Abstract:
Specific fluoroethoxy pyrimidines and triazines are useful as general or selective preemergent and postemergent herbicides. Ortho-ethoxy and ortho-propoxy substituted benzenesulfonamides, such as 2-ethoxy-N-[[4-methoxy-6-(2,2,2-trifluoroethyoxy)-1,3,5-triazin-2-yl]aminocarboxy]benzenesulfonamide and N-[[4-methoxy-6-(2,2,2-trifluoroethoxy)-1,3,5-triazin-2-yl]aminocarbonyl]-2-propoxybenzenesulfonamide, and their agriculturally suitable salts show preemergent and postemergent herbicial utility in corn.

Description:
RELATED APPLICATION 
     This application is a continuation-in-part of application U.S. Ser. No. 625,911, filed June 29, 1984, now abandoned which is a continuation-in-part of application U.S. Ser. No. 587,063, filed Mar. 7, 1984, now abandoned. 
    
    
     BACKGROUND OF THE INVENTION 
     The present invention relates to novel 2-fluoro-, 2,2-difluoro- and 2,2,2-trifluoroethoxy pyrimidine- and triazine-containing sulfonylureas which are useful as preemergent and postemergent herbicides. 
     Herbicidal benzenesulfonylureas of the formula ##STR1## wherein among the substituents disclosed R 4-6  can each be hydrogen, R 3  can be alkoxy of 1-4 carbon atoms, X can be alkoxy of 1-3 carbon atoms and Z is methyl or methoxy are disclosed in U.S. Pat. No. 4,127,405, issued Nov. 28, 1978 to Levitt. 
     European Patent Application (EP-A) No. 9419, published Apr. 2, 1980, discloses herbicidal benzene and thiophene sulfonylureas such as ##STR2## wherein among the substituents disclosed R 4  can be OCH 3 , X can be OCH 3 , and Y can be OCH 2  CF 3 . 
     South African Application No. 825671 (Swiss priority Aug. 6, 1981; EP-A-72,347, published Feb. 16, 1983) claims ortho-substituted alkoxy benzenesulfonylureas such as ##STR3## 
     South African patent application No. 835165 filed by Ciba-Geigy (Swiss Priority 7/16/82) discloses herbicidal sulfonylureas of the general structure shown below: ##STR4## wherein A is an unsubstituted or substituted bridge of 3 or 4 atoms which contains 1 or 2 oxygen, sulfur or nitrogen atoms and, together with the linking carbon atom, forms a non-aromatic 5- or 6-membered heterocyclic ring system, with the proviso that two oxygen atoms are separated by at least one carbon atom and that oxygen and sulfur atoms are only linked to each other if the sulfur atom takes the form of the --SO-- or SO 2  -- group; and R 3  and R 4  may be, among other values, a C 1  -C 4  haloalkoxy group. 
     SUMMARY OF THE INVENTION 
     This invention relates to novel compounds of Formula I, agriculturally suitable compositions containing them, and their method-of-use as general or selective preemergent and postemergent herbicides. ##STR5## wherein R is H or CH 3  ; 
     X is CH 3  or OCH 3  ; 
     Y is OCH 2  CH 2  F, OCH 2  CHF 2  or OCH 2  CF 3  ; 
     Z is CH or N; 
     L is ##STR6## R 1  is C 2  -C 4  alkyl, C 2  -C 4  alkoxy, SO 2  NR 8  R 9 , SO 2  N(OCH 3 )CH 3 , or 2-tetrahydrofuranyl; 
     R 2  is H, F, Cl, Br, CF 3 , CH 3 , OCH 3  or SCH 3  ; 
     R 3  is H, CH 3 , OCH 3 , F, Cl, Br, SO 2  N(CH 3 ) 2 , OSO 2  CH 3  or S(O) n  CH 3  ; 
     R 4  is C 1  -C 3  alkyl, F, Cl, Br, NO 2 , SO 2  NR 8  R 9 , SO 2  N(OCH 3 )CH 3  or S(O) n  R 10  ; 
     R 5  is H, C 1  -C 5  alkyl, CH 3  OCH 2  CH 2 , C 2  H 5  OCH 2  CH 2  or C 1  -C 4  alkyl substituted with 1-3 atoms of F or Cl or 1 Br; 
     R 6  is H or CH 3  ; 
     R 7  is H or CH 3  ; 
     R 8  is C 1  -C 3  alkyl; 
     R 9  is C 1  -C 3  alkyl; 
     R 10  is C 1  -C 3  alkyl or CH 2  CH═CH 2  ; 
     m is 0 or 1; and 
     n is 0, 1 or 2; 
     and their agriculturally suitable salts; provided that 
     (1) the total number of carbon atoms of R 8  and R 9  is less than or equal to four; 
     (2) when m is 1, R 6  is H; 
     (3) when L is L-1 and R 1  is SO 2  NR 8  R 9 , SO 2  N(OCH 3 )CH 3  or 2-tetrahydrofuranyl, then Y is OCH 2  CH 2  F or OCH 2  CHF 2  ; and 
     (4) when L is L-6, L-7, L-8, L-9 or L-10, then Y is OCH 2  CH 2  F or OCH 2  CHF 2 . 
     Preferred for reasons of their greater herbicidal activity, greater plant growth regulant activity and/or more favorable ease of synthesis are: 
     (1) Compounds of Formula I where L is L-1. 
     (2) Compounds of Formula I where L is L-2. 
     (3) Compounds of Formula I where L is L-3. 
     (4) Compounds of Formula I where L is L-4. 
     (5) Compounds of Formula I where L is L-5. 
     (6) Compounds of Formula I where L is L-6 or L-7. 
     (7) Compounds of Formula I where L is L-8 or L-9. 
     (8) Compounds of Formula I where L is L-10. 
     (9) Compounds of Preferred 1 where R is H; R 1  is C 2  -C 3  alkoxy; R 2  is H; and Z is N. 
     (10) Compounds of Preferred 2 where R is H; R 3  is CH 3 , OCH 3 , Cl, SCH 3  or Br; and Z is N. 
     (11) Compounds of Preferred 3 where R is H; R 4  is CH 3 , S(O) n  CH 3 , S(O) n  CH 2  CH 3  or SO 2  N(CH 3 ) 2  ; and Z is N. 
     (12) Compounds of Preferred 4 where R is H; R 4  is CH 3 , S(O) n  CH 3 , S(O) n  CH 2  CH 3  or SO 2  N(CH 3 ) 2  ; and Z is N. 
     (13) Compounds of Preferred 5 where R is H; R 4  is CH 3 , S(O) n  CH 3 , S(O) n  CH 2  CH 3  or SO 2  N(CH 3 ) 2  ; and Z is N. 
     (14) Compounds of Preferred 6 where R is H; R 2  is H; R 5  is H, C 1  -C 4  alkyl, CH 2  CH 2  OCH 3 , CH 2  CH 2  OC 2  H 5  or C 1  -C 4  alkyl substituted with 1-3 atoms of F or Cl or 1 Br; R 6  is H; and Z is N. 
     (15) Compounds of Preferred 7 where R is H; R 2  is H; R 5  is H, C 1  -C 4  alkyl, CH 2  CH 2  OCH 3 , CH 2  CH 2  OC 2  H 5  or C 1  -C 4  alkyl substituted with 1-3 atoms of F or Cl or 1 Br; and Z is N. 
     (16) Compounds of Preferred 8 where R is H; R 2  is H; and Z is N. 
     Specifically Preferred for their greatest herbicidal activity, greatest plant growth regulant activity and/or most favorable ease of synthesis are: 
     2-ethoxy-N-[[4-methoxy-6-(2,2,2-trifluoroethoxy)-1,3,5-triazin-2-yl]aminocarbonyl]benzenesulfonamide, m.p. 180°-181° (d); and 
     N-[[4-methoxy-6-(2,2,2-trifluoroethoxy)-1,3,5-triazin-2-yl]aminocarbonyl]-2-propoxybenzenesulfonamide, m.p. 161°-163° (d). 
     These compounds are excellent preemergent and postemergent herbicides for use in corn. 
     DETAILED DESCRIPTION OF THE INVENTION 
     Compounds of Formula I are prepared by the procedure of Equation 1 wherein L, R, X, Y and Z are as previously defined. This procedure is well known in the art. ##STR7## 
     The reaction is best carried out in inert aprotic organic solvents such as methylene chloride, tetrahydrofuran or acetonitrile, at ambient pressure and temperature. The mode of addition is not critical; however, it is often convenient to add the sulfonyl isocyanate to a stirred suspension of the aminotriazine. Since such isocyanates usually are liquids, their addition is more easily controlled. 
     The reaction is generally exothermic. In some cases, the desired product is insoluble in the warm reaction medium and crystallizes from it in pure form. Products soluble in the reaction medium are isolated by evaporation of the solvent, trituration of the solid residue with solvents such as 1-chlorobutane, ethyl ether, or pentane, and filtration. 
     The intermediate sulfonyl isocyanates of Formula II can be prepared by reacting corresponding sulfonamides with phosgene in the presence of n-butyl isocyanate at reflux in a solvent such as chlorobenzene, according to the procedure of H. Ulrich and A. A. Y. Sayigh, Newer Methods of Preparative Organic Chemistry, Vol. VI, pages 223-241, Academic Press, New York and London, W. Foerst Ed. In cases where formation of the desired sulfonyl isocyanate is difficult by the above procedure the sulfonylurea formed by reaction of butyl isocyanate with the appropriate sulfonamide is treated with phosgene according to the above reference. 
     Alternatively, compounds of Formula I can be prepared by contacting a sulfonyl carbamate of Formula IV with amine III as shown in Equation 2. ##STR8## 
     The reaction is carried out at 50° to 100° C. in a solvent such as dioxane for 0.5 to 24 hours as taught in EP-A-44,807. The required carbamates IV are prepared by contacting the corresponding sulfonamides V with diphenylcarbonate or phenylchloroformate in the presence of base. 
     The compounds of Formula I can also be prepared by contacting a sulfonamide of Formula V with an O-phenylcarbamate of Formula VI in the presence of base as shown in Equation 3. ##STR9## 
     The reaction is carried out at 0° to 50° C. in an inert solvent such as acetonitrile for 0.1 to 24 hours in the presence of a base such as 1,8-diazabicyclo[5.4.0]undec-7-ene (DBU) as taught in EP-A-44,807. The required carbamate VI is prepared by reacting amine III with diphenylcarbonate or phenylchloroformate in the presence of base. 
     The sulfonamides used as intermediates for this invention can be prepared by methods known in the art. The preparation of LSO 2  NH 2  where L is L-1 can be prepared as taught in U.S. Pat. No. 4,127,405; 4,310,346 or 4,435,205. When L is L-3, L-4 or L-5, methods such as those referred to in EP-A-64,804 and U.S. Pat. No. 4,398,939 can be used for the preparation of the sulfonamide intermediates. Naphthalenesulfonamides (L is L-2) can be prepared according to procedures referred to or described in U.S. Pat. No. 4,370,479. Sulfonamides where L is L-6, L-7, L-8, L-9 or L-10 can be prepared as described in EP-A-107,979. 
     Aminotriazines of structure III can be prepared by methods described in EP-A-9,419 (published Apr. 2, 1980). Pyrimidine intermediates of structure III can be prepared by similar procedures by substituting an appropriately substituted pyrimidine for triazines used in the procedures referred to above. 
     Agriculturally suitable salts of compounds of Formula I are also useful herbicides and can be prepared in a number of ways known to the art. For example, metal salts can be made by contacting compounds of Formula I with a solution of an alkali or alkaline earth metal salt having a sufficiently basic anion (e.g., hydroxide, alkoxide, carbonate or hydroxide). Quaternary amine salts can be made by similar techniques. 
     Salts of compounds of Formula I can also be prepared by exchange of one cation for another. Cationic exchange can be effected by direct contact of an aqueous solution of a salt of a compound of Formula I (e.g., alkali or quaternary amine salt) with a solution containing the cation to be exchanged. This method is most effective when the desired salt containing the exchanged cation is insoluble in water and can be separated by filtration. 
     Exchange may also be effected by passing an aqueous solution of a salt of a compound of Formula I (e.g., an alkali metal or quaternary amine salt) through a column packed with a cation exchange resin containing the cation to be exchanged for that of the original salt and the desired product is eluted from the column. This method is particularly useful when the desired salt is water-soluble. 
     Acid addition salts, useful in this invention, can be obtained by reacting a compound of Formula I with a suitable acid, e.g., p-toluenesulfonic acid, trichloroacetic acid or the like. 
    
    
     The compounds of this invention and their preparation are further illustrated by the following examples wherein temperatures are given in degrees centigrade. 
     EXAMPLE 1 
     2-Amino-4-(2,2,2-trifluoroethoxy)-6-methoxy-1,3,5-triazine 
     A. A solution of 300 g (1.63 mol) of cyanuric chloride in 1 liter THF and 0.24 liter diglyme was cooled to 0° C. and 81.6 mL (3.36 mol) of liquid ammonia added dropwise over 90 min. keeping the temperature between 10°-15°. The mixture was stirred for one hour at -10° to 0° and then allowed to warm to ambient temperature over one hour. The resulting suspension was filtered, the solid washed with THF, the filtrate reduced to 1/2 its original volume, and poured over 1 liter of ice water to give a white solid which was collected, washed with water, and dried in vacuo to give 244.3 g of 2-amino-4,6-dichloro-1,3,5-triazine with m.p. 221°-223.5° (dec). 
     B. To a suspension of 50.0 g (0.3 mol) of 2-amino-4,6-dichloro-1,3,5-triazine in 600 mL of methanol was added portionwise 19.5 g (0.3 mol) of 85% potassium hydroxide pellets with the temperature being kept between 15°-20°. The resulting suspension was stirred at 10°-15° for one hour and then allowed to warm to room temperature over 1.5 hours. The white solid was collected, washed three times with water, and dried in vacuo to give 37.1 g of 2-amino-4-chloro-6-methoxy-1,3,5-triazine with m.p. 221°-223.5° (dec). 
     C. To a suspension of 10.0 g (0.06 mol) of 2-amino-4-chloro-6-methoxy-1,3,5-triazine and 6.2 g (0.06 mol) of 2,2,2-trifluoroethanol in 150 mL of methylene chloride was added portionwise over five minutes 4.1 g (0.06 mol) of 85% potassium hydroxide pellets. After an initial exotherm to 27° the reaction mixture was stirred at ambient temperature overnight. The suspended solid was removed by filtration and filtrate concentrated in vacuo to give 13.21 g of white solid with m.p. 77°-80°. This was recrystallized from n-butyl chloride to give 11.16 g of 2-amino-4-(2,2,2-trifluoroethoxy)-6-methoxy-1,3,5-triazine as a white powder with m.p. 78°-80°. 
     NMR: (CDCl 3  +DMSO-d 6 ) δ3.96 (s, OCH 3 ), 4.79 (q, OCH 2  CF 3 ), 6.5 (br s, NH 2 ). 
     EXAMPLE 2 
     2-Ethoxy-N-[[4-methoxy-6-(2,2,2-trifluoroethoxy)-1,3,5-triazin-2-yl]aminocarbonyl]benzenesulfonamide 
     To 1.9 g of 2-amino-4-(2,2,2-trifluoroethoxy)-6-methoxy-1,3,5-triazine suspended in 50 mL of dry methylene chloride was added 2.4 g of 2-ethoxybenzenesulfonyl isocyanate. The mixture was stirred at ambient temperature for three days, filtered, and the filtrate stripped to an oil which crystallized. The solid was triturated with n-butyl chloride and collected to give 2.94 g of white solid with m.p. 180°-181° (dec). 
     NMR: (CDCl 3  +DMSO-d 6 ) δ1.25 (t, CH 3 ), 4.0 (s, OCH 3 ), 4.2 (q, OCH 2 ), 5.2 (Q, OCH 2  CF 3 ), 7.0-8.0 (m, aromatics), 10.8 (br s, NH), 11.7 (br s, NH). 
     EXAMPLE 3 
     N-[[4-methoxy-6-(2,2,2-trifluoroethoxy)-1,3,5-triazin-2-yl]aminocarbonyl]-2-propoxybenzenesulfonamide 
     To 2.0 g of 2-amino-4-(2,2,2-trifluoroethoxy)-6-methoxy-1,3,5-triazine suspended in 35 mL of dry methylene chloride was added 4.4 g of a 50% solution of 2-n-propoxybenzenesulfonyl isocyanate in methylene chloride. The mixture was stirred overnight at ambient temperature and the resulting solution stripped to an amber oil which was triturated with ethanol to give 1.42 g of white solid with m.p. 161°-163° (dec). 
     NMR: (CDCl 3  +DMSO-d 6 ) δ0.9 (t, CH 3 ), 1.7 (m, CH 2 ), 4.1 (m, OCH 3  and OCH 2 ), 5.1 (q, OCH 2  CF 3 ), 7.0-8.0 (m, aromatics), 10.7 (br s, NH), 11.6 (br s, NH). 
     The following compounds can be prepared by one skilled in the art using the proper reactants and the procedures outlined above. 
     
         ______________________________________General Structures for Tables______________________________________General Structure I ##STR10##General Structure II ##STR11##General Structure III ##STR12##General Structure IV ##STR13##General Structure V ##STR14##General Structure VI ##STR15##General Structure VIa ##STR16##General Structure VII ##STR17##General Structure VIII ##STR18##General Structure IX ##STR19##General Structure X ##STR20##______________________________________ 
    
     
                                           TABLE I__________________________________________________________________________General Structure IR.sub.1       R.sub.2               R   X    Y       Z   m.p. (°C.)__________________________________________________________________________C.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NC.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NC.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NC.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHC.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHC.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHC.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NC.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NC.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NC.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHC.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHC.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHCH.sub.2 CH.sub.2 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHCH.sub.2 CH.sub.2 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHCH.sub.2 CH.sub.2 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHCH.sub.2 CH.sub.2 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NCH.sub.2 CH.sub.2 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NCH.sub.2 CH.sub.2 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NCH.sub.2 CH.sub.2 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NCH.sub.2 CH.sub.2 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NCH.sub.2 CH.sub.2 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NCH.sub.2 CH.sub.2 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHCH.sub.2 CH.sub.2 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHCH.sub.2 CH.sub.2 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHOC.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                N   138-142OC.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                N   125-131 (d)OC.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                N   132-137OC.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CH  198-202OC.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOC.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHOC.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                N    94-102: 112 (d)OC.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NOC.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                N   180-181 (d)OC.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOC.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOC.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CH  165-168OCH.sub.2 CH.sub.2 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOCH.sub.2 CH.sub.2 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOCH.sub.2 CH.sub.2 CH.sub.3         H     H   OCH.sub. 3                        OCH.sub.2 CF.sub.3                                CH  168-170OCH.sub.2 CH.sub.2 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                N   120-124 (d)OCH.sub.2 CH.sub.2 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NOCH.sub.2 CH.sub.2 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                N   161-163 (d)OCH.sub.2 CH.sub.2 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                N   139-141 (d)OCH.sub.2 CH.sub.2 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NOCH.sub.2 CH.sub.2 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                N   121-126 (d)OCH.sub.2 CH.sub.2 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CH  176-179OCH.sub.2 CH.sub.2 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOCH.sub.2 CH.sub.2 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHCH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NCH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NCH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NCH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHCH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHCH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CH(CH.sub.2).sub.3 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CH(CH.sub.2).sub.3 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CH(CH.sub.2).sub.3 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CH(CH.sub.2).sub.3 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                N(CH.sub.2).sub.3 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                N(CH.sub.2).sub.3 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NCH.sub.2 CH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NCH.sub.2 CH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NCH.sub.2 CH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NCH.sub.2 CH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHCH.sub.2 CH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHCH.sub.2 CH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHCH(CH.sub.3)C.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHCH(CH.sub.3)C.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHCH(CH.sub.3)C.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHCH(CH.sub.3)C.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NCH(CH.sub.3)C.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NCH(CH.sub.3)C.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NCH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NCH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NCH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NCH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHCH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHCH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CH(CH.sub.2).sub. 3 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CH(CH.sub.2).sub.3 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CH(CH.sub.2).sub.3 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CH(CH.sub.2).sub.3 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                N(CH.sub.2).sub.3 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                N(CH.sub.2).sub.3 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NCH.sub.2 CH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NCH.sub.2 CH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NCH.sub.2 CH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NCH.sub.2 CH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHCH.sub.2 CH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHCH.sub.2 CH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHCH(CH.sub.3)C.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHCH(CH.sub. 3)C.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHCH(CH.sub.3)C.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHCH(CH.sub.3)C.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NCH(CH.sub.3)C.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NCH(CH.sub.3)C.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NOCH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOCH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NOCH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NOCH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOCH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOCH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHO(CH.sub.2).sub.3 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHO(CH.sub.2).sub.3 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHO(CH.sub.2).sub.3 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHO(CH.sub.2).sub.3 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NO(CH.sub.2).sub.3 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NO(CH.sub.2).sub.3 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NOCH.sub.2 CH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOCH.sub.2 CH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NOCH.sub.2 CH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NOCH.sub.2 CH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOCH.sub.2 CH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOCH.sub.2 CH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHOCH(CH.sub.3)C.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOCH(CH.sub.3)C.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOCH(CH.sub.3)C.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHOCH(CH.sub.3)C.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOCH(CH.sub.3)C.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NOCH(CH.sub.3)C.sub.2 H.sub.5         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NOCH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOCH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NOCH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NOCH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOCH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOCH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHO(CH.sub.2).sub.3 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHO(CH.sub.2).sub.3 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHO(CH.sub.2).sub.3 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHO(CH.sub.2).sub.3 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NO(CH.sub.2).sub.3 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NO(CH.sub.2).sub.3 CH.sub.3         H     H   OCH.sub.3                        OCH.sub. 2 CF.sub.3                                NOCH.sub.2 CH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOCH.sub.2 CH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NOCH.sub.2 CH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NOCH.sub.2 CH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOCH.sub.2 CH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOCH.sub.2 CH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHOCH(CH.sub.3)C.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOCH(CH.sub.3)C.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOCH(CH.sub.3)C.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHOCH(CH.sub.3)C.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOCH(CH.sub.3)C.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NOCH(CH.sub.3)C.sub.2 H.sub.5         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NOC(CH.sub.3).sub.3         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOC(CH.sub.3).sub.3         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NOC(CH.sub.3).sub.3         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NOC(CH.sub.3).sub.3         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOC(CH.sub.3).sub.3         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOC(CH.sub.3).sub.3         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHOC(CH.sub.3).sub.3         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOC(CH.sub.3).sub.3         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NOC(CH.sub.3).sub.3         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NOC(CH.sub.3).sub.3         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOC(CH.sub.3).sub.3         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOC(CH.sub.3).sub.3         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHC(CH.sub.3).sub.3         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHC(CH.sub.3).sub.3         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHC(CH.sub.3).sub.3         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHC(CH.sub.3).sub.3         H     H   OCH.sub.3                        OCH.sub.2 CH.sub. 2 F                                NC(CH.sub.3).sub.3         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NC(CH.sub.3).sub.3         H     H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NC(CH.sub.3).sub.3         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NC(CH.sub.3).sub.3         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NC(CH.sub.3).sub.3         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NC(CH.sub.3).sub.3         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHC(CH.sub.3).sub.3         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHC(CH.sub.3).sub.3         H     H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHSO.sub.2 N(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                N   159-164 (d)SO.sub.2 N(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NSO.sub.2 N(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHSO.sub.2 N(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHSO.sub.2 N(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                N   152-156SO.sub.2 N(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NSO.sub.2 N(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHSO.sub.2 N(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHSO.sub.2 N(C.sub.3 H.sub.5).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHSO.sub.2 N(C.sub.3 H.sub.5).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHSO.sub.2 N(C.sub.3 H.sub.5).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(C.sub.3 H.sub.5).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NSO.sub.2 N(C.sub.3 H.sub.5).sub.2         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(C.sub.3 H.sub.5).sub.2         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NSO.sub.2 N(C.sub.3 H.sub.5).sub.2         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHSO.sub.2 N(C.sub.3 H.sub.5).sub.2         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHSO.sub.2 N(CH.sub.3)CH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3 )CH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NSO.sub.2 N(CH.sub.3)CH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHSO.sub.2 N(CH.sub.3)CH(CH.sub.3).sub.2         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHSO.sub.2 N(CH.sub.3)CH.sub.2 CH.sub.2 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHSO.sub.2 N(CH.sub.3)CH.sub.2 CH.sub.2 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHSO.sub.2 N(CH.sub.3)CH.sub.2 CH.sub.2 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3)CH.sub.2 CH.sub.2 CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NSO.sub.2 N(OCH.sub.3)CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(OCH.sub.3)CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NSO.sub.2 N(OCH.sub.3)CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHSO.sub.2 N(OCH.sub.3)CH.sub.3         H     H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHSO.sub.2 N(CH.sub.3).sub.2         5-OCH.sub.3               H   CH.sub.3                        OCH.sub. 2 CH.sub.2 F                                CHSO.sub.2 N(CH.sub.3).sub.2         5-OCH.sub.3               H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHSO.sub.2 N(CH.sub.3).sub.2         5-OCH.sub.3               H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3).sub.2         5-OCH.sub.3               H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NSO.sub.2 N(CH.sub.3)CH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3)CH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NSO.sub.2 N(CH.sub.3)CH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHSO.sub.2 N(CH.sub.3)CH(CH.sub.3).sub.2         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHSO.sub.2 N(CH.sub.3)CH.sub.2 CH.sub.2 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHSO.sub.2 N(CH.sub.3)CH.sub.2 CH.sub.2 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHSO.sub.2 N(CH.sub.3)CH.sub.2 CH.sub.2 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3)CH.sub.2 CH.sub.2 CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub. 2                                NSO.sub.2 N(OCH.sub.3)CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(OCH.sub.3)CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NSO.sub.2 N(OCH.sub.3)CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHSO.sub.2 N(OCH.sub.3)CH.sub.3         H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHSO.sub.2 N(CH.sub.3).sub.2         5-OCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHSO.sub.2 N(CH.sub.3).sub.2         5-OCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHSO.sub.2 N(CH.sub.3).sub.2         5-OCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3).sub.2         5-OCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NC.sub.2 H.sub.5         5-OCH.sub.3               H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NC.sub.2 H.sub.5         5-OCH.sub.3               H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NC.sub.2 H.sub.5         5-OCH.sub.3               H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NC.sub.2 H.sub.5         5-OCH.sub.3               H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHC.sub.2 H.sub.5         5-OCH.sub.3               H   CH.sub.3                        OCH.sub.2 CHF.sub. 2                                CHC.sub.2 H.sub.5         5-OCH.sub.3               H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHC.sub.2 H.sub.5         5-OCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NC.sub.2 H.sub.5         5-OCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NC.sub.2 H.sub.5         5-OCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NC.sub.2 H.sub.5         5-OCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHC.sub.2 H.sub.5         5-OCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHC.sub.2 H.sub.5         5-OCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHCH.sub.2 CH.sub.2 CH.sub.3         5-Cl  H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHCH.sub.2 CH.sub.2 CH.sub.3         5-Cl  H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHCH.sub.2 CH.sub.2 CH.sub.3         5-Cl  H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHCH.sub.2 CH.sub.2 CH.sub.3         5-Cl  H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NCH.sub.2 CH.sub.2 CH.sub.3         5-Cl  H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NCH.sub.2 CH.sub.2 CH.sub.3         5-Cl  H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NCH.sub.2 CH.sub.2 CH.sub.3         5-Cl  H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NCH.sub.2 CH.sub.2 CH.sub.3         5-Cl  H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NCH.sub.2 CH.sub.2 CH.sub.3         5-Cl  H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NCH.sub.2 CH.sub.2 CH.sub.3         5-Cl  H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHCH.sub.2 CH.sub.2 CH.sub.3         5-Cl  H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHCH.sub.2 CH.sub.2 CH.sub.3         5-Cl  H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHOC.sub.2 H.sub.5         5-OCH.sub.3               H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOC.sub.2 H.sub.5         5-OCH.sub.3               H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NOC.sub.2 H.sub.5         5-OCH.sub.3               H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NOC.sub.2 H.sub.5         5-OCH.sub.3               H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOC.sub.2 H.sub.5         5-OCH.sub.3               H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOC.sub.2 H.sub.5         5-OCH.sub.3               H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHOC.sub.2 H.sub.5         5-OCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOC.sub.2 H.sub.5         5-OCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NOC.sub.2 H.sub.5         5-OCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NOC.sub.2 H.sub.5         5-OCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOC.sub.2 H.sub.5         5-OCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOC.sub.2 H.sub.5         5-OCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-OCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-OCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-OCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-OCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-OCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-OCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-OCH.sub.3               H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-OCH.sub.3               H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-OCH.sub.3               H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-OCH.sub.3               H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-OCH.sub.3               H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-OCH.sub.3               H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHOC.sub.2 H.sub.5         5-Cl  H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOC.sub.2 H.sub.5         5-Cl  H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NOC.sub.2 H.sub.5         5-Cl  H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NOC.sub.2 H.sub.5         5-Cl  H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOC.sub.2 H.sub.5         5-Cl  H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOC.sub.2 H.sub.5         5-Cl  H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHOC.sub.2 H.sub.5         5-Cl  H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOC.sub.2 H.sub.5         5-Cl  H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NOC.sub.2 H.sub.5         5-Cl  H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NOC.sub.2 H.sub.5         5-Cl  H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOC.sub.2 H.sub.5         5-Cl  H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOC.sub.2 H.sub.5         5-Cl  H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-CF.sub.3               H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-CF.sub.3               H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-CF.sub.3               H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-CF.sub.3               H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-CF.sub.3               H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-CF.sub.3               H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-CF.sub.3               H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-CF.sub.3               H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-CF.sub.3               H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-CF.sub.3               H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-CF.sub.3               H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-CF.sub.3               H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHOC.sub.2 H.sub.5         5-SCH.sub.3               H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOC.sub.2 H.sub.5         5-SCH.sub.3               H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NOC.sub.2 H.sub.5         5-SCH.sub.3               H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NOC.sub.2 H.sub.5         5-SCH.sub.3               H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOC.sub.2 H.sub.5         5-SCH.sub.3               H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOC.sub.2 H.sub.5         5-SCH.sub.3               H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHOC.sub.2 H.sub.5         5-SCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOC.sub.2 H.sub.5         5-SCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NOC.sub.2 H.sub.5         5-SCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NOC.sub.2 H.sub.5         5-SCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOC.sub.2 H.sub.5         5-SCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOC.sub.2 H.sub.5         5-SCH.sub.3               H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHOC.sub.2 H.sub.5         5-Br  H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOC.sub.2 H.sub.5         5-Br  H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOC.sub.2 H.sub.5         5-Br  H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHOC.sub.2 H.sub.5         5-Br  H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOC.sub.2 H.sub.5         5-Br  H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NOC.sub.2 H.sub.5         5-Br  H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NOC.sub.2 H.sub.5         5-Br  H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOC.sub.2 H.sub.5         5-Br  H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NOC.sub.2 H.sub.5         5-Br  H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NOC.sub.2 H.sub.5         5-Br  H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOC.sub.2 H.sub.5         5-Br  H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOC.sub.2 H.sub.5         5-Br  H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHOC.sub.2 H.sub.5         5-F   H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOC.sub.2 H.sub.5         5-F   H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NOC.sub.2 H.sub.5         5-F   H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NOC.sub.2 H.sub.5         5-F   H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOC.sub.2 H.sub.5         5-F   H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOC.sub.2 H.sub.5         5-F   H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHOC.sub.2 H.sub.5         5-F   H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOC.sub.2 H.sub.5         5-F   H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NOC.sub.2 H.sub.5         5-F   H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NOC.sub.2 H.sub.5         5-F   H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOC.sub.2 H.sub.5         5-F   H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOC.sub.2 H.sub.5         5-F   H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-F   H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-F   H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-F   H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-F   H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-F   H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-F   H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-F   H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-F   H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-F   H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-F   H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-F   H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-F   H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHOC.sub.2 H.sub.5         5-CH.sub.3               H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOC.sub.2 H.sub.5         5-CH.sub.3               H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NOC.sub.2 H.sub.5         5-CH.sub.3               H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NOC.sub.2 H.sub.5         5-CH.sub.3               H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOC.sub.2 H.sub.5         5-CH.sub.3               H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOC.sub.2 H.sub.5         5-CH.sub.3               H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHOC.sub.2 H.sub.5         5-CH.sub.3               H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOC.sub.2 H.sub.5         5-CH.sub.3               H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NOC.sub.2 H.sub.5         5-CH.sub.3               H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NOC.sub.2 H.sub.5         5-CH.sub.3               H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOC.sub.2 H.sub.5         5-CH.sub.3               H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOC.sub.2 H.sub.5         5-CH.sub.3               H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-CH.sub.3               H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-CH.sub.3               H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-CH.sub.3               H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-CH.sub.3               H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-CH.sub.3               H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-CH.sub.3               H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-CH.sub.3               H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-CH.sub.3               H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-CH.sub.3               H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NOCH.sub.2 CH.sub.2 CH.sub.3         5-CH.sub.3               H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-CH.sub.3               H   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHOCH.sub.2 CH.sub.2 CH.sub.3         5-CH.sub.3               H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHOC.sub.2 H.sub.5         3-Cl  H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NOC.sub.2 H.sub.5         3-Cl  H   CH.sub.3                        OCH.sub.2 CF.sub.3                                NOC.sub.2 H.sub.5         3-Cl  H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHOC.sub.2 H.sub.5         3-Cl  H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHC.sub.2 H.sub.5         6-Cl  H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHC.sub.2 H.sub.5         6-Cl  H   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHC.sub.2 H.sub.5         6-Cl  H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NC.sub.2 H.sub.5         6-Cl  H   OCH.sub.3                        OCH.sub.2 CF.sub.3                                N ##STR21##    H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                N ##STR22##    H     H   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                N ##STR23##    H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                N ##STR24##    H     H   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CH ##STR25##    H     H   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHC.sub.2 H.sub.5         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NC.sub.2 H.sub.5         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NC.sub.2 H.sub.5         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CF.sub.3                                NC.sub.2 H.sub.5         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHC.sub.2 H.sub.5         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHC.sub.2 H.sub.5         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHC.sub.2 H.sub.5         H     CH.sub.3                   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NC.sub.2 H.sub.5         H     CH.sub.3                   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NC.sub.2 H.sub.5         H     CH.sub.3                   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NC.sub.2 H.sub.5         H     CH.sub.3                   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHC.sub.2 H.sub.5         H     CH.sub.3                   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHC.sub.2 H.sub.5         H     CH.sub.3                   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHCH.sub.2 CH.sub.2 CH.sub.3         H     CH.sub.3                   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHCH.sub.2 CH.sub.2 CH.sub.3         H     CH.sub.3                   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                CHCH.sub.2 CH.sub.2 CH.sub.3         H     CH.sub.3                   OCH.sub.3                        OCH.sub.2 CF.sub.3                                CHCH.sub.2 CH.sub.2 CH.sub.3         H     CH.sub.3                   OCH.sub.3                        OCH.sub.2 CH.sub.2 F                                NCH.sub.2 CH.sub.2 CH.sub.3         H     CH.sub.3                   OCH.sub.3                        OCH.sub.2 CHF.sub.2                                NCH.sub.2 CH.sub.2 CH.sub.3         H     CH.sub.3                   OCH.sub.3                        OCH.sub.2 CF.sub.3                                NCH.sub.2 CH.sub.2 CH.sub.3         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NCH.sub.2 CH.sub.2 CH.sub.3         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NCH.sub.2 CH.sub.2 CH.sub.3         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CF.sub.3                                NCH.sub.2 CH.sub.2 CH.sub.3         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHCH.sub.2 CH.sub.2 CH.sub.3         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHCH.sub.2 CH.sub.2 CH.sub.3         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHCH(CH.sub.3).sub.2         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NCH(CH.sub.3).sub.2         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NCH(CH.sub.3).sub.2         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CF.sub.3                                NCH(CH.sub.3).sub.2         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHCH(CH.sub.3).sub.2         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHCH(CH.sub.3).sub.2         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CF.sub.3                                CH(CH.sub.2).sub.3 CH.sub.3         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CH(CH.sub.2).sub.3 CH.sub.3         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CH(CH.sub.2).sub.3 CH.sub.3         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CF.sub.3                                CH(CH.sub.2).sub.3 CH.sub.3         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                N(CH.sub.2).sub.3 CH.sub.3         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CHF.sub.2                                N(CH.sub.2).sub.3 CH.sub.3         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CF.sub.3                                NCH.sub.2 CH(CH.sub.3).sub.2         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NCH.sub.2 CH(CH.sub.3).sub.2         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NCH.sub.2 CH(CH.sub.3).sub.2         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CF.sub.3                                NCH.sub.2 CH(CH.sub.3).sub.2         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHCH.sub.2 CH(CH.sub.3).sub.2         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHCH.sub.2 CH(CH.sub.3).sub.2         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHCH(CH.sub.3)C.sub.2 H.sub.5         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                CHCH(CH.sub.3)C.sub.2 H.sub.5         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CHF.sub.2                                CHCH(CH.sub.3)C.sub.2 H.sub.5         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CF.sub.3                                CHCH(CH.sub.3)C.sub.2 H.sub.5         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CH.sub.2 F                                NCH(CH.sub.3)C.sub.2 H.sub.5         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CHF.sub.2                                NCH(CH.sub.3)C.sub.2 H.sub.5         H     CH.sub.3                   CH.sub.3                        OCH.sub.2 CF.sub.3                                N__________________________________________________________________________ 
    
     
                       TABLE II______________________________________General Structure IIR.sub.3  R      X       Y         Z    m.p.(°C.)______________________________________H        H      CH.sub.3                   OCH.sub.2 CH.sub.2 F                             CHH        H      CH.sub.3                   OCH.sub.2 CF.sub.3                             CHH        H      CH.sub.3                   OCH.sub.2 CHF.sub.2                             CHH        H      OCH.sub.3                   OCH.sub.2 CHF.sub.2                             NH        H      OCH.sub.3                   OCH.sub.2 CF.sub.3                             NH        H      OCH.sub.3                   OCH.sub.2 CH.sub.2 F                             NF        H      OCH.sub.3                   OCH.sub.2 CF.sub.3                             NF        H      OCH.sub.3                   OCH.sub.2 CH.sub.2 F                             NF        H      CH.sub.3                   OCH.sub.2 CF.sub.3                             CHCl       H      CH.sub.3                   OCH.sub.2 CF.sub.3                             CHCl       H      CH.sub.3                   OCH.sub.2 CHF.sub.2                             CHCl       H      CH.sub.3                   OCH.sub.2 CH.sub.2 F                             CHCl       H      OCH.sub.3                   OCH.sub.2 CF.sub.3                             CHCl       H      OCH.sub.3                   OCH.sub.2 CH.sub.2 F                             CHCl       H      OCH.sub.3                   OCH.sub.2 CF.sub.3                             N    193-197(d)Cl       H      OCH.sub.3                   OCH.sub.2 CHF.sub.2                             NCl       H      OCH.sub.3                   OCH.sub.2 CH.sub.2 F                             NBr       H      CH.sub.3                   OCH.sub.2 CH.sub.2 F                             NBr       H      CH.sub.3                   OCH.sub.2 CF.sub.3                             NBr       H      CH.sub.3                   OCH.sub.2 CHF.sub.2                             NBr       H      OCH.sub.3                   OCH.sub.2 CHF.sub.2                             NBr       H      OCH.sub.3                   OCH.sub.2 CF.sub.3                             NBr       H      OCH.sub.3                   OCH.sub.2 CH.sub.2 F                             NOCH.sub.3    H      CH.sub.3                   OCH.sub.2 CH.sub.2 F                             CHOCH.sub.3    H      CH.sub.3                   OCH.sub.2 CF.sub.3                             CHOCH.sub.3    H      OCH.sub.3                   OCH.sub.2 CF.sub.3                             CHOCH.sub.3    H      OCH.sub.3                   OCH.sub.2 CF.sub.3                             NOCH.sub.3    H      OCH.sub.3                   OCH.sub.2 CH.sub.2 F                             NOCH.sub.3    H      OCH.sub.3                   OCH.sub.2 CHF.sub.2                             NCH.sub.3 H      CH.sub.3                   OCH.sub.2 CH.sub.2 F                             CHCH.sub.3 H      CH.sub.3                   OCH.sub.2 CF.sub.3                             CHCH.sub.3 H      OCH.sub.3                   OCH.sub.2 CF.sub.3                             CHCH.sub.3 H      OCH.sub.3                   OCH.sub.2 CF.sub.3                             NCH.sub.3 H      OCH.sub.3                   OCH.sub.2 CH.sub.2 F                             NCH.sub.3 H      OCH.sub.3                   OCH.sub.2 CHF.sub.2                             NSO.sub.2 N(CH.sub.3).sub.2    H      CH.sub.3                   OCH.sub.2 CF.sub.3                             CHSO.sub.2 N(CH.sub.3).sub.2    H      CH.sub.3                   OCH.sub.2 CH.sub.2 F                             CHSO.sub.2 N(CH.sub.3).sub.2    H      CH.sub.3                   OCH.sub.2 CH.sub.2 F                             NSO.sub.2 N(CH.sub.3).sub.2    H      CH.sub.3                   OCH.sub.2 CF.sub.3                             NSO.sub.2 N(CH.sub.3).sub.2    H      OCH.sub.3                   OCH.sub.2 CF.sub.3                             NSO.sub.2 N(CH.sub.3).sub.2    H      OCH.sub.3                   OCH.sub.2 CH.sub.2 F                             NSO.sub.2 N(CH.sub.3).sub.2    H      OCH.sub.3                   OCH.sub.2 CHF.sub.2                             NOSO.sub.2 CH.sub.3    H      CH.sub.3                   OCH.sub.2 CF.sub.3                             CHOSO.sub.2 CH.sub.3    H      CH.sub.3                   OCH.sub.2 CH.sub.2 F                             CHOSO.sub.2 CH.sub.3    H      OCH.sub.3                   OCH.sub.2 CH.sub.2 F                             CHOSO.sub.2 CH.sub.3    H      OCH.sub.3                   OCH.sub.2 CH.sub.2 F                             NOSO.sub.2 CH.sub.3    H      OCH.sub.3                   OCH.sub.2 CF.sub.3                             NOSO.sub.2 CH.sub.3    H      OCH.sub.3                   OCH.sub.2 CHF.sub.2                             NSCH.sub.3    H      OCH.sub.3                   OCH.sub.2 CF.sub.3                             N    115-118(d)SCH.sub.3    H      OCH.sub.3                   OCH.sub.2 CH.sub.2 F                             NSCH.sub.3    H      CH.sub.3                   OCH.sub.2 CH.sub.2 F                             CHSOCH.sub.3    H      CH.sub.3                   OCH.sub.2 CH.sub.2 F                             CHSOCH.sub.3    H      OCH.sub.3                   OCH.sub.2 CH.sub.2 F                             NSOCH.sub.3    H      OCH.sub.3                   OCH.sub.2 CF.sub.3                             NSO.sub.2 CH.sub.3    H      OCH.sub.3                   OCH.sub.2 CF.sub.3                             NSO.sub.2 CH.sub.3    H      OCH.sub.3                   OCH.sub.2 CH.sub.2 F                             NSO.sub.2 CH.sub.3    H      CH.sub.3                   OCH.sub.2 CH.sub.2 F                             CHCl       CH.sub.3           OCH.sub.3                   OCH.sub.2 CF.sub.3                             NCl       CH.sub.3           OCH.sub.3                   OCH.sub.2 CH.sub.2 F                             NCl       CH.sub.3           OCH.sub.3                   OCH.sub.2 CHF.sub.2                             NCl       CH.sub.3           CH.sub.3                   OCH.sub.2 CF.sub.3                             CHOCH.sub.3    H      CH.sub.3                   OCH.sub.2 CH.sub.2 F                             NOCH.sub.3    H      CH.sub.3                   OCH.sub.2 CHF.sub.2                             NOCH.sub.3    H      CH.sub.3                   OCH.sub.2 CF.sub.3                             NCH.sub.3 H      CH.sub.3                   OCH.sub.2 CH.sub.2 F                             NCH.sub.3 H      CH.sub.3                   OCH.sub.2 CHF.sub.2                             NCH.sub.3 H      CH.sub.3                   OCH.sub.2 CF.sub.3                             NCl       H      CH.sub.3                   OCH.sub.2 CH.sub.2 F                             NCl       H      CH.sub.3                   OCH.sub.2 CHF.sub.2                             NCl       H      CH.sub.3                   OCH.sub.2 CF.sub.3                             NSCH.sub.3    H      OCH.sub.3                   OCH.sub.2 CHF.sub.2                             NSCH.sub.3    H      CH.sub.3                   OCH.sub.2 CHF.sub. 2                             NSCH.sub.3    H      CH.sub.3                   OCH.sub.2 CF.sub.3                             NSCH.sub.3    H      CH.sub.3                   OCH.sub.2 CH.sub.2 F                             N______________________________________ 
    
     
                       TABLE III______________________________________General Structure III                                     m.p.R.sub.4       R     X       Y        Z    (°C.)______________________________________CH.sub.3      H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHCH.sub.3      H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NCH.sub.3      H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NCH.sub.3      H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NC.sub.2 H.sub.5         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHC.sub.2 H.sub.5         H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                CHC.sub.2 H.sub.5         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NC.sub.2 H.sub.5         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NC.sub.2 H.sub.5         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                Nn-C.sub.3 H.sub.7         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                Nn-C.sub.3 H.sub.7         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                Nn-C.sub.3 H.sub.7         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                Nn-C.sub.3 H.sub.7         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHF             H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHF             H     OCH.sub. 3                       OCH.sub.2 CF.sub.3                                NF             H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NCl            H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NCl            H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NCl            H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NCl            H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHCl            H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NBr            H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NBr            H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NBr            H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NBr            H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NNO.sub.2      H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHNO.sub.2      H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NNO.sub.2      H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NNO.sub.2      H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3).sub.2         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3).sub.2         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSO.sub.2 N(CH.sub.3).sub.2         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 N(CH.sub.3).sub.2         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSO.sub.2 N(C.sub. 2 H.sub.5).sub.2         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSO.sub.2 N(C.sub.2 H.sub.5).sub.2         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 N(C.sub.2 H.sub.5).sub.2         H     OCH.sub.3                       OCH.sub.2 CHF.sub.3                                NSO.sub.2 N(C.sub.2 H.sub.5).sub.2         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3)n-C.sub.3 H.sub.7         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3)n-C.sub.3 H.sub.7         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 N(CH.sub.3)n-C.sub.3 H.sub.7         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSO.sub.2 N(CH.sub.3)OCH.sub.3         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 N(CH.sub.3)OCH.sub.3         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3)OCH.sub.3         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSCH.sub.3     H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSCH.sub.3     H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSCH.sub.3     H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSOCH.sub.3    H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSOCH.sub.3    H     OCH.sub. 3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                CHSC.sub.2 H.sub.5         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSC.sub.2 H.sub.5         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSC.sub.2 H.sub.5         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 C.sub.2 H.sub.5         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 C.sub.2 H.sub.5         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 C.sub.2 H.sub.5         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSO.sub.2 CH(CH.sub.3).sub.2         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSO.sub.2 CH(CH.sub.3).sub.2         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 CH(CH.sub.3).sub.2         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSCH.sub.2 CH═CH.sub.3         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSCH.sub.2 CH═CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSCH.sub.2 CH═CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSCH.sub.2 CH═CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 CH.sub.2 CH═CH.sub.2         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 CH.sub.2 CH═CH.sub.2         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSO.sub.2 CH.sub.2 CH═CH.sub.2         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 CH.sub.2 CH═CH.sub.2         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHCH.sub.3      H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NCH.sub.3      H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                NCH.sub.3      H     CH.sub.3                       OCH.sub.2 CHF.sub.2                                NSCH.sub.3     H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSCH.sub.3     H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSCH.sub.3     H     CH.sub.3                       OCH.sub.2 CHF.sub.2                                NSCH.sub.3     H     CH.sub.3                       OCH.sub.2 CF.sub. 3                                NSOCH.sub.3    H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSOCH.sub.3    H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSOCH.sub.3    H     CH.sub.3                       OCH.sub.2 CHF.sub.2                                NSOCH.sub.3    H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSO.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CHF.sub.2                                NSO.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NSCH.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSCH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSCH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CHF.sub.2                                NSCH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NSOCH.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSOCH.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSOCH.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSOCH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSOCH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CHF.sub.2                                NSOCH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 CH.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSO.sub.2 CH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 CH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CHF.sub.2                                NSO.sub.2 CH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 N(CH.sub.3).sub.2         H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3).sub.2         H     CH.sub.3                       OCH.sub.2 CHF.sub.2                                N______________________________________ 
    
     
                       TABLE IV______________________________________General Structure IV                                     m.p.R.sub.4       R     X       Y        Z    (°C.)______________________________________CH.sub.3      H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHCH.sub.3      H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NCH.sub.3      H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NCH.sub.3      H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NC.sub.2 H.sub.5         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHC.sub.2 H.sub.5         H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                CHC.sub.2 H.sub.5         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NC.sub.2 H.sub.5         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NC.sub.2 H.sub.5         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                Nn-C.sub.3 H.sub.7         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                Nn-C.sub.3 H.sub.7         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                Nn-C.sub.3 H.sub.7         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                Nn-C.sub.3 H.sub.7         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHF             H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHF             H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NF             H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NCl            H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NCl            H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NCl            H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NCl            H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHCl            H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NBr            H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NBr            H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NBr            H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NBr            H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NNO.sub.2      H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHNO.sub.2      H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NNO.sub.2      H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NNO.sub.2      H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3).sub.2         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3).sub.2         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSO.sub.2 N(CH.sub.3).sub.2         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 N(CH.sub.3).sub.2         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSO.sub.2 N(C.sub.2 H.sub.5).sub.2         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSO.sub.2 N(C.sub.2 H.sub.5).sub.2         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 N(C.sub.2 H.sub.5).sub.2         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSO.sub.2 N(C.sub.2 H.sub.5).sub.2         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3)n-C.sub.3 H.sub.7         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3)n-C.sub.3 H.sub.7         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 N(CH.sub.3)n-C.sub.3 H.sub.7         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSO.sub.2 N(CH.sub.3)OCH.sub.3         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 N(CH.sub.3)OCH.sub.3         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3)OCH.sub.3         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSCH.sub.3     H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSCH.sub.3     H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSCH.sub.3     H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSOCH.sub.3    H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSOCH.sub.3    H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                CHSC.sub.2 H.sub.5         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSC.sub.2 H.sub.5         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSC.sub.2 H.sub.5         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 C.sub.2 H.sub.5         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 C.sub.2 H.sub.5         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 C.sub.2 H.sub.5         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSO.sub.2 CH(CH.sub.3).sub.2         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSO.sub.2 CH(CH.sub.3).sub.2         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 CH(CH.sub.3).sub.2         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub. 2 CH.sub.2 CH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSCH.sub.2 CH═CH.sub.3         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSCH.sub.2 CH═CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSCH.sub.2 CH═CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSCH.sub.2 CH═CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 CH.sub.2 CH═CH.sub.2         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 CH.sub.2 CH═CH.sub.2         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSO.sub.2 CH.sub.2 CH═CH.sub.2         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 CH.sub.2 CH═CH.sub.2         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHCH.sub.3      H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NCH.sub.3      H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                NCH.sub.3      H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSCH.sub.3     H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSCH.sub.3     H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSCH.sub.3     H     CH.sub.3                       OCH.sub.2 CHF.sub.2                                NSCH.sub.3     H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NSOCH.sub.3    H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSOCH.sub.3    H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSOCH.sub.3    H     CH.sub.3                       OCH.sub.2 CHF.sub.2                                NSOCH.sub.3    H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSO.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CHF.sub.2                                NSO.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NSCH.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSCH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSCH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CHF.sub.2                                NSCH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NSOCH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSOCH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CHF.sub.2                                NSOCH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NSOCH.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSOCH.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CHF.sub. 2                                NSOCH.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 CH.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSO.sub.2 CH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 CH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CHF.sub.2                                NSO.sub.2 CH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 N(CH.sub.3).sub.2         H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3).sub.2         H     CH.sub.3                       OCH.sub.2 CHF.sub.2                                NSO.sub.2 N(CH.sub.3).sub.2         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                N______________________________________ 
    
     
                       TABLE V______________________________________General Structure V                                     m.p.R.sub.4       R     X       Y        Z    (°C.)______________________________________CH.sub.3      H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHCH.sub.3      H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NCH.sub.3      H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NCH.sub.3      H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NC.sub.2 H.sub.5         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHC.sub.2 H.sub.5         H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                CHC.sub.2 H.sub.5         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NC.sub.2 H.sub.5         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NC.sub.2 H.sub.5         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                Nn-C.sub.3 H.sub.7         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                Nn-C.sub.3 H.sub.7         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                Nn-C.sub.3 H.sub.7         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                Nn-C.sub.3 H.sub.7         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHF             H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHF             H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NF             H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NCl            H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NCl            H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NCl            H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NCl            H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHCl            H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NBr            H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NBr            H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NBr            H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NBr            H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NNO.sub.2      H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHNO.sub.2      H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NNO.sub.2      H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NNO.sub.2      H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3).sub.2         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3).sub.2         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSO.sub.2 N(CH.sub.3).sub.2         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 N(CH.sub.3).sub.2         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSO.sub.2 N(C.sub.2 H.sub.5).sub.2         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSO.sub.2 N(C.sub.2 H.sub.5).sub.2         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 N(C.sub.2 H.sub.5).sub.2         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSO.sub.2 N(C.sub.2 H.sub.5).sub.2         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3)n-C.sub.3 H.sub.7         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3)n-C.sub.3 H.sub.7         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 N(CH.sub.3)n-C.sub.3 H.sub.7         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSO.sub.2 N(CH.sub.3)OCH.sub.3         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 N(CH.sub.3)OCH.sub.3         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3)OCH.sub.3         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSCH.sub.3     H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSCH.sub.3     H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSCH.sub.3     H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSOCH.sub.3    H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSOCH.sub.3    H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                CHSC.sub.2 H.sub.5         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSC.sub.2 H.sub.5         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSC.sub.2 H.sub.5         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 C.sub.2 H.sub.5         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 C.sub.2 H.sub.5         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 C.sub.2 H.sub.5         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSO.sub.2 CH(CH.sub.3).sub.2         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSO.sub.2 CH(CH.sub.3).sub.2         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 CH(CH.sub.3).sub.2         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub. 2 CH.sub.2 CH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSCH.sub.2 CH═CH.sub.3         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHSCH.sub.2 CH═CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSCH.sub.2 CH═CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSCH.sub.2 CH═CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 CH.sub.2 CH═CH.sub.2         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 CH.sub.2 CH═CH.sub.2         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSO.sub.2 CH.sub.2 CH═CH.sub.2         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 CH.sub.2 CH═CH.sub.2         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                CHCH.sub.3      H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NCH.sub.3      H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                NCH.sub.3      H     CH.sub.3                       OCH.sub.2 CHF.sub.2                                NSCH.sub.3     H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSCH.sub.3     H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSCH.sub.3     H     CH.sub.3                       OCH.sub.2 CHF.sub.2                                NSCH.sub.3     H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NSOCH.sub.3    H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSOCH.sub.3    H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSOCH.sub.3    H     CH.sub.3                       OCH.sub.2 CHF.sub.2                                NSOCH.sub.3    H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSO.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CHF.sub.2                                NSO.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NSCH.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSCH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSCH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CHF.sub.2                                NSCH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NSOCH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSOCH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CHF.sub.2                                NSOCH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NSOCH.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSOCH.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CHF.sub. 2                                NSOCH.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 CH.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CHF.sub.2                                NSO.sub.2 CH.sub.2 CH.sub.3         H     OCH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 CH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CHF.sub.2                                NSO.sub.2 CH.sub.2 CH.sub.3         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                NSO.sub.2 N(CH.sub.3).sub.2         H     CH.sub.3                       OCH.sub.2 CH.sub.2 F                                NSO.sub.2 N(CH.sub.3).sub.2         H     CH.sub.3                       OCH.sub.2 CHF.sub.2                                NSO.sub.2 N(CH.sub.3).sub.2         H     CH.sub.3                       OCH.sub.2 CF.sub.3                                N______________________________________ 
    
     
                                           TABLE VI__________________________________________________________________________General Structure VIR.sub.2R.sub.5     R.sub.6               R X   Y      Z  m.p.(°C.)__________________________________________________________________________H    CH.sub.3    H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            CHH    CH.sub.3    H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.3    H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.3    H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.3    H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.3    H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    C.sub.2 H.sub.5            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    C.sub.2 H.sub.5            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    C.sub.2 H.sub.5            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3).sub.2            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3).sub.2            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3).sub.2            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.2 CH.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.2 CH.sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.2 CH(CH.sub.3).sub.2            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.2 CH(CH.sub.3).sub.2            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH(CH.sub.3).sub.2            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)C.sub.2 H.sub.5            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)C.sub.2 H.sub.5            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)C.sub.2 H.sub.5            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.4 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    (CH.sub.2).sub.4 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.4 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)(CH.sub.2).sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)(CH.sub.2).sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)(CH.sub.2).sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            CHH    CH.sub.2 CH.sub.2 OCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.2 CH.sub.2 OCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 OCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub. 5            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CHF.sub.2   H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CHF.sub.2   H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CHF.sub.2   H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CF.sub.3    H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CF.sub.3    H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 F            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 F            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CF.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CF.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CCl.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CCl.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHCl.sub.2            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHCl.sub.2            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 Cl            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 Cl            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 Cl            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            CHH    (CH.sub.2).sub.4 Cl            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            CHH    (CH.sub.2).sub.4 Cl            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.4 Cl            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CH.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CH.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 Br            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 Br            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 Br            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 Br            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            N6-Cl CH.sub.3    H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            N6-Cl CH.sub.3    H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            N5-Cl CH.sub.3    H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            N5-OCH.sub.3CH.sub.3    H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            N5-Br CH.sub.3    H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.3    CH.sub.3               H CH.sub.3                     OCH.sub.2 CHF.sub.2                            CHH    CH.sub.3    CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.3    CH.sub.3               H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.3    CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.3    CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.3    CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    C.sub.2 H.sub.5            CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    C.sub.2 H.sub.5            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    C.sub.2 H.sub.5            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3).sub.2            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3).sub.2            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3).sub.2            CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.2 CH.sub.2 CH.sub.3            CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.2 CH.sub.2 CH.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 CH.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 CH.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 CH.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 CH.sub.3            CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.2 CH(CH.sub.3).sub.2            CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.2 CH(CH.sub.3).sub.2            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH(CH.sub.3).sub.2            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)C.sub.2 H.sub.5            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)C.sub.2 H.sub.5            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)C.sub.2 H.sub.5            CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.4 CH.sub.3            CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    (CH.sub.2).sub.4 CH.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.4 CH.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)(CH.sub.2).sub.2 CH.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)(CH.sub.2).sub.2 CH.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)(CH.sub.2).sub.2 CH.sub.3            CH.sub.3               H CH.sub.3                     OCH.sub.2 CHF.sub.2                            CHH    CH.sub.2 CH.sub.2 OCH.sub.3            CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.2 CH.sub.2 OCH.sub.3            CH.sub.3               H OCH.sub. 3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 OCH.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CHF.sub.2   CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CHF.sub.2   CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CHF.sub.2   CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CF.sub.3    CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CF.sub.3    CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 F            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 F            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CF.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CF.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CCl.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CCl.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 Cl            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 Cl            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHCl.sub.2            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHCl.sub.2            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 Cl            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 Cl            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 Cl            CH.sub.3               H CH.sub.3                     OCH.sub.2 CHF.sub.2                            CHH    (CH.sub.2).sub.4 Cl            CH.sub.3               H CH.sub.3                     OCH.sub.2 CHF.sub.2                            CHH    (CH.sub.2).sub.4 Cl            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.4 Cl            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CH.sub.2 Cl            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CH.sub.2 Cl            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 Br            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 Br            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 Br            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 Br            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            N6-Cl CH.sub.3    CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            N6-Cl CH.sub.3    CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            N5-Cl CH.sub.3    CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            N5-OCH.sub.3CH.sub.3    CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            N5-Br CH.sub.3    CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            N5-Cl CH.sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            N5-Cl CH.sub.2 CH.sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            N5-Cl CH(CH.sub.3).sub.2            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            N5-Cl CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            N5-Cl CH.sub.2 CH(CH.sub.3).sub.2            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            N5-Cl CH(CH.sub.3)C.sub.2 H.sub.5            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            N5-Cl (CH.sub.2).sub.4 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            N5-Cl CH.sub.2 CH.sub.2 OCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            N5-Cl CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            N5-Cl CH.sub.2 CH.sub.2 CH.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    H           H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    H           H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    H           H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    H           H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3).sub.2            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3).sub.2            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH(CH.sub.3).sub.2            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH(CH.sub.3).sub.2            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)C.sub.2 H.sub.5            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 OCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 OCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CHF.sub.2   H  H CH.sub.3                     OCH.sub.2 CH.sub.2                            NH    CHF.sub.2   H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CF.sub.3    H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CF.sub.3    H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 F            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 F            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CF.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CF.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHCl.sub.2            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHCl.sub.2            H  H CH.sub. 3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CCl.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CCl.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 Cl            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 Cl            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)CH.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CH.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.4 Cl            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.4 Cl            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.4 F            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.4 F            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.4 F            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.4 F            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 Br            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 Br            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 Br            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 Br            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.4 Br            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.4 Br            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.4 Br            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.4 Br            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 F            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 F            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 F            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 F            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHF.sub.2            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHF.sub.2            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHF.sub.2            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHF.sub.2            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 F  H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 F  H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 F  H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 F  H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 (CH.sub.3)CH.sub.2 Br            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 (CH.sub.3)CH.sub.2 Br            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 (CH.sub.3)CH.sub.2 Br            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 (CH.sub.3)CH.sub.2 Br            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 (CH.sub.3)CH.sub.2 F            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 (CH.sub.3)CH.sub.2 F            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 (CH.sub.3)CH.sub.2 F            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 (CH.sub.3)CH.sub.2 F            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHClCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHClCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHClCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHClCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHClCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHBrCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHBrCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHBrCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHBrCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHFCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHFCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHFCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHFCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.2 Cl).sub.2            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.2 Cl).sub.2            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.2 Cl).sub.2            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.2 Cl).sub.2            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.2 F).sub.2            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.2 F).sub.2            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.2 F).sub.2            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.2 F).sub.2            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)CCl.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CCl.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)CCl.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CCl.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 CHClCH.sub.3            H  H CH.sub. 3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 CHClCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 CHClCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 CHClCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 CHBrCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 CHBrCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 CHBrCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 CHBrCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 CHFCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 CHFCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 CHFCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 CHFCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHlCH.sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub. 2 CH.sub.2 F                            NH    CH.sub.2 CHlCH.sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHlCH.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHlCH.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHBrCH.sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHBrCH.sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHBrCH.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHBrCH.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHFCH.sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHFCH.sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHFCH.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHFCH.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)CHClCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CHClCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)CHClCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CHClCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)CHBrCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CHBrCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)CHBrCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CHBrCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)CHFCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CHFCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)CHFCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CHFCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CCl.sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CCl.sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CCl.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CCl.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Br            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Br            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Br            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Br            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 F            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 F            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 F            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 F            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CF.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CF.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CF.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CF.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CHCl.sub.2)CH.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CHCl.sub.2)CH.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CHCl.sub.2)CH.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CHCl.sub.2)CH.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CHCl.sub.2)CH.sub.2 F            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CHCl.sub.2)CH.sub.2 F            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CHCl.sub.2)CH.sub.2 F            H  H OCH.sub. 3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CHCl.sub.2)CH.sub.2 F            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.2 Cl)CH.sub.2 CH.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.2 Cl)CH.sub.2 CH.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.2 Cl)CH.sub.2 CH.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.2 Cl)CH.sub.2 CH.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 Br H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 Br H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 Br H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 BR H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 Cl H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 Cl H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 Cl H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 Cl H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CHCl.sub.2  H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CHCl.sub.2  H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CHCl.sub.2  H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CHCl.sub.2  H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CCl.sub.2   H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CCl.sub.3   H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CCl.sub.3   H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CCl.sub.3   H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            N__________________________________________________________________________ 
    
     
                                           TABLE VIa__________________________________________________________________________General Structure VIaR.sub.2R.sub.5     R.sub.6              R X   Y      Z  m.p. (°C.)__________________________________________________________________________H    CH.sub.3    H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           CHH    CH.sub.3    H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           CHH    CH.sub.3    H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.3    H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.3    H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.3    H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    C.sub.2 H.sub.5            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           CHH    C.sub.2 H.sub.5            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    C.sub.2 H.sub.5            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CH.sub.3).sub.2            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CH.sub.3).sub.2            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH(CH.sub.3).sub.2            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           CHH    CH.sub.2 CH.sub.2 CH.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           CHH    CH.sub.2 CH.sub.2 CH.sub.3            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH.sub.2 CH.sub.3            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    (CH.sub.2).sub.3 CH.sub.3            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    (CH.sub.2).sub.3 CH.sub.3            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    (CH.sub.2).sub.3 CH.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           CHH    CH.sub.2 CH(CH.sub.3).sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           CHH    CH.sub.2 CH(CH.sub.3).sub.3            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH(CH.sub.3).sub.3            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CH.sub.3)C.sub.2 H.sub.5            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CH.sub.3)C.sub.2 H.sub.5            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH(CH.sub.3)C.sub.2 H.sub.5            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    (CH.sub.2).sub.4 CH.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           CHH    (CH.sub.2).sub.4 CH.sub.3            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    (CH.sub.2).sub.4 CH.sub.3            H H OH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CH.sub.3)(CH.sub.2).sub.2 CH.sub.3            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CH.sub.3)(CH.sub.2).sub.2 CH.sub.3            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH(CH.sub.3)(CH.sub.2).sub.2 CH.sub.3            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           CHH    CH.sub.2 CH.sub.2 OCH.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           CHH    CH.sub.2 CH.sub.2 OCH.sub.3            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH.sub.2 OCH.sub.3            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           CHH    CHF.sub.2   H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           CHH    CHF.sub.2   H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CHF.sub.2   H H OH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CF.sub.3    H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CF.sub.3    H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH.sub.2 F            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH.sub.2 F            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CF.sub.3            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CF.sub.3            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CCl.sub.3            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CCl.sub.3            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH.sub.2 Cl            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH.sub.2 Cl            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CHCl.sub.2            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CHCl.sub.2            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    (CH.sub.2).sub.3 Cl            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    (CH.sub.2).sub.3 Cl            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    (CH.sub.2).sub.3 Cl            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           CHH    (CH.sub.2).sub.4 Cl            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           CHH    (CH.sub.2).sub.4 Cl            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    (CH.sub.2).sub.4 Cl            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    (CH(CH.sub.3)CH.sub.2 Cl            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    (CH(CH.sub.3)CH.sub.2 Cl            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH.sub.2 Br            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH.sub.2 Br            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    (CH.sub.2).sub.3 Br            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    (CH.sub.2).sub.3 Br            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           N5-Cl CH.sub.3    H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           N5-Cl CH.sub.3    H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           N6-Cl CH.sub.3    H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           N6-OCH.sub.3CH.sub.3    H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           N6-Br CH.sub.3    H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    H           H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    H           H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    H           H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    H           H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH.sub.3            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CH.sub.3).sub.2            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH(CH.sub.3).sub.2            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH.sub.2 CH.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH.sub.2 CH.sub. 3            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    (CH.sub.2).sub.3 CH.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    (CH.sub.2).sub.3 CH.sub.3            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH(CH.sub.3).sub.2            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH(CH.sub.3).sub.2            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CH.sub.3)C.sub.2 H.sub.5            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH.sub.2 OCH.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH.sub.2 OCH.sub.3            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CHF.sub.2   H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CHF.sub.2   H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CF.sub.3    H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CF.sub.3    H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH.sub.2 F            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH.sub.2 F            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CF.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CF.sub.3            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH.sub.2 Cl            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH.sub.2 Cl            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CHCl.sub.2            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CHCl.sub.2            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CCl.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CCl.sub.3            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    (CH.sub.2).sub.3 Cl            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    (CH.sub.2).sub.3 Cl            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CH.sub.3)CH.sub.2 Cl            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH(CH.sub.3)CH.sub.2 Cl            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    (CH.sub.2).sub.4 Cl            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    (CH.sub.2).sub.4 Cl            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    (CH.sub.2).sub.4 F            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    (CH.sub.2).sub.4 F            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    (CH.sub.2).sub.4 F            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    (CH.sub.2).sub.4 F            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH.sub.2 Br            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH.sub.2 Br            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    (CH.sub.2).sub.3 Br            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    (CH.sub.2).sub.3 Br            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    (CH.sub.2).sub.4 Br            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    (CH.sub.2).sub.4 Br            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    (CH.sub.2).sub.4 Br            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    (CH.sub.2).sub.4 Br            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    (CH.sub.2).sub.3 F            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    (CH.sub.2).sub.3 F            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    (CH.sub.2).sub.3 F            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    (CH.sub.2).sub.3 F            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CHF.sub.2            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CHF.sub.2            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CHF.sub.2            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CHF.sub.2            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 F  H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 F  H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 F  H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 F  H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 (CH.sub.3)CH.sub.2 Br            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 (CH.sub.3)CH.sub.2 Br            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 (CH.sub.3)CH.sub.2 Br            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 (CH.sub.3)CH.sub.2 Br            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 (CH.sub.3)CH.sub.2 F            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 (CH.sub.3)CH.sub.2 F            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 (CH.sub.3)CH.sub.2 F            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 (CH.sub.3)CH.sub.2 F            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CHClCH.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CHClCH.sub.3            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CHClCH.sub.3            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub. 2 CHClCH.sub.3            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CHBrCH.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CHBrCH.sub.3            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CHBrCH.sub.3            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CHBrCH.sub.3            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CHFCH.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CHFCH.sub.3            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CHFCH.sub.3            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CHFCH.sub.3            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CH.sub.2 Cl).sub.2            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH(CH.sub.2 Cl).sub.2            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CH.sub.2 Cl).sub.2            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH(CH.sub.2 Cl).sub.2            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CH.sub.2 F).sub.2            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH(CH.sub.2 F).sub.2            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CH.sub.2 F).sub.2            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH(CH.sub.2 F).sub.2            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CH.sub.3)CCl.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH(CH.sub.3)CCl.sub.3            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CH.sub.3)CCl.sub.3            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH(CH.sub.3)CCl.sub.3            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH.sub.2 CHClCH.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH.sub.2 CHClCH.sub.3            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH.sub.2 CHClCH.sub.3            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH.sub.2 CHClCH.sub.3            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH.sub.2 CHBrCH.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH.sub.2 CHBrCH.sub.3            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH.sub.2 CHBrCH.sub.3            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH.sub.2 CHBrCH.sub.3            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH.sub.2 CHFCH.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH.sub.2 CHFCH.sub.3            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH.sub.2 CHFCH.sub.3            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH.sub.2 CHFCH.sub.3            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CHClCH.sub.2 CH.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CHClCH.sub.2 CH.sub.3            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CHClCH.sub.2 CH.sub.3            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CHClCH.sub.2 CH.sub.3            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CHBrCH.sub.2 CH.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CHBrCH.sub.2 CH.sub.3            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CHBrCH.sub.2 CH.sub.3            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CHBrCH.sub.2 CH.sub.3            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CHFCH.sub.2 CH.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CHFCH.sub.2 CH.sub.3            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CHFCH.sub.2 CH.sub.3            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CHFCH.sub.2 CH.sub.3            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CH.sub.3)CHClCH.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH(CH.sub.3)CHClCH.sub.3            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CH.sub.3)CHClCH.sub.3            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH(CH.sub.3)CHClCH.sub.3            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CH.sub.3)CHBrCH.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH(CH.sub.3)CHBrCH.sub.3            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CH.sub.3)CHBrCH.sub.3            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH(CH.sub.3)CHBrCH.sub.3            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CH.sub.3)CHFCH.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH(CH.sub.3)CHFCH.sub.3            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CH.sub.3)CHFCH.sub.3            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH(CH.sub.3)CHFCH.sub.3            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CCl.sub.2 CH.sub.3            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CCl.sub.2 CH.sub.3            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CCl.sub.2 CH.sub.3            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CCl.sub.2 CH.sub.3            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Cl            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Cl            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Cl            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Cl            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Br            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Br            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Br            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Br            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 F            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 F            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 F            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 F            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CF.sub.2 Cl            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CF.sub.2 Cl            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 CF.sub.2 Cl            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 CF.sub.2 Cl            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CHCl.sub.2)CH.sub.2 Cl            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH(CHCl.sub.2)CH.sub.2 Cl            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CHCl.sub.2)CH.sub.2 Cl            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH(CHCl.sub.2)CH.sub.2 Cl            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CHCl.sub.2)CH.sub.2 F            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH(CHCl.sub.2)CH.sub.2 F            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CHCl.sub.2)CH.sub.2 F            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH(CHCl.sub.2)CH.sub.2 F            H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CH.sub.2 Cl)CH.sub.2 CH.sub.2 Cl            H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH(CH.sub.2 Cl)CH.sub.2 CH.sub.2 Cl            H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH(CH.sub.2 Cl)CH.sub.2 CH.sub.2 Cl            H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH(CH.sub.2 Cl)CH.sub.2 CH.sub.2 Cl            H H OCH.sub.3                    OCH.sub. 2 CHF.sub.2                           NH    CH.sub.2 Br H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 Br H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 Br H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 Br H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 Cl H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 Cl H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CH.sub.2 Cl H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CH.sub.2 Cl H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CHCl.sub.2  H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CHCl.sub.2  H H CH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CHCl.sub.2  H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CHCl.sub.2  H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           NH    CCl.sub.3   H H CH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CCl.sub.3   H H CH.sub.3                    OCH.sub.2 CFH.sub.2                           NH    CCl.sub.3   H H OCH.sub.3                    OCH.sub.2 CH.sub.2 F                           NH    CCl.sub.3   H H OCH.sub.3                    OCH.sub.2 CHF.sub.2                           N__________________________________________________________________________ 
    
     
                                           TABLE VII__________________________________________________________________________General Structure VIIR.sub.2R.sub.5     R X   Y      Z  m.p. (°C.)__________________________________________________________________________H    CH.sub.3    H CH.sub.3                  OCH.sub.2 CHF.sub.2                         CHH    CH.sub.3    H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         CHH    CH.sub.3    H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.3    H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.3    H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.3    H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    C.sub.2 H.sub.5            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         CHH    C.sub.2 H.sub.5            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    C.sub.2 H.sub.5            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.3).sub.2            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.3).sub.2            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.3).sub.2            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         CHH    CH.sub.2 CH.sub.2 CH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         CHH    CH.sub.2 CH.sub.2 CH.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH.sub.2 CH.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    (CH.sub.2).sub.3 CH.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    (CH.sub.2).sub.3 CH.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    (CH.sub.2).sub.3 CH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         CHH    CH.sub.2 CH(CH.sub.3).sub.2            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         CHH    CH.sub.2 CH(CH.sub.3).sub.2            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH(CH.sub.3).sub.2            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.3)C.sub.2 H.sub.5            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.3)C.sub.2 H.sub.5            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.3)C.sub.2 H.sub.5            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    (CH.sub.2).sub.4 CH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         CHH    (CH.sub.2).sub.4 CH.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    (CH.sub.2).sub.4 CH.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.3)(CH.sub.2).sub.2 CH.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.3)(CH.sub.2).sub.2 CH.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.3)(CH.sub.2).sub.2 CH.sub.3            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         CHH    CH.sub.2 CH.sub.2 OCH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         CHH    CH.sub.2 CH.sub.2 OCH.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH.sub.2 OCH.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         CHH    CHF.sub.2   H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         CHH    CHF.sub.2   H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CHF.sub.2   H OCH.sub. 3                  OCH.sub.2 CHF.sub.2                         NH    CF.sub.3    H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CF.sub.3    H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH.sub.2 F            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH.sub.2 F            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CF.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CF.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CCl.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CCl.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.2 Cl            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.2 Cl            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CHCl.sub.2            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CHCl.sub.2            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    (CH.sub.2).sub.3 Cl            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    (CH.sub.2).sub.3 Cl            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    (CH.sub.2).sub.3 Cl            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         CHH    (CH.sub.2).sub.4 Cl            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         CHH    (CH.sub.2).sub.4 Cl            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    (CH.sub.2).sub.4 Cl            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.3)CH.sub.2 Cl            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.3)CH.sub.2 Cl            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.2 Br            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.2 Br            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    (CH.sub.2).sub.3 Br            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    (CH.sub.2).sub.3 Br            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         N5-Cl CH.sub.3    H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         N5-Cl CH.sub.3    H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         N6-Cl CH.sub.3    H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         N6-OCH.sub.3CH.sub.3    H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         N6-Br CH.sub.3    H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.3    H CH.sub.3                  OCH.sub.2 CHF.sub.2                         CHH    CH.sub.3    H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         CHH    CH.sub.3    H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.3    H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.3    H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.3    H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    C.sub.2 H.sub.5            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         CHH    C.sub.2 H.sub.5            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    C.sub.2 H.sub.5            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.3).sub.2            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.3).sub.2            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.3).sub.2            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         CHH    CH.sub.2 CH.sub.2 CH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         CHH    CH.sub.2 CH.sub.2 CH.sub. 3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH.sub.2 CH.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    (CH.sub.2).sub.3 CH.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    (CH.sub.2).sub.3 CH.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    (CH.sub.2).sub.3 CH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         CHH    CH.sub.2 CH(CH.sub.3).sub.2            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         CHH    CH.sub.2 CH(CH.sub.3).sub.2            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH(CH.sub.3).sub.2            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.3)C.sub.2 H.sub.5            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.3)C.sub.2 H.sub.5            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.3)C.sub.2 H.sub.5            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    (CH.sub.2).sub.4 CH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    (CH.sub.2).sub.4 CH.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    (CH.sub. 2).sub.4 CH.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.3)(CH.sub.2).sub.2 CH.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.3)(CH.sub.2).sub.2 CH.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.3)(CH.sub.2).sub.2 CH.sub.3            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         CHH    CH.sub.2 CH.sub.2 OCH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         CHH    CH.sub.2 CH.sub.2 OCH.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH.sub.2 OCH.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         CHH    CHF.sub.2   H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         CHH    CHF.sub.2   H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CHF.sub.2   H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CF.sub.3    H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CF.sub.3    H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH.sub.2 F            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH.sub.2 F            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CF.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CF.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CCl.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CCl.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.2 Cl            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.2 Cl            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CHCl.sub.2            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CHCl.sub.2            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    (CH.sub.2).sub.3 Cl            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    (CH.sub.2).sub.3 Cl            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    (CH.sub.2).sub.3 Cl            H CH.sub.3                  OCH.sub. 2 CHF.sub.2                         CHH    (CH.sub.2).sub.4 Cl            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         CHH    (CH.sub.2).sub.4 Cl            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    (CH.sub.2).sub.4 Cl            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.3)CH.sub.2 Cl            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.3)CH.sub.2 Cl            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.2 Br            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.2 Br            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    (CH.sub.2).sub.3 Br            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    (CH.sub.2).sub.3 Br            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         N5-Cl CH.sub.3    H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         N5-Cl CH.sub.3    H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         N6-Cl CH.sub.3    H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         N6-OCH.sub.3CH.sub.3    H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         N6-Br CH.sub.3    H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    H           H CH.sub.3                  OCH.sub. 2 CH.sub.2 F                         NH    H           H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    H           H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    H           H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH.sub.3            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.3).sub.2            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.3).sub.2            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.2 CH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH.sub.2 CH.sub.3            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    (CH.sub.2).sub.3 CH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    (CH.sub.2).sub.3 CH.sub.3            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH(CH.sub.3).sub.2            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH(CH.sub.3).sub.2            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.3)C.sub.2 H.sub.5            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub. 2 CH.sub.2 OCH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH.sub.2 OCH.sub.3            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CHF.sub.2   H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CHF.sub.2   H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CF.sub.3    H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CF.sub.3    H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.2 F            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH.sub.2 F            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CF.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CF.sub.3            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.2 Cl            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH.sub.2 Cl            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CHCl.sub.2            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CHCl.sub.2            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CCl.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CCl.sub.3            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    (CH.sub.2).sub.3 Cl            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    (CH.sub.2).sub.3 Cl            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.3)CH.sub.2 Cl            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.3)CH.sub.2 Cl            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    (CH.sub.2).sub.4 Cl            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    (CH.sub.2).sub.4 Cl            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    (CH.sub.2).sub.4 F            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    (CH.sub.2).sub.4 F            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    (CH.sub.2).sub.4 F            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    (CH.sub.2).sub.4 F            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.2 Br            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH.sub.2 Br            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    (CH.sub.2).sub.3 Br            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    (CH.sub.2).sub.3 Br            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    (CH.sub.2).sub.4 Br            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    (CH.sub.2).sub.4 Br            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    (CH.sub.2).sub.4 Br            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    (CH.sub.2).sub.4 Br            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    (CH.sub.2).sub.3 F            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    (CH.sub.2).sub.3 F            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    (CH.sub.2).sub.3 F            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    (CH.sub.2).sub.3 F            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CHF.sub.2            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CHF.sub.2            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CHF.sub.2            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CHF.sub.2            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 F  H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 F  H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 F  H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 F  H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 (CH.sub.3)CH.sub.2 Br            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 (CH.sub.3)CH.sub.2 Br            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 (CH.sub.3)CH.sub.2 Br            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 (CH.sub.3)CH.sub.2 Br            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 (CH.sub.3)CH.sub.2 F            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 (CH.sub.3)CH.sub.2 F            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 (CH.sub.3)CH.sub.2 F            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 (CH.sub.3)CH.sub.2 F            H OCH.sub.3                  OCH.sub. 2 CHF.sub.2                         NH    CH.sub.2 CHClCH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CHClCH.sub.3            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CHClCH.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CHClCH.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CHBrCH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CHBrCH.sub.3            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CHBrCH.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CHBrCH.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CHFCH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CHFCH.sub.3            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CHFCH.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CHFCH.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.2 Cl).sub.2            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.2 Cl).sub.2            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.2 Cl).sub.2            H OCH.sub. 3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.2 Cl).sub.2            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.2 F).sub.2            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.2 F).sub.2            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.2 F).sub.2            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.2 F).sub.2            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.3)CCl.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.3)CCl.sub.3            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.3)CCl.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.3)CCl.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.2 CHClCH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH.sub.2 CHClCH.sub.3            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.2 CHClCH.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH.sub.2 CHClCH.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.2 CHBrCH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH.sub.2 CHBrCH.sub.3            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.2 CHBrCH.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH.sub.2 CHBrCH.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.2 CHFCH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH.sub.2 CHFCH.sub.3            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH.sub.2 CHFCH.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH.sub.2 CHFCH.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CHClCH.sub.2 CH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CHClCH.sub.2 CH.sub.3            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CHClCH.sub.2 CH.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CHClCH.sub.2 CH.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CHBrCH.sub.2 CH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CHBrCH.sub.2 CH.sub.3            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CHBrCH.sub.2 CH.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CHBrCH.sub.2 CH.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CHFCH.sub.2 CH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CHFCH.sub.2 CH.sub.3            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CHFCH.sub.2 CH.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CHFCH.sub.2 CH.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.3)CHClCH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.3)CHClCH.sub.3            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.3)CHClCH.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.3)CHClCH.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.3)CHBrCH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.3)CHBrCH.sub.3            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.3)CHBrCH.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.3)CHBrCH.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.3)CHFCH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.3)CHFCH.sub.3            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.3)CHFCH.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.3)CHFCH.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CCl.sub.2 CH.sub.3            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CCl.sub.2 CH.sub.3            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CCl.sub.2 CH.sub.3            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CCl.sub.2 CH.sub.3            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Cl            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Cl            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Cl            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Cl            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Br            H CH.sub. 3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Br            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Br            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Br            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 F            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 F            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 F            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 F            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CF.sub.2 Cl            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CF.sub.2 Cl            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 CF.sub.2 Cl            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 CF.sub.2 Cl            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CHCl.sub.2)CH.sub.2 Cl            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CHCl.sub.2)CH.sub.2 Cl            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CHCl.sub.2)CH.sub.2 Cl            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CHCl.sub.2)CH.sub.2 Cl            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CHCl.sub.2)CH.sub.2 F            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CHCl.sub.2)CH.sub.2 F            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CHCl.sub.2)CH.sub.2 F            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CHCl.sub.2)CH.sub.2 F            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.2 Cl)CH.sub.2 CH.sub.2 Cl            H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.2 Cl)CH.sub.2 CH.sub.2 Cl            H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH(CH.sub.2 Cl)CH.sub.2 CH.sub.2 Cl            H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH(CH.sub.2 Cl)CH.sub.2 CH.sub.2 Cl            H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 Br H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 Br H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 Br H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 Br H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 Cl H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 Cl H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CH.sub.2 Cl H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CH.sub.2 Cl H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CHCl.sub.2  H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CHCl.sub.2  H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CHCl.sub.2  H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CHCl.sub.2  H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CCl.sub.3   H CH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CCl.sub.3   H CH.sub.3                  OCH.sub.2 CHF.sub.2                         NH    CCl.sub.3   H OCH.sub.3                  OCH.sub.2 CH.sub.2 F                         NH    CCl.sub.3   H OCH.sub.3                  OCH.sub.2 CHF.sub.2                         N__________________________________________________________________________ 
    
     
                                           TABLE VIII__________________________________________________________________________General Structure VIIIR.sub.2R.sub.5     R.sub.7               R X   Y      X  m.p. (°C.)__________________________________________________________________________H    CH.sub.3    H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            CHH    CH.sub.3    H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.3    H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.3    H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.3    H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.3    H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    C.sub.2 H.sub.5            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    C.sub.2 H.sub.5            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    C.sub.2 H.sub.5            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3).sub.2            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3).sub.2            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3).sub.2            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.2 CH.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.2 CH.sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.2 CH(CH.sub.3).sub.2            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.2 CH(CH.sub.3).sub.2            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH(CH.sub.3).sub.2            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)C.sub.2 H.sub.5            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)C.sub.2 H.sub.5            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)C.sub.2 H.sub.5            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.4 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    (CH.sub.2).sub.4 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.4 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)(CH.sub.2).sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)(CH.sub.2).sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)(CH.sub.2).sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            CHH    CH.sub.2 CH.sub.2 OCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.2 CH.sub.2 OCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 OCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CHF.sub.2   H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CHF.sub.2   H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CHF.sub.2   H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CF.sub.3    H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CF.sub.3    H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 F            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 F            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CF.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CF.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CCl.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CCl.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHCl.sub.2            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHCl.sub.2            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 Cl            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 Cl            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 Cl            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            CHH    (CH.sub.2).sub.4 Cl            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            CHH    (CH.sub.2).sub.4 Cl            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.4 Cl            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CH.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CH.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 Br            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 Br            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 Br            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub. 3 Br            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            N5-Cl CH.sub.3    H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            N5-Cl CH.sub.3    H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            N6-Cl CH.sub.3    H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            N6-OCH.sub.3CH.sub.3    H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            N6-Br CH.sub.3    H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.3    CH.sub.3               H CH.sub.3                     OCH.sub.2 CHF.sub.2                            CHH    CH.sub.3    CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.3    CH.sub.3               H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.3    CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.3    CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.3    CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    C.sub.2 H.sub.5            CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    C.sub.2 H.sub.5            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    C.sub.2 H.sub.5            CH.sub.3               H OCH.sub.3                     OCH.sub. 2 CHF.sub.2                            NH    CH(CH.sub.3 ).sub.2            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3 ).sub.2            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3 ).sub.2            CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.2 CH.sub.2 CH.sub.3            CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.2 CH.sub.2 CH.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 CH.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 CH.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 CH.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 CH.sub.3            CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.2 CH(CH.sub.3).sub.2            CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.2 CH(CH.sub.3).sub.2            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH(CH.sub.3).sub.2            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)C.sub.2 H.sub.5            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)C.sub.2 H.sub.5            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)C.sub.2 H.sub.5            CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.4 CH.sub.3            CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    (CH.sub.2).sub.4 CH.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.4 CH.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)(CH.sub.2).sub.2 CH.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)(CH.sub.2).sub.2 CH.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)(CH.sub.2).sub.2 CH.sub.3            CH.sub.3               H CH.sub.3                     OCH.sub.2 CHF.sub.2                            CHH    CH.sub.2 CH.sub.2 OCH.sub.3            CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CH.sub.2 CH.sub.2 OCH.sub.3            CH.sub. 3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 OCH.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CHF.sub.2   CH.sub.3               H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            CHH    CHF.sub.2   CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CHF.sub.2   CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CF.sub.3    CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CF.sub.3    CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 F            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 F            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CF.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub. 2                            NH    CH.sub.2 CF.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CCl.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CCl.sub.3            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 Cl            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 Cl            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHCl.sub.2            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHCl.sub.2            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 Cl            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 Cl            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 Cl            CH.sub.3               H CH.sub.3                     OCH.sub.2 CHF.sub.2                            CHH    (CH.sub.2).sub.4 Cl            CH.sub.3               H CH.sub.3                     OCH.sub.2 CHF.sub.2                            CHH    (CH.sub.2).sub.4 Cl            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.4 Cl            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CH.sub.2 Cl            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CH.sub.2 Cl            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 Br            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 Br            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 Br            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 Br            CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            N5-Cl CH.sub.3    CH.sub.3               H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            N5-Cl CH.sub.3    CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            N6-Cl CH.sub.3    CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            N6-OCH.sub.3CH.sub.3    CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            N6-Br CH.sub.3    CH.sub.3               H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    H           H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    H           H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    H           H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    H           H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3).sub.2            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3).sub.2            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH(CH.sub.3).sub.2            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH(CH.sub.3).sub.2            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3) C.sub.2 H.sub.5            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 OCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 OCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 OC.sub.2 H.sub.5            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CHF.sub.2   H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CHF.sub.2   H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CF.sub.3    H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CF.sub.3    H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 F            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 F            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CF.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CF.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHCl.sub.2            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHCl.sub.2            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CCl.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CCl.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 Cl            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 Cl            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)CH.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CH.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CHf.sub.2                            NH    (CH.sub.2).sub.4 Cl            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.4 Cl            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.4 F            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.4 F            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.4 F            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.4 F            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 Br            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 Br            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 Br            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 Br            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.4 Br            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.4 Br            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.4 Br            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.4 Br            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 F            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 F            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    (CH.sub.2).sub.3 F            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    (CH.sub.2).sub.3 F            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHF.sub.2            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHF.sub.2            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHF.sub.2            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHF.sub.2            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 F  H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 F  H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 F  H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 F  H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 (CH.sub.3)CH.sub.2 Br            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 (CH.sub.3)CH.sub.2 Br            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 (CH.sub.3)CH.sub.2 Br            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 (CH.sub.3)CH.sub.2 Br            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 (CH.sub.3)CH.sub.2 F            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 (CH.sub.3)CH.sub.2 F            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 (CH.sub.3)CH.sub.2 F            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 (CH.sub.3)CH.sub.2 F            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHClCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHClCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHClCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHClCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHBrCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHBrCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHBrCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHBrCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHFCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHFCH.sub.3            H  H CH.sub. 3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHFCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHFCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.2 Cl).sub.2            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.2 Cl).sub.2            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.2 Cl).sub.2            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.2 Cl).sub.2            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.2 F).sub.2            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.2 F).sub.2            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.2 F).sub.2            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.2 F).sub.2            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)CCl.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CCl.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)CCl.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CCl.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 CHClCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 CHClCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 CHClCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 CHClCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 CHBrCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 CHBrCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 CHBrCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 CHBrCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 CHFCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 CHFCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH.sub.2 CHFCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH.sub.2 CHFCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHClCH.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHClCH.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHClCH.sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHClCH.sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHBrCH.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHBrCH.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHBrCH.sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHBrCH.sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHFCH.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHFCH.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CHFCH.sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CHFCH.sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)CHClCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CHClCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)CHClCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CHClCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)CHBrCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CHBrCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)CHBrCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CHBrCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)CHFCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CHFCH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.3)CHFCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.3)CHFCH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CCl.sub.2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CCl.sub. 2 CH.sub.3            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CCl.sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CCl.sub.2 CH.sub.3            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Br            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Br            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Br            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 Br            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 F            H  H CH.sub.3                     OCH.sub.2 CH.sub. 2 F                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 F            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 F            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CH(CH.sub.3)CH.sub.2 F            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CF.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CF.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 CF.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 CF.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CHCl.sub.2)CH.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CHCl.sub.2)CH.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CHCl.sub.2)CH.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CHCl.sub.2)CH.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CHCl.sub.2)CH.sub.2 F            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CHCl.sub.2)CH.sub.2 F            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CHCl.sub.2)CH.sub.2 F            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CHCl.sub.2)CH.sub.2 F            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.2 Cl)CH.sub.2 CH.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.2 Cl)CH.sub.2 CH.sub.2 Cl            H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH(CH.sub.2 Cl)CH.sub.2 CH.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH(CH.sub.2 Cl)CH.sub.2 CH.sub.2 Cl            H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 Br H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 Br H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 Br H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 Br H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 Cl H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 Cl H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CH.sub.2 Cl H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CH.sub.2 Cl H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CHCl.sub.2  H  H CH.sub. 3                     OCH.sub.2 CH.sub.2 F                            NH    CHCl.sub.2  H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CHCl.sub.2  H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CHCl.sub.2  H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CCl.sub.3   H  H CH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CCl.sub.3   H  H CH.sub.3                     OCH.sub.2 CHF.sub.2                            NH    CCl.sub.3   H  H OCH.sub.3                     OCH.sub.2 CH.sub.2 F                            NH    CCl.sub.3   H  H OCH.sub.3                     OCH.sub.2 CHF.sub.2                            N__________________________________________________________________________   PG,79 
    
     
                       TABLE IX______________________________________General Structure IXR.sub.2  R.sub.7         R      X     Y        Z     m.p. (°C.)______________________________________H      H      H      CH.sub.3                      OCH.sub.2 CHF.sub.2                               NH      H      H      OCH.sub.3                      OCH.sub.2 CHF.sub.2                               NH      H      H      OCH.sub.3                      OCH.sub.2 CH.sub.2 F                               NH      CH.sub.3         H      OCH.sub.3                      OCH.sub.2 CH.sub.2 F                               NH      CH.sub.3         H      OCH.sub.3                      OCH.sub.2 CHF.sub.2                               NH      CH.sub.3         H      CH.sub.3                      OCH.sub.2 CHF.sub.2                               N6-OCH.sub.3  CH.sub.3         H      CH.sub.3                      OCH.sub.2 CHF.sub.2                               NH      H      H      CH.sub.3                      OCH.sub.2 CH.sub.2 F                               NH      CH.sub.3         H      CH.sub.3                      OCH.sub.2 CH.sub.2 F                               NH      H      H      OCH.sub.3                      OCH.sub.2 CH.sub.2 F                               CHH      H      H      OCH.sub.3                      OCH.sub.2 CHF.sub.2                               CH______________________________________ 
    
     
                       TABLE X______________________________________General Structure XR.sub.2  R.sub.7         R      X     Y        Z     m.p. (°C.)______________________________________H      H      H      CH.sub.3                      OCH.sub.2 CHF.sub.2                               NH      H      H      OCH.sub.3                      OCH.sub.2 CHF.sub.2                               NH      H      H      OCH.sub.3                      OCH.sub.2 CH.sub.2 F                               NH      CH.sub.3         H      OCH.sub.3                      OCH.sub.2 CH.sub.2 F                               NH      CH.sub.3         H      OCH.sub.3                      OCH.sub.2 CHF.sub.2                               NH      CH.sub.3         H      CH.sub.3                      OCH.sub.2 CHF.sub.2                               N6-OCH.sub.3  CH.sub.3         H      CH.sub.3                      OCH.sub.2 CHF.sub.2                               NH      H      H      CH.sub.3                      OCH.sub.2 CH.sub.2 F                               NH      CH.sub.3         H      CH.sub.3                      OCH.sub.2 CH.sub.2 F                               NH      H      H      OCH.sub.3                      OCH.sub.2 CH.sub.2 F                               CHH      H      H      CH.sub.3                      OCH.sub.2 CHF.sub.2                               CH______________________________________ 
    
     Formulations 
     Useful forrmulations of the compounds of Formula I can be prepared in conventional ways. They include dusts, granules, pellets, solutions, suspensions, emulsions, wettable powders, emulsifiable concentrates and the like. Many of these may be applied directly. Sprayable formulations can be extended in suitable media and used at spray volumes of from a few pints to several hundred gallons per acre. High strength compositions are primarily used as intermediates for further formulation. The formulations, broadly, contain about 1-99% by weight of active ingredient(s) and at least one of (a) about 0.1-20% surfactant(s) and (b) about 5-99% solid or liquid diluent(s). More specifically, they will contain these ingredients in the following approximate proportions: 
     
         ______________________________________      Percent by Weight      Active      Ingredient              Diluent(s)                        Surfactant(s)______________________________________Wettable Powders        20-90      0-75     1-10Oil Suspensions,         5-50     40-95     0-15Emulsions, Solutions(including Emulsifi-able Concentrates)Aqueous Suspensions        10-50     40-95     0-15Dusts         1-25     70-99     0-5Granules and Pellets         1-95      5-99     0-15High Strength        90-99      0-10     0-2Compositions______________________________________ 
    
     Lower or higher levels of active ingredient can, of course, be present depending on the intended use and the physical properties of the compound. Higher ratios of surfactant to active ingredient are sometimes desirable, and are achieved by incorporation into the formulation or by tank mixing. 
     Typical solid diluents are described in Watkins, et al., Handbook of Insecticide Dust Diluents and Carriers, 2nd Edition, Dorland Books, Caldwell, NJ. The more absorptive diluents are preferred for wettable powders and the denser ones for dusts. Typical liquid diluents and solvents are described in Marsden, Solvents Guide, 2nd Edition, Interscience, New York 1950. Solubility under 0.1% is preferred for suspension concentrates; solution concentrates are preferably stable against phase separation at 0° C. McCutcheon&#39;s Detergents and Emulsifiers Annual, Allured Publishing Corp., Ridgewood, NJ, as well as Sisely and Wood, Encyclopedia of Surface Active Agents, Chemical Publishing Co., Inc., New York, 1964, list surfactants and recommended uses. All formulations can contain minor amounts of additives to reduce foam, caking, corrosion, microbiological growth, etc. Preferably, ingredients should be approved by the U.S. Environmental Protection Agency for the use intended. 
     The methods of making such compositions are well known. Solutions are prepared by simply mixing the ingredients. Fine solid compositions are made by blending and, usually, grinding as in a hammer or fluid energy mill. Suspensions are prepared by wet milling (see, for example, Littler, U.S. Pat. No. 3,060,084). Granules and pellets may be made by spraying the active material upon preformed granular carriers or by agglomeration techniques. See J. E. Browning, &#34;Agglomeration&#34; Chemical Engineering, Dec. 4, 1967, pages 147ff and Perry&#39;s Chemical Engineer&#39;s Handbook, 4th Edition, McGraw-Hill, New York 1963, pages 8-59ff. 
     For further information regarding the art of formulation, see for example: H. M. Loux, U.S. Pat. No. 3,235,361, issued Feb. 15, 1966, Col. 6, lines 16  through Col. 7, line 19, and Examples 10 through 41; R. W. Luckenbaugh, U.S. Pat. No. 3,309,192, issued Mar. 14, 1967, Col. 5, lines 43 through Col. 7, line 62, and Examples 8, 12, 15, 39, 41, 52, 53. 58, 132, 138-140, 162-164, 166, 167, 169-182; H. Gysin and E. Knusli, U.S. Pat. No. 2,891,855 issued June 23, 1959, Col. 3, lines 66 through Col. 5, line 17 and Examples 1-4; G. C. Klingman, Weed Control As a Science, John Wiley &amp; Sons, Inc., New York 1961, pages 81-96; and J. D. Fryer and S. A. Evans, Weed Control Handbook, 5th Edition, Blackwell Scientific Publications, Oxford, 1968, pages 101-103. 
     EXAMPLE 4 
     Wettable Powder 
     
         ______________________________________2-ethoxy-N--[[4-methoxy-6-(2,2,2-trifluoroethoxy)-                       40%1,3,5-triazin-2-yl]aminocarbonyl]benzene-sulfonamidedioctyl sodium sulfosuccinate                       1.5%sodium ligninsulfonate       3%low viscosity methyl cellulose                       1.5%attapulgite                 54%______________________________________ 
    
     The ingredients are thoroughly blended, passed through an air mill, to produce an average particle size under 15 microns, reblended, and sifted through a U.S.S. No. 50 sieve (0.3 mm opening) before packaging. 
     All compounds of the invention may be formulated in the same manner. 
     EXAMPLE 5 
     Wettable Powder 
     
         ______________________________________N--[[4-methoxy-6-(2,2,2-trifluoroethoxy)-1,3,5-                     50%triazin-2-yl]aminocarbonyl]-2-propoxybenzene-sulfonamidesodium alkylnaphthalenesulfonate                      2%low viscosity methyl cellulose                      2%diatomaceous earth        46%______________________________________ 
    
     The ingredients are blended, coarsely hammer milled and the air milled to produce particles of active essentially all below 10 microns in diameter. The product is reblended before packaging. 
     EXAMPLE 6 
     Wettable Powder 
     
         ______________________________________2-ethoxy-N--[[4-methoxy-6-(2,2,2-trifluoroethoxy)-                       80%1,3,5-triazin-2-yl]aminocarbonyl]benzenesulfon-amidesodium alkylnaphthalenesulfonate                        2%sodium ligninsulfonate       2%synthetic amorphous silica   3%kaolinite                   13%______________________________________ 
    
     The ingredients are blended, hammermilled until all the solids are essentially under 50 microns in diameter, and then reblended before packaging. 
     EXAMPLE 7 
     Wettable Powder 
     
         ______________________________________N--[[4-methoxy-6-(2,2,2-trifluoroethoxy)-1,3,5-                     65%triazin-2-yl]aminocarbonyl]-2-propoxybenzene-sulfonamidedodecylphenol polyethylene glycol                      2%ethersodium ligninsulfonate     4%sodium silicoaluminate     6%montmorillonite (calcined)                     23%______________________________________ 
    
     The ingredients are thoroughly blended. The liquid surfactant is added by spraying upon the solid ingredients in the blender. After grinding in a hammermill to produce particles essentially all below 100 microns, the material is reblended and sifted through a U.S.S. No. 50 sieve (0.3 mm opening) and packaged. 
     EXAMPLE 8 
     High Strength Concentrate 
     
         ______________________________________2-ethoxy-N--[[4-methoxy-6-(2,2,2-trifluoroethoxy)-                     98.5%1,3,5-triazin-2-yl]aminocarbonyl]benzenesulfon-amidesilica aerogel            0.5%synthetic amorphous fine silica                     1.0%______________________________________ 
    
     The ingredients are blended and ground in a hammer-mill to produce a high strength concentrate essentially all passing a U.S.S. No. 50 sieve (0.3 mm opening). This material may then be formulated in a variety of ways. 
     EXAMPLE 9 
     Aqueous Suspension 
     
         ______________________________________N--[[4-methoxy-6-(2,2,2-trifluoroethoxy)-1,3,5-                     25%triazin-2-yl]aminocarbonyl]-2-propoxybenzene-sulfonamidehydrated attapulgite       3%crude calcium ligninsulfonate                     10%sodium dihydrogen phosphate                      0.5%water                     61.5%______________________________________ 
    
     The ingredients are ground together in a ball or roller mill until the solid particles have been reduced to diameters under 10 microns. 
     EXAMPLE 10 
     Oil Suspension 
     
         ______________________________________2-ethoxy-N--[[4-methoxy-6-(2,2,2-trifluoroethoxy)-                       25%1,3,5-triazin-2-yl]aminocarbonyl]benzenesulfon-amidepolyoxyethylene sorbitol hexaoleate                        5%highly aliphatic hydrocarbon oil                       70%______________________________________ 
    
     The ingredients are ground together in a sand mill until the solid particles have been reduced to under about 5 microns. The resulting thick suspension may be applied directly, but preferably after being extended with oils or emulsified in water. 
     EXAMPLE 11 
     Granule 
     
         ______________________________________2-ethoxy-N--[[4-methoxy-6-(2,2,2-trifluoroethoxy)-                       80%1,3,5-trizain-2-yl]aminocarbonyl]benzenesulfon-amideWetting Agent                1%Crude Ligninsulfonate salt (containing                       10%5-20% of the natural sugars)Attapulgite clay             9%______________________________________ 
    
     The ingredients are blended and milled to pass through a 100 mesh screen. This material is then added to a fluid bed granulator, the air flow is adjusted to gently fluidize the material, and a fine spray of water is sprayed onto the fluidized material. The fluidization and spraying are continued until granules of the desired size range are made. The spraying is stopped, but fluidization is continued, optionally with heat, until the moisture in the material is reduced to the desired level, generally less than 1%. The material is then discharged, screened to the desired size range, generally 14-100 mesh (140-149 microns), and packaged for use. 
     EXAMPLE 12 
     Extruded Pellet 
     
         ______________________________________N--[[4-methoxy-6-(2,2,2-trifluoroethoxy)-1,3,5-                     25%triazin-2-yl]aminocarbonyl]-2-propoxybenzene-sulfonamideanhydrous sodium sulfate  10%crude calcium ligninsulfonate                      5%sodium alkylnaphthalenesulfonate                      1%calcium/magnesium bentonite                     59%______________________________________ 
    
     The ingredients are blended, hammermilled and then moistened with about 12% water. The mixture is extruded as cylinders about 3 mm diameter which are cut to produce pellets about 3 mm long. These may be used directly after drying, or the dried pellets may be crushed to pass a U.S.S. No. 20 sieve (0.54 mm openings). The granules held on a U.S.S. No. 40 sieve (0.42 mm openings) may be packaged for use and the fines recycled. 
     UTILITY 
     Test results indicate that the compounds of the present invention are active herbicides. They should have utility for broad spectrum pre- and/or post-emergence weed control in areas where complete control of all vegetation is desired, such as around fuel storage tanks, ammunition depots, industrial storage areas, parking lots, drive-in theaters, around billboards, highway and railroad structures. Alternatively, the subject compounds are useful for the selective pre- or post-emergence weed control in corn. 
     The rates of application for the compounds of the invention are determined by a number of factors, including their use as selective or general herbicides, the crop species involved, the types of weeds to be controlled, weather and climate, formulations selected, mode of application, amount of foliage present, etc. In general terms, the subject compounds should be applied at levels of around 0.002-5 kg/ha, the lower rates being suggested for use on lighter soils and/or those having a low organic matter content, for selective weed control or for situations where only short-term persistence is required. 
     The compounds of the invention may be used in combination with any other commercial herbicide; examples of which are those of the triazine, triazole, uracil, urea, amide, diphenylether, carbamate, and bipyridylium types. They may also be used in combination with mefluidide. 
     
         ______________________________________Com-pound                          m.p. (°C.)______________________________________  ##STR26##               180-181(d)2  ##STR27##               161-163(d)3  ##STR28##               121-126(d)4  ##STR29##               120-124(d)5  ##STR30##               132-1376  ##STR31##               94-102; 112(d)7  ##STR32##               115-118(d)8  ##STR33##               193-197(d)9  ##STR34##               198-20210  ##STR35##               176-17911  ##STR36##               165-16812  ##STR37##               168-17013  ##STR38##               152-156______________________________________ 
    
     TEST A 
     Seeds of crabgrass (Digitaria spp.), barnyardgrass (Echinochloa crusgalli), wild oats (Avena fatua), sickelpod (Cassia obtusifolia), morningglory (Ipomoea spp.), cocklebur (Xanthium pensylvanicum), sorghum, corn, soybean, cotton, sugar beet, rice, wheat, and purple nutsedge (Cyperus rotundus) tubers were planted and treated preemergence with the test chemicals dissolved in a nonphytotoxic solvent. At the same time, these crop and weed species were treated with a soil/foliage application. At the time of treatment, the plants ranged in height from 2-18 cm. Treated plants and controls were maintained in a greenhouse for sixteen days, after which all species were compared to controls and visually rated for response to treatment. The ratings, summarized in Table A, are based on a numerical scale extending from 0=no injury, to 10=complete control. The accompanying descriptive symbols have the following meanings: 
     C=chlorosis/necrosis 
     E=emergence inhibition 
     G=growth retardation 
     H=formative effect 
     The herbicidal properties of the subject compounds were discovered in a number of greenhouse tests. The test procedures and results follow: 
     
                                           TABLE A__________________________________________________________________________   Cmpd. 1        Cmpd. 2             Cmpd. 3                  Cmpd. 4                       Cmpd. 5                            Cmpd. 6                                 Cmpd. 7                                      Cmpd. 8Rate kg/ha   0.05 0.05 0.05 0.05 0.05 0.05 0.05 0.05__________________________________________________________________________POSTEMERGENCEMorningglory   9C   9C   5C,8H                  10C  9C   10C  0    5C,9GCocklebur   10C  10C  10C  10C  6C,9G                            2C,9G                                 2C,5G                                      9CSicklepod   5C,9G        5C,9G             4C,9G                  9C   9C   9C   2C   2C,3GNutsedge   4C,9G        4C,8G             5G   4C,9G                       6C,9G                            9C   0    2C,8GCrabgrass   2C,5G        2G   0    5G   5G   5G   2G   3C,5GBarnyardgrass   3C,8H        0    2C,2H                  3C,9H                       5C,9H                            3C,9H                                 3H   2C,3HWild Oats   8G   0    0    5G   6G   2C,9G                                 0    0Wheat   4G   0    0    3G   0    8G   0    0Corn    4G   1C   0    1H   6G   3G   0    0Soybean 4C,9G        9C   5C,9G                  9C   5C,9G                            9C   2C,3G                                      4C,9GRice    5C,9G        4C,7G             3C,8G                  2C,9G                       9C   9C   2C   1GSorghum 2C,9G        1C,3G             3C,5G                  2C,9H                       2C,9H                            3C,9H                                 2G   1GSugar beet   5C,9G        9C   9C   9C   10C  10C  3C,6G                                      5C,9GCotton  9C   9C   5C,9G                  5C,9G                       9C   9C   0    4C,8HPREEMERGENCEMorningglory   4C,9G        9G   9G   9C   9G   9G   0    8GCocklebur   9H   9H   --   --   8H   8H   4G   8HSicklepod   9G   6G   9G   10C  9G   9C   --   2C,8GNutsedge   10E  8G   4C,9G                  3C,8G                       2C,8G                            3C,9G                                 0    3C,5GCrabgrass   0    3G   3G   5G   2G   1C   3G   1CBarnyardgrass   3C,6G        1G,3G             2G   5G   7H   9H   3G   2C,2HWild Oats   2C,8G        0    2C,6G                  2C,6G                       5G   6C,9G                                 0    2C,2GWheat   0    0    0    0    0    6G   5C   4GCorn    1C,5G        2C   5G   5G   7G   5G   3G   3C,6GSoybean 9H   8H   9H   9H   8H   9H   0    1CRice    10E  6G   3C,8H                  3C,9H                       9H   10E  2C,5G                                      3C,7GSorghum 4C,9H        5G   2C,8G                  3C,9G                       3C,8H                            5C,9H                                 2C,6G                                      3C,6GSugar beet   10E  10E  10E  10E  9C   9C   6G   9CCotton  9G   9G   9G   9G   9G   9G   2G   7G__________________________________________________________________________                  Cmpd. 9                       Cmpd. 10                            Cmpd. 11                                 Cmpd. 12                                      Cmpd. 13          Rate kg/ha                  0.05 0.05 0.05 0.05 0.05__________________________________________________________________________          POSTEMERGENCE          Morningglory                  2C,7H                       2C,4G                            2C,8G                                 3C,7H                                      10C          Cocklebur                  3G   2C,2G                            1C   3G   10C          Sicklepod                  4C,9H                       2C,4G                            2C,3H                                 2C,6G                                      5C,9G          Nutsedge                  3C,8G                       5G   4C,8G                                 2C,4G                                      5C,9G          Crabgrass                  2C,8G                       3G   2G   0    4C,8G          Barnyardgrass                  4C,9H                       3C,9H                            1H   0    9C          Wild Oats                  4C,7G                       2C,3G                            0    0    5C,9G          Wheat   2C,8G                       2C,3G                            0    0    9C          Corn    3C,9H                       1G   1H   0    5U,9C          Soybean 3C,7G                       2C,2H                            2C,2H                                 2H   9H          Soybean 3C,9H                       4C,9G                            2C,5H                                 3C,6H                                      5C,9G          Rice    5C,9G                       8G   6G   0    6C,9G          Sorghum 3C,9G                       2C,9G                            5G   2G   4U,9G          Sugar beet                  4C,9G                       3C,5G                            2C,6G                                 8G   9C          Cotton  9C   3C,8G                            8G   4C,9G                                      9C          PREEMERGENCE          Morningglory                  7G   2G   9G   7G   9G          Cocklebur                  --   8H   7H   0    9H          Sicklepod                  5C,9G                       2C   8G   2H   3C,9G          Nutsedge                  3C,7G                       4G   5G   0    4G          Crabgrass                  6G   2G   3G   0    2C,5G          Barnyardgrass                  5C,9H                       2C,8H                            3C,9H                                 6G   3C,9H          Wild Oats                  6C,9G                       8G   2C,5G                                 0    3C,8H          Wheat   4C,9H                       9H   5G   0    7C,9H          Corn    3C,9H                       1C,6G                            5G   3G   3C,9H          Rice    3C,8H                       2C,8G                            5G   0    10E          Sorghum 3C,9H                       2C,9G                            2C,8G                                 7G   5C,9H          Sugar beet                  4C,9G                       8G   8G   7H   5C,9G          Cotton  2C,9G                       8G   8G   2G   2C,9G__________________________________________________________________________ 
    
     TEST B 
     Postemergence 
     Two round pans (25 cm diameter by 12.5 cm deep) were filled with Woodstown sandy loam soil. One pan was planted with blackgrass (Alopecurus myosuroides), sugar beets, nutsedge (Cyperus rotundus) tubers, crabgrass (Digitaria sanguinalis), sickelpod (Cassia obtusifolia), teaweed (Sida spinosa), jimsonweed (Datura stramonium), velvetleaf (Abutilon theophrasti), and giant foxtail (Setaria faberii). The other pan was planted with wheat, cotton, rice, corn, soybean, wild oats (Avena fatua), cocklebur (Xanthium pensylvanicum), morninglory (Ipomoea hederacea), johnsongrass (Sorghum halepense) and barnyard grass (Echinochloa crusgalli). The plants were grown for approximately fourteen days, then sprayed postemergence with the chemicals dissolved in a nonphytotoxic solvent. 
     Preemergence 
     Two round pans (25 cm diameter by 12.5 cm deep) were filled with Woodstown sandy loam soil. One pan was planted with blackgrass (Alopecurus myosuroides), sugar beets, nutsedge, crabgrass, sicklepod, teaweed, jimsonweed, velvetleaf, and giant foxtail. The other pan was planted with wheat, cotton, rice, corn, soybeans, wild oats, cocklebur, morningglory, johnsongrass and barnyardgrass. The two pans were sprayed preemergence with the chemicals dissolved in a nonphytotoxic solvent. 
     Treated plants and controls were maintained in the greenhouse for 28 days, then all treated plants were compared to controls and visually rated for plant response as described for Test A. 
     Reponse ratings are contained in Table B. The data show that both test compounds have utility for selective pre- and postemergence weed control in corn. 
     
                                           TABLE B__________________________________________________________________________   Compound 1   Compound 2   Compound 8                                       Compound 10                                               Compound 13Rate g/ha   62 16 4  1   62 16 4  1   250                                62 16  250 62  62 16 4  1__________________________________________________________________________POSTEMERGENCECorn    3G 0  0  0   0  0  0  0   0  0  0   4G  0   10G                                                  10C                                                     9G 5GWheat   3G 0  0  0   0  0  0  0   0  0  0   4G  0   10C                                                  7G 0  0Rice    10G      9G 3G 0   2G 0  0  0   4G 2G 0   4G  3G  10C                                                  10G                                                     8G 4GSoybean 10G      10G         9G 8G  9G 9G 6G 2G  10G                                9G 7G  8G  5G  10G                                                  10g                                                     9G 6GCotton  10C      8G 4G 2G  9G 5G 2G 0   4G 3G 0   7G  3G  10G                                                  8G 6G 3GSugar beet   10C      10C         10C            8G  9G 9G 7G 4G  10G                                10G                                   4G  5G  3G  10C                                                  8G 5G 4GCrabgrass   0  0  0  0   3G 0  0  0   3G 0  0   0   0   5G 3G 0  0Johnsongrass   10G      5G 3G 0   0  0  0  0   0  0  0   6G  0   10C                                                  9G 4G 3GBlackgrass   10C      9G 3G 0   0  0  0  0   4G 0  0   7G  0   10C                                                  6G 0  0Barnyardgrass   5G 2G 0  0   0  0  0  0   0  0  0   7G  4G  10C                                                  9G 5G 0Nutsedge   10C      10C         4G 0   0  0  0  0   7G 4G 0   0   0   3G 0  0  0Giant foxtail   3G 0  0  0   0  0  0  0   0  0  0   4G  0   10C                                                  3G 0  0Wild Oats   5G 0  0  0   0  0  0  0   0  0  0   3G  0   10C                                                  5G 0  0Cocklebur   10C      10G         7G 3G  10C                   8G 6G 3G  10G                                9G 7G  0   0   10G                                                  7G 4G 0Morningglory   10G      10G         9G 5G  9G 7G 2G 0   10G                                8G 6G  3G  0   10G                                                  7G 3G 0Teaweed 9G 5G 0  0   4G 0  0  0   0  0  0   4G  0   6G 2G 0  0Sicklepod   10G      9G 4G 0   4G 2G 0  0   4G 0  0   3G  0   6G 4G 0  0Jimsonweed   10C      7G 5G 0   7G 7G 0  0   4G 0  0   7G  5G  6G 5G 0  0Velvetleaf   10C      10C         8G 2G  9G 7G 4G 0   9G 7G 3G  9G  7G  10G                                                  5G 0  0__________________________________________________________________________   Compound 1   Compound 2   Compound 8                                       Compound 10                                               Compound 13Rate kg/ha   250      62 16 4   250                   62 16 4   250                                62 16  250 62  250                                                  62 16 4__________________________________________________________________________PREEMERGENCECorn    2G 0  0  0   2G 0  0  0   2G 0  0   4G  2G  10E                                                  10G                                                     6G 0Wheat   0  0  0  0   2G 0  0  0   0  0  0   7G  4G  7G 2G 0  0Rice    10E      10E         9G 5G  9G 5G 2G 0   7G 5G 2G  10G 6G  10E                                                  10E                                                     10G                                                        6GSoybean 10G      9G 7G 2G  8G 4G 0  0   2G 0  0   5G  2G  10G                                                  9G 4G 0Cotton  10G      10G         6G 0   9G 4G 0  0   3G 0  0   7G  0   8G 6G 0  0Sugar beet   10G      10E         9G 5G  10G                   8G 3G 0   10G                                7G 4G  9G  7G  10G                                                  10G                                                     10G                                                        3GCrabgrass   0  0  0  0   0  0  0  0   3G 0  0   2G  0   10G                                                  7G 4G 2GJohnsongrass   10G      9G 4G 0   7G 3G 2G 0   2G 0  0   7G  0   10C                                                  10C                                                     9G 4GBlackgrass   10G      9G 8G 2G  9G 5G 4G 0   7G 5G 2G  10G 7G  10E                                                  9G 7G 2GBarnyardgrass   6G 6G 2G 0   3G 0  0  0   4G 0  0   6G  0   10G                                                  10G                                                     7G 3GNutsedge   10E      10E         7G 3G  9G 5G 3G 2G  9G 3G 0   4G  0   10E                                                  3G 0  0Giant foxtail   -- -- -- --  -- -- -- --  -- -- --  8G  5G  10E                                                  10G                                                     9G 4GWild Oats   7G 5G 0  0   3G 0  0  0   0  0  0   7G  6G  8G 4G 2G 0Cocklebur   10G      10G         8G 3G  10G                   9G 6G 2G  8G 0  0   0   0   10G                                                  7G 3G 0Morningglory   10G      10G         7G 3G  9G 6G 4G 2G  6G 0  0   0   0   10G                                                  7G 2G 0Teaweed 10G      9G 6G 3G  9G 4G 0  0   9G 5G 3G  3G  0   8G 3G 0  0Sicklepod   10E      10G         6G 4G  9G 4G 0  0   5G 0  0   8G  0   7G 3G 0  0Jimsonweed   10G      10G         9G 3G  9G 4G 0  0   7G 3G 0   8G  4G  9G 8G 4G 0Velvetleaf   10G      10G         9G 3G  9G 5G 0  0   7G 2G 0   6G  2G  10G                                                  5G 2G 0__________________________________________________________________________ 
    
     TEST C 
     Three 25-cm diameter plastic pots were filled with a light soil. One pot was planted to short rows of corn, soybeans and cotton, planting depth 2.5 cm. The other two pots were planted to the following weed species, 8 or 9 species per pot: crabgrass (Digitaria sp.), johnsongrass (Sorghum halepense), barnyardgrass (Echinochloa crusgalli), nutsedge (Cyperus rotundus), giant foxtail (Setaria faberi), green foxtail (Setaria viridis), cocklebur (Xanthium pensylvanicum), morning-glory (Ipomoea hederacea), teaweed (Sida spinosa), sicklepod (Cassia obtusifolia), jimsonweed (Datura stramonium), velvetleaf (Abutilon theophrasti), bindweed (Convolvulus arvensis), coffeeweed (Sesbania exaltata), lambsquarters (Chenopodium album), pigweed (Amaranthus retroflexus) and purslane (Portulaca oleracea). All of the foregoing weed species were planted at a depth of 0.5-1.0 cm except for cocklebur and nutsedge which were planted at a depth of 2.5 cm. The plantings were treated preemergence with the test chemicals dissolved in a nonphytotoxic solvent. At the same time, the same crops and weed species, from plantings made 10-21 days previously, were treated with soil/foliage applications. Treated plants and controls were maintained in a greenhouse for 3-4 weeks after which all species were compared to controls and visually rated for response to treatment utilizing the same rating system as described for Test A. The data for three tests for Compound 1 and two tests for Compound 2 are summarized in Table C. 
     It will be seen that both compounds can be used for selective weed control in corn, either applied pre- or postemergence. 
     
                                           TABLE C__________________________________________________________________________   Compound 1Rate g/ha   16 31 62 125               250                  4  16 62 250                              1000                                 16 31 62 125                                             250__________________________________________________________________________POSTEMERGENCECorn    0  0  0  0  3G 0  0  0  3G 0  0  0  0  0  0Cotton  10C      10C         10C            10C               10C                  5G 10C                        10C                           10C                              10C                                 9G 10C                                       10C                                          10C                                             10CSoybean 10C      10C         10C            10C               10C                  10C                     10C                        10C                           10C                              10C                                 10C                                    10C                                       10C                                          10C                                             10CGreen foxtail   0  0  0  0  3G 0  0  0  2G 5G 0  0  0  0  3GGiant foxtail   0  0  0  2G 4G 0  0  0  3G 5G 0  0  0  0  3GBarnyardgrass   0  0  0  0  3G 0  0  0  3G 7G 0  0  0  3G 6GJohnsongrass   0  3G 6G 8G 10C                  0  0  5G 8G 10C                                 0  2G 6G 8G 9GCrabgrass   0  0  0  0  0  0  0  0  0  0  0  0  0  0  0Nutsedge   -- 7G 8G 9G 10C                  0  0  10C                           10C                              10C                                 0  3G 9G 10C                                             10CVelvetleaf   10C      10C         10C            10C               10C                  5G 9G 10C                           10G                              10C                                 10C                                    10C                                       10C                                          10C                                             10CSicklepod   6G 9G 8G 10G               10C                  0  6G 9G 10G                              10C                                 8G 9G 9G 9G 10CLambsquarter   0  0  5G 8G 10C                  4G 8G 9G 10C                              10C                                 -- -- -- -- --Pigweed 10C      10C         10C            10C               10C                  5G 8G 9G 10C                              10C                                 10C                                    10C                                       10C                                          10C                                             10CBindweed   9G 10C         10C            10C               10C                  5G 7G 8G 10C                              10C                                 9G 10C                                       10C                                          10C                                             10CJimsonweed   8G 10C         10C            10C               10C                  6G 8G 10C                           10C                              10C                                 10C                                    10C                                       10C                                          10C                                             10CPrickly sida   6G 8G 9G 9G 10G                  4G 7G 9G 10G                              10C                                 8G 10C                                       10C                                          10C                                             10CSesbania   10C      10C         10C            10C               10C                  9G 10C                        10C                           10C                              10C                                 9G 10C                                       10C                                          10C                                             10CPurslane   10G      10G         10G            10C               10C                  8G 10G                        10G                           10C                              10C                                 5G 8G 10C                                          10C                                             10CMorningglory   10C      10C         10C            10C               10C                  8G 10C                        10C                           10C                              10C                                 10C                                    10C                                       10C                                          10C                                             10CCocklebur   10C      10C         10C            10C               10C                  9G 10C                        10C                           10C                              10C                                 10C                                    10C                                       10C                                          10C                                             10C__________________________________________________________________________Rate g/ha   8  16 31 62 125                  4  16 62 250                              1000                                 16 31 62 125                                             250__________________________________________________________________________PREEMERGENCECorn    0  0  0  0  0  0  1G 3G 5G 6G 0  0  0  3G 6GCotton  2G 5G 6G 8G 9G 3G 9G 10G                           10G                              10G                                 9G 9G 10G                                          10G                                             10GSoybean 2G 5G 5G 8G 8G 2G 7G 9G 10G                              10G                                 7G 8G 10G                                          10G                                             10GGreen foxtail   0  0  0  2G 2G 0  0  3G 6G 9G 0  0  2G 6G 8GGiant foxtail   0  0  0  0  4G 0  0  3G 6G 9G 0  0  2G 5G 8GBarnyardgrass   0  0  0  0  6G 0  2G 3G 9G 10G                                 0  0  0  2G 8GJohnsongrass   0  0  3G 8G 9G 3G 7G 9G 10G                              10G                                 0  4G 6G 9G 10GCrabgrass   0  0  0  0  0  0  0  0  0  2G 0  0  0  0  0Nutsedge   0  7G 9G 10E               10E                  2G 3G 6G 10G                              10G                                 2G 9G 10E                                          10E                                             10EVelvetleaf   8G 9G 10G            10G               7G 5G 8G 10G                           10G                              10G                                 9G 10G                                       10E                                          10G                                             10GSicklepod   7G 8G 10G            10G               10E                  3G 8G 10G                           10G                              10G                                 8G 8G 10G                                          10E                                             10GLambsquarter   5G 8G 10G            10G               10G                  4G 9G 10G                           10G                              10G                                 8G 9G 10G                                          10E                                             10EPigweed 7G 8G 10G            10G               10G                  5G 9G 10G                           10G                              10G                                 9G 10E                                       10G                                          10E                                             10EBindweed   7G 10G         10G            10G               10G                  5G 8G 10G                           10G                              10G                                 9G 10G                                       10G                                          10G                                             10EJimsonweed   5G 9G 9G 10G               10G                  2G 9G 10G                           10G                              10G                                 9G 10G                                       10G                                          10G                                             10EPrickly sida   6G 7G 7G 10G               10G                  0  8G 10G                           10G                              10G                                 7G 9G 10G                                          10G                                             10ESesbania   0  2G 4G 9G 10G                  2G 6G 10G                           10G                              10G                                 7G 8G 10G                                          10G                                             10EPurslane   4G 3G 9G 10G               10G                  5G 9G 10G                           10G                              10G                                 7G 10G                                       10G                                          10G                                             10EMorningglory   3G 7G 9G 9G 10G                  4G 9G 10G                           10G                              10G                                 10G                                    10G                                       10G                                          10G                                             10GCocklebur   2G 4G 9G 10G               10G                  4G 8G 10G                           10G                              10G                                 7G 10G                                       10G                                          10G                                             10G__________________________________________________________________________                     Compound 2             Rate g/ha                     16 62 250                              1000                                 62 125                                       250                                          500                                             1000__________________________________________________________________________             POSTEMERGENCE             Corn    0  0  0  2G 7G 9G 10C                                          10C                                             10C             Cotton  7G 9G 10C                              10C                                 8G 9G 10C                                          10C                                             10C             Soybean 10C                        10C                           10C                              10C                                 10C                                    10C                                       10C                                          10C                                             10C             Green foxtail                     0  0  0  0  0  0  0  0  2G             Giant foxtail                     0  0  0  0  0  0  0  0  0             Barnyardgrass                     0  0  0  0  0  0  0  3G 6G             Johnsongrass                     0  0  3G 8G 0  0  0  2G 7G             Crabgrass                     0  0  0  2G 0  0  0  0  0             Nutsedge                     0  2G 7G 10C                                 0  3G 6G 7G 9G             Velvetleaf                     5G 9G 10C                              10C                                 9G 9G 10C                                          10C                                             10C             Sicklepod                     2G 7G 9G 10C                                 7G 8G 9G 9G 10C             Lambsquarter                     2G 6G 9G 10C                                 -- -- -- -- --             Pigweed 0  6G 9G 10C                                 8G 10C                                       10C                                          10C                                             10C             Bindweed                     0  5G 8G 10C                                 8G 9G 9G 10C                                             10C             Jimsonweed                     5G 7G 10C                              10C                                 8G 8G 10C                                          10C                                             10C             Prickly sida                     0  7G 8G 9G 7G 8G 9G 10C                                             10C             Sesbania                     8G 10C                           10C                              10C                                 8G 10C                                       10C                                          10C                                             10C             Purslane                     4G 8G 10C                              10C                                 7G 9G 9G 10C                                             10C             Morningglory                     4G 8G 10C                              10C                                 8G 9G 10C                                          10C                                             10C             Cocklebur                     10C                        10C                           10C                              10C                                 10C                                    10C                                       10C                                          10C                                             10C__________________________________________________________________________             Rate g/ha                     16 62 250                              1000                                 31 62 125                                          250                                             500__________________________________________________________________________             PREEMERGENCE             Corn    0  0  2G 5G 0  2G 6G 7G 9G             Cotton  4G 7G 10G                              10G                                 0  2G 9G 9G 10G             Soybean 4G 7G 10G                              10G                                 3G 6G 8G 9G 9G             Green foxtail                     0  0  0  0  0  0  0  0  0             Giant foxtail                     0  0  0  0  0  0  0  0  2G             Barnyardgrass                     2G 3G 4G 5G 0  0  0  0  4G             Johnsongrass                     2G 3G 6G 7G 0  0  0  4G 7G             Crabgrass                     0  0  0  0  0  0  0  0  0             Nutsedge                     0  3G 6G 9G 0  5G 9G 10E                                             10E             Velvetleaf                     3G 8G 10G                              10G                                 2G 6G 6G 8G 9G             Sicklepod                     0  7G 8G 10G                                 0  4G 6G 7G 9G             Lambsquarter                     6G 10C                           10E                              10E                                 0  3G 5G 8G 9G             Pigweed 8G 10C                           10G                              10E                                 0  5G 8G 10G                                             10G             Bindweed                     6G 9G 10G                              10G                                 4G 8G 9G 10G                                             10G             Jimsonweed                     6G 9G 10G                              10E                                 0  2G 7G 8G 9G             Prickly sida                     3G 7G 9G 10G                                 0  2G 6G 8G 9G             Sesbania                     0  5G 8G 10G                                 0  0  4G 7G 9G             Purslane                     7G 9G 10G                              10G                                 5G 8G 10G                                          10G                                             10G             Morningglory                     5G 8G 10G                              10G                                 0  0  4G 8G 9G             Cocklebur                     5G 10G                           10E                              10E                                 5G 6G 9G 10G                                             10G__________________________________________________________________________ 
    
     TEST D 
     This test was conducted utilizing 25 cm and 12.5 cm diameter pots filled with a light soil. The large size pots were planted to either corn or soybeans, 5-8 plants per pot. The small pots were planted to the following weed species, one species per pot: morning-glory (Ipomoea Hederacea var. hederacea), velvetleaf (Abutilon theophrasti), cocklebur (Xanthium pensylvanicum), pigweed (Amaranthus retroflexus), giant foxtail (Setaria faberi), johnsongrass (Sorghum halepense), crabgrass (Digitaria sp.) and barnyardgrass (Echinochloa crusgalli). The plantings were treated preemergence with the test chemical dissolved in a nonphytotoxic solvent. At the same time, the same crops and weed species, from plantings made 10-22 days previously, were treated with soil/foliage applications. There were three replications of each treatment. Reponse data were collected approximately 17 days after treatment for the postemergence phase of the test and approximately 27 days after treatment for the preemergence phase. The weed species were visually rated for injury. The crop plantings contained an equal number of plants per pot for each crop. At the time of rating, total fresh weights per pot were determined of the above-ground portions of the crop plants. Growth since treatment was then calculated and expressed as a percentage of untreated controls. The response data were averaged for the three replications and are shown in Table D. 
     Compound No. 1 controlled several weed species at rates of application which were noninjurious to corn. 
     
                       TABLE D______________________________________      Compound 1      % injury/% controlRate g/ha    250     125     62   31   16   8______________________________________POSTEMERGENCECorn         23      22      11   6    --   --Soybean      80      78      79   77   --   --Velvetleaf   --      --      98   97   95   93Pigweed      --      --      88   95   88   60Ivyleaf morningglory        --      --      96   96   93   90Cocklebur    --      --      99   98   97   91Crabgrass    --      --      0    0    0    0Giant foxtail        --      --      21   13   0    0Johnsongrass --      --      80   50   0    0Barnyardgrass        --      --      0    0    0    0PREEMERGENCECorn         54      38      25   23   --   --Soybean      81      79      74   66   --   --Velvetleaf   --      --      98   85   75   36Pigweed      --      --      97   95   86   78Ivyleaf morningglory        --      --      95   78   46   11Cocklebur    --      --      85   90   75   46Crabgrass    --      --      0    0    0    0Giant foxtail        --      --      10   6    0    0Johnsongrass --      --      71   33   50   0Barnyardgrass        --      --      18   6    0    0______________________________________      Compound 1      % injury/% controlRate g/ha    125     62     31  16  8    4    2______________________________________POSTEMERGENCECorn         30      22     12  15  --   --   --Soybean      --      --     79  75  70   67   --Velvetleaf   --      --     --  95  95   81   31Pigweed      --      --     --  86  91   78   46Ivyleaf morningglory        --      --     --  96  96   91   81Cocklebur    --      --     --  98  98   94   76Crabgrass    --      0      0   0   0    --   --Giant foxtail        --      6      0   0   0    --   --Johnsongrass --      60     30  13  0    --   --Barnyardgrass        --      0      0   0   0    --   --PREEMERGENCECorn       33      23     8    9    --   --   --Soybean    --      --     53   36   28   5    --Velvetleaf --      --     --   86   50   43   0Pigweed    --      --     --   89   73   56   0Ivyleaf morningglory      --      --     --   63   13   0    0Cocklebur  --      --     --   83   56   16   0Crabgrass  --      0      0    0    0    --   --Giant foxtail      --      40     33   20   0    --   --Johnsongrass      --      86     46   13   0    --   --Barnyardgrass      --      16     0    0    0    --   --______________________________________