baber/WOPTO huggingface dataset:
Patent UA-117533-C2 (UA)
Title: Спосіб інгібування грибів роду candida у хворих на вульвовагініт на тлі віл-інфекції
IPC: A61P31/10
Filed: 2017-02-02
Abstract: Винахід належить до медицини, а саме до дерматології, і може бути використаний для інгібування грибів роду Candida у хворих на вульвовагініт на тлі ВІЛ-інфекції. Спосіб інгібування грибів роду Candida у хворих на вульвовагініт на тлі ВІЛ-інфекції включає при гострому та хронічному вагінальному кандидозі в стадії загострення призначення флуконазолу 100 мг однократно або клотримазолу 500 мг однократно на першій лінії лікування, на другій лінії лікування, що передбачає призначення кетоконазолу 200 мг 2 рази на добу курсом 3 дні або кетоконазолу 200 мг 1 раз на добу курсом 7 днів, як підтримуючу терапію - призначення ністатину 2000-4000 мг 2 рази на добу курсом 10 діб або флуконазолу 50-200 мг 1 раз на добу тривало, крім того, пацієнту під контролем біологічних зразків за показниками мікроскопічних досліджень та бакпосіву на середовище Сабуро при гострому та хронічному перебігу процесу, в тому числі в стадії загострення, додатково призначають зовнішній засіб цидипол у вигляді кожнодобових аплікацій інтравагінально курсом до нормалізації контрольованих вимірів.
Patent UA-127176-C2 (UA)
Title: Herbicide-tolerant maize plant dbn9858, and nucleotide sequence and method for detecting same
Inventor: KANG YUEJING
Filed: 2016-04-28
Abstract: Provided are a nucleotide sequence for detecting a maize event DBN9858 existing in a biological sample, and a detecting method therefor.
Patent UA-126272-C2 (UA)
Title: Anti-tau antibodies and methods of use
Inventor: ADOLFSSON OSKAR
Filed: 2016-06-02
Abstract: The invention provides anti-Tau antibodies and methods of using the same.
Patent UA-127447-C2 (UA)
Title: Methods for transfecting plants and for reducing random integration events
Inventor: TIJSTERMAN MARCEL
Filed: 2017-03-23
Abstract: The present disclosure provides methods for transfecting plants and for expressing RNA or polypeptide molecules in plants. In particular, plants having reduced POLQ expression and/or activity are transfected in order to reduce random integration events. The disclosure further provides transfected plants and plant progeny produced by the methods disclosed herein.
Patent UA-126026-C2 (UA)
Title: Поліетергуанідин як регулятор росту пшениці
Filed: 2019-07-17
Abstract: Поліетергуанідин загальної формули, дe R=CH2CH2OCH2CH2, n=20, як регулятор росту пшениці.
Patent UA-123810-C2 (UA)
Title: Potassium channel modulators
Inventor: AMRUTKAR DIPAK VASANTRAO
Filed: 2018-01-23
Abstract: Provided are compounds and pharmaceutically acceptable salts thereof, which are useful for treating a variety of diseases, disorders or conditions, associated with potassium channels.
Patent UA-124999-C2 (UA)
Title: Основа для супозиторіїв
Filed: 2020-07-15
Abstract: Основа для супозиторіїв містить твердий жир, воду очищену, емульгатор, натрію альгінат, кальцію стеарат, консерванти - ніпагін та ніпазол.
Patent UA-69866-C2 (UA)
Title: A method for producing a high-clean germanium
Inventor: TELIN VLADYSLAV VOLODYMYROVYCH
IPC: C22B41/00
Filed: 2003-12-11
Abstract: A method for producing a high-clean germanium involves charging germanium dioxide into the reactor, reducing thereof with hydrogen, alloying, directed crystallization and zone purification at multiplepassages of melted zone through the obtained ingot. After charging germanium dioxide to the reactor it is dried in the nitrogen atmosphere, with subsequent roasting in the nitrogen atmosphere. As germanium dioxide it is used the hydrated germanium dioxide. The invention allows to increase germanium output with simultaneous reducing expenses for producing thereof.
Patent UA-72840-C2 (UA)
Title: Method for repairing a liner section of a pipeline
Inventor: RUDNYK ANATOLII ANDRIIOVYCH
IPC: F16L55/175
Filed: 2004-07-07
Abstract: A method for repairing a linear section of a pipeline is in cleaning the section of the pipeline being repaired, with installation on it of a split muff, centering and fixation of its parts, with installation of circular elastic gaskets between the outer surface of the pipeline and the inner surface of the muff at its ends, installation at two ends of the muff of flanges connected with tightening, with filling the space between the pipeline and the inner surface of the muff with glue composition, with simultaneous air pressing out fro the cavity being filled. At that, after fixation of the parts of the split muff, to the pipeline, at both sides of the muff, one first winds one turn of flexible hose, this is pressed and placed between the pipeline and the inner surface of the muff; at that the hoses are placed in parallel arrangement with respect to the outer ends of the muff, and the ends of the hoses are let through the tightening in the body of the muff. After that one installed the flanges to the pipeline at two sides of the muss. After that, to the hoses, under pressure, liquid is supplied, or gaseous substance pressing the hoses between the pipeline and the inner surface of the muff. The flanges are tightened in long direction by means of bracing wire. After that, by means of high-pressure syringe, one fills the space between the pipeline and the inner surface of the muff with glue self-curing composition, hen the pressure is increased up to the maximally possible calculated value and soaked till the end of the curing process.
Patent UA-78555-C2 (UA)
Title: Method for immunizing plants against bacterioses and compounds used
IPC: A01N37/36
Filed: 2003-03-10
Abstract: The invention relates to a method for immunizing plants against bacterioses, characterized in that the plants, the soil, or seeds are treated with an effective quantity of a compound of formula (I), wherein: X represents halogen, C1-C4 alkyl or trifluoromethyl; m is equal to 0 or 1; Q represents C (=CH-CH3) -COOCH3, C (=CH-OCH3)-COOCH3, C(=CH-OCH3) -CONHCH3, C(=N-OCH3)-COOCH3, C(=N-OCH3) -CONHCH3 or N(-OCH3)-COOCH3; A represents -O-B, -CH2O-B, -CH2S-B, -OCH2-B, -CH=CH-B, -C=C-B, -CH2O-N=C(R1)-B or -CH2O-N=C(R1)-C(R2)=N-OR3, whereby B represents optionally substituted phenyl, naphthyl, 5-membered or 6-membered hetary) or 5-membered or 6-membered heterocyclyl, containing one to three N atoms and/or one 0 atom or S atom or one or two 0 atoms and/or S atoms; R1 represents hydrogen, cyano, alkyl, alkyl halide, cycloalkyl, alkoxy; R2 represents optionally substituted phenyl, phenylcarbonyl, phenylsulfonyl, 5-membered or 6-membered hetaryl, 5-membered or 6-membered hetarylcarbonyl or 5-membered or 6-membered hetarylsulfonyl, and; R3 represents hydrogen, optionally substituted alkyl, alkenyl and alkynyl. This effective quantity of the compound is absorbed by the plants or seeds.
Patent UA-79788-C2 (UA)
Title: Air distributor of brake of railroad transportation means
Inventor: TAMKOV MYKOLA LEONTIOVYCH
IPC: B60T15/18
Filed: 2004-12-20
Abstract: An air distributor of the brake of railroad transportation means contains a main part, in housing of which valve chamber and main chamber are formed which are divided by a mobile partition equipped with a hollow stock with radial openings at the end. In the stock the pusher is located for interaction from one side with the valve at the end of the plunger, which has channels and sleeve, and from other side - with the valve, which interacts with the bleeder valve and separates the cavity of additional discharging from accelerating cavity with the sleeve of check valve mounted in it. The unit of the softness of action is executed with a mobile partition. In the housing of main part a mobile partition is located, which separates the equalizing cavity from the atmosphere. For increasing the reliability of operation of the air distributor at all modes of braking in the wall of hollow stock a choke opening is made for connecting of main chamber and accelerating cavity. The control cavity of the unit of softness of action is connected with the equalizing cavity in the main part of air distributor.
Patent RU-2670955-C9 (RU)
Title: Обжимной контакт
Inventor: WANG XIAFU
IPC: H01R4/20
Filed: 2015-08-05
Granted: 2018-11-21
Abstract: Изобретение относится к штекерному соединителю для высокой нагрузки. Штекерный соединитель содержит по меньшей мере один обжимной контакт (1), переход (10) между образованной из алюминия обжимной зоной (11) и образованной из меди контактной зоной (12) перенесен в цилиндрический или по меньшей мере ротационно-симметричный обжимной контакт (1). За счет этого многопроволочный провод можно обжимать с помощью обжимного контакта (1). Кроме того, в обжимной зоне (11) предусмотрены дополнительная внутренняя резьба (112) и ввинчиваемый дорн (113). Технический результат - обеспечение сравнительно не затратного присоединения алюминиевого многопроволочного провода, а также обеспечение хорошей электрической проводимости. 3 н. и 7 з.п. ф-лы, 15 ил.
Patent RU-2735485-C9 (RU)
Title: Переключаемый амортизатор
Inventor: BAUER MICHAEL
IPC: F16F7/09
Filed: 2017-05-03
Granted: 2021-01-26
Abstract: Изобретение относится к переключаемому амортизатору 1, который содержит корпус 2, имеющий продольную ось 3, плунжер 4, выполненный с возможностью перемещения вдоль упомянутой продольной оси 3, поршень 20, расположенный между упомянутыми корпусом 2 и плунжером 4, фрикционную накладку 21, расположенную на упомянутом поршне 20, и узел переключения 23, переключаемый между состоянием блокирования, в котором поршень 20 заблокирован от перемещения вдоль продольной оси 3, и состоянием свободного перемещения, в котором для поршня 20 обеспечена возможность перемещения вдоль продольной оси 3. Фрикционная накладка 21 расположена на упомянутом поршне 20 и содержит область, которой она приводится в непосредственный контакт с торцевыми поверхностями продольных ребер 16 крышки или продольных ребер 18 основания и служит в качестве ограничительного буфера. Обеспечивается создание амортизатора с улучшенными рабочими характеристиками, в частности такого, изготовление и (или) работа которого не представляли бы сложности. 19 з.п. ф-лы, 12 ил.
Patent DK-122489-D0 (DK)
Inventor: ANDERSEN ANDERS JOERGEN
IPC: C12P21/02
Filed: 1989-03-14
Abstract: Pentapeptides having the formula H-Asp-Ser-C-Pro-Arg-OH, where Asp, Ser, Pro and Arg may have L- or D-configuration, and C denotes Asp or Asn in L or D configuration, are synthesized by reacting in an aqueous medium Y2-Pro-OH, wherein Y2 is a protective group, with Arg-Ro, wherein Ro is OH or is as defined below for R1 below, to form Y2-Pro-Arg-Ro, which is deprotected, if necessary under conversion to Pro-Arg-R1, wherein R1 is an enzymatically cleavable  alpha -carboxy substituting group selected from esters, amides, anilides, hydrazides or L-amino acid esters, and thereafter reacting Y3-C(Z3)-OH with Pro-Arg-R1 to form Y3-C(Z3)-Pro-Arg-R1, which is deprotected to C-Pro-Arg-R1, and then reacting Y4-Ser-OH with C-Pro-Arg-R1 to form Y4-Ser-C-Pro-Arg-R1, which is deprotected to Ser-C-Pro-Arg-R1, and reacting Y5-Asp(Z5)-OH with Ser-C-Pro-Arg-R1 to form Y5-Asp(Z5)-Ser-C-Pro-Arg-R1, which is deprotected to the intermediate Asp-Ser-C-Pro-Arg-R1, and finally removing the group R1 with an enzyme, preferably trypsin to form Asp-Ser-C-Pro-Arg, or removing R1 from Y5-Asp(Z5)-Ser-C-Pro-Arg-R1 before deprotection to Asp-Ser-C-Pro-Arg-OH. The groups Y2, Y3, Y4, Y5, Z3 and Z5 are protective groups which apart from Y2 are removable by catalytic hydrogenation. The employed synthesis strategy based on the combination hydrogenation/enzyme, both proceeding under mild conditions, leads to the peptides, in particular HEPP, in good yield without risk of formation of  beta -aspartyl peptides and cleavage of Asp-Pro bonds.
Patent DK-360688-D0 (DK)
Inventor: FAVRE ERIC
IPC: A47G19/22
Filed: 1988-06-30
Abstract: This drinking vessel comprises a bottom (2) and a lateral wall (3), the bottom having the shape of an ellipsoid, a paraboloid or a hyperboloid. 
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Patent DK-369785-D0 (DK)
Inventor: BELKA HEINRICH
IPC: B62J7/02
Filed: 1985-08-14
Abstract: A front wheel side luggage carrier (1) for bicycles comprises a strut arrangement (4) having two struts (7, 8), which when in the position of use extend substantially vertically and approximately parallel to a plane that intersects the front axle of the bicycle at right angles, and having an upper and a lower attachment arrangement (5, 6). Via these arrangements, the side luggage carrier (1) is secured to adjacent legs of the front wheel fork (2) at two points, one of which is located near the front axle and the other is spaced apart therefrom. In order to provide a simple structure, which even under adverse conditions will not tend to vibrate during the ride and which will be largely independent of the shape of the front wheel fork (2), the two vertical struts (7, 8) are joined integrally together at their lower end by means of a connecting cross portion (11), which bears the lower attachment arrangement (6). At their upper ends, the two vertical struts (7, 8) are bent toward one another, forming two transverse bent-over portions (23, 24) in alignment with one another, which in turn are bent at their free ends, forming two support struts (27, 28), towards the lower attachment arrangement (6) on which the support struts (27, 28) are anchored. The upper attachment arrangement (5) is provided on the support struts (27, 28).
Patent DK-376685-D0 (DK)
Inventor: STEER PETER LESLIE
IPC: A61F5/448
Filed: 1985-08-19
Abstract: An ostomy appliance having two interengaging coupling elements is described. One of the elements is an annular plate which includes an engaging member formed by two ribs which diverge from each other to define a V-formation. One of the ribs has a stepped formation on its distal region. The other coupling element has an annular channel having cooperating formation adapted to engage the stepped formation, thereby connecting the coupling elements.
Patent DK-520586-D0 (DK)
Inventor: BERGSTROEM CHRISTER
IPC: B32B27/00
Filed: 1986-10-30
Abstract: The invention concerns a chemically modified ethylene copolymer having good adhesion to metals and other polar substances. The ethylene copolymer consists of ethylene alkyl-(meth)acrylate copolymer to which has been grafted an unsaturated acid or anhydride.
Patent DK-527283-D0 (DK)
Inventor: PAUST JOACHIM
IPC: C07D307/60
Filed: 1983-11-17
Abstract: Dihydro-4,4-dimethylfuran-2,3-dione is prepared by oxidation of racemic dihydro-3-hydroxy-4,4-dimethyl-2(3H)-furanone by a process in which the oxidation is carried out by gradually adding powdered calcium oxide to a solution of racemic dihydro-3-hydroxy-4,4-dimethyl-2(3H)-furanone and chlorine in the inert organic solvent.
Patent DK-558688-D0 (DK)
Inventor: RAGNARSSON GERT ANDERS
IPC: A61K45/06
Filed: 1988-10-06
Abstract: Preparation giving a controlled and extended release of both a dihydropyridine, e.g. felodipine and a  beta -adrenoreceptor antagonist, namely metoprolol as well as a method for the manufacture of the new preparation.
Patent HU-903488-D0 (HU)
Title: Preparatives containing sulfonyl-carbamide derivatives as active substance
Inventor: FOERY WERNER
IPC: C07D401/12
Filed: 1990-06-05
Abstract: N-pyridinesulphonyl-N-pyrimidinyl- and -triazinylureas of the formula I <IMAGE>  in which R1 represents hydrogen, halogen, C1-C4-alkyl, C1-C4-alkoxy, C1-C4- alkylthio, C1-C4-haloalkoxy or CF3;  R2 represents hydrogen or C1-C4-alkyl; A represents C1-C6-alkyl or C3-C6-cycloalkyl, each of which is mono- to trisubstituted by halogen, or represents C1-C4-alkyl or C3-C6- cycloalkyl, each of which is substituted by C1-C4-alkoxy, C1-C4- alkylthio, C1-C4-alkylsulphonyl, C1-C4-alkylsulphinyl, C2-C4-alkenyl, C5-C6-cycloalkenyl, amino, C1-C4-alkylamino, C1-C4-dialkylamino or C2- C4-alkynyl, it also being possible for the C2-C4-alkenyl radical and for the C5-C6-cycloalkenyl radical to be monosubstituted to trisubstituted by halogen, or represents a 4- to 6-membered saturated heterocycle which contains a hetero atom selected from amongst the group comprising O, N and SO2, or represents C1-C4-alkyl which is substituted by a 4- to 6-membered saturated heterocycle which contains a hetero atom selected from amongst the group comprising O, N and SO2; X represents C1-C3-alkyl, C1-C3-alkyl which is monosubstituted to trisubstituted by halogen, or represents C1-C3-alkoxy or C1-C3-alkoxy which is monosubstituted to trisubstituted by halogen; Y represents halogen, C1-C3-alkyl, C1-C3-alkyl which is monosubstituted to trisubstituted by halogen, or C1-C3-alkoxy, C1-C3-alkoxy which is monosubstituted to trisubstituted by halogen, or cyclopropyl, methylamino or dimethylamino; and E represents nitrogen or the methine group, and the salts of these compounds with amines, alkali metal bases or alkaline earth metal bases or with quaternary ammonium bases, have good selective herbicidal and growth-regulating properties, both pre- and post-emergence.
Patent HU-9204036-D0 (HU)
Title: Anti-coagulant preparatives
Inventor: NORDFANG OLE JUUL
IPC: A61P7/02
Filed: 1991-05-30
Abstract: For prophylaxis or treatment of coagulation disorders or cancer an extrinsic pathway inhibitor (EPI) is administered together with heparin or other mucopolysaccharide to the patient. Thereby an increase in coagulant activity is obtained as well as an increase of half-life of injected EPI in plasma.
Patent HU-9204185-D0 (HU)
Title: Automatic clutch for regulator capable to define pivot point
Inventor: LIU CHIA-HSIANG
IPC: B60W30/19
Filed: 1992-12-30
Abstract: This invention provides automatic and reliable determination of the touch point of a clutch controlled by an automatic clutch actuation controller. This invention determines the touch point while idling the engine, with the transmission in neutral and an inertial brake applied. The clutch actuation controller engages the clutch so that the measured transmission input speed matches a reference speed signal preferably between 40% and 60% of the idle speed. This reliably provides the degree of clutch engagement at a small torque matching the braking torque. When the transmission input speed is within a predetermined amount of the reference speed signal, such as 4%, this invention determines the clutch touch point corresponding to the degree of clutch engagement. This degree of clutch engagement may be a clutch position signal or a clutch pressure signal produced by an existing sensor used in the automatic clutch control. If no measured clutch engagement signal is available, this degree of clutch engagement may be the clutch engagement signal used to control the degree of clutch engagement. The touch point is set as the difference between this degree of clutch engagement for the small torque and a clutch touch point offset. <IMAGE>
Patent HU-895246-D0 (HU)
Title: New peptidase inhibitors
Inventor: BEY PHILIPPE
IPC: C07F7/10
Filed: 1989-10-06
Abstract: This invention relates to analogs of peptidase substrates in which the nitrogen atom of the scissile amide group of the substrate peptide has been replaced by a substituted malonyl moiety. The contemplated peptidase inhibitors of the foregoing enzymes are selected from the generic formula <CHEM> the hydrates, isosteres or the pharmaceutically acceptable salts thereof wherein X is <CHEM> R1 is hydrogen, an amino protecting group selected from Group K, an alpha -amino acid or a peptide comprised of a number of  alpha -amino acid building blocks, said  alpha -amino acid or peptide optionally bearing on its terminal nitrogen atom an amino protecting group selected from Group K, R2 is the "R group" residue of the  alpha -amino acid responsible for directing the inhibitor to the active site of the enzyme or is -A-SiR7R8R9, C1-10 alkyl, aralkyl or aryl with R7, R8 and R9, each being selected from C1-10, alkyl, aralkyl or aryl and A is a C1-6 alkylene, R4 is the specific R-group residue of the  alpha -amino acid for that peptidase substrate analog, R5 is an  alpha -amino acid or peptide comprised of  alpha -amino acids or is deleted,  Y is NHR3 or OR3 with R3 being H, C1-7 alkyl, benzyl or phenethyl. These analogs of the peptidase substrates provide specific enzyme inhibitors for a variety of proteases, the inhibition of which will have useful physiological consequences in a variety of disease states.
Patent NO-870117-D0 (NO)
Inventor: VANGAEVER MARC
IPC: E01C19/15
Filed: 1987-01-12
Abstract: 1. Sweeping method comprising the combined use of a mechanical brush (9) and a container (10) at the front of a motor vehicle, in which the front edge (26) of the forwardly open container (10) is arranged almost against the ground to be swept, the ground is swept by driving the brush in rotation so that the swept material is projected rearwardly through the container opening and the material in the container is removed by raising the container (10) and inclining its opening downwardly and in which the brush is moved freely and automatically away from the container so as to clear its opening when an obstacle is encountered and the brush is automatically returned to its initial position when the obstacle disappears, characterized in that, during sweeping, the brush (9) is freely and automatically lowered under the effect of gravity towards the ground adjacent to the opening of the container (10) and in that, in the removal position, when the opening of the container is inclined downwardly well above the ground, the brush is freely and automatically moved away under the effect of gravity from the front edge of the container so as to clear the container opening and the brush (9) is possibly used to help remove the granular material from the container.
Patent NO-870826-D0 (NO)
Inventor: GASSNER THEO
IPC: B25C1/18
Filed: 1987-02-27
Abstract: An explosive powder charge operated fastening member driving tool has a muzzle part which can be locked within and released and removed from the tool housing by rotational movement and axial movement relative to the housing. When the tool is not ready to be fired, a contact pressure sensor projects from the front end of the muzzle part. By pressing the sensor opposite to the firing direction it compresses a firing mechanism spring and the tool is ready to be fired. Stop elements are provided on the muzzle part and stop surfaces are located on the tool housing. When the muzzle part is in the unlocked condition, the stop elements can abut the stop surfaces and block the displacement of the contact pressure sensor preventing it from compressing the firing spring mechanism so that the driving tool cannot be placed in the ready-to-fire condition.
Patent NO-873231-D0 (NO)
Inventor: WELTER ANDRE
IPC: C07D333/36
Filed: 1987-08-03
Abstract: The present invention is related to new diselenobis benzoic acid amides of primary heterocyclic amines of the general formula I <CHEM>  wherein R<1> and R<2>, which are equal or different from another, represent hydrogen, halogen, C1-4-alkyl, C1-4-alkoxy, trifluoromethyl, nitro or, both together, methylenedioxy,  n is zero or a numeral from 1 to 4 and R<3> is a saturated or unsaturated heterocyclic residue with one or two heteroatoms in the cyclic nucleus selected from the group of nitrogen, sulphur and oxygen, said residues being unsubstituted or substituted onces or twice, equally or in different manner, by halogen, C1-2-alkyl, C1-2-alkoxy, nitro or hydroxy. processes for producing the same and pharmaceutical compositions comprising the same. The compounds of formula I are useful in the treatment of diseases which are caused by cell damage due to the increased formation of active oxygen metabolites such as liver damages, heart infarctions, infections, psoriasis or damages by radiation.