baber/WOPTO huggingface dataset:
Patent FR-2862304-A1 (FR)
Title: New racemic or achiral dual molecules comprising cyclic peroxide linked to antimalarially active and/or bioavailability improving residue, useful as broad-spectrum antimalarial agents
Inventor: CAZELLES JEROME
IPC: C07D491/113
Filed: 2003-11-14
Abstract: New racemic or achiral dual molecules (I) consist of coupling products of (a) a cyclic peroxide having a spiro-bonded azacyclic ring and (b) a molecule with antimalarial activity and/or a residue for improving bioavailability, (a) and (b) being linked by a coupling arm bonded to the N-atom of (a). New racemic or achiral dual molecules consist of coupling products of formula (I) or their acid addition salts. Corresponding molecules in the form of pure optical isomers or their mixtures in all proportions are also claimed. [Image] A : residue of a molecule with antimalarial activity and/or a residue for improving bioavailability, the latter comprising one or more N, O or S heteroatoms in a 6-18C saturated or unsaturated cyclic moiety or in an optionally substituted (os) 1-18C linear chain; p, p', p'' : 0 or 1, provided that at least one of p and p'' is 1; Y 1, Y 21-5C alkylene, optionally containing one or more amine, amide, sulfonamide, carboxy, thiocarboxy, carbonyl, ether, thioether or thiocarbonyl radicals and os by 1-5C alkyl; U : amine, amide, thioamide, sulfonyl, carbonyl, thiocarbonyl, carboxy, thiocarboxy, ether, thioether or sulfonate function; Z 1, Z 2linear, branched or cyclic, saturated or unsaturated 1-4C alkylene, one of Z 1 and Z 2 optionally being absent; Z 1 + Z 2polycyclic structure including N and the junction carbon C j; R 1, R 2H or water-solubilizing group (specifically COOH, OH or NR aR b); R a, R bH or 1-5C linear, branched or cyclic alkyl; R x + R ygroup completing a 4-8 membered cyclic peroxide containing 1 or 2 additional O atoms in the ring structure and including C j in the ring structure, the ring being substituted by 1-4 groups R 3; R 3H, halo, OH, CF 3, NO 2, aryl, heteroaryl, Q, OQ or 3-18C mono-, bi- or tricyclic structure (optionally containing one or more O, N or S heteroatoms and os by Q), provided that at least one R 3 group other than H is present; or two adjacent R 3 groups together for a 5- or 6-membered saturated or unsaturated cyclic structure, os by one or more groups R 3 as defined above; Q : 1-5C linear, branched or cyclic alkyl. An independent claim is included for the preparation of (I). ACTIVITY : Antimalarial. Racemic 7-chloro-N-(2-(6-isopropyl-8a-methyl-4a,7,8,8a-tetrahydro-1'H-spiro-(1,2,4-benzotrioxin-3,4'-piperidine)-1'-yl)-ethyl)-quinoline-4-amine (Ia) (designated 'PA 1010') had IC 5 0 less than 0.1 MicroM against Plasmodium falciparum strains FcB1-Columbia (moderately resistant to chloroquine) and FcM29-Cameroon (highly resistant to chloroquine), cultured in vitro in media containing human erythrocytes. MECHANISM OF ACTION : Parasite heme and/or protein alkylating agent.
Patent FR-2863045-A1 (FR)
Title: Projectile stabilizer fin deployment system has inertia valve between gas generator and differential piston(s) driven by gas pressure
Inventor: AGNELOT GREGOIRE
IPC: F42B10/20
Filed: 2003-11-27
Abstract: A fin (3) deployment system comprises at least one gas generator (6) initiated on firing, and at least one differential piston (7) that receives gas pressure from firing on one face and gas pressure from the generator on the other, and incorporates at least one inertial valve (31) between the gas generator and piston(s). The valve has a peg (32) located in a bore parallel to the projectile's axis (11). The peg moves against a return spring and has a cylindrical section and recess that close and open a channel connecting the gas generator to the differential piston(s).
Patent FR-2863274-A1 (FR)
Title: Quantitative evaluation of specific genetic rearrangements or recombinations, useful e.g. for monitoring treatment of disease, comprises selective amplification of genomic DNA
Inventor: MARCHE PATRICE
IPC: C12Q1/68
Filed: 2003-12-05
Abstract: Process for quantitative evaluation of a targeted genetic rearrangement or recombination by selective amplification of genomic DNA. Process for quantitative evaluation of a targeted genetic rearrangement or recombination comprises: (a) extracting human genomic DNA (I) from a sample; (b) amplifying segments (II) of (I) of size from a few hundred to a few tens of thousands of bases by multiplex PCR; (c) separating the amplified (II) and; (d) detecting the rearranged/recombined segments. Step (b) is done in presence of: (i) one or more primer pairs, where at least one primer hybridizes upstream of and/or at the 5'-end of, one gene (Vx) being amplified, and the other hybridizes downstream of, and/or at the 3'-end of, the other gene (Jy) being analyzed, where Vx and Jy may be involved in a genetic rearrangement, and (ii) at least one DNA polymerase that can amplify (II) (preferably of over 10 kb) and has correction activity to improve the elongation reaction. The amplification step also includes initial denaturation; cycles of denaturation, hybridization and elongation, with the elongation being for at least 10 minutes at 68-72[deg]C. Independent claims are also included for the following: (1) kit comprising the specified primers and probes, also usual buffers and reagents for performing a PCR; (2) primer for use in the new process having any of 21 sequences reproduced; and (3) detection probe for use in the new process having any of 16 sequences reproduced.
Patent FR-2864510-A1 (FR)
Title: Mechanical unit e.g. articulation bearing, fixing arrangement for motor vehicle, has reinforcement unit with lower wall having holes coinciding with holes of side rail, and discharge opening coinciding with opening of lower wall of rail
Inventor: HLUBINA THIERRY
IPC: B62D21/04
Filed: 2003-12-31
Abstract: The arrangement has a side rail (14) with a tubular section having a lower wall (18) at its end part. A stiffening unit has a common reinforcement unit (24) with a lower wall (26) fixed on the wall (18) and having two holes (28) coinciding with fixation holes of the wall (18). A discharge opening (32) arranged in the wall coincides with an opening in the wall (18) for discharging condensation products formed in the rail.
Patent FR-2852472-A1 (FR)
Title: Appareil et procede pour le filtrage par modele de flux de trafic dans un systeme de communication mobile
Inventor: AHN HONG JIN
IPC: H04W92/00
Filed: 2004-02-20
Abstract: Un système de communication mobile effectuant un filtrage par Modèle de Flux de Trafic (ou TFT) conformément à des versions de Protocole Internet (IP), supporte une adresse d'une première version d'IP incluant des premiers bits et une adresse d'une seconde version d'IP incluant des seconds bits contenant les premiers bits. Une information basée sur la version d'IP est extraite de l'adresse IP de source. Une information de TFT contenant l'information extraite est générée et l'information de TFT générée est transmise à un Noeud de Support GPRS de Passerelle (ou GGSN) (1519).
Patent FR-2869106-A1 (FR)
Title: Procede d'estimation de distance pour aeronef avec prise en compte de contraintes de navigation aerienne
Inventor: BITAR ELIAS
IPC: G05D1/10
Filed: 2004-04-20
Abstract: Ce procédé met en oeuvre pour l'estimation d'une distance, une transformée de distance par propagation ne considérant que les trajets qui sont à la fois accessibles de l'aéronef compte tenu de son profil vertical de vol et respectueux de la réglementation aérienne. La distance propagée (DP) est accompagnée d'une altitude propagée (AP) qui suit en tout point le profil vertical de vol de l'aéronef, tout en étant supérieure aux altitudes de ces points et en respectant les contraintes de la réglementation aérienne en ces points. Cela est obtenu en soumettant la propagation à la satisfaction du profil vertical de vol de l'aéronef, des contraintes des élévations des points du relief et des contraintes de la réglementation aérienne.
Patent FR-2871586-A1 (FR)
Title: Verre ophtalmique a fonction electro-optique
Inventor: CANO JEAN PAUL
IPC: G02C7/10
Filed: 2004-06-11
Abstract: Un verre ophtalmique comprend un substrat transparent (3) et des moyens électro-optiques (5) intégrés au substrat pour procurer une fonction optique en réponse à un stimulus électrique. Le verre ophtalmique comprend en outre au moins une cellule photovoltaïque (6) intégrée au substrat pour alimenter les moyens électro-optiques en réponse à une lumière incidente. La cellule photovoltaïque (6) peut être incorporée à un élément opaque occupant une petite partie de la surface du verre. Alternativement, la cellule photovoltaïque (6) peut être transparente et peut recouvrir au moins en partie la surface du verre.
Patent FR-2873536-A1 (FR)
Title: Cubical bundles handling and turning over device for e.g. loader, has four lower teeth fixed on frame for supporting stack of five bundles, and five rows of four horizontal upper teeth fixed to axles and rotating with respect to frame
Inventor: COMBRET JULIEN
IPC: A01D87/12
Filed: 2004-08-02
Abstract: The device has a frame (1) to which four lower teeth (2) are fixed for supporting a stack of five bundles, and five rows of four horizontal upper teeth (6) fixed to axles (4) and rotating with respect to the frame. The axles are rotated using lever arms (7) that are connected to a linkage (9) through axles (8). The linkage is actuated by a jack using a third axle, where jack is connected to the frame using a fourth axle.
Patent FR-2880109-A1 (FR)
Title: Firearm system for use on e.g. flatbed truck, has cradle integrated with plate that can be disposed on ground by vehicle using operating arm, where plate has pivoting stabilizing arm fixed to each one of corners of plate
Inventor: BALBO PATRICK
IPC: B60P1/64
Filed: 2004-12-28
Abstract: The system has a barrel (2) mounted on a cradle (3) and intended to be carried by a vehicle (4). The cradle is integrated with a plate (8) that can be disposed on the ground by the vehicle using an operating arm. The barrel fires from the plate disposed at the ground. The plate has a pivoting stabilizing arm (12) fixed to each one of corners of the plate.
Patent FR-2871651-A1 (FR)
Title: Capot en verre et boitier d'encapsulation de composants electroniques dote d'un tel capot
Inventor: BETTINELLI ARMAND
IPC: H01L51/50
Filed: 2004-06-09
Abstract: Le capot d'encapsulation (1) comprend au moins deux couches de verre de compositions différentes, une première couche (2) dite de fond qui est continue et au moins une deuxième couche (3, 6) qui est discontinue et adaptée pour délimiter des cavités (4, 5) ou des anfractuosités dans ce capot.On forme de préférence les couches de verre autres que la première à partir de frittes à bas point de fusion, ce qui permet de fabriquer économiquement de tels capots, sans recourir à l'usinage de verre.
Patent FR-2884665-A1 (FR)
Title: Procede d'alerte lors d'une modification de contenu et systeme pour la mise en oeuvre du procede
Inventor: CASTAIGNET LAURENT
IPC: H04L29/00
Filed: 2005-04-19
Abstract: Procédé pour alerter un utilisateur (17) muni d'un terminal (4;5;6;7) lors d'une modification d'un contenu selon une technologie de syndication de contenu dans un système de communication supportant un protocole d'initiation de session et de notification et incluant un serveur d'alertes (1) et un serveur de contenu (2). Selon ce procédé :- on transmet, depuis un terminal (4) de l'utilisateur (17) vers le serveur d'alertes (1), un message de souscription (9; 18) dudit protocole identifiant un contenu conforme à ladite technologie de syndication de contenu stocké sur le serveur de contenu (2) ;- on reçoit au serveur d'alertes (1), depuis le serveur de contenu (2), une indication relative à une modification dudit contenu ; et- on transmet un message de notification (11;20;23) dudit protocole audit utilisateur (17), depuis le serveur d'alertes (1), lorsqu'une indication relative à une modification dudit contenu a été reçue.
Patent FR-2888290-A1 (FR)
Inventor: DORE MARTIAL
IPC: F02M35/104
Filed: 2005-07-07
Abstract: The manifold has a plenum connected to inlet valves and divided into lower part (5) and upper part (6). The upper part is integrated to a part of air intake ducts and the lower part is integrated to another part of the ducts. The upper part and lower part of the plenum are connected with respect to each other by a hinge (7). The plenum has a sealing joint situated between the lower part and upper part. An independent claim is also included for a motor vehicle comprising an air intake manifold.
Patent FR-2890846-A1 (FR)
Title: Electrocardiographic data acquisition and processing system for e.g. medical application, has calculating module calculating output value corresponding to interval between respective spikes of wave of pulse and wave of preceding pulse
Inventor: GREVOZ FRANCK
IPC: A61B5/352
Filed: 2005-09-16
Abstract: The system has an acquisition unit (31) for acquiring electrocardiographic data comprising digital values (Si) of samples of an electric signal representative of cardiac pulses as well as digital value indicating the detection of QRS wave of a determined cardiac pulse. A processing unit (32) e.g. computer, has a calculating module (344) for calculating an output value, pulse by pulse, corresponding to an interval between respective spikes of the wave of the pulse and the wave of preceding pulse from the electrocardiographic data. Independent claims are also included for the following: (1) a unit for acquisition of electrocardiographic data (2) a unit for processing electrocardiographic data.
Patent FR-2893324-A1 (FR)
Title: Procede de collage sur chape a base de sulfate de calcium.
Inventor: JALLA SEBASTIEN
IPC: C04B40/00
Filed: 2005-11-14
Abstract: L'invention a pour objet un procédé de collage sur une chape à base de sulfate de calcium ayant une humidité résiduelle de plus de 1% et/ou après une durée, mesurée après coulage de la chape, inférieure à 3 semaines, à l'aide d'un mortier-colle à base de sulfate de calcium hydrofugé et/ou sur une chape hydrofugée.L'invention a aussi pour objet l'utilisation d'un mortier-colle à base de sulfate de calcium hydrofugé pour le collage sur une chape à base de sulfate de calcium ayant une humidité résiduelle de plus de 1% et/ou après une durée, mesurée après coulage de la chape, inférieure à 3 semaines.
Patent FR-2882096-A1 (FR)
Title: Twin-shaft turbine engine for aircraft, has main drive pinion module driving movement transmission shafts extending coaxially, and driving unit comprising high and low pressure drive pinions integrated to high and low pressure rotors
Inventor: BART JACQUES
IPC: F02C7/36
Filed: 2005-02-11
Abstract: The engine has a driving unit comprising a high pressure drive pinion (9) integrated to a high pressure rotor (2) at the proximity of an upstream end of the rotor. The driving unit has a low pressure drive pinion (7) integrated to a low pressure rotor (1) in the downstream of the rotor (2). A main drive pinion module (29) drives movement transmission shafts (11, 12) that extend coaxial to each other. An independent claim is also included for a turbine engine mounting method.
Patent FR-2895995-A1 (FR)
Title: Pavement kerbstone has upper surface that slopes down to road level to facilitate passage for persons of reduced mobility, pedestrians and push chairs
Inventor: GAILLARD PASCAL
IPC: E01C11/22
Filed: 2006-01-10
Abstract: The kerbstone (1), made from natural stone or concrete with a preferable length of 100 cm between its two ends (9, 10), has an upper surface with a flat strip adjoining the pavement and a sloping section that is angled down to meet the road surface (2) with no difference in height from it. The vertical front edge of the kerbstone preferably measures some 14 cm in height, which is covered by the road surface, while its rear surface adjoining the pavement is preferably about 18 cm high. Kerbstones (13) with gradually sloping surfaces can be laid on either side of it.
Patent FR-2898265-A1 (FR)
Title: Oral irrigating device for cleaning impurity between teeth of individual, has dip-tube permitting to rise sterilizing liquid contained in reservoir when manual pressure is exerted on reservoir, where reservoir is made of flexible plastic
Inventor: ROUSSEL PHILIPPE
IPC: A61C17/02
Filed: 2006-03-08
Abstract: The device has a conduit (2) terminated by a curved and frayed mouth (3), and a threaded stopper (8) screwed on a thread (6) of a reservoir (1). The reservoir is made of flexible plastic and is filled with sterilizing liquid. The reservoir has a rigid plastic boring needle (12) at its base for piercing a sealing cap (11) of the reservoir. A dip-tube (5) permits to rise the liquid contained in the reservoir when manual pressure is exerted on the reservoir.
Patent FR-2898870-A1 (FR)
Title: Nacelle for turbojet engine of aircraft, has air inlet structure providing peripheral inner surface that is partially equipped with acoustic attenuation structure, where space is arranged between attenuation structure and casing
Inventor: VAUCHEL GUY
IPC: B64D33/02
Filed: 2006-03-24
Abstract: The nacelle has an air inlet structure channeling air flow towards a fan of a turbojet engine. A median structure (5) includes a casing (9) which surrounds the fan, where the inlet structure is attached to the casing. The inlet structure provides a peripheral inner surface that is partially equipped with an acoustic attenuation structure (13). The attenuation structure extends on a part of the casing, where a space (14) is provided between the attenuation structure and the casing.
Patent FR-2909887-A1 (FR)
Title: Dispositif de suspension a triangulation automatique.
Inventor: DUSSENNE FRANCOIS
IPC: A62B35/00
Filed: 2006-12-15
Abstract: Dispositif de suspension destiné à être appliqué à un utilisateur ou un objet quelconque pour lui permettre d'être suspendu à une corde le long de laquelle il va ainsi pouvoir se déplacer et comportant un premier point de support de charge principal, par exemple une ceinture (1) à dosseret destiné à entourer le bassin de l'utilisateur et au moins deux points de support de charge auxiliaires, par exemple deux cuissardes (4) destinées à chacune entourer une cuisse de l'utilisateur, et un système de liaison pour relier le premier point de support de charge principale au aux moins deux points de support de charge auxiliaires constitué d'au moins une première courroie (7) reliant le point de support de charge principale à l'un des deux points de support auxiliaire et une deuxième courroie (8) reliant le point de support principal au deuxième point de support auxiliaire et une courroie (9) centrale reliée à chacune des au moins deux courroies auxiliaires, la courroie centrale étant destinée à être suspendue à une corde principale le long de laquelle l'utilisateur souhaite pouvoir se déplacer dans un sens ou dans l'autre, est caractérisé en ce qu'il est prévu des moyens de réglage automatique de l'équilibre.
Patent FR-2898136-A1 (FR)
Title: Process for installing and/or deinstalling a hollow/filled magnetic target on a cathode magnetron for cathodic pulverization, comprises generating a permanent magnetic field above the target for controlling a magnetron magnetic field
Inventor: COULON JEROME
IPC: C23C14/35
Filed: 2006-03-03
Abstract: The process for installing and/or deinstalling a hollow/filled magnetic target (14) on a cathode magnetron (10) for cathodic pulverization, comprises generating a permanent magnetic field above the target for controlling a magnetron magnetic field. The permanent magnetic field is adapted with the cathode.
Patent FR-2900917-A1 (FR)
Title: Flexible irrigation sheath rolling and unrolling device for agriculture field, has disengageable mobilization module mounted on chassis and rotating reels when it is engaged with reels, and nozzles located in upstream of sheath rolling path
Inventor: JAULENT GERARD
IPC: A01G25/00
Filed: 2006-04-28
Abstract: The device (D) has preformed reception cradles (300a, 300b) positioned on a chassis (200) for receiving and rotatably guiding reels (100a, 100b) by supporting and guiding rollers. The chassis has a disengageable mobilization module (400) rotating the reels installed in the cradles when the module is engaged with the reels. The module movably mounted on the chassis has a motor moving a shaft co-operating with the reel (100a). Guiding nozzles are located in upstream of a rolling path of a flexible irrigation sheath.
Patent FR-2910811-A1 (FR)
Title: Use of riluzole for preparation of drug e.g. to reestablish immune function, to treat inflammatory diseases, infection, cancer, viral infection and their virological and immunitary symptoms, leishmaniasis, malaria or bilharziasis
Inventor: ACHOUR AMMAR
IPC: A61K31/428
Filed: 2007-01-03
Abstract: Use of riluzole (I) or its salt for the preparation of medicament to reestablish the immune function for the treatment of inflammatory diseases, infection and cancer, is claimed. ACTIVITY : Antiinflammatory; Antimicrobial; Cytostatic; Virucide; Anti-HIV; Hepatotropic; Protozoacide; Antimalarial; Schistosomacide. MECHANISM OF ACTION : None given.
Patent FR-2916830-A1 (FR)
Title: Sections e.g. post and frame crossmember, assembly for manufacturing e.g. transom frame, of door, has arm with wedging immobilization zone wedged with section at state, where zone is located in or at vicinity of connection zone of two arms
Inventor: GOUBIN JEAN JACQUES
IPC: E06B3/968
Filed: 2007-05-29
Abstract: The assembly has an angle bracket (10) with arms (11, 12) inserted at interior of two sections (20, 30) e.g. post and frame crossmember. Each of the arms has a wedging immobilization zone wedged with one section at an engaged state of the arms in the sections. The wedging immobilization zone is located in or at vicinity of a connection zone of the arms. The arms have support surfaces (13, 14) for allowing relative displacement of the angle bracket and the arms in direction of addition and/or reinforcement of the wedging immobilization of one section, when the effort is exerted on the supports. An independent claim is also included for a method for assembling two sections and an angle bracket for forming an assembly.
Patent FR-2917117-A1 (FR)
Title: Well or buried/non-buried piping casing method for water/crude oil production field, involves achieving radial expansion at certain areas spaced from each other by non-expanded portions, such that total length of expanded areas is smaller
Inventor: NICOLAS FREDERIC
IPC: E21B33/12
Filed: 2007-06-05
Abstract: The method involves inserting a long length cylindrical tube (1) into a well or a piping to be cased, and proceeding a radial expansion of the tube using an inflatable bladder (3) so that a wall (C) bears against the wall of the well or the piping. The radial expansion is achieved at certain areas spaced from each other by non-expanded portions (5) and not on the entire length of the tube, such that a total length of expanded areas (4) is smaller than a total length of non-expanded areas, and a number of expanded areas is equal to three. An independent claim is also included for a method for controlling a production of fluid inside a well.
Patent FR-2917910-A1 (FR)
Title: Dispositif de lumiere optimisee par l'utilisation de materiaux artificiels et procede de fabrication associe
Inventor: LEE BOUHOURS MANE-SI LAURE
IPC: H01S3/10
Filed: 2007-06-22
Abstract: La présente invention concerne un dispositif de lumière, et notamment un dispositif émetteur de lumière. Plus particulièrement, elle vise à obtenir un émetteur de lumière au rendement amélioré par l'utilisation de matériaux artificiels permettant d'effectuer des traitements antireflet ou haute réflectivité.A cette fin, des structures sub-longueur d'onde sont gravées sur les faces externes d'une cavité émissive, permettant de contrôler la réflectivité de ces faces.L'invention s'applique à tout émetteur de lumière et donc notamment aux lasers, et plus particulièrement encore aux lasers à cascade quantique (ou QCL pour Quantum Cascade Laser en anglais).Par ailleurs, le présent brevet indique un procédé collectif de fabrication associé.