baber/WOPTO huggingface dataset:
Patent FI-943231-A (FI)
Inventor: BJOERN SOEREN ERIK
IPC: A61P9/10
Filed: 1994-07-06
Abstract: A variant of the C-terminal Kunitz-type protease inhibitor domain of the  alpha 3 chain of human type VI collagen, the variant comprising the following amino acid sequence X1 X16 Asp Ile Cys Lys Leu Pro Lys Asp X2 Gly X3 Cys X4 X5 X6 X7 X8 X9 Trp Tyr Tyr Asp Pro Asn Thr Lys Ser Cys Ala Arg Phe X10 Tyr Gly Gly Cys X11 X12 X13 Glu Asn Lys Phe X14 Ser Gln Lys Glu Cys Glu Lys Val Cys Ala Pro X15 (SEQ ID NO. 1) wherein X1, X15, and X16 represents a naturally occurring amino acid residues except Cys and X2-X14 each independently respresents a naturally occurring amino acid residue, with the proviso that at least one of the amino acid residues X1-X16 is different from the corresponding amino acid residue of the native sequence. Alternatively, the N-terminal Asp may be preceded by H or 3-5 amino acid residues and the C-terminal Pro may be followed by OH or 3-5 amino acid residues.
Patent FI-945052-A (FI)
Inventor: HAIKALA HEIMO OLAVI
IPC: C07D237/08
Filed: 1994-10-27
Abstract: PCT No. PCT/FI93/00191 Sec. 371 Date Nov. 22, 1994 Sec. 102(e) Date Nov. 22, 1994 PCT Filed May 5, 1993 PCT Pub. No. WO93/21921 PCT Pub. Date Nov. 11, 1993.A method for preventing or treating myocardial ischemia in a mammalian organism is disclosed. The compound [[4-(1,4,5,6-tetrahydro-4-methyl-6-oxo-3-pyridazinyl)phenyl]hydrazono]propanedinitrile or its enantiomer or a pharmaceutically acceptable salt there is administered to a mammalian organism in need of such prevention or treatment. The compound may be administered in its racemic form or in a form which is substantially free of the (+)-enantiomer or substantially free of the (-)-enantiomer.
Patent FI-950562-A (FI)
Inventor: NILSSON HUGO
IPC: B65D43/08
Filed: 1995-02-09
Abstract: PCT No. PCT/SE93/00677 Sec. 371 Date Jan. 27, 1995 Sec. 102(e) Date Jan. 27, 1995 PCT Filed Aug. 12, 1993 PCT Pub. No. WO94/04422 PCT Pub. Date Mar. 3, 1994A container (1) for a lubricant has a cap (2) for sealing off one end (4) of a cylindrical tube (2). The cap (2) shows a bottom (19), from the periphery of which extends in an axial direction a circumferential interior ring part (17), which faces the inside of said tube end (4). The cap (3) rests, with a radially extended ring part (16) connected to said interior ring part (17), upon a radial end surface of said tube end (4). According to the invention, the latter end shows a circumferential flange edge pointed obliquely inwardly towards the central part of the tube (2) and being intended to act upon an exterior circumferential bulge (24) on the outside of cap wall (17). For optimal insertion into the tube (2) and passing said edge (18), said bulge (24) downwardly forms a longer bevel (24) with a minor style in relation to said wall (17), while for optimal locking, said bulge (24) is upwardly more acutely rounded close to said lateral wall (17).
Patent FI-954447-A (FI)
Inventor: PATTERSON ALAN
IPC: A61K9/00
Filed: 1995-09-20
Abstract: A sustained release veterinary composition, for intra-muscular and subcutaneous administration comprises Tylosin and an oily vehicle containing a gelling agent, wherein the gelling agent may be an aluminium salt of a fatty acid such as stearic acid and the oily vehicle may be a low viscosity polyol diester of a short chain naturally derived fatty acid such as propylene glycol dicaprylate/dicaprate.
Patent FI-955661-A (FI)
Inventor: BUZZETTI FRANCO
IPC: C07D209/22
Filed: 1995-11-24
Abstract: PCT No. PCT/EP95/00758 Sec. 371 Date Nov. 21, 1995 Sec. 102(e) Date Nov. 21, 1995 PCT Filed Mar. 2, 1995 PCT Pub. No. WO95/26341 PCT Pub. Date Oct. 5, 1995The present invention relates to new compounds of formula    <IMAGE>  (I)  wherein A is a bicyclic ring chosen from naphthalene, tetrahydronaphthalene, quinoline, isoquinoline and indole. B is a R2 substituted benzene ring or an unsubstituted pyridine or thiophene ring; R is hydrogen, C1-C6 alkyl, halogen, nitro, cyano, carboxy or a group NR3R4 wherein each of R3 and R4 is independently hydrogen or C1-C6 alkyl; R1 is hydrogen, C1-C6 alkyl or C1-C6 alkanoyl; R2 is hydrogen, C1-C6 alkyl, halogen, nitro, cyano, carboxy, hydroxy, C1-C6 alkoxy, C1-C6 alkanoyloxy or a group NR3R4 wherein R3 and R4 are as defined above; n is zero or an integer of 1 to 2; x is zero or an integer of 1 to 5; and the pharmaceutically acceptable salts thereof. The compounds of the invention are useful as tyrosine kinase inhibitors.
Patent FI-961503-A (FI)
Inventor: HOERMANN THOMAS J
IPC: E05F15/00
Filed: 1996-04-03
Abstract: Described is a door unit with a door which can be raised overhead, such as a jointed pull-up door, and with vertical frame spars fixed round the edge of the doorway and with a guide-rail system in whose rails the door is fitted so that it can be displaced along the rails and with ropes which hold the door, the ropes passing over pulleys and being attached to a fixed shaft. In order to prevent unauthorized opening of the door, the door has a latch assembly which is attached to at least one side of the door and which acts on the rope on this side of the door, the latch assembly having a latch which engages, when the door is raised, with a catch in the vicinity of at least one of the spars if this rope becomes slack.
Patent GB-849812-A (GB)
Title: Improvements in or relating to electric ignition systems
Inventor: FRANKLIN SIDNEY HENRY
Filed: 1956-01-12
Abstract: 849,812. Ignition systems. BRITISH THOMSON-HOUSTON CO. Ltd. Jan. 8, 1957 [Jan. 12, 1956], No. 1118/56. Class 7(4). [Also in Group XXXV] In an ignition system of the kind comprising a generator, a capacitor 5 charged from an armature of the generator and a plug 12 supplied with sparking voltage from the capacitor, the generator is adapted to produce a peaked wave and the shaft of the generator carries the armature also a rotating contact such as a conducting segment 7 connected to the armature and co-operating with a stationary contact such as a brush supplying the sparking plug, the angular-position of the contacts in relation to that of the armature being such as to cause engagement at a point on the front of the wave near the peak. The spark may be retarded by displacing the brush holder 8, Fig. 3, angularly about the axis of the generator. The capacitor 5 is carried as shown in a plate 4 carried by one end of the generator rotor 1. The system may use surface discharge plugs or spark plugs of any other conventional type. A short circuiting switch can be provided in the ignition circuit or in the circuit of an additional winding which is arranged in the electromagnetic field of the armature winding of the generator.
Patent GB-1409326-A (GB)
Title: Preparation of stilbene-azo dyes
IPC: C09B56/04
Filed: 1973-01-09
Abstract: 1409326 Preparation of stilbene-azo dyestuffs IMPERIAL CHEMICAL INDUSTRIES Ltd 7 Jan 1974 [9 Jan 1973] 1126/73 Heading C4P Stilbene-azo dyes are prepared by condensing 4,4<SP>1</SP> - dinitro - 2,2<SP>1 </SP>- stilbenedisulphonic acid or a salt thereof with an aminoazo compound in an aqueous alkaline medium containing lithium hydroxide. Preferably the dilithium salt of 4,41 - dinitro - 2,21 - stilbenedisulphonic acid is used. Concentrated aqueous solutions of the products may be obtained and are used for dyeing cotton and paper. The orange dye C.I. Direct Orange 34 (C.I. 40215) may be obtained in the form of a lithium salt by the above process using 4<SP>1</SP>-aminoazobenzene-4-sulphonic acid as the aminoazo compound.
Patent GB-1409490-A (GB)
Title: Meter interrogation systems
IPC: H02J13/00
Filed: 1973-05-15
Abstract: 1409490 Electric selective signalling GENERAL PUBLIC UTILITIES CORP 15 May 1973 1159/75 Divided out of 1409489 Heading G4H The disclosure of the present Specification is identical to that of Specification 1,409,489, but the claims are directed to determining the maximum delay of information signals transmitted over an electric power distribution network connecting a central station to a plurality of remotely located utility meters, to adjust the rate of transmission of the signals in accordance therewith.
Patent GB-562288-A (GB)
Title: Improvements in or relating to the printing cylinders of rotary off-set printing machines
IPC: B41F33/00
Filed: 1943-01-25
Abstract: 562,288. Printing cylinders. PIRIE, W. J. Jan. 25,1943, No. 1207. [Class 100 (ii)] [Also in Group XXIV] A rotary machine cylinder having a longitudinal gap, particularly the printing cylinder of a rotary offset printing press, is provided with a safety guard for the gap comprising a plate or member of substantially the same size as the gap but lying somewhat nearer the centre of the cylinder than the ungapped periphery of the cylinder, the guard being constructed or arranged to give access to the gap when the cylinder is stationary without the necessity of removing the guard. Figs. 1 and 2 show a printing cylinder with two gaps 11 housing the clamps 15 of the printing plate 17, each gap having a guard plate 19 secured by a screw 23 to a support 22 extending from the cylinder hub 10. To provide access to the clamps 15 without removing the guard, the front edge of the guard is provided with notches 20 which may be normally substantially covered by a cover-plate 28 slidable on the plate 19 and guided by slots 29, 32 and pins 31 and fixed by the screw 23. In a modification, instead of providing notches such as 20, the edge of the plate is bent down to lie under the clamps 15.
Patent GB-1332882-A (GB)
Title: Process for producting a pressure-resistant temperature-resistant temperature-resistant foam
IPC: C08G14/06
Filed: 1972-01-10
Abstract: 1332882 Bituminous/carbazole modified novolak foams RUTGERSWERKE AG 10 Jan 1972 [18 Jan 1971] 1214/72 Headings C3C C3R and C3N A foam is made by simultaneously foaming and hardening a mixture of a bituminous substance and a novolak resin, produced by condensing a phenol, carbazole and formaldehyde, e.g. in the presence of an acid. The foaming may occur either by means of gases liberated during hardening, e.g. with hexamethylenetetramine, or by means of an expanding agent. The bituminous substance may be natural or petroleum asphalt, a tar, e.g. coal, lignite or wood, or a pitch, e.g. coal tar, lignite tar or wood. The phenol may be phenol, a cresol and or a xylenol. The mixture may also contain a filler, e.g. talc, asbestos or soot, and polyethylene, polyvinyl chloride or polystyrene.
Patent GB-574250-A (GB)
Title: Improvements relating to thermally responsive devices
IPC: H01R13/595
Filed: 1944-01-21
Abstract: 574,250. Thermometers. NEGRETTI, H. N., NEGRETTI, P. E., and HOTCHEN, C. W. Jan. 21, 1944, No. 1216. [Class 97 (iii)] In a thermometer the indication lag caused by the time occupied in transferring heat to or from the filling fluid is reduced by arranging that the expansion and contraction of the bulb wall predominates in effecting the temperature indication, the function of the fluid filling being purely or mainly to act as a hydraulic transmission medium. As shown in Fig. 1, a tubular bulb 1 of good thermal conductivity and high coefficient of thermal expansion contains a solid core 2 having a relatively low coefficient of thermal expansion. A thin annular space 3 between the bulb and core is filled with the transmitting fluid and communicates by means of capillary tubing 6 with a Bourdon tube 7. In a modification, Fig. 3, wherein the temperature of fluid passing through a pipe line may be measured, the thermometer has screwed ends 14, 15 for connecting it in the pipe line and comprises a non-expansible outer tube 8 and an expansible inner tube 9 leaving an annular space 10 communicating with the Bourdon tube by capillary tubing 13. Suitable low or non-expansible materials for the core 2 are quartz or fused silica or nickel-iron alloy. The core may consist of several rods or beads. Specification 167,000, [Class 97 (iii)], is referred to.
Patent GB-994546-A (GB)
Title: Dithiocarbamic acid esters
Inventor: KUEHLE ENGELBERT
IPC: C07C333/18
Filed: 1964-01-10
Abstract: The invention comprises dithiocarbamic acid esters of the formula <FORM:0994546/C2/1> wherein X represents oxygen or sulphur and R represents an alkyl, aralkyl, aryl, alkaryl or cycloalkyl radical which may be optionally substituted, e.g. by Cl, Br, nitro or alkoxy. The above compounds are prepared by reacting methylamine and carbon disulphide with a vinyl compound of the formula CH2 = CH.X.R.ALSO:Fungicidal and nematicidal compositions contain as the active ingredient dithiocarbamic acid esters of the formula <FORM:0994546/A5-A6/1> wherein X represents oxygen or sulphur and R represents an unsubstituted or substituted alkyl, aralkyl, aryl, alkaryl or cycloalkyl radical.
Patent GB-582206-A (GB)
Title: Improvements in tailless airplanes
IPC: B64C9/00
Filed: 1944-01-25
Abstract: 582,206. Tailless aircraft. NORTHROP AIRCRAFT, Inc. Jan. 25, 1944, No. 1417. Convention date, Sept. 24, 1942. [Class 4] A tailless aircraft is rendered longitudinally stable by disposing the aerodynamic centre 15 of the wing ahead of the centre of gravity 13 of the machine, and by providing control surfaces having negative trailing characteristics, i.e. surfaces whose angles of attack increase with increase of incidence of the wing. In the arrangement shown in Fig. 5, the control surface 17 is pivoted at 19 so as to be overbalanced, and a balance tab 23 is provided, while in the construction according to Fig. 7 the surface 11 is controlled by a weight 24, or a spring may be used in place of a weight, Fig. 8 (not shown). Alternatively, the control surface may be provided at its leading edge with a vane projecting into a sealed recess at the trailing of the wind, the recess being in communication with selected points on the wing surface, Fig. 6 (not shown), or gyroscopic control mechanism may be used to impart the negative trailing characteristic. The aircraft illustrated in Fig. 9 is provided with control surfaces 27 incorporating balance tabs 29, as in the arrangement according to Fig. 5, and trimming tabs 31, together with rudders 33. The surfaces 27 may be used as combined elevators and ailerons, and as landing flaps. Alternatively, the members 27 may be employed only as elevators and stabilizing flaps, in which case the members 33 serve as ailerons. Instead of employing trimming tabs, a hydraulic or electric booster may be incorporated in the elevator control system, the position of the control column determining the elevator hinge moment. The control forces are applied by movements of the pilot's control member in the conventional directions.
Patent GB-110462-A (GB)
Title: Means for Locking Electric Lamps in their Sockets.
IPC: H01R33/97
Filed: 1917-01-29
Abstract: 110,462. Beith, G. R., and British Agencies, Ltd. Jan. 29, 1917. Electro-magnets.-A magnet for disengaging an enclosed catch in an electric lamp holder has a pointed pole 15 for insertion in a depression in the casing enclosing the catch, a coil 16, a handle 18, a press switch 17, and flexible conductors leading to a portable battery.
Patent GB-344595-A (GB)
Title: Improvements relating to bowls or containers
IPC: D01D7/02
Filed: 1930-01-16
Abstract: 344,595. Centrifugal spinning pots. WESTINGHOUSE ELECTRIC & MANUFACTURING CO., East Pittsburg, U.S.A. -(Assignees of Schmidt, H. F. ; 85, S. Lansdown Avenue, Lansdowne, Kempton, W. H. ; Newport Road, Wilkinsburg, and Gudge, B. J. ; 144, Avenue A, East Pittsburg, all in Pennsylvania, U.S.A.) Jan. 16, 1930, No. 1578. Convention date, Jan. 18, 1929. [Class 23.] Bowls or containers, particularly bowls used in the manufacture of artificial silk, comprise a base 2 formed of agglomerated material such as shredded fabric or ground asbestos, impregnated with a binder, such as a phenolic condensation product, and a wall 1 formed of laminated sheets of fibrous material impregnated with a similar binder, the base and wall being moulded under heat and pressure into a unitary structure. The inner sheets of the wall are formed of finely woven material such as cambric and the outer sheets of coarsely woven material such as canvas or duck, or comminuted material may be used as an interior facing. The lower edges of the sheets forming the wall are bent inwardly to form a ragged-edged flange which intimately associates with the material forming the base. The base is preferably moulded around a bush 5 which forms the bearing for the driving-shaft. The wall is formed with an annular shoulder 8, and the cover 3 which is also formed of impregnated sheet material, is provided with inwardly extending lugs 11 adapted to slide into notched channels 13 in the rim, the channels being bevelled so that, during the rotation of the bowl when spinning, the cover tends to tighten the engagement.
Patent GB-865649-A (GB)
Title: Improvements in or relating to over-temperature protective systems for electric motors
IPC: G05D23/24
Filed: 1959-01-16
Abstract: 865,649. Protective cut-out systems; control of motors. WESTINGHOUSE ELECTRIC CORPORATION. Jan. 16, 1959 [Jan. 20, 1958], No. 1651/59. Classes 38 (3) and 38 (5). [Also in Group XXXV] A protective system for a motor comprises at least one temperature-sensitive resistance element 24 having a positive temperature coefficient of resistance and embedded in or attached to a current carrying winding 30 of the motor, a relay 45 having a coil 46 in series with the element 24 and a low voltage source, and a contactor 34 having an operating coil 36 in series with a voltage supply and the contacts 44 of the relay 45. Under normal conditions the coil 46 of the relay 45 is energized and the contacts 44 are closed, but under overload conditions the rise in temperature of the motor winding causes a sudden increase in the resistance of the element 24 and the relay 45 opens to de-energize the contactor coil 36. A threephase motor may have an element 24 associated with each phase winding. Fig. 3 (not shown) illustrates a modified circuit in which a starting relay provides for automatic resetting when the temperature of the motor returns to normal.
Patent GB-1374741-A (GB)
Title: Window plane having a radio antenna
IPC: H01Q1/32
Filed: 1973-01-12
Abstract: 1374741 Aerials SAINT-GOBAIN INDUSTRIES 12 Jan 1973 [14 Jan 1972] 1784/73 Heading H4A A window pane such as a motor vehicle windscreen incorporates an aerial which comprises two aerial elements of different configurations. The said elements are connected together, and have a common feed terminal. One element is made up of two parts which are arranged with relative electrical asymmetry with respect to the other element. Both elements are tuned to the same frequency, e.g. a frequency in the range 80 to 220 mHz. In one embodiment, a windscreen la, Fig. 3, comprises a central vertical conductor 2 which extends from a terminal 4 to connect at a point 5 with an upper horizontal conductor 3. Each conductor has a length equivalent to #/2 (# = wavelength at frequency of operation) and the point 5 is offset from the centre of the conductor 3 to provide optimum feed conditions. In a second embodiment a central vertical conductor is provided with a symmetrically disposed upper horizontal member (forming a "T") and is associated with a lower asymmetrically disposed horizontal conductor, the two conductors being connected together adjacent a feed terminal (Fig. 4, not shown). In a third embodiment a T-shaped central conductor 13, 14, Fig. 5, is associated with a U-shaped conductor having two symmetrical branches 15a, 15b. Asymmetry is provided by capacitive loading of the branch 15b, a conductor 16 being disposed parallel thereto, and connected to the vehicle body. Alternatively, inductive loading may be used. In a fourth embodiment, somewhat similar to the third, asymmetry is provided by omitting the upper horizontal part of one of the branchesof the U-shaped conductor (Fig. 6, not shown). In other embodiments, also somewhat similar to the embodiment shown in Fig. 5, asymmetry is provided in the lower horizontal portions of the two branches of the U-shaped conductor, in one case by duplication of unequal portions thereof (Fig. 7, not shown), and in the other case by inserting zig-zag portions of unequal lengths (Fig. 8, not shown). In a seventh embodiment, a windscreen lg, Fig. 9, comprises a T-shaped central conductor 36, 37, which extends from a terminal 38, and an associated U-shaped conductor 39a, 39b. The lower part of the U-shaped conductor comprises three parallel conductors 40a-40b, 41a-41b, 42a-42b. On one side, the three conductors 40b, 41b, 42b are connected in parallel. Before they reach the central conductor 36, they are connected to a conductor 43, Fig. 10, which is arranged around the terminal 38. The conductors 40a, 41a form branches having free ends, whereas the conductor 42a is connected at 47 to the conductor 43. The conductor 43 is extended by conductors 44, 45 arranged in a loop and connected at 46 to the central conductor 36. It is stated that when such an aerial is installed in a car radiation diagram minima in the fore and aft directions are improved (Fig. 11, not shown).
Patent GB-170785-A (GB)
Title: An element for use in building constructional toys or models
IPC: A63H33/04
Filed: 1921-01-13
Abstract: 170,785. Hornby, F. Jan. 13, 1921. Mechanical constructions, details for building up.-An element for use with constructional toys consists of a pawl having two teeth so positioned that the pawl may be turned on its pivot to engage one or the other of two gear-wheels. The pawl consists of a tubular boss 1 to which is secured a blade 6 having two oppositely-directed teeth 9, 9<a>. The boss is provided with a pinch. ing-screw to enable it to be secured to a rod if desired. A pivot bolt a, Fig. 4, for use with the pawl has a plain shank 11 and a threaded tip 12. The plain shank forms a pivot for the bars 1, while the threaded end enables the bolt to be secured to the usual perforated strips 13 by means of two nuts 14, 15.
Patent GB-764226-A (GB)
Title: Diaryl disulphonamides
Filed: 1955-01-21
Abstract: The invention comprises diaryl disulphonamides of the general formula <FORM:0764226/IV(b)/1> in which X is a carbonyl or dicarbonyl radical or an alkylene radical containing from 1 to 5 carbon atoms, and their preparation by two methods: (1) reacting the corresponding disulphonyl halide with ammonia or a substance producing ammonia under the reaction conditions such as an ammonium salt or hexamethylene tetramine, and (2) oxidizing the corresponding disulphenamide.  The first method is preferably conducted in the presence of a diluent such as water or dioxan at temperatures below about 100 DEG  C. and preferably at room temperature.  Specified oxidizing agents for use in the second method are hydrogen peroxide in acid solution and alkaline permangate solutions.  Examples illustrate the preparation of the 4,41-di-sulphonamides of diphenylmethane, benzophenone, benzil and a ,a  - dimethyldiphenylmethane.  Starting materials.  Diaryl disulphonyl halides may be obtained by direct sulphochlorination, by reacting an alkali-metal salt of the corresponding disulphonic acid with an acid halide or by replacing amino groups by sulphonyl halide groups by diazotization followed by reaction with sulphur dioxide in the presence of a catalytic amount of cuprous chloride.  Disulphenamides may be obtained by direct halogenation of a dimercaptan in an inert solvent followed by reaction of the resulting disulphene chloride with ammonia.