baber/WOPTO huggingface dataset:
Patent CZ-9902436-A3 (CZ)
Title: Quinolines and quinozalines, process and intermediates for their preparation, their use and pharmaceutical preparations based thereon
Inventor: FOX DAVID NATHAN ABRAHAM
IPC: C07D413/04
Filed: 1998-01-06
Abstract: Compounds of formula (I), wherein R<1> represents C1-4 alkoxy optionally substituted by one or more fluorine atoms; R<2> represents H or C1-6 alkoxy optionally substituted by one or more fluorine atoms; R<3> represents a 5- or 6-membered heterocyclic ring, the ring being optionally substituted; R<4> represents a 4-, 5-, 6- or 7-membered heterocyclic ring, the ring being optionally fused to a benzene ring or a 5- or 6-membered heterocyclic ring, the ring system as a whole being optionally substituted; X represents CH or N; and L is absent, or represents a cyclic group of formula (Ia), or represents a chain of formula (Ib), and pharmaceutically acceptable salts thereof; are useful in therapy, in particular in the treatment of benign prostatic hyperplasia.
Patent CZ-261999-A3 (CZ)
Inventor: JOHANSSON LEIF
IPC: H02G1/14
Filed: 1998-02-02
Abstract: Řešeníse týká provedení spojek kabelu, zvláště spojek ohnutých
kabelů. Spojka kabelu zahrnuje dvakabely/6,7,18,19,45,46/ a
spojovací spojku /9,16,43/umístěnou mezi kabely. Provedeníje
charakteristicetím, že zahrnuje opěru/1, 15,40,41/, unístčnou
nad spojkou tak, žedíly/6,7,9,16,18,19,43,45,46/ tvořící
spojku zůstávají vůči sobě nepohyblivé, a dále tím, že zahrnuje
alespoňjeden spojovací prvek /11,12,21,22,50,51/, ktetý
ptužně cpěru ke kabelu připojuje, kdyje tento spojovací prvek
schopnýabsorbovat změny rozměrů kabelu, způsobené tepelnou
roztažností asmštěním Řešeníse rovněž týká otáčivá»
elektrická» stroje, ktaý zahrnuje statcr s vinutímprotaženým
štětbinani ve statoru, dále zahrnuje rotor, přičemžtento stroj
zahrnuje popsaná provedeníspojky kabelu.
Patent CZ-310799-A3 (CZ)
Title: Edible spray emulsion packaged in pressure vessel
Inventor: MEIJER MARGARETHE JENNIE
IPC: A23L9/20
Filed: 1999-03-31
Abstract: A description is given of an edible fat emulsion, packed in a pressurized container, and a method for producing it. The fat constituents come from different sources, the particle size distributions of the various fat constituents being selected in such a manner that, optionally after suitable processing, they substantially correspond to one another, in order to form a stable product.
Patent CZ-340898-A3 (CZ)
Title: Compound, process of its preparation and pharmaceutical composition containing thereof
Inventor: SANDERSON PHILIP E
IPC: C07D241/20
Filed: 1997-04-18
Abstract: Compounds of the invention are useful in inhibiting thrombin and associated thrombotic occlusions having structure (a), for example (b).
Patent CZ-345696-A3 (CZ)
Title: Cable coupling
Inventor: BOGG WALTER
IPC: H02G15/113
Filed: 1995-05-04
Abstract: Described is a cable coupling box (1) consisting of two casing halves (2 and 3) sealed together round the edges by means of seals (10, 11). The seals (10, 11) end near cable lead-ins (4) in the coupling box (1), leading in to a splice joint inside the coupling box (1). In order to seal the two casing halves (2 and 3) together, they are held together by means of screws so that the seals (10 and 11), fitted in grooves, provide a seal round the edge of the coupling box (1). Fitted in the lead-ins (4) are sealing rings (20) whose outside surfaces rest against the end surfaces (14) of the seals (10, 11). The inside surfaces of the sealing rings (20) rest against the surface of the cable inserted in the lead-in. In addition, pressure elements (25) are screwed into the lead-ins (4), elastically deforming each sealing ring (20) so that the outside surface of the sealing ring (20) is pressed against the inside surface (15) of the lead-in (4), including the end surface (14) of the seal (10, 11), and its inside surface is pressed against the surface of the cable.
Patent CZ-348499-A3 (CZ)
Title: Process for preparing ice-cream
Inventor: BEER RICHARD
IPC: A23B7/08
Filed: 1997-07-23
Abstract: The invention relates to a method for the production of ice cream containing soft and/or pasty chip-shaped added ingredients, such as fruit or chocolate. The invention also relates to the ice cream products obtained by this method.
Patent CZ-348896-A3 (CZ)
Inventor: BRDLIK MIROSLAV
IPC: C02F3/00
Filed: 1996-11-28
Abstract: Gravitační čistírna odpadních vod je tvořena
nádrží /1/, která obsahuje osazený dílec pro
zachycení plovoucích nečistot /4/, na němž je
vytvořen vertikální průtok /5/ do usazovacího
prostoru /8/ ve štěrbinovém žlabu a vytvořeny
plynotěsné závěsy /13, 14/ a na protilehlé
straně /10/ jsou vytvořeny plynotěsné
závěsy /15, 16/. Nádrž /1/ dále obsahuje
usazovací prostor ve štěrbinovém žlabu vytvořený
osazením desek /11, 12/ do plynotěsných
závěsů /13, 14, 15, 16/. Odtokový
žlab /21/ z usazovacího prostoru /8/je zaústěný
do první komory filtru /22/. Osazený
ponořený komorový anaerobní filtr je vyústěný
do odtoku /31/ a vytvořený ze sestavy
komor /22, 23, 24/, opatřených nornou stěnou
/25/ a zarážkami /27/ pro osazení vysunovatelného
roštu /28/ s filtrační náplní z
plastických hmot /30 /.
Patent CZ-9903587-A3 (CZ)
Inventor: MUELLER GERMAR
IPC: H02K3/40
Filed: 1998-10-08
Abstract: Elektrický stroj je dimenzován pro napětí až 6,6 kV. Výroba
jeho vinutí je z výrobně technického hlediskajednodušší než
výroba šablonového vinutí s plochými dráty. Používá se
vsypávaného vinutí (1) z kulatého drátu, lakovaného nebo
holého. Drát včetně vývodů je překryté obandážován pásem
slídové fólie. Každá cívka leží vždy ve dvou polootevřených
drážkách (2) aje rozdělena do alespoň dvou nad sebou
ležících, za sebou zapojených a vzájemně mezivrstvou (5)
izolovaných dílčích cívek (4,6). Vyložení (3) drážky a fázová
izolace se provádí plochým izolantem, obsahujícím slídu.
Patent LV-5042-A3 (LV)
Inventor: WALS LOURENS
IPC: C07D211/04
Filed: 1992-11-27
Abstract: Novel  alpha , alpha -diaryl-4-aryl-4-hydroxy-1-piperidinebutanamide, N-oxides of formula <CHEM>  wherein  R is hydrogen or methyl;  Ar<1> and Ar<2> are, each independently, phenyl or halophenyl;  Alk is -CH2-CH2- or -CH2-CH(CH3)-; R<1> and R<2> are, each independently, hydrogen, C1-6alkyl, phenylmethyl or 2-propenyl or R<1> and R<2> combined with the nitrogen atom bearing said R<1> and R<2> may form a pyrrolidinyl, piperidinyl, C1-6alkylpipridinyl, 4-morpholinyl or 2,6-di(C1-6alkyl)-4-morpholinyl radical; Ar<3> is phenyl being optionally substituted with up to 3 substituents selected from the group consisting of C1-6alkyl, C1-6alkyloxy, halo and trifluoromethyl; the pharmaceutically acceptable acid addition salts and possible stereochemically isomeric forms thereof, which compounds are anti-diarrheal agents; pharmaceutical compositions containing such compounds as an active ingredient and methods of preparing said compounds and pharmaceutical compositions.
Patent SK-114893-A3 (SK)
Title: Process for the production of a seasoning sauce from bread
Inventor: MULLER RUDI
IPC: A23L7/25
Filed: 1993-10-21
Abstract: A process for the production of a seasoning sauce in which an enzyme-containing, fungus-covered substrate comprising divided bread of wheat gluten. The substrate is mashed with salt water, the mash is subjected to a three stage fermentation and then clarified by squeezing pasteuring and filtration.
Patent SK-122197-A3 (SK)
Title: Frontal superstructure member of undercarriage and deformation element on vehicles, in particular rail vehicles
Inventor: ERDMANN MARC
IPC: B61D15/06
Filed: 1997-09-10
Abstract: With the using up of the stroke of the coupling (10), the failure of a wear element (11), and the receding of the coupling into the coupling sleeve, load is directed through two deformation elements (1) side-mounted on the underframe (4). The deformation elements are attached to the underframe by a mounting plate (18). The enclosed casing (14) is built onto the underframe and has only one opening (15) for the coupling.
Patent SK-122398-A3 (SK)
Title: Substituted sulfonic acid n-[(aminoiminomethyl)phenylalkyl]- -azaheterocycloamide compounds
Inventor: EWING WILLIAM R
IPC: C07D223/10
Filed: 1997-12-01
Abstract: The compounds of formula (I) exhibit useful pharmacological activity and accordingly are incorporated into pharmaceutical compositions and used in the treatment of patients suffering from certain medical disorders. More specifically, they are inhibitors of the activity of Factor Xa. The present invention is directed to compounds of formula (I), compositions containing compounds of formula (I), and their use, which are for treating a patient suffering from, or subject to, physiological condition which can be ameliorated by the administration of an inhibitor of the activity of Factor Xa.
Patent SK-150797-A3 (SK)
Title: Antifungal composition
Inventor: MEINGASSNER JOSEF G
IPC: A61P31/04
Filed: 1996-05-10
Abstract: PCT No. PCT/EP96/02022 Sec. 371 Date Nov. 12, 1997 Sec. 102(e) Date Nov. 12, 1997 PCT Filed May 10, 1996 PCT Pub. No. WO96/35423 PCT Pub. Date Nov. 14, 1996Use of a combination of the squalene epoxidase inhibitor terbinafine and an azole 14-alpha-methyldemethylase inhibitor (fluconazole or itraconazole) in mycotic infections caused by azole-resistant fungal strains, and corresponding pharmaceutical compositions, process and method.
Patent SK-152015-A3 (SK)
Inventor: TREBUNA PETER
IPC: G08G1/087
Filed: 2015-03-13
Abstract: Systém automatického vytvárania trasy voľného prejazdu pre vozidlá rýchleho zásahu pozostáva z centralizovaného systému (7) riadenia svetelných križovatiek, ktorý je diaľkovo prepojený so svetelnými križovatkami (3) a zároveň je prepojený aj s navigačným systémom (5) na automatické vyhľadanie trasy (2) z východiskového miesta (1) do miesta zásahu (4), pričom navigačný systém (5) je prepojený s aktívnym navigačným systémom (8) vo vozidle rýchleho zásahu prostredníctvom vidiaceho systému (6) dispečingu.
Patent SK-162299-A3 (SK)
Title: Process for preparing a reactive pharmaceutical product for the detection of gastrointestinal disorder caused by bacteria in the gastrointestinal superior tract
Inventor: MARSHALL BARRY J
IPC: A61K47/26
Filed: 1998-05-28
Abstract: The invention relates to the diagnosis in a human or lower animal subject of a gastrointestinal disorder of the upper gastrointestinal tract caused by bacteria using a breath test. In one aspect the invention provides a process for the preparation of a reactive pharmaceutical product for the detection of gastrointestinal disorder caused by bacteria in the superior gastrointestinal tract, characterized by the preparation of a dense powdered vehicle or granules of sugar, or granules of Nu-pareil seeds, of a specific diameter between 0.12 to 3.0 mm and soluble in gastric fluids; dispersing in or coating on the vehicle a micro dose of <14>C-urea; and coating or encapsulating the resulting blend with an inert gelatin substance that dissolves rapidly, thereby obtaining a capsule, wherein the density of the vehicle is such that it allows deposition of the isotope contained in the capsule onto the gastrointestinal tract mucosa. In another aspect the invention provides a pharmaceutical product for breath tests for the detection of gastrointestinal disorder that comprises an isotope of <14>C-urea dispersed in or coated on a dense powdered or granulated vehicle of sugar, Nu-pareil seeds, and the resulting blend being coated with or enclosed in inert gelatin substance that dissolves rapidly in the presence of gastric juice, wherein the vehicle has a density sufficient to allow the capsule contents to be deposited onto the gastrointestinal tract mucosa, and wherein the granules have a diameter of between 0.12 to 3.0 mm.
Patent SK-184299-A3 (SK)
Title: A paste container
Inventor: AMBERG GUNTHER
IPC: D06F39/02
Filed: 1998-06-15
Abstract: The invention relates to a paste container with a follower plate tightly sealing the open side of the container. A multiblade mixing propeller is fitted to the follower plate in such a way that it can be rotated, a short distance beneath the follower plate, around an axle (5) which juts through the middle of the plate. The paste container includes a removal device with an external drive mechanism with which paste can be removed from the container through an opening in the follower plate. The agitator blades and the removal device have the same drive mechanism. The paste container is used in particular for receiving thixotropic pastes.
Patent SK-719789-A3 (SK)
Title: Xantine derivatives, method for producing thereof, pharmaceutical composition containing them and their use
Inventor: KUFNER-MUHL ULRIKE
IPC: C07H19/04
Filed: 1989-12-19
Abstract: Xanthines of formula (I) and their optical isomers and acid-addn. salts are new: R1 = 1-6C alkyl, 3-4C alkenyl or 3-4C alkynyl; R2 = 1-6C alkyl, 3-4C alkenyl, 3-4C alkynyl or opt. substd. benzyl; R3 = (a) C-bonded satd. or unsatd. 5- to 7-membered heterocyclyl contg. one or more O and/or S atoms, opt. substd. by 1-6C alkyl, oxo, CHO, CH2OR4, CH2OR7, COOR4 or CONR5R6; where furyl and thienyl gps. are opt. also substd. and tetrahydrofuryl gps. are opt. also substd; (b) 4-8C cycloalkenyl opt. substd. by 2-4C alkenyl; (c) a 4-8C cycloalkanone or cycloalkanol gp. opt. alpha-substd. by 2-6C alkenyl, 2-6C alkynyl, opt. substd. benzyl, CH2OR4, CH2COOR7 or CH2CH2CN; (d) 3-8C cycloalkyl opt. substd. by 1-6C alkyl, =CH2, =NNHAr, =NNHR, =NOH, OCONHAr, OCONHR, OR4, OR7, (CH2)xCOOR4, (CH2)xNR4R4, (CH2)xCONR5R6, (CH2)xOR4, (CH2)xOR7 or =CHA; (e) 3-8C cycloalkyl gem-substd. by OH and 1-6C alkyl, vinyl, allyl or opt. substd. phenyl or (1-4C alkyl)phenyl; (f) 3-8C cycloalkyl gem-substd. by ORa and ORb, or (g) 3,4-methylenedioxyphenyl, 3,4-ethylenedioxyphenyl, 2-fluorenyl, 9-fluorenyl or a bicyclic gp., e.g. of formula (i)-(iii). Ar = opt. substd. aryl; R = 1-6C alkyl, x = 0-4; A = COOR4, CN, CONR5,R6, CH=CHCOOR4, CH=CHCONR5R6, CH2OR4 or CH2OR7; Ra and Rb = 1-4C alkyl, or Ra+Rb = 2-3C alkylene opt. substd. by 1 or 2 of 1-5C alkyl, 2-6C alkoxycarbonyl and 1-5C hydroxyalkyl; R4 = H, 1-13C alkyl, 3-13C alkenyl, propargyl, trityl or opt. substd. 3-6C cycloalkyl or benzyl; R5 = H, 1-6C alkyl or opt. substd. 3-6C cycloalkyl; R6 = H, 1-6C alkyl, opt. substd. benzyl, (CH2)nNR5R5, ((CH2)nO(CH2)mO)k(CH2)nNR5R5, (CH2)nQ(CH2)nNR5R5, or C-bonded piperidinyl opt. substd. ; or NR5R6 is a 5- to 7-membered ring opt. contg. another heteroatom and opt. substd. ; n = 2-8; m = 2-6; k = 0 or 1; Q = piperazine-1,4-diyl opt. substd. ; R7 = acyl derived from a natural amino acid, 2-14C alkanoyl, methyloxyacetyl, camphanoyl, abietoyl, 4-aminobutyryl, opt. substd. benzoyl or COB1; B1 = opt. substd.
Patent SK-872020-A3 (SK)
Inventor: CÍSAR MIROSLAV
IPC: A63B21/062
Filed: 2020-07-16
Abstract: Zariadenie na uchopovanie bremien pozostáva zo základnej konštrukcie (2), ku ktorej sú pripevnené vodiace tyče (3), na ktorých sú umiestnené cez otvory (27) bremená (1), pričom každé jedno bremeno (1) obsahuje zahĺbenie (11) a drážku na vodiaci element (13). Zariadenie ďalej obsahuje držiak (8) motora, na ktorom je upevnený prvý motor (7), ku ktorému je pomocou spojky (14) pripevnená závitová tyč (6), na ktorej sa pohybuje guľôčková matica (5) pripevnená k rúrke (4) obsahujúcej drážku na kábel (15). Na konci rúrky (4) je upevnený druhý motor (16) uložený v medzikuse motora (17), spojený prostredníctvom hriadeľa (25) s hlavicou (12). Hlavica (12) pozostáva zo spodného krytu (19) a vrchného krytu (20), ktoré sú k sebe priskrutkované a fixované kolíkmi (24). Cez hlavicu (12) prechádza hriadeľ (25), ku ktorému (25) sú pripevnené pomocou čapov (22) ramená (23), a tie sú pomocou čapov (22) pripevnené k výsuvným elementom (21), pričom každý výsuvný element (21) je umiestnený na aretačnom čape (28).
Patent BE-1003825-A3 (BE)
Title: Dispositif telephonique numerique sans fil.
Inventor: KAEWELL JOHN DAVID JR
IPC: H04M1/72505
Filed: 1990-02-16
Granted: 1992-06-23
Abstract: Un dispositif téléphonique numérique sans fil contient au moins une station de base émulée (96) plus une ou plusieurs stations d'abonné (90), la station de base émulée comportant une station semblable à la station d'abonné mais ayant la possibilité d'initialiser un processus de synchronisation, d'où il résulte qu'elle peut affecter des secteurs à la station d'abonné dans la configuration de trame d'un signal d'amplitude en surveillant les fronts positifs du signal.
Patent BE-1007590-A3 (BE)
Title: Videosignaalverwerkingsschakeling.
Inventor: VAN ROOIJ JOHANNES H J M
IPC: H04N9/68
Filed: 1993-10-01
Granted: 1995-08-16
Abstract: In een videosignaalverwerkingsschakeling wordt een adaptieve signaalcompressie gerealiseerd door de kleurverzadiging door vermenigvuldiging van kleurverschilsignalen (R-Y,G-Y) met eenzelfde correctiefactor dusdanig bij te regelen dat kleursignaalwaarden (R,G,B) beneden hun respectievelijke maximaal toegestane waarden blijven zonder dat daarbij tevens de luminantie (Y) begrensd wordt.
Patent WO-0178320-A3 (WO)
Title: Systeme et procede notification destine a un dispositif mobile de transmission de donnees
Inventor: MAJOR HARRY
IPC: H04M1/72436
Filed: 2001-04-10
Abstract: L'invention concerne un système et un procédé de notification destinés à un dispositif mobile de transmission de données. Un logiciel client fonctionnant au niveau dudit dispositif mobile permet de gérer et d'exécuter des systèmes de notification (« unités de notification ») pouvant être sélectionnés par l'utilisateur, en réponse à des éléments de donnée transmis au dispositif mobile depuis un système hôte via un réseau de communication. L'utilisateur configure l'unité de notification afin d'exécuter certaines notifications sonores, visuelles et/ou tactiles en réponse à certains types de messages reçus par le dispositif mobile.
Patent WO-0219064-A3 (WO)
Title: Procede et systeme permettant d'empecher des modifications non souhaitees de donnees et de programmes stockes dans un systeme informatique
Inventor: BUCKLEY CONLETH
IPC: G06F21/56
Filed: 2001-08-31
Abstract: La présente invention concerne un procédé et un système permettant d'empêcher des modifications non souhaitées de données et de programmes stockés dans un système informatique. Le système décrit dans cette invention utilise un réseau de portes programmable par l'utilisateur afin de commander l'accès à un dispositif de stockage. L'utilisateur peut accéder à différents profils par l'intermédiaire de mots de passe. Les différents profils constituent différents paramètres de commande permettant d'accéder au dispositif de stockage. Le réseau de portes peut être reprogrammé de temps en temps à l'aide de fichiers électroniques téléchargeables. La sécurité est assurée pendant le téléchargement grâce à des clés et à des techniques de chiffrement.
Patent WO-03097690-A3 (WO)
Title: Derives de la pth resistants aux proteases de la peau
Inventor: KRISHNA G PERI
IPC: C07K14/635
Filed: 2003-05-16
Abstract: L'invention concerne des analogues, résistants aux protéases, de dérivés biologiquement actifs de la parathormone humaine (PTH). Ces analogues sont destinés à être utilisés dans des préparations thérapeutiques servant à traiter divers états pathologiques associés à une perte osseuse ou à un risque de perte osseuse. Les analogues spécifiés sont des hPTH(1-34) et hPTH(1-31). Plus particulièrement, l'invention concerne des analogues de la PTH, résistants aux protéases, qui sont conçus pour l'administration transdermique.
Patent CH-623713G-A3 (CH)
IPC: G04C21/02
Filed: 1976-12-23
Abstract: An electro-acoustic transducer of electromagnetic type is composed of an exciting part having a magnetic core wound with an exciting coil, a vibrating plate provided opposite to the magnetic core at an interval and a ferromagnetic thin plate mounted to the vibrating plate. The thin plate is provided on the surface of the vibrating plate on the side of the magnetic core, so that the thin plate is not exposed to the open air. Furthermore, the thin plate is connected to the vibrating plate at plural points more than three or at a part with some area. Such connection restrains undesirable vibration of the thin plate.
Patent WO-8402493-A3 (WO)
Title: Plant for the continuous and automated manufacturing of agglomerated, sintered, vulcanized and pressed articles
Inventor: MILISAVLJEVIC MILORAD
IPC: B28B21/90
Filed: 1983-12-14
Abstract: The plant for the continuous and automated manufacturing of articles obtained by compression of products comprises a supply means arranged in a central cylinder (6) and secured to the plant frame consisting of a central cylinder (1) and fixed platforms (2, 4, 5, 7). The plant comprises one or a plurality of working units mounted on the frame. Each working unit is divided into sectors, each of them comprising a press-forming means consisting of an auxiliary press mounted in the cylinder (3) and a main press arranged within the cylinder (95), and/or processing means and/or unmolding or discharging means. The working unit comprises a carrousel driven by a central shaft (226) to displace the mold elements (222, 231, 232) and the frames (213) to support the mold elements from one working unit sector to the next sector. Said plant is characterized by reduced overall dimensions, a high productivity and may be adapted to the manufacturing of various articles.
Patent CZ-2001225-A3 (CZ)
Inventor: BOETTCHER HENNING
IPC: C07D295/18
Filed: 1999-07-08
Abstract: Derivát bifenylu obecného vzorce I, kde znamená R -C(=NH)-
NH2, -C(=NH)-NHA3, -C(=NH)-NHAc, -C(=NH)-
NHSO2CH3, R2, -CO-NH-Z-R3, nebo -CO-R1; X -CONH-,
SOjNH-, -NHCO- nebo -NHSO2-; Y CH nebo N; A1 atom H,
C].6alkyl, přičemž několik atomů H může být nahrazeno
, 's atomy F, SO2CH3 nebo SC>2CF3; A2 atom H nebo Ci^alkyl;
A3, A4 vždy na sobě nezávisle C).6alkyl, A5, A6 vždy na sobě
nezávisle atom H nebo (CH2)DCH3; Q atom H nebo skupina
OA1, R1 4-A5-piperazin-l-yl, 4-A5-homopiperazinyl, 1-
pyrrolidinyl, který je substituován jednou skupinou R4 nebo -
Z-R4, piperidinyl, který je substituován jednou skupinou R4
nebo Z-R4, nebo znamená N-A5-pyrrolidinylamino, N-A5-
piperidinylamino, N-A5-pyrrolidinyl-Z-amino nebo N-Apiperidinyl-Z-amino,
skupinu -N(A6)(ZR3) nebo NA6A7; R2 5-
methyl-l,3,4-oxadiazol-2-yl nebo 5-methyl-l,2,4-oxa-diazol3-yI;
R3, R4 vždy na sobě nezávisle NHA5, N(A5)2, 4-
morfolinyl, 1-pyrrolidinyl nebo 1 piperidinyl; Z Ci.ealkylen; n
0 nebo 1; p 0,1 nebo 2 jeho racemáty a enantiomery ajeho
fyziologicky přijatelné soli a solváty jsou jakožto serotoninové
(5-HZib/id) antagonisty vhodné pro výrobu farmaceutických
prostředků k ošetřování a k předcházení poruch centrálního
nervového systému, zvláště depresí, všeobecné úzkosti,
nutkavého chování a bulimie.
Patent CZ-2002323-A3 (CZ)
Title: Substituted oxoazaheterocyclyl compounds and pharmaceutical preparations in which they are comprised
Inventor: EWING WILLIAM R
IPC: A61K31/517
Filed: 2000-07-26
Abstract: This invention is directed to oxoazaheterocyclyl compounds which inhibit Factor Xa, to oxoazaheterocyclyl compounds which inhibit both Factor Xa and Factor IIa, to pharmaceutical compositions comprising these compounds, to intermediates useful for preparing these compounds, to a method of directly inhibiting Factor Xa and to a method of simultaneously directly inhibiting Factor Xa and Factor IIa.