baber/WOPTO huggingface dataset:
Patent BR-PI1000087-B1 (BR)
Title: Calçado, acessório, combinação calçado/acessório e processo para sua produção
Inventor: EDSON MATSUO
IPC: A43B3/12
Filed: 2010-01-07
Abstract: calçado, acessório, combinação calçado/acessório e processo para sua produção a presente invenção proporciona calçados, acessórios e uma combinação calçado/acessórios, bem como um processo para sua obtenção. a invenção proporciona, entre outras vantagens: o ajuste do calçado às necessidades do usuário; o uso de diferentes acessórios em combinação com o calçado, dependendo da situação específica; e o uso de acessórios individuais da combinação separadamente do calçado. além disso, a invenção inclui um processo que confere grande versatilidade na produção industrial, visto que com um modelo único o fabricante é capaz de adequá-lo às várias tendências de sua linha de produção, diminuindo sensivelmente o custo da produção dos calçados.
Patent BR-PI1008975-B1 (BR)
Title: Meios de dispensação/espalhamento para dispensar uma substância colorante em pó sobre a superfície de uma mistura, aparelho para distribuir em uma camada fina uma mistura com base em material de pedra ou cerâmico sobre um suporte subjacente, e, método para distribuir em uma camada fina uma mistura com base em material de pedra ou cerâmico e/ou um aglutinante sobre um suporte
Inventor: LUCA TONCELLI
IPC: B28B1/00
Filed: 2010-03-09
Abstract: meios de dispensação/espalhamento para dispensar uma substância colorante em pó sobre a superfície de uma mistura, aparelho para distribuir em uma camada fina uma mistura com base em material de pedra ou cerâmico sobre um suporte subjacente, e, método para distribuir em uma camada fina uma mistura com base em material de pedra ou cerâmico e/ou um aglutinante sobre um suporte meios para dispensar uma substância colorante em pó sobre a superfície de uma mistura (14) que compreende material de pedra, material similar a pedra, vidro ou cerâmica. o dispositivo compreende, pelo menos, um meio de dispensação (28) para conter e dispensar uma substância colorante em pó (11) e no, mínimo, um dispositivo de espalhamento (30). o dispositivo de espalhamento (30) compreende, pelo menos, uma placa perfurada móvel (100) que recebe uma quantidade dosada da dita substância colorante (11) a partir do dispositivo de dispensação (28) e a distribui sobre a superfície da mistura (14).
Patent EA-003706-B1 (EA)
Title: A process for preparation of 1,4,7,10-tetraazacyclododecane
Inventor: ARGESE MARIA
IPC: C07C/
Filed: 2000-03-06
Abstract: 1. A process for the preparation of the compound of formula (I), 1,4,7,10-tetraazacyclododecane, according to the following scheme 1: Scheme 1: a) condensation of triethylenetetramine (TETA) with glyoxal hydrate in water or water-soluble solvents or mixtures thereof, at a temperature ranging from 0 to 5 degree C, in the presence of stoichiometric amounts or of a slight excess of calcium hydroxide, to give the compound of formula (IV); b) reaction of compound of formula (IV) with 1,2-dichloroethane, in amounts from 1 to 5 mol per mol of compound (IV), in dimethylacetamide (DMAC) and in the presence of Na2CO3, in amounts from 5 to 10 mol per mol of compound (IV), adding NaBr in amounts from 0.1 to 2 mol per mol of compound (IV) at a temperature from 25 to 150 degree C, to give the compound of formula (III) which is isolated in the form of a salt of an inorganic acid selected from the group consisting of hydrochloric acid and phosphoric acid; c) hydrolysis of compound (III) by reaction with diethylenetriamine in water, at pH ranging from 5 to 9, at a temperature ranging from 90 to 120 degree C, in the presence of 5-10 mols of diethylenetriamine per mol of compound (III), under inert gas atmosphere or in the air, for 12-48 h, recovering compound (II) as the tetrahydrochloride; and optionally d) quantitative liberation of the base to give compound of formula (I). 2. A process as claimed in claim 1, in which condensation of compound (III) in step b) is carried out with 3-5 mol of 1,2-dichloroethane per mol of compound (III), in dimethylacetamide (DMAC), in the presence of sodium carbonate, and with the addition of NaBr as a catalyst in amounts from 0.1 to 2 mol per mol of compound (IV). 3. A process as claimed in claim 2, in which 3 mol of 1,2-dichloroethane, 10 mol of sodium carbonate and 0.5 mol of NaBr are used. 4. A process according to claims 1 to 3, in which the final reaction mixture from step b) is added with an amount of concentrated HCl equivalent to 2-4 mol/mol of compound (IV). 5. A process as claimed in claim 4, wherein the concentration of the solution is 6 L of DMAC/mol of compound (IV). 6. A process according to claims 1 to 3, in which the final reaction mixture from step b) is added with an amount of 85% H3PO4 equivalent to at least 2 mol/mol of compound (IV). 7. A process as claimed in claim 6, wherein the concentration of the solution is equivalent to 4.5 L of DMAC/mol of compound (IV). 8. A process according to claims 1 to 7, in which in step c) the molar ratio of salt of compound (III) to diethylenetriamine is 1: 5.
Patent EA-007403-B1 (EA)
Title: Device for discharging liquids, a cartridge suited therefor, and a system comprised of the device for discharging liquids and of the cartridge
Inventor: SCHIEWE JOERG
IPC: A61M15/00
Filed: 2003-08-26
Abstract: The invention relates to a propellant gas-free device for discharging liquids, to a cartridge, which is adapted thereto and which is provided for storing the liquid, and to the ensemble comprised of both the device and cartridge. The invention consists of a device (1) for supplying pressure and for accommodating a cartridge (10), and of a cartridge (10) inside of which a discharging device (29) is integrated.
Patent EA-007584-B1 (EA)
Title: A seed tape including successively arranged germinating units
Inventor: AHM POUL HENRIK
IPC: A01C1/04
Filed: 2004-07-02
Abstract: A seed tape (1) including successively arranged germinating units (la, l b, 1c). The seed tape includes at least one carrier strip (3) as well as at least one auxiliary layer (5) arranged thereon and made of a biodegradable, flexible, non-woven, film-like material. Locally, the auxiliary layer (5) can be interrupted over a short distance along the seed tape (1). Each germinating unit (la, l b, 1c) includes a mixture (6) of granulated carrier, at least one granulated additive and optionally an adjuvant in addition to one or more seeds (7). This mixture (6) is kept together to form at least one core portion (8) in the germinating unit. The core portion (8) includes locally adhered bicomponent fibres (18) of one or more thermoplastic materials which form a coherent open network (8a) for keeping the granules (6a) of the mixture (5) and possibly also one or more seeds (7) together. In this manner it is possible in a very simple and reliable manner to retain the carrier, the additive and the adjuvant, if any.
Patent EA-009533-B1 (EA)
Title: Process for the preparation of urea granules
Inventor: MUTSERS STANISLAUS MARTINUS PETRUS
IPC: B01J2/16
Filed: 2004-10-15
Abstract: Process for the preparation of urea granules in a fluid-bed granulator, by using at least one feeding device to feed a urea melt in the form of a film to a fluidized bed of solid urea nuclei, upon which the nuclei grow by solidification of the urea melt on the nuclei, in which the amounts of biuret and water in the urea melt and in the urea granules fulfill the following relation (I) ) b∙b/w(w-w) = 0,1-20, wherein b= the % by weight of biuret in the urea melt; b= the % by weight of biuret in the urea granules; w= the % by weight of water in the urea melt; w= the % by weight of water in the urea granules.
Patent EA-011714-B1 (EA)
Title: N-(1h-indolyl)-1h-indole-2-carboxamide derivatives, their preparation and their therapeutic use
Inventor: DUBOIS LAURENT
IPC: C07D209/42
Filed: 2005-08-02
Abstract: A compound of the formula (I) in which X, X, X, X, Z, Z, Z, Zand Zrepresent, independently of one another, a hydrogen or halogen atom or a C-C-alkyl, C-C-cycloalkyl, C-C-fluoroalkyl, C-C-alkoxy, C-C-fluoroalkoxy, cyano, C(O)NRR, nitro, NRR, C-Cthioalkyl, -S(O)- C-C-alkyl, -S(O)- C-C-alkyl, SONR1R, NRCOR, NRSORor aryl group; Xrepresents a hydrogen or halogen atom or a C-C-alkyl or C-C-fluoroalkyl group; R represents a 4-, 5-, 6- or 7-indolyl group, optionally substituted, Y represents a hydrogen atom or a C-C-alkyl group; n is equal to 0, 1, 2 or 3; Rand Rrepresent, independently of one another, a hydrogen atom or a C-C-alkyl, C-C-cycloalkyl, C-C-cycloalkyl-C-C-alkyl or aryl group; or Rand Rform, together with the nitrogen atom which carries them, an azetidine, pyrrolidine, piperidine, azepine, morpholine, thiomorpholine, piperazine or homopiperazine group, said group optionally being substituted by a C-C-alkyl, C-C-cycloalkyl, C-C-cycloalkyl-C-C-alkyl or aryl group; Rand Rrepresent, independently of one another, a hydrogen atom or a C-C-alkyl or aryl group; Rrepresents a C-C-alkyl or aryl group; in base or acid addition salt, hydrate or solvate form. The invention also concerns a method for preparing said compounds and their therapeutic use.
Patent EA-015146-B1 (EA)
Title: Compositions and methods relating to anti igf-1 receptor antibodies
Inventor: CALZONE FRANK J
IPC: A61P37/00
Filed: 2005-12-20
Abstract: The present invention provides compositions and methods relating to or derived from anti-IGF-1R antibodies. In particular embodiments, the invention provides fully human, humanized, or chimeric antiIGF-1R antibodies that bind human IGF-1R, IGF-1R-binding fragments and derivatives of such antibodies, and IGF-1R-binding polypeptides comprising such fragments. Other embodiments provide nucleic acids encoding such antibodies, antibody fragments and derivatives and polypeptides, cells comprising such polynucleotides, methods of making such antibodies, antibody fragments and derivatives and polypeptides, and methods of using such antibodies, antibody fragments and derivatives and polypeptides, including methods of treating or diagnosing subjects having IGF-1R-related disorders or conditions.
Patent EA-010386-B1 (EA)
Title: Method for simultaneous recovering a c3+ hydrocarbon-rich cut and ethane-rich stream from natural gas and installation therefor
Inventor: PARADOWSKI HENRI
IPC: F25J3/00
Filed: 2005-12-19
Abstract: The invention concerns a method comprising cooling the initial natural gas (13) and introducing same into a C2+ hydrocarbon recovery column (35). It comprises recovering the overhead stream (131) of the column (35) to form the treated natural gas (15), and recovering the bottoms stream (171) of the column (35) to introduce same at a supply level (P1) of the fractionating column (61) provided with an overhead condenser (63). The column (61) produces in the bottoms said C3+ hydrocarbon cut (17). The method comprises recovering the ethane-rich stream (19) from the intermediate level (P2) of the column (61), located above said supply level (P1) and the production of a secondary reflux stream (191) from said overhead condenser (63) introduced in reflux into the recovery column (35).
Patent EA-015254-B1 (EA)
Title: Triazole derivatives
Inventor: CEZANNE BERTRAM
IPC: C07D487/04
Filed: 2006-11-24
Abstract: Novel triazole derivatives, inhibitors of TGF-beta receptor I kinase, of application, amongst other things, to the treatment of tumours.
Patent EA-015939-B1 (EA)
Title: Polypropylene composition, process for preparing and use thereof
Inventor: AASETRE SVEINUNG
IPC: B29C48/08
Filed: 2007-02-13
Abstract: The present invention provides a polymer composition comprising: (i) 0.05 to 15 wt.% of a propylene polymer comprising a polymeric nucleating agent, said agent preferably containing vinyl compound units; and (ii) 85 to 99.95 wt.% of a heterophasic propylene polymer which does not comprise a polymeric nucleating agent, wherein the weight ratio of (i):(ii) is 10:90 to 1:99, and the amount of polymeric nucleating agent based on the total weight of the composition is 0.01 to 100 ppm wt. The invention also provides the process for preparing said polymer composition comprising blending (i) and (ii) in the defined ratio and use thereof for preparing articles by moulding, thermoforming or extrusion.
Patent EA-013420-B1 (EA)
Title: A device for delivering medical treatment
Inventor: FIERENS JOOST J
IPC: A61M25/10
Filed: 2007-03-20
Abstract: The present invention provides a medical device for the delivery of treatment fluid to body vessels, having a distal (21) and a proximal (20) end, comprising a self-expanding, hollow tubular member (9) and a delivery catheter (10) suitable for deploying a self-expanding, tubular member (9), wherein the tubular member (9) is configured to expand radially to form a central part (11) flanked by two annular ridges, which creates, in situ, an annular lumen for that can apply treatment fluid locally to a vessel and a passageway that can maintain the flow of blood though the vessel. The device is particularly suited for minimally invasive and repeatable organ perfusion. It also relates to a method for organ perfusion.
Patent EA-016948-B1 (EA)
Title: Nicotinic acetylcholine receptor modulators
Inventor: GHIRON CHIARA
IPC: A61K31/4155
Filed: 2008-01-16
Abstract: The present invention provides compounds of formula (I) and compositions thereof, methods of making them, and methods of using them to modulate alpha7 nicotinic acetylcholine receptors and/or to treat any of a variety of disorders, diseases, and conditions. Provided compounds can affect, among other things, neurological, psychiatric and/or inflammatory system.
Patent EA-014669-B1 (EA)
Title: Interferon-based formulation
Inventor: PROKULEVICH VLADIMIR ANTONOVICH
IPC: A61K38/21
Filed: 2009-06-08
Abstract: The invention relates to the field of medicine, veterinary medicine, chemical and pharmaceutical industry, biotechnology and can be used at production of medical and preventive immunobiological drugs, having durable immunomodulatory and antiviral action. In particular, the invention relates to the bioactive formulations on the basis of recombinant interferons. It is suggested an interferon based formulation, comprising α-interferon, stabilizer and water, which contains at least one fat-soluble vitamin in the form of colloidal particles as the stabilizer and additionally contains sodium benzoate as a preservative and sodium chloride as an agent, providing osmoticity of solution at the following components content per 1 liter of solution:A formulation can preferably contain as a stabilizer one fat-soluble vitamin in the form of colloidal particles, chosen from the group of vitamins A, D, E, B or a mixture of fat-soluble vitamins A, D, E in the form of colloidal particles, if necessary, with the water-soluble vitamins C and B12. The preparation presents a stable solution, having improved therapeutic action and providing preservation of a high level of immunomodulatory and antiviral activity in the body for a long period of time, as well as a faster and more effective action of interferon at early stages after administration into the body.
Patent EA-017552-B1 (EA)
Title: Method of stratified deposit development for chamber mining
Inventor: SMYCHNIK ANATOLIJ DANILOVICH
IPC: E21C41/16
Filed: 2010-06-28
Abstract: This invention relates to the mining, it extends the field of application of mining equipment used at deposits with seam inclinations bigger than maximum permissible ones for series-produced mining equipment which became common use at horizontal and low-inclined seams. The way comprises main, panel and block openings where main and block openings are driven at an angle α to dip direction, and angle α is determined fromwhere j is maximum permissible inclination angle of main and block openings to horizontal plane at which usage of mining equipment is possible, degree; β - dip angle, degree, with j≤β.
Patent EA-018747-B1 (EA)
Title: Method for producing catalysts
Inventor: WALLER DAVID
IPC: B01D46/24
Filed: 2008-07-04
Abstract: The invention relates to a process to produce catalysts by powder injection moulding and the catalysts thereof, wherein the catalysts are made by preparing a ceramic formulation with temperature controlled rheological properties comprising catalytic components, heating the powder formulation up to at least the fluid state transition temperature, shaping a sample by injecting the fluid powder formulation into an injection mould followed by cooling the injected powder formulation below the fluid state transition temperature, de-binding the shaped sample, and sintering the shaped sample to form a ceramic catalyst. Alternatively the ceramic structure may be formed initially followed by a coating of the ceramic structure by one or more catalytic compounds.
Patent EA-018784-B1 (EA)
Title: Compositions and methods for controlling nematodes
Inventor: WILLIAMS DERYCK J
IPC: A01N43/64
Filed: 2008-08-13
Abstract: The present invention provides processes for controlling plant parasitic nematodes comprising administering to plants, seeds or soil a composition comprising an effective amount of a compound of formula (IV) or a compound of formula (V).
Patent EA-017154-B1 (EA)
Title: Amino arylsulfonamide compounds and their use as 5-htligands
Inventor: RAMAKRISHNA NIRODI VENKATA SATYA
IPC: A61K31/404
Filed: 2008-05-02
Abstract: The present invention relates to novel amino arylsulfonamide compounds of the formula (I), their derivatives, their stereoisomers, their pharmaceutically acceptable salts and pharmaceutically acceptable compositions containing them. The present invention also relates to a process for the preparation of above said novel compounds, their derivatives, their stereoisomers, their pharmaceutically acceptable salts and pharmaceutically acceptable compositions containing them. The compounds of the invention are useful in the treatment of various disorders that are related to 5-HT6 receptor functions. Specifically, the compounds of this invention are also useful in the treatment of various CNS disorders, hematological disorders, eating disorders, obesity, anxiety, depression, diseases associated with pain, respiratory diseases, gastrointestinal, cardiovascular diseases and cancer.
Patent EA-030512-B1 (EA)
Title: High polymer content hybrid drag reducers
Inventor: MILLIGAN STUART N
IPC: C08L23/00
Filed: 2008-07-30
Abstract: A drag reducing composition comprising particles of at least two different drag reducing polymers. The different drag reducing polymers can be formed by different processes, such as bulk polymerization or emulsion polymerization, and the particles of the different drag reducing polymers can have different mean particle sizes. The drag reducing compositions can be added to a hydrocarbon-containing fluid to decrease the pressure drop associated with the turbulent flow of the hydrocarbon-containing fluid through a conduit.
Patent EA-021940-B1 (EA)
Title: Pharmaceutical composition based on rotigotine dihydrophosphate
Inventor: BOUWSTRA J A
IPC: C07D333/20
Filed: 2010-06-24
Abstract: The present invention relates to pharmaceutical compositions for prevention or treatment of CNS disorders like Parkinson Disease, Restless Legs Syndrome, Parkinson Plus Syndrome, depression, fibromyalgia and/or Parkinson's accessory symptoms comprising rotigotine dihydrophosphate, wherein pH≤5. The compositions can be used in a transdermal delivery system, for example, in an ionophoretic system. The use of said compositions is characterised by improved transdermal delivery of a formulation in a patient.
Patent EA-025274-B1 (EA)
Title: Reusable auto-injector
Inventor: JENNINGS DOUGLAS IVAN
IPC: A61M5/20
Filed: 2009-06-10
Abstract: The invention is related to the field of medical equipment. Claimed is an automatic injection device (110) with an adaptor for transfer of a fluid medium from a container to a chamber comprising a first assembly including a chamber (116) accommodating fluid medium, said chamber comprising an inner surface and an outlet opening (144); a stopper (112) made of an elastic material, movable inside the chamber and having an outside surface substantially contacting the inner surface over its periphery; and an adaptor able to transfer fluid medium to the chamber where the adaptor includes a means for moving the stopper (112) through the chamber (116), and a means for transfer of fluid medium into the chamber (116) as the stopper (112) moves from the closed outlet opening; the adaptor being able to receive a fluid medium container (132) and to transfer fluid medium from the container to the chamber (116) by means of a fluid medium channel; characterized in that it comprises a second assembly including a detachable drive mechanism, said drive mechanism including an elongated rod that acts directly on the stopper after activation of the drive mechanism, the means for transfer of fluid medium into the chamber (116) comprising a hollow fluid medium transfer needle (128) engageable with the fluid medium container for fluid medium transfer from the fluid medium container through the hollow needle when the stopper is shifted away from the outlet opening; and the hollow needle is able to pierce the stopper (112) so that the hollow needle extends from the container to the chamber to feed fluid medium through the stopper to the chamber (116). Also claimed is a method for introduction of fluid medium into the automatic injection device and a set for injections including the automatic injection device. The invention provides versatility and reduction of labour efforts while using.
Patent EA-021587-B1 (EA)
Title: Haloalkyl heteroaryl benzamide compounds
Inventor: ROSSIGNOL JEAN-FRANCOIS
IPC: C07C233/00
Filed: 2010-05-11
Abstract: A new class of haloalkyl heteroaryl benzamides is described. These compounds show strong activity against hepatitis viruses.
Patent EA-024365-B1 (EA)
Title: Pharmaceutical composition comprising tamsulosin and process for preparing the same
Inventor: SEDMAK GREGOR
IPC: A61K9/20
Filed: 2010-05-26
Abstract: The present invention relates to a pharmaceutical composition comprising tamsulosin or a pharmaceutically acceptable salt or solvate thereof in a solid dosage form and to a process for preparing such a composition.
Patent EA-022149-B1 (EA)
Title: Absorbent article
Inventor: TAKINO SHUNSUKE
IPC: A61F13/49
Filed: 2008-09-03
Abstract: The invention is aimed at creating an absorbent article providing the discharge of evaporations from the article for alleviating dampness feeling experienced otherwise by the article user. The present invention provides an absorbent article, comprising belt members 4, forming correspondingly a front belt region 1 and a rear belt region 2, and a moisture absorption structure 5, which forms an intermediate region 3, wherein the belt members 4 have elastic elements 18, surrounding the waist and causing shrinking said belt members 4 in the circumferential direction R. The moisture absorption structure 5 has a first edge 24 and a second edge 25, wherein the outer surface of the first edge 24 overlaps the inner surface of the front belt region 6, forming a first overlapping region 26, and the outer surface of the second edge 25 overlaps the inner surface of the rear belt region 7, forming a second overlapping region 27. The moisture absorption structure 5 is bonded to the front and rear belt regions 6 and 7 in the first and second overlapping regions 26 and 27 by butt regions 32 extending in the vertical direction Z and arranged in spaces in the circumferential direction R. First joinless regions 45 formed between each pair of the adjacent butt regions 32 form ventilation passages 34 and 35, which provide the intermediate region 3 to cooperate with the front and rear belt regions 1 and 2.