baber/WOPTO huggingface dataset:
Patent IL-74837-A0 (IL)
Title: 7-oxo 8-dimethylaminomethylene hexahydrobenzo(de)quinolines
IPC: A61P25/00
Filed: 1985-04-08
Abstract: 8-dimethylaminomethylene compounds of the formula <CHEM>  wherein R is H, benzyl, (C1-C3)alkyl or allyol; and R<4> and R<5> are independently H or (C1-C3)alkoxy; and  7-oxo-hexahydrobenzo[de]quinolines of the formula <CHEM>  wherein  R<7> is (C1-C3)alkyl, ally, or benzyl; R<4> and R<5> are independently (C1-C3)alkoxy, or H, with the limitation that when R<4> and R<5> are both (C1-C3)alkoxy, then R<7> can not be methyl; are intermediates useful in the preparation of 6-substituted hexahydroindazolo or hexahydroisoindolo isoquinolines, having dopamine agonist and dopamine antagonist activity.
Patent IL-76815-A0 (IL)
Title: Process and apparatus for joining protective plastic films to an extruded plastic sheet,with the aid of an auxiliary plastic film
IPC: B32B38/10
Filed: 1985-10-24
Abstract: A process and apparatus are described wherein a honeycombed sheet of plastic (13) is extruded from an extruding means (10) and at least one protective film of plastic is joined onto at least one of its surface layers, said protective film having a softening temperature lower than that for extruding the sheet.According to the invention the protective film (14), combined with the auxiliary film or support film (15), is layed onto the surface of the sheet (13) leaving the extruding means; then said sheet (13), protective film (14) and support film (15) are subjected to the calibrating and cooling stage; and lastly said support film (15) is separated from the sheet. The protective film has now been made an integral part of the sheet, (protected honeycombed sheet).
Patent IL-94654-A0 (IL)
Title: Apparatus for separating a light liquid from a liquid mixture
IPC: E03F5/16
Filed: 1990-06-06
Abstract: PCT No. PCT/DE90/00429 Sec. 371 Date Mar. 27, 1991 Sec. 102(e) Date Mar. 27, 1991 PCT Filed Jun. 5, 1990 PCT Pub. No. WO90/14874 PCT Pub. Date Dec. 13, 1990.The present invention is directed to a light-liquid separator with an inlet for a light liquid/heavy liquid mixture at least one separator chamber for the light liquid from the heavy liquid located behind the inlet, a heavy liquid outlet located behind the separator chamber, an overflow edge being located in front of the heavy liquid outlet, a light liquid outlet including a light liquid balance room, a dip tube extending from a point below the overflow edge of the separator chamber downwardly into the light liquid balance room, and a light liquid discharge tube extending from the light liquid balance room upwardly, as well as a light liquid reservoir with which the light liquid discharge tube is in communication.
Patent AU-PP109097-A0 (AU)
Title: Napthalene derivatives
IPC: A61K31/27
Filed: 1997-12-22
Abstract: A compound of formula (I), wherein R1 is carboxy or protected carboxy, R2 and R3 are each independently hydrogen, hydroxy, or protected hydroxy, R4 is hydrogen or halogen, R5 is aryl substituted with halogen, amino, hydroxy or protected hydroxy, R6 is aryl optionally substituted with halogen, amino, hydroxy or protected hydroxy, A1 and A2 are each independently lower alkylene, and (II) is (III), (IV), (V) or (VI) or its salt, process for preparing it, a pharmaceutical composition including it, and a use thereof.
Patent FI-20061017-A0 (FI)
Inventor: PEACOCK MARK
IPC: B66B/
Filed: 2006-11-17
Abstract: The method involves utilizing a temporary machine room (6) movable in an elevator shaft. The machine room of an elevator provided with the temporary machine room is dismounted and the elevator is converted into an elevator without machine room by placing a hoisting machine (4). The hoisting machine is placed into a mounting position in the elevator shaft by releasing the hoisting machine together with a traction sheave (30). An independent claim is also included for an apparatus for installing an elevator without machine room during a building construction.
Patent IL-112606-A0 (IL)
Title: Mercaptoacetylamido 1,3,4,5-tetrahydro- benzo Úc¾ azepin-3-one disulfide derivatives useful as inhibitors of enkephalinase and ace
IPC: A61K38/00
Filed: 1995-02-09
Abstract: The present invention relates to certain novel mercaptoacetylamido 1,3,4,5-tetrahydro-benzo[c]azepin-3-one disulfide derivatives of the formula   <IMAGE>   useful as inhibitors of enkephalinase and of ACE.
Patent IL-117306-A0 (IL)
Title: Process for the synthesis of hydrocarbon compounds which are fluorinated on a carbon of an alkyl chain
IPC: C07C317/10
Filed: 1996-02-28
Abstract: A process for the synthesis of fluorinated derivs. comprises a step in which a substrate is reacted with a cpd. comprising the association of a Bronsted base with a defined number (n) of HF species (n=3-20, pref. 15, and esp. 10). The substrate comprises at least one halo-carrying C of sp<3> hybridisation, attached to at least two halogens, of which at least one is a halogen of atomic number greater than F, bonded to at least one chalcogen.
Patent IL-124472-A0 (IL)
Title: Contraceptive process and kit for female mammals comprising a combination of gestagen and estrogen
IPC: A61P15/18
Filed: 1996-12-20
Abstract: The present invention relates to a female mammal contraceptive process consisting of the sequential administration for at least 28 days of (a) a gestagen in an ovulation-preventing dose for at least 28 days in combination with (b) a natural oestrogen for 5 to 10 days at the end of the sequential dosage of at least 28 days, and a contraception kit.
Patent IL-132336-A0 (IL)
Title: Method for charging the combustion unit of a coal-fuelled power station
IPC: F23J15/02
Filed: 1998-03-28
Abstract: The invention relates to a method for charging the combustion unit of a coal-fuelled power station in which the coal is fed into said combustion unit at least partially using a stream of flue gas. According to prior art, said flue gas stream consists of the recycled flue gas of the coal-fuelled power station. The aim of the invention is to provide another stream of flue gas. To this end, the flue gas stream of a waste incineration plant is used as a flue gas stream, said flue gas stream having already been treated to large extent to remove mercury and other heavy metals, flue ash and hydrochloric acid.
Patent IL-138792-A0 (IL)
Title: Method for preparing hydrazine hydrate
IPC: C01B21/16
Filed: 1999-05-06
Abstract: The invention concerns a method for making hydrazine hydrate which consists in hydrolyzing methyl ethyl ketone azine to obtain hydrazine hydrate and methyl ethyl ketone, characterised in that it consists in purging heterocyclic compounds of the pyrazoline family to prevent coloration of the hydrazine hydrate.
Patent IL-140276-A0 (IL)
Title: Processes to generate submicron particles of water-insoluble compounds
IPC: B01J3/00
Filed: 1999-06-18
Abstract: Submicron particles of water-insoluble compounds, particularly drugs, are prepared by simultaneously stabilizing microparticulate suspensions of same with surface modifier molecules by rapid expansion into an aqueous medium from a compressed solution of the compound and surface modifiers in a liquefied gas and optionally homogenizing the aqueous suspension thus formed with a high pressure homogenizer.
Patent IL-144412-A0 (IL)
Title: Fast dispersing dosage forms free of gelatin
IPC: A61K9/00
Filed: 2000-01-27
Abstract: The present invention relates to fast dispersing solid dosage forms that preferably dissolve in the oral cavity within sixty (60), more preferably within thirty (30), most preferably within ten (10) seconds. A novel feature of the solid dosage forms according to the invention reside in the fact that the composition is essentially free or absolutely free of mammalian gelatin. It has been discovered that the use of certain modified starches at concentrations from 20 to 90 % by weight of the solid dosage form prepares dosage forms that are mechanically and chemically stable and are able to deliver higher concentrations of an active ingredient than the heretofore utilized gelatin based fast dispersing solid dosage forms. Further, the solid dosage forms according to the invention are obtainable by removing a solvent, such as water, from a mixture comprising an active ingredient, a modified starch and a matrix forming agent via freeze drying.
Patent IL-145385-A0 (IL)
Title: Methods and compositions for treating leukemia
IPC: C07D277/74
Filed: 2000-03-13
Abstract: Compounds of general formula (I), wherein R1 is H or C1 to C3 alkyl; R2 is aryl or -(CH2)n-aryl and n is 1 to 4; R3 is H or CH3; and R4 is substituted or unsubstituted phenyl, pyridyl, thiophene, furan, indole, pyrrole, thiazole or imidazole are described, as well as methods for treating cell proliferative disorders and neoplastic disorders.
Patent IL-147263-A0 (IL)
Title: Method for decoding and retrieving a sound signal in an asynchronous transmission system
IPC: H04L12/64
Filed: 2000-06-22
Abstract: The invention concerns a method for decoding and retrieving a sound signal in an asynchronous transmission system which consists in detecting an backfilling overload in said buffer memory and/or a second memory in the input or the output of the decoding unit and comparing the backfilling rate to at least a threshold. The invention is characterised in that, depending on the value of the backfilling rate, it consists in using a detection of voice activity and in eliminating the frames considered as being non-active by said detection; carrying out a concatenation processing on two successive frames.
Patent IL-149158-A0 (IL)
Title: Tailored peptide synthetases, a method for their production and the use thereof
Inventor: MARAHIEL MOHAMED A
IPC: C12N9/00
Filed: 2000-10-18
Abstract: Novel tailor-made artificial non-ribosomal peptide synthetases (NRPSs) for non-ribosomal synthesis and/or modification of peptides of a predetermined length and composition and/or for modification of individual amino acids are described. The fusion of building units of said peptide synthetases in particular linker regions makes it possible to specifically prepare by means of “modular molecule construction kits” NRPSs which are capable of synthesizing peptides of a desired structure.
Patent IL-153469-A0 (IL)
Title: Electrochemical cell connector
IPC: G01N27/327
Filed: 2002-12-16
Abstract: The present invention relates to electrochemical cells including a connector which mates with a connection device to provide electrical connection to meter circuitry.
Patent IL-155702-A0 (IL)
Title: Piperazinylpyrazine compounds as agonist or antagonist of serotonin 5-ht2 receptor
IPC: A61P25/30
Filed: 2001-11-20
Abstract: A compound of the general formula (I), wherein R1, R2, X, Y and Z are as described in the specification.
Patent IL-163781-A0 (IL)
Title: Purine derivatives as kinase inhibitors
IPC: A61K31/55
Filed: 2003-03-04
Abstract: The present invention provides kinase inhibitors of Formula.
Patent IL-166822-A0 (IL)
Title: 6,7-dihydro-5h-pyrazoloÄ1,2-aÜpyrazol-1-ones whichcontrol inflammatory cytokines
IPC: A61P29/00
Filed: 2005-02-10
Abstract: The present invention relates to 2-(4-fluorophenyl)-3-(2-phenoxy-pyrimidin-4-yl)-6,7-dihydro-5H-pyrazolo-[1,2-a]pyrazol-1-one, including all enantiomeric and diasteriomeric forms and pharmaceutically acceptable salts thereof, having the formula: and pharmaceutical compositions thereof, and methods for controlling the level of one or more inflammation inducing cytokines selected from the group consisting of, interleukin-1 (IL-1), Tumor Necrosis Factor-alpha (TNF-alpha), interleukin-6 (IL-6), and interleukin-8 (IL-8), thereby controlling, mediating, or abating disease states affected by the level of extracellular inflammatory cytokines in humans.
Patent IL-183063-A0 (IL)
Title: Phenylpiperazine derivatives with a combination of partial dopamine d2 receptor agonism and serotonin reuptake inhibition
Filed: 2007-05-08
Abstract: The invention relates to a group of novel phenylpiperazine derivatives with a dual mode of action: serotonin reuptake inhibition and partial agonism on dopamine -D2 receptors. The invention also relates to the use of a compound disclosed herein for the manufacture of a medicament giving a beneficial effect. The compounds have the general formula (1) wherein the symbols have the meanings given in the specification.
Patent IL-215487-A0 (IL)
Title: Submersible vehicle and method of operation thereof
IPC: B63H5/14
Filed: 2011-10-02
Abstract: A submersible vehicle having an outer hull which defines a hull axis and appears substantially annular when viewed along the hull axis, the interior of the annulus defining a duct which is open at both ends so that when the vehicle is submerged in a liquid, the liquid floods the duct. The vehicle further comprises a buoyancy control system. Various methods of deploying and using the vehicle are described.
Patent RO-129070-A0 (RO)
Title: Thermostating vessel
Inventor: AMARIEI SONIA
IPC: B01L3/00
Filed: 2013-03-13
Abstract: The invention relates to a modular system intended for thermostating some cylinder-shaped glass jars containing a working reagent or solution. According to the invention, the thermostating system comprises a cylindrical vessel (1) made of polymeric material, a thermostating solution (2), a ring (3) made of polymeric material which exhibits a circular cavity wherein there is arranged a thin-walled resilient closed sealing ring (4) made of silicone rubber, a micro compressor (11) and a pneumatic valve (5) for inflating the sealing ring (4), an intake nozzle (6) and an outlet nozzle (7) for a liquid heating medium, a cylinder-shaped glass jar (8) which contains the working fluid (9) and a thermostat (10) provided with a pump for recycling the heating medium.
Patent RO-132212-A0 (RO)
Title: Differential speed amplifier with two counter-rotating outputs
Inventor: SĂULESCU RADU GABRIEL
IPC: F03D7/00
Filed: 2017-05-30
Abstract: The invention relates to a differential speed amplifier with two inputs and two counter-rotating outputs meant to be integrated in wind turbine systems with two counter-rotating wind rotors and a counter-rotating generator, in order to harmonize the low nominal speeds of the two wind rotors with the high nominal speed of the electric generator. According to the invention, the amplifier comprises a central toothed wheel (1) with external toothing, made integral with a mobile rotor (8) of a counter-rotating electric generator, a central toothed wheel (2) with internal toothing, made integral on the one hand with a mobile stator (9) of the electrical generator and on the other hand with a secondary wind rotor (10), the central wheels (1 and 2) engaging simultaneously with a satellite wheel (3) made integral with a satellite wheel (4) which engages with an internal-toothing wheel (5) made integral with a main wind rotor (11), where the satellite wheels (3 and 4) form a double satellite (6) which keeps the contact with central wheels (1, 2 and 5) by means of a satellite-holder element (7), the planetary amplifier having two or more double satellites (6) mounted in parallel, and the wheels (1, 2, 3, 4 and 5) can be toothed wheels or friction wheels, in case of low power systems.
Patent LU-74030-A1 (LU)
IPC: A47F3/04
Filed: 1975-12-16
Abstract: 1506655 Refrigerators LINDE AG 11 Dec 1975 [20 Dec 1974] 50760/75 Heading F4H In a refrigerated display case in which air is drawn into a duct, cooled and passed out to form an air curtain, the air passes out from the duct through open-celled foamed material, e.g. polyester foam. As shown, the duct 3 includes an evaporator 4 and a fan 5 and the duct outlet is covered by polyester foam strips 7 supported so as to have two inlet faces and one outlet face. In a second embodiment, Fig. 3 (not shown), in which the duct is defined by the back wall of the goods compartment and the back wall of the casing, the back wall of the goods compartment being perforated or slotted and faced with open-celled foamed material through which the air passes and passes over shelves supported on the back wall.
Patent LU-88187-A1 (LU)
Inventor: COUTSOMITROS CONSTANTIN
IPC: G03H1/00
Filed: 1992-11-03
Abstract: Detector of variations in a physical quantity such as temperature, light intensity or pressure. According to the invention, the detector comprises an optical interferometric cavity (6) composed of two holographic glass plates on which three-dimensional interferometric networks have been previously recorded, said glass plates being placed adjacent to one another with a thin air layer in between, said physical quantity being capable of acting on said cavity; a laser beam generator (1) directing its coherent beam on said cavity; and a receiver (8) which captures light (7) reflected by said optical cavity or having traversed said optical cavity and capable of showing variations in the interference fringes induced by said variations in the physical quantity.
Patent MA-21026-A1 (MA)
Inventor: FREDDY FRANCOIS VLAEMINCK
IPC: C07D211/58
Filed: 1987-07-02
Abstract: The use for the manufacture of a medicament for the treatment of diarrhea of a compound of formula <CHEM> wherein Ar is thienyl, halothienyl, furanyl, halofuranyl, pyridinyl, aminopyridinyl, thiazolyl, imidazolyl or a radical of formula <CHEM> Ar<1> and Ar<2> are, each independently, phenyl or halophenyl; the pharmaceutically acceptable acid addition salts and possible stereochemically isomeric forms thereof; pharmaceutical compositions containing such compounds as an active ingredient and methods of preparing said compounds and pharmaceutical compositions; novel compounds of formula (I).
Patent MA-23292-A1 (MA)
Inventor: FOLSBERG JAN
IPC: B02C15/06
Filed: 1994-07-29
Abstract: The present invention relates to a ring roller mill which, among other things, can be used in connection with the manufacture of cement for grinding of mineral clinker materials, slags, and similar materials. The mill has a grinding ring 1 and a roller 2. Between the roller 2 and the grinding ring 1, the partially crushed material forms a grinding bed 4 and on each side of the grinding ring 1 dam rings 5 are fitted. On the outer side of the dam rings 5 are fitted collecting jackets 6, to which scoop plates 7 are fixed. The jacket collects the material which flows over the dam ring and by means of the scoop plates the material is lifted round with the collecting jacket. Since the speed of the jacket is lower than the critical speed, the material will drop off from the uppermost part of the jacket, being dispersed towards the bottom of the latter, and is subsequently returned to the grinding path. Effective internal conveyance is achieved with the mill according to the invention, hence eliminating the need for any external conveyance of overflow material.
Patent MA-23642-A1 (MA)
Inventor: REINHARD RIES
IPC: A62C3/02
Filed: 1995-08-08
Abstract: PCT No. PCT/EP95/02964 Sec. 371 Date Sep. 27, 1996 Sec. 102(e) Date Sep. 27, 1996 PCT Filed Jul. 26, 1995 PCT Pub. No. WO96/04960 PCT Pub. Date Feb. 22, 1996What is disclosed is a device for extinguishing fires, and utilization of the device for stationary protection of specific objects, and for dust abatement during blasting operations, and a method for extinguishing forest or terrain fires with the extinguishing device. The extinguishing device comprises a container for receiving an extinguishing agent, and an explosive in or on this container, by means of detonation of which the extinguishing agent is atomized to form a mist and brought into the fire. In order to increase the flexibility and effectiveness in practical use, the container consists of a flexible hose which may be closed at both ends. The method of extinguishing forest or terrain fires with this device provides for the hose to be laid out in front of the fire front, filled with the extinguishing agent, and exploded by detonation of the explosive.
Patent MA-38205-A1 (MA)
Title: Procédé d'obtention d'un revêtement antireflet pour dispositifs optiques et thermoélectriques
Inventor: CAPARROS JIMENEZ SEBASTIAN
IPC: C03C17/00
Filed: 2013-12-19
Abstract: La présente invention concerne un procédé sol-gel pour l'obtention d'un revêtement antireflet à partir de précurseurs de type alcoxyde, qui peuvent ensuite être appliqués sur des substrats de verre ou de plastique par pulvérisation. L'invention concerne également des dispositifs optiques et thermoélectriques revêtus dudit matériau antireflet. Ce revêtement augmente le facteur de transmission des substrats transparents sur lesquels il est appliqué, et convient par conséquent pour être appliqué sur des modules solaires haute concentration (hcpv), aussi bien sur les lentilles primaires que secondaires, sur du silicium classique ou sur des tubes csp.
Patent MA-39163-A1 (MA)
Title: Forme cristalline de (s)-(2-(6-chloro-7-methyl-1h-benzo[d]imidazol-2-yl)-2-methylpyrrolidin-1 -yl)(5-methoxy-2-(2h-1,2,3-triazol-2-yl)phenyl)methanone et utilisation de celle-ci en tant qu'antagonistes des recepteurs de l'orexine
Inventor: BOSS CHRISTOPH
IPC: C07D403/14
Filed: 2014-12-02
Abstract: L'invention concerne des formes cristallines de (s)-(2-(6-chloro-7-méthyl-1h-benzo[d]imidazol-2- yl)-2-méthylpyrrolidin-1-yl)(5-méthoxy-2-(2h-1,2,3-triazol-2-yl)phényl)méthanone, des procédés de préparation de celles-ci, des compositions pharmaceutiques contenant de telles formes cristallines, des compositions pharmaceutiques préparées à partir de telles formes cristallines ainsi que leur utilisation en tant que médicament, notamment en tant qu'antagonistes des récepteurs de l'orexine.
Patent UY-23373-A1 (UY)
Inventor: DHIRAJ SHANTILAL MODY
IPC: A61K31/19
Filed: 1992-02-10
Abstract: The invention provides a topical analgesic composition comprising an oil-in-water emulsion containing about 5% to about 12% by weight of ibuprofen and about 60% to about 90% by weight of water, the oil phase of the emulsion consisting essentially of emollient constituents that do not dissolve the ibuprofen to any great extent at a pH of 4-7, the composition having a pH of about 4 to about 7.2 such that the ibuprofen is suspended in substantially solid crystalline form and the ibuprofen which is dissolved is partially in the neutral or non-charged state. The invention also includes a process for preparing this composition.
Patent UY-26206-A1 (UY)
Title: Antagonistas del receptor de il-8.
Inventor: BENSON KATHERINE L WIDDOWSON Y
IPC: A61P31/04
Filed: 2000-06-13
Abstract: Esta invención se refiere a nuevas fenil-ureas útiles en el tratamiento de estados de enfermedad mediados por la quimiocina interleucina-8 (IL-8)
Patent UY-26666-A1 (UY)
Title: Compuestos y composiciones antipicornavirales, sus usos farmaceuticos y los materiales para su sintesis
Inventor: DRAGOVICH PETER S
IPC: C07D/
Filed: 2001-04-16
Abstract: Compuestos de la fórmula: donde las variables de la fórmula son como se define aquí, que ventajosamente inhiben o bloquean la actividad biológica de la proteasa 3C picornaviral. Estos compuestos, así como las composiciones farmacéuticas que contienen estos compuestos, son útiles para el tratamiento de pacientes o anfitriones infectados con uno o más picornaviruses, tal como RVP. También se describen métodos intermediarios y sintéticos para preparar estos compuestos.
Patent UY-29221-A1 (UY)
Title: Derivados de octahidropirrolo(3,4-c)pirrol
Inventor: LANE CHARLOTTE ALICE LOUISE
IPC: C07D233/20
Filed: 2005-11-21
Abstract: La presente invención se refiere a derivados de octahidropirrolo(3,4-c)pirrol de fórmula (I): y a procedimientos para su preparación, a composiciones que los contienen y a sus usos.
Patent UY-31608-A1 (UY)
Title: Derivados de carboxamidas n-azabicíclicas, su preparación y su aplicación en terapéutica
Inventor: ODILE LECLERC
IPC: A61K31/404
Filed: 2009-01-22
Abstract: Compuestos derivados de carboxamidas azabicíclicas de fórmula general (I) en el estado de base o de sal de adición a un ácido, así como en el estado de hidrato o de solvato, en cuya fórmula los sustituyentes e índices son tales como se especifican en la memoria descriptiva y en las reivindicaciones. Procedimiento de preparación o el tratamiento de patologías en las que estén implicados los receptores de tipo TRPV1