baber/WOPTO huggingface dataset:
Patent JP-H09512258-A (JP)
Title: 複素環式ベンゾニトリル類
IPC: C07D209/48
Filed: 1995-04-18
Abstract: (57)【要約】
本発明は一般式（Ｉ）
 式中、Ｒ 1 、Ｒ 2 、Ｒ 3 及びＨｅｔは本文に記載される意味を有する、の新規な複素環式ベンゾニトリルに関する。本発明は、更に、その製造に対する新規な方法及び新規な中間体生成物並びにその除草剤としての使用にも関する。
Patent JP-2000506578-A (JP)
Title: 地下資源の探査装置
IPC: G01N3/40
Filed: 1997-12-17
Abstract: (57)【要約】
本発明は、その最も下方に工具を支持する一連のロッドによる地下資源探査装置に関し、該ロッド（７）は、互いに関節で繋がれ、リールの周りに巻き付けられており、塔（１０）での交互の直線状の運動及び連続的にロッドを降ろすための回転運動により作動し、それから、それらをリール（１）の上に再び巻き付ける。
Patent JP-H09512193-A (JP)
IPC: A61B7/02
Filed: 1995-04-21
Abstract: The headset comprises left and right elongate ear pieces having respective first ends to receive ear tips and respective, interconnected second ends. Each ear piece includes a one-piece elongate body made of flexible and resilient material and curved outwardly to skirt round the user's head when the ear tips are applied to a user's ears. The elongate body is formed with a first length of smaller cross section and therefore of greater flexibility proximate the second end of the corresponding ear piece and with a second length of lower flexibility situated between that first length and the corresponding ear tip. Bending of the elongate bodies when the ear pieces are spread apart is therefore concentrated in the first lengths and pressure applied to the user's ears by the ear tips is mainly produced by the bent first lengths and transmitted to the ear tips through the second lengths of lower flexibility. The elongate ear pieces have respective second end sections assembled laterally adjacent to each other, and a threaded sleeve is mounted on these laterally adjacent second end sections and is rotated and displaced longitudinally to adjust the level of pressure applied to the user's ears by the ear tips.
Patent JP-H09512682-A (JP)
Title: 連続交流電源を使用したゲート駆動回路
IPC: H03K17/567
Filed: 1995-04-17
Abstract: (57)【要約】
電源スイッチング装置（４７）用のゲート駆動回路は四個の整流器（３８、４０、４２、４４）を有するＨブリッジ整流装置を備え、第一、第二の整流器（３８、４０）の各陽極が互いに中間点で第三、第四の整流器（４２、４４）の陰極に結合される。この中間点は電源スイッチング装置（４７）のゲート端子に結合される。連続交流波形発生器（１０）が、出力選択制御論理回路（１２）に結合され、出力選択論理回路（１２）は、電源スイッチング装置（４７）をオンにするために、第三、第四整流器（４２、４４）の各陽極に二次側が結合された第一変圧器（３２ａ、３２ｂ）に、あるいは電源スイッチング装置（４７）をオフにするために、第一、第二整流器（３８、４０）の各陰極に二次側が結合された第二変圧器（３４ａ、３４ｂ）に連続交流波形を印加する。
Patent JP-H10505958-A (JP)
Title: 自動車用の制御装置
IPC: B60R16/02
Filed: 1996-03-08
Abstract: (57)【要約】
受容体内に差込み体を収容するための構成である。差込み体１内で電気回路装置が支持体２上に配置され、支持体２の少なくとも２つの縁区域が、差込み体１から突出し、受容体９の案内溝１６，１７内に係合している。エアバッグ制御装置に使用可能である。
Patent JP-2000506034-A (JP)
Title: 電気療法およびその装置
IPC: A61N1/39
Filed: 1996-03-01
Abstract: (57)【要約】
本発明は、細動除去およびカルジオバージョンのための電気療法パルスの伝達において、患者ごとのインピーダンス差を自動的に補償する外部細動除去器および細動除去の方法を提供する。好適な実施形態では、細動除去器は患者に置いた電極を通して放電し、２相の電圧または電流パルスを供給することができるエネルギ源を備えている。本発明の一局面では、第１および第２の位相の持続時間および最初の第１の位相の振幅は、予め設定した値である。本発明の第２の局面では、パルスの第１の位相の持続時間は、パルスの第１の位相の振幅が閾値よりも小さければ、所定の第１の位相の持続時間の終わりに高インピーダンスの患者で発生するように延長することができる。本発明の第３の局面では、第１の位相は、低いインピーダンスから平均のインピーダンスの患者で発生することがあるように、第１の位相の振幅が閾値より低くなるか、または第１の位相の持続時間が閾時間値に到達するか、いずれか先に生ずるとき終了する。伝達される２相パルスを変えるというこの方法および装置は、それにより伝えられる電気治療パルスの性格を変えることにより患者のインピーダンスの差を補償し、より小さい一層効率的なあまり高価でない細動除去器を生ずる。
Patent JP-H11503329-A (JP)
Title: グリコシド結合の酵素的合成
IPC: C12P19/18
Filed: 1996-04-10
Abstract: (57)【要約】
本発明はグリコシド結合の形成方法を提供する。これらの方法は、式：ＮｅｕＡｃα（２→３）Ｇａｌβ（１→４）（Ｆｕｃα１→３）ＧｌｃＮ（Ｒ’）β（１→３）Ｇａｌβ−ＯＲの化合物の製造に有効である。
Patent JP-H11506476-A (JP)
IPC: C08F36/04
Filed: 1996-04-17
Abstract: A high yield of three armed radial anionic polymers is produced by the process of coupling metal terminated anionic polymers with a trialkoxysilane having a silicon-hydrogen bond, preferably trimethoxysilane. The metal terminated anionic polymer is preferably produced by initiating polymerization with a protected functional initiator which is readily converted to terminal hydroxyl groups or derivatives thereof for use in adhesives, sealants, and coatings.
Patent JP-2000507274-A (JP)
IPC: A61K39/385
Filed: 1998-01-20
Abstract: The present invention is concerned with a fragment of IgA1-protease having 40 to 200 amino acid residues and comprising at least 40 amino acids of an amino acid sequence as shown in SEQ ID NO:1, beginning with the amino acid in any one of positions 1 to 5 and ending with an amino acid in any one of positions 40 to 104 or a homologous sequence, its use as a carrier for a conjugate, particularly in combination with a polysaccharide, and a process for producing the peptide as well as vaccines comprising said peptide.
Patent JP-2001510569-A (JP)
Title: 血漿容積の測定
IPC: G01N33/68
Filed: 1998-02-05
Abstract: (57)【要約】
患者の血液流内に第一の低投与量の低分子量高分子物質を導入し、該物質の分布容積を決定することから成る毛管漏れの存在または発生を確認する方法。前記分布容積をここでは見かけの分布容積と呼ぶ。ここで決定される分布容積の値は毛管壁を通っての溢出による影響をうけるばかりでなく、小さい分子が毛管壁の細孔または受容体結合部位に結合することによる影響をも受ける。この結合は溢出よりもずっと大きな速度で起り、毛管漏れ発生の重要な指標となる。前記過程を、高投与量の高分子量高分子物質によって繰り返し、もう一つの分布容積を決定する。この分布容積をここでは時間循環血漿容積と呼ぶ。前記二つの分布容積の値を比較して、毛管漏れの存在または発生を確認する。
Patent JP-2001512475-A (JP)
Title: 抗病原性合成ペプチドおよびこれらを含む組成物
IPC: A61P31/04
Filed: 1998-02-19
Abstract: (57)【要約】
ペプチド、束になったペプチドの複合体、ペプチドまたはランダムペプチドコポリマーの混合物から選択される非溶血性細胞溶解性物質は、病原性細胞（体内では自然に存在せず、かつ病原性生物および悪性細胞を含む細胞）に対する細胞溶解活性を有すること；および非溶血性であること、すなわち、赤血球に対する細胞溶解作用がないこと、により表される選択的細胞溶解活性を有する。ペプチドは、パーダキシンやメリチンのような天然のペプチドおよびこれらの断片の環状誘導体（ここで、Ｌ−アミノ酸残基は対応するＤ−アミノ酸残基により置換されるか、または種々の比の、少なくとも１つの正に荷電したアミノ酸と少なくとも１つの疎水性アミノ酸からなる線状ペプチドのジアステレオ異性体よりなり、そして、少なくとも１つのアミノ酸残基がＤ−アミノ酸である）でもよい。非溶血性細胞溶解性物質を含む薬剤組成物は、細菌、真菌、ウイルス、マイコプラズマおよび原生動物感染症を含む病原体により引き起こされるいくつかの疾患の治療、および癌の治療のために使用することができる。
Patent JP-2001522232-A (JP)
IPC: C07K14/12
Filed: 1998-03-10
Abstract: Disclosed are compositions comprising a recombinant nucleic acid vector including a nucleotide sequence encoding a syncytium-inducing polypeptide expressible on a eukaryotic cell surface, and a host cell containing the recombinant vector and expressing the syncytium inducing polypeptide on its cell surface, the vectors and resultant host cells expressing the syncytium inducing polypeptide being useful for selective elimination of unwanted cells.
Patent JP-H11510981-A (JP)
Title: 通信装置のための自己較正装置および方法
IPC: H04W24/00
Filed: 1997-04-17
Abstract: (57)【要約】
通信装置７０の適応アンテナ・アレイ素子８６のビーム・パターンに関する重みづけ率を提供する較正ネットワーク１１０〜１３０，１８０，１８２は、狭帯域チャネルを、比較的短いビット当たりのパルス速度と、狭帯域信号チャネルのノイズ閾値の電力レベルより相対的に低い電力レベルとを有する疑似乱数シーケンス（ＰＲＮＳ）を含む共通広帯域信号で変調および復調することにより、自己較正される。受信経路１１６および送信経路１１４のうち選択された相補経路によりＰＲＮＳ内に導入される誤差は、ＰＲＮＳに導入される誤差に基づいて較正ネットワークの処理利得を計算することにより決定される。次に、収束アルゴリズム１３０を適応して、選択された経路のコンポーネント１１２〜１１８により導入される振幅および位相変動を解明して、次にこの変動を補正するために適切な修正率１２６を決定することにより、これらの振幅および位相変動が第３図の通信装置７０により軽減される。
Patent JP-2001504571-A (JP)
Title: プッシュプルチェーン駆動型ドア作動装置
IPC: F16H19/06
Filed: 1998-05-12
Abstract: (57)【要約】
プッシュプルチェーン型ガレージドア用作動装置が、駆動モジュール及びキャリジ組立体に連結されたプッシュプルチェーンの細長い案内レールを有し、キャリジ組立体は、案内レールに取り付けられている。チェーンは、全体として矩形の板状成形プラスチック支持部材に取り付けられたスプロケットに係合でき、支持部材には、蛇行状遊びチェーン収納スロットが設けられている。支持部材は、収納スロットを覆うと共に駆動モジュールを支持するプレス加工金属フレーム板に解除自在に連結されている。支持部材の底壁は、駆動モータに連結された直角形減速駆動ユニットを支持し、駆動モータは、支持部材に設けられた一体ボスにより形成されているクレードル内に保持されている。モータ及びこのための始動用コンデンサは、着脱自在な保持ストラップによりボスのそれぞれ対応したクレードル部分内に保持されている。制御回路板が、支持部材の下側に取り付けられ、作動機構の２部品構成シュラウドがフレーム板に解除自在に固定されている。
Patent JP-H06316475-A (JP)
Title: Method for coating of fiber-reinforced ceramic composite material and its coated composite material
Inventor: HAABAATO DEIITORITSUCHI
IPC: C04B41/88
Filed: 1989-11-15
Abstract: PURPOSE: To enhance the adhesive strength of a coating and to prevent the occurrence of cracks, etc., by etching the surface of a fiber reinforced ceramic composite material to be coated with an etchant and coating the etched surface with a coating compsn.  
     CONSTITUTION: A matrix material selected from carbon, silicon carbide, silicon nitride, etc., is combined with fibers such as carbon fibers or silicon carbide fibers to produce a fiber reinforced ceramic composite material. The surface of the composite material is etched with an etchant at a suitable temp. for an effective time to expose the fibers in the composite material to the surface while maintaining the bound flawless state. An active gas such gas chlorine, hydrogen or hydrogen fluoride is suitable for use as the etchant and the suitable etching depth is about 0.5-10 mils. The etched surface of the composite material is coated with a coating compsn. contg. a ceramic, a metal, etc. 
     COPYRIGHT: (C)1994,JPO
Patent MX-154023-A (MX)
Inventor: GONZALEZ EDUARDO BARNETCHE
IPC: E21B10/24
Filed: 1981-04-23
Abstract: An automatic depth compensating system is provided for controlling the pressure in a volume such as the interior of a rotary drill bit in response to pressure changes in the environment adjacent to the volume. The system comprises at least one pressure compensating device positioned between the volume and the environment for changing the pressure in the volume in response to pressure changes in the environment. The system further includes a pressure surge compensating device which is positioned between the volume and the environment for compensating for positive and negative pressure surges when the pressure in the volume changes relative to the pressure in the environment. The pressure compensating devices each comprises differential piston devices having a spring for biasing the differential piston and the pressure surge compensating device comprises a cylinder, a piston positioned in the cylinder and forming a chamber therein and first and second check valves for opening in response to predetermined pressure differentials between the environment and the interior of the volume.
Patent NZ-201953-A (NZ)
Title: Combating nematodes by applying macrolides to foliage
Inventor: CLAYTON J
IPC: A01N43/90
Filed: 1982-09-20
Abstract: Soil dwelling nematode pests of growing plants are combated and controlled by applying to the aerially exposed foliar parts of the plants an effective amount of an insecticidally active macrolide substance, such as, for example, an avermectin or milbemycin.
Patent NZ-210309-A (NZ)
Title: Blot-overlay immunoassay using colloidal metals
Inventor: MOEREMANS M K J J
IPC: G01N33/58
Filed: 1984-11-23
Abstract: A method for detecting and/or determining an agglomerate formed by the reaction between a specific binding agent and the corresponding acceptor substance according to the general methodology of blot overlay assays by using colloidal metal particles labelled components which may be visualized as a coloured signal at the surface of the blotting medium characteristic for the colloidal metal particles used or quantitatively determined following art-known spectopho- tometric procedures such as densitometry.
Patent NZ-217679-A (NZ)
Title: Antibiotic fermentates from kibdelosporangium aridum largum and compositions
Inventor: DINGERDISSEN J J
IPC: A23K20/195
Filed: 1986-09-24
Abstract: A novel subspecies of Kibdelosporangium aridum, subsp. largum (SK&F-AAD-609) produces AAD-216 antibiotics and AAD-609 antibiotics, the AAD-609 antibiotics differing from the AAD-216 antibiotics in presence of glucosamine in the glycolipid radical in place of amino glucuronic acid.
Patent NZ-222310-A (NZ)
Title: N,n-disubstituted aminopropionic acids and their use as emulsifying agents, wetting agents and surfactants in cleaning agents and for waterproofing leather and skins
Inventor: STOCKHAYSEN DOLF
IPC: C07C275/16
Filed: 1987-10-27
Abstract: A process for the preparation of compounds of the formula I <IMAGE> in which R1 denotes a saturated or unsaturated alkyl radical or alkoxyalkyl radical having 1 - 22 carbon atoms, preferably 12 - 18 carbon atoms, R2 denotes an alkyl radical having 1 - 18 carbon atoms, a saturated or unsaturated carboxyalkyl radical having 3 - 4 carbon atoms, a carboxyphenyl radical or a carboxyl radical (-COOH),  R3 denotes hydrogen or CH3 and X denotes hydrogen, alkali metal, alkaline earth metal, ammonium, alkylammonium or alkanolammonium  and  A represents <2bL>C=O, <2bL>SO2, <IMAGE> or an alkylene radical having 0-3 C atoms, which is characterised in that alkylamines of the formula R1-NH2, in which R1 has the meaning described above, are added to (meth)acrylic acid and the resulting N-alkylaminopropionic acids are reacted with carboxylic anhydrides, carbonyl chlorides, sulphonyl chlorides, isocyanates, halocarboxylic acids or (meth)acrylic acids and are then optionally at least partially neutralised. Novel N-alkyl-N-(2-carboxyethyl)sulphonamides and N-alkyl-N-(2-carboxyethyl)ureas are additionally described.
Patent NZ-226490-A (NZ)
Title: Bar code verification requires two bar codes presented simultaneously
Inventor: MAY LANCE
IPC: G07D7/00
Filed: 1988-10-13
Abstract: The Invention relates to a method and machine for use in coupon verification. At least two juxtaposed coupons, each having a bar code printed or formed thereon, are passed substantially simultaneously through or relative to bar code reader means provided in a machine for verifying coupons. The machine additionally includes holding and dispensing means and a programmed processor. In use, at least two juxtaposed coupons are passed substantially simultaneously, into and through the bar code reader means of the machine. On the juxtaposed coupons being accepted and verified by the bar code reader means, matter is caused to be dispensed from the holding and dispensing means of the machine.
Patent NZ-230193-A (NZ)
Title: A radioiodinated benzodiazepine derivative and brain imaging composition
Inventor: CARMANN HEINZ
IPC: C07C59/00
Filed: 1989-08-03
Abstract: Radioiodinated 5,6-dihydro-5-methyl-6-oxo-4H-imidazo [1,5-a][1.4]benzodiazepine derivatives and the use thereof as brain-imaging agents are described.
Patent NZ-238121-A (NZ)
Title: Packaging items using cavitated and apertured plates
Inventor: BOYHAN LAURENCE ANTHONY
IPC: B65B5/06
Filed: 1991-05-10
Abstract: Apparatus and process in which one plate, or several accurately superimposed plates (10, 16) carry items (12, 18) to be packaged. On inversion of the plates, items either fall directly into the voids of a partitioned box (26) or fall into individual packages held by a plate, which packaged items are then ejected by pushrods, etc. into a single box. A plate may have cut-away portions (e.g. V-shaped grooves) which receive upstanding edges or partition walls of a box to accurately register box with plate (and contents) and nest the box into the plate to achieve configuration-accurate inversion of the items to be packaged.
Patent NZ-238223-A (NZ)
Title: Human bile salt-stimulated lipase related proteins and their production and use
Inventor: BJURSELL GUNNAR KARL
IPC: A61K8/37
Filed: 1991-05-22
Abstract: Bile-salt stimulated lipase (BSSL) may comprise amino acids 1-722, 1-535, 1-278, 1-341, 1-409, 1-474, 279-341, 279-409, 279-474, 342-409, 342-474 or 536-722 of the sequence given at the end. Also claimed are (1) a functionally equivalent variant or mutant of BSSL; (2) a DNA sequence (I) encloding BSSL, comprising nucleotides 151-2316, 151-1755, 151-985, 151-1172, 151-1376, 151-1574, 986-1172, 986-1376, 986-1574, 1173-1376 or 1173-1574 of the sequence given in the specification; (3) a vector comprising (I); and (4) a host organism transformed with the vector of (3); and (5) an infant food formulation comprising BSSL. Pref. BSSL may be in combination with one or more of the direct repeats of the sequence given in the specification. BSSL may posses Met as additional N-terminal amino acid.
Patent NZ-240009-A (NZ)
Title: Process for preparation of carboxylic acid anhydrides by reaction of co with a carboxylic acid ester or alkyl ether
Inventor: BEEVOR ROBERT GEORGE
IPC: C07C51/09
Filed: 1991-09-30
Abstract: The solubility and stability of rhodium catalysts in rhodium-catalysed carbonylation of alkyl esters or alkyl ethers under substantially anhydrous conditions to produce carboxylic acid anhydrides is improved by the use of co-promoters selected from the group:  1,3-dialkyl-4-methylimidazolium iodide;  1,3-dialkyl-4-ethylimidazolium iodide;  1,3-dialkyl-4-n-propylimidazolium iodide;  1,3-dialkyl-4-isopropylimidazolium iodide;  1,3-dialkyl-4-n-butylimidazolium iodide  1,3-dialkyl-4-sec-butylimidazolium iodide  1,3-dialkyl-4-tert-butylimidazolium iodide; 1,3-dialkyl-2,4,5-trimethylimidazolium iodide and mixtures thereof where the alkyl groups are independently C1 to C20 alkyl.
Patent NZ-243784-A (NZ)
Title: N-(isoquinolin-5-ylsulphonyl) azacycloalkane derivatives and pharmaceutical compositions
Inventor: PEGLION JEAN-LOUIS
IPC: A61K31/42
Filed: 1992-07-30
Abstract: Compounds of formula (I):  (* CHEMICAL STRUCTURE *) (I) (* CHEMICAL STRUCTURE *)  wherein R1, R2, U, X, Y, Z, n, m, p and r are as defined in the description, and medicaments containing the same.
Patent NZ-244773-A (NZ)
Title: Carboxamide substituted isoquinoline derivatives and pharmaceutical compositions
Inventor: THOMPSON WAYNE J
IPC: C12N9/99
Filed: 1992-10-16
Abstract: Oligopeptide analogs are described. These compounds are useful in the inhibition of HIV protease, the prevention or treatment of infection by HIV and the treatment of AIDS, either as compounds, pharmaceutically acceptable salts, pharmaceutical composition ingredients, whether or not in combination with other antivirals, immunomodulators, antibiotics or vaccines. Methods of treating AIDS and methods of preventing or treating infection by HIV are also described.
Patent NZ-253623-A (NZ)
Title: Plastic blow moulded bottle with hollow legs around base: tapered, curved ribs between legs
Inventor: YOUNG WILLIAM C
IPC: B65D1/02
Filed: 1993-06-09
Abstract: A plastic blow molded container (10) is disclosed as including a freestanding base structure (20) that is constructed with a plurality of alternating hollow legs 22 and curved ribs (34), and a hub (41) from which the legs and ribs extend radially with a construction that provides good stability against tipping as well as the capability of withstanding internal pressure. Each rib (34) has an outer upper end (36) with a circumferential width Wu and an inner lower end (38) with a circumferential width Wl that is greater than the circumferential width Wu of the upper rib end so the lower rib end is capable of resisting stress cracking. An intermediate rib portion (40) of a curved shape tapers between the ends with an included angle B in the range of about 1 degrees to 8 degrees and preferably about 2 degrees.
Patent NZ-283259-A (NZ)
Title: Multiple compartment package suitable for two different articles of food
Inventor: PERRY MICHAEL R
IPC: B65D51/28
Filed: 1995-03-22
Abstract: A multiple compartment package for use in the packaging of foodstuff articles includes a first compartment portion, a second compartment portion, and a retaining mechanism for retaining the first compartment portion in close relation to the second compartment portion.
Patent NZ-285442-A (NZ)
Title: Corticotropin-releasing factor antagonists comprising pyridines, pyrimidines, purinoses, pyrrolopyrimidinones and pyrrolopyridinone compounds
Inventor: CHEN YUHPYNG L
IPC: A61P11/00
Filed: 1995-06-06
Abstract: PCT No. PCT/IB95/00439 Sec. 371 Date Dec. 6, 1996 Sec. 102(e) Date Dec. 6, 1996 PCT Filed Jun. 6, 1995 PCT Pub. No. WO95/33750 PCT Pub. Date Dec. 14, 1995Corticotropin-releasing factor (CRF) antagonists having formulae (I), (II) or (III) wherein the dashed lines, A, B, Y, Z, G, R3, R4, R5, R6, R16 and R17 are as defined in the description, and processes for preparing them. These compounds and their pharmaceutically acceptable salts are useful in the treatment of CNS and stress-related disorders.
Patent NZ-293626-A (NZ)
Title: The fungus gliocladium catenulatum and use in controlling plant diseases
Inventor: TAHVONEN RISTO TAPIO
IPC: A01N63/30
Filed: 1995-09-29
Abstract: PCT No. PCT/FI95/00536 Sec. 371 Date Jul. 14, 1997 Sec. 102(e) Date Jul. 14, 1997 PCT Filed Sep. 29, 1995 PCT Pub. No. WO96/10626 PCT Pub. Date Apr. 11, 1996The present invention relates to biological control of plant diseases and concerns new Gliocladium catenulatum fungi and their use for controlling fungal infections in plants. The invention concerns also compositions comprising new strains of Gliocladium catenulatum and their use to said purpose.
Patent NZ-295410-A (NZ)
Title: Recycling fibre products by deinking with lanolin (or derivative) as collector chemical
Inventor: BENTLEY THOMAS RICHARD
IPC: C11D1/04
Filed: 1995-11-13
Abstract: PCT No. PCT/GB95/02651 Sec. 371 Date May 7, 1997 Sec. 102(e) Date May 7, 1997 PCT Filed Nov. 13, 1995 PCT Pub. No. WO96/15315 PCT Pub. Date May 23, 1996A process for recycling fiber products employs an aqueous deinking medium containing an effective amount of a collector chemical. The collector chemical comprises a surface active agent which is or can be derived from lanolin. Alkoxylated lanolin derivatives are preferred.
Patent NZ-299659-A (NZ)
Title: Amidine derivatives; compounds, preparation and medicaments with anti-thrombin activity
Inventor: OH YEONG SOO
IPC: C07C311/42
Filed: 1996-10-29
Abstract: The present invention relates to a novel selective thrombin inhibitor having the following formula (I), which is also effective by oral administration: <CHEM>  in which   R<1>   represents acetyl substituted with aryl or aryloxy, or represents sulfonyl substituted with substituted or unsubstituted aryl or N-containing heterocyclic group, X   represents a group of formula <CHEM>   R<2> and R<3>   independently of one another represent hydrogen; cycloalkyl substituted or unsubstituted with carboxyl or alkoxycarbonyl; arylalkyloxy; hydroxy; or lower alkyl substi tuted or unsubstituted with carboxyl, alkoxycarbonyl or hydroxy, or R<2> and R<3>   together with nitrogen atom to which they are attached can form a piperidine group substituted with carboxyl or alkoxycarbonyl, R<4>   represents hydrogen, lower alkyl or lower alkoxy, R<5>   represents alkanesulfonyl; alkoxycarbonyl; alkylcarbonyl; formyl; lower alkyl; aryl substituted or unsubstituted with alkoxy or haloalkyl; or hydroxy-substituted lower alkyl,  and R<6> and R<7>   independently of one another represent hydrogen, lower alkyl or amino, and to a process for preparation thereof and a pharmaceutical composition for thrombin inhibition which comprises the compound of formula (I) as an active ingredient.
Patent NZ-331463-A (NZ)
Title: Use of rapamycin derivatives in vasculopathies and xenotransplantation
Inventor: SCHULER WALTER
IPC: A61P9/00
Filed: 1997-03-26
Abstract: 40-O-(2-hydroxy)ethyl-rapamycin is used to prevent or treat neointimal proliferation and thickening, restenosis and /or vascular occlusion following vascular injury or for preventing or combating manifestation of chronic rejection in a recipient of organ or tissue allotransplant or xenograft transplant.
Patent NZ-332157-A (NZ)
Title: Fire extinguishing system, liquid inert gas mixed with extinguishing agent
Inventor: RUSSWURM MANFRED
IPC: A62C35/02
Filed: 1997-03-26
Abstract: In a fire extinguishing system, a liquid inert gas, such as liquid CO2, is mixed with the fire extinguishing agent in mixer 3 to produce a two phase bubble flow.  The inert gas is introduced at a higher pressure than that of the extinguishing agent.  The flow of liquid gas may be controlled by signals from sensor 6 which monitors the progress of the fire.
Patent NZ-336296-A (NZ)
Title: A road barrier
Inventor: WILLIAMS JAMES RICHARD
IPC: A01K3/00
Filed: 1999-06-15
Abstract: A barrier (32) to prevent passage of vehicles or animals includes two posts (13) that contain or support mechanisms to raise or lower the barrier (32) vertically as required.  When not active, the actual barrier (5) is lowered into a channel inside a frame (7) across the road (3) for protection from wheels or passing vehicles.  A portable road barrier has a ramp on each side of the frame so that it may (if lowered) be driven over when in place.  One version of barrier is a single horizontal rod, beam, and rope or chain (5) raised or lowered from the posts (13) at both ends.   Dependent chains or straps (21-23) and further horizontal beams (15) may be added to form a more effective though collapsible (when lowered) stock barrier.  An actuator mechanism raises and lowers the barrier assembly to a height sufficient to cause the road barrier to become closed, or lower the barrier back into the surface of the road.  The device may also for example be used to prevent "ram raids" in shops.  The barrier serves as a lockable gate and can be controlled by an (remotely controlled) electronic lock.