baber/WOPTO huggingface dataset:
Patent AU-5356986-A (AU)
Title: Teilchen aus euner hydrophoben oder schwerloslichen substanz und verfahren zur ihrer hydrophilisierung
Inventor: GERGELY THOMAS
IPC: A61K9/16
Filed: 1985-12-12
Abstract: The surface of micronized and hydrophilized powder particles of a hydrophobic or sparingly soluble substance is covered with a cohesive layer of not more than 0.1 part by weight of surfactant in not more than 10 parts by weight of a binder (based on 100 parts by weight of the substance). A sparingly soluble or insoluble antibiotic is converted to instant granules or instant tablets, while a hydrophobic, moderately soluble to readily soluble pharmaceutical substance, such as, for example, acetylsalicylic acid or paracetamol, is converted to effervescent granules or effervescent tablets. The particles are preferably applied to carbohydrate crystals by means of a binder. The preparation is carried out by a method in which a solution which contains at least one surfactant in an amount of 0.01 to 0.1% by weight, based on the weight of the particles to be hydrophilized, and a binder in an amount corresponding to 5 to 10 times the weight of the surfactant used is sucked through a bed of the particles under a pressure of less than 800, preferably less than 100, mbar.
Patent AU-5602280-A (AU)
Title: Processes
Inventor: OSTERMAYER FRANZ
IPC: C07C231/02
Filed: 1980-02-29
Abstract: Derivatives of 3-aminopropane-1,2-diol of the formula    <IMAGE>  (I) in which Ar represents optionally substituted aryl, _n represents the number 0 or 1, and _a represents alkylene having 2 to 5 carbon atoms, the nitrogen atom and the oxygen atom, or, if _n is zero, the phenyl radical, being separated from one another by at least two carbon atoms, and R1 and R2, independently of one another, each represents hydrogen or lower alkyl, or together they represent lower alkylene, oxa-lower alkylene, thia-lower alkylene, aza-lower alkylene or N-lower alkyl-aza-lower alkylene, and salts of such compounds, processes for their manufacture, medicaments containing the new compounds and their use for the treatment of Angina pectoris and cardiac arrhythmia, and as blood pressure-reducing agents, as well as for the treatment of reactive or endogenic states of depression.
Patent AU-5742799-A (AU)
Title: Carbon black, method for producing carbon black and use of the same
Inventor: VOGLER CONNY
IPC: C09C1/50
Filed: 1999-08-28
Abstract: The inventive carbon black is characterised by an STSA surface of between 20 and 180 m<2>/g, a 24M4-DBP-absorption of between 40 and 140 ml/100g, a specific BET surface of between 20 and 250 m<2>/g, in that it contains 0.01 to 20 wt % silicon in relation to its total weight and in that it has a ratio of tan delta 0/tan delta 60 greater than 3.37-0.0068•STSA. The inventive carbon black is produced by adding silicon-containing compounds are added and mixed with the of carbon black raw material during the oxidative pyrolysis of the same and optionally, using carbon black oil as the fuel. The inventive carbon black can be used as a filler in rubber mixtures, preferably for tyres.
Patent AU-5764186-A (AU)
Title: Refuse bin with compactor means
Inventor: MASSONNET HENRY
IPC: B65F1/14
Filed: 1986-05-21
Abstract: This invention relates to improvements in refuse bins incorporating compacting means for domestic use, wherein the compacting plate comprises two upwardly oriented tabs which are placed in housings in the lid to be slidably associated with a control member. Catches facing opposite each other and borne by said tabs come into slides in the control member embedded in a groove in the lid. In this way, by subjecting the control member to a translation, it may, at the end of a stroke, be pivoted with respect to the catches in order to orient it vertically with a view to vertically actuating the compacting plate.
Patent AU-5800900-A (AU)
Title: Medicament for treatment of neuropathies
Inventor: LAREIDA JURG
IPC: A61K31/519
Filed: 2000-07-27
Abstract: Compounds of formula (I) in which R<SUP>1</SUP>=C<SUB>1-6 </SUB>alkyl, optionally halosubstituted; R<SUP>2</SUP>=H, C<SUB>1-4 </SUB>alkyl, optionally halosubstituted or replaced by halogen; R<SUP>3</SUP>=C<SUB>2-4 </SUB>alkyl, optionally halosubstituted; R<SUP>4</SUP>=SO<SUB>2</SUB>NR<SUP>5</SUP>R<SUP>6</SUP>, CO<SUB>2</SUB>R<SUP>7 </SUP>or halogen, C<SUB>2-4 </SUB>alkenyl; optionally substituted with NR<SUP>5</SUP>R<SUP>6</SUP>, SONR<SUP>5</SUP>R<SUP>6</SUP>, CONR<SUP>5</SUP>R<SUP>6</SUP>, CO<SUP>2</SUP>R<SUP>7 </SUP>or halogen, C<SUB>2-4 </SUB>alkanoyl, optionally substituted with NR<SUP>5</SUP>R<SUP>6</SUP>, SONR<SUP>5</SUP>R<SUP>6</SUP>, CONR<SUP>5</SUP>R<SUP>6</SUP>, CO<SUB>2</SUB>R<SUP>7 </SUP>or halogen; R<SUP>5 </SUP>and R<SUP>6</SUP>=independently H or C<SUP>1-4 </SUP>alkyl, or, together with the N atom to which they are attached, a pyrrolidino, piperidino, morpholino, 4-(NR<SUP>8</SUP>)-1-piperazinyl or 1-imidazolyl ring optionally substituted with one or two C<SUB>1-4 </SUB>alkyl groups; R<SUP>7</SUP>=H, C<SUP>1-4 </SUP>alkyl, optionally fluorosubstituted, and R<SUP>8</SUP>=H,C<SUP>1-3 </SUP>alkyl or hydroxyalkyl with 1-4 C atoms, or the pharmaceutically acceptable salts thereof are useful for the chemotherapeutic treatment of neuropathies.
Patent AU-5875898-A (AU)
Title: Horizontal moving and stirred bed reactor
Inventor: ROY CHRISTIAN
IPC: C10B7/06
Filed: 1998-01-30
Abstract: Provided is a reactor having: 1 a housing inlet means for admitting therein a particulate material to be heat treated and an outlet means for discharging the heat treated material, 2 at least one tray disposed horizontally inside the housing between the inlet and outlet means and having a support surface for supporting a bed of the particulate material, 3 a heating means for heating the bed of particulate material on the support surface, and 4 a conveyor system for moving the bed of particulate material while being heated along a predetermined direction on the support surface. The conveyor system includes a plurality of horizontally spaced-apart rake members extending across the support surface transversely of the predetermined direction and each having a plurality of spaced apart fingers in sliding contact with the support surface, and means for moving the rake members to displace with the finger the particulate material along the predetermined direction, the fingers of any one of the rake members being misaligned with the fingers of any other one of the rake members and being displaced relative to one another such the at the fingers rake across substantially the entire support surface of the tray and constantly stir the particulate material which displacing same, thereby constantly exposing the fresh surfaces of the particulate material to heat and increasing heat transfer in the bed.
Patent AU-5992199-A (AU)
Title: Tool component
Inventor: FRIES ROBERT
IPC: B23B27/14
Filed: 1999-10-08
Abstract: A tool component comprising an abrasive element presenting a cutting edge or point and a thermally conductive element having a thermal conductivity greater than the thermal conductivity of the abrasive element, wherein the thermally conductive element is in thermal contact with the abrasive element so as to conduct heat generated at the cutting edge or point away from such cutting edge or point. The thermally conductive element may be bonded to a substrate. The abrasive element may be PCBN and the thermally conductive element may be either CVD diamond or PCD or else the abrasive element may be PCD and the thermally conductive element may be CVD diamond.
Patent AU-6012201-A (AU)
Title: Supragingival powder spraying
Inventor: FLEMMIG THOMAS
IPC: A61K8/00
Filed: 2001-03-15
Abstract: Fine-grained powders or powder mixtures can be used to provide for spray cleaning of supragingival tooth surfaces. The abrasion of the tooth surface by the spraying of powder does not exceed 0.15 mm<SUP>3 </SUP>in relation to a tooth surface of 10 mm<SUP>2 </SUP>during a spray period lasting 2 minutes at a pressure of 4 bars and a distance of no more than 2.5 mm between the tooth surface and nozzle of the spray jet.
Patent AU-6055996-A (AU)
Title: Multiple data stream searching method and apparatus
Inventor: TSUKAGOSHI IKUO
IPC: H04N21/488
Filed: 1996-07-17
Abstract: Multiple data stream searching is achieved by encoding a video broadcast into multiple types of data streams including video, audio and subtitle data. Addresses are generated for each of the data streams pointing to a position of the data stream to be stored on a record medium. These addresses are stored in areas of the record medium reserved by type of data stream Such that location of any event represented by data in a data stream can be achieved by locating the data streams at the same type as that of the data to be located. A computer-readable memory directs a computer to store these addresses and to decode data streams at these addresses which correspond to the type of data stream to be searched. The data streams which are of the type to be searched are decoded and the event to be searched is found in these decoded data streams. <IMAGE>
Patent AU-6083100-A (AU)
Title: Bag style container with bullet resistant deployable panels
Inventor: NORRIS GAIL
IPC: B65D33/00
Filed: 2000-07-10
Abstract: A combination container for transporting articles which can concurrently be used as a ballistic shield from high speed projectiles such as bullets and/or shrapnel. The container, which can be a backpack, purse, computer carrying case, or similar bag style device, features a forward wall and a rear wall each having forming a compartment therebetween and at least one ballistic shield, attachable to one or both of the forward wall and said rear wall. Upper flaps and lower flaps attached to the bag afford deployable additional protection from attached ballistic shields. A handle provides a means for elevating the deployed elongated flaps and attached bag in front of the user to provide a large area of protection from such high speed projectiles.
Patent AU-6290400-A (AU)
Title: Use of nitriles as polar aprotic solvents
Inventor: LAURAIN NATHALIE
IPC: C07C205/12
Filed: 2000-06-30
Abstract: The invention concerns the use of aliphatic nitriles with relatively high molecular weight, as polar aprotic solvents, in particular in nucleophilic substitution reactions of the aromatic type. Said nitriles have a molecular mass more 79, preferably more than 90. The invention is useful for synthesis of fluorinated aromatic compounds.
Patent AU-6302694-A (AU)
Title: Lysosomal enzyme-cleavable antitumor drug conjugates
Inventor: FIRESTONE RAYMOND ARMAND
IPC: A61K47/48
Filed: 1994-05-12
Abstract: The present invention relates to drug-ligand conjugates wherein the drug is linked to the ligand through a protein peptide linker and a connector, a process for the preparation of said conjugates, method of controlling the growth of undesirable cells, pharmaceutical compositions, and intermediates thereof.
Patent AU-6403099-A (AU)
Title: Fuel injector with direct needle valve control
Inventor: LEI NING
IPC: F02M45/00
Filed: 1999-09-28
Abstract: A hydraulically-actuated unit fuel injector of the intensifier type is provided with two independently operable active control valves. A selectively actuable fuel pressure control valve is disposed on the hydraulic actuation fluid side to control the fuel pressure actuation process and provide a window of injection opportunity wherein the fuel pressure is maintained at high pressure. A selectively actuable timing control valve is disposed on the high pressure fuel side to provide precise control of injection timing events and duration, such as start of injection, end of injection, timing of interruption and duration of interruption, which all may occur during a single injection event within the window of opportunity. Both control valves are independently controlled to prevent reverse motion of the intensifier piston and plunger during dwell or interruption of injection while maintaining the full injection pressure. Dwell or interruption is controlled by using the timing control valve to port fuel under pressure to a fuel injector needle valve surface to generate a force on the fuel injector needle valve surface acting to close the fuel injector needle valve. Methods of defining a fuel injection event fuel injector having a fuel pressure intensifier, includes the steps of (a) preparing fuel pressure with a fuel injection pressure control valve, and (b) controlling the timing of a fuel injection event with a fuel injection timing control valve, the fuel pressure preparation and the timing of the fuel inject event being independently controllable. Preferably, full intensified fuel pressure is made available to the injector throughout a single injection event which may include a pilot injection, a main injection, a rate-shaped injection, and dwell periods wherein no injection occurs. Various methods of operating the fuel injector to provide various functions during a single injection event are also disclosed.
Patent AU-6480700-A (AU)
Title: Fungicidal compounds having a fluorovinyl- or fluoropropenyl-oxyphenyloxime moiety and process for the preparation thereof
Inventor: KIM BUM TAE
IPC: C07D317/54
Filed: 2000-08-16
Abstract: A fungicidal compound of formula (I) having a fluorovinye- or fluoropropenyl-oxyphenyloxime moiety and stereoisomers thereof are useful for protecting crops from fungal diseases: wherein, X is CH or N; Y is O or NH; R1 is hydrogen, C1-4 alkyl, or halogen-substituted C1-4 alkyl, R2 is a phenyl group optionally carrying one or more substituents selected from the group consisting of C1-4 alkyl, C1-4 alkoxy, methylenedioxy and halogen; or a naphthyl group; andR3 is hydrogen or CF3.
Patent AU-6482899-A (AU)
Title: Mixer-faucet cartridge with tangential spring
Inventor: MAGOCSI TAMAS
IPC: F16K11/078
Filed: 1999-10-25
Abstract: The present invention relates to cartridge for a mixer faucet mainly intended for mixing hot and cold water, wherein said cartridge comprises a housing (3) as well as two superimposed plates, i.e. an inlet plate (6) and a control plate (5), forming together a flat seal for controlling the mixing ratio and the volume of the flowing liquids. The inlet plate (6) is attached in the cartridge housing (3) while the control plate (5) is capable of sliding movement and rotation on the inlet plate (6). A lever support (2) is further provided at least partially in the cartridge housing (3), wherein said support is capable of rotation about he axis of the cartridge housing (3). A displacement lever (1) capable of rotation globally about the control rod (7) is mounted in the lever support (2). At least one elastic member (12) is provided or formed in the gap between the lever support (2) and the housing (3) and co-operates mechanically with said lever support (2) or housing (3). An actuation member (403) or an insert (13) or another elastic member is provided or formed from the housing (3) or the lever support (2) on the portion which is not connected to the elastic member (12) so that the stroke of said elastic member (12) comprises at least partially a covering member according to the rotation of the lever support (2).
Patent AU-6508994-A (AU)
Title: Chiral synthesis of tertiary alcohols with a hydrolase
Inventor: BLACKER ANDREW JOHN
IPC: C07D249/10
Filed: 1994-04-15
Abstract: PCT No. PCT/GB94/00793 Sec. 371 Date Dec. 11, 1995 Sec. 102(e) Date Dec. 11, 1995 PCT Filed Apr. 15, 1994 PCT Pub. No. WO94/24305 PCT Pub. Date Oct. 27, 1994Method of preparing an optically active compound of formula, wherein R and R1 are independently alkyl, alkenyl, alkynyl, alkoxy, alkoxyalkyl, cycloalkyl, aryl, aralkyl, a heterocyclic group or a C1-C4 alkyl-heterocycle, each being optionally substituted, procided that R and R1 are not identical and * is an optically active chiral center, from the corresponding racemic ester or diol by treating with a hydrolase enzyme. In particular, racemic 2-(2,4-difluorophenyl)-3-(1H-1,2,4-triazol-1-yl)propan-1,2 diol, an intermediate in fluconazole synthesis, is resolved using porcine pancreatic lipase or lipase from Chromobacterium viscosum.
Patent AU-6660796-A (AU)
Title: Synchronizing a telecommunications connection in a mobile communications system
Inventor: KINNUNEN KIMMO
IPC: H04B7/26
Filed: 1996-08-13
Abstract: PCT No. PCT/FI96/00437 Sec. 371 Date Apr. 14, 1997 Sec. 102(e) Date Apr. 14, 1997 PCT Filed Aug. 13, 1996 PCT Pub. No. WO97/07604 PCT Pub. Date Feb. 27, 1997A method for synchronizing a telecommunications connection in a mobile communications system including a database, at least one base station communicating with mobile stations on system channels which include control channels and traffic channels. Mobile stations communicate with other mobile stations using the base station and the system channels or communicate directly using a direct mode channel. Time slots and frame structures of the system channels are synchronized with time slots and frame structures of the direct mode channels.
Patent AU-6760694-A (AU)
Title: Compounds for reversing drug resistance
Inventor: SARKADI BALAZS
IPC: C07K5/02
Filed: 1994-05-12
Abstract: The invention features novel peptide derivatives called Reversins, and provides for their use in a method of reducing the activity of the multi-drug transporter protein MDR1 in order to overcome multidrug resistance in a mammal. The peptide derivatives are of the formula (I) X1n-X2-X3(X4)n-X5, wherein n is 0 or 1, and each n is the same or different; X1 is BOC, BOC-Asu, Z-Asu, benzyloxycarbonyl, Glu(OBzl)-OBzl, Trp-OMe, Trp-Phe-OMe, Phe-Trp-OMe, Phe-Phe-OtBu, Trp-Trp-OtBu, indoloacetyl, benzoyl, an alkylanine of 1-4 carbons, dibenzylamide, tryptamide, 1-amino-adamantine, aminomethylcyclohexane, indoline, phenylethylamide or dicyclohexylamide; X2 is Glu(OBzl), Asp(OBzl), succinyl, O,O-dibenzoyltartaroyl, diphenoyl, muconyl, Thx, Cpa, Asu, Nal, Pen, Phg, Dbt, Lys(BOC), Lys(Z), Cys(Bzl), Thr(Bzl), Glu(OtBu), tert.-Leu, Leu, Nle, Pro, Phe, Tyr(Bzl), or Ser(Bal); X3 is Asp, Asu, Lys, Glu, Trp, Thx, Cpa, Nal, Pen, Phg, Dbt, Glu(OtBu), tert.-Leu, Leu, Nle, Pro, Tyr, Phe, or Tyr(Bzl); X4 is BOC-Glu(OBzl), Glu(OBzl), Asu, OBzl, Bzl, BOC, BOC-Lys(BOC), Z-Glu(OtBu), Asp(OBzl), Asp(OBz)-OBzl, benzyloxycarbonyl, O-(cyclo-hexyl), fluorenylmethyl ester, Glu(OtBu), Glu(OtBu)-OBzl, 1-amino-adamantine, aminomethylcyclohexane, indoline, phenylethylarnide, or dicyclohexylamide; and X5 is OMe, OBzl, OtBu, Phe-OMe, -O-(cyclohexyl), Trp-OMe, (chlorophenyl)-isobutylamide, fluorenylmethyl ester, ONp, 1-aminoadamantane, aminomethylcyclohexane, indoline, phenylethylamide, or dicyclohexylamide.
Patent AU-6916487-A (AU)
Title: Azolyl-ketone derivatives
Inventor: ELBE HANS-LUDWIG
IPC: C07D/
Filed: 1987-02-11
Abstract: 1. Substituted di- or triazolylalkyl-carbinols of the general formula   see diagramm : EP0120276,P20,F1   in which A represents a nitrogen atom or the CH group ; B represents a nitrogen atom or the CH group ; X represents hydrogen and straight-chain or branched alkyl with 1 to 6 carbon atoms ; Y represents straight-chain or branched alkyl with 1 to 6 carbon atoms ; and, if X represents hydrogen, also straight-chain or branched alkenyl and alkinyl with in each case 3 to 6 carbon atoms and benzyl which is optionally mono- to trisubstituted in the phenyl part by identical or different substituents, substituents which may mentioned being : halogen, alkyl with 1 to 4 carbon atoms, alkoxy and alkylthio with in each case 1 to 4 carbon atoms, halogenoalkyl, halogenoalkoxy and halogenoalkylthio with in each case 1 to 2 carbon and 1 to 5 identical or different halogen atoms, such as preferably fluorine and chlorine atoms, nitro and cyano ; R represents phenyl which is optionally mono- to tri-substituted by identical or different substituents, preferred substituents which may be mentioned being : halogen, alkyl with 1 to 4 carbon atoms, alkoxy and alkylthio with in each case 1 to 4 carbon atoms, halogenoalkyl, halogenoalkoxy and halogenoalkylthio with in each case 1 to 2 carbon and 1 to 5 identical or different halogen atoms, such as preferably fluorine and chlorine atoms, nitro, cyano, hydroxyl, hydroxycarbonyl with 1 to 4 carbon atoms in the alkyl part, hydroximinoalkyl with 1 to 4 carbon atoms, alkoximinoalkyl with 1 to 4 carbon atoms in each alkyl part, and phenyl, phenoxy, benzyl and benzyloxy, each of which is optionally substituted by halogen and/or alkyl with 1 to 2 carbon atoms ; R furthermore preferably represents the grouping   see diagramm : EP0120276,P20,F2   wherein Alk**1 represents straight-chain or branched alkyl with 1 to 4 carbon atoms ; Alk**2 represents straight-chain or branched alkyl with 1 to 4 carbon atoms ; Alk**1 and Alk**2, together with the carbon atom to which they are bonded, represent a 3- to 7-centered cycloaliphatic ring ; and R**1 represents, straight-chain or branched alkyl with 1 to 6 carbon atoms, alkenyl with 2 to 4 carbon atoms and phenyl, phenylalkyl with 1 to 4 carbon atoms in the alkyl part, phenoxy, phenylthio, phenoxyalkyl with 1 to 4 carbon atoms in the alkyl part, phenylthioalkyl with 1 to 4 carbon atoms in the alkyl part, benzyloxy and benzylthio, each of which is optionally mono- to trisubstituted in the phenyl part by identical or different substituents, preferred possible substituents being the phenyl substituents alreadly mentioned for R.
Patent AU-6975694-A (AU)
Title: Salmonella identification by the polymerase chain reaction
Inventor: OLSEN JOHN ELMERDAHL
IPC: C12Q1/689
Filed: 1994-06-17
Abstract: PCT No. PCT/GB94/01316 Sec. 371 Date Mar. 11, 1996 Sec. 102(e) Date Mar. 11, 1996 PCT Filed Jun. 17, 1994 PCT Pub. No. WO95/00664 PCT Pub. Date Jan. 5, 1995The invention provides nucleic acid molecules for the detection and identification of Salmonella species, methods for detecting one or more Salmonella serotpes using the nucleic acid molecules of the invention as probes or primers in DNA-based detection systems and kits for carrying out the invention.
Patent AU-7028998-A (AU)
Title: Retroviral vectors, method for the production and the use thereof for gene transfer in cd4-positive cells
Inventor: CICHUTEK KLAUS
IPC: C12N15/867
Filed: 1998-02-27
Abstract: The invention relates to the production and use of retroviral vectors for cell specific gene transfer, specially to a production method of retroviral vectors containing capsid particles of murine leukemia virus (MLV) and envelope proteins of human immunodeficiency vises (HIV) or simian immunodeficiency viruses (SIV). Said vectors can be used for gene transfer in selected cell types, specially in CD4-positive mammal cells.
Patent AU-7036991-A (AU)
Title: Three laser optical disk drive system
Inventor: GOLDSMITH PAUL
IPC: G11B7/13
Filed: 1990-12-12
Abstract: An erasable optical disk drive system is disclosed which utilizes an electron trapping media coated on the disk surface to store data in the form of light energy and which utilizes three laser beams, each having a wavelength range distinct from each other as well as distinct from the wavelength range of the emission produced by the impingement of the read laser onto the electron trapping media. Data is written onto the disk, which is contained in a light-tight contamination-free environment, using a visible light laser beam. Data is read from the disk and the disk is erased by using a near infrared light laser beam. The focus and tracking functions of the disk drive system are accomplished by using a laser beam having yet another range of wavelengths, which are greater than those of the visible light laser beam and those of the photon emission from the electron trapping optical memory media, but less than those of the read/erase laser.