baber/WOPTO huggingface dataset:
Patent BG-63777-B1 (BG)
Title: Aromatic compounds and pharmaceutical compositions containing them
Inventor: BREAULT GLORIA A
IPC: A61K31/455
Filed: 1998-01-09
Abstract: The invention relates to a compound with the formula where A optionally means substituted ring system provided that the groups -CH(R3)N(R2)B-R1 and -OR4 are in position 1,2 towards each other in ring-type carbon atoms and the ring carbon atom placed in ortho-place in respect of -OR4-connection group (and in 3rd place, therefore, in respect of the connecting group -CHR3NR2-) has not been substituted; B optionally is a substituted ring-type system; R1 is in ring B in position 1,3 or 1,4 in reespect of the binding group -CH(R3)N(R2)- and has the meanings listed in the description; R2 is hydrogen, C1-C6 alkyl, optionally substituted with hydroxy, cyano or trifluoromethyl, C2-C6 alkyenyl provided that the double bond is not in first place, C2-C6 alkynyl provided that the triple bond is not in the first place, phenyl C1-C3 alkyl or pyridyl or pyridyl C1-C3 alkyl; R3 is hydrogen, methyl or ethyl; R4 optionally is substituted C1-C6 alkyl, C3-C7 cycloalkyl, C1-C3 alkyl or C3-C7 cycloalkyl and N- oxide of -NR2 when it is chemically possible, and 5-oxides of sulphur-containing rings when it is chemically possible. The invention also relates to pharmaceutically acceptable salts and in vivo hydrolizable esters and their amides. The invention also applies to methods for the preparation of the compounds, to their usage as therapeutical preparations and to pharmaceutical compositions containing them. 16 claims
Patent BG-64970-B1 (BG)
Title: Spisulosine compounds having antitumour activity
Inventor: RINEHART KENNETH
IPC: A61K35/618
Filed: 2000-11-09
Abstract: Investigation of the activity of extract of the clam Spisula polynyma has led to antitumour long-chain, straight-chain and alkene compounds which have a 2-amino group and a 3-hydroxy group.
Patent BG-65492-B1 (BG)
Title: Method for precise determinating the location of an object, preferably a vehicle moving along a known course
Inventor: FRANCKART JEAN-PIERRE
IPC: G01S19/48
Filed: 2002-12-27
Abstract: The invention concerns a method for determining the location and/or positioning of an object, in particular a vehicle such as a train moving along a known course, and this securely in terms of railway transport. The invention is characterised in that it consists in determining said location and/or positioning of said object by a valid calculation at a given time based on an elementary measurement involving at least a satellite and on a secure mapping of said known course.
Patent BG-66893-B1 (BG)
Title: Internal combustion engine
Inventor: TODORIN IVAN
IPC: F02B71/00
Filed: 2013-09-25
Abstract: The invention relates to an internal combustion engine finding application in transport equipment. The engine includes pistons (1) with two opposite fronts each, which pistons (1) are located in two adjacent pairs of working cylinders (2) and compression cylinders (3),as each pair of the working cylinders (2) and compression cylinders (3) are opposite to one axis, in which bleed valves (5) are mounted in the working cylinders (2) of each opposite pair of cylinders, and suction valves (4) are mounted in the compression cylinders (3) of each opposite pair of cylinders. and valves (8) in grooves to back valves (9) mounted on combustion chambers (6), between which combustion chambers (6) and the working cylinders (2) are mounted valves (7). The pistons are connected to a generator. The design allows both a high degree of expansion and high speed with less friction, thus maintaining the efficiency while reducing power.
Patent BG-67357-B1 (BG)
Title: Remuneration method and system at billing
Inventor: TSIGOV BORIS
IPC: H04M1/00
Filed: 2017-08-04
Abstract: The method and system are related to the field of telecommunications and, in particular, to a communication remuneration method and system at billing that can be used by all subscribers and users of digital, mobile, satellite, computer, network, Internet devices connected via digital communication. It is done via a connection between a digital communication device (2) of a dialling user and between a digital communication device (3) of a target user-object by means of a module-register (4) and at least one digital communication system (1). According to the method, the dialling user through the digital communication device (2) and by means of the register-module (4) selects a specific name of the target user-object included in the register-module (4), as after selecting the specific name, in the database for selected names of the register-module (4) are recorded the identification data of the dialling user and the thus selected specific name of the target user-object, and the notification module (9) notifies the target user-object of the selection of the dialling user after the dialling user makes a payment to the target user-object by means of the payment module (5), connects to the database of the validation module (6) and enters its identification data and data certifying the payment to the target user-object, and the notification module (9) notifies the target user-object for the input of the dialling user, then the target user-object connects via their digital communication device (3) to the database of the validation module (6) and confirms the correctness of the data entered by the dialling user, after that the billing-remuneration module (7) determines billing of the target user-object and determines the remuneration of the dialling user thereof. The system for remuneration at billing includes a dialling module (8) which has an option of an audio/voice connection between at least two devices for voice digital communication (2 and (3) and a payment module (5) which has an option of performing and/or authentication of payment of the dialling user to the target user-object and validation module (6) which has an option of recording the identification data and data verifying the payment of the dialling user to the target user-object in the cells of its database; and their confirmation from the target user-object, as well as a module for billing-remuneration (7), which has an option of setting the charging and remuneration.
Patent CU-24380-B1 (CU)
Title: Derivados de 3- [2- (3,4-dihidroisoquinolin-2 (1 h) -ilcarbonil) fenil] -n- (4-hidroxifenil) -n-fenil-5,6,7,8 - tetrahidroindolizina -1-carboxamida útiles como inhibidores bcl-2 antiapoptóticos, y composiciones farmacéuticas que los contienen
Inventor: CHEN I-JEN
IPC: C07D519/00
Filed: 2014-07-22
Abstract: <p>La invención se refiere a compuestos de fórmula I como inhibidores selectivos de las proteínas de la familia Bcl-2 y composiciones farmaceúticas que los contienen, que pueden ser útiles en la fabricación de medicamentos destinados al tratamientos de cánceres , enfermedades autoinmunes y enfermedades del sistema inmune:</p> <p> </p> <p>ESPACIO PARA FÓRMULA I</p> <p> </p> <p>en el que Ra, Rb, Rc, Rd, T, R3, R4, R5, y G son como se definen en la descripción.</p>
Patent EP-1033539-B1 (EP)
Inventor: CASTELLETTI LUIGI
IPC: F24D19/10
Filed: 2000-02-25
Granted: 2006-04-26
Abstract: The present modular collector is mounted on a heating plant with radiating panels arranged in either the floor or walls or ceiling. This modular collector is basically formed by a series of sectional continuous modules. Compared with the known solutions, the modular collector in question has the important advantage of ensuring a rapid, precise balancing of each circuit since the setting up can be accomplished in a short time. In general, the present collector consists of two series of modules, i.e. a series of return modules (2) and a series of delivery modules (3). The series of return modules (2) is provided with a further delivery module (6) while the series of delivery modules (3) is provided with a further return module (7). The modules (6, 7) act as mixing valve . The delivery and return modules are connected through a pump (8). During the operation, the pump (8) generates both a depression in the return collector, modules (2), and a pressure in the delivery collector, modules (3), proportionally to the load losses of the plant. <IMAGE>
Patent EP-1187431-B1 (EP)
Inventor: HIRSCH HANS-GUENTER
IPC: G10L15/26
Filed: 2000-09-05
Granted: 2005-12-21
Abstract: A portable terminal (100) for accessing an external database (120), wherein the external database (120) is removably connectable to the terminal (100) and contains a plurality of strings with one or more alphanumerical characters, is described. The portable terminal (100) comprises an automatic speech recognizer (160) adapted to access a reference database (170) containing information relating to spelled alphanumerical characters comprising at least letters or digits. The portable terminal (100) further comprises a processing unit (140) for searching at least one matching string among the plurality of strings on the basis of one or more alphanumerical characters recognized by the automatic speech recognizer (160) and an interface (180) for accessing the external database (120). Prior art speech recognition methods do not restrict the recognition to admissible characters at all times. This problem is solved in that a syntax database comprising the admissible characters is generated when the terminal is switched on.
Patent EP-1106147-B1 (EP)
Inventor: SALZ ULRICH DR
IPC: A61C5/60
Filed: 2000-10-19
Granted: 2005-03-23
Abstract: A one shot mixing system for dental material, or for other mixed materials, has a blister pack with a reaction substance (catalyst) in the bottom of a recess, sealed by a cover film. The recess has level marks (34) to indicate how much material to add prior to mixing. The disposable mixing tool (42) can be included in the blister pack.
Patent EP-1096156-B1 (EP)
Inventor: OSTROWSKI WOLFGANG
IPC: F16B5/02
Filed: 2000-10-20
Granted: 2005-05-04
Abstract: The mounting bolt (1) for vehicle bodywork, fitted in advance, is held in place in the preassembled position where the lower bolt section (3) is wholly covered by the damping sleeve (5). The dia. of the upper bolt section (2) is smaller than the nominal dia. of the thread. The bolt (1) has a collar (9) at the upper bolt section (2) and of a larger dia. than it. The damping sleeve (5) has an upper (10) and a lower (11) section, bonded together by an adhesive or by vulcanizing. The collar (9) dia. is larger than the drilling (8) through the upper damping sleeve section (10) and smaller than the drilling (8) through the lower damping sleeve section (11).
Patent EP-1101908-B1 (EP)
Inventor: ENGELER WERNER
IPC: F02M25/00
Filed: 2000-11-13
Granted: 2005-12-07
Abstract: Apparatus (A) for reducing harmful components in the exhaust gas from an engine (particularly a diesel engine), includes a nitrogen oxides (NOX) storage catalyst (12). Apparatus (A) for reducing harmful components in the exhaust gas from an engine (particularly a diesel engine), includes, in order in the direction of gas flow and in the exhaust line (4), an oxidation catalyst (9) and filter (11) for removing particles, also an exhaust gas recycle device that includes a recycle line (25) that by-passes the cylinders (2) of the engine. The new feature is that a nitrogen oxides (NOX) storage catalyst (12) is present in (4), behind (9).
Patent EP-1193387-B1 (EP)
Inventor: PRESS ROMAN
IPC: F02M51/06
Filed: 2000-09-27
Granted: 2005-07-27
Abstract: A gaseous fuel injector for an internal combustion engine or a propulsion system using fuel cells has an electromagnetic solenoid with a flat rectangular armature (13) which seats agains a seat member (15) to form a valve. The valve is kept in a closed position by the differential between the fuel pressure on one side and the atmospheric pressure or the ambient pressure in the discharge chamber on the other side with additional closing force being provided by a spring (23) which abuts against the armature. With each pulsating actuation of the coil (12) of the solenoid, the armature is driven away from its seat to open the valve formed thereby providing an injection of gas from the injector. The injector has a discharge nozzle which is integrally formed therewith. A centrally located aperture (13a) is formed in the armature which along with the side space (10a,10b) afforded by the rectangular shape of the armature provides dual apertures for the flow of gas through the injector. <IMAGE>
Patent EP-1077085-B1 (EP)
Inventor: DUFRESNE PIERRE
IPC: B01J37/08
Filed: 2000-08-03
Granted: 2005-11-16
Abstract: The precarbonation of the catalyst improves its hydrodesulfurising and hydrogenating properties, and also reduces the selectivity in cracking and isomerisation, possibly due to the attenuation of the acidity of the support. Process for the presulfuration of a hydrocarbon hydroconversion catalyst in the presence of hydrogen and a sulfurised compound includes a precarbonation stage to deposit a non-leachable carbonated compound in the pores of the catalyst. An Independent claim is also included for the presulfurised catalyst obtained by the process.
Patent EP-1098657-B1 (EP)
Inventor: ROMBI MAX
IPC: A23L33/20
Filed: 2000-01-14
Granted: 2002-07-10
Abstract: The invention relates to a composition for the treatment of obesity, comprising a catechol-rich extract of green tea, in particular containing from 20% to 50% by mass of catechols expressed as epigallocatechol gallate (EGCG).
Patent EP-1159233-B1 (EP)
Inventor: COSTA UMBERTO
IPC: C04B28/00
Filed: 2000-03-02
Granted: 2003-02-12
Abstract: The present invention refers to a hydraulic binder made from Portland clinker containing calcium fluoroaluminate 11CaO.7Al2O3.CaF2, to which sodium aluminate, lime, and optionally, sodium bicarbonate are added. The added lime has not undergone the formation process of clinker. The cement mix that can be obtained with this binder has a very short hardening time, scarcely influenced by temperature variations during laying operations.
Patent EP-1165540-B1 (EP)
Inventor: OWEN SIMON NEIL
IPC: C07D309/10
Filed: 2000-03-16
Granted: 2003-08-13
Abstract: The present invention relates to compounds of the formula (I):wherein R1, R2, R3, R4, R5, R6, R7, R8, R9, R10 and n are defined herein. The compounds are of particular use in the treatment or prevention of depression, anxiety, pain, inflammation, migraine, emesis and postherpetic neuralgia.
Patent EP-1157347-B1 (EP)
Inventor: GULATI SANDEEP
IPC: G16B25/10
Filed: 2000-02-17
Granted: 2004-10-20
Abstract: A biochip output pattern (OP) is analyzed to identify mutations in biological samples applied to it. The OP is tessellated and a stimulus pattern (SP) associated with known mutations is generated. A resonance pattern (RP), of resonance between SP and tessellated OP, is generated and interpreted to yield confirmed mutations. Independent claims are also included for the following: (1) preconditioning the OP of a biochip, comprising: (a) tessellating the output pattern to match a predetermined stimulus pattern yielding a tessellated output pattern; (b) extracting local parametrics from the tessellated output pattern; (c) determining if a degree of amplitude wandering representative of the local parametrics is within an allowable generator function limit; and (d) if not, renormalizing the tessellated output pattern to match spectral properties of the stimulus pattern and repeating (b)-(d); (2) performing a convergent reverberant dynamics resonance analysis on the OP of a biochip to identify mutations, comprising: (a) determining resonance dynamics relaxation values based on the preconditioned output pattern and resonance stimulus; (b) filtering the dynamics relaxation values using ensemble boundary and CSR filters to yield a second set of values; (c) applying bulk property estimators to the dynamics relaxation values to yield a third set of values; (d) evaluating the second and third sets of values to determine if resonance convergence has been achieved; and (e) determining if dynamic paralysis has occurred, and repeating the method if it has; (3) system for analyzing OP of a biochip to identify mutations comprising: (a) a tessellation unit operative to tessellate the output; (b) a stimulus pattern generation unit; (c) a resonance pattern generation unit and (d) a resonance pattern interpretation unit; and (4) system for performing method (2), comprising: (a) a determination unit; (b) a filter to filter dynamics relaxation values using ensemble boundary and CSR filters; (c) an estimator unit; (d) an evaluation unit; and (e) a paralysis detection unit.
Patent EP-1196365-B1 (EP)
Inventor: LINA MARIE-JOSE
IPC: C07C43/13
Filed: 2000-03-29
Granted: 2004-03-03
Abstract: The subject-matter of the invention is a fluorinated diol and its process of preparation. The fluorinated diol corresponds to the formula (I):in which n has a value from 2 to 20 and A means -CH=CH- or -CH2CH2- and R is an alkyl group comprising 1 to 4 carbon atoms.
Patent EP-1185771-B1 (EP)
Title: Procede de reduction d'emissions des gaz d'echappement d'un moteur a combustion interne
Inventor: ALMKVIST GOERAN
IPC: F02D41/02
Filed: 2000-06-08
Granted: 2004-03-24
Abstract: L'invention concerne un procédé de réduction d'émissions des gaz d'échappement d'un moteur à combustion interne (1) comprenant au moins un cylindre (2) auquel est acheminé un mélange air/carburant lorsque le vilebrequin du moteur (1) tourne, au moins une soupape d'admission (4), au moins une soupape d'échappement (6) et un piston (10) à mouvement alternatif entre une position centrale supérieure et une position centrale inférieure dans le cylindre (2). Le procédé consiste à acheminer vers le cylindre (2) un mélange air/carburant avec une valeur lambda supérieure à 1, à faire en sorte qu'un moteur/générateur électrique (17) relié au vilebrequin (3) maintienne une vitesse prédéterminée essentiellement constante du vilebrequin (3) et à commander une soupape d'échappement (6) de manière qu'elle s'ouvre avant que le piston (10) ne passe la position centrale inférieure.
Patent EP-1197025-B1 (EP)
Inventor: CARLSSON TORSTEN
IPC: H04B17/00
Filed: 2000-06-29
Granted: 2009-01-28
Abstract: A mobile station with a receiver having antenna diversity where the diversity processing is controlled from the base band processing circuit and only turned on when the performance gain justifies extra power consumption. The base band processing circuit may be instructed by the network that it can cease diversity reception after evaluating cell leads within a system.
Patent EP-1206320-B1 (EP)
Inventor: UNNO GARRETT
IPC: G01N35/00
Filed: 2000-08-10
Granted: 2007-06-06
Abstract: L'invention concerne des dispositifs et des systèmes microfluidiques, comprenant des éléments de manipulation, d'enregistrement ou d'indication qui communiquent une fonctionnalité du dispositif microfluidique à l'instrumentation utilisée avec lesdits dispositifs. Les éléments d'indicateurs comprennent des indicateurs structurels, des indicateurs électriques, des indicateurs optiques, et des indicateurs chimiques. Les différents éléments d'indicateurs indiquent différentes fonctionnalités, par exemple, des applications nouvelles quant à leur utilisation, et analogues.
Patent EP-1313958-B1 (EP)
Inventor: KORPIOLA KARI
IPC: D21F1/40
Filed: 2000-08-28
Granted: 2005-08-10
Abstract: Gas bearing for use in rolls (1) and rollers having a shaft (2) and a rotating envelope part (3) supported by bearings on the shaft, said bearing comprising an inner part fitted to the shaft (2) and an outer part fitted to the envelope (3), with a clearance (6) between the inner and outer parts, into which clearance a gas used for lubrication is supplied via nozzles (20) or a porous material. The inner part fitted on the outer surface of the shaft of the roll or roller consists of separate detachable sleeves or segments forming an inner ring (127), that the outer part rotating around the inner ring and having a cylindrical inner surface or consisting of cylindrical segments forms an outer ring (125), and that the inner and outer rings are attached via flexible or articulated joints to the shaft and the rotating envelope so that they allow the inner and outer rings to adapt to a common axis of rotation formed by the shaft and the envelope.
Patent EP-1217989-B1 (EP)
Inventor: GREGORIADIS GREGORY
IPC: C12N15/88
Filed: 2000-10-02
Granted: 2005-12-14
Abstract: An oral vaccine contain liposomes and complexed or, preferably entrapped, DNA operatively encoding an antigen in which the liposomes are formed from components including cationic compounds and zwitterionic phospholipids. The hydrophobic groups within the liposome forming components must include at least one group which is saturated. This is believed to raise the transition temperature, rendering the liposomes more stable when delivered orally. The compositions have been found to give detectable increased in IgA levels, secreted immunoglobulins of importance in efficacious oral vaccine delivery.
Patent EP-1118727-B1 (EP)
Inventor: BAERVELDT KONRAD
IPC: E01C11/10
Filed: 2001-01-16
Granted: 2003-05-02
Abstract: The present invention relates to a joint seal for use in joints that may be exposed to water, comprising at least one layer of a compressible impregnated open cell foam, on at least a portion of the surface of which is positioned a hydrophilic material. <IMAGE>
Patent EP-1142918-B1 (EP)
Inventor: USUI KAZUHIRO
IPC: C09D11/108
Filed: 2001-03-21
Granted: 2004-12-08
Abstract: The invention provides a novel chlorine-free modified polyolefin resin composition with excellent adherence to nonpolar substrates, with excellent solubility into solvent and compatibility with other resins, and with no tack after painting and drying. It relates to a modified polyolefin resin composition obtainable by graft modifying a mixed resin comprising 40 to 99 parts by weight of polyolefin resin (A) and 1 to 60 parts by weight of ethylenic compound-unsaturated carboxylic acid copolymer (B) that contains 0.1 to 50% by weight of unsaturated carboxylic acid derivative, with unsaturated carboxylic acid derivative and/or its anhydride (C), the modified polyolefin resin composition having weight average molecular weight of 20,000 to 150,000 and the grafting weight of (C) being 0.1 to 20% by weight.
Patent EP-1148309-B1 (EP)
Inventor: HOWARD LEE JARVIS
IPC: F25J3/02
Filed: 2001-04-12
Granted: 2004-03-03
Abstract: C<sub>2</sub> and C<sub>3</sub> hydrocarbons, particularly ethylene and propylene, are recovered from refinery or petrochemical plant gas mixtures by cooling and fractionating a feed gas mixture containing these hydrocarbons and lighter components. Refrigeration for the process is provided by a closed-loop gas expander (147) refrigeration process cycle which preferably uses nitrogen as the recirculating refrigerant. Cooling and fractionation may be effected in a dephlegmator (121).
Patent EP-1143035-B1 (EP)
Inventor: CARLSON DAVID K
IPC: H01L21/00
Filed: 1996-05-21
Granted: 2005-12-14
Abstract: An apparatus and a concomitant method for controlling coolant (air) flow proximate a reaction chamber (102) within a workpiece processing system (100) such that the temperature of a wall of the reaction chamber (102) is maintained at a predefined target temperature. The target temperature is typically a temperature that optimizes a process concurrently being accomplished within the chamber (102), e.g., utilizing one temperature during deposition processes and a different temperature during cleaning processes. The apparatus contains a temperature measuring device (140) to measure the temperature of the chamber wall. The measured temperature is compared to the predefined target temperature. A closed loop system controls the air flow proximate the chamber walls such that the measured temperature becomes substantially equal to the target temperature. Air flow control is provided by an air flow control device (138) located within an inlet conduit (120) that supplies air to a shroud for channeling the air past the reaction chamber (102). The shroud forms a portion of a housing (118) which supports and encloses the reaction chamber (102).