Patent MY-133385-A (MY)
Title: Benzazoles: benzoxazoles, benzthiazole and benzimidazole derivatives
Inventor: MATHEWS CHRISTOPHER JOHN
IPC: A01N43/80
Filed: 1999-07-28
Abstract: A COMPOUND OF FORMULA (I):WHEREIN X IS 0 OR S; N IS 0 OR 1; Y IS 0, S OR NR 7; R I IS HYDROGEN, HALOGEN, CI-6 ALKYL, CI-6 HALOALKYL, CI-6 ALKOXY, CI-6 HALOALKOXY, CI-6 ALKYLTHIO, CI-6 HALOALKYLTHIO, C3-6 CYCLOALKYL, CI-6 ALKOXY(CI-6)ALKYL OR SF5; R2 IS HYDROGEN, HALOGEN, CI-6 ALKYL, CI-6 ALKOXY, CI-6 HALOALKOXY, CI-6 ALKYLTHIO, CI-6 HALOALKYLTHIO, CI-6 ALKYLSULFINYL, CI-6 HALOALKYLSULFINYL, CI-6 ALKYLSULFONYL, CI-6 HALOALKYL~LFONYL, CI-6 HALOALKYL, CYANO, NITRO, CHO, CH=NOR5, CI-6 ALKYLCARBONYL, CI-6 ALKOXYCARBONYL OR SF5; OR TOGETHER R1 AND R2 FONN A FIVE OR SIX MEMBERED SATURATED OR UNSATURATED CARBOCYCLIC RING, OPTIONALLY SUBSTITUTED BY ONE OR TWO CI-6 ALKYL GROUPS; R3 IS HYDROGEN, CI-6 ALKYL, CH2(CI-4 HALOALKYL), CI-6 CYANOALKYL, C3-6 ALKENYL, C3-6 ALKYNYL, CI-6 ALKOXY(CI-6)ALKYL, CI-6 ALKYLTHIO(CI-6)ALKYL, CI-6 ALKOXY(CI-6)ALKOXY(CI 6)ALKYL, CI-6 ALKYLCARBONYL, CI-6 ALKOXYCARBONYL, FONNYL, CI-6 ALKYLCARBONYL(CI-6)ALKYL, CI-6 ALKOXYCARBONYL( C 1-6)ALKY 1, C 1-6 ALKY LAMINOCARBONYL, DI( C 1-6)ALKY LAMINOCARBONY 1, OPTIONALLY SUBSTITUTED PHENOXYCARBONYL, OPTIONALLY SUBSTITUTED PHENYL(CI-4)ALKYL OR S(O)QR6; R4 IS HYDROGEN, HALOGEN, CYANO, CI-8 ALKYL, CI-6 HALOALKYL, CI-6 CYANOALKYL, C2-6 ALKENYL, C2-6 ALKYNYL, C3-7 CYCLOALKYL, C3-7 HALOCYCLOALKYL, C3-7 CYANOCYCLOALKYL, CI-3 ALKYL(C3-7)CYCLOALKYL, CI-3 ALKYL(C3-7)HALOCYCLOALKYL, C3-6 CYCLOALKYL(CI-6)ALKYL, C5-6 CYCLOALKENYL, CS-6 CYCLOALKENYL(CI-6)ALKYL, C2-6 HALOALKENYL, CI-6 CYANOALKENYL, CI-6 ALKOXY(CI-6)ALKYL, FORMYL, C1- 6 CARBOXYALKYL, CI-6 ALKYLCARBONYL(CI-6)AIKYL, CI-6 ALKOXYCARBONYL(CI-6)ALKYL, CI-6 ALKYLTHIO(C1- 6)ALKYL, CI-6 ALKYLSULFINYL(CI-6)ALKYL, CI-6 ALKYLSULFONYL(CI-6)ALKYL, AMINOCARBONYL(CI-6)ALKYL, CI-6 ALKYLAMINOCARBONYL(CI-6)ALKYL, DI(CI-6JALKYLAMINOCARBONYL(CI-6)ALKYL, CI-6 ALKOXYCARBONYL, CI-6 ALKYLCARBONYL, AMINOCARBONYL, CI-6 ALKYLAMINOCARBONYL, DI(C1- 6)ALKYLAMINOCARBONYL, OPTIONALLY SUBSTITUTED PHENYL, OPTIONALLY SUBSTITUTED.PHENYL(CI-4)ALKYL, OPTIONALLY SUBSTITUTED PHENYL(C2-4)ALKENYL, OPTIONALLY SUBSTITUTED HETEROARYL, OPTIONALLYSUBSTITUTED HETEROARYL(CI-4)ALKYL, OPTIONALLY SUBSTITUTED HETEROCYCLYL, OPTIONALLY SUBSTITUTED HETEROCYCLYL(CI-4)ALKYL, A GROUP OR8, A GROUP SH, A GROUP S(O)PR9, A GROUP NR10RII OR A GROUP C(R12)=NORI3; R'''' IS HYDROGEN, CI-6 ALKYL, OPTIONALLY SUBSTITUTED PHENYL OR OPTIONALLY SUBSTITUTED PHENYL(CI-4)ALKYL; R6 IS CI-6 ALKYL, CI-6 HALOALKYL OR OPTIONALLY SUBSTITUTED PHENYL;R7 IS HYDROGEN, CYANO, CI-8 ALKYL, CI-6 HALOALKYL, CI-6 CYANOALKYL, C2-6 ALKENYL, C2-6 ALKYNYL, C3-7 CYCLOALKYL, C2-6 HALOALKENYL, C3-6 CYCLOALKYL (CI-6)ALKYL, CI-6 ALKOXY(C''''-6)ALKYL, CI-6 ALKOXYCARBONYL, CI-6 ALKYLCARBONYL, CI-6 ALKYLARNINOCARBONYL, DI(C''''-6)ALKYLARNINOCARBONYL, OPTIONALLY SUBSTITUTED PHENYL OR OPTIONALLY SUBSTITUTED HETEROARYL; R8 IS HYDROGEN, CI-6 ALKYL, CI-6 HALOALKYL, C3-6 ALKENYL, CI-4 CYANOALKYL, CI-6 ALKOXYCARBONYL (CI-6)ALKYL, OPTIONALLY SUBSTITUTE~ PHENYL, OPTIONALLY SUBSTITUTED PHENYL(C''''-4)ALKYL, OPTIONALLY SUBSTITUTED HETEROARYL, N=C(CH3);; R9 IS CI-6 ALKYL, CI-6 HALOALKYL, C3-6 ALKENYL, CYANO, CI-4 CYANOALKYL, CI-6 ALKOXYCARBONYL(CI-6)ALKYL, OPTIONALLY SUBSTITUTED PHENYL, OPTIONALLY SUBSTITUTED PHENYL(CI- 4)ALKYL OR OPTIONALLY SUBSTITUTED HETEROARYL; RIO AND R II ARE, INDEPENDENTLY, HYDROGEN, CI-8 ALKYL, C3-7 CYCLOALKYL, C3-6 ALKENYL, C3-6 ALKYNYL, C2-6 HALOALKYL, CI-6 ALKOXY(CI-6)ALKYL, CI-6ALKOXYCARBONYL, OPTIONALLY SUBSTITUTED PHENOXYCARBONYL, FONNYL, CI-6 ALKYLCARBONYL, CI-6 ALKY1SO2'''' OPTIONALLY SUBSTITUTED PHENYLSO2 OR OPTIONALLY SUBSTITUTED PHENYL(CI-4)ALKYL; R 12 IS CI-3 ALKYL; R 13 IS CI-6 ALKYL, OPTIONALLY SUBSTITUTED PHENYL(C1_JALKYL; AND P AND Q ARE, INDEPENDENTLY, 0, 1 OR 2, PROCESSES FOR PREPARING THESE COMPOUNDS, COMPOSITIONS COMPRISING THEM, METHODS OF USING THEM TO COMBAT FUNGAL DISEASES AND METHODS OF USING THEM TO COMBAT OR CONTROL INSECT, ACARINE, MOLLUSC AND NEMATODE PESTS.