baber/WOPTO huggingface dataset:
Patent IL-151519-A0 (IL)
Title: Anti-infective active substance combinations and the use thereof for the topical treatment of fungus disease of toe and finger nails
IPC: A61K9/08
Filed: 2001-02-28
Abstract: A preparation comprising a combination of a topical and a systemic antimycotic and a physiologically acceptable lacquer base is suitable for the treatment and prophylaxis of onychomycoses. Preference is given to the use of water-insoluble lacquer preparations and a combination of at least one systemic antimycotic from the group of itraconazole, terbinafine and fluconazole or salts thereof with at least one topical antimycotic from the group of ciclopirox, 6-(2,4,4-trimethylpentyl)-1-hydroxy-4-methyl-2(1H)pyridone, amorolfine and butenafine or salts thereof.
Patent IL-153682-A0 (IL)
Title: Variolin derivatives, processes for the preparation thereof and pharmaceutical compositions containing the same
IPC: C07B61/00
Filed: 2001-07-11
Abstract: The invention provides variolin derivatives of formula (I), wherein: R<SUB>1 </SUB>and R<SUB>2 </SUB>are each independently selected from the group consisting of H, OH, OR, SH, SR, SOR, SO<SUB>2</SUB>R, NO<SUB>2</SUB>, NH<SUB>2</SUB>, NHR, N(R)<SUB>2</SUB>, NHCOR, N(COR)<SUB>2</SUB>, NHSO<SUB>2</SUB>R, CN, halogen, C(-O)H, C(-O)R, CO<SUB>2</SUB>H, CO<SUB>2</SUB>R, C<SUB>1</SUB>-C<SUB>12 </SUB>alkyl, C<SUB>1</SUB>-C<SUB>12 </SUB>haloalkyl, C<SUB>2</SUB>-C<SUB>12 </SUB>alkenyl, C<SUB>2</SUB>-C<SUB>12 </SUB>alkynyl, substituted or unsubstituted aryl, substituted or unsubstituted aralkyl and substituted or unsubstituted heteroaromatic; and R<SUB>3 </SUB>is selected from the group consisting of H, OH and OMe; wherein the or each group R is independently selected from the group consisting of OH, C<SUB>1</SUB>-C<SUB>12 </SUB>alkyl, C<SUB>1</SUB>-C<SUB>12 </SUB>haloalkyl, C<SUB>2</SUB>-C<SUB>12 </SUB>alkenyl, C<SUB>2</SUB>-C<SUB>12 </SUB>alkynyl, substituted or unsubstituted aryl, substituted unsubstituted aralkyl, substituted or unsubstituted arylalkenyl and substituted or unsubstituted heteroaromatic, and wherein the group R<SUB>1</SUB>, R<SUB>2 </SUB>or R<SUB>3 </SUB>is a group of formula N(R)<SUB>2 </SUB>or N(COR)<SUB>2</SUB>, each of the R groups may be the same or different, or the two R groups, together with the nitrogen atom to which they are attached, may form a 5-14 membered heterocyclic ring. These compounds display activity against a range of mammalian cancer cell lines. New synthetic routes to new and known variolin compounds, together with novel intermediates, are also disclosed. New antitumour activity of known variolin compounds is also described.
Patent IL-189128-A0 (IL)
Title: Aerated product
Filed: 2008-01-30
Abstract: A product comprising a container which contains an aerated composition is provided, the container having a dispensing aperture through which the aerated composition can be dispensed, characterized in that the aerated composition comprises hydrophobin.
Patent IL-197598-A0 (IL)
Title: Device for a pram and use of a push bar
Filed: 2009-03-15
Abstract: One embodiment of the present invention relates to a device for a pram, including a collapsible undercarriage provided with at least one moving device and at least a sub-frame which is releasable from the undercarriage and which is provided with device for supporting a child, and wherein the sub-frame is provided with a tiltable push bar. The sub-frame is reversible relative to the undercarriage. Another example embodiment of the present invention also relates to the use of a bar on a device for displacing a child, such as a pram, wherein the bar forms part of a sub-frame which can be coupled to an undercarriage for a pram, wherein the sub-frame is provided with a device for supporting a child, wherein the bar is used as push bar in the coupled situation of undercarriage to sub-frame, and wherein the bar is used in the uncoupled situation as carrying bar for the sub-frame.
Patent RO-130183-A0 (RO)
Title: Linear lighting fixture with leds
Inventor: HERŢANU RADU MIHAI
IPC: F21Y101/02
Filed: 2014-12-02
Abstract: The invention relates to a linear lighting fixture with LEDs, exhibiting an easy construction and being meant to illuminate indoor spaces. According to the invention, the lighting fixture consists of an upper profile (1), a lower profile (2) on which LED modules (6), an optical element (3) and a deflector (8) are mounted, where the lower profile (2) is secured to the upper profile (1) by means of four fastening clamps (11) and four fastening supports (12).
Patent AP-2001002138-A0 (AP)
Title: System and method for delineating spatially dependant objects, such as hydrocarbon accumulations.
Inventor: BUSH RONALD R
IPC: G01V3/38
Filed: 1999-08-31
Abstract: A neural network bases system, method, and process for the automated delineation of spatially dependent objects is disclosed. The method is applicable to objects such as hydrocarbon accumulations, aeromagnetic profiles, astronomical clusters, weather clusters, objects from radar, sonar, seismic and infrared returns, etc. One of the novelties in the present invention is that the method can be utilized whether or not known data is available to provide traditional training sets. The output consists of a classification of the input data into clearly delineated accumulations, clusters, objects, etc. That have various types and properties. A preferred but non-exclusive application of the present invention is the automated delineation of hydrocarbon accumulations and sub-regions within the accumulations with various properties, in an oil and gas field, prior to the commencement of drilling operations.
Patent AP-2004002961-A0 (AP)
Title: Rotary heat engine
Inventor: JARMAN JOHN WARNER
IPC: B60K16/00
Filed: 2004-01-06
Abstract: The engine consists of an annular array of chambers (hot leg), individually 5 connected to an adjacent continuous condenser (cold leg), and containing a quantity of working fluid and gas - the gas usually being the fluid's own saturated vapor. When a temperature differential exists between the chambers and condenser - either by means of heat being applied to the chambers or cooling being applied to the condenser, or both - a resultant difference in vapor pressure 10 is created; and while fluid within chambers on one lateral side is forced into the condenser, the positioning of the interconnecting ducts allows fluid to run freely from the condenser into chambers on the opposite upper lateral side. The weight imbalance and resultant torque created by such displacement of fluid causes the whole device to rotate, together with the axle to which it is secured.
Patent MA-22133-A1 (MA)
Inventor: R GILS
IPC: A61K31/40
Filed: 1991-04-15
Abstract: PCT No. PCT/GB91/00587 Sec. 371 Date Oct. 14, 1992 Sec. 102(e) Date Oct. 14, 1992 PCT Filed Apr. 15, 1991 PCT Pub. No. WO91/16306 PCT Pub. Date Oct. 31, 1991.There is disclosed a process for the preparation of a compound of structure (I)    <IMAGE>  (I)  in which n is 1 to 3 and each group R is hydrogen or C1-4 alkyl, which comprises, reaction of compound of structure (II)    <IMAGE>  (II)  (prepared by esterifying the hydroxyl compound) in which R1 is C1-4alkyl, phenyl or substituted phenyl and n is 1 to 3, with an amine HNR2 in which R is as described for structure (I), and optionally thereafter forming a salt. Intermediates are also disclosed.
Patent MA-24135-A1 (MA)
Inventor: BISCONTI BRUNO
IPC: B29C65/66
Filed: 1997-04-08
Abstract: This invention concerns an injection moulding process for soles in expansible and cross-linking "EVA" based compounds characterised in that during the cooling stage of the moulded sole (1) the spontaneous shrinkage of the same is arrested by means of a template (3) consisting of a rigid shaped plate placed on the sole (1) so that its edge connects with a perimeter edge (2) realised specifically on the upper surface (1a) of the sole (1), whose dimensions reduce no further either during the remaining cooling phase or after cooling.
Patent MA-24717-A1 (MA)
Title: Terminateur flexible de reseau synchrone
Inventor: SOLONE DE QUESADA JUAN IGNACIO
IPC: H04L25/38
Filed: 1998-12-09
Abstract: TERMINATEUR FLEXIBLE DE RÉSEAU SYNCHRONE QUI COMPREND LE TRASPORT DU MODE DE TRANSFERT ASYNCHRONE (ATM), DONT LA FINALITÉ EST D'eTRE INTÉGRÉ AUSSI BIEN à DES RÉSEAUX DIGITAUX DE SERVICES INTÉGRÉS à LARGE BANDE (RNIS-LB) QU'à DES RÉSEAUX DE TRANSPORT DE COMMUNICATIONS BASÉS SUR LA HIÉARCHIE DIGITALE SYNCHRONE (HDS), QUI EST CONFIGURABLE DANS UN  PREMIER MODE HDS-ATM,  DANS LEQUEL IL RÉALISE LES FONCTIONS DE LA SOUS-COUCHE DE CONVERGENSE DE TRANSMISSION, ET UN SECOND MODE HDS DANS LEQUEL IL SE COMPORTE COMME POINT DE TERMINAISON DE LA SECTIONDE MULTIPLEXAGE DE LA HDS, UN MODULE DE TRAITEMENT DE ATM, TOUS DEUX CONFIGURABLES DE FAÇON DYNAMIQUE, AINSI QU'UNE INTERFACE DE CONNECTION AVEC UN MICROPROCESSEUR EXTERNE POUR LA PROGRAMMATION DE CES MODULES, DIFFÉRENTS TYPES DE TRAMES SYNCHRONES ET DE TRAMES ATM POUVANT eTRE MANIPULÉES POUR RÉALISER DES INTERFACES ASYMÉTRIQUES EN VERTU DE L'INDÉPENDANCE DE LA SELECTION DANS DES PROCESSUS DE TRANSMISSION ET DE RECEPTION.
Patent MA-38105-A1 (MA)
Title: Immunoglobulines hétérodimères
Inventor: KANNAN GUNASEKARAN
IPC: C07K19/00
Filed: 2013-11-21
Abstract: La présente invention concerne des anticorps hétérodimères et des méthodes d'utilisation associées.
Patent MA-38323-A1 (MA)
Title: Dérivés pyrimidone et leur utilisation dans le traitement, l'amélioration ou la prévention d'une maladie virale
Inventor: ZHANG ZHUMING
IPC: C07D487/04
Filed: 2014-01-07
Abstract: La présente invention concerne un composé de formule générale (i), éventuellement sous la forme d'un sel, solvate, polymorphe, comédicament, cocristal, promédicament, tautomère, racémique, énantiomère ou diastéréoisomère pharmaceutiquement acceptable ou d'un mélange de ceux-ci, qui sont utiles dans le traitement, l'amélioration ou la prévention d'une maladie virale. De plus, l'invention concerne des polythérapies spécifiques.
Patent MA-40307-A1 (MA)
Title: Raccord à raccorder à un élément tubulaire, raccord de tubage et procédé de raccordement d'un raccord à un élément tubulaire
Inventor: SALEHI BAKHTIARI MANOUCHEHR
IPC: F16L13/14
Filed: 2015-10-29
Abstract: Cette invention concerne un raccord (3, 3') destiné à être raccordé à un élément tubulaire (5, 5') présentant une première section d'extrémité (9, 9') comprenant au moins un premier élément de raccordement (21, 21'), le diamètre d'au moins une partie du premier élément de raccordement (21, 21') pouvant être réduite dans une direction radiale de manière à former une connexion. Ledit premier élément de raccordement (21, 21') comprend au moins un premier élément formant crochet (21, 21') et/ou au moins un pr
Patent UY-26746-A1 (UY)
Title: Liberación controlada de fármacos administrados por via sublingual o bucal
Inventor: EL-RASHIDY RAGAB
Filed: 2001-06-01
Abstract: Una composición que proporciona una liberación relativamente lenta de fármacos solubles en agua, tales como apomorfina, por suministro a través de las rutas sublingual o bucal
Patent UY-26860-A1 (UY)
Title: Nuevo compuesto farmacéutico
Inventor: BARBIER PIERRE
IPC: A61K31/718
Filed: 2001-07-27
Abstract: La presente invención se refiere a combinaciones , composiciones y procedimientos farmacéuticos, para el tratamiento de la obesidad. De una forma más particular, la presente invención, se refiere a una combinación o composición, que comprende un inhibidor de lipasa, preferiblemente orlistat, y un secuestrante de ácidos biliares.
Patent UY-27706-A1 (UY)
Title: Bencimidazoles útiles en el tratamiento de la disfunción sexual.
Inventor: DAANEN JEROME F
Filed: 2003-03-07
Abstract: Uso de compuestos de fórmula ( I ) para el tratamiento de la disfunción sexual y composiciones que contienen compuestos de fórmula ( I ) para el tratamiento de la disfunción sexual.
Patent UY-30840-A1 (UY)
Title: Derivados de isoquinolina e isoquinolinona sustituidos
Inventor: LOHN DR MATTHIAS
IPC: A61K31/472
Filed: 2007-12-26
Abstract: La invencion se refiere a derivados de isoquinolina e isoquinolona 6-sustituidos de la formula (I), utiles para el tratamiento y/o prevencion de enfermedades asociadas con la Rho-quinasa de la fosfatasa de la cadena ligera de miosina, y a sus composiciones que contienen tales compuestos.
Patent UY-31074-A1 (UY)
Title: Maquina descortezadora
Inventor: ESQUENET JUAN
Filed: 2008-05-08
Abstract: La descortezadora que se propone, consiste en un chasis sobre ruedas, sobre el cual se encuentran dos conos o cilindros truncados de forma paralela y con giro opuesto. Los cuales poseen cada uno un aletado en forma de tornillo de Arquimedas con diferente " pase" y velocidad de giro, lo que provoca un efecto de "rascado" el cual despega la cascara de las tozas. También posee un precortador delantero en sentido transversal, que le hace el primer corte a la cascara y ayuda a ingresar a la linea central formada por los cilindros.
Patent ES-151140-A1 (ES)
Title: PROCEDIMIENTO PARA LA OBTENCIoN DE DERIVADOS DE AMUDINA
Filed: 1940-12-18
Abstract: Procedimiento para la obtención de derivados de amidina de la fórmula general **(Ver fórmula)** en la cual R1 representa un núcleo benzóico que en la p-posición posee un grupo nitroso o un sustituto reemplazable por tal grupo R2 un radical sustituido o no sustituido de la serie alifáticaalicíclicaaralifáticaaromáticahidroaromática o heterocíclica R3 y R4 hidrógeno o radicales substituidos o no substituidosen caso dado también combinados entre síalifáticosaralifáticosaromáticoshidroaromáticos o heterocíclicoscaracterizado porque se llevan a la transformación halogenuros imídicos de benzolsulfonacilamidas substituidas en la p-posición con un grupo nitroso o transformable en dicho grupo de la fórmula general **(Ver fórmula)** en la cual los radicales R1 y R2 tienen el mismo significativo como antescon amoníacoaminas primarias o secundariassimples o mezcladas incluso substituidas alifáticascon aminas primarias aralifáticasaromáticasheterocíclicas o primarias y secundarias hidroaromáticas.
Patent ES-177754-A1 (ES)
Title: UN QUEMADOR, ESPECIALMENTE PARA COMBUSTIBLES LiQUIDOS
IPC: F23D11/00
Filed: 1947-04-25
Abstract: Un quemador que comprende una caja cerrada para el aire primario abierta en su extremo de descarga una caja de aire secundario abierta en su extremo de descarga dispuesta dentro de dicha caja de aire primario y que define un paso anular entre dichas cajas una tobera de combustible contenida dentro de dicha caja de aire secundario y que define un paso anular con la misma y medios que se aplican a la caja del aire secundario y se extienden a través de la caja del aire primario y exteriormente a ella para ajustar la posición longitudinal de la caja del aire secundario con respecto a la caja del aire primario y la tobera del combustible.
Patent ES-181255-A1 (ES)
Title: MEJORAS EN O RELATIVAS A TELÉMETROS Y ALTiMETROS PARA ARTILLERiA ANTIAÉREA
Filed: 1947-12-30
Abstract: Mejoras en o relativas a telémetros y altímetros para artillería antiaérea y en especial en los mecanismos reguladores del telémetro, que comprenden un engranaje de velocidad variable movido continuamente por una fuerza, medios para aplicar al mecanismo un movimiento en concordancia con la variación del ángulo del rumbo del blanco (conjunto vacio), y usualmente también en conformidad con la variación del ángulo de la vista o mira del blanco (alfa), los cuales dos factores son variables y mensurables, sirviendo el mecanismo para combinar estos movimientos en conformidad con una relación matemática predeterminada, para dar un movimiento resultante correspondiente a la proporción de cambio de un valor seleccionado relacionado con la distancia, movimiento resultante que se utiliza para efectuar la regulación continua del engranaje de velocidad variable en conformidad con la indicada proporción de variación o cambio, y uniéndose el mecanismo motor del engranaje de velocidad variable con el prisma deflector del telémetro para la actuación del prisma, comprendiendo también el mecanismo un medio sintonizador maniobrado a mano para variar la potencia del mecanismo en conformidad con la variación de la altura y (o) la velocidad del blanco.
Patent ES-186769-A1 (ES)
Title: Perfeccionamientos en amplificadores de onda progresiva transversal
Filed: 1949-01-27
Abstract: Perfeccionamientos en amplificadores de onda progresiva transversal que constituyen un dispositivo traductor de energía de descarga electrónica en el que se intercambia energía entre electrones y ondas electromagnéticas progresivas que comprenden medios de enfoque para controlara dichos electrones respondiendo dichos medios de enfoque al vector de intensidad de campo magnético de dichas ondas electromagnéticas.
Patent ES-199674-A1 (ES)
Title: Un método de fabricar un material luminiscente
Filed: 1951-09-20
Abstract: Método para fabricar un material luminiscente para ser empleado en una válvula de descarga eléctrica de acuerdo con la Patente 191.176 caracterizado por el hecho de que se mezcla sulfuro de zinc con sulfuro de cadmio y una cantidad de sulfuro de zinc sobre la cual se ha depositado oro en forma de sulfuro siendo humedecido seguidamente la mezcla con una solución acuosa de nitrato de plata y una solución acuosa de nitrato de aluminio siendo agitada la masa y calentada una vez secada en una atmósfera de azufre e hidrógeno.
Patent ES-319960-A1 (ES)
Title: Carboxymethyl derivatives of tetracycline antibiotics
IPC: A61K31/65
Filed: 1965-11-24
Abstract: The invention comprises tetracycline derivatives of formula <FORM:1120821/C2/1> and their physiologically acceptable salts and complexes, wherein R represents the nucleus of a tetracycline antibiotic RCONH2, selected from tetracycline, or one of the following derivatives thereof: 7-chloro- 7-bromo- 5-oxy- 4-desdimethylamino- 4-desdimethylamino - 7 - chloro - 4 - desdimethylamino - 5-oxy- 6-deoxy- 6-deoxy-5-oxy- 6-demethyl- 6 - demethyl - 7 - chloro - 6 - deoxy - 6 - demethyl - 6 - deoxy - 6 - demethyl - 4 - desdimethylamino, metacycline or meclocycline, and <FORM:1120821/C2/2> is the residue of a primary or secondary amine which may be (1) a mono- or di-alkyl-amino or hydroxyalkylamino group, (2) a secondary saturated heterocyclic amino group containing one nitrogen atom, or a carboxy-, alkyl-, hydroxyalkyl-, dialkyl-amino-, or dialkyl-amino alkyl derivative thereof (3) an N1-substituted piperazino group wherein the N-substituent is alkyl, hydroxyalkyl, or dialkylaminoalkyl, or a carboxymethyl tetracycline group corresponding to the formula <FORM:1120821/C2/3> wherein R is as above or (4) the residue of a o -aminoalkanoic acid or an a , o -diaminoalkanoic acid, having 3 to 6 carbon atoms, or a suitable salt thereof "alkyl" refers to such groups having up to 5 carbons. The compounds are prepared by reacting in an inert solvent, at -10 DEG to 60 DEG C., stoichiometric amounts of the tetracycline antibiotic, glyoxylic acid, and the appropriate amine. The product may be formed into a salt, or the reaction carried out in the presence of the appropriate base to give the corresponding salt as the reaction product. Preferred cations are Na, K, Ca, Mg, Al, NH4, or amine groups, possibly being as defined above, or lidocaine or mepivacaine, but preferably tertiary alkylamines. <FORM:1120821/C2/4> may be piperidine, pyrrolidine, morpholine, N - (2 - hydroxyethyl) - piperazine or lysine. The reaction process, which may be performed in, e.g. ketones, lower alkanols, ethers or cyclic ethers, envisages the use of reacting derivatives of the reactants, such as amine or metal salts or lower alkanol hemi-acetals of glyoxylic acid, and acid addition salts of the tetracycline and amine. The product of the reaction may be obtained by cooling and crystallization of the mixture, precipitation with added miscible non-solvents, or by evaporating or lyophilizing off the solvent. As well as the salts of the inventive compounds mentioned above, complexes with calcium or magnesium may be formed, the proportion of complexing metal affecting the aqueous solubility and the stability of the complex. Pharmaceutical oral or parenteral compositions comprise the inventive compounds, together with excipients such as sterile water or tabletting substances, or in capsule form.
Patent ES-334670-A1 (ES)
Title: Milling machine with pivotal spindle head
IPC: B23Q1/48
Filed: 1966-12-19
Abstract: A milling machine comprises a cutter spindle head 40 rotatable about a horizontal axis 38 on a part 26 rotatable on a parallel second axis 28 on a slide 16, the second axis being parallel to and spaced from the axis of a cutter spindle 18 in the slide. The slide 16 is manually- or motor-driven and carries a spindle motor 20 and an upper slide 24 which carries the part 26. A worktable 14 is vertically adjustable. The head 40 may carry a double-ended tool spindle. In the milling position of Fig. 1, the part 26 is bolted to the slides 24 and 16 with the spindle 18 being inoperative. In the drilling position of Fig. 3, the part 26 is bolted to the slide 24 only. The spindle nose 42 then has a clearance b enabling the slide 24 to be completely retracted.
Patent ES-334966-A1 (ES)
Title: Improvements in or relating to pneumatic removal of waste from carding machines
IPC: D01G15/82
Filed: 1966-12-10
Abstract: In a cotton carding-engine, impurities in the form of short fibres, husk fragments and nips are pneumatically removed from beneath the feed roller 10, taker-in 11, main carding cylinder 12 and doffer 13, by an air flow directed from a blast box 27 through an opening 26, along the continuous surface of a guide plate extending the full width of the machine and comprising sections 25, 24 (which may be the supporting floor for the machine) 28, and a downwardly directed section which, together with a lead-in plate 34, forms a funnel or collecting device 29 for the impurities, thence to a suction outlet 35. An air duct, for the main flow and secondary currents created by the rotating cylinders, is defined by these sections, the cylinders themselves, the grid 22 with a perforated section 23 and side and end covers such as 31, 32. The section 28 may comprise separate sections set at an angle to each other in order to ensure that the duct cross-section between section 28 and the grid 22 is constant.
Patent ES-340667-A1 (ES)
Title: Endless belt for paper or board making machine and a method of weaving cloth therefor
IPC: D03D25/00
Filed: 1967-04-29
Abstract: A fourdrinier fabric is twill woven and has the twill pattern reversed at intervals along its length so that the tension of the weft bends the warp threads into transversely directed chevron formations. The reversal may take place at nine inch intervals to deflect the warp threads one-sixth inch. The fabric may be of 40 to 110 mesh and have sixty 0.0096 inch dia. warp threads per inch and fourty five 0.0108 dia. weft threads per inch. The warp and weft may be of metal or synthetic threads or the warp may be metal and the weft synthetic or vice versa. The heald frames for a 2 x 1 twill are shed by levers acted on by cams 23 on a shaft 5 and to reverse the direction of rotation of the shaft 5 is driven by a axially movable clutch 6 that engages either cog wheels 9, 10 or a chain drive 12.