baber/WOPTO huggingface dataset:
Patent CZ-284798-B6 (CZ)
Title: Oral pharmaceutical preparation against cough
Inventor: GALLI ANGELI DEPALMO
IPC: A61P11/14
Filed: 1995-02-22
Abstract: PCT No. PCT/EP95/00658 Sec. 371 Date Dec. 24, 1996 Sec. 102(e) Date Dec. 24, 1996 PCT Filed Feb. 22, 1995 PCT Pub. No. WO95/23602 PCT Pub. Date Sep. 8, 1995Oral antitussive pharmaceutical composition which allows a significant contact of its components with mucous membranes of the buccal cavity and comprises a centrally acting antitussive or a pharmaceutically acceptable salt thereof and benzydamine or a pharmaceutically acceptable acid addition salt thereof.
Patent CZ-286695-B6 (CZ)
Title: 1,5-Benzodiazepine derivatives, process of their preparation, their use and pharmaceutical preparations in which they are comprised
Inventor: SUGG ELIZABETH ELLEN
IPC: C07K5/08
Filed: 1994-04-14
Abstract: In the present invention there are disclosed 1,5-benzodiazepine derivatives of the general formula I, in which the individual symbols are as specified in the main Claim. These substances exhibit agonistic activity on CCK-A receptors and they can be therefore used for preparing pharmaceutical preparations, which also form the part of the present invention and which are intended for modulation of gastrin and CCK cholecystokinin in mammals, i.e. for inducing anorectic effect and treating obesity. In the present invention, there are also claimed processes for preparing said derivatives.
Patent CZ-292792-B6 (CZ)
Title: Quinoxalinediones, process and intermediates for their preparation as well as pharmaceutical compositions based thereon
Inventor: BULL DAVID JOHN
IPC: C07D401/04
Filed: 1997-02-27
Abstract: The present invention provides quinoxalinediones of the general formula I and the pharmaceutically acceptable salts thereof, wherein R is a 5-membered ring heteroaryl group containing 3 or 4 nitrogen heteroatoms which is linked to the quinoxalinedione ring by a ring carbon or nitrogen atom, or is a 6-membered ring heteroaryl group containing from 1 to 3 nitrogen heteroatoms which is linked to the quinoxalinedione ring by a ring carbon atom, either of said groups being optionally benzo-fused and optionally substituted, including in the benzo-fused portion, by 1 or 2 substituents each independently selected from alkyl, alkenyl,  cycloalkyl, halo, hydroxy, alkoxy, cycloalkyloxy, -COOH, alkoxycarbonyl, -CONRe3Re4, -NRe3Re4, -S(O)ip-alkyl), -SO2NRe3Re4, aryl, aryloxy, arylalkoxy and heterocycle, said alkyl being optionally substituted by cycloalkyl, halo, hydroxy, alkoxy, haloalkoxy, cycloalkyloxy, cycloalkylalkoxy, -COOH, alkoxycarbonyl, -CONRe3Re4, -NRe3Re4, -S(O)ip-alkyl, -SOi2NRe3Re4 aryl, aryloxy, arylalkoxy and a heterocycle, and said alkyl or alkenyl being optionally further substituted; Re1 and Re2 are each independently selected from hydrogen, fluoro, chloro, bromo, alkyl and haloalkyl; Re3 and Re4 are either each independently selected from hydrogen or alkyl or, when taken together, are alkylene; p is 0, 1 or 2; together with the preparation of, compositions containing, the uses of and intermediates used in the synthesis of, such compounds. The compounds are useful as NMDA receptor antagonists for treating acute neurodegenerative and chronic neurological disorders, for example apoplexy.
Patent CZ-290252-B6 (CZ)
Title: Process for preparing 4H-4-oxo-quinolizine-3-carboxylic acid derivatives
Inventor: WANG WEI-BO
IPC: C07D455/02
Filed: 1998-02-06
Abstract: In the present invention there is disclosed a process for preparing carboxylic acid of the general formula II, in which the substituents Re1 through Re5 have specific meaning, by reacting enamine with acid chloride and further by reacting the resulting intermediate with malonamic acid ester in the presence of a base. Subsequently the obtained compound is protected on the hydroxy position by treatment thereof for example with methyl chloride. The resulting compound then reacts with an alkali metal base and subsequently with 3-alkoxyacryloyl compound and the formed intermediates is reacted with a catalytic amount of acid in order to close a ring and finally the resulting acid is reacted with a halogenating agent.
Patent CZ-298488-B6 (CZ)
Title: Pharmaceutical composition containing tumor suppressor nucleic acid
Inventor: NIELSEN LORETTA
IPC: A61K31/4545
Filed: 1998-02-17
Abstract: In the present invention, there are disclosed methods of treating mammalian cancer or hyperproliferative cells, said methods comprising contacting said cells with a tumor suppressor protein or tumor suppressor nucleic acid and also contacting said cells with at least one adjuvant antitumor agent. There are also disclosed pharmaceutical compositions comprising a tumor suppressor protein or a tumor suppressor nucleic acid and at least one adjuvant antitumor agent as well as kits for the treatment of mammalian cancer or hyperproliferative cells.
Patent SK-284560-B6 (SK)
Title: A load-bearing structure of a glass wall or glass roof made of glass panels
Inventor: FISCHER KLAUS
IPC: E04B1/32
Filed: 1996-02-13
Abstract: A load-bearing structure of a glass wall or glass roof made of glass panels (56), which load-bearing structure comprises a plurality of bars (12 through 22). Each bar have an end region (28) of lesser height than the remainder of the bar, each end region (28) define a pair of end faces (30, 32); two cover disks (34, 36) and a plurality of threaded bolts (40). Bars (12 through 22) are joined together at their end regions (28) such that said end faces (30, 32) are in abutment and form thereby upper and lower countersunk areas of lesser height. The bar end regions (28) lying in the node (10) have a reduced bar height (15) by comparison with the remaining bar region and are held bolted together (40) between two cover disks (34, 36), which mutual spacing (17) is less than the height (15) of the bar (12 through 22).
Patent SK-284108-B6 (SK)
Title: Novel 2,3-disubstituted-4(3H)-quinazolinones
Inventor: ELLIOTT MARK LEONARD
IPC: C07D239/91
Filed: 1997-02-17
Abstract: The present invention relates to novel 2,3-disubstituted- 4(3H)-quinazolinones compounds of formula (I), and their pharmaceutically acceptable salts, and pharmaceutical compositions and methods of treating neurodegenerative and CNS-trauma related conditions.
Patent SK-284780-B6 (SK)
Title: Process of optical cleaning enantiomeric enriched benzimidazole derivatives
Inventor: UNGE SVERKER VON
IPC: C07D401/12
Filed: 1996-06-26
Abstract: Described is process for the optical purification of the single enantiomers of some 2-sulphinyl-1H-benzimidazole derivatives and another structurally related sulphoxide from the respective enantiomerically enriched preparation thereof.
Patent SK-281179-B6 (SK)
Title: N-acyl derivatives of ll-e33288 antibiotics, methods of their preparation, their use for the preparation of medicaments
Inventor: LEE MAY DEAN-MING
IPC: C12P19/60
Filed: 1990-04-13
Abstract: N-acyl derivatives of the LL-E33288 antibiotics of the general formula (I) wherein W represents the general formula (II), where R1 is H or a group of the formula (III), R4 is a hydroxyl group when R5 is H or R4 and R5 taken together are a carbonyl; and X is a iodine or bromine atom, R is H or a branched or unbranched alkyl (C1-C10) optionally substituted by one or more hydroxyl or carboxyl groups and R2 is a methyl group, ethyl group or CH(CH3)2 with the proviso that if R1 represents a group of the formula (III), R2 is an ethyl group, R4 and R5 taken together are carbonyl group and X is a iodine atom then R is not a methyl group. Also disclosed is a method of preparation of said derivatives. These derivatives are effective antibacterial and antitumor agents.
Patent SK-289058-B6 (SK)
Title: High gain boost converter with the coupled inductors and the resetting of the magnetic flux
Inventor: PRAŽENICA MICHAL
IPC: H02M3/00
Filed: 2018-08-11
Abstract: The high gain boost converter with the coupled inductors and the resetting of the magnetic flux, consists of the DC source (1) and the boost converter (2). The latter consists of the power switches (3), the coupled boost inductors (4), coupled desaturating block (5) and the output part (7) comprising the output condenser with the load and the control circuit (8).  The connection is characterized by the converter that obtains a high constant gain due to reciprocal magnetic coupling between the inductors. The desaturating inductor ensures resetting of a magnetic flux of the coupled inductors hence it prevents the magnetic circuit of oversaturation and this energy is moved via desaturating rectifier to the load, so that the efficiency of the connection is higher.
Patent SK-279320-B6 (SK)
Title: Automatic gearbox
Inventor: MICHALKO JAN
IPC: F16H15/48
Filed: 1989-11-03
Abstract: An automatic gearbox has two epicyclical arrangements rotating round the axis of a flywheel. A first arrangement being driven by the flywheel (2) is represented by rollers (3). A second arrangement is represented by balls (7). Once the gearbox is working, these two arrangements are, through a thread (10), nut (20) and spring (21), pressed against each other by means of a force which varies depending on a degree of a transmitted torque.
Patent CZ-300133-B6 (CZ)
Title: Process for preparing fatty acid methyl esters by transesterification of triglycerides, particularly from rapeseed oil and apparatus for making the same
Inventor: MACEK RADOVAN
IPC: C07C67/03
Filed: 2005-04-06
Abstract: The present invention relates to a process for preparing fatty acid methyl esters by transesterification of triglycerides, particularly from rapeseed oil and apparatus for making the same wherein the process is characterized by separating residues of glycerin phase form ester phase by cooling the ester phase leaving a third reactor (4) within a cooler (5) down to 30 to 50 degC and than supplying thereof in a coagulator (6) at the inlet of which the glycerin phase from a second separator (7) is supplied along with the glycerin phase from a first separator (3) in such a ratio as to make the ratio of the glycerin phase to the ester phase in the coagulator (6) within the range of 1:3 to 3:1.
Patent CZ-308920-B6 (CZ)
Title: Method and device for redundant optical measurement and / or calibrating the position of a body in space
Inventor: Valášek Michael
IPC: G01B21/00
Filed: 2013-03-11
Abstract: Method for redundant optical measurement and / or optical calibration of the position of a body in space by at least one laser tracker (4) placed on the measured or calibrated body (3) or on the frame (1) of the body and at least two laser beam reflectors (5) placed on the measured or calibrated body (3) and / or on the body frame (1), so that the laser tracker (4), which uses an absolute method of measuring the positions of the laser reflectors, is set to at least one position on the frame (1), in which the position of at least three laser reflectors (5) of the laser beam (6) on the frame (1) is measured, then the position of these laser reflectors (5) of the laser beam (6) on the frame (1) is calibrated, then the laser tracker (4) is set in at least one further position on the frame (1), in which the position of at least these three calibrated laser reflectors (5) of the laser beam (6) on the frame (1) is measured and the position of the at least three laser reflectors (5) on the measured or calibrated body (3), and on the basis of these measurements the position of the measured or calibrated body (3) is determined, or a measured or calibrated body (3) on which a laser tracker (4) is arranged, which uses an absolute method of measuring the positions of laser reflectors, sets at least one position in space, in which the position of at least three laser reflectors (5) on the frame (1) is measured by a laser tracker (4), subsequently, the positions of the laser reflectors (5) on the frame (1) is calibrated from these measurements and at the same time determining the position of the measured or calibrated body (3). Equipment for redundant optical measurement and / or optical calibration of the position of a body in space, consisting of at least one laser tracker that uses an absolute method of measuring the positions of laser reflectors, placed on the measured or calibrated body or on the frame, and a number of laser beam reflectors located on the frame and / or on the measured or calibrated body, so that at least three laser reflectors (5) placed on the frame (1) or on a measured or calibrated body (3) are arranged in a triangle or a polygon.
Patent CZ-305389-B6 (CZ)
Title: Layered product of animal material particles and binder, process for its preparation and apparatus for making the same
Inventor: NIEDOBA KRZYSZTOF
IPC: B44F9/08
Filed: 2014-04-28
Abstract: The present invention relates to a layered product that is characterized in that the animal material are particles (2) optionally fractions of egg shells bonded by a suitable binding agent (3), further to a process for its production, which comprises crushing the shells, sorting thereof, selection of fraction size of the used particles (2), their arrangement into a monolayer (1) and encapsulating thereof in the binding agent (3), whereby after layering several monolayers (1) and incorporation of a tension-resistant material, hardening thereof takes place. Apparatus for producing the above-described product consists of a shell crushing device (10), having its outlet directed into a sorting device (11) with an outlet gap of a monolayer (1) removable mold (12) that can be positioned and opened by a positioning and tipping device (13) being followed up with a monolayer (1) vacuum transfer device (14) to a solid back plate (15), particularly non-wettable for the binding agent, wherein a positionable binder (3) dosing device (16) is arranged close thereto. The solid back plate (15) is situated in working area of a composite vacuum transfer device (17) to molding and hardening device (18) optionally a press.
Patent CZ-307611-B6 (CZ)
Title: Zásobník nábojů pro střelné zbraně
Inventor: ŠIMEK VLADIMÍR
IPC: F41A9/64
Filed: 2017-11-22
Abstract: Zásobník nábojů (4) pro střelné zbraně pro více typů nábojů (4) s různou ráží je tvořen tělesem (1) zásobníku, ve kterém je pohyblivě upraven podavač (2) nábojů (4) opatřený pružinou (3), přičemž na vnitřní stěně (6) zásobníku jsou upraveny minimálně dvě dvojice protilehlých vodicích žeber, a to zadních vodicích žeber (a) a středních vodicích žeber (b). V tělese (1) zásobníku je na vnitřní stěně (6) zásobníku uspořádána před zadními vodicími žebry (a) a středními vodicími žebry (b) alespoň jedna dvojice protilehlých předních vodicích žeber (c), přičemž výška předních vodicích žeber (c) je větší než výška zadních vodicích žeber (a) a středních vodicích žeber (b).
Patent CZ-308162-B6 (CZ)
Title: Process for preparing a nanostructured superhydrophobic surface layer with a radially symmetric wettability gradient
Inventor: KRATOCHVÍL JIŘÍ
IPC: B82Y30/00
Filed: 2019-03-13
Abstract: The solution is a device (1) for preparing a nanostructured superhydrophobic coating (8) on a carrier substrate (6) with a radially symmetrical wettability gradient comprising at least one deposition chamber (2) for receiving the carrier substrate (6) and at least one nanoparticle source (3) for generating a nanoparticle beam (7) into the deposition chamber (2), at least one ECWR electrode (4) is between the nanoparticle source (3) and the deposition chamber (2) so that a negative electric field generated by the ECWR electrode (4) ) surrounds the nanoparticle beam (7), and in the deposition chamber (3) there is at least one negatively charged control electrode (5) arranged in projection of the nanoparticle beam (7) on the surface of the carrier substrate (6).
Patent CZ-309281-B6 (CZ)
Title: Galvanic cell
Inventor: MUŠÁLEK OTO
IPC: H01M6/14
Filed: 2021-05-17
Abstract: A galvanic cell including at least two electrodes, each in the form of a collector (1), which is formed by a flat body made of electrically conductive material. The collectors (1) are parallel and the space between them is divided by a flat separator (2), while between each collector (1) and the separator (2) there is at least one layer of active mass (3) containing an electrolyte. The active mass (3) is stored in the flexible peripheral frame guardrails (4), inserted between each separator (2) and collector (1). The guard (4) rests closely on one side to the surface of the marginal part of the collector (1) and on the opposite side to the surface of the marginal part of the separator (2).
Patent SK-285266-B6 (SK)
Title: Particle-shaped, expandable styrol polymers and method for the production thereof
Inventor: EBERSTALLER ROMAN
IPC: C08K3/00
Filed: 2000-01-20
Abstract: Particle-shaped expandable styrol polymers that can be processed to hard foamed material having a low density and a fine cellular structure and containing a foaming agent and aluminium in the form of particles, which are reflecting infrared rays and this styrol polymer particles are homogeneously distributed in particle of styrol polymer. Method for the production styrol polymers by polymerization styrol and foaming agent in reactor, where during this polymerisation process,the aluminium articles are added in the polystyrol carrier to the limit 6 % weight, in which general participation has a laminar shape in the form of the concentrate.
Patent CZ-288471-B6 (CZ)
Title: Process for producing glass-making grindstones
Inventor: NETOPIL JIRI ING
IPC: C08J5/14
Filed: 2000-04-19
Abstract: Stirred up mixture with cement binding agent is put into a mold where it is treated by vibrations with frequency ranging from 180 to 250 Hz and amplitude level within the range of 0.05 to 0.40 mm for a period of escape of free air from the mixture being treated. After finish of vibrations and levelling of surface the product is kept for a period of 24 hours in the mold and subsequently it is removed from the mold and put for a period of at least 27 days in a water bath with temperature ranging from 18 to 25 degC.
Patent CZ-299522-B6 (CZ)
Title: Process for preparing lactone group-containing diol
Inventor: TAOKA NAOAKI
IPC: C07D319/06
Filed: 1999-12-10
Abstract: In the present invention, there is disclosed a process for preparing a lactone group-containing diol of the general formula 3, which diol can be further used for synthesis of simvastatin finding a great use as an HMG-CoA reductase inhibitor, wherein the preparation process comprises deacylation of lovastatin with an inorganic base and a secondary or tertiary alcohol to obtain a triol containing a carboxyl group, from which the required diol is obtained by acylation and lactonization thereof.
Patent CZ-302236-B6 (CZ)
Title: Feeding device for sewing machine
Inventor: KADOWAKI SHINJIROU
IPC: D05B55/14
Filed: 2000-09-05
Abstract: In the present invention, there is disclosed a feeding device (52) for a sewing machine (51) comprising a needle feed driving force transmission mechanism (90) and a lower feed driving force transmission mechanism (87). The needle feed driving force transmission mechanism (90) includes an eccentric cam (63) for horizontal movement of a needle bar (80), a crankshaft (64), an output shaft (65) and a connecting arm (76). The eccentric cam (63) is connected to an upper shaft (60). One end of the crankshaft (64) is connected to the eccentric cam (63), and the second end of the crankshaft (64) is connected to one end of the output shaft (65) for driving motion. The connecting arm (76) is fixed at its one end to the second end of the output shaft (65). The lower feed driving force transmission mechanism (87) is provided with a second connecting rod (84) and a driving arm (85). One end of the second connecting rod (84) is connected to one of the other ends of the connecting arm (76) and the drive shaft of the needle bar (80). The driving arm (85) is connected via its upper end to the second end of the second connecting rod (84). A lower part of the driving arm (85) is connected to the lower feed driving shaft (59).
Patent CZ-294760-B6 (CZ)
Title: Valve, particularly thermostatic valve for heating systems
Inventor: WIWE JORGEN SEINDAL
IPC: F16K31/64
Filed: 2000-11-16
Abstract: The present invention relates to a valve, particularly thermostatic valve for heating systems wherein the valve is provided with a housing (150, 170), a valve seat (153, 173), a closing piece (154, 176) that is operated by means of a pin (156, 178) penetrating a sealing arrangement (157, 179), and a connecting arrangement (166, 167, 185, 186) suited for the fixing of an operating adapter. The connecting arrangement has a bearing surface (162, 182) at a first distance (A, B) from the pin (156, 178) free end, and a corresponding first clamping surface (161, 181). In order to fasten at least one second type of the operating adapter, there are arranged in combination: a) an internal connecting member (158, 172) supporting the sealing arrangement (157, 179), having a first clamping surface (161, 181) performed thereon and being adjustable by a predetermined path (D) in the direction of the pin (156, 178) axis, and b) an external connecting member (163, 183) encompassing said internal connecting member (158, 172), having outside thread (165, 184) and with a bearing surface (162, 182) performed thereon, and being also adjustable by a predetermined path (E) in the direction of the pin (156, 178) axis but oppositely relative to said internal connecting member (158, 172).
Patent CZ-292473-B6 (CZ)
Title: Process for producing packaging materials exhibiting antimicrobial properties
Inventor: DOBIAS JAROSLAV DOC ING CSC
IPC: B65D81/24
Filed: 2000-11-16
Abstract: The present invention relates to a process for producing packaging materials exhibiting antimicrobial properties wherein the packaging materials containing at least one group of amino, carboxylic, aldehyde and isocyanide group are brought into contact with at least one antimicrobial agent containing each at least one group being selected from the group comprising carboxylic, amino or aldehyde groups whereby at least one such group of at least one antimicrobial agent reacts with at least one group being selected from the group comprising   carboxylic, amino, aldehyde and isocyanide groups present on the surface of the packaging material in the presence of substances containing at least one group being selected from the group comprising amino, carboxylic, aldehyde and isocyanide groups that is absent on the packaging material surface to thereby retaining the antimicrobial agent on the packaging material surface.
Patent CZ-295367-B6 (CZ)
Title: Chucking head
Inventor: ROHM GUNTER HORST
IPC: B23B31/16
Filed: 2000-11-21
Abstract: In the present invention, there is disclosed a chucking head (1) having at least two chuck jaws consisting of one draw jaw (9) and one base jaw (8) adjustable in radial guide holders (3), set by a clamping rod (6) which slides axially through the chuck body (2). The two jaws (8, 9) are provided with grooves (10) to come flush together, with a centering unit with reversible distortion as a hollow roller fitted into the base jaw (8).
Patent CZ-294708-B6 (CZ)
Title: Hydraulic turbine with non-bladed rotor
Inventor: SEDLACEK MIROSLAV ING CSC
IPC: F03B5/00
Filed: 2001-09-13
Abstract: In the present invention, there is disclosed a hydraulic turbine with a non-bladed rotor and comprising a liquid tank (1) provided with an inflow opening, and at least one stator (3). At least one non-bladed rotor (5) formed by a body of rotational shape is mounted on a holding-down device (4) within the stator (3). A distributor (2) formed by an enclosed chamber having an inlet opening (6) and an outlet opening (7) is arranged between the liquid tank (1) and the stator (3). Said inlet opening (6) is connected through the mediation of a supply pipe (8) with said liquid tank (1) while said outlet opening (7) is turned toward the rotor (5), whereby the area of the inlet opening (6) is less than that one of the outlet opening (7).