baber/WOPTO huggingface dataset:
Patent CZ-286325-B6 (CZ)
Title: N-(endo-9-methyl-9-azabicyclo/3,3,1/non-3-yl)-1-methylindazole-3-carboxamide, use thereof for preparing a pharmaceutical preparation and the pharmaceutical preparation containing thereof
Inventor: KING FRANCIS D
IPC: C07D487/08
Filed: 1991-11-01
Abstract: In the present invention there is disclosed N-(endo-9-methyl-9-azabicyclo/3,3,1/non-3-yl)-1-methylindazole-3-carbo xamide of the general formula I, pharmaceutically acceptable salts thereof and use of this substances for preparing a pharmaceutical preparation suitable particularly for treating migraine, vomiting, trigeminal neuralgia and other disorders of central nervous system. In the present invention there is also claimed a pharmaceutical preparation in which the above indicated compound is comprised.
Patent CZ-283757-B6 (CZ)
Title: PROCESS FOR PREPARING 5-CARBAMOYL-5H-DIBENZO[b,f]AZEPINE
Inventor: ACKLIN GEORG DR
IPC: C07D223/22
Filed: 1988-06-16
Abstract: Prodn. of dibenzazepine-N-carboxamides (I), esp. dibenz(b,f)-azepine -5-carboxamide (Ia), is effected by reacting the corresp. dibenzazepine with HOCN. The reaction is pref. effected at 0-120 (esp. 40-80) deg.C in an organic solvent in the presence of an acid. The HOCN is introduced in gaseous form or is formed in situ from NaOCN. The solvent is toluene, xylene, 1,2-dichloroethane, HOAc or EtOAc. The acid is HCl, H2SO4, trichloroacetic acid (TCA) or HOAc.
Patent CZ-285369-B6 (CZ)
Inventor: BOTTCHER HENNING DR
IPC: C07D401/14
Filed: 1995-04-21
Abstract: Derivát 3-indolylpiperidin obecného vzorce I, kde znamená R.sup.1.n., R.sup.2.n., R.sup.3.n. a R.sup.4.n. vždy na sobě nezávisle H, A, OH, OA, F, Cl, Br, J, CN, CF.sub.3.n., COOH, CONH.sub.2.n., CONHA, CONA.sub.2.n. nebo COOA nebo R.sup.1.n. a R.sup.2.n., jakož i R.sup.3.n. a R.sup.4.n. vždy spolu dohromady také methylendioxyskupinu, R.sup.5.n. H nebo OH, R.sup.6.n. H nebo R.sup.5.n. a R.sup.6.n. spolu dohromady vazbu, A C.sub.1-6.n.alkyl a n 2, 3, 4, 5 nebo 6, a jeho fysiologicky vhodné soli jsou účinné na centrální nervový systém a vykazuje zvláště dopamin-agonistické nebo dopaminantagonistické působení.
ŕ
Patent CZ-291572-B6 (CZ)
Title: 4-(Arylaminoethylene)-2,4-dihydropyrazol-3-one derivative, process of its preparation and pharmaceutical preparation in which the derivative is comprised
Inventor: ARLT MICHAEL DR
IPC: A61K31/4427
Filed: 1996-05-16
Abstract: The present invention relates to a 4-(arylaminomethylene)-2,4-dihydropyrazol-3-one derivative of the general formula I, in which Re1 represents benzyl, alkoxybenzyl having 1 to 3 carbon atoms in the alkoxy moiety, phenyl being optionally substituted with 1, 2 or 3 substituents that are selected from a group comprising amino, halogen, NOi2, CN, AO-, carboxyl, sulfonyl, A-O-CO-, A-CO-NH-, A-CO-NA-, carbamoyl, N-alkylcarbamoyl containing 1 to 6 carbon atoms in the alkyl moiety, N,N-dialkylcarbamoyl containing 1 to 6 carbon atoms in the dialkyl moiety, A-O-CO-NH-, A-O-CO-NA-, A-SOi2-, SOi2NRe4Re5, wherein Re4 and Re5 represents hydrogen or alkyl having 1 to 6 carbon atoms, or NRe4Re5 denotes 5- or 6-membered ring having optionally 1 to 2 hetero atoms such as nitrogen, sulfur or oxygen being optionally substituted with A, further the group A-CO-NH-SOi2, A-CO-NA-SOi2-, A-SOi2-NH-, A-SOi2-NA, (A-SOi2)i2N, tetrazolyl and phosphonyl; or Re1 represents pyridyl, Re2 denotes alkyl containing 1 to 5 carbon atoms, alkoxycarbonylalkyl containing 1 to 5 carbon atoms in the alkoxy moiety and 1 to 4 carbon atoms in the alkyl moiety, hydroxyalkyl with 1 to 4 carbon atoms in the alkyl moiety, hydroxycarbonylalkyl containing 1 to 4 carbon atoms in the alkyl moiety, Re3 represents alkyl containing 1 to 5 carbon atoms, alkoxy having 1 to 5 carbon atoms, fluorine- or chlorine-substituted alkyl, A denotes alkyl containing 1 to 6 carbon atoms, fluorine- or chlorite-substituted alkyl with 1 to 6 carbon atoms, and salts thereof. These compounds functioning as selective cGMP inhibitors of specific phosphodiesterases (PDE) are suitable for preparing pharmaceutical preparations intended particularly for treating diseases of heart circulation system and heart insufficiency.
Patent CZ-294506-B6 (CZ)
Title: Clear, concentrated liquid fabric softener microemulsion composition
Inventor: GRANDMAIRE JEAN PAUL
IPC: C11D1/40
Filed: 1995-12-19
Abstract: In the present invention, there is disclosed a clear fabric softener aqueous microemulsion concentrate composition, capable of conversion to a milky macroemulsion upon dilution with water consisting essentially of: (A) a diester quaternary ammonium surfactant fabric softener of the general formula (1) wherein R is an alkylene group having 2 to about 4 carbon atoms, R' is an alkyl or alkenyl group having 8 to about 22 carbon atoms, n is an integer having values of 1 to about 4, and R" is a lower alkyl radical having 1 to about 4 carbon atoms, and/or a diamido ammonium surfactant fabric softener of the general formula (2) wherein n, R and R' are as defined above, Re1 represents a lower alkyl group having 1 to about 4 carbon atoms and X denotes R"Soi4e-, Bre- or Cle- wherein R" represents a lower alkyl group having 1 to about 4 carbon atoms, (B) an organic solvent, (C) an optional water-immiscible oil perfume, (D) an optional fabric co-softener being selected from the group consisting of fatty alcohols, fatty acids, fatty acid esters, fatty amines and/or amidoamines, and (E) a sufficient amount of water to convert the aqueous microemulsion to a milky macroemulsion.
Patent CZ-293747-B6 (CZ)
Title: Aqueous pharmaceutical solution suitable for injection into a host and use thereof
Inventor: BOETTNER WAYNE ALAN
IPC: A61K33/30
Filed: 1996-11-13
Abstract: The present invention relates to an aqueous pharmaceutical solution, which is suitable for injection into a host comprising danofloxacin or a pharmaceutically acceptable salt thereof in an amount ranging from 60 to 200 mg/ml, and (1) a magnesium oxide, or (2) a zinc oxide or zinc acetate in admixture with a co-solvent, whereby the magnesium and zinc compounds and said co-solvent being present in amounts which are sufficient for improved toleration at the injection site. Claimed is also the use of the above-described solution for the preparation of a medicament intended for the treatment of bacterial infections in a host, such as cattle.
Patent CZ-287222-B6 (CZ)
Title: Isolation process of citric acid
Inventor: PENDL JIRI ING
IPC: C07C59/265
Filed: 1999-07-07
Abstract: In the present invention there is disclosed an isolation process of citric acid by fermentation of saccharide sources by making use of Aspergillus niger production strain with subsequent removal of production mycelium from fermentation aqueous solution after fermentation, with the removal of higher-molecular ballast substances by ultrafiltration, decolorizing solutions on activated charcoal, removal of ballast mineral anions on anion-exchange resin and removal ballast cations and residual saccharides on a second anion-exchange resin at simultaneous selective entrapping citric acid, whereby the process is characterized by separate processes for obtaining three different fractions of eluates from the anion-exchange resin. The first fraction contains in addition to residual citric acid residual saccharides, too. This fraction is liquidated in waste water bio-aeration treatment plant or after optional thickening it can be treated by reversible osmosis to citric acid. The second fraction is recycled to a feed on the second anion-exchange resin. The third fraction containing pure citric acid being first subjected to thickening by reversible osmosis and subsequently to thickening in vacuum evaporator is then subjected to a simple crystallization or a multistage recrystallisation and washing with potable water or a condensate under obtaining a product with parameters complying with medicamentous or foodstuff standards.
Patent CZ-293233-B6 (CZ)
Title: Hydroxamic acid derivatives and pharmaceutical composition containing thereof
Inventor: BERTOLINI GIORGIO
IPC: C07D217/04
Filed: 1997-05-12
Abstract: In the present invention, there are disclosed hydroxamic acid derivatives of the general formula  I, in which the individual symbols have meaning indicated in the main Claim. These derivatives are compounds exhibiting antiphlogistic and immunosuppressive activities. Claimed is also a pharmaceutical formulation that can be used for the treatment of inflammatory diseases and immune system disorders.
Patent SK-286337-B6 (SK)
Title: Radioactive contaminated waste dump
Inventor: PLSKO JULIUS
IPC: B09B1/00
Filed: 2005-02-21
Abstract: An invention related waste dump of radioactivity contaminated materials, by which is solution sealing file layers (6), which consists minimum one of least basic drainage and sorptive layer (62), which consists of lignite brash of modification lignite with content humin acid in form of calcium and magnesium salts.
Patent SK-279355-B6 (SK)
Title: Heat treatable sputter-coated product
Inventor: HARTIG KLAUS W
IPC: C23C14/58
Filed: 1992-12-08
Abstract: A heat treatable sputter-coated layer system for glass substrates may be applied before heat treatment if the layer system includes: a) a substantially non-oxidated metallic layer (C) of nickel or a high nickel content alloy containing more than 50 percent by weight of nickel, with a thickness ranging from 2 to 25 nm; b) a protective layer (E) of a metal oxide being different from the metal used in the layer (C), with a thickness ranging from 2 to 100 nm; c) a separate layer (D) of metallic silicon or an oxide or nitride of nickel or the high nickel content alloy and containing more than 50 percent by weight of nickel which is inserted in between the layers (C) and (E). The layer (D), firmly binding the layer (C) with the layer (E), is as thick as 0.5-10 nm.
Patent SK-278148-B6 (SK)
Title: Method of mixed combustion of coal and device for realization of this method
Inventor: BOROSS LASZLO
IPC: A01N29/08
Filed: 1988-10-26
Abstract: By method of mixed combustion of coal in combustion of fluid and powder combustion, is into fluid combustion chamber forced the fluidizating air with flow velocity higher than 4 m/s and into powder combustion chamber is blown the mixture of air and coal powder with flowing speed 15 to 25 m/s. Device consists of fluid combustion chamber (11) and over it is arranged the powder combustion chamber with common fireplace (2). Into space of fluid combustion chamber (11) is orificed the first coal pipe (18) or second coal pipe (19) with coal supply from first coal mill (10) and first or second air pipe (9,16) for supply of fluidization air. Powder combustion chamber is equipped with at least one torch (6), connected with leading of combustion air and with blowing pipe (5) for blowing mixture of air and coal powder leaded from second coal mill (1).
Patent CZ-305394-B6 (CZ)
Title: Grounding device for high voltage instruments
Inventor: VOSTRACK ZDENĚK
IPC: H02B13/075
Filed: 2009-03-30
Abstract: The present invention relates to a grounding device for high voltage instruments, particularly for earthing switches and earthing switches disposed on a power plant disconnecting switch, consisting of a frame (1) with a drive shaft (9) bearing (3) located at the point of a central insulator (2) on the frame (1), wherein the drive shaft (9) is connected at its one end with a drive (10). Two “V” or “U” shaped grounding bars (4), being located on the drive shaft (9) are connected above with each other by a first electrically conducting cross bar (5) with electrically conducting contacts (8) that are fixedly attached at the point of insulators (2), whereby on the ground potential, both the grounding bars (4) are connected with each other by means of a second electrically conducting cross bar (11) and joined with the frame by an elastic electrically conducting coupling (6).
Patent CZ-307091-B6 (CZ)
Title: A stable pharmaceutical preparation containing Vardenafil hydrochloride
Inventor: LINEK JAN
IPC: A61K47/12
Filed: 2012-09-14
Abstract: The invention relates to a pharmaceutical formulation for oral administration, the formulation containing an effective quantity of Vardenafil hydrochloride or Vardenafil hydrochloride trihydrate, stearic acid and at least one further pharmaceutically acceptable excipient. A further solution provides a process for the preparation of said formulation.
Patent CZ-309039-B6 (CZ)
Title: Biodegradable sports shoes
Inventor: Sáha Tomáš
IPC: C08L67/00
Filed: 2021-03-12
Abstract: The biodegradable sports shoes consist of a textile upper with a sewing insole and a sole with an integrated insole attached to the upper. The upper part is made of biodegradable cotton woven fabric with seams of threads, which, like shoelaces, are made exclusively of biodegradable fibres, the sewing insole is cotton or linen. The sole is based on a reactive biodegradable polyurethane and is attached to the upper without adhesives, directly during the synthesis of polyurethane from the polyol component and the isocyanate component in a weight ratio from 1: 0.4 to 1 : 4. The polyol component consists of a mixture of 100 by weight parts of polyester polyol with a molecular weight of 500 to 5000 g / mol and a hydroxyl number of 20 to 100 mgKOH / g, 1 to 30 by weight parts of a diol-based chain extender with a molecular weight of 50 to 400 g / mol and a hydroxyl number of 200 to 2000 mgKOH / g, 0.1 to 2 by weight parts of water as a blowing agent, 0.05 to 2 by weight parts of amine catalyst and 1 to 5 by weight dye parts. The isocyanate component consists of a polyisocyanate with an NCO group content of 5 to 30% by weight.
Patent CZ-309327-B6 (CZ)
Title: Audio dynamic range compressor
Inventor: KRAMPERA JIŘÍ
IPC: H03G7/00
Filed: 2021-04-15
Abstract: The solution is used to compress the dynamic range of an audio signal in audio technology. An input audio signal with a wide intensity range is compressed to a prescribed intensity range when entering an audio dynamic range compressor. Excessively high audio signal intensity values at the input are reduced, while low audio signal intensity values are passed through the dynamic range compressor of the audio signal without limiting. The compressor of the dynamic range of the audio signal is made up of a temperature-variable resistor, preferably a filament.
Patent CU-23389-B6 (CU)
Title: Combinación farmacéutica citoprotectora, útil en la prevención y tratamiento del síndrome de respuesta inflamatoria sistémica
Inventor: SELMAN-HOUSEIN SOSA MANUEL
IPC: A61K38/04
Filed: 2005-12-29
Abstract: La presente invención trata de una combinación farmacológica entre una proteína con propiedades citoprotectoras y un péptido inmunomodulador. El Péptido de la combinación farmacológica es el LALF 31-52 lineal, que incrementa los mecanismos de defensa inmunológica, sin inducir una respuesta inflamatoria exacerbada. La proteína de la combinación farmacológica es el Factor de Crecimiento Epidérmico que posee un efecto citoprotector y activa la transducción de senales de genes de sobrevida celular. La combinación farmacológica de la presente invención confiere resistencia a las células sistémicas e inmunocomponentes, para tolerar el dano inducido por las citoquinas inflamatorias y por endotoxinas bacterianas, sin activar vías moleculares de apoptosis. Además, atenúa los eventos inflamatorios de la primera etapa de la sepsis y de la respuesta inflamatoria ante traumatismos estériles, permitiendo la defensa del organismo contra la invasión de patógenos o contra los mediadores de la inflamación, sin que la respuesta inflamatoria sea deletérea a su integridad.
Patent CZ-293940-B6 (CZ)
Title: Escalator step
Inventor: HENNING GUNTER
IPC: B66B23/12
Filed: 2000-06-02
Abstract: The invented escalator step is substantially made of a material such as plastic and has its front edge (16) of tread surface (12) provided with an edge strip (22) that is anchored to the tread surface (12) by fasteners (26) passing therethrough and invisible from outside, whereby said edge strip (22) is made of material having greater hardness than that of the plastic. On said tread surface (12) inner side, there is arranged opposite to said edge strip (22) a support plate (30) provided with through holes for pin-like fasteners (26) of the edge strip (22).
Patent CZ-302123-B6 (CZ)
Title: Granules with hydrated barrier material
Inventor: BECKER NATHANIEL T
IPC: C11D11/00
Filed: 1998-12-21
Abstract: In the present invention, there are disclosed granules comprising an enzyme core and a hydrate barrier salt as a coating around said enzyme core and one or a plurality of layers coated over said hydrated barrier material wherein the barrier salt is selected from the group consisting of magnesium sulfate heptahydrate, zinc sulfate heptahydrate, copper sulfate pentahydrate, sodium phosphate dibasic heptahydrate, magnesium nitrate hexahydrate, sodium borate decahydrate, sodium citrate dihydrate and magnesium acetate tetrahydrate. The invention also provides a method of producing a granule comprising: a) providing an enzyme core; b) coating a hydrated barrier salt onto the enzyme core wherein the hydrated barrier salt is represented by magnesium sulfate heptahydrate, zinc sulfate heptahydrate, copper sulfate pentahydrate, sodium phosphate dibasic heptahydrate, magnesium nitrate hexahydrate, sodium borate decahydrate, sodium citrate dihydrate or magnesium acetate tetrahydrate; and c) applying an outer coating over the hydrated barrier salt.
Patent CZ-297095-B6 (CZ)
Title: Method and device for increasing recognition probability in voice recognition systems
Inventor: KAUSCHE ULRICH
IPC: G10L15/06
Filed: 1999-01-20
Abstract: The present invention relates to a method for increasing recognition probability in voice recognition systems and a device for making the same. According to the inventive method, selective post-training of the already stored homonymic term is carried out after inputting a term to be recognized. This makes it possible to improve the speaker-dependent recognition rate even in environments with prevailing acoustic interference.
Patent CZ-296267-B6 (CZ)
Title: Method and apparatus for measuring distribution of temperature within a material, particularly in a tissue
Inventor: POUSEK LUBOMIR
IPC: G01K11/22
Filed: 2000-12-20
Abstract: When measuring distribution of temperature within material of a measured objects, particularly a tissue, during which distribution ultrasonic waves with frequency ranging from 16 kHz to 1 GHz propagate as longitudinal waves within the material being measured and an ultrasonic cross section of the scanned area formed by a shot with different values of textural parameters is created from a reflected signal, whereby the textural parameter value corresponds to relative change in temperature. By comparing magnitude of the relative change with a predetermined reference values, there is determined temperature at the given point. Disclosed is also apparatus for carrying out the above-described method, which apparatus consists of an ultrasonic device being connected to a device for acquiring and processing ultrasonic data and for grabbing and analysis of shots, whereby said data acquiring and processing device is connected with a device for projecting a network into the given point and for determination of brightness average value, whereby said device is connected to a cathode-ray tube.
Patent CZ-305726-B6 (CZ)
Title: Securing and arming device
Inventor: ETTMUELLER PETER
IPC: G05G17/00
Filed: 2002-05-17
Abstract: In the present invention, there is disclosed a securing and arming device having an operating body (20), which, prior to an arming time, is secured in its position of rest on a support device (12) by means of a securing element (30), which is in a securing position, can, for the purpose of arming, be released by the securing element (30), which is moved into its release position in relation to the support device (12). After the arming time, said an operating body (20) can be brought into an operating position by a rotary movement around a trigger axis (E), and having a delay element (22), which is designed to be driven in the course of the rotational movement of the operating body (20) and to delay the rotational movement of the operating body (20), wherein the invention is characterized in that the operating body (20) and the delay element (22) are arranged one inside the other, so that they constitute an outer wheel without a wheel shaft and an inner wheel without a wheel shaft. Both the wheels have parallel geometric wheel axes and define a ring-like gap therebetween. At least one of the wheels is embodied to be wavy on its surface facing the other one of the wheels, with wave crests (20.1) and wave troughs (20.2) over its circumference, and with areas of their surfaces facing each other. The wheels rest against motion transfer bodies (24) located in the ring-like gap and being seated radially displaceable in the said gap.
Patent CZ-297734-B6 (CZ)
Title: Ski binding for cross-country skis and touring skis
Inventor: KOGLER HANNES
IPC: A63C9/20
Filed: 2002-04-11
Abstract: In the present invention, there is disclosed a ski binding for cross-country skis and touring skis with a step-in mechanism, said ski binding comprising two pressure-spring-loaded retention pins (1, 101) located in the toe region and extending substantially transversely to the ski longitudinal axis and provided with a rounding or chamfer at their outer ends. Said retention pins engaging in latching openings (4) of the boot sole (22) or parts of the latter in the manner of a step-in mechanism and can be brought out of the snapped-in position by a releasing mechanism. The wall of the latching opening (4) is cylindrical and in the clamped state of the boot in the binding (20) swivels along with the cylindrical peripheral surface of the retention pin (1, 101).
Patent CZ-301353-B6 (CZ)
Title: Plasma arc torch tip, plasma torch including such tip and method of operating the plasma arc torch
Inventor: CONWAY CHRISTOPHER J
IPC: B23K9/29
Filed: 2003-04-07
Abstract: In the present invention, there is disclosed a plasma arc torch tip (102) configured for electrical contact and passage of fluid between the tip (102) and an adjacent anode member (108) of the plasma torch, wherein the tip (102) comprises perimeter surface adjoining a perimeter surface of the anode member (108), and the adjacent perimeter surfaces ensure electrical contact, preferably for instance through raised ridges (290) and passage of cooling fluid, preferably for instance through areas extending between the raised ridges (290). There is further disclosed a plasma arc torch comprising an anode member (108) forming a perimeter surface, and a tip (102), configured for electrical contact with the anode member (108) and for passage of fluid between the tip (102) and the anode member (108), whereby the tip (102) forms a perimeter surface adjoining a perimeter surface of the anode member (108), and these adjacent perimeter surfaces ensure electrical contact and passage of a cooling fluid. There is also disclosed a method of operating the above-described plasma arc torch.
Patent SK-288049-B6 (SK)
Title: Coating and binding agent, its use for production of cover oral or dermal pharmaceutical dosage forms, process for its production and dosage form containing same
Inventor: PETEREIT HANS-ULRICH
IPC: A61K47/12
Filed: 2001-02-27
Abstract: A coating and binding agent for oral or dermal pharmaceutical dosage forms, consisting of a) a copolymer, consisting of radically polymerized C1-C4-esters of (meth)acrylic acid and other (meth)acrylate monomers having functional tertiary ammonium groups, wherein the copolymer being in powder form with an average particle size of 1 to 40 um and b) 3 to 15 % by weight based on a) of an emulsifier with an HLB value at least 14, optionally water and/or a pharmaceutical active substance and other conventional additives, wherein the agent comprising also c) 5 to 50 % by weight based on a) of a C12-C18-monocarboxylic acid or a C12-C18-hydroxyl compound. It is described the use this agent as a moisture-proof and/or a flavour insulating coating for pharmaceutical composition containing active substances, a process for preparing this cover and dosage form containing the same.