baber/WOPTO huggingface dataset:
Patent RU-2749437-C2 (RU)
Inventor: IN LEJ
IPC: A61P35/00
Filed: 2016-11-28
Granted: 2021-06-10
Abstract: Изобретение относится к соединениям формулы I, их дейтерированным производным и фармацевтически приемлемым солям, где в формуле I R1представляет собой атом водорода или C1-C6алкил; R2и R3представляют собой C1-C6алкил или R2и R3вместе с атомом C, к которому они присоединены, образуют C3-C6циклоалкил; R4и R5независимо выбраны из водорода и галогена, и по меньшей мере один из R4и R5представляет собой галоген; R6выбран из атома водорода или C1-C6алкила; R7представляет собой, Z представляет собой O или, и n равен целому числу от 0 до 4; каждый из W и Y независимо представляет собой C или N, но оба W и Y не могут одновременно представлять собой C, и если Z представляет собой O, W представляет собой C; R10, R11, R12и R13независимо выбраны из атома водорода, C1-C6алкила, C1-C6гидроксиалкила или циклопропилметила, или R6и R7вместе с атомами C, к которым они присоединены, образуют 6-членный гетероцикл, содержащий один атом N, который замещен; R8представляет собой C1-C6гидроксиалкил. Также изобретение относится к промежуточным соединениям формулы VI, способу получения и применению соединений формулы I, фармацевтической композиции, набору и способам лечения. Технический результат – соединения формулы I, обладающие ингибирующей активностью в отношении CDK 4/6. 9 н. и 20 з.п. ф-лы, 12 табл., 52 пр.
Patent RU-2736998-C2 (RU)
Title: Inbuilt meteorite
Inventor: RIGON MATTEO
IPC: A44C27/00
Filed: 2017-02-22
Granted: 2020-11-23
Abstract: FIELD: jewelry industry. 
     SUBSTANCE: invention relates to jewelry containing a meteorite enclosed in metal (hereinafter—built-in meteorite), and to a method of producing a built-in meteorite. Proposed method comprises the following operations: placing meteorite pieces into mold having flat bottom; metal is heated to temperature, equal to or greater than its melting point, for a time sufficient to melt the metal to produce molten metal; pouring said molten metal into said mold, containing meteorite pieces to produce initial combined material (ICM), which is a combination of said metal and meteorite; performing ICM cold pressing to produce sheet, having a predetermined thickness; said sheet is heated to a temperature equal to or greater than its melting point, but below the melting point of the meteorite pieces for a time sufficient to melt the metal, to obtain a built-in meteorite, and cold pressing of the built-in meteorite is performed. Method of making a jewelry product containing a built-in meteorite involves the following operations: obtaining a built-in meteorite containing a first metal; attaching the built-in meteorite to the jewelry containing the second metal and having the body adapted to receive the built-in meteorite, and heating the combination of the jewelry product and the built-in meteorite to a temperature sufficient for melting said first and second metals. 
     EFFECT: invention discloses a method of fusing a meteorite into a metal and a method of making a jewelry product containing a fused meteorite obtained using said method. 
     18 cl, 2 dwg
Patent RU-2733199-C2 (RU)
Title: Vehicle having detachable panel assembly
Inventor: ST-PER DENI
IPC: B60P1/64
Filed: 2017-06-15
Granted: 2020-09-29
Abstract: FIELD: transport machine building. 
     SUBSTANCE: according to the first version, the vehicle comprises a frame, a driver's seat, a plurality of elements for engagement with the ground, a motor connected to the ground engaging element, an assembled panel. Panel assy comprises cargo platform, left and right side panels, and platforms. Motor is accessible to the user when the panel assembly is removed, located behind the driver's seat and under the cargo platform. According to the second version, vehicle contains left and right doors connected with frame, and side panels are connected to frame near door hinges. According to the third version, the vehicle comprises the frame front part, the frame central part and the frame rear part. According to the first version, the method of access to the motor of the vehicle includes the stage, at which the fastening elements are dismantled, the frame parts are disconnected from the rest part of the frame, and removing assemblies and frame parts from vehicle. According to the second version, the method of access to the motor of the vehicle includes the stage, at which the rear instrument panels are disconnected from the frame. 
     EFFECT: easier access to the motor installed behind the vehicle. 
     16 cl, 14 dwg
Patent RU-2738422-C2 (RU)
Inventor: HOCKER JON A
IPC: A22C17/00
Filed: 2017-07-25
Granted: 2020-12-14
Abstract: FIELD: food industry. 
     SUBSTANCE: disclosed are treatment system (10) and corresponding method (158) for processing workpieces (WP), including food products, for cutting and removing undesirable components from food products and/or separating said products into parts during their movement in conveyor system (12). X-ray scanning station (14) is located in the upper by conveyor section (12) technological flow and is intended for determination of food products size and/or shape parameters, as well as location of any undesirable components of these products, such as bones, fat or cartilages. Further, the food products are transferred to lower conveyor (20), where optical scanner (102) is located, intended for determination of size and/or shape parameters of food products. X-ray and optical scanning results are transmitted to processor (18) to confirm that the food product scanned by the optical scanner is the same product, previously scanned by X-ray scanner. After confirmation of this identity (if necessary) data from X-ray scanner are translated or converted into data from optical scanner. Such translation may include one or more of the following: movement of food products in direction X and/or Y, rotation of food product, food product size changing and food product shear deformation. Further, the location of the undesirable material within the food product is displayed from the X-ray scanning data into the optical scanning data. After that unwanted material is removed by means of cutting device(s) (28). Food product (or alternatively) can be divided into parts by cutting device(s) (28). 
     EFFECT: proposed cutting/separation into parts using combined X-ray and optical scanning. 
     21 cl, 10 dwg
Patent RU-2755000-C2 (RU)
Title: Ligands to receptor of follicle-stimulating hormone (fsh) in diagnostics and treatment of tumors
Inventor: CARPI ANDREA
IPC: C07K14/59
Filed: 2017-10-10
Granted: 2021-09-08
Abstract: FIELD: medicine.SUBSTANCE: invention relates to the use of a ligand of a receptor of follicle-stimulating hormone (hereinafter – RFSH) of a human, which is a β-subunit of follicle-stimulating hormone (FSHβ) of a human, and which is characterized by a sequence SEQ. ID. no. 2 or a sequence that is at least 90% similar to the sequence corresponding to SEQ. ID. no. 2, preferably 90-99.9% or more similar, and more preferably 95-97% similar, for the treatment and/or diagnostics of tumors. A method for obtaining the ligand of the receptor of follicle-stimulating hormone (RFSH) of a human, which is a β-subunit of follicle-stimulating hormone (FSHβ) of a human, using recombinant DNA technology, is also proposed. Forms of FSH subunits of the present invention bind to FSHR with high affinity.EFFECT: producing the ligand of RFSH for the treatment of tumors.21 cl, 21 dwg
Patent RU-2757847-C2 (RU)
Title: Controlling the heating mode of food processor
Inventor: DERCAR HEINZ
IPC: A47J43/08
Filed: 2017-12-11
Granted: 2021-10-21
Abstract: FIELD: kitchen equipment. 
     SUBSTANCE: device (1) for processing a liquid food product contains: container (10) limiting cavity (10') for placing the specified liquid food product; impeller (20) for driving the liquid food product in container (10); engine (30) for driving impeller (20); engine compartment (40) for placing engine (30) and means for removing heat from engine compartment (40). Such a means includes one or more movable elements (50) that are driven by engine (30) and are made with the possibility to ensure the circulation of air flows (2a, 2b) in engine compartment (40) to remove heat from it.  
     EFFECT: provided is possibility of controlling the heating mode of the food processor. 
     29 cl, 2 dwg
Patent RU-2743031-C2 (RU)
Title: Additive for construction chemical compositions
Inventor: GAEDT TORBEN
IPC: C04B28/02
Filed: 2017-10-23
Granted: 2021-02-12
Abstract: FIELD: construction. 
     SUBSTANCE: present invention relates to an additive for construction chemical compositions, particularly compositions of mortar and cement compositions. Additive includes at least one amide or sugar acid ester and at least one water-soluble comb polymer, which contains on the main chain acid functions and side chains having ether functions. Additive is useful for slowing down hardening of the building chemical composition. Also described is a construction chemical composition and use of an additive for slowing hardening of compositions of construction mixtures. 
     EFFECT: disclosed is an additive for construction chemical compositions. 
     17 cl, 2 dwg, 4 tbl
Patent RU-2745834-C2 (RU)
Title: Device for growing mushrooms
Inventor: JACOBUS ALEXANDER JOZEF LEMMEN
IPC: A01G18/00
Filed: 2019-06-04
Granted: 2021-04-01
Abstract: FIELD: mushroom growing. 
     SUBSTANCE: invention relates to a device for growing mushrooms. The device contains a rack made to support the beds for placing compost, while the beds are arranged at the same distance one above the other. The beds are designed to move between at least the first position, in which the second bed, located above the first bed, at least partially makes it difficult to access the first bed in a direction perpendicular to the plane in which the first bed runs, and the second position, in which at least a large part of the first bed is freely accessible from the direction perpendicular to the plane in which the first bed extends, compared to the first position. At the same elevation, there is at least one pair of beds, the beds run parallel to each other, while a pair of beds at or essentially at the same elevation can rotate in the opposite direction. When the bed is turned, the side of the bed that faces the bed at the same level rises up, and when the bed is turned, the side of the bed that faces outward from the rack goes down.  
     EFFECT: device makes the production of cultivated mushrooms easier. 
     14 cl, 3 dwg
Patent RU-2766797-C2 (RU)
Title: Method for making dental prosthesis having internal through channel located at angle
Inventor: ANITUA ALDECOA EDUARDO
IPC: A61C8/00
Filed: 2018-08-27
Granted: 2022-03-15
Abstract: FIELD: medicine; dentistry. 
     SUBSTANCE: invention is intended for use in making a denture fixed on a dental implant. A dental prosthesis intended for direct or indirect connection with a dental implant is made, which includes an internal through channel located at an angle, for which the main part of the denture is obtained, wherein said main part has a first end intended for orientation in the direction of the dental implant, and a second end opposite to said first end. A first hole is drilled in said first end in a first direction. Middle area of said first hole is milled and expanded to produce expanded area. A second hole is drilled in said second end in a second direction, which forms an angle other than zero with the first direction, note here that said second opening extends to first opening. Inner end of the first hole, which enters from the second hole with formation of bend, is milled and expanded in lateral direction. 
     EFFECT: method allows making a prosthesis located at an angle to implants, with possibility of its fixation. 
     12 cl, 11 dwg
Patent UA-72508-C2 (UA)
Title: Device for digging out roots
Inventor: DAVYDIUK VASYL PETROVYCH
IPC: A01D25/04
Filed: 2001-10-10
Abstract: The present invention relates to the field of agricultural machine-building, in particular to root-diggers. New arrangement of working elements and changes in the construction of attachment thereof simplifies the device and ensures setting them in one row and the proper feeling of a row. An element of radial attachment of the plates is made of separate units and consists of a bushing, arranged in such a manner as to allow the longitudinal movement on a horizontal shaft, which is figured in the cross-section. In doing so the opposite ends of the bushing in the cross-section are also made as figured ones, where flanges of the radial attachment of plates, the longitudinal movement of which is limited by screws adjusting the gap between the elements of digging up the roots, are arranged. In addition inside the bushing in a bearing a two-arm lever is installed, the front arm of which is immovably connected with the row-feeling plates, and the rear arm supports a plate for releasing the roots gripped.
Patent UA-72817-C2 (UA)
Title: Method and apparatus for increase of efficiency and economy of use of complex methods of control of boundary layer
Inventor: MOORE KENNETH J
IPC: B63B1/38
Filed: 2001-07-17
Abstract: In an apparatus and method for ejecting an additive for significantly reducing the drag of a first fluid moving relative to a wall, a drag-reducing substance is conditioned by causing a second fluid (5), which includes the drag-reducing substance as a dispersed solid, liquid or gas. to flow through a nozzle (13). The second fluid is then passed by a vortex chamber (4) prior to ejection of the second fluid into the first fluid via an aperture that includes a Coanda surface (8) on a portion thereof. Additional techniques are also disclosed which increase the effectiveness and efficiency of ejecting a drag-reducing substance into a fluid that is moving relative to a wall, and which thus enable multiple layer 10 be established without the undesirable disruption of the boundary layer und without the rapid diffusion of the additives across the boundary layer that occur in prior art ejection techniques.
Patent UA-73373-C2 (UA)
Title: Door handle-latch
Inventor: SHULHA HRYHORII FEDOROVYCH
IPC: E05B1/00
Filed: 2003-03-19
Abstract: The door handle-latch to the set of which is included the lever with handle, this is fixed through aperture in the sheet of the insert through door by means of a rotary couple. The lever is equipped with coupling element, this interacts with a respective element of the onlay of the door frame placed at the level of the lever arm. The axis of rotation of the arm is placed in vertical position, and the lever itself is made with one arm and is equipped by one handle at its end and a coupling element placed at the side in the middle part; at that the aperture in the door sheet for the lever arm is arranged as a slot opened from three sides. Absence of the handle on the door indicates purposive closing of the door.
Patent UA-79312-C2 (UA)
Title: Method of forming wheel billets having rim, disk and nave
Inventor: YAKOVCHENKO OLEKSANDR VASYLIOV
IPC: B21K1/28
Filed: 2005-04-11
Abstract: The invention relates to the branch of metal forming, namely to the branch of hot upset-forging and die forging, and it is intended for use at producing the railroad wheels. A method of forming the wheel billets, which have rim, disk and nave, includes preliminary upset-forging of billet with simultaneous or subsequent spread of metal from its centre section to peripheral section and final forging of wheel billet in the moulding dies. During spreading on one of the sides of billet a the part of the rim is formed, which makes by volume not less than 75.0 % of the volume of counterpart of the rim in forged wheel billet, while in during forging by moulding ring the billet is displaced in horizontal plane to the alignment of the axis of billet with the one of dies. Technical result consists in reduction of the force of forging, increase of accuracy and stability of sizes of obtained wheel billets and wheels, which are rolled from them.
Patent UA-87460-C2 (UA)
Title: microstructured nozzle with filter (embodiments), sprayer for inhalation therapy and method of manufacturing nozzle
Inventor: EICHER JOACHIM
IPC: B05B15/00
Filed: 2004-06-23
Abstract: The invention relates to a microstructured nozzle comprising a plurality of channels, which are produced by microstructuring a plate-like body. The channels of said nozzle are disposed between projections which are arranged in rows next to each other and which project out of the base plate. Said microstructured base plate is covered with a cover plate. The channels are defined within narrow boundaries according to shape, cross-sectional area and length. Said nozzle contains a filter as a primary structure and a secondary structure is arranged downstream from the filler. The nozzle is, for example, used with a sprayer enabling an aerosol to be produced from a liquid, which contains a medicament.
Patent UA-82532-C2 (UA)
Title: Normal;heading 1;heading 2;FLUCONAZOLE CAPSULES WITH IMPROVED RELEASE
Inventor: FEKETE PAL
IPC: A61K9/48
Filed: 2004-06-30
Abstract: The object of the invention is to provide fluconazole containing capsules with improved active ingredient release. The in vitro dissolution as well as in vivo absorption of the fluconazole capsules according to the invention is faster and more consistent that) those of commercial compositions containing fluconazole. The invention is based on the fact that granulation of fluconazole particles with an agent capable to provide hydrophilic surface, e.g. lactose, to said particles results in fast an consistent release of the active ingredient. In this way, capsules according to the invention are suitable to provide enhanced absorption of said active ingredient.
Patent UA-86030-C2 (UA)
Title: Methods for the preparation of benzoxazole sulfonamide compounds and intermediates thereof
Inventor: DE KOCK HERMAN AUGUSTINUS
IPC: C07D417/12
Filed: 2004-09-30
Abstract: The present invention relates to methods for the preparation of benzoxazole sulfonamide compounds of formula (9) as well as novel intermediates of formula (6) for use in said method. More in particular the invention relates to methods for the preparation of 2-amino-benzoxazole sulfonamide compounds which make use of 2-mercapto-benzoxazole sulfonamide intermediates, more in particular methods employing the intermediate [-benzyl-2-hydroxy-3-[isobutyl(2-methylsulfanyl-benzoxazole-6-sulfonyl)-amino)-propyl)-carbamic ester, and to methods amenable to industrial scaling up. Said benzoxazole sulfonamide compounds arc particularly useful as HIV protease inhibitors. The substituents are defined in the claims.
Patent UA-79053-C2 (UA)
Title: Anticorrosive priming
Inventor: KONIUSHENKO VOLODYMYR PETROVYC
IPC: C08L61/00
Filed: 2006-03-09
Abstract: An anticorrosive priming for protective covering of pipelines contains butadiene-styrene rubber, n-tret-buthylphenol-formaldehyde resin, magnesium oxide, industrial carbon and aminomethyl derivatives of nonylphenoles as corrosion inhibitor, gallic acid propyl ether or pyrogallol as stabilizer, solvent petroleum as organic solvent and also polyethylene terephthalate and ethylene-vinyl-acetate resin. This priming provides advanced adhesive durability of polyethylene terephthalate cover against polyethylene and steel, the advanced adhesive durability against cathode layering at the elevated temperature, underfilm corrosion speed decreasing, priming's durability against aging increasing.
Patent UA-87501-C2 (UA)
Title: High-voltage power cable
Inventor: ZOLOTARIOV VOLODYMYR MYKHAILOVYCH
IPC: H01B9/00
Filed: 2007-01-18
Abstract: A power high-voltage cable comprises a water-blocking layer, its insulation is made of high-purity melt which is vulcanized and cooled in compressed nitrogen, and triing resistant polyethylene. The cable is triing resistant in case of using thereof for power supply networks of 100 kV and higher.
Patent UA-88023-C2 (UA)
Title: Information post of stand
Inventor: L HOTEL FRANCOIS
IPC: G09F1/06
Filed: 2005-10-05
Abstract: The invention concerns a support comprising at least one panel (2) made of substantially rigid and collapsible material including a display surface (3), return and stressing elastic bands (44) for dishing the display surface of the panel and a plurality of inserts (18-20) for maintaining the convexity of the display surface of the panel, countering the stressing rubber bands, and whereof the action is exerted discretely distributed along said display surface of the panel. The inserts (18-20) are equal in length to the distance between the two side edges (8, 9) of the panel (2), when it is dished, said panel being extended by two series of side flaps (12, 13, 14, 15, 16, 17) designed to form two series of dihedrals for receiving the inserts, the rubber bands (44) co-operating with the inserts and the flaps (12-17) and exerting, additionally to their horizontal stressing force, opposite vertical forces (49. 50) to maintain the inserts heightwise when the display surface is dished.
Patent UA-95771-C2 (UA)
Title: Device for electrochemical purification of waste water
Inventor: DONSKA MARIIA DMYTRIVNA
IPC: C02F101/32
Filed: 2007-05-16
Abstract: The invention relates to a device for electrochemical purification of waste water and can be used in chemical, gas and oil industries. The device comprises a body with nozzles for supply of initial water and discharge of purified one with arrangement of a cathode and an anode therein, made in the form of cylindrical tubes located coaxially to each other with a radial gap. The cathode is fixed in the inner cavity of anode and is made of several adjacent cylinder rings, separated from each other by cross annular channels, and on the external surface of each ring helical channels are made, and the anode is made of two semicylindrical electrodes, located in a tube of dielectric material.
Patent UA-93241-C2 (UA)
Title: New concept card and a selling system and method based on a buyer using the card
Inventor: LEE KIL-JIN
IPC: G06Q30/06
Filed: 2007-04-17
Abstract: A new concept card and a selling system and method based on a buyer using the card are disclosed. The system includes a card system 4 which issues a new concept card for allowing a card company to identify a seller or registers or grants information to a seller, a seller system 3 or terminal 31 which allows the seller to receive the UC or information and to advertise the card or information to a buyer and allows the buyer to purchase merchandise, a buyer terminal 1 which allows the buyer to access the seller system or terminal so as to purchase merchandise or acquire the UC information and to access the card company to rapidly/accurately input the UC or seller information such that credit card approval is requested, and a bank system 2 which processes the credit car approval when the buyer requests the credit card approval.