub-unit by using the synchronous bus. Where the data transfer between the core and the sub-unit is to be effected by the synchronous bus, the data may be parallelly transferred to a plurality of sub-units.
Patent EP-0574725-A1 (EP)
Inventor: SEIDEL ANDREAS DR
IPC: C07C67/10
Filed: 1993-05-21
Abstract: A process for the preparation of vinyl esters of haloacetic acids of the general formula (I> HalnHmC-COO-CH=CH2 (I> in which     Hal is equal to Cl or Br,   n is equal to 1, 2 or 3,   m is 3-n, is given, which is characterised in that a haloacetic acid of the general formula (II> HalnHmC-COOH (II> in which Hal, n and m have the abovementioned meaning, is allowed to react with a vinyl ester of the general formula (III> R-CH2-COO-CH=CH2 (III> in which R denotes hydrogen or an alkyl radical having 1 to 6 C atoms, in liquid phase in the presence of a palladium(II) compound as a catalyst, a copper(II) compound as a co-catalyst and an alkali metal compound as a promoter at 20 DEG C to 100 DEG C over a period of 0.1 to 10 hours, then the evaporable fractions of the catalyst components are removed from the reaction mixture in a flash evaporation and the catalyst components are subsequently oxidatively treated, the evaporated fractions are condensed and the condensate is separated by means of distillation into unreacted vinyl ester, crude vinyl ester of haloacetic acid and unreacted haloacetic acid, the crude vinyl ester of haloacetic acid is extracted with water at 5 DEG  to 20 DEG C, as a result of which the carboxylic acid formed from the vinyl ester employed is transferred to the aqueous phase, and the vinyl ester of haloacetic acid removed as the organic phase is optionally treated with a drying agent.
Patent EP-0574726-A1 (EP)
Inventor: BRENDEL JOACHIM DR
IPC: C07D498/04
Filed: 1993-05-21
Abstract: The present invention relates to fused 1,2,5-oxadiazole 2-oxides of the general formula I <IMAGE>  in which  A denotes <IMAGE>  -(CH2)n-Y-, -CH2-Z-CO-, <IMAGE>  or <IMAGE> and X, Y, Z and also R<1>, R<2>, R<3> and n are defined as indicated in Claim 1, to processes for their preparation and to their use.
Patent EP-0580988-A1 (EP)
Inventor: GRATZER FRANZ DIPL-ING
IPC: F16D41/08
Filed: 1993-06-01
Abstract: A roller clutch consists of an outer race (5), an inner race (2) and a cage (7) with rolling elements (1). The cage (7) and the outer race (5) are frictionally connected and a pawl (11) actuated by centrifugal force mounted on the inner race (2) interacts with a projection (14) on the cage (7). As a result, the clutch acts in both directions of rotation and torque application and the free-wheel action comes into play only at relatively high speed. <IMAGE>
Patent EP-0575791-A1 (EP)
Inventor: OHNISHI NORIAKI
IPC: C08F2/50
Filed: 1993-06-03
Abstract: The present invention relates to a liquid crystal composite layer of polymer dispersion type in which
     (a) a liquid crystal material comprising compounds selected from the group consisting of compounds represented by the following chemical formula (1) and compounds represented by the following chemical formula (2) is dispersed in   (b) a matrix polymer;
           
 wherein
   A₁ and A₂   represented respectively a benzene ring, cyclohexane ring, pyrimidine ring or trans-1,3-dioxane ring;   X₁, X₂,X₃, X₄, X₅ and X₆   represent respectively H, F or Cl;   Z₁ and Z₂   represent respectively a single bond, -CH₂-, -CH₂CH₂-, -CH=CH-, -C≡C-, -COO- or -OCO-;   Q   represents a single bond, -CH₂-, -CH₂CH₂-, -CF₂-, OCF₂-, -C₂F₄-, -CCl₂- or -C₂Cl₄-;   Y   represents H, F or Cl;   R   represents -C n H 2n+1 -,-C n H 2n+1 O-, -C n H 2n+1 CH=CH- (in which n represents an integer of 2-10);   m   represents 0, 1 or 2;
           
 in which B and C represent respectively -C n H 2n+1 -, -C n H 2n+1 O-, -C n H 2n+1 -CH=CH- or -C n H 2n+1 -C 6 H 10  (in which n is the same as mentioned above, and L is H or F.
Patent EP-0584699-A1 (EP)
Inventor: SATO SHINICHIRO C O CASIO COMP
IPC: G06F17/30
Filed: 1993-08-17
Abstract: A data searching apparatus is capable of searching for an image of an object, relevant combined data or character data corresponding to the image of the object based on part data which compose the object image. At least one of a plurality of part data composing the object image is designated by operation a key input unit (12), and image data including the part data which coincides with the designated part data is read out from among a plurality of combined data stored in a memory unit (14) or among from a plurality of relevant image data stored in a memory unit (13). The object image to be searched for is displayed on 3 display unit (19) based on the read out image data or combined data. Further character data representing the object are displayed on the display unit (19) together with the object image.
Patent EP-0585757-A1 (EP)
Inventor: MEZZOLI GIORGIO
IPC: A61F13/36
Filed: 1993-08-20
Abstract: Nasal and/or rhinopharyngeal tampon including an elongated core (2), with aspiration holes (7), around which there is a shaped body (3) made of elastic spongy material covered by a thin deformable membrane (4) made of impermeable material; the core has a stem (5) for connection to an aspiration unit (6) suitable to make the body assume an insertion or extraction configuration having a limited volume in a vacuum state; the flow of air through the stem into the shaped body is suitable to make the body resume an active configuration having a large volume at atmospheric pressure.
Patent EP-0598224-A1 (EP)
Inventor: OGALE KUMAR
IPC: D04H1/42
Filed: 1993-10-15
Abstract: Disclosed is a nonwoven textile material comprising fibers of a propylene polymer material blended with an olefin polymer material.
Patent EP-0603870-A1 (EP)
Inventor: SMITH RONALD T
IPC: G02B5/32
Filed: 1993-12-22
Abstract: A hologram structure for use in a holographic center high mounted stoplight system for a vehicle is disclosed. The hologram structure includes a hologram layer (49) having a plurality of holographic lenses (C) formed therein, each holographic lens (C) being configured to diffract light into a predetermined solid angular region.
Patent EP-0570063-A1 (EP)
Inventor: BREDOL MICHAEL DR
IPC: C09K11/56
Filed: 1993-05-07
Abstract: The invention relates to a luminescent zinc sulphide having a cubic structure (zinc blende) which has been activated with aluminium and copper in such a way as to produce a green luminophor. It combines ease of manufacture with high X-chromaticity values and a high light yield as a result of incorporating copper in an amount from 200 to 450 mol-ppm and aluminium in an amount from 700 to 2000 mol-ppm. <IMAGE>
Patent EP-0588435-A1 (EP)
Inventor: VAN DEN AARSEN GERARDUS FRANCI
IPC: B65F3/08
Filed: 1993-09-15
Abstract: The invention relates to a container loading and emptying device for a refuse vehicle with an endless carrier consisting of two chains(10,11), which runs in a substantially vertical plane along a substantially rectangular path, one or more pick up members(13), which are fitted to a shaft(12) connected to the endless carrier(10,11) and which are rotatable around this shaft(12) and tilting means consisting of rolls (15,16,17,18) mounted to the pick up member(13) and guides(27a,27b,28,27a',27b',28',30,31) for the said rolls mounted on the frame(3), with which at the upper angular points and a successive part of the upper part of the path the pick up member(13) rotates over an angle of 180°, wherewith seen in the lowermost vertical position, the pick up member(13) is provided with two rolls(17,18) mounted symmetrically with respect to the vertical central line of the pick up member(13) below the pivot point of the pick up member(13), with guides(27a,27b,28,27a',27b',28') for the said rolls(17,18) mounted at the upper angular points of the path and that the shaft(12) which connects the chains(10,11) to each other and whereto the pick up member(13) is fitted, is a straight shaft.
Patent EP-0656172-A1 (EP)
Inventor: CAPPON WILFRIED J M
IPC: A01F29/10
Filed: 1993-12-04
Abstract: A forage harvester is provided with a cutterhead frame (34), mounted on a support (40) which can be pivoted about a cylindric beam (80) at the top thereof. The cutterhead frame (34) can be pivoted about the axis (39) of the cutterhead (36) under the action of hydraulic cylinders (90). Lower feedrolls (26,27) are installed in a lower feeder frame (24), attached to the cutterhead frame (34), and upper feedrolls (20,21) are installed in an upper feeder frame (18), which can be tilted forwardly about a cylindric beam (67) attached to the front of the lower feeder frame (24). Means (61,62) for the coupling of a crop collecting apparatus (10) also serve to support the upper feeder frame (18), when the latter is separated from the lower feeder frame (24). Other means (96,95) enable the attachment of the upper feeder frame (18) to a tractor (110). Thus can be gained access for inspection and servicing between the upper (20,21) and lower feedrolls (26,27) and to the cutterhead (36). The support (40) can be secured to the cutterhead frame (34) in order to raise both together and gain access between the cutterhead (34) and the blower rotor (49).
Patent EP-0590746-A1 (EP)
Inventor: ALDRIDGE IRENE YEATMAN
IPC: C11D3/386
Filed: 1993-09-24
Abstract: A method for inhibiting or removing biofilm from surfaces which are in contact with an aqueous system comprising adding to the system an enzyme composition consisting essentially of proteases, optionally in combination with certain other enzymes and/or surfactants, in amounts effective to inhibit or remove the biofilm.
Patent EP-0564154-A1 (EP)
Inventor: MITANI YOUKO
IPC: A61K9/10
Filed: 1993-03-24
Abstract: A pharmaceutical formulation in the form of aqueous suspension which comprises an ion exchange resin carrying an active ingredient and a suspending agent, characterized in that the formulation further contains a basic or neutral amino acid or a salt thereof as a dispersion stabilizer.
Patent EP-0586056-A1 (EP)
Inventor: REEVES GEOFF
IPC: A61M1/00
Filed: 1993-07-06
Abstract: A medical coupling device (8) to form part of a medical system designed to withdraw an ovum from a follicle, said system comprising a first conduit means (9), extending from the follicle, via the coupling device (8) to an aspiration arrangement at which the ovum is to be collected, said system also comprising a second conduit means (10) extending from a source of flushing media to the coupling device (8) in which connection between the first and second conduit means (9,10) occurs, whereby flushing media can be applied to the follicle to assist in the withdrawal of the ovum, the coupling device (8) comprises an inner chamber (3) and first means for terminating the said second conduit (10) means in the chamber (3), in that the first conduit means (9) has a lumen therein adapted (11) to be in fluid communication with the said inner chamber (3), and in that the device (8) also comprises means (16,17) for sealing the first and second conduit means (9,10) with respect to the said chamber (3).
Patent EP-0581464-A1 (EP)
Inventor: BIRD THOMAS GEOFFREY COLERICK
IPC: C07D407/12
Filed: 1993-07-08
Abstract: The invention concerns ester derivatives of the formula I
       
wherein Ar is phenyl, naphthyl, indenyl, indanyl, a 10-membered bicyclic heterocyclic moiety containing one or two nitrogen heteroatoms and optionally containing a further heteroatom selected from nitrogen, oxygen and sulphur, or a 9-membered or 10-membered bicyclic heterocyclic moiety containing one heteroatom group selected from oxygen, sulphur, sulphinyl, sulphonyl and imino;
     A 1  is a direct link to the oxygen atom of the ester group or A 1  is (1-3C)alkylene ;   each of R 4  and R 5  is hydrogen or (1-4C)alkyl;   R 1  is (1-4C)alkyl, (3-4C)alkenyl or (3-4C)alkynyl ; and   R 2  and R 3  together form a group of the formula -A 2 -X-A 3 - wherein each of A 2  and A3 is independently (1-3C)alkylene and X is oxy, thio, sulphinyl, sulphonyl or imino;   or pharmaceutically-acceptable salts thereof ;   processes for their manufacture; pharmaceutical compositions containing them and their use as 5-lipoxygenase inhibitors.
Patent EP-0595527-A1 (EP)
Inventor: PAPPALARDO ROMANO G
IPC: C09K11/72
Filed: 1993-10-19
Abstract: A fluorescent lamp having a plurality of lamp phosphors for converting ultraviolet radiation to visible illumination, in which the lamp phosphor comprises a plurality of metameric blends. The metameric blends of lamp phosphors having substantially identical color coordinates. Cheaper phosphor blends may then be used in conjunction with more expensive fluorescent coatings of the same color coordinate to produce a cheaper fluorescent lamp of the same color coordinates.