baber/WOPTO huggingface dataset:
Patent CN-100567944-C (CN)
Inventor: YANFA GAO
IPC: G01N11/00
Filed: 2006-10-24
Granted: 2009-12-09
Abstract: 本发明公开了一种材料流变扰动效应实验系统及实验方法，包括恒载加载系统，通过加载装置、曲轴扩力装置和传力连杆实现对试件施加恒定载荷；还包括扰动加载系统，通过冲击扰动加载装置和爆破扰动加载装置实现对试件施加冲击扰动载荷及爆破扰动载荷；还包括围压加载系统，通过三轴压力箱对试件施加围压载荷。三轴压力箱包括密闭箱体，密闭箱体内设有环形胶囊，可实现对试件施加围压载荷。通过上述材料流变扰动效应实验系统可以实现对试件进行单轴流变实验、单轴流变扰动实验、三轴流变试验、三轴流变扰动实验。结构简单、成本低、测试精确，适用于对各种材料试件进行流变扰动试验，尤其适用于对岩石试件进行长时间流变扰动实验。
Patent CN-100582576-C (CN)
Title: 无氧碳化危险固体废物处置装置
Inventor: XUEJIANG WANG
IPC: F23G5/027
Filed: 2006-07-24
Granted: 2010-01-20
Abstract: 一种无氧碳化固体危险废物处置装置，无氧热解区有一个耐火保温壳体，其下部是加热炉、中部是可燃气体燃烧室，上部是炉膛火道，炉膛火道的内部悬置热解罐，热解罐的顶部的密封开启加料口与上方加料器对应，热解罐的顶侧与可燃气体排出管连通，可燃气体排出管的下端与可燃气体燃烧室连通，热解罐底部侧面连接出碴器，耐火保温壳体的顶侧开有与风动急冷区连通烟气出口，风动急冷区外壳上部开有高温烟气入口，下部开有低温烟气出口，内部置有冷风管束和烟气导向板，风动急冷区外壳的底部置有风机，顶部有排气口。可将有机化合物转化为无害可燃气体和固体碳化废物。适用于各种工业固体废物、医疗废物的处置，达到无害化，减量化，保护环境。
Patent CN-100533973-C (CN)
Inventor: CAIYONG LIU
IPC: H03H21/00
Filed: 2007-07-10
Granted: 2009-08-26
Abstract: 本发明提供了一种最小均方差自适应滤波器及其实现方法。所述最小均方差自适应滤波器充分利用了滤波器的半并行结构，从而实现了乘法器的复用，进而减少了乘法器的使用量；采用延时器的方法解决了滤波器半并行结构导致的抽头系数的存储控制问题，从而使得抽头系数不需存储，而且系数更新也可以实现流水的方式；所述方法可以还可以通过动态地对最小均方差自适应滤波器中使用的抽头个数进行调整，以适应不同抽头数量的需求。
Patent CN-100541232-C (CN)
Inventor: DIFENG WANG
IPC: G01S17/89
Filed: 2007-09-04
Granted: 2009-09-16
Abstract: 本发明公开了一种无姿态信息条件下的航空多光谱扫描仪几何粗校正方法。包括如下步骤：1)对多光谱扫描仪数据进行坐标转换，将WGS-84大地坐标系下的测量观测值转换为高斯平面直角坐标下的值；2)根据理想飞行模型，利用1秒模式模拟滚动角；3)在竖直平面内根据高度数据拟合一条曲线，然后根据曲线的切向计算每一个更新数据点处的飞行俯仰角；4)利用中心投影构像方程求得机下点坐标；5)由扫描方式，根据飞行高度、扫描角、瞬时扫描角求取同一扫描行其它点的坐标；6)利用直接法生成粗校正后的图像。本发明提高了航空遥感的地理精度，是对无姿态信息条件下遥感技术的一项创新，提高时效性，使航空遥感技术能够更好的应用于国民经济生产生活中。
Patent CN-100523522-C (CN)
Title: 一种万向液压联结器
Inventor: PING WU
IPC: F15B15/20
Filed: 2007-03-14
Granted: 2009-08-05
Abstract: 本发明属于一种联接装置，具体公开一种万向液压联结器。其特点是作为整体的支耳、横轴和供油回转轴一起转动，供油回转轴在轴套内转动，从而形成一个回转自由度；由于支耳与供油回转轴的槽孔沿供油回转轴的轴向有一定的间隙，所以支耳可以在间隙形成的空间内绕横轴发生一定旋转，从而形成另一个回转自由度。此外，由于供油回转轴的油路与横轴的油路相通，横轴的油路与支耳的油路相通，支耳的油路与液压缸的油路相通，因此，本发明不需要软管，避免了软管破裂对安全性能的影响，因此，本发明的显著优点是回转灵活、安全性能好。本发明可用于承载的联接装置。
Patent CN-100452056-C (CN)
Title: 解析存储器内容的系统及方法
Inventor: YIHONG KE
IPC: G06F17/30
Filed: 2007-06-25
Granted: 2009-01-14
Abstract: 本发明提供一种解析存储器内容的系统及方法。其中该方法提供一定义文件，该定义文件包括至少一存储器地址及与其对应的至少一参数值，该参数值对应于一事件描述，接着，经由该存储器地址的载入，撷取一存储器内对应该存储器地址的至少一内容信息，之后，比对该参数值与该内容信息，以自动取得并显示对应该参数值的该内容信息的该事件描述，借此，透过自动化的技术，让使用者可便于得知该内容信息对应的事件描述，且进一步达成提升使用者的工作效率的目的。
Patent CN-100516564-C (CN)
Inventor: MIAOGEN YU
IPC: F16B41/00
Filed: 2007-09-18
Granted: 2009-07-22
Abstract: 螺旋楔锁紧式螺母防松防盗装置，由薄壁套筒、圆形螺垫片和螺旋楔组成，薄壁套筒的筒底内孔设有一周左右的螺旋面，在螺旋面的最前端有一穿通的开口，这样筒底的螺旋面就能把螺旋楔压紧在圆形螺垫片的内孔锥面上，而螺旋面前端的缺口又能顶住螺旋楔大端的尾部，由于薄壁套筒的大端内孔与圆形螺垫片的外圆之间为过盈配合，因此薄壁套筒可以把螺旋楔、圆形螺垫片连接成一体。只要控制好螺旋楔安装的初始位置，就可把它们一起顺利地拧在所要保护的螺栓螺母上，安装十分方便无须专用工具。而当该装置逆时针反转时，薄壁套筒内的螺旋面缺口即与螺旋楔大端尾部脱开，这时圆形螺垫片内的不完整螺牙牙顶则压紧螺旋楔，当该装置在螺栓上反转角度越大，则锁紧效果越好，达到螺母防松防盗的目的。
Patent CN-100507335-C (CN)
Inventor: FENGCHUN WANG
IPC: F16L3/08
Filed: 2007-10-31
Granted: 2009-07-01
Abstract: 本发明公开了一种海缆锚固装置，它包括底座，底座上设置有倒锥孔，倒锥孔中设置有倒锥形套，倒锥形套外表面与倒锥孔内表面相互配合，底座上方设置有压板，压板通过连接件与底座固定连接，压板上设置有环形夹紧面，环形夹紧面与倒锥形套上段弧面相互配合，底座边缘设置有与外部连接的安装孔，本发明的优点在于由于压板的环形夹紧面与倒锥形套上段弧面的相互配合及倒锥形套与底座上的倒锥孔的相互配合，当使用利用压板使倒锥形套基本与倒锥孔内表面密合，由于海缆的自重，使得倒锥形套与倒锥孔内表面更为夹紧，从而海缆被有效地固定于工作平台上；本发明具有高机械强度、高耐海水腐蚀性；本发明结构简单，工作可靠，还可用于深井作业等其他平台中。
Patent CN-100538377-C (CN)
Title: 确定特高压交流线路与调幅广播电台间防护距离的缩比模型试验方法
Inventor: ZHEYUAN GAN
IPC: G01R31/00
Filed: 2007-12-20
Granted: 2009-09-09
Abstract: 本发明涉及一种确定特高压交流线路与调幅广播电台间防护距离的缩比模型试验方法，所采用的方法是：将实物尺寸按照一定比例缩小制成缩比模型，将天线建立为形状与实物完全或近似相同的微缩天线模型，且使激励模型的源波长与被研究的实际波长相比也按照同一比例缩小，这样就使得长度与波长之比保持不变，模型天线与被研究对象在工作波长下有相同的电参数和特性，测量模型天线的参数就能够得的被研究对象的性能。本发明可应用于高压输电线路与其他类型相邻无线电台站间电磁防护间距的精确计算。
Patent MX-3055-E (MX)
Title: Procedimiento para la preparacion de derivados de histidina
Inventor: MORGAN BARRY ARNOLD
IPC: C07K5/097
Filed: 1976-03-08
Abstract: La presente invención se refiere a procedimiento para la preparación de derivados de histidina de la fórmula: (VER FIGURA) en la cual R es hidrógeno o alquilo C1-3'R1 es alquilo o alcoxi(ver gaceta ), C1-3'R2 es hidrógeno, alquilo o alcoxi, C1-3'R3 es higrógeno, alquilo C1-6 o cicloalquilo, C3-6 y R4 es hidrógeno o alquilo, C1-6' caracterizado porque un compuesto de la fórmula II: en donde A e Y son respectivamente un grupo protector o un grupo capaz de formar un enlace de péptido, en primer lugar se acopla con (VER FIGURA) (a) un copuesto de la fórmula III, en donde B es hidrógeno o un grupo protector y X es un grupo capaz de formar un enlace de péptido; o bien (b) un compuesto de la fórmula IV; y en segundo término, el dipéptido resultante se acopla con el otro compuesto, y en seguida se remueven los grupos protectores.
Patent FR-84892-E (FR)
Inventor: BARCLAY JOHN LYNN
IPC: B01J23/18
Filed: 1963-12-06
Granted: 1965-04-30
Abstract: Acrylonitrile or methacrylonitrile are prepared by reacting propylene or isobutene at an elevated temperature in the vapour phase with oxygen and ammonia over an oxidation catalyst comprising (i) a mixture of the oxides of antimony and tin, and/or (ii) a compound of antimony, tin and oxygen (see Group III).ALSO:Catalysts suitable for the production of acrylonitrile and methacrylonitrile (see Group IV(b)) comprise (i) a mixture of the oxides of antimony and tin, and/or (ii) a compound of antimony, tin and oxygen, such as tin antimonate.  The catalyst may be prepared from the oxides or from compounds, such as the hydroxides, which on heating in the presence of an oxygen-containing gas are converted to the oxides.  Specified oxides are antimony trioxide, tetroxide and pentoxide and their mixtures; stannic oxide, stannous oxide, metastannic acid and their mixtures.  Hydrated forms of the oxides may be used, such as those formed by the action of aqueous nitric acid on antimony or tin metals or their mixtures.  The catalyst mixture may be pre-heated in the presence of an oxygen-containing gas such as air, for instance at a temperature between 550 and 1100 DEG C. Cationic salts of the metals, such as the chlorides may be hydrolysed with water or aqueous ammonia and the resulting precipitate heated.  The catalyst may be supported, e.g. on silica.
Patent PT-1057851-E (PT)
Inventor: KOEHLER BURKHARD
IPC: B32B5/18
Filed: 2000-05-12
Abstract: A composite material comprises (A) a layer of polyurethane (PUR) directly bonded with (B) a layer of a different thermoplastic. (A) contains homogeneously dispersed particles, of size 1-10 nm, coated with a thermoplastic other than (A) and showing a total surface area at least equal to the total interfacial area between (A) and (B). An Independent claim is also included for a process for the production of this material by applying layer (A) to layer (B).
Patent PT-1219104-E (PT)
Title: Method for changing the charge type during an established connection
Inventor: COSTA JEAN-PAUL
IPC: H04M3/51
Filed: 2000-02-28
Abstract: The invention relates to a method with which the charge rate for an established connection between a caller (10) and an agent (12) can be changed while said connection persists. The connection is guided through at least one switch (110), said switch (110) being controlled by an overriding server (SCP) (111/119). Said agent (12) can change the charge rate by transmitting a corresponding instruction directly to said server (111/119).
Patent PT-1270555-E (PT)
Inventor: RAMON BERENGUER MAIMO
IPC: A61P1/04
Filed: 2001-03-08
Abstract: The present invention relates to a procedure for the oxidation of a thioether group to a sulfoxide group, with aqueous sodium percarbonate in the presence of a molybdenum salt as a catalyst. The procedure is of application to oxidize the thioether group of a compound (I), where R1 is a C1-C6 alkyl, a halogenated C1-C6 alkyl, or -(CH2)n-OR9, where n is an integer between 1 and 6 and R9 is H or a C1-C6 alkyl; R2, R3, R4, R5, R6 and R8, independently form each other represent H, a C1-C6 alkyl, or C1-C6 alkoxy; and R7 is H, a C1-C6 alkyl, a C1-C6 alkoxy or a C1-C6 fluorinated alkoxy, in order to obtain the sulfinyl derivative (II). <CHEM>
Patent PT-1323222-E (PT)
Title: Island network and method for operation of an island network
Inventor: WOBBEN ALOYS
IPC: F03D9/00
Filed: 2001-09-05
Abstract: The arrangement has at least one first energy generator using a regenerative energy source, preferably a wind power system (10) with a generator, and a second generator (32) for coupling to an internal combustion engine (30). The revolution rate and blade setting of the wind power generator can be controlled and there is an electromagnetic coupling (34) between the second generator and internal combustion engine. Independent claims are also included for the following: a method of operational control of an electrical island network with at least one wind power system and the use of a synchronous generator as a network mimic for a mains inverter.
Patent PT-1281790-E (PT)
Inventor: REINHARD GEORG
IPC: C23F11/02
Filed: 2002-06-12
Abstract: A corrosion inhibiting composition comprises: (a) an inorganic salt of nitric acid, (b) a water-insoluble multi-substituted phenol, (c) an aliphatic ester of a di-hydroxybenzoic acid and (d) tocopherol (2,5,7,8-tetramethyl-2-(4',8',12'-trimethyltridecyl) chroman-6-ol). An Independent claim is also included for a process for the production of a sublimatable corrosion inhibiting composition (I) by mixing together components (a)-(d).
Patent PT-1372892-E (PT)
Inventor: DI DOMENICO GIAMPIERO
IPC: B22D41/30
Filed: 2002-03-04
Abstract: The invention relates to a process for repairing refractory plate (1), having a pouring hole (3), circumscribed by a circle C of center (4), at least a portion of the edges (15, 16, 17, 18) of the plate (1) are angularly oriented so as to focus the clamping forces optimally in the throttling area and around the pouring hole.
Patent PT-1401652-E (PT)
Inventor: MICHAEL EISELE
IPC: B32B27/08
Filed: 2002-06-12
Abstract: The invention relates to a dielectric response elastomer-composition and the use thereof for producing a laminate and a composite, in addition to the linkage of said composite.  The dielectric response elastomer-composition is obtained by the homogeneous distribution of small thermoplastic-particles (7) in an elastomer (8).  A composition of said type can be excited by a dielectric field (6) and has good mechanical properties.
Patent PT-1408142-E (PT)
Title: Saw tooth wire for card clothing
Inventor: GRAF RALPH A
IPC: D01G15/88
Filed: 2003-10-06
Abstract: Both sides (32, 34) of the teeth have regions (40, 50) with lengthwise profiling, comprising projections (42) or grooves (52), both bow-shaped, e.g. with a radius of 0.15 mm, interspersed by straight segments. The depth of the profiling varies along the tooth height in a specified manner. The profiled regions (40, 50) on either tooth flank (32, 34) alternate between grooves and projections and are staggered along the tooth height.  An Independent claim is also included for the following:  (1) A method for making wire of this kind that includes profiling of the wire section along its length while being formed; (2) A doffer roller for a card clothed with this kind of wire.
Patent PT-1608838-E (PT)
Title: Climbing aid for ladders
Inventor: BLASEK FRANK
IPC: E06C7/18
Filed: 2005-02-18
Abstract: The invention relates to a climbing aid for ladders or the like, comprising an endless traction means running between guide pulleys, from which a person may optionally hang by means of a suspension device, with a drive device (20) comprising a drive motor (21), by means of which one of the guide pulleys may be driven as the drive disc (12) for the drive means (13), with a traction force limitation device and with a device for switching the drive device on/off, which can be actuated by the endless traction means (13). According to the invention, the traction force limitation device consists of a slip clutch (30) with torque limitation interposed between the drive disc (12) and the drive motor (21), and the device for switching the drive device on/off comprises sensor means (70) with which a movement of the traction means (13) can be detected, whereby the sensor means (70) are formed in such a manner that a detection of a sensor pulse switches the drive motor (21) on and an absence of sensor pulses within a time span switches the drive motor (21) off.
Patent PT-1841254-E (PT)
Title: Method for defining a zone for location based billing and/or location based services
Inventor: MARSDEN ROGER
IPC: H04W4/02
Filed: 2006-03-29
Abstract: The invention refers to a method for defining a zone for location based billing and/or services, wherein the zone is a part of a geographical area which is served by nodes of a telecommunications network, the method comprising the steps of: 
a) defining a zone within the geographical area, 
b) determining all serving nodes of the telecommunications network which serve said zone defined in step a), 
c) determining an initial area whose geographical perimeter envelopes the physical location of all of said serving nodes, 
d) determining a density vector which has its basis in the centroid of said initial area defined in step c) and which points into the direction of the smallest density of said serving nodes being located in said initial area 
and 
e) determining a final area which has its centroid on said density vector and which is enlarged compared to the initial area so that no serving nodes are located in said final area which are not located in said initial area, wherein the final area is said zone for location based billing.
Patent PT-1945943-E (PT)
Title: Wind turbine blade
Inventor: SCHUON GOTTFRIED
IPC: F03D1/06
Filed: 2006-10-11
Abstract: Wind turbine blade (10) which comprises a root area (13), an enclosure (20) inside the blade at the root area, and means for draining off water that condensates inside the blade. The draining means comprise four bores (30) formed on the surface of the blade at the root area, two at one side of the enclosure and two at the other side; as for their angular position on the surface of the blade, two bores are located on the suction side of the blade and two other bores are located on the pressure side of the blade. The bores (30) are provided with a protrusion (35) protruding outwards from the outer surface of the blade, so that water flowing down the outer surface of the blade is prevented from entering the blade.
Patent PT-2189459-E (PT)
Title: Stable crystalline salt of 5-methyl-(6s)-tetrahydrofolic acid
Inventor: MUELLER HANS RUDOLF
IPC: A23L33/15
Filed: 2000-04-08
Abstract: Crystalline salts of 5-methyl-(6R,S)-, -(6S)- and -(6R)-tetrahydrofolic acid are new. Independent claims are also included for: (1) crystalline calcium salt of 5-methyl-(6S)- and -(6R)-tetrahydrofolic acid; and (2) the preparation of crystalline salts of 5-methyl-(6R,S)-, -(6S)- and 5-methyl-(6R)-tetrahydrofolic acid.
Patent PT-2276821-E (PT)
Title: Electrochromic formulation and organic electrochromic switchable electronic component
Inventor: KANITZ ANDREAS
IPC: C09K9/02
Filed: 2009-05-18
Abstract: An electrochemical formulation has an active dye. An organic electrochromic switchable electronic component of high switching speed is made using the dye. The component is used to make electrochromic displays. The dye has substituents limiting or preventing a π-merisation of the aromatic moieties.
Patent PT-2189088-E (PT)
Title: Beverage distribution apparatus with support system and droplet recuperation for containers with different sizes
Inventor: CAHEN ANTOINE
IPC: B67D7/84
Filed: 2006-06-16
Abstract: The device (1) has a base (2), and a drop recuperation and support system (9), which has a support element (10) to receive a small size container. The element is movable along a deployed support position, to receive the container, and a partially moved position, to push the element so as to liberate a free space permitting to position a large size container in the place of the former container, below an outlet (7) of a beverage. The system has a liquid storage container receiving the liquid recuperated by the element during the moved position, where the element and the container form a slide.
Patent PT-611767-E (PT)
Inventor: KAZDA STANISLAV
IPC: A61K31/41
Filed: 1994-02-02
Abstract: Derivatives of the formula <IMAGE>  in which     B and D together form a radical of the formula <IMAGE>     T is a radical of the formula <IMAGE>  or tetrazolyl.   The compounds can be employed as active ingredients in medicaments for the treatment of arterial high blood pressure and atherosclerosis.
Patent PT-640353-E (PT)
Inventor: DAVIDSON JAMES A
IPC: A61C8/00
Filed: 1994-08-15
Abstract: An implant has a core comprising (a) a Zr-contg. Ti alloy core, (b) a layer surrounding the core comprising an oxygen-rich alloy soln. and (c) a surface layer of mixed oxides of the metals present in the core. Also claimed is a surface-hardened medical implant made by heating a Zr-contg. Ti implant in an environment able to provide oxygen so as to allow oxygen to diffuse into the implant surface, and soaking at this temp. long enough to oxidise the metal at the surface of the implant. This gives a hard mixed-oxide surface layer and an oxygen-rich layer beneath the surface layer. Also claimed is the implant as defined above where the process involves heating to and soaking at 200-1200[deg]C.
Patent PT-608180-E (PT)
Inventor: LETEMPS BERNARD
IPC: H01Q1/32
Filed: 1994-01-19
Abstract: The invention relates to windows, especially compound windows, consisting of at least one sheet (5) of a rigid material, permanently including a surface antenna (13) consisting of at least one microstrip separated from an earth plane by a dielectric. These windows including such an antenna (13) are used for reception and transmission of frequencies higher than 1 GHz, and preferably for the frequency bands 5795-5815 MHz, 63-64 GHz and 74-77 GHz. <IMAGE>
Patent PT-692250-E (PT)
Inventor: BOMBARDELLI EZIO
IPC: A61K31/353
Filed: 1995-07-05
Abstract: The present invention relates to the use of esculoside alone or in combination with adenylate cyclase stimulators, such as forskolin or Salvia miltiorrhiza diterpenes and/or with phosphodiesterase inhibitors, such as apigenine-skeleton dimeric flavones, in topical formulations for the treatment of peripheral vasculopathies related to an impaired peripheral microcirculation, cellulitis or unesthetisms connected with a deposit of superfluous fat. For the reduction of the deposits of superfluous fat of any origin, the above mentioned products are advantageously also combined with caffeine, theophylline and derivatives thereof.
Patent PT-709093-E (PT)
Inventor: SHANNON HARLAN E
IPC: A61K31/4545
Filed: 1995-10-30
Abstract: The present invention provides the use of a compound <CHEM>  wherein  X is oxygen or sulphur; R is hydrogen, amino, halogen, -CHO, -NO2, -OR<4>, -SR<4>, -SOR<4>, -SO2R<4>, C3-7-cycloalkyl, C4-8-(cycloalkylalkyl), -Z-C3-7-cycloalkyl, and -Z-C4-8-(cycloalkylalkyl) wherein R<4> is straight or branched C1-15-alkyl, straight or branched C2-15-alkenyl, straight or branched C2-15-alkynyl, each of which is optionally substituted with one or more halogens, -CF3, -CN, phenyl or phenoxy wherein phenyl or phenoxy is optionally substituted with halogen, -CN, C1-4-alkyl, C1-4-alkoxy, -OCF3, -CONH2 or -CSNH2; or R is phenyl or benzyloxycarbonyl, each of which is optionally substituted with halogen, -CN, C1-4-alkyl, C1-4-alkoxy, -OCF3, -CONH2 or -CSNH2; or R is -OR<5>Y, -SR<5>Y, -OR<5>ZY, -SR<5>ZY, -O-R<4>-Z-R<5> or -S-R<4>-Z-R<5> wherein Z is oxygen or sulphur, R5 is straight or branched C1-15-alkynyl, and Y is a 5 or 6 membered heterocyclic group containing one to four N, O or S atom(s) or a combination thereof, which heterocyclic group is optionally substituted at carbon or nitrogen atom(s) with straight or branched C1-6-alkyl, phenyl or benzyl, or which heterocyclic group is optionally fused with a phenyl group; and G is selected from one of the following azabicyclic rings <CHEM> wherein the thiadiazole or oxadiazole ring can be attached at any carbon atom of the azabicyclic ring; R<1> and R<2> may be present at any position, including the point of attachment of the thiadiazole or oxadiazole ring, and independently are hydrogen, straight or branched C1-5-alkyl, straight or branched C2-5 alkenyl, straight or branched C2-5-alkynyl, straight or branched C1-10-alkoxy, straight or branched C1-5-alkyl substituted with -OH, OR<4>, halogen, -NH2 or carboxy; R<3> is H, straight or branched C1-5-alkyl, straight or branched C2-5-alkenyl or straight or branched C2-5-alkynyl; n is 0, 1 or 2; m is 0, 1 or 2; p is 0, 1 or 2; q is 1 or 2; and --- is a single or double bond; or a pharmaceutically acceptable salt thereof for the manufacture of a medicament for the treatment of anxiety.
Patent PT-820376-E (PT)
Inventor: EVRARD ALAIN
IPC: B29C35/08
Filed: 1996-04-10
Abstract: PCT No. PCT/FR96/00538 Sec. 371 Date Dec. 16, 1997 Sec. 102(e) Date Dec. 16, 1997 PCT Filed Oct. 10, 1996 PCT Pub. No. WO96/32243 PCT Pub. Date Oct. 17, 1996A preform (3) for use in making a container such as a bottle from a thermoplastic material is selectively heated prior to at least one step of blow molding or stretch-blow molding the heated preform. For this purpose, at least most (7A) of the radiation (4) transmitted generally towards the preform by a source (1A) is focused (8) onto a preferred area (A) thereof, the source is located substantially opposite the preferred area of the preform, whereby said the preferred area (A) receives most (7A) of the radiation (4) while the areas adjacent to the preferred area (A) do not receive the radiation fraction initially transmitted towards them by the source.
Patent PT-833818-E (PT)
Inventor: CASELLAS PIERRE
IPC: C07D209/08
Filed: 1996-06-20
Abstract: The use of human CB2 receptor-specific agonists of formula (I) or (I') for preparing immunomodulating drugs is disclosed. In formulae (I) and (I'), R1 is a group selected from -CH2CHR10NR6R11, -(CH2)2NR'6R'11, -CHR9CH2NR'6R'11, -(CH2)nZ and -COR8; R'1 is a -CH2CHR10NR6R11 or -(CH2)2NR'6R'11 group; R2 and R'2 are hydrogen, halogen or C1-4 alkyl; R3 is hydrogen, C1-4 alkyl or a group selected from -CH2CHR10NR6R11, -(CH2)2NR'6R'11 and -COR8; R'3 is a =CR6R8 group; R4 has one of the meanings given for R5 or is a -COR8 group; R5 is hydrogen, C1-4 alkyl, C1-4 alkoxy, a halogen atom, a CF3 group, an OCF3 group or C1-4 alkylthio; R'5 has one of the meanings given for R5 and is in the 5 or 6 position of the indene ring; R6 is hydrogen or C1-4 alkyl; R'6 is C1-4 alkyl; R7 has one of the meanings given for R5 or R7 and R9 together form a -Y-CH2- group attached to the indole ring in the 7 position by a group Y; R8 is phenyl substituted one to four times by a substituent selected from halogen, C1-4 alkyl or C1-4 alkoxy; a polycyclic ring selected from naphth-1-yl, naphth-2-yl, 1,2,3,4-tetrahydronaphth-1-yl, 1,2,3,4-tetrahydronaphth-5-yl, anthryl, benzofuryl, benzothien-2-yl, benzothien-3-yl, 2-, 3-, 4- or 8-quinolyl, said polycyclic rings optionally being substituted once or twice by a substituent selected from C1-4 alkyl, C1-4 alkoxy, C1-4 alkylthio, halogen, cyano, hydroxyl, trifluoromethyl and imidazol-1-yl; R10 and R11 together are a group selected from -CH2-O-CH2-CR12R13- and -(CH2)p-CR12R13-, wherein the carbon atom substituted by R12 and R13 is attached to the nitrogen atom; R'11 is C1-4 alkyl; or R'11 and R'6, taken together with the nitrogen atom to which they are attached, form a group selected from morpholin-4-yl, thiomorpholin-4-yl, piperidin-1-yl and pyrrolidin-1-yl; each of R12 and R13 is independently hydrogen or C1-4 alkyl; n is 2, 3, 4 or 5; p is 2 or 3; Z is a methyl group or a halogen atom; and Y is a methylene group or an oxygen atom.
Patent PT-888353-E (PT)
Inventor: ALTMANN EVA
IPC: C07D487/04
Filed: 1997-03-05
Abstract: PCT No. PCT/EP97/01095 Sec. 371 Date Sep. 10, 1998 Sec. 102(e) Date Sep. 10, 1998 PCT Filed Mar. 5, 1997 PCT Pub. No. WO97/34895 PCT Pub. Date Sep. 25, 1997There are described pyrrolo[2,3]pyrimidines of formula I wherein R1-R5, m and n are as defined in the description. The compounds have valuable pharmaceutical properties and are effective especially as tyrosine protein kinase inhibitors. They can be used in the treatment of bone diseases and other diseases in warm-blooded animals that can be favorably influenced by the inhibition of tyrosine protein kinase.