baber/WOPTO huggingface dataset:
Patent SG-11201809560Q-A (SG)
Title: Enhancer of zeste homolog 2 inhibitors
Inventor: KNIGHT STEVEN DAVID
IPC: C07D495/04
Filed: 2017-05-01
Abstract: WO 17 / 19 15 45 Al (12) INTERNATIONAL APPLICATION PUBLISHED UNDER THE PATENT COOPERATION TREATY (PCT) (19) World Intellectual Property Organization International Bureau (43) International Publication Date 09 November 2017 (09.11.2017) WIPO I PCT omit IIl mum 0 mu OH 100 oimIE (10) International Publication Number WO 2017/191545 Al (51) International Patent Classification: C07D 495/04 (2006.01) (21) International Application Number: (84) Designated States (unless otherwise indicated, for every kind of regional protection available): ARIPO (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW), Eurasian (AM, AZ, BY, KG, KZ, RU, TJ, TM), European (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR), OAPI (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG). Declarations under Rule 4.17: as to applicant's entitlement to apply for and be granted a patent (Rule 4.1 7(ii)) as to the applicant's entitlement to claim the priority of the earlier application (Rule 4.1 7(iii)) of inventorship (Rule 4.1 7(iv)) PCT/IB2017/052523 (22) International Filing Date: 01 May 2017 (01.05.2017) (25) Filing Language: English (26) Publication Language: English (30) Priority Data: 62/332,131 05 May 2016 (05.05.2016) US 62/359,904 08 July 2016 (08.07.2016) US 62/454,143 03 February 2017 (03.02.2017) US 62/482,964 07 April 2017 (07.04.2017) US (71) Applicant: GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED [GB/GB]; 980 Great West Road, Brentford Middlesex TW89GS (GB). (72) Inventors: KNIGHT, Steven David; 1250 South Col- legeville Road, Collegeville, Pennsylvania 19426 (US). LAFRANCE, III, Louis Vincent; 1250 South Collegeville Road, Collegeville, Pennsylvania 19426 (US). TIAN, Xin- rong; 1250 South Collegeville Road, Collegeville, Pennsyl- vania 19426 (US). (81) Designated States (unless otherwise indicated, for every kind of national protection available): AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DJ, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JP, KE, KG, KH, KN, KP, KR, KW, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW. Published: with international search report (Art. 21(3)) (54) Title: ENHANCER OF ZESTE HOMOLOG 2 INHIBITORS (57) : This invention relates to novel compounds according to Formula (I) which are inhibitors of Enhancer of Zeste Homolog 2 (EZH2), to pharmaceutical com- positions containing them, to processes for their preparation, and to their use in therapy for the treatment of cancers. R 2 L-. R3 (I)
Patent AT-396081-B (AT)
Inventor: AUZINGER JOHANN
IPC: B23Q1/48
Filed: 1991-02-12
Granted: 1993-05-25
Abstract: In order to greatly increase the disposal periods for troughs in production lines as well as the entire disposal capacity without increasing the cost and in order to also minimize production- and processing-line stoppage times related to disposal, a device having at least two U-shaped supports 1 is provided. All the tubes deposited in the trough can be lifted out of the trough at the same time with this device. The supports 1 are rotatably mounted at their holders 2, so that they can be slipped under the ends of tubes in the trough. In the top holding position of the supports 1, a loose bunch can be bunched together by an automatic bunching device before it is disposed of. <IMAGE>
Patent AT-391036-B (AT)
IPC: G11B33/04
Filed: 1986-03-13
Granted: 1990-08-10
Abstract: The device has a shelf (1), sloping from front to back, which can be swivelled about a swivel spindle (7) running transversely to the longitudinal axis of this shelf (1), the design being such that the swivel spindle (7) is accommodated in foot parts (8), that each foot part (8) bears a short swivel spindle (7), the free end face of which can be inserted into an aligned bore (14) of a bearing part and/or further foot part, and that neighbouring foot parts with in each case a separate short swivel spindle can be locked immoveably in the axial direction with respect to one another, in particular by means of positive locking elements (15). <IMAGE>
Patent AT-407780-B (AT)
IPC: F16H41/02
Filed: 1986-03-20
Granted: 2001-06-25
Abstract: A multistage turbine is, via an engine, acted on by a high-pressure oil flow by means of a connected oil pump. The admission is carried out by an electromagnet and dynamo as a function of the travelling speed of a motor vehicle. A gearshift lever can be used for the reverse gear and can, if appropriate, be replaced by an electromagnet. In conjunction with the shift lever scale, the gearshift lever also has the function of shifting gear only by means of the shift lever itself, or that is to say it affords the opportunity of prebraking or fully braking the vehicle by appropriate acceleration in the reverse gear position. <IMAGE>
Patent AT-396120-B (AT)
IPC: C23C4/06
Filed: 1988-04-13
Granted: 1993-06-25
Abstract: For the provision of durable and easily legible inscriptions by jet spraying on steel ingots when they are at an elevated temperature, a nickel or iron metal powder having a largest particle dimension not in excess of 0.075 mm and a zirconium oxide powder or aluminum oxide powder having a largest particle dimension not in excess of 0.075 mm and used in an amount that is not in the excess of 10% by weight of the metal powder are jointly sprayed onto the surface of the steel ingots to form dots or lines thereon.
Patent HU-185691-B (HU)
Title: Process for preparing a new analgetic pharmaceutical composition
Inventor: CSILLI BERTALAN
IPC: A61N1/30
Filed: 1982-02-09
Abstract: A method of treating chronic pain is disclosed which comprises the step of topically administering to the skin of a human patient, 1 to 100  mu g/cm2 of body surface of a compound of the Formula (I) <IMAGE>  (I)  in which R is -CH3 or -CHO R1 is methoxy or amino; R2 is hydrogen, hydroxyl or acetoxy; R3 is hydrogen or ethyl; R4 and R5 together form a valency bond or an epoxy bridge, or R4 is hydroxy or ethyl; and R5 is hydrogen; or a pharmaceutically acceptable acid addition salt thereof, by iontophoresis.
Patent HU-183356-B (HU)
Title: Cutter holding device for turning polygon surfaces
Inventor: TAJNAFOEI JOZSEF
IPC: B23Q27/00
Filed: 1981-03-10
Abstract: The cutter-holder is also suitable for processing epicycloid, hypocycloid, ribbed and relieved polygonal surfaces. The advantageous feature of the cutter-holder according to the invention lies in that on a work piece of any size or weight polygonal surfaces of optional shape and number may be processed without the occurrence of detrimental dynamic forces or moments; processing may be performed with a high accuracy, it does not contain quickly abrading components; changing over to processing of surfaces of different size and shape can be easily performed; eccentricities can be adjusted quickly and without difficulties, ideal cutting conditions may be achieved. The most important characteristic of the cutter-holder according to the invention lies in that on the actuating camshaft there is a cutter-holder with adjustable eccentricity supported in bearings, furthermore it is provided with a second camshaft keeping said cutter-holder in a position being parallel with the adjusted position or with a structural part preventing turn-off; on one or more camshafts there are the eccentric journals having been displaced by 180` in relation to the journals of the cutter-holder; said eccentric journals are putting the balance-bridge into motion; at last, the cutter-holder is provided with a centralized resp. automatized organ for the simultaneous adjusting of the eccentricities of the eccentrics.
Patent YU-48281-B (YU)
Title: Legura na bazi nikla za centrifuge za staklena vlakna i postupak za termičku obradu izlivene centrifuge
Inventor: VASSEUR S
IPC: C22F1/10
Filed: 1992-03-30
Abstract: LEGURA NA BAZI NIKLA ZA CENTRIFUGE ZA STAKLENA VLAKNA I POSTUPAK ZA TERMIČKU OBRADU IZLIVENE CENTRIFUGE. Legura na bazi nikla za centrifuge za staklena vlakna, naznačena time, čiji sastav sadrži sledeće elemente u masenim procentima: Cr 27,5 - 29,5% W 6,5 - 7,8% C 0,69 - 0,73% Fe 7 - 10% pri čemu je ostatak u suštini nikl i predstavlja u svojoj kristalnoj strukturi karbide tipa M23C6 pri čemu je M hrom i/ili najmanje jedan "ekvivalentni" metal, karbidi M23 C6 i u suštini sekundarni. - Prijava sadrži još 2 nezavisna i 8 zavisnih zahteva.
Patent ZA-81473-B (ZA)
Title: 5-amino-tetayole derivatives of retinoic acids, their preparation and pharmaceutical formulations containg these derivatives
Inventor: NUERRENBACH A
IPC: A61P35/00
Filed: 1981-01-23
Abstract: 5-Amino-tetrazole derivatives of retinoic acids and their physiologically tolerated salts, processes for their preparation and pharmaceutical formulations which contain these derivatives and salts and which may, in particular, be used in the treatment of dermatoses.
Patent ZA-87309-B (ZA)
IPC: A61K31/35
Filed: 1987-01-16
Abstract: Racemic and chiral (2R,4R)-4-c-hydroxy-2-r-(substituted) chroman (and thiochroman)-4-acetic acids and their pharmaceutically acceptable salts useful in the treatment of diabetic complications, and intermediates therefor.
Patent ZA-95692-B (ZA)
Title: Neuroprotective compounds
Inventor: BUTLER TODD W
IPC: A61P39/02
Filed: 1995-01-30
Abstract: PCT No. PCT/IB94/00365 Sec. 371 Date Oct. 24, 1996 Sec. 102(e) Date Oct. 24, 1996 PCT Filed Nov. 21, 1994 PCT Pub. No. WO95/20587 PCT Pub. Date Aug. 3, 19953R*4S*3-[4-(4-fluorophenyl)-4-hydroxy-piperidin-1-yl]-chroman-4,7-diol, its enantiomers and pharmaceutically acceptable salts are effective oral agents for treating diseases and conditions susceptible to treatment by NMDA blocking drugs.
Patent AT-399160-B (AT)
Inventor: WILFINGER WERNER DR
IPC: C09C1/64
Filed: 1992-07-30
Granted: 1995-03-27
Abstract: The process described in AT Patent 386 000, for stabilising aluminium pigments by mixing them with optionally (partially) neutralised carboxyalkylenephosphoric acid esters and/or carboxyalkylenephosphonic acids and/or carboxyalkylenephosphinic acids is modified to the effect that the aluminium pigments stabilised in this way are mixed with an acid-curing binder combination comprising a resin containing hydroxyl groups and an amino resin, and leaving these mixtures to develop fully for from 2 to 24 hours at from 40 to 80 DEG C. This additional process step achieves a further improvement in the stability of aluminium pigments in aqueous or non-aqueous coating formulations.
Patent AT-406028-B (AT)
Title: Tool for machining workpieces
Inventor: KIRCHBERGER PETER DIPL ING
IPC: B23C5/08
Filed: 1995-09-27
Granted: 2000-01-25
Abstract: The invention relates to a tool, in particular a milling or rotary broaching tool, for machining workpieces having regions of round or rounded cross sections, e.g. crankshafts or camshafts. A tool 1 according to the invention is formed by a parent body 2 with a plane bearing surface 21 directed perpendicularly to its axis and with at least one cylindrical radial supporting surface 22 for the block cassettes, in which case the latter, for absorbing tangential forces, has at least one nose or projection 23 having a contact surface 231 cooperating with the parent body, and in each case at least one fastening element 5, with an oblique angle of the resulting direction of the angle of force relative to the perpendiculars of the cooperating surfaces, produces a surface pressure on the latter. <IMAGE>
Patent AT-402095-B (AT)
Title: Connecting piece, in particular having a threaded connection, for pressing onto the end of a pipe
Inventor: JAEGGI STEFAN
IPC: F16L13/14
Filed: 1995-09-27
Granted: 1997-01-27
Abstract: A connecting piece, in particular having a threaded connection 1 or on a fitting, comprises a projecting supporting sleeve 3 as well as a compression sleeve 7 arranged concentrically thereto, for pressing-on an unthreaded pipe 15. The compression sleeve 7 is held at a distance from the supporting sleeve 3 by means of an insulating ring 8. The pipe 15 is pushed into the annular gap 13 between the two sleeves 3, 7 and is compressed. Apertures 14 which make it possible to look into the annular gap 13 are provided in a cylindrical part 10 of the insulating ring 8. Since the insulating ring 8 is located in the region of the greatest insertion depth into the annular gap 13, the apertures 14 make it possible to check whether the pipe 15 has been pushed far enough into the annular gap 13 to produce a good compression joint. <IMAGE>
Patent AT-405813-B (AT)
Inventor: FILSEGGER HERMANN
IPC: B64C1/10
Filed: 1997-11-10
Granted: 1999-11-25
Abstract: A pressure frame, designed in particular for an aircraft, including a dome-shaped cover made of composite materials reinforced with fibers, preferably in one single piece, and cover reinforcing devices connected to the cover or produced integrally therewith. To reduce weight and cost while still fulfilling strain requirements, particularly of large aircraft, and to reduce the risk of destruction due to the cover being turned inside out towards the inside of the aircraft, the cover is of essentially uniform thickness and includes at least one cover reinforcing device which is mounted in the central area on the concave side of the cover. Advantageously, this cover reinforcing device in the central area is formed by a reinforcing structure oriented against the curvature of the cover, such as at truncated cone-shaped, mug-shaped or parabolic structure, with a cavity being arranged between the cover and the reinforcing structure.
Patent AT-387854-B (AT)
Title: Heat meter on the evaporation principle for determining the heat discharged by a heating surface
IPC: G01K17/02
Filed: 1985-08-28
Granted: 1989-03-28
Abstract: The invention relates to a heat meter on the evaporation principle for determining the heat discharged by a heating surface, provision being made for at least one ampoule 1 that can be or is filled with a measuring liquid and which has at least one surface section which is in surface contact with a heat bridge made of highly thermally conductive material. The invention is characterized in that the ampoule 1 is of non-round design, specifically substantially prism-shaped or with a semicircular cross section, at least one of the planar surfaces being in surface contact with the heat bridge. <IMAGE>
Patent AT-397025-B (AT)
Title: Process and apparatus for preparing a roasted soya snack product
IPC: A23L11/00
Filed: 1990-12-21
Granted: 1994-01-25
Abstract: To prepare a roasted soya snack product, the raw soya beans are allowed to swell in cold water, cooked until soft in salt water and then rapidly roasted at high temperature with constant turning. For the roasting, a drum 3 which is furnished with a double-wall drum casing is mounted so as to be able to rotate within a heat- insulated shell 1, the hot exhaust air of the burner 2 being passed through the drum 3 and the perforated base 7 of the same. <IMAGE>
Patent AT-384959-B (AT)
Title: Process for preparing communal waste
Inventor: LUGSCHEIDER WALTER DIPL ING DR
IPC: B03B9/06
Filed: 1985-12-20
Granted: 1988-02-10
Abstract: In order to prepare communal waste, the waste is first fed to a mill 1 after which, following first coarse screening on a coarse screen 2 and further screening on a dividing screen 4, it is led over hard material separators 5 and 6 and magnetic separators 7 and 9. The screen overflow from the first coarse screen 2 is likewise divided into two fractions, after magnetic separation 3, with the aid of a further coarse screen 16 with a larger mesh size. The fractions obtained are fed to wet preparation and, optionally, at least to some extent to a composting operation. A plurality of fine screens 8, 10 and 17 is provided in order to separate out adhesive granules and extremely fine granules and in this way to be able to work up separately fractions rich in heavy metals. As a result, the wet preparation permits building-material and coloured metal fractions to be obtained, and also separate fibrous raw materials and separate plastic fractions, non-ferrous metal fractions, waste fuel fractions and raw materials for hydrolysis. <IMAGE>
Patent DK-162065-B (DK)
Inventor: SVENGREN ANDERS GUSTAF
IPC: A21D8/02
Filed: 1985-04-12
Abstract: A process for preparing a rolled pastry product in which a sheet of pastry material advancing on a conveyor belt is cut and folded into discrete pieces of a predetermined size and then rolled. The cutting and folding operation is carried out by an oscillating knife positioned above the conveyor belt which has a cutting edge extending laterally across the width of the conveyor belt, and which immediately after contacting and cutting through the advancing pastry sheet by means of its cutting edge, ascends and rotates in a direction such that the motional vector of the cutting edge is counter to the conveying direction thereby causing the forward edge of the pastry sheet to be lifted up and folded over. The knife then descends and rotates in the reverse direction so that the cutting edge contacts and cuts through the advancing pastry sheet behind the folded portion to separate a folded piece from the remainder of the pastry sheet.
Patent DK-160393-B (DK)
Title: System for the manufacture of chocolate mass
Inventor: CHAVERON HENRI
IPC: A23G1/10
Filed: 1985-04-26
Abstract: Apparatus for preparing a chocolate paste in which the various ingredients comprising at least cocoa and powdered sugar are subject to operations of grinding to a predetermined degree of particle size, of fluidification by dispersion of the particles of sugar and of cocoa into a continuous fatty phase and of degasification for the removal of water and undesirable volatile compounds. At least part of the treatment is carried out in a conveyor with several screws and an arrangement for regulating the temperature of the entrained material. After preliminary grinding of the ingredients to obtain a refined paste having the desired degree of particle size in the screw conveyor, dry-conching of the refined paste is carried out and then the liquefaction of the paste is obtained by the incorporation of additives in accordance with the receipe.
Patent DK-150353-B (DK)
Title: Ceiling element
Inventor: FRIIS JESPER ACHTON
IPC: E04F/
Filed: 1983-11-11
Abstract: Ceiling element for hanging at the ends between supporting rails and including a surface (2) whose side edges (3) are bent upwards to form side flanges, between which insulation material in the form of mineral wool is positioned, and where the side flanges have a profile that is designed to hold together adjacent pieces. So that the adjacent elements in a ceiling are able to reinforce one another, without consequently making it impossible to remove any one element, and to achieve high resistance to smoke gasses travelling through the air in the event of a fire, the side flanges' free edge (4, 5) is bent to form a channel open on the bottom, in that the one edge (5) is bent inwards and the other (4) outwards, and approximately in the middle of the one flange a depression (6) running along the length of the side flange and a corresponding protrusion (7) on the other side flange.<IMAGE>
Patent DK-166269-B (DK)
Inventor: BARMENTLOO ADRIANUS
IPC: B65F3/20
Filed: 1988-10-26
Abstract: A container (2) for a refuse lorry is divided by means of at least one horizontal partition (3) into several compartments (4,5) lying above each other. The filling openings of the compartments (4,5) are disposed on the rear of the container (2). The container (2) is provided on the rear with a rear loader (6) having a filling opening (7) and a compacting mechanism (8). The rear loader (6) has a trough (21) which is divided in by means of at least one horizontal partition (22) into several compartments (23,24) lying above one another and corresponding to the compartments (4,5) of the container (2). The compartments (23,24) connect to the filling opening (7) via slide plates (25,26). With this container (2) different types of refuse separated from each other, can be deposited each in one of the compartments (4,5) of the container (2).
Patent FI-77051-B (FI)
Inventor: ZAGEFKA HANS-DIETER
IPC: B27K3/15
Filed: 1983-04-13
Granted: 1988-09-30
Abstract: 1. An aqueous composition for treating wood containing 1) a water-soluble or water-dispersible, oxidatively drying binder which has a double-bond content corresponding to an iodine value of at least 100 [g iodine/100 g] and is based on a 1,3-butadiene polymer optionally modified by isomerisation, partial cyclisation or partial hydrogenation, the polymer having a relative molecular weight (-Mn ) of 500 to 6000 and containing at least 70 mol % of units obtained by polymerisation of 1,3-butadiene and not more than 30 mol % of units obtained by polymerisation of one or more other copolymerisable 1,3-diolefins and alpha-monoolefins, 2) a water-insoluble organic wood preserving agent or mixture of agents and optionally also a watersoluble organic wood preserving agent or mixture of agents, and 3) optionally one or more additives conventional in the impregnating and coating industries, but excluding pore-closing additives, characterized in that 4) the binder satisfies the additional criterion that it is a polymer carrying amino groups but not quaternary ammonium groups and containing from more than 50 up to 600 mg-atom of titratable amine nitrogen per 110 g, and 5) the composition contains acid and has a pH of from 2 to 8, the acid strength and amount of acid (degree of neutralisation) on the one hand and the amount of amino groups on the other hand being selected so that the binder is water-soluble or water-dispersible.
Patent FI-77529-B (FI)
Inventor: OESTBO KARL
IPC: F28F21/08
Filed: 1985-04-25
Granted: 1988-11-30
Abstract: PCT No. PCT/SE84/00282 Sec. 371 Date Apr. 16, 1985 Sec. 102(e) Date Apr. 16, 1985 PCT Filed Aug. 22, 1984 PCT Pub. No. WO85/01101 PCT Pub. Date Mar. 14, 1985.In order to improve the transfer of heat within a heat exchanger one or more tubes are provided for a heat transporting medium, and are embedded by casting into a block of an aluminum alloy, or some other metal having high heat conducting capacity. The block is at its outward faces provided with surface-enlarging flanges, and is enclosed in a casing which defines a passage for a second heat transporting medium flowing around the block. A block can be prismatic or annular, and a number of blocks can be fitted within the same casing.
Patent FI-91958-B (FI)
Inventor: ADOLFSSON BENGT
IPC: B01F3/04
Filed: 1991-11-27
Granted: 1994-05-31
Abstract: PCT No. PCT/SE90/00371 Sec. 371 Date Nov. 27, 1991 Sec. 102(e) Date Nov. 27, 1991 PCT Filed May 30, 1990 PCT Pub. No. WO90/15011 PCT Pub. Date Dec. 13, 1990.In a method for simultaneously carbonating and cooling liquid carbon dioxide under high pressure which is introduced under the liquid surface and is allowed to expand and dissolve in the liquid. Carbon dioxide not dissolved in the liquid is re-introduced under the liquid surface through a compressor and a cooler. A device for carrying out the method includes a closed vessel (1), a liquid inlet (2) opening into the vessel, a carbon dioxide inlet (12) opening into the vessel (1) under the liquid surface, a discharge conduit (5) for carbonated vessel, and, leading from the vessel (1) above the liquid surface, a re-circulation conduit (6,3) for carbon dioxide not dissolved in the liquid, compressor (7) and a cooler (8) being arranged in the re-circulation conduit (6,3).