baber/WOPTO huggingface dataset:
Patent SK-284392-B6 (SK)
Title: Anthracycline analog, use thereof and pharmaceutical composition based thereon
Inventor: SCHALLY ANDREW V
IPC: A61K47/48
Filed: 1996-11-14
Abstract: Anthracycline analog represented by general formula Q14-O-R-P wherein Q has the general formula (II) wherein -R- represents a single bond or -C(O)-(CH2)n-C(O)-, n is 0-7, R' is NH2 or an aromatic, saturated 5 or 6 membered heterocyclic compounds having at least one ring nitrogen and optionally having a butadiene moiety bonded to adjacent carbon atoms of said ring to form a bicyclic system and P is H or a peptide moiety, suitably an LHRH, somatostatin or bombesin analogs, when R' is NH2 then R and P are other than H and when R and P are H, then R' is other than NH2 and its use for the manufacture of a medicament for the treatment of various tumors bearing receptors for the somatostatin analogs such as breast cancer, gastric cancer, pancreatic cancer, colorectal cancer, prostate cancer, small cell and non-small cell lung cancer, kidney carcinoma, osteosarcoma and brain tumor. Pharmaceutical composition based on the analogs.
Patent SK-280352-B6 (SK)
Title: Process of forming surfaces of holes by extrusion and device for making the same
Inventor: REGENT MIROSLAV
IPC: B21K21/08
Filed: 1992-03-17
Abstract: A raw product (3) to be moulded is accommodated into an extrusion die reduction (5). An extruder core (1) is inserted, at its lateral part (2), into the product (3). Upon applying force on a face (15) of the product (3) in the direction its longitudinal axis said product (3) is extruded via the reduction (5) with a bevel. This operation is followed by separating lateral part of the extruder core from a compressed moulded object. This separation is processed in an auxiliary appliance by applying force on an end (16) of the extruder core (1). A device for this method comprises a die, extrusion die with a punch (7), extruder core (1), extrusion die with a base (9) and an auxiliary appliance. A recess (10) made at an end part (17) of the punch (7) accommodates the extruder core (1) via the lateral part (2) thereof, during the operation. A first centring ring (11) is attached to the base (9) of the extrusion die, which ring has a clip (14) positioned therein. The clip (14) contains the reduction (5) with a bevel. A second centring ring (4) is attached on that reduction (5) inside a fastening ring (18), and, the fastening ring (18) is attached to the first centring ring (11).
Patent CS-276135-B6 (CS)
Inventor: HUCALA LUDOVIT ING
IPC: B67B7/10
Filed: 1989-03-10
Abstract: Na jednom konci tyče /11/ ja upevněná
rukovat /12/ a druhý koniec ja opatřený
bodcom /13/. Tyč /11/ ja u avojho druhého
konca opatřená dvojramenným pružným
zvleračom /14/. ktorého každé rameno ja
zakončené zahnutím /Yíf, orientovaným
smarom k tyči /11/. Dvojramenný pružný
zviarač /14/ Ja uložený otočná v otvore
/16/ tyče /11/, ktorého os Je kolmá na
tyč /11/.
Patent CZ-279296-B6 (CZ)
Inventor: KIENER ANDREAS DR
IPC: C12P17/12
Filed: 1992-08-28
Abstract: Je popsán mikrobiologický způsob výroby kyseliny  6-hydroxy-pyrazinkarboxylové a/nebo jejích solí  pomocí mikroorganismů zpracujících kyselinu  pikolinovou a/nebo její soli. Vytvořená kyselina  6-hydroxy-pyrazinkarboxylová se přitom akumuluje  v mediu a pak se izoluje.ŕ
Patent CS-277153-B6 (CS)
Inventor: HAZDRA FRANTISEK ING
IPC: H03K4/08
Filed: 1990-11-27
Abstract: Zapojení sestává ze synchronizačního tvarovaného
obvodu pro každou fázi (9.1, 9.2,
9.n) napětové soustavy, jehož výstup je
spojen s řídícím vstupem příslušného spínače
(7.1, 7.2, 7.n), kterého prvni pól je
společně s prvním pólem integračního kondenzátoru
(6.1, 6.2, 6.n) ukostřen, zatímco
druhé póly obou, tvořící zároveň jednu
z výstupních svorek (10.1, 10.2, 10.n)
jednotlivých složek referenčního signálu,
jsou současné připojeny k výstupu vlastního
proudového zdroje. Jeho podstatou jsou
výstupy proudových zdrojů, tvořených regulovatelnými
napětové proudovými převodníky
(3.1, 3.2, 3.n) jsou jednotlivé zapojeny do
vstupů (5.1, 5.2, 5.n) obvodu (5) výběru
maximální hodnoty amplitudy pilovitého
napětí, jehož výstup je přes amplitudový
demodulátor (4) zpětnovazebně zapojen do
regulátoru (2) amplitudy pilovitého napětí,
jehož výstup je spojen s řídícími vstupy
všech napětověproudových převodníků (3.1,
3.2, 3.n).
Patent CZ-297494-B6 (CZ)
Title: Apparatus for shearing at least one stream of molten glass
Inventor: DIFRANK FRANK J
IPC: C03B7/11
Filed: 1998-04-17
Abstract: The present invention relates to a parallel shear apparatus (10) for sequentially shearing each of a plurality of streams of molten glass from a glass feeder into gobs for processing into glass containers by a glass-forming machine. The apparatus (10) has first and second opposed carriages (12, 14), which are reciprocable along parallel slides (16, 18, 20) toward and away from one another, each of the carriages (12, 14) carrying one or more opposed knife elements (32a, 32b, 32c, 32d, 34a,34b, 34c, 34d), corresponding to the number of streams of molten glass, and the opposed knife elements overlap at the innermost limits of their travel to perform the shearing action. Motion of the carriages (12, 14) is actuated by a unidirectionally acting servomotor (36), which imparts oscillating motion to a bell crank (22) through a connecting rod (46). The oscillating motion of the bell crank (22) imparts simultaneous, opposed, rectilinear motion to the carriages (12, 14) through connecting rods (26, 30), wherein the rods (26, 30) are pivotally attached to the bell crank (22) at diametrically spaced apart locations. The servo motor (36) is mounted on a pivoting bracket (40) that is urged to its normal operating position by a pneumatic cylinder (44) and is spring biased (50) away from its normal operating position in the event of the apparatus (10) stoppage. The pneumatic cylinder (44) is cushioned to minimize shock loads caused by a sudden retraction of the servomotor (36) mounting bracket (40) and is adjustably mounted relative to fixed structure of the shear apparatus (10).
Patent CZ-285134-B6 (CZ)
Title: Absorption article and process for producing thereof
Inventor: RONNBERG PETER
IPC: A61F13/514
Filed: 1993-11-11
Abstract: PCT No. PCT/SE93/00964 Sec. 371 Date Aug. 1, 1995 Sec. 102(e) Date Aug. 1, 1995 PCT Filed Nov. 11, 1993 PCT Pub. No. WO94/10952 PCT Pub. Date May 26, 1994An absorbent article, particularly a diaper, has a central absorbent unit (1) which is comprised of an elongated absorbent body (2) enclosed between a liquid-permeable inner casing sheet (3) which lies proximal to the wearer in use, and a liquid-impermeable, outer casing sheet (4) which lies distal from the wearer in use. The absorbent unit is provided along its longitudinal edges (9) with liquid-impermeable folds (6) which are upstanding from the inner casing sheet and which form side-leakage barriers. The article has a side-flap (18) on each side of the absorbent unit (1). The side-flaps (18), optionally with associated edge (21, 23), are produced in the form of rectangular strips (10) completely separated from the absorbent unit (1) and are thereafter jointed thereto. A longitudinally extending edge-part (13) of each strip (10) is suitably folded double and the backwardly fold part (19) is joined to the outer casing sheet (3a, 4b or 4) of the absorbent unit (1)along a curved fastening line (21). When the aper is to be used, the side-flaps (18) are pulled-out laterally, the length of this extension, and therewith the width of the resulting side-flaps (18), being dependent on the curved shape of the fastening line (21). It is therewith possible to produce a curved contour (16) of the diaper for conforming to the wearer's legs with side-flaps (18) which originally have straight edges (11) The material from which the side-flaps (18) are made can be chosen quite independently of the inner and the outer casing sheets (3, 4), so as to avoid irritation of the wearer's skin while still fitting closely to the wearer's legs.
Patent CZ-287560-B6 (CZ)
Title: Process for taking off fibrous material from working cylinder in textile machines and apparatus for making the same
Inventor: RYBICKA JOSEF
IPC: D01G15/46
Filed: 1997-05-07
Abstract: When taking off fibrous material (2) from a worker roller (1) the fibrous material (2) fibers being taken off therefrom are maintained separated from fibers of the fibrous material (2) being just transferred by the transfer roller ot a take-off roller to which they are resiliently forced after transfer is done. The apparatus for making the process comprises a take-off flexible sheet (4) reaching in the space between the worker roller (1) and the transfer roller (3) and fitting close to the transfer roller (3).
Patent CZ-284995-B6 (CZ)
Title: Use of substituted cyclohexane derivatives
Inventor: HEMMERLE HORST DR
IPC: C07C69/65
Filed: 1993-09-08
Abstract: Esters of cyclohexane derivatives of the formula I <IMAGE>  in which A-B, R<3>, R<4>, R<5>, Y and Z have the stated meanings, for use as inhibitors of the glucose-6-phosphatase system in the liver of mammals are described. The compounds are suitable for producing pharmaceutical products.
Patent CZ-294817-B6 (CZ)
Title: Movable wall
Inventor: KORDES HERBERT
IPC: E04B2/82
Filed: 1996-09-17
Abstract: The present invention relates to a movable wall comprising individual door and/or wall elements mounted in a suspended manner, the individual elements being both movable in a stationary hollow guide strip (1) attached to the ceiling (41) and provided with bifurcation and branches. The individual door and/or wall elements are not guided in the floor (3) region and are provided with a profiled foot strip (5) with a locking device (6) arranged therein. When at least two door and/or wall elements get into mutual contact said locking device locks them to one another and in the floor (3), too. Inside the locking device (6) there is performed a recess (20) with an actuating plate (22) for conversion of horizontal direction of a lifter (11) movement to vertical direction of a locking pin (21) movement arranged therein. In the actuating plate (22) there is performed a skew recess (28), such as a through hole, communicating with a guide pin (12) fastened in the locking pin (21) and sliding in said a through hole (13) made in the locking device (6) fundamental body (7).
Patent CZ-290711-B6 (CZ)
Title: 1-Arylcycloalkylsulfides, -sulfoxides and -sulfones, process of their preparation, pharmaceutical preparations in which these compounds are comprised and their use
Inventor: HARRIS PAUL JOHN
IPC: A61P25/28
Filed: 1994-05-07
Abstract: In the present invention there are disclosed compounds of the general formula I, in which m is 0, 1 or 2, n is 2 through 5, X represents carbonyl or the group of the general formula II, Y and Z represent an optionally substituted alkylene, R represents an optionally substituted phenyl, or R represents naphthyl and Ri1 a Ri2 represent hydrogen, alkyl or phenylalkyl, their pharmaceutically acceptable salts, process of their synthesis, pharmaceutical preparation containing the compound of the general formula I as well as use of this compound for neuroprotective treatment or for treatment of depression, anxiety, Parkinson?s disease, obesity, consciousness disorders, paroxysms and neurological disorders.
Patent CZ-291693-B6 (CZ)
Title: Apparatus for producing water glass by hydrothermal synthesis
Inventor: ANTOS PETR DR ING
IPC: C01B33/32
Filed: 1999-12-22
Abstract: In the present invention there is disclosed an apparatus having the form of a horizontal cylinder with the cylinder length-to-diameter ratio ranging between 2.9 to 4.0. Inner circumference of the cylinder jacket is provided with mixing blades and the inner surface thereof is metal coated with pure nickel containing alloying ingredients such as manganese, chromium, titanium, niobium, tantalum, or molybdenum in an amount ranging from 0.1 to 10 percent by weight.
Patent SK-284919-B6 (SK)
Title: Method of producing powder agglomerates and dosage form comprising thereof
Inventor: YANG TSONG-TOH
IPC: A61K31/404
Filed: 1998-03-16
Abstract: Described is a method of producing agglomerates of drug and solid binder, starting from said components in a form of fine particles having proper amount of convertible amorphous content. Agglomerates are formed from these dry particles and convertible amorphous content present in agglomerates is converted to a crystalline form upon exposure to atmospheric moisture. Finished agglomerates have crush strength, thought an average amount of fine particles fraction is provided by breaking apart thereof during administration. Dosage forms for oral and nasal administration of these agglomerates are described.
Patent SK-279294-B6 (SK)
Title: Method of hydrogenated conjugated diolefin polymers and copolymers preparation
Inventor: CHAMBERLAIN LINDA R
IPC: C08C19/44
Filed: 1991-05-13
Abstract: A method of hydrogenated conjugated diolefin polymers preparation which is terminating a living polymer obtained by polymerising or copolymerising at least a conjugated diolefin with an organo-alkali metal polymerisation initiator in a suitable solvent, by the addition of hydrogen, and effecting selective hydrogenation of the unsaturated double bonds in the conjugated diolefin units of the terminated polymer by contacting the polymer, in the absence of hydrocarbon lithium and alkoxy lithium compounds, with hydrogen in the presence of at least one bis(cyclopentadienyl)titanium compound.
Patent SK-279240-B6 (SK)
Title: Cookie with high cereal content
Inventor: RUSSO CLAUDIO
IPC: A21D13/08
Filed: 1992-08-31
Abstract: A cookie with a high cereal content has an expanded cellular structure and includes from 7 to 20 percent by weight of at least one protein and from 10 to 65 percent by weight of cereal flakes being dispersed and incorporated into the expanded cellular structure. The expanded cellular structure consists, preferably, of at least one foam producing protein, which might be whipped, and is selected from the group containing the white protein, lactic and cereal proteins, vegetable proteins and compounds thereof as they are or partially hydrolyzed.
Patent CZ-299225-B6 (CZ)
Title: Process for preparing crystalline dibenzothiazepine derivative, crystalline dibenzothiazepine derivative so prepared and medicaments containing thereof
Inventor: SNAPE EVAN WILLIAM
IPC: A61K31/55
Filed: 1998-07-28
Abstract: In the present invention, there is disclosed a process for preparing crystalline 11-(4-[2-(2-hydroxyethoxy)ethyl]-1-piperazinyl)dibenzo [b, f] [1, 4]thiazepine of the general formula I by crystallizing from a non-aromatic solvent such as ethyl acetate, isobutyl acetate, methyl iso-butylketone or methyl tert-butyl ether, preferably in the absence of water. The obtained crystalline substance can be converted to a pharmaceutically acceptable salt, such as fumarate and it can be used for the treatment of psychoses, or more precisely for preparing medicaments for treating psychoses.
Patent CZ-302750-B6 (CZ)
Title: Pharmaceutical composition and a vial for containing formulation based on erythropoietin and method of inhibiting microbial growth in a solution comprising erythropoietin
Inventor: GAYED ATEF
IPC: A61K/
Filed: 2000-07-21
Abstract: In the present invention, there is disclosed a pharmaceutical composition comprising erythropoietin and an amount of benzethonium chloride effective to inhibit microbial growth in said composition, wherein the composition can further comprise a preservative being selected from the group consisting of benzethonium chloride, phenoxyethanol and phenylethyl alcohol. There is also disclosed a vial for containing formulation of the same composition as the above-described pharmaceutical composition and containing multiple dosages of erythropoietin. Further disclosed is a method of inhibiting microbial growth in a solution comprising erythropoietin, said method comprising adding benzethonium chloride to said solution.
Patent CZ-305056-B6 (CZ)
Title: Precession liquid turbine
Inventor: SEDLÁČEK MIROSLAV
IPC: H02K7/18
Filed: 2013-09-05
Abstract: In the present invention, there is disclosed a precession liquid turbine having a stator (1) with a liquid inlet opening (3) and a liquid outlet opening (4). A vaneless roller runner (2) consisting of body of rotational shape is mounted on retention device (6) within the stator (1). The retention device (6) is adapted for enabling gyratory rolling of the runner (2) on inner wall of the stator (1). The roller rotor (2) is coupled by means of a mechanism (5) with an electric current generator (7) that is arranged inside a waterproof casing (8). The mechanism (5) comprises a crankshaft (9), arranged between the roller rotor (2) and the electric current generator (7), whereby the crankshaft (9) is provided with a magnetic clutch (10).
Patent CZ-305281-B6 (CZ)
Title: Implant introduction device
Inventor: KUBĚNA PETR
IPC: A61M25/095
Filed: 2013-09-16
Abstract: In the present invention, there is disclosed a device being provided with a base tube (2) with an olive (12) arranged for insertion of a cover tube (4) thereon. In front of the olive (12), the base tube (2) is provided with an insertion hole (13). A control wire (3) provided at its end with a clip (5) and a securing element (21) of the control wire (3) position, passes all over the length inside the base tube (2). The proximal end of the control wire (3) serves for passing into an eye (27) of the implant tubular part (26) stranded wire. A front definition element (15) and a rear definition element (16) serve for securing the position of the implant stent part (25) onto the base tube (2). The base tube (2) has a proximal portion (2.1) and a distal portion (2.2), which portions are coupled with each other in the rear definition element (16). An extensible stop (17) for release the implant tubular part (26) and an extensible stop (18) for release of the implant stent part (25) are arranged on the distal portion (2.2). The base tube (2) is coupled by means of a coupling (19) with a Y connector (20), The control wire (3) passes through the side outlet (23) of said Y connector while a guide wire passes through horizontal arm of the same. The guide wire (6) is arranged within an internal tube (14) passing all over the length of the base tube (2).
Patent CZ-306692-B6 (CZ)
Title: Telescopic hydraulic lines
Inventor: Hovanec Dušan
IPC: F16J7/00
Filed: 2015-11-03
Abstract: The telescopic hydraulic lines consist of the hollow pressure cylinder (3) mounted on the rigid frame (1). The pressure cylinder (3) is provided, in the axis of one of the bottoms, with the pressure oil inlet (4), while the flange (5) of the pressure oil inlet (4) is provided with elements for connecting the hydraulic lines. In the opposite bottom of the pressure cylinder (3), there is formed the opening (6) in which there is slidably placed the piston rod (7) provided with the piston (11) slidable in the pressure cylinder (3). In the axis of the piston rod (7), there is, along its entire length, created the through opening (8) which is connected to the coaxial through opening (12) of the same diameter formed in the piston (11) further provided with the longitudinal through openings (13) for pressure equalization, whose centres are located on a circle in the annulus formed by the through opening (12) and the outer circumference of the piston (11). The diameter of the longitudinal openings (13) for equalizing the pressure corresponds to one third of the diameter of the axial through opening (8, 12) in the piston (11) and in the piston rod (7). The outlet part of the piston rod (7), located in the movable frame (2), is arranged for connection to the hydraulic lines of the pressure oil outlet (9).
Patent CZ-307846-B6 (CZ)
Title: Fire protection box for sensitive equipment
Inventor: TIPEK MICHAL
IPC: A62C35/02
Filed: 2018-03-23
Abstract: Fire protection box for sensitive equipment containing a fireproof lining. The box has a coolant tank (140) which is coupled to the internal cooling block (2) in the housing and comprising of a pump (20), coolant, air heat exchanger / coolant in the tank (140) and an indoor air ventilation unit ( 21) assigned to the heat exchanger, the pump (20) and the ventilation unit (21) are connected to a power source and a control unit (3) which is inside the box and coupled to at least one temperature sensor (4), and at least one smoke sensor (6) which are also in the housing.
Patent CZ-308303-B6 (CZ)
Title: Lighted radiator grille and front of the car with this mask
Inventor: KRAMULE MICHAL
IPC: B60R19/52
Filed: 2018-09-17
Abstract: The illuminated radiator grille comprises a light source (6), an outer transparent part (1) with a semi-permeable layer (8) applied to the back, an inner transparent part (2) with a reflective layer (7) applied to the back, and a housing (3). The semi-permeable layer (8) partially transmits and partially reflects light. The outer transparent part (1) is permanently connected to the housing (3) at the periphery and together they form a closed inner space. The rear of the outer transparent part (1) is oriented to the interior. In the interior space there is an inner transparent part (2) with its front side towards the rear side of the outer transparent part (1). Furthermore, a light source (6) is located in the inner space. The front of the car includes the headlights, the front bumper, the bonnet and the illuminated radiator grille of the car. The illuminated radiator grille is located approximately in the middle of the front of the car between the headlights, above the front bumper, under the bonnet.
Patent SK-283507-B6 (SK)
Title: Method of making (+/-)-3-(aminomethyl)-5-methylhexanoic acid
Inventor: GROTE TODD MICHEL
IPC: C07C227/04
Filed: 1996-05-13
Abstract: A method of making (+/-)-3-(aminomethyl)-5-methylhexanoic acid usable for making of (S)-3-(aminomethyl)-5-methylhexanoic acid.
Patent CZ-296305-B6 (CZ)
Title: Ventilation unit
Inventor: HOEPLER KLAUS
IPC: F24F13/24
Filed: 2000-06-27
Abstract: The present invention relates to a ventilation unit (10) intended for a ventilating shaft wherein the ventilation unit (10) is provided with supporting casing (12) accommodating a fan (14) whereby on said casing (12) bottom side, there is performed a suction opening (22) for intake air and on said casing (12) upper side, there is performed an outlet opening (32) for exhausted air. The fan (14) is fastened within the casing (12) by means of shaped blocks (16, 18, 20) made of sound and heat insulating parts (16,18,20).
Patent CZ-298559-B6 (CZ)
Title: Isothiazole derivative, process and intermediates for its preparation and pharmaceutical composition in which the derivative is comprised for treating hyperproliferative diseases
Inventor: LARSON ERIC ROBERT
IPC: C07C327/38
Filed: 1999-05-03
Abstract: In the present invention, there is disclosed an isothiazole derivative of the general formula 1, process and intermediates for its preparation and pharmaceutical composition in which the derivative is comprised for treating hyperproliferative diseases such as cancer of brain, lung, squamous cell, bladder, gastric, breast and the like. Disclosed is also the use of the above-described derivative for preparing a medicament.
Patent CZ-303238-B6 (CZ)
Title: Insecticidal coating of seeds and use thereof for protection of agricultural produces
Inventor: CHEN YUGUANG
IPC: A01N57/24
Filed: 1998-12-14
Abstract: The present invention relates to an insecticidal coating for a seed comprising one or more binders selected from the group consisting of polymers and copolymers of polyvinyl acetate, methyl cellulose, polyvinyl alcohol, vinylidene chloride, acrylic acid, cellulose, polyvinylpyrrolidone and polysaccharide and an insecticide and filler wherein the binder forms a matrix for the insecticide and filler resulting in a substantially non-phytotoxic seed coating; methods for producing said coating and the seed treated with the above described coating. Additionally the invention concerns a method of controlling soil-borne insect pests, particularly from the order of Coleoptera, such as Diabrotica spp., comprsing applying to a seed an insecticidal coating as described above.