baber/WOPTO huggingface dataset:
Patent EP-0461141-B1 (EP)
Inventor: LEE KUO-HSIUNG
IPC: C07D493/04
Filed: 1990-02-23
Granted: 1999-11-03
Abstract: Compounds that are analogs of etoposide and exhibit antitumor activity are disclosed. The compounds of the present invention have formula (I), where R1 is  beta -OCH2CH2NH2,  beta -NHCH(CH3)CH2OH, beta -NHCH2CH(CH3)OH,  beta -Cl,  beta -Br,  beta -OH,  alpha -OH, beta -NH2,  alpha -NH2,  beta -NHCH2CH2OH,  alpha -NHCH2CH2OH,  beta -NHCH2CH2CH3,  beta -NHCH2CH2OCH3,  beta -NHCH2CH=CH2,  beta -NHCH2CH(OH)CH3,  beta -NHCH2CH2CH2OH,  beta -OCH2CH2OH, (a), (b), (c), (d), (e), (f), (g), (h), (i), (j), (k), (l), (m), (n), (o), (p), (q), (r), (s), (t), (u), (v) or (w). R2 is H, or Br; R3 is H, or Br; R4 is H, or Br; R5 is H, or Br; and R6 is H, or -CH3.
Patent EP-0450080-B1 (EP)
Inventor: AVETISOV EDUARD SERGEEVICH
IPC: A61K47/24
Filed: 1990-05-02
Granted: 1994-03-16
Abstract: Une composition de traitement de la myopie évolutive comprend les composants suivants, exprimés en pourcentage en poids: un mélange de polyvinylpyrrolidone, et d'acrylamidehydrazide d'acrylate d'éthyle (en proportions égales) 18,8 à 29,5, une solution aqueuse contenant les composants suivants en mg/l: acide muriatique 940,0, acide borique 4,12, oxyde ferreux 115,0, citrate de cuivre 16,0, ladite solution étant comprise entre 69,5 et 80,1, une solution aqueuse à 3 % de peroxyde d'hydrogène 0,79 à 0,89, du dichlordi[2-méthyl-3-oxy-4,5 di(oxyméthyl)-pyridine] de cuivre (II) 0,11 à 0,31.
Patent EP-0491749-B1 (EP)
Inventor: PRINZHAUSEN FRIEDRICH
IPC: G01D5/30
Filed: 1990-09-07
Granted: 1994-06-01
Abstract: Un dispositif permet de mesurer la position absolue d'une pièce (10) sur deux dimensions par rapport à un dispositif de mesure (11), la surface de la pièce (10) ayant la forme d'un hologramme. Les informations contenues dans l'hologramme sont lues au moyen d'une onde de mesure (13) dirigée sur l'hologramme (18) et diffractée par celui-ci, par interférence avec une onde de référence (14). Les ondes (13, 14) ayant subi l'interférence sont captées par un dispositif détecteur optique (20) qui comprend au moins deux capteurs (21, 22). Un agencement (23) de traitement de signaux détermine la position absolue à partir de l'intensité des rayonnements détectés par les capteurs (21, 22) ou des relations de phases entre les signaux émis par les capteurs (21, 22), dans les deux cas par comparaison avec une valeur enregistrée dans une mémoire.
Patent EP-0552143-B1 (EP)
Inventor: KELLY JOHN HAMILTON
IPC: G01N33/20
Filed: 1990-10-10
Granted: 1995-01-11
Abstract: On détermine d'une manière rapide la qualité interne des coulées en continu et d'autres échantillons en acier se présentant sous forme de lingots, de billettes, de blooms, de brames et de barres pour identifier et corriger dans un temps approprié les conditions de coulage pouvant potentiellement provoquer des problèmes. Un échantillon d'acier provenant de la coulée est tout d'abord meulé pour éliminer les zones endommagées par la chaleur et pour obtenir un degré prédéterminé de dureté de la surface, puis il est attaqué par procédé anodique avec de l'acide chlorhydrique dilué dans des conditions de température ambiante pour éliminer par attaque à l'acide le métal se trouvant en surface afin de faire apparaître la qualité interne. Lorsque l'échantillon sort de l'appareil de mordançage, on le lave, on le sèche puis on l'examine visuellement pour déterminer la qualité interne.
Patent EP-0443469-B1 (EP)
Inventor: HOELZEMANN JUERGEN
IPC: B01D29/39
Filed: 1991-02-16
Granted: 1995-02-01
Abstract: A rotor filter press is described, in which filter discs 7 are placed on a carrier 13 and are penetrated by a shaft 3, a collecting tube 15 runs under the filter discs 7, which tube is connected in an attachable manner via a connecting piece 16 to an outlet orifice 17 of each assigned filter disc 7, and each filter disc 7 is divided into filter disc sectors 19, 20 and a lower filter disc sector 19 is provided with the outlet orifice 17, is separated from the shaft 3 by a distance 25 and the collecting tube 15 is pushed by means of a rotary movement between the shaft 3 and the carrier 13. It is required in this case that the installation and removal of the lower filter disc sector be simplified. This is achieved by every connecting piece being a connecting nozzle 16, over which the assigned lower filter disc sector 19 with the outlet orifice 17 is pushed along a drop distance, by the drop distance being adapted to the distance 25 between the lower filter disc sector 19 and the shaft 3 and by a ring segment 26 being pushed by means of a rotary movement about the shaft 3 between the shaft 3 and the lower filter disc sector 19. The lower filter disc sectors are pushed onto the connecting nozzles and the ring segments are pushed under the shaft. <IMAGE>
Patent EP-0543049-B1 (EP)
Inventor: VOGEL IGNAZ
IPC: B60N2/427
Filed: 1991-11-22
Granted: 1994-10-12
Abstract: When the seats of passenger transport vehicles are arranged in rows, the space between the backrest and rearside of the backrest of the seat in front constitutes the survival space for the passengers in the event of an accident. Therefore, the backrests should not be too greatly deformed by the impacting passengers in the event of an accident so that this survival space is not excessively reduced. According to the invention, this is achieved, and nevertheless the peak impact energy resulting from deformation is absorbed, by virtue of an extension of the backrest frame which becomes embedded in an angled portion. <IMAGE>
Patent EP-0492497-B1 (EP)
Inventor: SCHUDOK MANFRED DR
IPC: C12N11/08
Filed: 1991-12-20
Granted: 1996-08-28
Abstract: The invention relates to a process for acylating alcohols with Pseudomonas lipases which have been immobilised on polystyrene- or phenol/formaldehyde-based carriers.
Patent EP-0433273-B1 (EP)
Inventor: DONALD ROBERT ARCHIBALD
IPC: B65D75/26
Filed: 1986-10-02
Granted: 1995-09-13
Abstract: Components for aseptic packaging, a method of forming such a package and an aseptically filled package using a construction of flexible plastics material (12,13) sandwiching a material (10,11) which is impervious to micro-organisms, the longitudinal seal being made between two surfaces of the same material. The specification also discloses a form of end closure (20) including a plug (22) of resilient material which ensure the integrity of the closure.
Patent EP-0454494-B1 (EP)
Inventor: DANISHEFSKY SAMUEL J
IPC: A61P35/00
Filed: 1991-04-26
Granted: 1995-09-20
Abstract: Calicheamicinone, the aglycone portion of calicheamicin, derivatives and analogs thereof are disclosed as are a method of preparing and using the same.
Patent EP-0466314-B1 (EP)
Inventor: MORISAWA NOBUO
IPC: G09F9/00
Filed: 1991-05-29
Granted: 1995-11-15
Abstract: A parking time display device, in or for a motor vehicle (3), to display the parking time of the vehicle (3). The device comprises display means (5) visible from outside the vehicle (3) for indicating a parking time of said vehicle (3) and means for operating said display means (5) according to said parking time. <IMAGE>
Patent EP-0467690-B1 (EP)
Inventor: DAIGLE RONALD E
IPC: G10K11/34
Filed: 1991-07-18
Granted: 1995-11-29
Abstract: An ultrasonic diagnostic imaging system is provided for scanning with a linear transducer array and displaying an image area which is truncated with respect to a conventional triangular image sector to take the form of a trapezoid. Uniformity of image resolution and ease of signal processing enhancement is provided by transmitting adjacent ultrasonic beams at equal angular increments over the sector area. The ultrasonic beams transmitted are focused around predetermined transmit focal points and the transmit aperture employed for each transmission is determined by a transducer sensitivity criterion applied to the focal point. Means are provided for delaying signal components received from the beam directions so that the sum of the components will form a coherent echo signal. Means are provided for dynamically focusing received signal components by dynamically focusing received signal components by dynamically varying the sampling frequencies of laterally disposed signal components, and the receive aperture is dynamically varied in correspondence with the number of array elements which satisfy a sensitivity criterion at different depths of field. <IMAGE>
Patent EP-0449727-B1 (EP)
Inventor: GARDNER JAMES F
IPC: F16J15/34
Filed: 1991-03-26
Granted: 1996-01-03
Abstract: A dry-running gas seal (12) includes a stationery seal ring carrier (14) holding a stationary seal ring (16), a rotary seal ring carrier (18) holding a rotary seal ring (22) facing the stationary seal ring (16), scoops (26) radially outside and extending toward the rotary seal ring carrier (18), and a heat exchanger (32) in fluid communication with the scoops (26), whereby the portion of the gas is trapped by the scoops (26) and transferred to and cooled by the heat exchanger (32) and returned to and the high pressure area adjacent to the seal. <IMAGE>
Patent EP-0544961-B1 (EP)
Inventor: MESNEL FRANCOIS
IPC: B60J10/00
Filed: 1991-11-29
Granted: 1995-04-12
Abstract: The subject of the invention is a weather strip for framing a motor vehicle bodywork opening, this strip comprising a reinforced section (1) forming a grip with a U-shaped cross-section made from a thermoplastic material, and a tubular sealing element (2) made from an elastically deformable material which adheres laterally to the external surface of the section with a U-shaped cross-section (1). In accordance with the invention, along at least part of its length, corresponding to the position of a corner of the opening frame to be equipped, the tubular element (2) has a length which is greater than that of the corresponding part of the section (1), the portion of the tubular element (2) of length greater than that of the corresponding part of the section (1) being laterally offset with respect to the latter. <IMAGE>
Patent EP-0528030-B1 (EP)
Inventor: OKANISHI MASANORI
IPC: C07H19/23
Filed: 1991-02-20
Granted: 1997-09-17
Abstract: A 12,13-dihydro-6H-indolo[2,3-a]pyrrolo[3,4-C]-carbazole-5,7(6H)-dione derivative of general formula (I), pharmaceutically acceptable salt thereof, production thereof, and uses thereof, wherein R<1> represents a monosaccharide group with 5 to 7 carbon atoms, and the hydroxyl group(s) of the monosaccharide group may be substituted with one to three groups which may be the same or different from each other and are selected from among hydrogen, lower alkyl, lower alkylcarbonyloxy and lower alkoxy. <CHEM>
Patent EP-0535115-B1 (EP)
Inventor: COCHRAN WILLIAM H
IPC: B32B27/00
Filed: 1991-06-19
Granted: 2006-02-01
Abstract: A flexible composite comprising a high tensile strength fibrous component dispersed within a flexible or resilient polymeric matrix, the matrix and fibrous component being essentially unbonded to each other so that the composite retains essentially the flexibility of the polymeric matrix.
Patent EP-0546038-B1 (EP)
Inventor: WONG PATRICK S-L
IPC: A61K31/55
Filed: 1991-08-28
Granted: 1994-07-27
Abstract: A dosage form is disclosed that comprises means inside the dosage form for providing a substantially drug-free interval before the dosage form delivers a drug from inside the dosage form. The dosage form in an embodiment comprises a drug on the exterior of the dosage form, which drug is available for immediate delivery.
Patent EP-0519022-B1 (EP)
Inventor: EBERBACH MARK ALLEN
IPC: A61B19/00
Filed: 1991-10-11
Granted: 1997-12-17
Abstract: Apparatus and method for laparoscopic hernia repair including the use of an introducer sheath housed around an inner tubular plunger. The plunger houses an elongated ribbon formed into a loop, the loop being formed by a bipartite distal end of the ribbon. A patch with a passageway is attached to the loop with each of the two ends of the bipartite distal end of the ribbon being introducible into one end of the passageway for opening the patch into a planar configuration once it is pushed out of the sheath by the plunger.
Patent EP-0515864-B1 (EP)
Inventor: DOHERTY CHERYL A
IPC: A23G3/34
Filed: 1992-04-30
Granted: 1995-11-29
Abstract: A low or no fat confection is prepared containing 80% soluble solids wherein at least 70% of the solids are carbohydrates. The mixture containing carbohydrate, a cationic reactive and thermalsensitive hydrocolloid and an edible cation containing material is cooked or its solids concentration adjusted to 80% solids while hot. The molten mixture is then cooled to form a solid confection having a water activity being 0.30 to 0.65 Aw and a pH from 3.0 to 8.5.
Patent EP-0530531-B1 (EP)
Inventor: WAESCHENBACH GUIDO DR
IPC: A61K8/20
Filed: 1992-08-06
Granted: 1998-11-18
Abstract: The invention relates to preservative-free cosmetics in the form of emulsions of the O/W or W/O type of conventional composition, which contain at least 2% by weight, preferably at least 5% by weight (calculated as anhydrous salt) of water-soluble, emulsifier-compatible alkali metal or alkaline earth metal salts of inorganic or organic anions.
Patent EP-0528382-B1 (EP)
Inventor: SCHIEVELBUSCH ULRICH PROF DIPL
IPC: F16H15/28
Filed: 1992-08-14
Granted: 1995-02-22
Abstract: A drive hub for a vehicle, in particular bicycle, comprising a hub axle (1, 2), a hub sheath (9) which encloses the hub axle, a driver (13), a friction gear (17), a coupling device and a control device (50) for infinite adjustment of the transmission ratio of the friction gear (17) is constructed with a ball-and-socket friction gear, comprising one drive ring (25) and one drive ring (27), several friction balls (35) which connect the rings to one another in a frictionally engaging fashion, one friction ball carrier (39a,b) which is connected fixed in terms of rotation to the hub axle (4) and one control device (50) for jointly swivelling the bore axes, the drive ring (25) and the drive ring (27) each being in frictional contact with the friction balls on their side facing away from the axle. The drive hub is of simple, inexpensive design and is highly efficient. 
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Patent EP-0547297-B1 (EP)
Inventor: KADER KARL-WILHELM
IPC: B65B39/08
Filed: 1992-08-17
Granted: 1996-10-30
Abstract: Bag-clamping device for the retention of a bag to be filled, especially a side-folding bag, on a filling connection, the bag-clamping device having the following features:
 a first pair of clamps having respective clamping bodies (15), in order to retain mutually opposite first bag-wall parts on the filling connection, and a second pair of clamps having respective pairs of clamping bodies (25), the pairs of second clamping bodies having first surface parts (26) which are laid against one another in pairs in such a way that bag-wall parts located in front of the end faces are grasped and held in the edge region, and respective second surface parts (27) which are angled relative to these and which are matched with the end faces (3) and to the guide plates of the swung-out spreading flaps (10), in order to retain the remaining free bag-wall parts on the filling connection. 
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Patent EP-0548613-B1 (EP)
Inventor: WUJCIK STEVEN E
IPC: C08G18/28
Filed: 1992-12-03
Granted: 1997-05-21
Abstract: Addition of minor quantities of mono- or dicarboxylic acids to polyurethane foam formulations which employ polyisocyanate polyaddition polymer polyol dispersions prevents shrinkage and tightness in polyurethane foams prepared therefrom. If acid addition is made directly after dispersion preparation, reduction of polyol viscosity and more rapid stabilization against viscosity change is observed.
Patent EP-0498510-B1 (EP)
Inventor: BOUMANS JOHANNES ADRIANES
IPC: B27F5/12
Filed: 1992-02-05
Granted: 1997-04-16
Abstract: Milling template assembly for use in milling recesses, openings etc. for mortise locks and lock plates in a door and/or door-frame, comprising a milling template defining at least one milling aperture corresponding to said recess, opening, etc., and means (2, 3; 12, 13, 14) for attaching the template means to a door or door-frame. The attaching means comprise adjustable gauge means (2; 14) provided with gauge indication and means for adjustably mounting the gauge means on the template, wherein the gauge means are provided with abutment surfaces for abutting against the abutting, closure edge of the door or door-frame in order to enable accurate positioning of the milling aperture with respect to that abutting closure edge. The milling template comprises a master milling template (1, 11) and an insert cassette (4;15.1, 15.2), wherein the milling template is provided with the attaching means and with an opening adapted to positively receive and accommodate the insert cassette, the latter being provided with and defining the milling aperture. The insert cassette (4) may be U-shaped and comprises an end plate (3) and side plates (4, 5) with work passages for router and mandrel hole augering and tapping tools for carving the openings required in the door. Alternatively, the insert cassette (15.1) may be shaped as a plate which is provided with an aperture corresponding to the contours of a locking plate. Moreover, the insert cassette (15.2) may be shaped as a plate that is provided with apertures for day and night bolts. <IMAGE>
Patent EP-0519530-B1 (EP)
Inventor: ERLACH JOSEF
IPC: H02P9/04
Filed: 1992-05-05
Granted: 1995-01-25
Abstract: In a hydraulic turbine with a distributor with adjustable guide blades and a rotor wheel with adjustable rotor blades indirect optimisation of the operating parameters is achieved in that fluctuations in the intensity of the generator power and/or the bearing oscillations of the hydraulic turbine are determined without reference to the absolute values and set at or adjusted to a minimum.
Patent EP-0522854-B1 (EP)
Inventor: HANCOCK JOHN EDWIN
IPC: E04B2/76
Filed: 1992-07-09
Granted: 1997-04-23
Abstract: A structure and method of making same is described, which comprises at least four elongate members (10), joined to form a rectangular framework for supporting panelling (90), the join between pairs of elongate members (10) is provided by locating in an axially extending bore (22) of one of them an expansion element (100) which is engaged by a bolt (102) passing through an aperture formed to extend transversely of the axis of the other of said pair. Each elongate member (10) may have two axially extending parallel bores (22, 22 min ) formed therein with pairs of expansion elements (100, 100 min ) and bolts (102, 102 min ) used with them. The elongate members (10) are formed with walls (26, 36) defining cavities (30, 34) extending parallel to the or each bore (22) therein. The walls (26, 36) are adapted to engage legs (46, 48, 56) of elongate cover elements (42, 52) to be fitted to said members (10). The walls and cover elements may be used to define sets of slots running parallel to said cavities (22) of the elongate members, in which slots edges of panelling (90) are received. The panelling may comprise a rectangular cut piece of solid material with lugs at each edge received in said slots, or be two laminar layers (90) (possibly glass) the edges of which are fitted said slots. The volume between layers (90) may be void or filled with insulating material. Resilient inserts may be placed in the slots to hold edges of panelling received therein. The slots may be used to support brushes or other sealing elements. One form of cover element (150) described for use on a door structure has a part (162) extending past the elongate member (10) on which it is supported and itself supports a resilient sealing strip (170) engagable with a surface of a cover element (54) of an elongate member (10 min ) adjacent the door when the door is closed. <IMAGE>
Patent EP-0533385-B1 (EP)
Inventor: COUPLAND DUNCAN ROY
IPC: B22C21/14
Filed: 1992-09-08
Granted: 1999-04-14
Abstract: Pinning wires suitable for use in turbine blade manufacture comprise palladium alloyed with one or more noble and/or refractory metals, and are substantially more cost effective than conventional pinning wires.
Patent EP-0639199-B1 (EP)
Inventor: THORN DAVID LINCOLN
IPC: C08G69/04
Filed: 1992-01-02
Granted: 1997-08-27
Abstract: A process for producing phosphonate esters containing the 2-(pyridyl)ethyl group by reacting a vinylpyridine with a di- or trihydrocarbylphosphite in the presence of a selected silane, protic acid, or Lewis acid is disclosed. Also disclosed are novel silylphosphonate esters containing the 2-(pyridyl)ethyl group. All of the compounds produced herein are useful as catalysts for increasing the molecular weight of polyamides.
Patent EP-0575366-B1 (EP)
Inventor: BALTZ ROLF
IPC: G01N3/30
Filed: 1992-02-26
Granted: 1994-09-21
Abstract: PCT No. PCT/EP92/00401 Sec. 371 Date Jan. 28, 1994 Sec. 102(e) Date Jan. 28, 1994 PCT Filed Feb. 26, 1992 PCT Pub. No. WO92/15856 PCT Pub. Date Sep. 17, 1992.A method of dynamically testing the functionality of a multi-part specimen comprises the steps of applying a predetermined reproducible shock loading to one part of the specimen and measuring the resulting shock load both at the point of application on said one part and at at least one point on another part of the specimen. Said measured shock loads are also recorded. Apparatus for carrying out this method comprises a drop carriage with means for coupling to one part of the specimen, and at least one acceleration transducer for attachment to the drop carriage and also to at least one part of the test specimen. The apparatus thus produces reproducible shocks up to 40,000 g to enable the structural optimization of severely shock-loaded articles such seat-belt buckles and their functionality both during and after the shock-loading to be demonstrated.
Patent EP-0572559-B1 (EP)
Inventor: CLARKE ROBERT LEWIS
IPC: H01M4/62
Filed: 1992-02-19
Granted: 1997-05-21
Abstract: A particulate composition having improved stability in typical electrolytes consisting essentially of Magneli phase substoichiometric titanium oxides.
Patent EP-0542956-B1 (EP)
Inventor: LANG HUGO
IPC: G01F23/26
Filed: 1992-06-05
Granted: 1994-12-07
Abstract: Un dispositif de fixation de l'électrode métallique d'une sonde de façon électriquement isolée dans l'ouverture d'un boîtier, de préférence d'une sonde de mesure de niveau dans l'ouverture du boîtier de tête pour sonde, comprend une électrode métallique en baguette et une électrode métallique de protection sur lesquelles sont disposées avec écartement deux bagues bicônes qui, à l'aide de couches isolantes, isolent électriquement et renferment de manière étanche à la pression l'électrode en baguette par rapport à l'électrode de protection, et les deux électrodes par rapport au boîtier dans l'ouverture duquel elles sont fixées. Les deux électrodes sont connectées de manière électriquement isolée à un circuit électronique.
Patent EP-0551459-B1 (EP)
Title: Method for the preparation of 3-amino-2-chloro-4-alkylpyridines
Inventor: GROZINGER KARL G
IPC: C07D213/85
Filed: 1992-05-29
Granted: 1996-11-20
Abstract: A process for the preparation of a 3-amino-2-chloro-4-alkylpyridine of the formula:   <IMAGE>   wherein R is alkyl of from one to three carbon atoms, an intermediate in the preparation of certain 5,11-dihydro-6H-dipyrido[3,2-b:2',3'-e][1,4]diazepine compounds useful in the prevention and treatment of HIV infection.