baber/WOPTO huggingface dataset:
Patent HU-194232-B (HU)
Title: Process for preparing 1-/amino-carbonyl-methyl/-imidazo/1,2-a/quinoline derivatives and pharmaceuticals comprising these compounds
Inventor: GEORGE PASCAL
IPC: A61K31/435
Filed: 1987-01-21
Abstract: 1. Claims for the Contracting States : BE, CH, DE, FR, GB, IT, LI, LU, NL, SE Imidazo[1,2-_a]quinoline derivatives corresponding to the formula (I)  see diagramm : EP0233800,P14,F1  in which X denotes hydrogen, a halogen or a (C1-4 )alkyl, (C1-4 )-alkoxy, (C1-4 )alkylthio, methylsulphonyl, amino, (C1-4 )-alkylamino, di(C1-4 )alkylamino, nitro or trifluoroalkyl group, Y denotes hydrogen, a halogen or a methyl group at position 6, 7 or 8, and R1 and R2, taken separately, each denote hydrogen or a (C1-6 )alkyl group, or alternatively R1 and R2 together form a tetramethylene, pentamethylene, 3-methyl-3-azapentamethylene or 3-oxapentamethylene chain, as well as their addition salts which are acceptable in pharmacology. 1. Claims for the Contracting States : AT, ES, GR Process for the preparation of imidazo[1,2-_a]quinoline derivatives corresponding to the formula (I)  see diagramm : EP0233800,P16,F1  in which X denotes hydrogen, a halogen or a (C1-4 )alkyl, (C1-4 )-alkoxy, (C1-4 )alkylthio, methylsulphonyl, amino, (C1-4 )-alkylamino, di(C1-4 )alkylamino, nitro or trifluoroalkyl group, Y denotes hydrogen, a halogen or a methyl group at position 6, 7 or 8, and R1 and R2, taken separately, each denote hydrogen or a (C1-6 )alkyl group, or alternatively R1 and R2 together form a tetramethylene, pentamethylene, 3-methyl-3-azapentamethylene or 3-oxapentamethylene chain, which process is characterized in that the quinoline of formula (II)  see diagramm : EP0233800,P16,F2  is first subjected to the action of an alpha-bromoacetophenone bearing the substituent X defined above, in the heated state in a solvent such as methylene chloride or 1,2-dichloroethane ; an ionic compound of formula (III)  see diagramm : EP0233800,P16,F3  is obtained, which is cyclized in the presence of ammonium acetate, in an acidic organic solvent such as acetic or propionic acid, at a temperature of 90 degrees C, to obtain the compound of formula (IV)  see diagramm : EP0233800,P16,F4  the compound obtained (IV) is reacted with glyoxylic acid in a solvent such as acetic acid at 80 degrees C ; the alpha-hydroxy acid obtained (V)  see diagramm : EP0233800,P17,F1  is acetylated using acetic anhydride in the presence of pyridine, and then converted to the alpha-acetoxyacetamide  see diagramm : EP0233800,P17,F2  via the imidazolide, which is prepared in situ ; the compound (VI) is deacetylated to the alpha-hydroxyacetamide (VII) see diagramm : EP0233800,P17,F3  by treatment with potassium carbonate in ethanol ; the compound (VII) is reacted with sulphonyl chloride SOCl2 in a chlorinated solvent such as dichloromethane, to obtain the chlorinated compound (VIII)  see diagramm : EP0233800,P17,F4  which is reduced using Rongalite**(r) in methylene chloride to the compound (I).
Patent HU-185877-B (HU)
Inventor: OPITZ RUDOLF
IPC: D06L4/75
Filed: 1980-03-05
Abstract: A találmány tárgya fehérítőszer előnyösen mosó- és tisztítószrekhez, különösen alacsonyabb hőmérsékleten történő felhasználásra, amely 10—90%, szervetlen peroxivegyüleíből, vagy 90—89%, szerves peroxivegyületből és/vagy 15—70%, szervetlen peroxivegyület aktiválására alkalmas aktivátorból valamint 0,1—10%, mennyiségben fémkelátkomplexből áll, és fémkelátkomplexként egy M.íMzUXmjY képletű, előnyösen (M2UXJY Mi jelentése egy vagy több alkáli- és/vagy alkáliföldfémion, M2 jelentése réz, cink, króm, mangán, vas, kobalt vagy nikkel, L jelentése egy kelátképző ligandum, X jelentése semleges ligandum, éspedig víz vagy komplex amion éspedig etilén-diamin-tetraaeetát-ion, nitrát-, szulfát-, klorid-, vagy hidroxilion. Y jelentése egy vagy több anion, n jelentése 1 és 3 közötti egész szám, m jelentése 0 és 4 közötti egész szám. -1-
Patent HU-187553-B (HU)
Title: Building member for making model particularly for building toys
Inventor: BOLLI PETER
IPC: A63H33/04
Filed: 1984-02-13
Abstract: A building block is provided having side walls and a top face with two rows of coupling pins on the one side of the top face and counter-coupling tubes on the other side for mechanically coupling two such building blocks by means of a clamping action. On their side faces, the coupling pins have electrically conducting regions, which extend over an angular range. The angular range of one row being turned by 180 DEG  relative to those of the other row. All the conducting regions are connected to a contact bar, which is arranged on the side of the counter-coupling tubes along one side wall. When two building blocks are coupled arbitrarily, at least one conducting region of each row of coupling pins of the one building block makes contact with a contact bar of the other building block in such a way, that a short circuit cannot occur in the two electrical circuits assigned to each row of coupling pins or each contact bar.
Patent HU-210148-B (HU)
Title: Process for producing quinoline and pyridine derivatives and pharmaceutical compositions containing them
Inventor: ROBL JEFFREY ADAM
IPC: C07F9/58
Filed: 1991-02-25
Abstract: Compounds which are useful as inhibitors of cholesterol biosynthesis and thus as hypocholesterolemic agents are provided which have a quinoline or a pyridine anchor attached by means of a linker to a binding domain sidechain, which compounds inhibit the enzyme 3-hydroxy-3-methylglutaryl-coenzyme A reductase.
Patent LT-4162-B (LT)
Title: Mower-collector for use on embankments
Inventor: RAGAUSKAS STASYS
IPC: A01D34/42
Filed: 1995-07-13
Abstract: Invention belongs to agriculture, drainage domain and may be used to cut the grass on the embankments of drainage trenches or roadside slopes.The hay cutting and collecting device consists of a girder-type arm (2) with cutting device (1) hinge-connected at its end, as well as a turning column (3), frame (4) and container (5).  Inside the arm (2), beginning from its end the following parts are respectively installed: a collector (10), a shaping chamber (11) and a passive transporter (12), which consists of parallel (in respect of the arm axis) guides (13).  Inside the collector (10) and shaping chamber (11) there is installed a transporting screw (14), which consists of a conical part (19) and two cylindrical parts (20, 21) of different diameter.  The diameter of the cylindrical part of the screw (21) corresponds to the inner diameter of the collector's (10) gutter (15), and the diameter of the conical part (19) and the cylindrical part (20) correspond respectively to the inner diameter of the two parts (17, 18) of the shaping chamber (11).The operating part (22) of the cutting device (1) cuts hay and directs it towards the collector (10).  The cut hay, on hitting the guide (16), falls down on the screw (14), which shapes it into a cylinder of hay and pushes it upwards by transporter (12) guides (13) until the cylinder of hay, having reached the end of the transporter, falls to the container (5), and is further unloaded onto a vehicle.
Patent YU-49057-B (YU)
Inventor: TRBOJEVIC RADMILA
Filed: 1992-05-26
Abstract: Postupak za dobijanje 1,1-dioksida penicilanske kiseline i njenih alkalnih soli, koji se izvodi u jednoj fazi i sa kraćim vremenom izvođenja, naznačen time, što se 6-amino penicilanska kiselina prvo diazotuje sa 0,4 do 0,8 masenih udela NaNO2 i zatim bromuje u smeši sumporne kiseline i etil-acetata pri čemu je odnos smeše 12ml do 16ml po 1g 6-APK, u temperaturnom intervalu od 0В°C do 10В°C, pri čemu se na pH=7, na izdvojeni vodeni sloj deluje oskidacionom smešom koja se sastoji od 1,1 masena udela KMnO4, 0,35ml 85% H3PO4 i 11ml H2O po 1g 6-APK, u temperaturnom intervalu od t=-5В°C do t=+5В°C, posle čega se dobijeni proizvodi oksidacije, posle ekstrahovanja sa 15ml do 25ml etil-acetata po 1g 6-APK, bez izolovanja dehalogenuju sa cinkom u prahu u količini od 0,6g do 1g po 1g 6-APK u prisustvu 5M HCl. Prijava sadrži još 3 zavisna zahteva.
Patent AT-399228-B (AT)
Inventor: MOESTL ANTON DIPL ING
IPC: G01N21/11
Filed: 1990-06-08
Granted: 1995-04-25
Abstract: Method of analysing gaseous or liquid samples using a disposable measuring element having a measuring channel which contains at least one optical or electrochemical sensor and provided with closure devices at both ends. To achieve an accurate measurement in a simple way, in carrying out the measurement a storage medium is first replaced in the measuring channel by a separating medium and the separating medium is then replaced by the sample. Sample and storage medium are retained when the measuring element is disposed of.
Patent AT-395540-B (AT)
Title: Articulated model railway vehicle
IPC: A63H19/10
Filed: 1989-07-21
Granted: 1993-01-25
Abstract: The invention relates to an articulated model railway vehicle 1, having two independently runnable vehicle parts 2, 3 which can be connected together by a coupling apparatus 15 and each have their own running gear 4, 5, wherein each running gear 4, 5 is provided with a drive arrangement 6, 7 of its own, and having a coupling arrangement 18 parallel to the coupling apparatus 15 and connected for movement, so as to be releasable as necessary, to drive elements of the two drive arrangements 6, 7, with the interposition of a cardan arrangement 19, 20. Arranged between the drive elements of the two drive arrangements 6, 7 is a longitudinal adjustment apparatus 34 comprising two parts adjustable relative to one another and integrated into the cardan arrangement 19, 20. A cardan sleeve 29 has a greater length in the direction of cardan shaft 33 than a diameter 36 of a counterpart 30, especially a cardan head, arranged in this cardan sleeve 29 and connected for movement to the cardan shaft 33. The cardan head engages, via dogs projecting in the radial direction, in slots 32 in the cardan sleeve 29. The cardan sleeve 29 is elastically deformable and provided with radially inward- directed projections 38 in its end region remote from the drive arrangement 6, 7 and facing the cardan shaft 33. A clear width 39 between these projections 38 is at least slightly smaller than the diameter 36 or an outer dimension of the counterpart 30. Each of the drive arrangements 6, 7 comprises a drive motor 23, 24. <IMAGE>
Patent AT-401747-B (AT)
Title: Panel element of solid wood and process for its production
IPC: B27D1/00
Filed: 1994-11-14
Granted: 1996-11-25
Abstract: In a process for the production of a panel element, such as a furniture coreboard, a panel or the like, with essentially vertical annual rings, forest-thinning round timber with sound knots is respectively divided into a thicker central plank 3, containing the core, and, if the thickness is suitable, thin side boards 4 flanking this thicker plank and having essentially horizontal annual rings 5 over its width, whereafter from this cut material there are cut out by cuts 7 parallel to the narrow sides only those strips 8 or 4a which have essentially horizontal annual rings 5 over their width, which strips are subsequently glued to form a matt of strips 10, whereupon this matt of strips 10 is divided into strips 12, which are placed one on top of the other and glued to form a beam 14 with annual rings running essentially in one direction. By making cuts perpendicularly with respect to the direction of the annual rings, panels 18 are cut from this beam 14, are glued to one another on the narrow sides and cut into blanks 22, which after a grinding operation are provided on at least one side directly with a fair covering 23. <IMAGE>
Patent CA-1042511-B (CA)
Title: Self-cleaning aperture tube for coulter study apparatus
Inventor: HOGG WALTER R
IPC: G01N15/12
Filed: 1978-02-01
Granted: 1978-11-14
Abstract: ABSTRACT     Improved apparatus for obtaining signals from particles passing through a scanning aperture without extraneous interference from other particles.  The apparatus is improved by providing a pump device interposed between the inlet and outlet chambers which operates to draw the particle suspension up through the outlet chamber and back into the inlet chamber.          The flow created by the pump is such as to ensure that all particles introduced into the aperture device are caught by the orifice of the outlet chamber so as to prevent the occurrence of extraneous signals.
Patent CA-1226832-B (CA)
Inventor: LADT CARROLL H
IPC: B65G67/06
Filed: 1987-02-23
Granted: 1987-09-15
Abstract: ABSTRACT     A load out chute system for controlling and directing the flow of relatively large quantities of bulky material, such as coal, is disclosed.  The chute system includes an upper chute defining an  upper flow path and a hydraulically operated sliding gate valve positioned above the upper chute for controlling the supply of material thereto.  A lower chute defines a lower flow path and is capable of pivotal movement from a horizontal stored position to an operative position wherein the upper and lower flow paths are aligned.  The lower chute is mounted by means of a triangular skirt pivotal secured to an overhead structure.  The triangular skirt includes an arcuate bottom plate enabling the lower chute to cover the upper chute discharge opening when the lower chute is being pivoted toward its horizontal stored position, thereby preventing material spillage from the upper chute.  A corresponding curved retainer plate is operative to cover the lower chute inlet opening during pivoting movement for preventing spillage.          A blade gate valve operated by hydraulic cylinders, is positioned at the bottom portion of the lower chute, the blade being operative to control material flow along the lower flow path.  By positioning the blade gate valve in proximity to the bottom discharge opening of the lower chute, precise topping off at the end of the loading cycle may be achieved and material spillage is minimized.  The topping off feature is particularly applicable in a leading and trailing two chute system disclosed for filling a moving open top box car where material flow through the trailing chute is controlled to top off the load.  Rapid pivotal movement of the lower chute is achieved with a power cylinder interconnected to the chute with a cable and pulley arrangement.          A power winch is also interconnected with the chute by the cable means and is capable of incrementally adjusting the lower flow path to ensure proper alignment with the upper flow path.
Patent CA-1244899-B (CA)
Inventor: ALEXANDROV NICOLAI
IPC: H01F41/02
Filed: 1988-01-14
Abstract: Un transformateur de distribution comportant au moins un circuit magnétique fermé en forme de tore creux constitué d'un ruban enroulé en acier ferromagnétique. Un circuit électrique est formé d'un enroulement primaire et d'un enroulement secondaire, chacun étant constitué d'un ou de plusieurs sous-ensembles en forme de galette double, ces sous-ensembles étant juxtaposés et moulés ensemble au moyen d'une matière isolante solide qui forme avec les enroulements qu'elle entoure et qu'elle infiltre, un cadre rigide isolé sur lequel se trouve enroulé le circuit magnétique en forme d'un ou de plusieurs tores. Le cadre rigide isolé constitué par les enroulements électriques et la matière aussi isolante de moulage renferme des tubes destinés à la circulation du fluide qui refroidi intérieurement le bloc des conducteurs électriques moulés ainsi que le circuit magnétique.
Patent DK-164482-B (DK)
Inventor: OLOFF HORST
IPC: A61K47/00
Filed: 1984-09-11
Abstract: A device for transdermal administration of active medicinal agents is based on the active medicinal agent dissolved to an extent of at least 50% in a nonflowable, physiologically acceptable gel, which latter is distributed in a microdisperse mode in a crosslinked silicone elastomer.
Patent DK-162366-B (DK)
Inventor: BOCKHACKER BERND
IPC: A01K1/015
Filed: 1987-08-24
Abstract: The invention relates to a slatted floor grate for livestock housing, consisting of an elongate profile produced from sheet metal, the metal profile being enamelled and the top of the bearing side being provided with an additional, rough and hence slip-proof acid-resistant layer of silicate enamel.
Patent DK-155692-B (DK)
Inventor: BARTHELMESS ULRICH
IPC: B02C17/16
Filed: 1985-10-16
Abstract: An agitating mill, particularly an agitating ball mill, comprising a housing having an inlet for material to be ground and for air, an outlet for fines and air, and at least one horizontal agitator shaft which is provided with agitating members. The outlet for fines and air has a large area and is provided in the top wall of the housing and extends throughout the length and width of the top wall of the housing. A plurality of agitator shafts are preferably provided which are juxtaposed and superposed.
Patent FI-65068-B (FI)
Inventor: STAEHLE HELMUT
IPC: C07D487/04
Filed: 1979-06-21
Granted: 1983-11-30
Abstract: Compounds of the formula   <IMAGE>   wherein R1, R2 and R3, which may be identical to or different from each other, are each hydrogen, fluorine, chlorine, bromine, methyl, methoxy or trifluoromethyl, provided that one of them is other than hydrogen; and R4 and R5, which may be identical to or different from each other, are each hydrogen or methyl; and non-toxic, pharmacologically acceptable acid addition salts thereof. The compounds as well as their salts are useful as bradycardiacs.
Patent FI-67809-B (FI)
Inventor: ARMSTRONG BO
IPC: B42F7/02
Filed: 1982-05-20
Granted: 1985-02-28
Abstract: A file, especially for paper or the like, for instance a magazine file (10), comprising a bottom (15) and side walls (11-14) and an opening opposite to the bottom, is designed so that its handling volume will be about half the normal volume. The magazine file (10) has at least one slit (16-19) extending from the free top edges of the side walls (11-14) and directed towards the bottom (15) and having such a width that it can receive a side wall. The slit is adapted to accommodate a side wall (31-34) of a second, similar file (30) when this is telescoped into said first file (10) with the opening (40) and the side walls (31-34) of said second file facing the opening (20) and side walls (11-14) of said second file (10) while being slightly displaced in parallel with the bottom (15, 35) plane.
Patent FI-74479-B (FI)
Inventor: LUEHMANN ERHARD
IPC: C08L1/08
Filed: 1982-10-05
Granted: 1987-10-30
Abstract: A viscous cellulose substance containing paste which is characterized by containing an alkoxylated plasticizer and a ratio of solid to the organic solvent phase of >/=1 and which can be used to prepare a lacquer consisting at most of 25% of an organic solvent.
Patent FI-73217-B (FI)
Inventor: VALLEE ERIC
IPC: C07D495/04
Filed: 1983-06-16
Granted: 1987-05-29
Abstract: This invention relates to a new thieno-pyridinone derivative of the formula:   <IMAGE>   and its pharmaceutically acceptable inorganic or organic acid addition salts. This invention relates also to a process for the preparation of said compound and to its therapeutic application as blood-platelet anti-aggregation agent and anti-thrombosis agent.
Patent FI-68731-B (FI)
Inventor: PAULUS HENRY P
IPC: C07K16/00
Filed: 1983-08-11
Granted: 1985-06-28
Abstract: A homogenous sample of identical bispecific antibody determinants, each determinant being composed of two L-H half-molecules linked by disulfide bonds, each L-H half-molecule being specific for a different antigenic determinant and including at least the F(ab') portion of a monoclonal IgG antibody. The bispecific antibody determinants are useful, e.g., in the formation of multilamellar assemblies and enzyme electrodes.
Patent FI-83351-B (FI)
Inventor: CHRISTENSEN JOHN MOSGAARD
IPC: D04H13/00
Filed: 1985-10-22
Granted: 1991-03-15
Abstract: PCT No. PCT/DK85/00017 Sec. 371 Date Oct. 28, 1985 Sec. 102(e) Date Oct. 28, 1985 PCT Filed Feb. 27, 1985 PCT Pub. No. WO85/03962 PCT Pub. Date Sep. 12, 1985.A desirable embossing of a fibrous web (6) as dry laid on a forming sheet (2) is effected by the web (6) in a still unglued condition passing a pair of embossing producing rollers (18, 20) carried on or by a pressure resistant support sheet (16) as also passing between the rollers. Problems as to web fractures are hereby widely eliminated.
Patent FI-87189-B (FI)
Inventor: DEVIC MICHEL
IPC: C07C46/00
Filed: 1985-10-28
Granted: 1992-08-31
Abstract: 1. Process for manufacturing 2-amylanthraquinone having a high content of the tert-isomer, by reaction of phthalic anhydride with tert-amylbenzene in the presence of a catalyst consisting of a mixture of hydrofluoric acid and boron trifluoride, followed by conversion of the amyl-orthobenzoylbenzoic acid obtained to 2-amylanthraquinone according to processes which are known per se, characterized in that the reaction of phthalic anhydride with tert-amylbenzene is performed at a temperature of between -60 C and -20 C in a two-phase liquid reaction medium formed as a result of the presence of a solvent for tert.amylbenzene which is inert and immiscible with the mixture of hydrofluoric acid and boron trifluoride under the conditions of the reaction.
Patent FI-86084-B (FI)
Inventor: AMBERG GUENTHER
IPC: D06L1/20
Filed: 1988-06-14
Granted: 1992-03-31
Abstract: A machine washing process with process-controlled dosing of water and detergent using a paste-form, phosphate-reduced or phosphate-free detergent which is substantially free from water, organic solvents and hydrotropic compounds. The paste comprises a phase liquid at a temperature below 10 DEG  C. and contains a nonionic surfactant selected from the group of polyglycolether compounds and of a solid phase dispersed therein in which the particles have a mean particle size of from 5 to 40  mu m and less than 5% of the particles have a particle size larger than 80  mu m, the solid phase comprising washing alkalis, sequestering compounds and other detergent constituents and, optionally, anionic surfactants. Under the control of a process-control computer, the paste is taken from a storage container, delivered to a mixer and diluted therein with water to at least such an extent that the formation of a gel phase is avoided. The aqueous mixture is fed to a washing machine and, unless this has already happened in the mixer, is diluted with more water to a concentration of 0.5 to 10 g/l, after which the washing process is started.
Patent FI-102615-B (FI)
Inventor: FATTORI MARIA
IPC: A01N63/27
Filed: 1992-04-16
Granted: 1999-01-15
Abstract: A method for the screening of potential antifungal agents comprises testing the inhibitory effect of the potential antifungal agent in two tests, a first test for inhibition of pathogen development in sterilised soil infested with mycelium of Pythium spp and a second test against for inhibition of disease development in a growing plant of a species susceptible to disease from damping-off disease complex in the presence of the said complex, identifying agents giving potential inhibitory effect in both tests compared with control and submitting same for further examination. Using this method four particularly useful microorganisms which display antifungal activity in a wide spectrum, shown in further testing and in field trials, of disease fungi have been provided. Methods of using such microorganisms and compositions and compositions containing same are also described.
Patent FI-96396-B (FI)
Inventor: JAERVENKYLAE JYRI
IPC: B29C48/09
Filed: 1992-12-28
Granted: 1996-03-15
Abstract: According to the invention, a core pipe (2) is formed, whose properties correspond to the requirements set by the fluid to be conducted. With a suitable coating method an outer protective layer (3) is formed around the core pipe (2) of such a plastic material, which properties meet the requirements set by the prevailing environment and/or pipelaying procedure. <IMAGE>