baber/WOPTO huggingface dataset:
Patent EP-1266898-A1 (EP)
Inventor: FUKUOKA KOICHIRO
IPC: C07D495/04
Filed: 2001-02-27
Abstract: The present invention provides a process for
producing an intermediate for thienopyrimidine derivatives
having the GnRH antagonistic activity at an industrial
large scale. 
     The process for production of the present invention
relates to a process for producing a compound represented
by the formula (III):
 
wherein respective symbols have the same meanings as those
described below, or a salt thereof, which comprises
subjecting a compound represented by the formula (I) :
 
wherein R 1  denotes hydrogen, nitro, halogen, phthalimido,
mono- or di-(alkylcarbonyl)amino or alkoxy, or a salt
thereof, to an acid halogenating reaction, which is
successively reacted with malonic acid ester and magnesium
alkoxide, treated with an acid, and reacted with sulfur
and a compound represented by the formula: NCCH 2 COOR 2 
[wherein R 2  denotes alkyl or aryl], or a salt thereof, in
the presence of primary amine. According to the process
of production of the present invention, thienopyrimidine
derivatives having the GnRH antagonistic activity can be
produced effectively and at an industrial large scale by a
high yield and simple method.
Patent EP-1267168-A1 (EP)
Inventor: TAJIMA HIDEJI
IPC: B01L3/00
Filed: 2001-03-15
Abstract: The present invention relates to the support of substances for detection, apparatus
for processing same, method of processing same, apparatus for making same, and
method of making same. The object of the present invention is to provide a reliable
and high quality technology that can perform a series of processes, consistently,
automatically and easily. A support of substances for detection of the present
invention is constructed so as to comprise a flexible base member formed to be slender
as thread, string or tape, a variety of substances for detection having predetermined
chemical structure thereof and being fixed side by side along the length of the base
member, and a supporting member for supporting the base member in a manner that
enables expansion, wherein a fixed location of each substance for detection corresponds
with the chemical structure thereof.
Patent EP-1277570-A1 (EP)
Inventor: MORIWAKI KEN
IPC: H01J29/89
Filed: 2001-03-19
Abstract: It is to provide a functional laminated film which
is useful for antireflection on the surface and which can
make the brightness of an image uniform, its production
process and a CRT having said film attached thereto. 
     A functional laminated film having an antireflection
layer, a substrate film, a colorant layer having a color
density distribution and an adhesive layer laminated. A
functional laminated film having an antireflection layer,
a substrate film and a colored adhesive layer having a
color density distribution laminated. A CRT having the
above film attached thereto.
Patent EP-1163780-A1 (EP)
Inventor: GUENTHER RAINER
IPC: H04M1/02
Filed: 2001-01-17
Abstract: The invention relates to a telephone connection box for an ISDN basic access. The telephone connection box comprises an electronic circuit of a network terminating device.
Patent EP-1267702-A1 (EP)
Title: Dispositif d'insertion pour endoscope
Inventor: BUTLER JOHN
IPC: A61B1/31
Filed: 2001-03-23
Abstract: La présente invention concerne un système de sonde comprenant un dispositif de guidage gonflable (10) et un coloscope (2). Le dispositif de guidage (10) comprend une gaine en matériau flexible retournée sur elle-même pour former un tube retournable présentant une partie de gonflage destinée à la connexion à un tube de gonflage (11). Une extrémité avant du dispositif de guidage (10) est fixé de façon non définitive au coloscope (2) durant l'insertion dans un colon. Après l'insertion, l'extrémité avant est détachée et le dispositif de guidage (10) est gonflé. Le coloscope (2) peut être avancé à travers le colon en étant espacé des parois du colon grâce à un mouvement de retournement du dispositif de guidage (10).
Patent EP-1279117-A1 (EP)
Inventor: BIORGE JAMES
IPC: G06Q20/00
Filed: 2001-03-08
Abstract: La présente invention concerne un dispositif portable (12) acheteur dans lequel est stockée une valeur, un dispositif de base (24) acheteur, et un dispositif (50) fournisseur acheteur. Une quantité d'achat est déduite du dispositif portable acheteur et envoyé au dispositif fournisseur acheteur. Le dispositif fournisseur acheteur génère et chiffre un fichier (122) de paiement et un fichier (120) de visualisation de paiement qui confirme l'existence du fichier de paiement. Le dispositif de base (64) vendeur transmet le fichier de visualisation de paiement et le fichier de paiement à un dispositif (102) fournisseur vendeur. Le dispositif fournisseur vendeur génère et chiffre un fichier (130) de produit et un fichier (128) de visualisation de produit qui confirme l'existence du fichier de produit. Le dispositif fournisseur acheteur et le dispositif fournisseur vendeur déchiffrent respectivement le fichier de visualisation de produit et le fichier de visualisation de paiement. Suite à l'approbation de l'acheteur et du vendeur, des clés d'utilisateur sont échangées afin de permettre le déchiffrement des fichiers de produit et de paiement.
Patent EP-1280486-A1 (EP)
Inventor: SANDERS STEVEN W
IPC: A61K9/16
Filed: 2001-04-24
Abstract: A pharmaceutical composition that minimises an adverse drug experience associated with oxybutynin therapy comprises oxybutynin, wherein the composition in use provides a plasma area under the curve (AUC) ratio of oxybutynin to an oxybutynin metabolite of from about 0.5:1 to about 5:1.
Patent EP-1293216-A1 (EP)
Inventor: TAKEDA YASUKATA
IPC: F02G3/00
Filed: 2001-05-17
Abstract: An ion generating device generates O 2   - (H 2 O)   n    (where  n  is a natural number) as
negative ions and H + (H 2 O)   m    (where  m  is a natural number) as positive ions, and discharges
those ions into the air so that airborne germs are killed through an oxidation reaction by
hydrogen peroxide H 2 O 2  or radical hydroxyl OH generated through as an active species a
chemical reaction between the negative and positive ions. Satisfactory sterilization is
achieved when the negative and positive ions are generated in such a way that the
concentrations of the negative and positive ions are both 10,000 ion/cc at a distance of 10 cm
from the point at which they are generated.
Patent EP-1300160-A1 (EP)
Inventor: TOMOHIRA YUSO
IPC: A61K31/4709
Filed: 2001-05-23
Abstract: Disclosed is a method for stabilizing a solid
pharmaceutical preparation containing a pharmacological
substance and sodium lauryl sulfate, the method comprising
incorporating into the preparation at least one member
selected from the group consisting of neutral salts, basic
salts and basic substances. The preparation containing
sodium lauryl sulfate prepared by the method of the
invention has superior performance, including high storage
stability, suppression of discoloration and deterioration,
and prevention of change in its properties, such as the
dissolution rate of pharmacological substance from the
preparation.
Patent EP-1283741-A1 (EP)
Inventor: VERTRIEST DANNY
IPC: B01D53/26
Filed: 2001-05-15
Abstract: The invention relates to a compressor unit comprising a compressor unit comprising compressor element (2), the outlet conduit (3) of which connects to an adsorption dryer (6) with a vessel (8) and a rotor (7) mounted therein. On each of the extremities of the vessel (8), two compartments (20, 21, 23, 24) are formed. The portion of the rotor (7) situated between one compartment (24) n he o extremity and a compartment (21) on the other extremity forms a drying chamber (9), whereas the portion of the rotor (7.) situated between the other compartments (20, 24) forms a regeneration chamber (10) and is situated in the outlet conduit (3) upstream of a cooler (4). Between the compartments (20, 21, 213, 24) on each extremity, a separation compartment (22, 25) is formed and means (30, 21) are provided to remove gas therefrom (22, 25).
Patent EP-1202484-A1 (EP)
Inventor: AIHARA KOICHI
IPC: H04B1/707
Filed: 2001-06-13
Abstract: A first-stage processing section 105 detects a
plurality of slot timings corresponding to a plurality
of correlation values equal to or greater than a threshold
value, a second-stage processing section 110 detects
scrambling code timing and a scrambling code group in
accordance with one of the slot timings, a third-stage
processing section 115 identifies a scrambling code in
accordance with the scrambling code timing, and a
controller 104 switches a switch 103 so that processing
by the second-stage processing section 110 and processing
by the third-stage processing section 115 are executed
for a plurality of slot timings each time processing by
the first-stage processing section 105 is executed once.
Patent EP-1284614-A1 (EP)
Inventor: BRETTERBAUER DIETER
IPC: A44C17/02
Filed: 2001-05-30
Abstract: The invention relates to a jewellery piece on which at least one decorative element, which can be a stone, a pearl or another piece of jewellery is movably mounted, whereby the decorative element in the jewellery piece runs in a pair of grooves facing each other, the cross-section of which matches the form of the decorative piece and which may optionally be arranged in guide rails.
Patent EP-1285528-A1 (EP)
Title: Tramage a operations multiples ayant des trames de lineature d'inclinaisons quelconques
Inventor: WADLE HEINRICH
IPC: H04N1/40
Filed: 2001-05-02
Abstract: L'invention concerne un procédé de tramage numérique à opérations multiples d'une image en demi-teinte ayant une trame (6) de linéature et d'inclinaison quelconques. Selon ce procédé, le tramage s'effectue par lecture de valeurs seuils et comparaison des valeurs seuils lues avec les valeurs de teintes de l'image en demi-teinte. A cet effet, on utilise des matrices de valeurs seuils dans lesquelles les valeurs seuils représentent au moins un point de trame d'une trame donnée (3), qui permet d'approcher la linéature et l'inclinaison de trame souhaitées. Pendant la lecture des valeurs seuils, on détermine une erreur entre les coordonnées de la trame souhaitée (6) et de la trame donnée (3), et l'erreur est compensée par une correction de l'adresse de lecture de la matrice de valeurs seuils dès que l'erreur dépasse une valeur limite donnée. On peut utiliser à la place des matrices de valeurs seuils des matrices de valeurs d'impression dans lesquelles sont mémorisées la répartition des valeurs d'impression à imprimer, cette répartition étant valable pour une valeur de nuance.
Patent EP-1308040-A1 (EP)
Inventor: BAZIN PASCAL
IPC: H04N7/16
Filed: 2001-06-25
Abstract: La présente invention concerne un réseau de télévision numérique interactive. Selon l'invention, le réseau comporte essentiellement un site diffuseur (1) connecté par un canal de diffusion (16, 10, 34) à au moins une station de client (4). Le site diffuseur (1) comporte principalement une centrale des régies (4) qui mobilisent des ressources (5) pour réaliser des projets (6) à l'aide de profils cibles (7) à destination d'un générateur ou transcodeur (11) qui interprète les programmes d'une application de télévision numérique interactive en un langage de bas niveau multi-plate-forme. Les stations de client comportent essentiellement un lecteur (26) des programmes qui exécutent chaque programme à l'aide d'une plateforme de télévision numérique (29), le programme exécuté ayant été transcodé en fonction de la plate-forme cible.
Patent EP-1236914-A1 (EP)
Title: Plain bearing
Inventor: KANAYAMA HIROSHI
IPC: C10M103/02
Filed: 2001-08-13
Abstract: An object of the present invention is to provide a sliding
bearing having an excellent initial conformability and seizure
resistance as well as desired durability and heat resistance
required particularly for high speed engine. 
     The present invention provides a sliding bearing having
a resin coating layer comprising a thermosetting resin being
soft and having a good elongation at high temperature and a solid
lubricant formed on a bearing alloy layer.
Patent EP-1422990-A1 (EP)
Inventor: LEGRAND EMMANUEL
IPC: B26B9/02
Filed: 2001-09-03
Abstract: The invention relates to a cutting wire (2) which is designed to trim or cut vegetation and which can be used on rotating head devices, such as brush cutters and edge trimmers.  The external surface of the cutting wire is provided with tooth-type (5) or similar formations along the length of said wire (2).  In the case of a wire having one or more longitudinal cutting edges (4), said tooth-type formations (5) are disposed on the cutting edge(s) along the length of each edge (4).  In this way, the sharpness of the wire (2) is improved.
Patent EP-1325244-A1 (EP)
Inventor: HULTEN JOHAN
IPC: F16D65/00
Filed: 2001-09-28
Abstract: L'invention concerne un dispositif de freinage comprenant une plaque arrière supportant une garniture de frein (14) présentant au moins une surface de contact (16), des bords latéraux (18) et des bords d'extrémité (19, 20). Pour empêcher un sifflement des freins, le coefficient de frottement de la garniture de frein (14) varie dans le sens longitudinal entre les deux bords d'extrémité (19, 20) de telle sorte qu'au moins une des parties de bord d'extrémité (19, 20) de la garniture de frein présente un coefficient de frottement inférieur à celui du reste de la garniture de frein.
Patent EP-1318991-A1 (EP)
Title: Benzoic acid derivatives and uses thereof
Inventor: KASTELIC TANIA
IPC: A61K31/365
Filed: 2001-09-21
Abstract: The present invention is provides benzoic acid derivatives and uses thereof. In accordance with one aspect there is provided a compound of formula (I): stereoisomers thereof, or pharmaceutically acceptable salts or hydrates thereof, or physiologically acceptable and hydrolysable esters thereof; wherein: R1 is H, OH, halogen, (C1-C4) alkyl, (C1-C4) alkenyl, (C1-C4) alkoxy, or (C1-C4)alkyl-COO-; R2 is H, OH, halogen, (C1-C4) alkyl, (C1-C4) alkenyl, (C1-C4)alkoxy, or (C1-C4) alkyl-COO-; r3 is H, OH, halogen, (C1-C4) alkyl, (C1-C4) alkenyl, (C1-C4)alkoxy, or (C1-C4) alkyl-COO-; R4 is H, OH, halogen, (C1-C4) alkyl, (C1-C4) alkenyl, (C1-C4)alkoxy, or (C1-C4) alkyl-COO-; R5 is H, OH, halogen, (C1-C4) alkyl, (C1-C4) alkenyl, (C1-C4)alkoxy, or (C1-C4) alkyl-COO-; Y is O or -NR', wherein R' is H or (C1-C4) alkyl; n is 0-8; R6 is a 5 to 8 membered lactone or lactam ring; R7 is H, (C1-C4) alkyl, (C1-C4) alkenyl, (C1-C4)alkoxy, phenyl or (C1-C4) alkyl-COO-, wherein the lactam or lactone ring optionally comprises one or more C=C double bonds and the lactam or lactone ring is optionally substituted with one or more (C1-C4)alkyl or (C1-C4) alkenyl groups.The compounds of the present invention are useful for the treatment or prevention of disorders with an etiology associated with or comprising excessive cytokine release. The compounds are also used in the treatment of cancer, inflammatory disorders and disorders associated with an increased stability of mRNA which has an mRNA instability sequence. The present invention further provides processes for preparing benzoic acid derivatives of Formula I.
Patent EP-1333983-A1 (EP)
Title: Marking device and extrusion system with a marking device of this type
Inventor: BERINGER ANDREAS
IPC: B41J2/175
Filed: 2001-10-23
Abstract: The invention relates to a marking device, comprising a pump (2), a marking liquid container (6) for holding a marking liquid (8) and a marking head (12). A first line (4) through which the pressurised air of the pump (2) can be pumped into the marking liquid container (6) is located between the pump (2) and said marking liquid container (6). A second line (10), through which the marking liquid (8) can be pumped from the marking liquid container (6) to the marking head (12) is also provided. A surveillance device (22, 24) for measuring the pressure and for comparing the pressure measurement with a predetermined limit pressure value is provided in said second line (10). Were a hole or similar to appear in the second line (10), the falling of the pressure measurement below the limit pressure value would be detected by the surveillance device (22, 24) and the marking liquid container (6) would be deaerated. The deaeration of the marking liquid container (6) causes to the pressure inside said marking liquid container (6) to decrease. This ensures that no more marking liquid (8), which would otherwise leak out through the hole, is pumped into the second line (10). The invention also relates to an extrusion system with a marking device of this type.
Patent EP-1352275-A1 (EP)
Inventor: LAUZON JOCELYN
IPC: G02B6/34
Filed: 2001-10-29
Abstract: L'invention concerne un dispositif de couplage optique comportant un substrat présentant au moins deux guides d'onde à canal (18, 20, 21). Les deux guides d'onde se situent côte à côte dans une région de couplage formée sur le substrat. Un changement périodique d'indice de réfraction (22) est apporté de façon permanente dans la région de couplage. Le changement d'indice de réfraction périodique présente en permanence une période Δ et permet la réalisation d'un couplage entre les guide d'onde lumineux dont la longueur d'onde de couplage correspond à : μ=Μ(θeff1 - θeff2), θeff1 et θeff2 représentant les valeurs moyennes de l'indice de réfraction des guides d'onde respectifs dans la région de couplage, et θeff1 étant différente de θeff2. Par ailleurs, on peut appliquer un champ électrique sur la région de couplage pour régler la longueur d'onde de couplage.
Patent EP-1332624-A1 (EP)
Inventor: BRUEKERS ALPHONS A M L
IPC: H04N19/467
Filed: 2001-09-21
Abstract: Disclosed are a method, device (100) and arrangement for inserting extra information in an input signal (111) in the acoustical or visual domain. A representation in the electrical domain is received, a watermark comprising the extra information is generated and a watermark signal (113) representing the watermark is output to the acoustical or visual. There it merges with the input signal (111). Any recording unit (114) which attempts to record the input signal (111) will automatically record the watermark signal (113) as well, so no unwatermarked specimens are made available. The device (100) can be realized as a computer program product, or as a small portable unit, which can be worn by a person to automatically watermark anything he says. The device (100) can be used to protect physical objects against unauthorized taking of photographs, by projecting a visual watermark signal towards the source.
Patent EP-1409763-A1 (EP)
Inventor: GREZES-BESSET CATHERINE
IPC: C23C14/54
Filed: 2001-11-08
Abstract: La présente invention est relative à un procédé et à un dispositif de dépôt de couches minces. Le domaine technique de l'invention est celui de la fabrication de dispositifs optiques à couches minces. Selon l'invention, un dispositif (27) de dépôt de couches minces (35, 36) sur plusieurs substrats (10, 11), comporte des moyens de production d'un faisceau lumineux (31, 31a, 31b, 32a) de contrôle de l'épaisseur optique des substrats.
Patent EP-1349632-A1 (EP)
Title: Mecanisme de valve pour systemes de goutte-a-goutte
Inventor: COLLINS GREGORY R
IPC: A61M1/34
Filed: 2001-12-07
Abstract: La présente invention concerne un procédé et un dispositif permettant de d'empêcher l'écoulement rétrograde d'un fluide, par exemple, de produits sanguins, dans une source de fluide de substitution stérile (50). Le dispositif décrit dans cette invention comprend un élément robinet-vanne à commande (110) placé sur une section du conduit (90) qui achemine le fluide de substitution stérile vers un circuit extra-corporel (30). Dans un mode de réalisation, la régulation de l'élément de valve (110) est fondé sur une unité de commande (120) à l'aide de pressions fluidiques qui sont détectées en amont et en aval de l'élément (110) par un capteur amont (121) et par une pression avale (122) respectivement. De préférence, l'élément (110) est ouvert uniquement lorsque la pression amont est supérieure à la pression avale; ce qui permet de garantir que le fluide de substitution s'écoule seulement dans un seul sens lorsque l'élément (110) obstrue complètement le conduit (90) dans une position fermée. De cette façon et grâce aux différences de pression, le sang ne contamine pas le fluide stérile lors de son acheminement à travers le conduit (90).
Patent EP-1231436-A1 (EP)
Title: Haushaltsgerät
Inventor: SCHMID DIETRICH DIPL-ING
IPC: F24C15/20
Filed: 2002-02-07
Abstract: Die Erfindung betrifft die Vermeidung von stärker anhaftenden Verunreinigungen, insbesondere von Fetten, an Haushaltsgeräten mit von Wrasen angeströmten beschichteten Teilen. Dazu ist vorgesehen, dass die Teile aus Polycarbonat mit einer Silikonhardcoatingbeschichtung versehen werden. Eine bevorzugte Anwendung betrifft Wrasenschirme (1), die tauchbeschichtet werden. Um zu verhindern, dass durch mechanische Spannungen die Schutzwirkung reduziert wird, sieht die Erfindung in ihrer Ausgestaltung vor, dass der beschichtete Wrasenschirm (1) schwimmend auf dem Trägerteil (2) der Esse (3) angeordnet wird. <IMAGE>
Patent EP-1237343-A1 (EP)
Inventor: GOURON FRANCK
IPC: H04L29/06
Filed: 2002-02-25
Abstract: The electronic unit interface mechanism has interface circuits (30)) and a second interface (20,22,24) to different circuit modules. There is a processing unit (10) and a memory. The processing unit only transfers the digital word programming assembly when a pass word furnished by the mechanism user is recognized.
Patent EP-1243587-A1 (EP)
Inventor: KUHN WALTER DR
IPC: C07B61/00
Filed: 2002-03-11
Abstract: The invention relates to a process for the preparation of 15-pentadecanolide by hydrogenating 15-pentadecenolide and to its use.
Patent EP-1348340-A1 (EP)
Inventor: BOURGUIGNON MICHEL
IPC: A23C19/076
Filed: 2002-03-28
Abstract: The present invention relates to a dairy product, which comprises ornamental
patterns mainly based on colour effects. The dairy product may comprise lateral
stripes that are preferably visible through a transparent pot of the dairy product.
Different lateral stripes of different colours are possible, and even a complete
coating of the dairy product.
Patent EP-1266900-A1 (EP)
Inventor: KAO WENDLING
IPC: C07D498/22
Filed: 1993-10-08
Abstract: The invention concerns a compound of the structure
 
wherein R 1  and R 2  are each, independently, hydrogen, 
-CONH-[(CR 3 R 4 ) m (-A-(CR 5 R 6 ) n ) p ] q -B;
 
R 3 , R 4 , R 5 , R 6 , R 9  and R 10  are each defined substitutents, and R 3-6  may each also
represent hydrogen, 
B is alkenyl of 2-7 carbon atoms, alkynyl of 2-7 carbon atoms, hydroxyalkyl of 1-6
carbon atoms, alkylthioalkyl of 2-12 carbon atoms, alkylaminoalkyl of 2-12
carbon atoms, dialkylaminoalkyl of 3-12 carbon atoms, -OR 7 , -SR 7 , -CN,
-COR 7 , -CONHR 7 , -OSO 3 R 7 , -NR 7 R 8 , -NHCOR 7 , -NHSO 2 R 7 , or Ar; 
A is -CH 2 -, -NR 7 -, -O-, -S-, -SO-, -PR 7 -, -NHCO-, -NHSO- or -P(O)(R 7 )-; 
Ar is naphthyl, pyridyl, quinolyl, isoquinolyl, quinoxalyl, thienyl, thionaphthyl, furyl,
benzofuryl, benzodioxyl, benzoxazolyl, benzoisoxazolyl, indolyl, thiazolyl,
isoxazolyl, pyrimidinyl, pyrazinyl, imidazolyl, benzopyranyl,
benz[b]thiophenolyl,  
benzimidazolyl, benzthiazolyl, benzodioxolyl, piperidinyl, morpholinyl,
piperazinyl, tetrahydrofuranyl, or pyrrolidinyl; wherein the Ar group may be
optionally mono-, di-, or tri- substituted with a group selected from alkyl of 1-6
carbon atoms, arylalkyl of 7-10 carbon atoms, alkoxy of 1-6 carbon atoms,
cyano, halo, hydroxy, nitro, carbalkoxy of 2-7 carbon atoms, trifluoromethyl,
amino, dialkylamino of 1-6 carbon atoms per alkyl group, dialkylaminoalkyl of
3-12 carbon atoms, hydroxyalkyl of 1-6 carbon atoms, alkoxyalkyl of 2-12
carbon atoms, alkylthio of 1-6 carbon atoms, -SO 3 H -PO 3 H, and -CO 2 H;
PO 3 H, and -CO 2 H;
 
is a nitrogen containing heterocycle that may be saturated, unsaturated,
or
partially unsaturated, and may be optionally mono-, di-, or tri- substituted with a
defined substituent, with the proviso that R 1  and R 2  are not both hydrogen; 
m=0-6; n=0-6; p=0-1; q=0-1; 
or a pharmaceutically acceptable salt thereof which is useful as an immunosuppressive,
antiinflammatory, antifungal, antiproliferative, and antitumor agent.