baber/WOPTO huggingface dataset:
Patent FI-881802-A0 (FI)
Inventor: MACHIDA YOSHIMASA
IPC: C07D519/00
Filed: 1988-04-18
Abstract: Novel thiadiazolylacetamide cephem derivatives of the following formula are described. <CHEM> wherein A represents a quaternary ammonio group: or a pharmaceutically acceptable salt thereof. These novel compounds are useful as antibacterial agents, because they have a broad antibacterial spectrum ranging from gram-negative bacteria to gram-positive bacteria. Processes for the preparation of these novel compounds are also described.
Patent FI-894747-A0 (FI)
Inventor: BEY PHILIPPE
IPC: C07C311/36
Filed: 1989-10-06
Abstract: This invention relates to analogs of peptidase substrates in which the nitrogen atom of the scissile amide group of the substrate peptide has been replaced by a substituted malonyl moiety. The contemplated peptidase inhibitors of the foregoing enzymes are selected from the generic formula <CHEM> the hydrates, isosteres or the pharmaceutically acceptable salts thereof wherein X is <CHEM> R1 is hydrogen, an amino protecting group selected from Group K, an alpha -amino acid or a peptide comprised of a number of  alpha -amino acid building blocks, said  alpha -amino acid or peptide optionally bearing on its terminal nitrogen atom an amino protecting group selected from Group K, R2 is the "R group" residue of the  alpha -amino acid responsible for directing the inhibitor to the active site of the enzyme or is -A-SiR7R8R9, C1-10 alkyl, aralkyl or aryl with R7, R8 and R9, each being selected from C1-10, alkyl, aralkyl or aryl and A is a C1-6 alkylene, R4 is the specific R-group residue of the  alpha -amino acid for that peptidase substrate analog, R5 is an  alpha -amino acid or peptide comprised of  alpha -amino acids or is deleted,  Y is NHR3 or OR3 with R3 being H, C1-7 alkyl, benzyl or phenethyl. These analogs of the peptidase substrates provide specific enzyme inhibitors for a variety of proteases, the inhibition of which will have useful physiological consequences in a variety of disease states.
Patent FI-900637-A0 (FI)
Inventor: ELORANTA ERKKI
IPC: A63K3/04
Filed: 1990-02-08
Abstract: PCT No. PCT/FI91/00041 Sec. 371 Date Aug. 10, 1992 Sec. 102(e) Date Aug. 10, 1992 PCT Filed Feb. 7, 1991 PCT Pub. No. WO91/12060 PCT Pub. Date Aug. 22, 1991.A cupholder for supporting a hurdle boom (10) includes a gliding part (1) which is sleeve-like and mounted around a pillar so as to be moved vertically on the pillar and a support (2) on which the end of the boom (1) is supported. The sleeve-like gliding part is broken at one point and a locking apparatus for the gliding part if formed by a tightening apparatus which pulls the opposite edges of the gliding part towards each other so that the gliding part presses against the pillar.
Patent FI-903446-A0 (FI)
Inventor: SAGAMI HIROSHI
IPC: C25B13/08
Filed: 1990-07-06
Abstract: A cation exchange membrane having high durability, which is adapted for use in electrolysis of an alkali metal chloride, which comprises a quadrilateral base membrane and, disposed on at least one marginal area of one surface of the base membrane, a diffusion coating having a capability for an alkali metal hydroxide to diffuse therethrough at a diffusion velocity greater than that at which the alkali metal hydroxide diffuses through a fluorocarbon polymer layer constituting the base membrane when the base membrane is composed of one fluorocarbon polymer layer or through one outermost layer of the base membrane which layer has thereon the diffusion coating and has a water sorption smaller than that of the opposite outermost layer of the base membrane, when the base membrane is composed of a plurality of fluorocarbon polymer layers. The cation exchange membrane is free, for a prolonged period of time, from the local lowering of the mechanical strength of the membrane as caused by the precipitation of an alkali metal chloride within and the formation of oxygen in nascent state within the base membrane during the electrolysis of an alkali metal chloride.
Patent FI-912436-A0 (FI)
Inventor: QUEEN CARY L
IPC: A61P21/04
Filed: 1991-05-20
Abstract: Compsn. comprises a pure human-like immunoglobulin (Ig) which (a) reacts specifically with p55 Tac protein and/or (b) inhibits binding of human interleukin-2 (IL-2) to its receptor. Also new are (1) human-like Ig having 2 pairs of light/heavy chains and able to react specifically with an epitope of a human IL-2 receptor with affinity at least 10 power 8 per mole, the chains including complementarily determg. regions (CDR's) and human-like framework regions (FR's), the CDR's being from different Ig molecules than FR's; (2) humanised Ig (hIg) which can bind to IL-2 receptors and contain at least one CDR from anti-Tac antibody in a human-like FR contg. at least one amino acid from the anti-Tac antibody; (3) nucleic acid encoding for human-like FR and at least one murine CDR, and (4) cells transfected with nucleic acid.
Patent FI-924458-A0 (FI)
Inventor: STERLING JEFF
IPC: A61P25/24
Filed: 1992-10-02
Abstract: N-propargyl-1-amonoindan monofluorinated in the phenyl ring and their use as selective inhibitors of monoamine oxidase (MAO). There are provided several processes for the preparation of these novel compounds. There are also provided as novel compounds 1-aminoindans monofluorinated in the phenyl ring, which serve as intermediates in the preparation of the corresponding novel N-propargyl derivatives.
Patent FI-933656-A0 (FI)
Inventor: COE JOTHAM W
IPC: C07D/
Filed: 1993-08-19
Abstract: 2,4-diaminoquinazoline derivatives as potentiators of chemotherapeutic agents in the treatment of cancer.
Patent FI-934805-A0 (FI)
Inventor: VON NORDENSKJOELD REINHART
IPC: C02F3/26
Filed: 1993-10-29
Abstract: The invention relates to a method and a device for purifying waste water in a plurality of sequentially following phases, the waste water (effluent) being aerated in a first phase A, and then being given a preliminary clarification in a second phase B, and then, in a third phase C, secondary aeration and, in a fourth phase D, secondary sedimentation being carried out. Phases with circulation only can be provided directly upstream of the phases, and filtering and storing phases can be provided directly downstream. In order to achieve a simple, space-saving, inexpensive and nevertheless reliable device, carrying out all four purification phases in one tank is provided according to the invention. In order to make possible adaptation to increasing loads and a changing ratio of hydraulic to biochemical load, the partitions between the phases are arranged to be slidable to change their volumes. <IMAGE>
Patent FI-934916-A0 (FI)
Inventor: RELIGA ZBIGNIEW
IPC: A61F2/24
Filed: 1993-11-05
Abstract: PCT No. PCT/EP92/01018 Sec. 371 Date Jan. 14, 1994 Sec. 102(e) Date Jan. 14, 1994 PCT Filed May 8, 1992 PCT Pub. No. WO92/19185 PCT Pub. Date Nov. 12, 1992.An elastic textile covering is applied over an annular support of a heart valve prosthesis by inserting the preferably collar shaped textile covering through the annular support, turning two projecting axial ends of the textile covering over the outer surface of the annular support and then joining the two axial ends to each other to form a seam that preferably extends entirely around an outer periphery of the annular support. This seam can be concealed by a collar, which also may be covered by the textile covering. An apparatus for applying the textile covering to the annular support includes two coaxial annular rings into which the annular support and textile covering are inserted. Each of the rings includes structure for attachment to a respective axial end of the textile covering.
Patent FI-935596-A0 (FI)
Inventor: TROUGOUBOFF EMILE
IPC: E01F13/00
Filed: 1993-12-13
Abstract: PCT No. PCT/FR92/00531 Sec. 371 Date Mar. 7, 1994 Sec. 102(e) Date Mar. 7, 1994 PCT Filed Jun. 12, 1992 PCT Pub. No. WO92/22709 PCT Pub. Date Dec. 23, 1992.A barrier for the protection of reserved areas including at least one upper element (1) rotatably mounted relative to a lower element (6) anchored in the ground (G). An elastic return spring (18) is interposed between the upper and lower elements (1,6). The upper element (1) is adapted to be displaced to either side of an upright reference position by rotating about a horizontal pin (2) provided on the lower element (6). A releasable mechanism selectively blocks rotation of the upper element in a first direction (F2) and a non-releasable mechanism blocks rotation of the upper element in the reverse direction (F1) at the end of a limited angular deflection. The elastic return spring provides a force opposing the limited deflection in the reverse direction.
Patent FI-940752-A0 (FI)
Inventor: GIACOBBE JAMES
IPC: C08F297/08
Filed: 1994-02-17
Abstract: A film or sheet material 95-60 wt. % heteroplastic olefin polymer compsn. (I) and 5-40 wt. % of an ethylene alpha-olefin copolymer (II) of density 0.890-0.940 g/cc in which the alpha-olefin is of formula CH2=CHR (R = 1-8C alkyl). The heteroplastic olefin polymer compsn. (I) comprises 10-50 wt. % propylene polymer (III), 5-20 wt. % semi-crystalline linear copolymer fraction (IV) and 40-80 wt. % xylene-soluble copolymer fraction (V). (III) has an isotactic index greater than 80 and is propylene homopolymer or a copolymer contg. over 80 wt. % propylene with ethylene and/or a 4-10C alpha-olefin. (IV) has a crystallinity of 20-60 % and is insoluble in xylene at room temp. (IV) is a copolymer of ethylene and propylene contg. over 55 wt. % ethylene, or a copolymer of ethylene, propylene and 1-10 wt. % 4-10C alpha-olefin in which the combined content of ethylene and 4-10C alpha-olefin is over 55 wt. %, as a copolymer of ethylene and a 4-10C alpha olefin contg. over 55 wt. % 4-10C alpha-olefin. (V) has a intrinsic viscosity of 1.5-4.0 dl/g and is a copolymer of ethylene and propylene contg. 20-40 wt. % ethylene at a copolymer of ethylene, propylene and 1-10 wt. % 4-10C alpha-olefin in which the combined content of ethylene and 4-10C alpha-olefin is 20-40 wt. % or a copolymer of ethylene, 4-10C alpha-olefin and opt. 0.5-10 wt. %, diene, in which the 4-10C alpha-olefin content is 20-40 wt. %. The wt. ratio of (IV):(V) is less than 0.4:1. (I) is prepd. by polymerisation in at least 2 stages.
Patent FI-942035-A0 (FI)
Inventor: FRYKLUND LINDA
IPC: A61M5/24
Filed: 1994-05-03
Abstract: PCT No. PCT/SE92/00654 Sec. 371 Date Sep. 26, 1994 Sec. 102(e) Date Sep. 26, 1994 PCT Filed Sep. 23, 1992 PCT Pub. No. WO93/08854 PCT Pub. Date May 13, 1993A liquid preparation of a pharmaceutically active agent having a defined composation is repeatedly dosed from a multi-dose container having a defined volume. The amount dosed is selected as 1/N of the volume of the multi-dose container, N being an integer having a value of 2 or higher. A device for dosing a liquid preparation comprises a holder (1) for a multi-dose container (2), which has a movable rear wall (5) acting as a piston for expelling the liquid preparation (6) from the container, and a piston rod (7), which is provided with releasable blocking means (11, 14, 19, 22), such that the movement of the piston rod is limited to a preset length (35) corresponding to an expelled volume of 1/N of the volume of said multi-dose container, N being an integer having a value of 2 or higher. A preferred embodiment of the device is as an injection device for repeated parenteral injections from an injection cartridge.
Patent FI-944949-A0 (FI)
Inventor: MORELLO FREDERICK
IPC: B21D13/04
Filed: 1994-10-21
Abstract: A metal building is formed of adjacent preformed panels of generally U-shape with crimpable edges, the edges of adjacent panels being crimped together to form the building, the building having straight side walls and a continuous arched curved roof in which the side walls are reinforced by similar shaped straight panels positioned against the side walls to form cavities, which cavities may be filled with reinforcing material, electrical conduits and the like.
Patent FI-945587-A0 (FI)
Inventor: MARTIN-COCHER JEAN-PAUL
IPC: B65B11/58
Filed: 1994-11-28
Abstract: Method of wrapping a load and device for carrying out said method. The method of wrapping a load placed on a pallet consists in covering the load with one or more plastic films which obstruct the pallet apertures. The invention is characterized by forming, in the film obstructing the pallet apertures, permanent passages for the forks of handling units. Application especially in wrapping loads transported on standard pallets.
Patent FI-952686-A0 (FI)
Inventor: SRIVATSA NARARDRA R
IPC: C09K23/44
Filed: 1995-06-01
Abstract: Deinking of impact and nonimpact printed paper is accomplished by repulping the printed paper in an alkali aqueous medium containing a deinking composition comprising one or more nonionic surfactants and/or alkanols. The presence of the deinking composition causes ink particles to agglomerate, which are removed from the aqueous medium by size and density separation. The invention provides an agglomeration method with high ink removal from all types of impact and nonimpact printed paper.
Patent FI-954304-A0 (FI)
Inventor: BAZIARD-MOUYSSET GENEVIEVE
IPC: C07D311/20
Filed: 1995-09-13
Abstract: Arylalkyl piperazino alkyl benzopyran derivs. of formula (I), their optical isomers and acid and base addn. salts, are new. Ar = phenyl or naphthyl (both opt. substd. by 1-3 OH, alkyl (opt. substd. by one or more halo), alkoxy or halo); n = 1-4; when Rb = alkyl, then A = bond and Ra, Rc = H, halo, alkyl (opt. substd. by one or more halo) or alkoxy; when Rb+Rc = -(CH2)q-, then A = -(CH2)p- and Ra = OH or alkoxy in position 5, or H or halo ; or when Rb+Rc = -CH= single bonded to the aromatic ring, then A = CH2 and Ra = H, OH or alkoxy in position 5; or Rb+Rc = bond, then A = -C(=O)-CH= and Ra = H, hydroxy or alkoxy; p = 0- 2; q = 0- 2; provided that p + q = 1 or 2; when Rb = alkyl, then X, Y = H; or CXY = CO and Rd = H or alkyl; when Rb+Rc = (CH2)2 or -CH= then X, Y = H and Rd = H; all alkyl, alkoxy = 1-6C.
Patent IL-70819-A0 (IL)
Title: Substituted diamine hardeners,epoxy compositions containing the same and composites formed therewith
IPC: C08L27/00
Filed: 1984-01-30
Abstract: Described herein is a composition comprising a select group of substituted diamine hardeners and an expoxy resin containing two or more 1,2-epoxide groups per molecule. These compositions exhibit reduced moisture absorption, and controlled reactivity which comprises the processing characteristics of the composition.
Patent IL-78369-A0 (IL)
Title: Quick-attachable connectors particularly for use as a hose coupler
IPC: F16L37/08
Filed: 1986-03-31
Abstract: A female connector member (4) for use in a quickly-attachable connector assembly with a male connector member (6) comprises a housing (10) formed with a socket for receiving the male connector member (6) and further formed with a pair of circumferentially-spaced openings (22) through a wall leading into said socket; and a locking member (8) having a flexible arcuate section (30) received on the outer face of the housing (10), and a pair of locking elements (32) normally projecting through the openings (22) into the socket for locking the male connector member (6) therein. The outer faces of the locking elements (32) are inclined at an acute angle to the longitudinal axis of the socket and converge in the direction of the mouth of the socket, such as not only to facilitate the insertion of the male connector member (6) into the socket by a small push force but also to lock the male connector member (6) against withdrawal from the socket even by a large pull force.
Patent AU-PP355798-A0 (AU)
Title: Process for the production of ultrafine powders
IPC: C01F17/235
Filed: 1998-05-15
Abstract: A process for the production of ultrafine powders that includes subjecting a mixture of precursor metal compound and a non-reactant diluent phase to mechanical milling whereby the process of mechanical activation reduces the microstructure of the mixture to the form of nano-sized grains of the metal compound uniformly dispersed in the diluent phase. The process also includes heat treating the mixture of nano-sized grains of the metal compound uniformly dispersed in the diluent phase to convert the nano-sized grains of the metal compound into a metal oxide phase. The process further includes removing the diluent phase such that the nano-sized grains of the metal oxide phase are left behind in the form of an ultrafine powder.
Patent IL-100865-A0 (IL)
Title: Formulations of crop protection agents
IPC: A01N53/08
Filed: 1992-02-04
Abstract: The invention relates to water-emulsifiable granules of plant protection agents comprising the pesticidal active substance in liquid or dissolved form and a coating- and structure-imparting material which is at least partially soluble in water, to the use of these granules as new, advantageous plant protection formulations, and to processes for their preparation. Furthermore, it relates quite generally to the use of polyvinyl alcohols as coating- and structure-imparting materials in the preparation of water-emulsifiable granules which contain organic compounds dissolved in a high-boiling solvent or solvent mixture.
Patent IL-106087-A0 (IL)
Title: The use of condensed bis-(3,4-dihydro-1-pyridinyl)methanes for the production of pharmaceutical preparations
IPC: A61P1/00
Filed: 1993-06-21
Abstract: Benzo- and thieno-3,4-dihydropyridine derivates having general formula (I), in which D stands for a group having formula (Ia), A and B standing for a benzo- or thieno residue, R2, R3, R5, R6, R7, R11, R12, m and n being as defined in the description, and their pharmaceutically tolerable salts, are used for preparing agents for treating chronic inflammatory processes, colitis ulcerosa and Crohn's disease, and antiproliferative agents.
Patent IL-106147-A0 (IL)
Title: 4-iminoquinolines,processes for their preparation,and their use
IPC: C07D401/12
Filed: 1993-06-25
Abstract: Compounds of the formula I <IMAGE>  and their tautomeric forms, of the general formula Ia <IMAGE>  Ib and Ic <IMAGE> in which the substituents R<1>-R<4> and X and Y have the meanings mentioned, have an antiviral activity.
Patent IL-110039-A0 (IL)
Title: Method for producing enzymatically active human superoxide dismutase in bacteria
IPC: A61K38/44
Filed: 1985-08-26
Abstract: (1) Vector that on introduction into a suitable bacterial host cell contg. the thermolabile repressor C (I) renders the host cell capable, when the temp. is raised to a level at which the repressor is inactivated, of effecting expression of a desired gene inserted in the vector to produce polypeptide (I) encoded by the gene is new when it comprises a double-stranded DNA molecule including in 5'- to 3'- order. (a) DNA sequence contg. the promoter and operator P(L)O(L) from lambda bacteriophage; (b) a N utilisation site for binding antiterminator N protein; (c) a first restriction enzyme site permitting replacement of the DNA sequence contg. the ribosomal binding site following after; (d) DNA sequence contg. a ribosomal binding site for making the MRNA of the desired gene capable of binding to ribosomes in the host cell; (e) ATG initiator codon or a DNA sequence converted into the codon on insertion of the desired gene into the vector; and (f) a second restriction enzyme site for inserting the desired gene into the vector in phase with the ATG initiation codon; and (g) a DNA sequence contg. an origin of replication from a bacterial plasmid capable of autonomous replication in the host cell; and for selection, DNA sequence contg. a gene associated with a selectable or identifiable phenotypic trait manifested when the vector is present in the host cell, or DNA sequence contg. fragment C (I) 434, including the gene for the C (I) 434 repressor protein and its associated promoter and operator sequence.
Patent IL-119450-A0 (IL)
Title: Process for preparing optically active carboxylic acids
IPC: C07D213/89
Filed: 1996-10-20
Abstract: This invention relates to a process for preparing optically active carboxylic acids by oxidizing an optically active aldehyde with a peracid in the presence of an amine and/or amine N-oxide catalyst selected from the group consisting of a substituted or unsubstituted alkyl amine, alkyl amine N-oxide, aromatic amine, aromatic amine N-oxide, heterocyclic amine, heterocyclic amine N-oxide and mixtures thereof, to produce the optically active carboxylic acid. Such optically active carboxylic acids have utility for example as pharmaceuticals.
Patent IL-123497-A0 (IL)
Title: System for transmission of electronic mail
IPC: H04W88/18
Filed: 1996-08-30
Abstract: The present invention relates to a system and to a host arrangement for transferring electronic mail over a mobile telephone network with the aid of SMS message routing means existing in the network. According to the invention, e-mail is coupled with a modified SMS message containing an agent which, through the medium of control characters, is recognized in the addressed mobile station. A client function in the computer decodes the agent and initiates the transfer of e-mail from the host arrangement, wherein the mail is loaded into the computer from the mobile station, via a PCMCIA connection.
Patent IL-137274-A0 (IL)
Title: Lubrificating oil reconditioning system
IPC: F01M11/03
Filed: 1999-01-12
Abstract: Apparatus and methods for improved in-line contaminant removal from engine lubricating oil are provided which employ gravity to achieve a desired flow rate of oil. The invention is adapted for use with an existing engine oil lubrication system and continuously processes a side stream that after processing, is returned to the engine oil. During processing, the oil is first filtered and then drained and deposited upon the upper central surface portions of a heated dome whereon the oil forms a thin film from which relatively low boiling volatile impurities (especially water) are rapidly separated in a gaseous state. The gas is vented through a pressure relief valve to the manifold while the recovered reconditioned oil is collected and recycled.
Patent IL-138632-A0 (IL)
Title: Multiple view endoscopes
IPC: A61B1/00
Filed: 2000-09-21
Abstract: An endoscope comprises a sheath, an articulation section adjacent to its distal tip, and two or more separate optical channels that produce two or more distinct views. Each of the optical channels comprises an objective lens and a means of capturing and/or viewing the image. The objective lens or lenses of the optical channel that produces the first distinct view, is located at a first location on the distal tip. The objective lens or lenses of the optical channel that produces the second distinct view is located at a second location on the proximal end of the articulation section or on the sheath of the endoscope adjacent to or located proximally of the articulation section.
Patent IL-140139-A0 (IL)
Title: Microgels and process for their preparation
IPC: C08F4/40
Filed: 1999-07-09
Abstract: A process for preparing microgel(s) that uses a wide range of activatable prepolymers; in the process, a polymer composition of crosslinked component A and soluble components B and C is formed from mono-olefinic and multi-olefinic monomers in the presence of catalyst and initiator; the process comprises:I) introducing mono-olefinic monomer, catalyst, and initiator into a reactor in the absence of multi-olefinic monomer and producing an activatable prepolymer, component B;II) contacting the product of I) with multi-olefinic monomer to produce components A and C, optionally in the presence of additional initiator; also optionally in the presence of additional mono-olefinic monomer and initiator; the ratio of components A/(B+C) can be controlled by varying the mole ratio of Component B/multi-olefinic monomer from 0.05/1 up to 5/1, by decreasing the mole ratio to increase the ratio of A/(B+C), and increasing the mole ratio to decrease the ratio of A/(B+C).