SUBSTITUTED PYRIDINE HERBICIDES

Abstract: Compounds of formula (I), in which the substituents are as defined in claim 1 and the agrochemically tolerated salts M<+> and all stereoisomers and tautomers of the compounds of formula (I) are suitable for use as herbicides.

Description: SUBSTITUTED PYRIDINE HERBICIDES The present invention relates to novel, herbicidally active pyridine ketones, to their preparation, to compositions comprising these compounds, and to their use for controlling weeds, especially in crops of useful plants, or for inhibiting plant growth. Herbicidally active pyridine ketones are described, for example, in WO 97/46530. There have now been found novel pyridine ketones which have herbicidal and growth-inhibitory properties. The present invention therefore relates to compounds of the formula I in which p is 0 or 1 ; R 5 is d-Cehaloalkyl; R 2 is hydrogen, Cι-C 6 alkyl, CrC 6 haloalkyl, C 2 -C 6 alkenyl, C 2 -C 6 haloalkenyl, vinyl which is substituted by d-C 2 alkoxycarbonyl or phenyl, or is C 2 -C 6 alkynyl, C 2 -C 6 haloalkynyl, ethynyl which is substituted by trimethylsilyl, hydroxyl, d-C 2 alkoxy, d-C 2 alkoxycarbonyl or phenyl, or is C 3 -C 6 allenyl, C 3 -C 6 cycloalkyl, C 3 -C 6 cycloalkyl which is substituted by halogen, or is d-C 6 alkoxy, C 3 -C 6 alkenyloxy, C 3 -C 6 alkynyloxy, d-C 6 haloalkoxy, C 3 -C 6 haloalkenyloxy, cyano-C C 4 alkoxy, d-C alkoxy-d-C 4 alkoxy, d-C 4 alkylthio-Cι-C 4 alkoxy, Cι-C 4 alkylsulfinyl- d-C alkoxy, Cι-C 4 alkylsulfonyl-CrC 4 alkoxy, Cι-C 4 alkoxycarbonyl-d-C alkoxy, Cι- 6 alkylthio, d-C 6 alkylsulfinyl, d-C 6 alkylsulfonyl, d-C 6 haloalkylthio, d-C 6 haloalkylsulfinyl, CrCehaloalkylsulfonyl, d-dalkoxycarbonyl-Cι-C 4 alkylthio, C C 4 alkoxycarbonyl- CrC 4 aIkylsulfinyl, d-C 4 alkoxycarbonyl-d-C 4 alkylsulfonyl, benzyI-S(O) n ι-, d-C 6 alkylamino, C 2 -C 6 dialkylamino, CrC 6 alkylaminosulfonyl, di-(d-C 6 alkylamino)sulfonyl, benzyloxy, benzyl, phenyl, phenoxy, phenylthio, phenylsulfinyl or phenylsulfonyl, it being possible for the phenyl- containing groups, in turn, to be substituted by d-C 3 alkyl, d-C 3 haloalkyl, Cι-C 3 alkoxy, d- C 3 haloalkoxy, halogen, cyano or nitro or R 2 is OS(O) n2 -R 2 i, N(R 23 )-S(O) n3 -R22, cyano, carbamoyl, d-C 4 alkoxycarbonyl, formyl, halogen, thiocyanato, amino, hydroxy-d-C 4 alkyl, d-dalkoxy-d-dalkyl, C 1 -C 4 alkyl-S(0) n4 -C 1 -C 4 alkyl, cyano-d-C 4 alkyl, C C 6 alkylcarbonyloxy-CrC 4 alkyl, CrC 4 alkoxycarbonyl-d-C 4 alkyI, d-C 4 alkoxycarbonyloxy-d- C 4 alkyl, C C thiocyanato-d-C 4 alkyl, benzoyloxy-d-C 4 alkyl, C 2 -C 6 oxiranyl, Cι-C 4 alkylamino- d-C alkyl, di-(Cι-C 4 -alkyl)amino-d-C alkyl, d-C 12 alkylthiocarbonyl-d-C 4 alkyl or formyl-d- C 4 alkyl, or R 2 is a five- to ten-membered monocyclic or fused bicyclic ring system which can be aromatic or partially saturated and can contain 1 to 4 hetero atoms selected from the group consisting of nitrogen, oxygen and sulfur, the ring system being bonded to the pyridine ring via a C C 4 alkylene, -CH=CH-, -C≡C-, -CH 2 O-, -CH 2 N(C 1 -C 4 alkyl)- I -CH 2 SO-, or -CH 2 SO 2 group and it not being possible for each ring system to contain more than 2 oxygen atoms and not more than 2 sulfur atoms, and it being possible for the ring system itself to be mono-, di- or trisubstituted by d-C 6 alkyl, d-C 6 haloalkyl, C 3 -C 6 alkenyl, C 3 -C 6 haloalkenyl, C 3 - C 6 alkynyl, C 3 -C 6 haloalkynyl, d-C 6 alkoxy, d-C 6 haloalkoxy, C 3 -C 6 alkenyloxy, C 3 - C 6 alkynyloxy, mercapto, d-C 6 alkylthio, d-C 6 haloalkylthio, C 3 -C 6 alkenylthio, C 3 - C 6 haloalkenylthio, C 3 -C 6 alkynylthio, C 2 -C 5 alkoxyalkylthio, C 3 -C 5 acetylalkylthio, C 3 - C 6 alkoxycarbonylalkylthio, C 2 -C 4 cyanoalkylthio, d-C 6 alkylsulfinyl, CrC 6 haloalkylsulfinyl, d- C 6 alkylsulfonyl, Cι-C 6 haloalkylsulfonyl, aminosulfonyl, d-C 2 alkylaminosulfonyl, di-(d- C 2 alkyl)aminosulfonyl, di-(d-C 4 alkyl)amino, halogen, cyano, nitro, phenyl and benzylthio, it being possible for phenyl and benzylthio, in turn, to be substituted on the phenyl ring by d- C 3 alkyl, d-C 3 haloalkyl, d-C 3 alkoxy, C C 3 haloalkoxy, halogen, cyano or nitro, and substituents on the nitrogen in the heterocyclic ring being other than halogen; R 3 is hydrogen, d-C 6 alkyl, d-C 6 haloalkyl, C 2 -C 6 alkenyl, C 2 -C 6 haloalkenyl, C 2 -C 6 alkynyl, C 2 -C 6 haloalkynyl, C 3 -C 6 cycloalkyl, d-C 6 alkoxy, d-C 6 haloalkoxy, d-Cβalkylthio, d-C 6 alkylsulfinyl, d-C 6 alkylsulfonyl, d-C 6 haloalkylthio, d-C 6 haloalkylsulfinyl, CrCehaloalkylsulfonyl, d-Cealkylamino, C 2 -C 6 dialkylamino, CrC 6 alkylaminosulfonyl, C 2 -C 6 dialkylaminosulfonyl, phenyl, phenylthio, phenylsulfinyl, phenylsulfonyl or phenoxy, it being possible for phenyl, in turn, to be substituted by d-C 3 alkyl, d-C 3 haloalkyl, d- C 3 alkoxy, C C 3 haloalkoxy, halogen, cyano or nitro, or R 3 is -N(R 23 )-S(O) n -R22, cyano, halogen, amino, d-C 4 alkoxy-Cι-C 4 alkyl or d-C 4 alkyl-S(O) n -Cι-C 4 .alkyl; R 4 is hydrogen, d-C 6 alkyl, hydroxyl, d-C 6 alkoxy, d-C 6 haloalkoxy, C 3 -C 6 alkenyloxy, C 3 -C 6 haloalkenyloxy, C 3 -C 6 alkynyloxy, d-C 4 alkylcarbonyloxy, d-C 4 alkylsulfonyloxy, tosyloxy, C C 4 alkylthio, d-C alkylsulfinyl, Cι-C 4 alkylsulfonyl, Cι-C 4 alkylamino, CrC dialkylamino, Cι-C 4 alkoxycarbonyl, C C 4 haloalkyl, formyl, cyano, halogen, phenyl or phenoxy, it being possible for phenyl, in turn, to be substituted by d-C 3 alkyI, d-C 3 haloalkyl, d-C 3 alkoxy, Cι-C 3 haloalkoxy, halogen, cyano or nitro; or R 4 is a five to ten-membered monocyclic or R 3 -fused bicyclic ring system which can contain 1 to 4 hetero atoms selected from the group consisting of nitrogen, oxygen and sulfur, the ring system, unless fused, being bonded to the pyridine ring directly or via a d-C 4 alkylene, -CH=CH-, -C≡C-, -CH 2 O- , -CH 2 N(Cι-C 4 alkyl)-, -CH 2 S-, -CH 2 SO- ( or -CH 2 SO 2 - group and it not being possible for the ring system to contain more than 2 oxygen atoms and not more than two sulfur atoms, and it being possible for the ring system itself to be mono-, di- or trisubstituted by d-C 6 alkyl, Cι-C 6 haloalkyl, C 2 -C 6 alkenyl, C 2 -C 6 haloalkenyl, C 2 -C 6 alkynyl, C 2 -C 6 haloalkynyl, d-C 6 alkoxy, d-C- 6 haloalkoxy, C 3 -C 6 alkenyloxy, C 3 -C 6 alkynyloxy, d-C 6 alkylthio, d-C 6 haloalkylthio, C 3 -C 6 alkenylthio, C 3 -C 6 haloalkenylthio, C 3 -C 6 alkynylthio, d-C 4 alkoxy-CrC 2 alkylthio, C 1 -C 4 alkylcarbonyl-C 1 -C 2 alkylthio, C 1 -C 4 alkoxycarbonyl-C C 2 alkylthio, cyano-d-C 4 alkylthio, d-C 6 alkylsulfinyl, Cj-Cehaloalkylsulfinyl, d-C 6 alkylsulfonyl, CrC 6 haloalkylsulfonyl, aminosulfonyl, d-C 2 alkylaminosulfonyl, di-(d-C 2 alkyl)aminosulfonyl, di-(d-C 4 alkyl)amino, halogen, cyano, nitro, phenyl and benzylthio, it being possible for phenyl and benzylthio, in turn, to be substituted on the phenyl ring by C C 3 alkyl, d-C 3 haloalkyl, d-C 3 alkoxy, d-C 3 haloalkoxy, halogen, cyano or nitro, and substituents on the nitrogen in the heterocyclic ring being other than halogen; R 21 is d-C 4 alkyl or d-C haloalkyl; R 22 is d-C alkyl, C C 4 haloalkyl or di-(d-C 4 alkyl)amino; R 23 , R 24 , R 2 5 independently of one another are hydrogen or Cι-C 4 alkyl; n, n^ n 2 , n 3 and n 4 independently of one another are 0, 1 or 2; Q is Qi in which R 6 , R , Re and R 9 independently of one another are hydrogen, d-C 6 alkyl, d-C 6 haloalkyI, C 2 -C 6 alkenyl, C 2 -C 6 alkynyl, d-C 6 alkoxycarbonyl, d-C 6 alkylcarbonyl, C 1 -C 6 alkyl-S(O) n ι , C 1 -C 6 alkyl-NHS(O) 2 , d-C 6 alkylamino, di-(CrC 6 alkyl)amino, hydroxyl, d-C 6 aIkoxy, C 3 -C 6 alkenyloxy, C 3 -C 6 alkynyloxy, hydroxy-d-C 6 alkyl, d-C 4 alkyIsulfonyloxy-Cι-C 6 alkyl, tosyloxy-d-C 6 alkyl, C C 6 alkoxy-CrC 6 alkyl, Cι-Cβalky.-S(0) π4 -Cι-Cβalkyl, cyano-d-C 6 alkyl, CrCβalkoxy-CrCealkoxy, benzyloxy-Cι-C 6 alkyl, CrC 6 alkoxycarbonyl-Ci-C 6 alkyl, d-Cealkoxycarbonyloxy-d-Cealkyl, thiocyanato-d-C 6 alkyl, oxiranyl, d-C 6 alkylamino- d-C 6 alkyl, di(C 1 -C 6 alkyl)amino-C 1 -C 6 alkyl, formyl-Cι-C 6 alkyl, d-Cealkyloximo, halogen, cyano, nitro, phenyl or phenyl which is substituted by C C alkyl, C C 4 haloalkyl, d-C alkoxy, C C 4 haloalkoxy, Cι-C alkylcarbonyl, Cι-C alkoxycarbonyl, amino, Cι-C 4 alkylamino, di- Cι-C 4 alkylamino, Cι-C 4 alkyl-S(O) n ι 8 , Cι-C 4 alkyl-S(O) 2 O, d-C 4 haloalkyl-S(O)n 5 , d-C 4 haloalkyl-S(O) 2 O, d-C 4 alkyl-S(O) 2 NH, d-C 4 alkyl-S(O) n19 N(Cι-C 4 alkyl) 2 , halogen, nitro, COOH or cyano; or adjacent R 6 and R 7 or R 8 and R 9 together are -(CH 2 )m- , C(O)O(CH 2 ) n 2o- or r) 5 , n 17 , n 18 , nι 9 and n 2 ι independently of one another are 0, 1 or 2; n 20 is 2 or 3; n 22 is 2, 3 or 4; m is 2, 3, 4, 5, or 6; W is oxygen, -C(O)- or -NR 13 ; R6 3 , 6 4 , Res and R 6 6 independently of one another are hydrogen or d-C 6 alkyl, or R 65 together with R 7 or R 9 forms a direct bond; n 6 is 0, 1 or 2; Rn is hydrogen, C C 4 alkyl, d-C 4 haloalkyl, Cι-C alkoxy-d-C 4 alkyl, C C 4 alkylthio-d- C 4 alkyl, d-C 4 alkylthio-C 3 -C 6 cycloalkyl, d-C 4 alkycarbonyloxy-d-C 4 alkyl, Ci- C 4 alkysulfonyloxy-Cι-C 4 alkyl, tosyloxy-C C alkyl, di-(Cι-C 3 alkoxyalkyl)methyl, di-(C C 3 aIkthioalkyl)methyl, (Cι-C 3 alkoxyalkyl)-(C 1 -C 3 alkthioalkyl)methyl, C 3 -C 5 oxacycloalkyl, C 3 - C 5 thiacycloalkyl, C 3 -C 4 dioxacycloalkyl, C 3 -C 4 dithiacycloalkyl, C 3 -C 4 oxathiacycloalkyl, formyl, C C 4 alkoxycarbonyl, carbamoyl, CrC 4 alkylaminocarbonyI, di-(C 1 -C 4 alkyl)aminocarbonyl, phenylaminocarbonyl, benzylaminocarbonyl or phenyl which, in turn, can be substituted by d-C 4 alkyl, d-C 4 haloalkyl, d-C 4 haloalkoxy, d-C 4 alkylcarbonyl, CrC 4 alkoxycarbonyl, amino, Cι-C 4 alkylamino, di-Cι-C 4 alkylamino, C C^lkyl-SCO),,^, d-C 4 alkyl-S(O) 2 O, d-C 4 haloalkyl-S(O) n 7, C C 4 haloalkyl-S(O) 2 O, d-C 4 alkyl-S(O) 2 NH, C 1 -C 4 alkyl-S(O) n20 N(C 1 -C 4 alkyl), halogen, nitro, COOH or cyano; n 7 , n 2o and n 2 ι independently of one another are 0, 1 or 2; or R 12 together with R 6 or R 9 is a group -(CH 2 ) 0 -; o is 1 , 2, 3, 4 or 5; R 12 is hydrogen, C C 4 alkyl or d-C 4 haloalkyl; or R12 together with Rn is a group -(CH 2 )mi; ITH is 2, 3, 4, 5, or 6; R 10 is hydroxyl, O " M + , halogen, cyano, SCN, OCN, C^C^alkoxy, C^dalkoxycarbonyl- C Cι 2 alkylsulfonyl, CrC 12 haloalkylthio, CrC^haloalkylsulfinyl, d-d ∑ haloalkylsulfonyl, CrCealkoxy-d-Cβalkylthio, d-C 6 alkoxy-Cr C 6 alkylsulfinyl, CrCealkoxy-Ci-Cβalkylsulfonyl, C 2 -Cι 2 alkenylthio, C 2 -Cι 2 alkenylsulfinyl, C 2 - C 12 alkenylsulfonyl, C 2 -C 12 alkynylthio, C 2 -C 2 alkynylsulfinyl, C 2 -Cι 2 alkynylsulfonyl, C 2 - C 12 haloalkenylthio, C 2 -C 12 haloalkenylsulfinyl, C 2 -C 12 haloalkenylsulfonyl, d-C 4 - alkoxycarbonyl-C C 4 alkylthio, C C 4 alkoxycarbonyl-Cι-C 4 alkylsulfinyl, C C 4 alkoxycarbonyl- d-C 4 alkylsulfonyl, (d-C 4 alkoxy) 2 P(O)O, d-C 4 alkyl-(Cι-C 4 alkoxy)P(O)O, H(C C 4 alkoxy)P(O)O, R 14 Rι 5 N, R 14 R 15 NNH, R 16 Rι 7 NC(O)O-, R 16 R 17 NC(O)NH-, C C 12 alkyl- S(O) 2 NR 18 , Cι-C 4 haloalkyl-S(O) 2 NR 19 , d-C 12 alkyl-S(O) 2 O, C C 4 haloalkyl-S(O) 2 O, d- C 18 alkylcarbonyloxy, it being possible for the alkyl group to be substituted by halogen, d- C 6 alkoxy, d-C 6 alkylthio or cyano, or is C 2 -Cι 8 alkenylcarbonyloxy, C 2 -Cι 8 alkynylcarbonyloxy, C 3 -C 6 cycloalkylcarbonyloxy, CrCi ∑ alkoxycarbonyloxy, d-Cι 2 alkylthiocarbonyloxy, C Cι 2 alkylthiocarbamoyl, d-C 6 alkyl-NH(CS)N(d-C 6 alkyl)-NH-, di-d-C 6 alkyl-N(CS)N(d- C 6 alkyl)-NH-, benzyloxy, benzylthio, benzylsulfinyl, benzylsulfonyl, phenoxy, phenylthio, phenylsulfinyl, phenylsulfonyl, phenylsulfonylamino, phenylsulfonyloxy or benzoyloxy, it being possible for the phenyl groups, in turn, to be substituted by C C 4 alkyl, Cι-C 4 haloalkyl, d- C 4 alkoxy, Cι-C 4 haloalkoxy, d-C 4 alkylcarbonyl, d-C 4 alkoxycarbonyl, d-C 4 alkylamino, di-C C 4 alkylamino, C C 4 alkylthio, d-C 4 alkylsulfinyl, d-C 4 alkylsulfonyl, d-C 4 alkyl-S(O) 2 O, d-C 4 haloalkylthio, C C 4 haloalkylsulfinyl, C C 4 haloalkylsulfonyl, d-C 4 haloalkyl-S(O) 2 O, d- C 4 alkyl-S(O) 2 NH, d-C 4 alkyl-S(O) 2 N(d-dalkyl), halogen, nitro or cyano; or R 10 is a group Ar thio, Ar 2 -sulfinyl, Ar 3 -sulfonyl, -OCO-Ar 4 or NH-Ar 5 in which Ar 1 ( Ar 2 , Ar 3 , Ar 4 and Ar 5 independently of one another are a five- to ten-membered monocyclic or fused bicyclic ring system which can be aromatic or partially saturated and can contain 1 to 4 hetero atoms selected from the group consisting of nitrogen, oxygen and sulfur, and it being possible for each ring system to contain not more than 2 oxygen atoms and not more than two sulfur atoms, and it being possible for the ring system itself to be mono-, di- or trisubstituted by d-C-ealkyl, d-C 6 haloalkyl, C 3 -C 6 alkenyl, C 3 -C 6 haloalkenyl, C 3 -C 6 alkynyl, C 3 -C 6 haloalkynyl, d-C 6 alkoxy, d-C 6 haloalkoxy, C 3 -C 6 alkenyloxy, C 3 -C 6 alkynyloxy, mercapto, d-C 6 alkylthio, d-C 6 haloalkylthio, C 3 -C 6 alkenylthio, C 3 -C 6 haloalkenylthio, C 3 - C 6 alkynylthio, C 2 -C 5 alkoxyalkylthio, C 3 -C 5 acetylalkylthio, C 3 -C 6 alkoxycarbonylalkylthio, C 2 -C - cyanoalkylthio, d-C 6 alkylsulfinyl, d-C 6 haloalkylsulfinyl, C C 6 alkylsulfonyl, C C 6 - haloalkylsulfonyl, aminosulfonyl, CrC 2 alkylaminosulfonyl, di-(Cι-C 2 alkyl)aminosulfonyl, di- (Cι-C 4 alkyl)amino, halogen, cyano, nitro, phenyl and benzylthio, it being possible for phenyl and benzylthio, in turn, to be substituted on the phenyl ring by d-C 3 alkyl, C C 3 haloalkyl, d-C 3 alkoxy, d-C 3 haloalkoxy, halogen, cyano or nitro, and where substituents on the nitrogen in the heterocyclic ring are other than halogen; Rι . R 15 , R 16 . R 17 and R 8 independently of one another are hydrogen or d-C 6 alkyl; n 8 , n 9 , n 10 , n 11 ? nι 2 , n 13 and n 14 independently of one another are 0, 1 or 2; R 13 is hydrogen, d-C 4 alkyl, Cι-C alkythio-d-C 4 carbonyl, CrC alkylsulfinyI-d-C 4 carbonyl, d-C 4 alkylsulfonyl-Cι-C 4 carbonyl, d-C 4 alkoxycarbonyl, Cι-C 4 alkylcarbonyl, phenylcarbonyl, or is phenyl which, in turn, can be substituted by Cι-C alkyl, d-C haloalkyl, Cι-C 4 alkoxy, CrC 4 haloalkoxy, Cι-C 4 alkylcarbonyl, C C 4 alkoxycarbonyl, Cι-C 4 alkylamino, di-d-C 4 - alkylamino, d-C 4 alkyl-S(O) n15 , d-C 4 alkyl-S(O) 2 O, C 1 -C 4 haloalkyl-S(0) n ιβ, C C 4 haloalkyl- S(O) 2 O, d-C 4 alkyl-S(O) 2 NH, C C 4 alkyl-S(O) 2 N(d-C 4 alkyl), halogen, nitro, or cyano; and n 15 and n 16 independently of one another are 0, 1 or 2; and the agrochemically tolerated salts M + and all stereoisomers and tautomers of the compounds of the formula I. The alkyl groups in the definitions of the substituents can be straight-chain or branched and are, for example, methyl, ethyl, n-propyl, iso-propyl, n-butyl, sec-butyl, iso-butyl, tert-butyl, pentyl, hexyl, heptyl, octyl, nonyl, decyi, undecyl and dodecyl and their branched isomers. Alkoxy, alkenyl and alkynyl radicals are derived from the abovementioned alkyl radicals. The alkenyl and alkynyl groups can be mono- or polyunsaturated. An alkylene group for example, -(CH 2 ) m -, -(CH 2 ) m ι- or -(CH 2 ) 0 - can be substituted by one or more methyl group; preferably, such alkylene groups are in each case unsubstituted. The same also applies to the -C(O)O(CH 2 ) n20 - and -S(O) n21 (CH 2 ) n22 - group and to all C 3 -C 6 - cycloalkyl-, C 3 -C 5 oxacycloalkyl-, C 3 -C 5 thiacycloalkyl-, C 3 -C 4 dioxacycloalkyl-, C 3 -C 4 - dithiacycloalkyl-, C 3 -C 4 oxathiacycloalkyl-containing groups. Halogen is, as a rule, fluorine, chlorine, bromine or iodine. This also applies analogously to halogen in conjunction with other meanings such as haloalkyl or halophenyl. Haloalkyl groups with a chain length of 1 up to 6 carbon atoms are, for example, fluoromethyl, difluoromethyl, trifluoromethyl, chloromethyl, dichloromethyl, trichioromethyl, 2,2,2-trifluoroethyl, 1 -fluoroethyl, 2-fluoroethyl, 2-chloroethyl, 2-fluoroprop-2-yl, pentafluoroethyl, 1 ,1-difluoro-2,2,2-trichloroethyl, 2,2,3,3-tetrafluoroethyl and 2,2,2- trichloroethyl, pentafluoroethyl, heptafluoro-n-propyl, perfluoro-n-hexyl; haloalkyl groups in the meanings R 2 , R 3 and, in particular, R 5 are preferably trichloromethyl, fluoromethyl, dichlorofluoromethyl, difluorochloromethyl, difluoromethyl, trifluoromethyl, pentafluoroethyl or heptafluoro-n-propyl. Suitable as haloalkyl are monohalogenated or polyhalogenated alkenyl groups, where halogen is fluorine, chlorine, bromine and iodine, and in particular fluorine and chlorine, for example 1 -chlorovinyl, 2-chlorovinyl, 2,2-difluorovinyl, 2,2-difluoroprop-1 -en-2-yl, 2,2-dichlorovinyl, 3-fluoroprop-1-enyl, chloroprop-1-en-1 -yl, 3-bromoprop-1-en-1 -yl, 2,3,3-trifluoroprop-2-en-1 -yl, 2,3,3-trichloroprop-2-en-1 -yl and 4,4,4-trif luorobut-2-en-1 -yl. Preferred amongst the monohalogenated, dihalogenated or trihalogenated C 2 -C 6 alkenyl groups are those which have a chain length of 2 to 5 carbon atoms. Suitable as haloalkynyl are, for example, monohalogenated or polyhalogenated alkynyl groups, where halogen is bromine, iodine and, in particular, fluorine and chlorine, for example 3-fluoropropynyl, 3-chloropropynyl, 3-bromopropynyl, 3,3,3-trifluoropropynyl and 4,4,4-trifluorobut-2-yn-1 -yl. Preferred amongst the monohalogenated or polyhalogenated alkynyl groups are those which have a chain length of 2 to 5 carbon atoms. A monohalogenated or polyhalogenated C 3 -C 6 cycloalkyl group is, for example, the 2,2- dichlorocyclopropyl, 2,2-dibromocyclopropyl, 2,2,3,3-tetrafluorocyclobutyl or 2,2-difluoro-3,3- dichlorocyclobutyl group. Alkoxy groups preferably have a chain length of 1 to 6 carbon atoms. Alkoxy is, for example, methoxy, ethoxy, propoxy, i-propoxy, n-butoxy, iso-butoxy, sec-butoxy and tert-butoxy and the pentyloxy and hexyloxy isomers; preferably methoxy and ethoxy. Alkylcarbonyl is preferably acetyl or propionyl. Alkoxycarbonyl is, for example, methoxycarbonyl, ethoxycarbonyl, propoxycarbonyl, iso-propoxycarbonyl, n-butoxycarbonyl, iso- butoxycarbonyl, sec-butoxycarbonyl or tert-butoxycarbonyl; preferably methoxycarbonyl, ethoxycarbonyl or tert-butoxycarbonyl. Haloalkoxy groups preferably have a chain length of 1 to 6 carbon atoms. Haloalkoxy is, for example, fluoromethoxy, difluoromethoxy, trifluoromethoxy, 2,2,2-trifluoro- ethoxy, 1 ,1 ,2,2-tetrafluoroethoxy, 1 -f luoroethoxy, 2-fluoroethoxy, 2-chloroethoxy, 2,2- difluoroethoxy and 2,2,2-trichloroethoxy; preferably fluoromethoxy, difluoromethoxy, 2-chloroethoxy and trifluoromethoxy. Alkylthio groups preferably have a chain length of 1 to 8 carbon atoms. Alkylthio is, for example, methylthio, ethylthio, propylthio, iso-propylthio, n-butylthio, iso-butylthio, sec- butylthio or tert-butylthio, preferably methylthio and ethylthio. Alkylsulfinyl is, for example, methylsulfinyl, ethylsulfinyl, propylsulfinyl, iso-propylsulfinyl, n-butylsulfinyl, iso-butylsulfinyl, sec-butylsulfinyl, tert-butylsulfinyl; preferably methylsulfinyl and ethylsulfinyl. Alkylsulfonyl is, for example, methylsulfonyl, ethylsulfonyl, propylsulfonyl, iso-propylsulfonyl, n-butylsulfonyl, iso-butylsulfonyl, sec-butylsulfonyl or tert-butylsulfonyl; preferably methylsulfonyl or ethylsulfonyl. Alkylamino is, for example, methylamino, ethylamino, n-propylamino, iso-propylamino or the butylamino isomers. Dialkylamino is, for example, dimethylamino, methylethylamino, diethylamino, n-propylmethylamino, di-butylamino and di-iso-propylamino. Preferred are alkylamino groups having a chain length of 1 to 4 carbon atoms. Alkoxyalkyl groups preferably have 1 to 6 carbon atoms. Alkoxyalkyl is, for example, methoxymethyl, methoxyethyl, ethoxymethyl, ethoxyethyl, n-propoxymethyl, n-propoxyethyl, iso- propoxymethyl or iso-propoxyethyl. Alkylthioalkyl groups preferably have 1 to 6 carbon atoms. Alkylthioalkyl is, for example, methylthiomethyl, methylthioethyl, ethylthiomethyl, ethylthioethyl, n-propylthiomethyl, n-propylthioethyl, iso-propylthiomethyl, iso-propylthioethyl, butylthiomethyl, butylthioethyl or butylthiobutyl. Phenyl, also as part of a substituent such as phenoxy, benzyl, benzyloxy, benzoyl, phenylthio, phenylalkyl, phenoxyalkyl or tosyl can be in monosubstituted or polysubstituted form. In this case, the substituents can be in any of the ortho, meta and/or para position(s). Allenyl is, for example, CH 2 =C=CH 2 CH 2 =CH-CH 2 -CH=CH 2 , CH 2 =CH-CH 2 -CH 2 -CH=CH 2 or The invention also extends to the salts M + which the compounds of the formula I, in particular those compounds of the formula I in which R 10 is O " M + , can form, preferably with amines, alkali metal bases, alkaline earth metal bases or quaternary ammonium bases. The following must be emphasized as salt formers amongst the alkali metal bases and alkaline earth metal bases: the hydroxides of lithium, sodium, potassium, magnesium or calcium, in particular those of sodium or potassium. Examples of amines which are suitable for ammonium salt formation are not only ammonia, but also primary, secondary and tertiary Cι-C 18 alkylamines, C 1 -C hydroxyalkylamines and C 2 -C 4 alkoxyalkylamines, for example methylamine, ethylamine, n-propylamine, iso-propylamine, the four butylamine isomers, n-amylamine, iso-amylamine, hexylamine, heptylamine, octylamine, nonylamine, decylamine, pentadecylamine, hexadecylamine, heptadecylamine, octadecylamine, methylethylamine, methylisopropylamine, methylhexylamine, methylnonylamine, methyl-pentadecylamine, methyloctadecylamine, ethylbutylamine, ethylheptylamine, ethyloctylamine, hexylheptylamine, hexyloctylamine, dimethylamine, diethylamine, di-n-propylamine, di-iso- propylamine, di-n-butylamine, di-n-amylamine, di-iso-amylamine, dihexylamine, diheptylamine, dioctylamine, ethanolamine, n-propanolamine, iso-propanolamine, N,N- diethanolamine, N-ethylpropanolamine, N-butylethanolamine, allylamine, n-butenyl-2-amine, n-pentenyl-2-amine, 2,3-dimethylbutenyl-2-amine, dibutenyl-2-amine, n-hexenyl-2-amine, propylenediamine, trimethylamine, triethylamine, tri-n-propylamine, tri-iso-propylamine, tri-n- butylamine, tri-iso-butylamine, tri-sec-butylamine, tri-n-amylamine, methoxyethylamine and ethoxyethylamine; heterocyclic amines for example, pyridine, quinoline, iso-quinoline, morpholine, piperidine, pyrrolidine, indoline, quinuclidine and azepine; primary arylamines for example anilines, methoxyanilines, ethoxyanilines, o-, m-, p-toluidines, phenylenediamines, naphthylamines and o-, m- and p-chloroanilines; but in particular triethylamine, isopropylamine and di-iso-propylamine. Examples of quaternary ammonium bases which are suitable for salt formation are, for example, [N(R a R b R c R d )] + OH " , where R a , R , R c and R d independently of one another are d-C alkyl. Other suitable tetraalkylammonium bases with other anions can be obtained, for example, by anion exchange reactions. M + preferably represents an ammonium salt, in particular NH 4 + , or an alkali metal, in particular potassium or sodium. The compounds of the formula I can occur in various tautomeric forms, for example, if R 10 is hydroxyl, in the preferred formulation I' and I'" Preferred among the compounds of the formula I are those in which p is 0; R 5 is Cι-C 6 haloalkyl; R 2 is hydrogen, d-C 6 alkyl, d-C 6 haloalkyl, C 2 -C 6 alkenyl, C 2 -C 6 haloalkenyl, C 2 -C 6 alkynyl, C 2 -C 6 haloalkynyl, C 3 -C 6 cycloalkyl, d-C 6 alkoxy, CrC 6 haloalkoxy, d-C 6 alkylthio, Cι-C 6 - alkylsulfinyl, d-C 6 alkylsulfonyl, Cι-C 6 haloalkylthio, d-C 6 haloalkylsulfinyl, d-C 6 - haloalkylsulfonyl, benzyl-S(O) n r, Cι-C 6 alkylamino, C 2 -C 6 dialkylamino, d-C 6 - alkylaminosulfonyl, C 2 -C 6 -dialkylaminosulfonyl, phenyl, phenoxy, phenylthio, phenylsulfinyl or phenylsulfonyl, it being possible for the phenyl group, in turn, to be substituted by d-C 3 - alkyl, d-C 3 haloalkyl, d-C 3 alkoxy, d-C 3 haloalkoxy, halogen, cyano or nitro, or is OS(O) n2 - 2 i, N(R 23 )-S(O) n3 -R 22 , cyano, halogen, amino, Cι-C 4 alkoxy-C C alkyl, d-C alkyl- S(O) n4 -Cι-C 4 alkyl, cyano-C C 4 alkyl or d-C alkoxy-d-C 4 alkoxy; R 3 is hydrogen, d-C 6 alkyl, d-C 6 haloalkyl, C 2 -C 6 alkenyl, C 2 -C 6 haloalkenyl, C 2 -C 6 alkynyl, C 2 -C 6 haloalkynyl, C 3 -C 6 cycloalkyl, d-C 6 alkoxy, C C 6 haloalkoxy, d-C 6 alkylthio, d-C 6 - alkylsulfinyl, d-C 6 alkylsulfonyl, d-C 6 haloalkylthio, C C 6 haloalkylsulfinyl, d-C 6 - haloalkylsulfonyl, d-C-ealkylamino, C 2 -C 6 dialkylamino, d-C-ealkylaminosulfonyl, C 2 -C 6 - dialkylaminosulfonyl, phenyl, phenylthio, phenylsulfinyl, phenylsulfonyl or phenoxy, it being possible for phenyl, in turn, to be substituted by d-C 3 alkyl, d-C 3 haloalkyl, d-C 3 alkoxy, Cι-C 3 haloalkoxy, halogen, cyano or nitro, or is -N(R 23 )-S(O) n -R 22 , cyano, halogen, amino, CrC 4 alkoxy-C 1 -C 4 alkyl or d-dalkyl-SCOJ n -d-dalkyl; R 4 is hydrogen, d-C 6 alkyl, Cι-C alkoxy, d-C 4 haloalkoxy, Cι-C alkylcarbonyloxy, C C 4 - alkylthio, d-C 4 alkylsulfinyl, C C 4 alkylsulfonyl, d-C 4 haloalkyl, formyl, cyano, halogen, phenyl or phenoxy, it being possible for phenyl, in turn, to be substituted by d-C 3 alkyl, Cι-C 3 haloalkyl, d-C 3 alkoxy, d-C 3 haloalkoxy, halogen, cyano or nitro; or R 4 is a five- to ten-membered monocyclic or R 3 -fused bicyclic ring system which can contain 1 to 4 hetero atoms selected from the group consisting of nitrogen, oxygen and sulfur, the ring system being bonded to the pyridine ring via a Cι-C alkylene group and it not being possible for the ring system to contain more than 2 oxygen atoms and not more than two sulfur atoms, and it being possible for the ring system itself to be mono-, di- or trisubstituted by d-C 6 alkyl, C C 6 haloalkyl, C 2 -C 6 alkenyl, C 2 -C 6 haloalkenyl, C 2 -C 6 alkynyl, C 2 -C 6 haloalkynyl, d-C 6 alkoxy, Cι-C 6 haloalkoxy, C 3 -C 6 alkenyloxy, C 3 -C 6 alkynyloxy, d-C 6 - Alkylthio, d-C 6 haloalkylthio, C 3 -C 6 alkenylthio, C 3 -C 6 haloalkenylthio, C 3 -C 6 alkynylthio, d-C 4 - alkoxy-C C 2 alkylthio, C -C 4 alkylcarbonyl-C 1 -C 2 alkylthio, d-C 4 alkoxycarbonyl-Ci-C 2 alkylthio, cyano-d-C 4 alkylthio, d-C 6 alkylsulfinyl, d-C 6 haloalkylsulfinyl, Cι-C 6 alkylsulfonyl, C C 6 - haloalkylsulfonyl, aminosulfonyl, CrC 2 alkylaminosulfonyl, C 2 -C 4 dialkylaminosulfonyl, halogen, cyano, nitro, phenyl and benzylthio, it being possible for phenyl and benzylthio, in turn, to be substituted on the phenyl ring by d-C 3 alkyl, d-C 3 haloalkyl, d-C 3 alkoxy, d-C 3 - haloalkoxy, halogen, cyano or nitro, and where substituents on the nitrogen in the heterocyclic ring are other than halogen; R 21 and R 22 independently of one another are C C 4 alkyl or d-C 4 haloalkyl; R 23 , R 24 and R 25 independently of one another are hydrogen or C C 4 alkyl; n, n 1 ( n 2 , n 3 and n 4 independently of one another are 0, 1 or 2; Q is Q ! in which R 6 , R 7 , R 8 and R 9 independently of one another are hydrogen, d-C 6 alkyl, d-C 6 haloalkyl, C 2 - C 6 alkenyl, C 2 -C 6 alkynyl, d-C 6 alkoxycarbonyl, Cι-C 6 alkyl-S(O) n17 , Cι-C 6 alkyl-NHS(O) 2 , Cι-C 6 aIkylamino, di-(d-C 6 alkyl)amino, hydroxyl, d-C 6 alkoxy, C 3 .C 6 alkenyloxy, C 3 -C 6 - alkynyloxy, hydroxy-CrC 6 alkyl, Cι-C 4 alkylsulfonyloxy-d-C 6 alkyl, tosyloxy-d-C 6 alkyl, halogen, cyano, nitro, phenyl or phenyl which is substituted by d-C 4 alkyl, d-C 4 haloalkyl, d-C 4 alkoxy, Cι-C 4 haloalkoxy, Cι-C 4 alkylcarbonyl, d-C 4 alkoxycarbonyl, amino, C C - alkylamino, di-d-C 4 alkylamino, d-C 4 alkyl-S(O) n18 , d-C 4 alkyl-S(O) 2 O, d-C 4 haloalkyl-S(O) n 5, d-C 4 haloalkyl-S(O) 2 O, d-C alkyl-S(O) 2 NH, d-C 4 alkyl-S(O) n ι 9 N(d-C 4 alkyl), halogen, nitro, COOH or cyano; or adjacent R 6 and R 7 or R 8 and R 9 together are -(CH 2 ) m -; n 5 nι , nι 8 and nι 9 independently of one another are 0, 1 or 2; m is 2, 3, 4, 5, or 6; W is oxygen, S(O) n6 , -CRn R. 2 -. -C(O)- or -NR 13 -; n 6 is 0, 1 or 2; Rn is hydrogen, d-C alkyl, d-C haloalkyl, d-C 4 alkoxy-Cι-C 4 alkyl, d-C alkylthio-d- C alkyl, d-C alkylcarbonyloxy-CrC alkyl, Cι-C 4 alkylsulfonyloxy-d-C 4 alkyl, tosyloxy-Ci- C 4 alkyl, di-(d-C 3 alkoxyalkyl)methyl, di-(d-C 3 alkylthioalkyl)methyl, (d-C 3 alkoxyalkyl)-(Cι- C 3 alkylthioalkyl)methyl, C 3 -C 5 oxacycloalkyl, C 3 -C 5 thiacycloalkyl, C 3 -C dioxacycloalkyl, C 3 -C 4 - dithiacycloalkyl, C 3 -C 4 oxathiacycloalkyl, formyl, Cι-C alkoxycarbonyl or phenyl which, in turn, can be substituted by d-C 4 alkyl, d-C 4 haloalkyl, d-C 4 alkoxy, C C 4 haloalkoxy, Cι-C 4 - alkylcarbonyl, d-C 4 alkoxycarbonyl, amino, Cι-C alkylamino, di-d-C alkylamino, d-C 4 alkyl- S(O) n2 ι, C dalkyl-S(O) 2 O, d-C 4 haloalkyl-S(O) n7 , Cι-C 4 haloalkyl-S(O) 2 O, C r C 4 alkyl- S(O) 2 NH, Cι-C 4 alkyl-S(O) n2 oN(d-C 4 alkyl), halogen, nitro, COOH or cyano; n 7 , n 20 and n 2 . independently of one another are 0, 1 or 2; or R 12 together with R 9 is a group -(CH 2 ) 0 -; o is 1 , 2, 3, 4 or 5; R 12 is hydrogen, C C alkyl or d-dhaloalkyl; or R 12 together with Rn is a group -(CH 2 ) m i; R 10 is hydroxyl, O " M + , halogen, d-Cι 2 alkoxy, CrC 12 alkylcarbonyloxy, C 2 -C 4 - alkenylcarbonyloxy, C 3 -C 6 cycloalkylcarbonyloxy, C Cι 2 alkoxycarbonyloxy, C 1 -C 12 - alkylcarbonyloxy, R 23 R 24 N-C(O)O, d-C 12 alkylS(O) n8 -, C 1 -C 4 haloalkyl-S(O) n9 -, C 2 -C 12 - alkenylS(O)nio-, C 2 -Cι 2 haloalkenylS(O) n n-, C2-C 12 alkynylS(O) n i2-; benzyloxy, phenoxy, phenylthio, phenylsulfinyl or phenylsulfonyl, where the phenyl group, in turn, can be substituted by Cι-C 4 alkyl, d-C 4 haloalkyl, d-C 4 alkoxy, C 1 -C 4 haloalkoxy, C C alkylcarbonyl, CrC 4 alkoxycarbonyl, C C 4 alkyIamino, di-C C 4 alkylamino, d-C 4 alkyl-S(O) n i 3 , C C 4 alkyl- S(O) 2 O, d-C 4 haloalkyl-S(O) n . . C C 4 haloalkyl-S(O) 2 O, C C 4 alkyl-S(O) 2 NH, C C 4 alkyl- S(O) 2 N(C C 4 alkyl), halogen, nitro or cyano, or is d-C 4 alkyl-S(O) 2 O, phenyl-S(O) 2 O, (C C 4 - alkoxy) 2 P(O)O, d-C 4 alkyl(d-C 4 alkoxy)P(O)O, or H(d-C 4 alkoxy)P(O)O; n 8 , n 9 , nio, nu, n 12 , n 13 and n 14 independently of one another are 0, 1 or 2; R 13 is hydrogen, d-C 4 alkyl, Cι-C 4 alkoxycarbonyl or phenyl which, in turn, can be substituted by Cι-C 4 alkyl, Cι-C 4 haloalkyl, C 1 -C 4 alkoxy, d-C 4 haloalkoxy, C C 4 alkylcarbonyl, d- C alkoxycarbonyl, C C 4 alkylamino, di-d-C 4 alkylamino, Cι-C 4 alkyl-S(O) n i 5 , C 1 -C alkyl- S(O) 2 O, C 1 -C 4 haloalkyl-S(0)mβ, Cι-C 4 haloalkyl-S(O) 2 O, d-C 4 alkyl-S(O) 2 NH, d-C 4 alkyl- S(O) 2 N(C 1 -C 4 alkyl), halogen, nitro or cyano; nι 5 and n 16 independently of one another are 0, 1 or 2; and the agrochemically tolerated salts M + and all stereoisomers and tautomers of the compounds of the formula I. In a preferred group of compounds of the formula I, R 10 is halogen, thiocyanato, d- Cι 2 alkylthio, d-C 12 alkylsulfinyl, d-C 2 alkylsulfonyl, d-Cι 2 haloalkylthio, d-C 12 - haloalkylsulfinyl, d-C^haloalkylsulfonyl, d-C^alkenylthio, C 2 -Cι 2 alkenylsulfinyl, C 2 -Cι 2 - alkenylsulfonyl, C 2 -C 2 haloalkenylthio, C -Ci 2 haloalkenylsulfinyl, C 2 -Cι 2 -haloalkenylsulfonyl, C 2 -Cι 2 alkynylthio, C 2 -Cι 2 alkynylsulfinyl, C 2 -d 2 alkynylsulfonyl, d-C 4 alkoxycarbonyl-d- C alkylthio, d-C 4 alkoxycarbonyl-d-C 2 alkylsulfinyl, d-C 4 alkoxycarbonyl-C 1 -C 2 alkylsulfonyl, Cι-C 8 alkyl-S(O) 2 NH, d-C 8 haloalkyl-S(O) 2 NH, d-C 8 alkyl-S(O) 2 θ, C C 18 alkylcarbonyloxy, C 2 -C 18 alkenylcarbonyloxy, C 3 -C 6 cycloalkylcarbonyloxy, d-C^alkoxycarbonyloxy, C Cι 2 - alkylthiocarbonyloxy, R 16 Rι 7 NC(O)O-, R 16 Rι 7 NC(S)O-, benzylthio, benzylsulfinyl, benzylsulfonyl, phenylthio, phenylsulfinyl, phenylsulfonyl, phenylsulfonyloxy or benzoyloxy, it being possible for the phenyl groups, in turn, to be substituted as indicated in claim 1 ; or is a group Ar-i-thio, Ari-sulfinyl, Arrsulfonyl in which An is a five- or six-membered monocyclic ring system which can be aromatic or partially saturated and can contain 1 to 2 hetero atoms selected from the group consisting of nitrogen, oxygen and sulfur and which, in turn, can be substituted as indicated in claim 1 ; or is thienylcarbonyloxy or furylcarbonyloxy, it being possible for these, in turn, to be substituted by methyl or halogen, or pyridylcarbonyloxy which, in turn, can be substituted as indicated in claim 1. In preferred compounds of the formula I, furthermore, R 10 is hydroxyl or O " M + . Other compounds of the formula I which must be emphasized are those in which W is oxygen, -CRnR 12 - or -C(O)-, where, in particular when W is -CRnRι 2 -, a) R 6 is hydrogen, methyl, ethyl, cyano, methoxycarbonyl, ethoxycarbonyl, methylthio, methylsulfinyl, methylsulfonyl or methoxy; and R 7 , R 8 , R 9 , Rn and R 12 independently of one another are hydrogen, Cι-C 4 alkyl, d-C 3 haloalkyl, C 2 -C 3 alkenyl or C 2 -C 3 alkynyl, or b) adjacent R 6 and R 7 and/or R 8 and R 9 together are -(CH 2 ) m -, -C(O)O(CH 2 ) 2 - or c) R 6 is hydrogen, methyl, ethyl, methoxycarbonyl, ethoxycarbonyl, methylthio, methylsulfinyl, methylsulfonyl or methoxy and R 12 together with R 9 is -(CH 2 ) 0 -- Furthermore, preferred groups of compounds of the formula I are those in which W is oxygen and R 6 , R 7 , R 8 and R 9 independently of one another are hydrogen or Cι-C 3 alkyl; or W is -C(O)- and R 6 , R 7 , R 8 and R 9 independently of one another are d-C 3 alkyl; or R 2 is hydrogen and R 3 is methyl; or R 2 is methyl, ethyl, n-propyl, i-propyl, vinyl, methoxymethyl, methoxycarbonyloxymethyl, ethoxycarbonyloxymethyl, acetoxymethyl, propionyloxymethyl, chloromethyl, bromomethyl, fluoromethyl, difluoromethyl, trifluoromethyl or cyanomethyl. Other compounds of the formula I which must be emphasized are those in which R 4 is hydrogen or methyl or R 5 is trifluoromethyl, difluorochloromethyl, pentafluoroethyl, heptafluoropropyl or difluoromethyl. In a further preferred group of compounds of the formula I, R 3 is hydrogen, R 2 is d-C 4 alkyl, CrC 3 haloalkyl, cyclopropyl, C 2 -C 3 alkenyl, C 2 -C 3 haloalkenyl, C 2 -C 3 alkynyl, allenyl, C C 2 - alkoxy-d-C 2 alkyl, Cι-C 2 alkylthio-Cι-C 2 alkyl, cyano-C -C 2 alkyl, C 1 -C 2 alkoxycarbonyl-Cι-C 2 - alkyl, C 1 -C alkylcarbonyloxy-C 1 -C 2 alkyl, d-C 3 alkoxy, CrC 3 haloalkoxy, allyloxy, propargyloxy, d-C 3 alkylthio, d-C 3 alkylsulfinyl or cyano. The compounds of the formula I in which Q is a group Q^ can be prepared using processes which are known per se, for example those described in EP-A-O 353 187 and EP-A- 0 316 491 , for example either by a) reacting a compound of the formula III in which R 2 , R 3 , R 4 and R 5 have the meaning given under formula I and X is a leaving group, for example halogen or cyano, with a compound of the formula II in which R 6 , R , R 8 , Rg and W have the meaning given under formula I in the presence of a base and in an inert organic solvent to give the compound of the formula IV and subsequently isomerizing the latter, for example in the presence of a base and a catalytic amount of dimethylaminopyridine (DMAP) or a cyanide source; or b) reacting a compound of the formula XVI in which R 2 , R 3 , R 4 and R 5 have the meaning given under formula I with compounds of the formula II in which R 6 , R , R 8 , R 9 and W have the meaning given under formula I in an inert organic solvent in the presence of a base and a coupling agent to give the compound of the formula IV and subsequently isomerizing the latter, for example as described under route a). The preparation of the compounds of the formula I is illustrated in greater detail in reaction scheme 1 below. Reaction scheme 1 Route a): Bas Route b): solvent, for example, CH 2 CI 2 , 0-110°C The compounds of the formula I with the group Qi in which R 10 is hydroxyl can preferably be prepared in accordance with this reaction scheme. The starting material for the preparation of the compounds of the formula I in which Q is the group Qi and R 10 is hydroxyl is, in accordance with reaction scheme 1 , route a), the carboxylic acid derivatives of the formula III in which X is a leaving group for example halogen, for example iodine, bromine and, in particular chlorine, N-oxyphthalimide or N,O-dimethylhydroxylamino or part of an activated ester, for example -N=C C--NNHH ■ -n (formed from dicyclohexylcarbodiimide (DCC) and O- the corresponding carboxylic acid) or 2 5 ι 2 3 3 2 (formed from N-ethyl-N'-(3- dimethylaminopropyl)carbodiimide (EDC) and the corresponding carboxylic acid). These are reacted with the dione derivatives of the formula II in an inert organic solvent, for example a halogenated hydrocarbon, for example dichloromethane, a nitrile, for example acetonitrile, or an aromatic hydrocarbon, for example toluene, and in the presence of a base, for example an alkylamine, preferably triethylamine, an aromatic amine, for example pyridine or 4-dimethylaminopyridine (DMAP) to give the isomeric enol ethers of the formula IV. This esterif ication is successfully carried out at temperatures from 0°C to 110°C. The isomerization of the ester derivatives of the formula IV to give the dione derivatives of the formula I (in which Rι 0 is OH) can be carried out, for example, in analogy to EP-A-0 353 187 or EP-A-O 316491 in the presence of a base, for example an alkylamine, for example triethylamine, a carbonate, for example potassium carbonate, and a catalytic amount of DMAP or a catalytic amount of a cyanide source, for example acetone cyanohydrin or potassium cyanide. Both reaction steps can be carried out in situ without isolation of the intermediates IV, in particular when using a cyanide compound of the formula III (X = cyano), or in the presence of a catalytic amount of acetone cyanohydrin or potassium cyanide. In accordance with reaction scheme 1 , route b), the desired diones of the formula I (in which R 10 is hydroxyl) can be obtained, for example, analogously to Chem. Lett. 1975, 1045 by esterifying the carboxylic acids of the formula XVI with the dione derivatives of the formula II in an inert solvent, for example a halogenated hydrocarbon, e.g. dichloromethane, a nitrile, e.g. acetonitrile or an aromatic hydrocarbon, e.g. toluene, in the presence of a base, for example an alkylamine, e.g. triethylamine, and a coupling agent, for example 2-chloro-1- methylpyridinium iodide. Depending on the solvent used, this esterification is successfully carried out at temperatures from 0°C to 110°C and first yields, as described under route a), the isomeric ester of the formula IV which can be isomerized as described under route a), for example in the presence of a base and a catalytic amount of DMAP, or a cyanide source, to give the desired dione derivatives of the formula I (R 10 = hydroxyl). The activated carboxylic acid derivatives of the formula III in reaction scheme I (route a) in which X is a leaving group, for example halogen, e.g. bromine, iodine or, in particular, chlorine, can be prepared by known standard methods, for example as described by C. Ferri "Reaktionen der organischen Synthese" ["Reactions in organic synthesis"], Georg Thieme Verlag, Stuttgart, 1978, page 460 et seq. This is shown in the reaction scheme 2 which follows. Reaction scheme 2 III XVI In accordance with reaction scheme 2, the compounds of the formula III in which X has the abovementioned meaning are prepared, for example, by using a halogenating agent, for example thionyl halides, e.g. thionyl chloride or thionyl bromide; phosphorus halides or phosphorus oxyhalides, e.g. phosphorus pentachloride or phosphorus oxychloride, or phosphorus pentabromide or phosphoryl bromide; or oxalyl halides, for example oxalyl chloride, or by employing a reagent for forming activated esters, for example N,N'- dicyclohexylcarbodiimide (DCC) or N-ethyl-N'-(3-dimethylaminopropyl)carbodiimide (EDC), of the formula XVII. Examples of meanings of X for the compound of the formula XVII as halogenating agent is a leaving group, for example halogen, e.g. fluorine, bromine or iodine and, in particular, chlorine, and Wi is, for example, PCI 2 , SOCI, SOBr or CICOCO. The reaction is preferably carried out in an inert organic solvent, for example in aliphatic, halogenated aliphatic, aromatic or halogenated aromatic hydrocarbons, e.g. n-hexane, benzene, toluene, xylenes, dichloromethane, 1 ,2-dichloroethane or chlorobenzene, at reaction temperatures in the range of -20°C to the reflux temperature of the reaction mixture, preferably at 40-150°C, and in the presence of a catalytic amount of N,N-dimethylformamide. Such reactions are generally known, and various variations with regard to the leaving group X are described in the literature. Compounds of the formula I in which R 10 is other than hydroxyl or halogen can be prepared by conversion methods which are generally known from the literature, for example by acylation or carbamoylation methods using appropriate acid chlorides in the presence of a suitable base, starting from compounds in which R 10 is hydroxyl, or can be prepared by nucleophilic substitution reactions on chlorides of the formula I in which Rι 0 is halogen, which can also be obtained by known methods by reaction with a chlorinating agent such as phosgene, thionyl chloride or oxalyl chloride. In this case, examples of compounds which are employed are suitably substituted amines, or, directly, hydroxylamines, or alkylsulfonamides, mercaptans, thiophenols, phenols, Ar 5 -NH 2 or Ar^SH, in the presence of a base, for example 5-ethyl-2-methylpyridine, diisopropylethylamine, triethylamine, sodium bicarbonate, sodium acetate or potassium carbonate. Compounds of the formula I in which R 10 contains thio groups can be oxidized in analogy to known standard methods, for example using peracids, e.g. meta-chloroperbenzoic acid (m-CPBA) or peracetic acid, to give the corresponding sulfones and sulfoxides of the formula I. The degree of oxidation on the sulfur atom (SO- or SO 2 -) can be controlled by the amount of oxidant. Also, the resulting derivatives of the formula I in which Rι 0 is other than hydroxyl can exist in various isomeric forms which, if appropriate, can be isolated in pure form. The invention therefore also extends to all of these stereoisomeric forms. Examples of these isomeric forms are the formulae I * , I ** and I *** below in which Q is the group Qi (see also note and scheme on page 10 above). All other compounds from within the scope of the formula I can be readily prepared taking into consideration the chemical properties of the pyridyl or Q moiety. The end products of the formula I can be isolated in the customary manner by concentration or by evaporating the solvent and purified by recrystallization or trituration of the solid residue in solvents in which they are not readily soluble, such as ethers, aromatic hydrocarbons or chlorinated hydrocarbons, by distillation or by means of column chromatography and a suitable eluent. Furthermore, the skilled worker knows in which sequence certain reactions are expediently carried out to avoid any side reactions. Unless a directed synthesis for isolating pure isomers is carried out, the product may be obtained as a mixture of two or more isomers. The isomers can be resolved by methods known per se. Compounds of the formula I in which n is 1 , i.e. the corresponding N-oxides of the formula I, can be synthesized by reacting a compound of the formula I in which n is 0 with a suitable oxidant, for example with the H 2 O 2 -urea adduct in the presence of an acid anhydride, e.g. trifluoroacetic anhydride. Compounds of the formula I in which R in the ortho-position relative to the pyridine nitrogen is 1 -chioro-d-C 2 alkyl, 1 -hydroxy-C C 2 alkyl, 1-(d-C 6 alkylcarbonyloxy)-d-C 2 alkyl, 1 -benzoyloxy-C C 2 alkyl, 1 -(C 1 -C alkoxycarbonyloxy)-Cι-C 2 alkyl, 1 -(Cι-C 4 alkylthio)-Cι-C 2 - alkyl, 1 -(Ci 1 -C 4 alkylsulfinyl)-d-C 2 alkyl, 1 -(C 1 -C 4 alkylsuifonyl)-d-C 2 alkyl, 1 -thiocyanato-C C 2 alkyl, 1 -cyano-d-C 2 alkyl, can also be prepared by, for example, heating an N-oxide of the formula I under known reaction conditions, for example in the presence of tosyl chloride (see, for example, Parham, W. E.; Sloan, K. B.; Reddy, K. R.; Olson, P. E.; J Org Chem 1973, 38, 927) or in the presence of an acid anhydride (see, for example, Konno, K.; Hashimoto, K.; Shirahama, H.; Matsumoto, T.; Heterocycles 1986, 24, 2169) and, if appropriate, subsequently further reacting the product. These reaction sequences may be demonstrated with reference to the following example: (z.B CIC0 2 Et, Ac 2 0 oder TsCI) E = OC(0)R, OH, Cl E = OC(0)R, Cl Compounds of the formula I in which R in the ortho-position relative to the pyridine nitrogen, in particular 1-bromo-Cι-C 2 alkyI, 1 -chloro-d-C 2 alkyl, 1-fluoro-Cι-C 2 alkyl, 1 ,1 -dibromomethyl, 1 ,1-dichloromethyl, formyl, 1-(d-C 4 alkylthio)-d-C 2 alkyl, 1-(C 1 -C 4 alkylsulfinyl)-Cι-C 2 alkyl, 1 -(Cι-C 4 alkylsulfonyl)-d-C 2 aIkyl, 1-thiocyanato-d-C 2 alkyl or 1-cyano-Cι-C 2 alkyl, can also be prepared, for example, by oxidizing a compound of the formula I in which R 10 is, in particular, chlorine, Cι-C 4 alkoxycarbonyloxy or benzoylcarbonyloxy under known halogenation conditions, for example with N-bromosuccinimide or N-chlorosuccinimide in the presence of light and a free-radical initiator, for example benzoyl peroxide, to give the 1 -bromo or 1 -chloro, 1 ,1 -dibromo or 1 ,1-dichloro compound, and subsequently refunctionalizing the latter to give the corresponding derivatives. Again, these reaction sequences may be demonstrated with reference to the example below. Aqueous work-up Conversion reactions X=CI, Br; X Q -, = H, X Compounds of the formula I can also be synthesized by reacting a compound of the formula I in which p is 0 and R 2 is d-C 6 alkyl with a suitable base, for example lithium diisopropylamide or n-butyllithium, at temperatures between -100 and -20°C (preferably -70 and -50°C) in an inert solvent (for example tetrahydrofuran) to give the corresponding dianion. The skilled worker knows how such carbanions can be converted by means of electrophilic substitution, for example with a chloroformic ester. This reaction sequence may be demonstrated with reference to the following example: Electrophile (e.g. CIC0 2 CH 3 ) Other compounds from within the scope of the formula I can be prepared with suitable electrophiles taking into consideration the chemical properties of the pyridyl or Q moiety. The compounds of the formula Ilia in which R 501 is d-Cehaloalkyl; R 30 ι is hydrogen; R 0 ι is hydrogen or d-C 6 aIkyl; and R 201 is d-C 6 alkyl, d-C 6 haloalkyl-Cι-C 4 alkyl, C 2 -C 6 alkenyl, C 2 -C 6 haIoalkenyl, or d-C 2 - alkoxycarbonyl- or phenyl-substituted vinyl, C 2 -C 6 alkynyl or C 2 -C 6 haloalkynyl; or trimethylsilyl-, hydroxyl-, Cι-C 2 alkoxy-, d-C 2 alkoxycarbonyl- or phenyl-substituted ethynyl or C 3 -C 6 allenyl; or C 3 -C 6 cycloalkyl, halogen-substituted C 3 -C 6 cycloalkyl, Cι-C 4 alkoxy-Cι-C 4 - alkyl, Cι-C 4 alkyl-S(O) n4 -C 1 -C 4 alkyl, cyano-d-C 4 alkyl, d-C 4 alkoxycarbonyl-d-C 4 alkyl, C C 4 - thiocyanato, oxiranyl, C C 4 alkylamino-Cι-C 4 alkyl, d-C 4 dialkylamino-Cι-C alkyl, hydroxy- Cι-C alkyl, Cι-Cι 2 alkylthiocarbonyl-d-C 4 alkyl or formyl-Cι-C 4 alkyl, or R 20 ι is a five- to ten- membered monocyclic or fused bicyclic ring system which can be aromatic or partially saturated and can contain 1 to 4 hetero atoms selected from the group consisting of nitrogen, oxygen and sulfur, the ring system being bonded to the pyridine ring via a Cι-C - alkylene, -CH=CH-, -C≡C-, -CH 2 O- , -CH 2 N(C 1 -C 4 alkyl)- ) -CH 2 S-, -CH 2 SO- or -CH 2 SO 2 - group and it not being possible for each ring system to contain more than 2 oxygen atoms and more than two sulfur atoms, and it being possible for the ring system itself to be mono-, di- or trisubstituted by d-C 6 alkyl, d-C 6 haloalkyl, C 3 -C 6 alkenyl, C 3 -C 6 haloalkenyl, C 3 - C 6 alkynyl, C 3 -C 6 haloalkynyl, d-C 6 alkoxy, Ci-Cehaloalkoxy, C 3 -C 6 alkenyloxy, C 3 - C 6 alkynyloxy, mercapto, d-C 6 alkylthio, d-Cehaloalkylthio, C 3 -C 6 alkenylthio, C 3 - C 6 haloalkenylthio, C 3 -C 6 -alkynylthio, C 2 -C 5 alkoxyalkylthio, C 3 -C 5 acetylalkylthio, C 3 - C 6 alkoxycarbonylalkylthio, C 2 -C 4 -cyanoalkylthio, d-C 6 alkylsulfinyl, d-C 6 haloalkylsulfinyl, d- C 6 alkylsulfonyl, d-C 6 -haloalkylsulfonyl, aminosulfonyl, d-C 2 alkylaminosulfonyl, di-(d- C 2 alkyl)aminosulfonyl, di-(d-C 4 alkyl)amino, halogen, cyano, nitro, phenyl and benzylthio, it being possible for phenyl and benzylthio, in turn, to be substituted on the phenyl ring by d- C 3 alkyl, Cι-C 3 haloalkyl, d-C 3 alkoxy, d-C 3 -haloalkoxy, halogen, cyano or nitro, and where the substituents on the nitrogen in the heterocyclic ring are other than halogen; and X is halogen or cyano, are novel and were developed specifically for the preparation of the compounds of the formula I and are therefore a further subject of the present invention. The compounds of the formula XVIa in which R 201 , R 30 ι, R 40 ι and R 50 ι have the abovementioned meaning, with the proviso that, if R50 1 is trifluoromethyl and, simultaneously, R 30 ι and R 401 are hydrogen, then R 20 ι is other than d.Cealkyl, are novel and therefore a further subject of the present invention. The compounds of the formula Q T (or formula II) are known and can be prepared by methods similar to those described, for example in J. Org. Chem. (1977), 42, 1163-9, Brit. UK Pat. Appl.GB 2205316, DE 3902818, GB 8706557, DE 4434987, WO 9213821 and Aust. J. Chem. (1976), 29(11 ), 2525-31 , Chem. Commun. (1998), (16), 1691-1692. The compounds of the formula XVI (or XVIa and XVIb) are synthesized by methods similar to known methods, for example as in Heterocycles, 46, 129 (1997) or Helvetica Chimica Acta 71 , 596 (1988), and is characterized in that either a) a compound of the formula V 01 (V) in which R 30 ι is hydrogen; R 0 ι is hydrogen, d-C 6 alkyl or phenyl, it being possible for phenyl, in turn, to be substituted by d-C 3 alkyl, Cι-C 3 haloalkyl, d-C 3 alkoxy, d-C 3 haloalkoxy, halogen, cyano or nitro; or R 40 i is a five- to ten-membered monocyclic or fused bicyclic ring system which can contain 1 to 4 hetero atoms selected from the group consisting of nitrogen, oxygen and sulfur and it not being possible for the ring system to contain more than 2 oxygen atoms and more than two sulfur atoms, and it being possible for the ring system itself to be mono-, di- or trisubstituted by d-C-ealkyl, d-C 6 haloalkyl, C 2 -C 6 alkenyl, C 2 -C 6 haloalkenyl, C 2 -C 6 alkynyl, drCehaloalkynyl, d-C 6 alkoxy, d-C 6 haloalkoxy, C 3 -C 6 alkenyloxy, C 3 -C 6 alkynyloxy, d- C 6 alkylthio, d-C 6 haloalkylthio, C 3 -C 6 alkenylthio, C 3 -C 6 haloalkenylthio, C 3 -C 6 alkynylthio, Cι-C 4 alkoxy-Cι-C 2 alkylthio, Cι-C 4 alkylcarbonyl-d-C 2 aIkylthio, d-C alkoxycarbonyl-d-C 2 - alkylthio, cyano-C C 4 alkylthio, Cι-C 6 alkylsulfinyl, Cι-C 6 haloalkylsulfinyl, Cι-C 6 alkylsulfonyl, Cι-C 6 haloalkylsulfonyl, aminosulfonyl, C C 2 alkylaminosulfonyl, di-(C 1 -C 2 alkyl)aminosulfonyl, halogen, cyano, nitro, phenyl and benzylthio, it being possible for phenyl and benzylthio, in turn, to be substituted on the phenyl ring by C C 3 alkyl, d-C 3 haloalkyI, d-C 3 alkoxy, d- C 3 haloalkoxy, halogen, cyano or nitro, and where substituents on the nitrogen in the heterocyclic ring are other than halogen; and Rι is C C 4 alkyl; is acylated with a compound of the formula VI in which R 50 ι is d-C 6 haloalkyl to give the compound of the formula VII in which R 30 ι, R 4 oι, R 501 and R 1 have the abovementioned meaning in the presence of a base, for example an aromatic amine, e.g. pyridine, and the alkoxy group is subsequently exchanged for the amino group with ammonia in an organic solvent, for example a halogenated hydrocarbon, e.g. dichloromethane, a nitrile, e.g. acetonitrile. The resulting compound of the formula VIII is subsequently subjected to a condensation reaction with a compound of the formula IX in which R 20 ι is CrCealkyl, Cι-C 6 haloalkyl-d-C 4 alkyl, C 2 -C 6 alkenyl, C 2 -C 6 haloalkenyl, C 2 -C 6 - alkynyl, C 2 -C 6 haloalkynyl, C 3 -C 6 cycloalkyl, Cι-C 4 alkoxy-d-C 4 alkyl, Cι-C 4 alkyl-S(O) n -d-d- alkyl, cyano-Cι-C alkyl, CrC 4 alkoxycarbonyl-C C 4 alkyl, d-C alkoxycarbonyloxy-Cι-C 4 alkyl, C 1 -C 4 thiocyanato-C 1 -C 4 alkyl, oxiranyl, C 1 -C 4 alkylamino-Cι-C alkyl, di-(d-C 4 alkyl)amino- C C 4 alkyl or formyl-d-C 4 alkyl; or R 20 ι is a group Ar 6 -d-C 4 alkyl in which Ar 6 is a five- to ten-membered monocyclic or fused bicyclic ring system which can be aromatic or partially saturated and can contain 1 to 4 hetero atoms selected from the group consisting of nitrogen, oxygen and sulfur, it not being possible for each ring system to contain more than 2 oxygen atoms and more than two sulfur atoms and it being possible for the ring system itself to be mono-, di- or trisubstituted by d- C 6 alkyl, d-C 6 haloalkyl, C 3 -C 6 alkenyl, C 3 -C 6 haloalkenyl, C 3 -C 6 alkynyl, C 3 -C 6 haloalkynyl, d- C 6 alkoxy, CrC 6 haloalkoxy, C 3 -C 6 alkenyloxy, C 3 -C 6 alkynyloxy, mercapto, d-C 6 alkylthio, C C 6 haloalkylthio, C 3 -C 6 alkenylthio, C 3 -C 6 haloalkenylthio, C 3 -C 6 -alkynylthio, C 2 - C 5 alkoxyalkylthio, C 3 -C 5 acetylalkylthio, C 3 -C 6 alkoxycarbonylalkylthio, C 2 -C 4 -cyanoalkylthio, Cι-C 6 alkylsulfinyl, d-C 6 haloalkylsulfinyl, d-C 6 alkylsulfonyl, Cι-C 6 -haloalkylsulfonyl, aminosulfonyl, d-C 2 alkylaminosulfonyl, di-(C 1 -C 2 alkyl)aminosulfonyl, di-(Cι-C 4 alkyl)amino, halogen, cyano, nitro, phenyl and benzylthio, it being possible for phenyl and benzylthio, in turn, to be substituted on the phenyl ring by d-C alkyl, Cι-C 3 haloalkyl, d-C- 3 alkoxy, C C 3 haloalkoxy, halogen, cyano or nitro, and where substituents on the nitrogen in the heterocyclic ring are other than halogen, and R 14 has the abovementioned meaning, and subsequently hydrolysing the resulting compound of the formula Xa is subsequently hydrolysed to give the compound of the formula XVIa in which R 20 ι, R 30 ι, R 4 oι and R 50 ι have the abovementioned meaning; or b) a compound of the formula XI in which R 14 has the abovementioned meaning is subjected to a condensation reaction with a compound of the formula XII R OR 14 ( XII) O and the resulting compound of the formula XIII in which R 3 , R 4 and R 5 have the abovementioned meaning and R 1 is Cι-C 4 alkyl, is chlorinated to give the compound of the formula XIV in which R 3 , R 4, R 5 and R have the abovementioned meaning (for example using POCI 3 ), and this compound is subsequently reacted with a nucleophile of the formula XV in which Z is SH, OH or amino and R 15 is d-C 6 alkyl, C 3 -C 6 alkenyl, C 3 -C 6 haloalkenyl, C 3 -C 6 - alkynyl, C 3 -C 6 haloalkynyl, d-C 6 alkylsulfonyl, C C 6 haloalkyl, phenyl or benzyl, it being possible for the phenyl group, in turn, to be substituted by Cι-C 3 alkyl, Cι-C 3 haloalkyl, d-C 3 - alkoxy, CrC 3 haloalkoxy, halogen, cyano or nitro, or is Cι-C 4 alkoxy-Cι-C 4 alkyl, d-C 4 - alkylthio-Cι-C 4 alkyl, Cι-C 4 alkylsulfinyl-Cι-C 4 alkyl, Cι-C 4 alkylsulfonyl-d-C alkyl, Cι-C 4 - alkylsulfonyl or di-(C C 4 alkyl)aminosulfonyl, or R 15 is a five- to ten-membered monocyclic or fused bicyclic ring system which can be aromatic or partially saturated and can contain 1 to 4 hetero atoms selected from the group consisting of nitrogen, oxygen and sulfur, it not being possible for each ring system to contain more than 2 oxygen atoms and more than two sulfur atoms and it being possible for the ring system itself to be mono-, di- or trisubstituted by d- C 6 alkyl, d-Cehaloalkyl, C 3 -C 6 alkenyl, C 3 -C 6 haloalkenyl, C 3 -C 6 alkynyl, C 3 -C 6 haloalkynyl, d- C 6 alkoxy, d-C 6 -haloalkoxy, C 3 -C 6 alkenyloxy, C 3 -C 6 alkynyloxy, mercapto, Cι-C 6 alkylthio, d- C-e-haloalkylthio, C 3 -C 6 alkenylthio, C 3 -C 6 haloalkenylthio, C 3 -C 6 alkynylthio, C 2 - C 5 alkoxyalkylthio, C 3 -C 5 acetylalkylthio, C 3 -C 6 alkoxycarbonylalkylthio, C 2 -C 4 cyanoalkylthio, Cι-C 6 alkylsulfinyl, d-C 6 haloalkylsulfinyl, Cι-C 6 alkylsulfonyl, d-C 6 haloalkylsulfonyl, aminosulfonyl, Cι-C 2 alkylaminosulfonyl, di-(Cι-C 2 alkyl)aminosulfonyl, (CH 2 ) n R 7 , NR 8 R 9 , halogen, cyano, nitro, phenyl and benzylthio, it being possible for phenyl and benzylthio, in turn, to be substituted on the phenyl ring by d-C 3 alkyl, Cι-C 3 haloalkyl, d-C 3 alkoxy, Ci- C 3 haloalkoxy, halogen, cyano or nitro, and substituents on the nitrogen in the heterocyclic ring being other than halogen, in the presence of a base to give compounds of the formula Xb in which R 14 , R 15 , R 3 , R 4 , R 5 and Z have the abovementioned meanings and the resulting compound is subsequently hydrolysed to give the compound of the formula XVIb in which R 15 , R 3 , R 4 , R 5 and Z have the abovementioned meaning. Compounds in which Z-R 15 and Z are oxygen and R 15 is d-C 6 alkyl, C 3 -C 6 alkenyl, C 3 -C 6 - alkynyl, Ci-Cehaloalkyl, C 3 -C 6 haloalkenyl, cyano-C C 4 alkyl, C C alkoxy-Cι-C 4 alkyl, Cι-C 4 - alkylthio-Cι-C 4 alkyl or d-C alkoxycarbonyl-d-C 4 alkyl can also be reacted starting from XIII by direct alkylation with the corresponding alkylating agent L-R 15 XVa in which L is a leaving group such as chlorine, bromine, iodine, mesyloxy or tosyloxy. Compounds of the formula XVIb in which Z-R 15 is fluorine are prepared by reacting a compound of the formula XIV with potassium fluoride and, if appropriate, a catalytic amount of 18-crown-6 in the presence of a polar aprotic solvent, for example acetonitrile, dimethylformamide or sulfolane. Compounds of the formula XVIc in which Z-R 15 is hydrogen are prepared by reducing the chlorine group in formula XIV, for example with hydrogen in the presence of a suitable metal catalyst or with ammonium formate, in a suitable solvent. The preparation of the compounds of the formula XVI or XVIa, XVIb and XVIc are illustrated in greater detail in reaction schemes 3 and 4 which follow. Reaction scheme 3 Reaction scheme 4 Reduction e.g. eOH/NH 4 HC0 2 MeOH XVIb Xb Compounds of the formula XVId in which R 2 is bromomethyl, cyanomethyl, thiocyanatomethyl, C 2 -C 6 alkenyl, C 2 -C 6 haloalkenyl, a d-C 2 aIkoxycarbonyl- or phenyl- substituted vinyl, C 2 -C 6 alkynyl, C 2 -C 6 haloalkynyl, a trimethylsilyl-, hydroxyl-, d-C 2 alkoxy-, Cι-C 2 alkoxycarbonyl- or phenyl-substituted ethynyl, C 3 -C 6 allenyl, C 3 -C 6 cycloalkyl or mono- or polyhalogenated C 3 -C 6 cycloalkyl can be prepared, for example, in accordance with generally known conversion methods which are shown in reaction scheme 4a. Reaction scheme 4a Intermediates of the formula XVIa in which R 50 ι is CF 2 CI are prepared as described in scheme 3 or by reacting a compound of the formula Xa in which R 501 is trichloromethyl with hydrofluoric acid in a pressurized vessel at temperatures between 0 and 220°C (preferably 60-200°C). Compounds of the formula XVIa in which R 50 ι is CHF 2 can be prepared as in scheme 3 or by heating a compound of the formula Xa in which R 30 ι, R 4 oι, Rι 4 and R 20 ι have the abovementioned meaning and R 50 ι is CF 2 CI in an inert solvent, for example toluene or benzene, at temperatures between 25 and 120°C (preferably 80-120°C) with tributyltin hydride or 1 ,1 ,1 ,3,3,3-hexamethyl-2-(trimethylsilyl)trisilane in the presence of a catalytic amount of azo-isobutyronitrile and subsequently hydrolysing the resulting compound to give the compound of the formula XVIa in which R 50 is CHF 2 . Compounds of the formula XVIa in which R 20 ι, R 30 ι, R 0 ι and R 50 ι have the abovementioned meaning can also be prepared by reacting a compound of the formula Xc in which R 14 , R 30 ι, R_ t oι and R 50 ι have the abovementioned meaning and R 20 ι is CH 2 CI by nucleophilic substitution, for example with an alkali metal iodide in an inert solvent, to give the corresponding iodides, or by means of gaseous hydrobromic acid in lower carboxylic acids such as glacial acetic acid to give the corresponding bromine derivatives (for example in accordance with US-3974166) or by means of alkali metal fluoride in a dipolar solvent such as sulfolane to give the corresponding fluorine derivatives, or, to prepare an alkoxy radical Xd, by reacting a halogen derivative Xc with an alcohol or phenol in the presence of a base such as sodium hydride or an alkaline earth metal oxide or alkaline earth metal carbonate or directly with an alkali metal alkoxide in an inert solvent such as dimethylformamide or in an excess of the alcohol ROH which corresponds to the group to be introduced at temperatures between -5 and 160°C, or, in order to prepare a corresponding aromatic or aliphatic thioether Xe, by reacting, analogously to what has been said above, either the halide Xc with an aliphatic or aromatic thiol in the presence of a base such as sodium hydride or with an alkali metal salt of a thiol in an inert solvent at -10 - 150°C, or, in order to prepare corresponding sulfinyl or sulfonyl derivatives Xe, by carrying out the reaction with an oxidant such as m-chloroperbenzoic acid or sodium periodate or sodium perborate, with the temperature control known in the art, depending on the degree of oxidation (for example -30°C - +50°C for n=1) or -20°C - +100°C for n=2) in an inert solvent such as dichloromethane to give Xf, or, in order to prepare cyanomethylene derivatives of the formula Xg, by reacting a halide of the formula Xc with an alkali metal cyanide or tetraalkylammonium cyanide or copper cyanide in an inert solvent such as dichloromethane, tetrahydrofuran or dimethylformamide at temperatures between 0°C and 220°C. The preparation of the compounds of the formula XVIa (R 50 ι = CF 2 CI) and of the intermediates of the formulae Xc, Xd, Xe, Xf, and Xg are illustrated in greater detail in the reaction schemes 5, 6 and 7 which follow. Reaction scheme 5 Xa (R ∞1 = CCI 3 ) Xa (R^ = CCIF 2 ) Reaction scheme 6 Xa (R 501 = CF 2 CI) or (n-Bu) 3 Sn-H χa ^ __ ^^ XVIa (R 501 = CHF, Reaction scheme 7 xg Xd To prepare all other compounds of the formula X and XVI which are functionalized in accordance with the definition of R 20 ι (Z-R 15 ) to R 50 ι, a multiplicity of known standard methods are suitable, for example alkylation, halogenation, acylation, amidation, oximation, oxidation and reduction, the choice of the preparation methods which are suitable depending on the properties (reactivities) of the substituents in the intermediates. The reactions to give compounds of the formula I are advantageously carried out in aprotic inert organic solvents. Such solvents are hydrocarbons such as benzene, toluene, xylene or cyclohexane, chlorinated hydrocarbons such as dichloromethane, trichloromethane, tetrachloromethane or chlorobenzene, ethers such as diethyl ether, ethylene glycol dimethyl ether, diethylene glycol dimethyl ether, tetrahydrofuran or dioxane, nitriles such as acetonitrile or propionitrile, amides such as N,N-dimethylformamide, diethylformamide or N-methylpyrrolidinone. The reaction temperatures are advantageously between -20°C and +120°C. In general, the reactions are slightly exothermic and, as a rule, they can be carried out at room temperature. To shorten the reaction time, or else to start the reaction, the mixture may be heated briefly to the boiling point of the reaction mixture. The reaction times can also be shortened by adding a few drops of base as reaction catalyst. Suitable bases are, in particular, tertiary amines such as trimethylamine, triethylamine, quinuclidine, 1 ,4-diazabicyclo[2.2.2]octane, 1 ,5-diazabicyclo[4.3.0]non-5-ene or 1 ,5-diazabicyclo- [5.4.0]undec-7-ene. However, inorganic bases such as hydrides, e.g. sodium hydride or calcium hydride, hydroxides, e.g. sodium hydroxide or potassium hydroxide, carbonates such as sodium carbonate and potassium carbonate, or hydrogen carbonates such as potassium hydrogen carbonate and sodium hydrogen carbonate, may also be used as bases. The compounds of the formula I can be isolated in the customary manner by concentrating and/or by evaporating the solvent and purified by recrystallization or trituration of the solid residue in solvents in which they are not readily soluble, such as ethers, aromatic hydrocarbons or chlorinated hydrocarbons. All application methods which are conventionally used in agriculture, for example pre- emergence application, post-emergence application and seed treatment, as well as various methods and techniques, for example the controlled release of active ingredients, are suitable for the use according to the invention of the compounds of the formula I or of compositions comprising them. To this end, the active ingredient in solution is applied to mineral carriers for granules or to polymerized granules (urea/formaldehyde) and dried. If appropriate, an additional coating can be applied (coated granules), which allows the active ingredient to be released in a controlled manner over a specific period of time. The compounds of the formula I can be employed as herbicides as such, i.e. as obtained from synthesis. However, they are preferably processed in the customary manner together with the auxiliaries conventionally used in the art of formulation, for example to give emulsifiable concentrates, directly sprayable or dilutable solutions, dilute emulsions, wettable powders, soluble powders, dusts, granules or microcapsules. Such formulations are described, for example, in WO 97/34485 on pages 9 to 13. The application methods such as spraying, atomizing, dusting, wetting, scattering or pouring, as well as the type of composition, are chosen to suit the intended aims and the prevailing circumstances. The formulations, i.e. the compositions, preparations or products which comprise the active ingredient of the formula I or at least one active ingredient of the formula I and, as a rule, one or more solid or liquid formulation auxiliaries are prepared in the known manner, for example by intimately mixing and/or grinding the active ingredients together with the formulation auxiliaries, for example solvents or solid carriers. Furthermore, surface-active compounds (surfactants) may additionally be used when preparing the formulations. Examples of solvents and solid carriers are indicated for example in WO 97/34485 on page 6. Suitable surface-active compounds are, depending on the nature of the active ingredient of the formula I to be formulated, non-ionic, cationic and/or anionic surfactants and surfactant mixtures which have good emulsifying, dispersing and wetting properties. Examples of suitable anionic, non-ionic and cationic surfactants are enumerated, for example, in WO 97/34485 on pages 7 and 8. The surfactants conventionally used in the art of formulation which are described, inter alia, in "McCutcheon's Detergents and Emulsifiers Annual" MC Publishing Corp., Ridgewood New Jersey, 1981 , Stache, H., "Tensid-Taschenbuch" ["Surfactants Guide"], Carl Hanser Verlag, Munich/Vienna, 1981 , and M. and J. Ash, "Encyclopedia of Surfactants", Vol l-lll, Chemical Publishing Co., New York, 1980-81 , are furthermore also suitable for preparing the herbicidal compositions according to the invention. As a rule, the herbicidal formulations comprise 0.1 to 99% by weight, in particular 0.1 to 95% by weight, of herbicide, 1 to 99.9% by weight, in particular 5 to 99.8% by weight, of a solid or liquid formulation auxiliary and 0 to 25% by weight, in particular 0.1 to 25% by weight, of a surfactant. While concentrated compositions are more preferred as commercially available goods, the end consumer uses, as a rule, dilute compositions. The compositions can also comprise further additives such as stabilizers, for example epoxidized or non-epoxidized vegetable oils (epoxidized coconut oil, rapeseed oil or soya oil), antifoams, e.g. silicone oil, preservatives, viscosity regulators, binders, tackifiers and fertilizers or other active ingredients. As a rule, the active ingredients of the formula I are applied to the plant or its environment at rates of 0.001 to 4 kg/ha, in particular 0.005 to 2 kg/ha. The dosage required for the desired action can be determined by experiments. It depends on the type of the action, the developmental stage of the crop plant and of the weed, and on the application (location, timing, method) and can, owing to these parameters, vary within wide limits. The compounds of the formula I are distinguished by herbicidal and growth-inhibitory properties which allow them to be employed in crops of useful plants, in particular in cereals, cotton, soya, sugar beet, sugar cane, plantation crops, rapeseed, maize and rice and for the non-selective control of weeds. Crops are also to be understood as including those which have been rendered tolerant to herbicides or classes of herbicides by means of conventional plant breeding or by genetic engineering methods. The weeds to be controlled may be both mono- and dicotyledonous weeds such as Stellaria, Nasturtium, Agrostis, Digitaria, Avena, Setaria, Sinapis, Lolium, Solanum, Echinochloa, Scirpus, Monochoria, Sagittaria, Bromus, Alopecurus, Sorghum halepense, Rottboellia, Cyperus, Abutilon, Sida, Xanthium, Amaranthus, Chenopodium, Ipomoea, Chrysanthemum, Galium, Viola and Veronica. The examples which follow illustrate the invention in greater detail without limiting it. Preparation Examples: Example H1 : Preparation of 3-hvdroxy-4,4-dimethyl-2-(2-methyl-6-trifluoromethylpyridine- 3-carbonyl)cvclohex-2-enone (compound A2-B24): 6.68 g (0.0305 mol) of methyl 2-methyl-6-trifluoromethylnicotinate (prepared as described in Heterocycles, 46, 129 (1997)) are dissolved in 250 ml of methanol/water (3:1 mixture), and 1.92 g (0.046 mol) of lithium hydroxide hydrate are added portionwise at a temperature of 22°C. After 4 hours at 22°C, the reaction mixture is poured onto ethyl acetate and 2 N hydrochloric acid, and the organic phase is washed three times with water, dried with sodium sulfate and evaporated, and the residue is triturated with a small amount of hexane. After filtration, 5.69 g (90% of theory) of 2-methyl-6-trifluoromethylnicotinic acid of melting point 147-149°C are obtained. The resulting 2-methyl-6-trifluoromethylnicotinic acid (1.026 g, 0.005 mol) is dissolved in 20 ml of oxalyl chloride. Three drops of dimethylformamide are added and the mixture is refluxed for 1 hour. The mixture is then concentrated on a rotary evaporator and the residue (2-methyl-6-trifluoromethylnicotinoyl chloride) is taken up in 100 ml of methylene chloride. At a temperature of 0°C, 1.6 ml (0.0115 mol) of triethylamine and 0.7 g (0.005 mol) of 4,4- dimethylcyclohexane-1 ,3-dione are added. After 2 hours at a temperature of 22°C, the solvent is removed on a vacuum rotary evaporator, the residue which remains is dissolved in 55 ml of acetonitrile, and 0.15 ml (0.0016 mol) of acetone cyanohydrin and 0.79 ml (0.0057 mol) of triethylamine are added in order to subject the intermediate to a rearrangement reaction. After the reaction solution has been stirred for 4 hours at room temperature, it is evaporated. The syrup which remains is chromatographed on silica gel. Elution with a mixture of toluene, ethyl alcohol, dioxane, triethylamine and water (100:40:20:20:5 parts by volume) gives a pale yellow viscous oil (Rf = 0.39 on the abovementioned mixture as mobile phase), which is dissolved in dichloromethane and washed in succession with 75 ml of 5% hydrochloric acid and 75 ml of water. Evaporation to dryness of the organic solution which has been dried with Na 2 SO 4 yields 1.05 g (63%) of pure 3-hydroxy-4,4-dimethyl-2-(2-methyl-6-trifluoromethylpyridine-3-carbonyl)cyclohex-2- enone in the form of white crystals of melting point 75-77°C. 1 H NMR (de-DMSO, δ in ppm): 1.342, s, 6H: 2.088, t, J 9Hz, 2H: 2.685, s, 3H: 2.982, t, J 9Hz, 2H:8.030, d, J 8.1 Hz, IH: 8.094, d, (J, 8.1 Hz), 1H. Example H2: Preparation of 5-methyl-5-trifluoromethylcvclohexane-1 ,3-dione (compound H-B1066 0.64 g of sodium were introduced into 40 ml of ethanol, and 3.23 ml of methyl acetoacetate and 4.9 g of isopropyl 4,4,4-trifluoro-3-methylbut-2-enoate were introduced, and the mixture was heated at the boil for 18 hours. After the mixture has been partitioned between dilute hydrochloric acid and ethyl acetate, the mixture is evaporated. The remaining unpurified methyl 2-methyl-4,6-dioxo-2-trifluoromethylcyclohexanecarboxylate is hydrolysed in a mixture of methanol and water at boiling point in the presence of 9.1 g of sodium hydroxide. The mixture is subsequently acidified with hydrochloric acid and extracted with fresh ethyl acetate. After recrystallization (ethyl acetate), pure 5-methyl-5-trifluoromethylcyclohexane- 1 ,3-dione of melting point 150-152°C is obtained. Example H3: Preparation of methyl 2-hvdroxy-1 -methoxy-5-methyl-4-oxocvclohex-2- enecarboxylate (Example H-B1069): A 30% solution of 35.8 g of sodium methoxide is introduced into 65 ml of dimethyl sulfoxide and, within 20 minutes, treated with a mixture of 16.7 g of 3-methyl-3-butene-2-one and 32.4 g of dimethyl methoxymalonate at a temperature of 30-35°C. The mixture is stirred for 1 hour at a temperature of 35°C, and is then acidified with hydrochloric acid and extracted repeatedly with dichloromethane. The organic phases are washed with water, dried and concentrated. Crystallization from hot ethyl acetate and hexane gives pure methyl 2-hydroxy- 1-methoxy-5-methyl-4-oxocyclohex-2-enecarboxylate of melting point 117-117.5°C. Example H4: Preparation of methyl 2-hvdroxy-1 -methoxy-5-methyl-3-(2-methyl-6- trifluoromethylpyridine-3-carbonv0-4-oxocvclohex-2-enecarboxylate (compound A2-B1069): 2.23 g of fresh 2-methyl-6-trifluoromethylnicotinoyl chloride are added to a mixture of 2.14 g of methyl 2-hydroxy-1-methoxy-5-methyl-4-oxocyclohex-2-enecarboxylate and 2.02 g of triethylamine in 30 ml of acetonitrile. After approximately 30 minutes, 0.065 g of potassium cyanide is added and the mixture is stirred for 18 hours. At pH 2, the mixture is subsequently partitioned between water and ethyl acetate, dried over magnesium sulfate and evaporated. Filtration on silica gel (mobile phase ethyl acetate/methanol/triethylamine 85:10:5) gives the pure methyl 2-hydroxy-1 -methoxy-5-methyl-3-(2-methyl-6-trifluoromethylpyridine-3-carbonyl)- 4-oxocyclohex-2-enecarboxylate as a viscous oil. Example H5: Preparation of 3-hvdroxy-4-methoxy-6-methyl-2-(2-methyl-6-trifluoromethyl- pyridine-3-carbonyl)cvclohex-2-enone (compound A2-B1070): 1.4 g of methyl 2-hydroxy-1-methoxy-5-methyl-3-(2-methyl-6-trifluoromethylpyridine-3- carbonyl)-4-oxocyclohex-2-enecarboxylate in dioxane/water (5:3) are treated with 0.586 g of potassium hydroxide and the mixture is stirred for 3 hours. The mixture is then acidified (pH 3) and extracted with fresh ethyl acetate. The crude product is purified by chromatography analogously to Example H4. 3-Hydroxy-4-methoxy-6-methyl-2-(2-methyl-6- trifluoromethyl-pyridine-3-carbonyl)cyclohex-2-enone is obtained as a viscous oil (according to 1 H-NMR as a mixture of 3 tautomeric forms). Example H6: 5-Chloro-2.2.6.6-tetramethyl-4-(2-methyl-6-trifluoromethylpyridine-3-carbonyl)- cvclohex-4-ene-1 ,3-dione (compound A2-B1 105) and 6-rchloro-(2-methyl-6-trifluoromethyl- pyridin-3-yl)methylene1-2,2,4,4-tetramethylcvclohexane-1 ,3,5-trione : 7.0 g (55 mmol) of oxalyl chloride are introduced into 18.5 g (50 mmol) of 5-hydroxy-2,2,6,6- tetramethyl-4-(2-methyl-6-trifluoromethylpyridine-3-carbonyl)cyclohex-4-ene-1 ,3-dione (compound A2-B354), dissolved in 50 ml of dichloromethane; 5 drops of dimethylformamide are added, and the mixture is slowly heated up to boiling point. After approximately 30 minutes, after the evolution of gas has ceased, the mixture is evaporated and the product is crystallized by adding n-hexane. The main product obtained is pure 5-chloro-2,2,6,6- tetramethyl-4-(2-methyl-6-trifluoromethylpyridine-3-carbonyl)cyclohex-4-ene-1 ,3-dione, m.p. 119.5-120°C. Further HPLC-separation of the mother liquor using 5-10% ethyl acetate in hexane gives the isomer 6-[chloro-(2-methyl-6-trifluoromethylpyridine-3-yl)methylene]- 2,2,4,4-tetramethylcyclohexane-1 ,3,5-trione, m.p. 92.5-93°C. Example H7: 5-Chloro-2,2,6,6-tetramethyl-4-(2-methyl-1 -oxy-6-trifluoromethylpyridine-3- carbonyl)cvclohex-4-ene-1 ,3-dione (compound A1210-B1105): 1.94 g (5 mmol) of 5-chloro-2,2,6,6-tetramethyl-4-(2-methyl-6-trifluoromethylpyridine-3- carbonyl)cyclohex-4-ene-1 ,3-dione are treated in 20 ml of dichloroethane at a temperature of -10°C with 0.94 g (10 mmol) of hydrogen peroxide/urea adduct and 1.89 g (9 mmol) of trifluoroacetic anhydride. The reaction mixture is warmed to room temperature, with stirring, and held for a further 4 hours at this temperature. The mixture is then partitioned between ethyl acetate and water of pH 5, washed with sodium chloride solution and evaporated. The residue which is filtered through silica gel is pure 5-chloro-2,2,6,6-tetramethyl-4-(2-methyl-1- oxy-6-trifluoromethylpyridine-3-carbonyl)cyclohex-4-ene-1 ,3-dione of melting point 145.5- 146°C. Example H8: 4-(2-Bromomethyl-6-trifluoromethylpyridine-3-carbonyl)-5-chloro-2.2,6,6- tetramethylcvclohex-4-ene-1 ,3-dione (compound A1029-B1105): 0.39 g (1 mmol) of 5-chIoro-2,2,6,6-tetramethyl-4-(2-methyl-6-trifluoromethylpyridine-3- carbonyl)cyclohex-4-ene-1 ,3-dione and 0.20 g (1.1 mmol) of N-bromsuccinimide are refluxed in the presence of a catalytic amount of dibenzoyl peroxide in 10 ml of carbon tetrachloride. After the reaction has subsided, the resulting succinimide is removed by filtration and the crude product is purified by column chromatography (mobile phase: ethyl acetate/hexane 1 :4). This gives pure 4-(2-bromomethyl-6-trifluoromethylpyridine-3-carbonyl)-5-chloro- 2,2,6,6-tetramethylcyclohex-4-ene-1 ,3-dione of melting point 94.5-95°C. Example H9: 2-(2-Acetoxymethyl-6-trifluoromethylpyridine-3-carbonyl)-4,4,6,6-tetramethyl- 3.5-dioxocvclohex-1 -enyl acetate (compound A1099-B1107): 0.4 g (1 mmol) of 5-chloro-2,2,6,6-tetramethyl-4-(2-methyl-1-oxy-6-trifluoromethylpyridine-3- carbonyl)cyclohex-4-ene-1 ,3-dione (Example H7) is refluxed for 25 minutes in the presence of 3 ml of acetic anhydride. The mixture is then concentrated and partitioned between ethyl acetate and sodium bicarbonate solution at pH 6.5. The crude product, separated on silica gel (mobile phase: ethyl acetate/hexane 1 :4) yields the pure 2-(2-acetoxymethyl-6- trifluoromethylpyridine-3-carbonyl)-4,4,6,6-tetramethyl-3,5-dioxocyclohex-1 -enyl acetate as an oil; 1 H-NMR (CDCI 3 ): 7.98 d, CH, 7.72 d, CH, 5.62 s, CH 2 , 2.22 and 2.20 2x OAc, 1.58, s, 2x CH 3 , 1.44 ppm, s, 2x CH 3 . Example H10: 5-Hvdroxy-2-methyl-4-(2-methyl-6-trifluoromethylpyridine-3-carbonyl)- bicvclor4.1.01hept-4-en-3-one (compound A2-D109) and 3-hvdroxy-7-methyl-2-(2-methyl-6- trifluoromethylpyridine-3-carbonyl)cvclohepta-2,6-dienone (compound A2-F5): 0.82 g (2 mmol) of ethyl trans-5-hydroxy-2-methyl-4-(2-methyl-6-trifluoromethylpyridine-3- carbonyl)-3-oxobicyclo[4.1.0]hept-4-en-2-carboxylate (compound A2-D111 )is stirred in a 2:1 mixture of dioxane/water together with 0.254 g (4.5 mmol) of potassium hydroxide at room temperature until all of the starting material is reacted. Then, ethyl acetate is added, the mixture is acidified to pH 3 using 4 N HCI, and the 2-phase mixture is then heated for approx. 1 hour at a temperature of 40°C. The aqueous phase which is saturated with sodium chloride is then separated off. The ethyl acetate extract is evaporated to dryness and the product is chromatographed on silica gel (mobile phase ethyl acetate/hexane 1 :2). The 1st fraction which is isolated is 3-hydroxy-7-methyl-2-(2-methyl-6-trifluoromethylpyridine-3- carbonyl)cyclohepta-2,6-dienone as pure tautomer mixture, 1 H-NMR (CDCI 3 ): 17.72 and 17.08, 2s, OH, 7.6-7.45, 2 arom. H, 6.68 and 6.62, 2t, CH, 2.84, m, 2.63, m, 2.52, m, 4H, 2.62 and 2.54, 2s, CH 3 , 2.03 and 1.77 ppm, 2s, CH 3 . Subsequent elution with 100% ethyl acetate gives, as the 2nd fraction, the isomer and tautomer mixture of 5-hydroxy-2-methyl-4- (2-methyl-6-trif luoromethylpyridine-3-carbonyl)bicyclo[4.1.0]hept-4-en-3-one, 1 H-NMR (CDCI 3 ): i.a. 17.62 and 17.48, 2s, OH, 7.6-7.45, 2 arom. H, 2.54, m, 2.48, 2s CH 3, 1.22 and 1.14, 2d, CH 3 , 1.00 to 0.05 ppm, 2H. Example H11 : 5-Hvdroxy-2-methanesulfinyl-2-methyl-4-(2-methyl-6-trifluoromethylpyridine-3- carbonyl)bicvclor4.1.01hept-4-en-3-one (compound A2-D114): 0.87 g (2.3 mmol) of 5-hydroxy-2-methyl-2-methyIsulfanyl-4-(2-methyl-6- trifluoromethylpyridine-3-carbonyl)bicyclo[4.1.0]hept-4-en-3-one (compound A2-D113), dissolved in 8 ml of methanol, is warmed for 3 hours at a temperature of 50°C in the presence of 0.56 g of sodium periodate. The mixture is then partitioned between ethyl acetate and sodium chloride solution, concentrated, and the crude product is purified by chromatography (mobile phase: ethyl acetate/methanol 19:1). Pure 5-hydroxy-2- methanesulfinyl-2-methyl-4-(2-methyl-6-trifluoromethylpyridine-3-carbonyl)bicyclo[4.1.0]hept- 4-en-3-one is obtained as tautomer and isomer mixture of melting point 159.5-160°C. Example H12: 2-Prop-2-vnyloxy-6-trifluoromethylnicotinic acid (compound A1025): 47 g (0.2 mol) of 2-oxo-6-trifluoromethyl-1 ,2-dihydropyridine-3-carboxylic acid, 20 ml (0.25 mol) of propargyl bromide and 43 g (0.31 mol) of potassium carbonate are heated to a temperature of 75°C in a mixture of 40 ml of dimethylformamide and 80 ml of acetonitrile in the presence of a catalytic amount of 18-crown-6 ether. After 5 hours, the mixture is partitioned between ethyl acetate and saturated sodium chloride solution. The crude product is filtered through a silica gel column using 15% ethyl acetate in hexane. The main component, which is obtained in the form of an oil, is the pure ethyl 2-prop-2-ynyloxy-6- trifluoromethylnicotinate; 1 H-NMR (CDCI 3 ): 8.31 , d, CH, 7.38, d, CH, 5.13, d, CH 2 , 4.41 , q, CH 2 , 2.48, t, CCH, 1.41 ppm, t, CH 3 . 36.3 g (0.13 mol) of this product is stirred over a period of 16 hours with a solution of 11.5 g (0.17 mol) of potassium hydroxide in 50 ml of water and 50 ml of dioxane. After acidification and extraction with ethyl acetate, crystalline 2-prop-2-ynyloxy-6-trifluoromethylnicotinic acid is obtained; 1 H-NMR (CDCI 3 ): 10.0, b, OH, 8.53, d, CH, 7.44, d, CH, 5.22, d, CH 2 , 2.54 ppm, t, CCH. Example H13: 2-Methylthio-6-trifluoromethylnicotinic acid (compound A15): 9.4 g (40 mmol) of 2-oxo-6-trifluoromethyl-1 ,2-dihydropyridine-3-carboxylic acid are introduced into a 1 -molar solution of 21.7 g of phosphorus tribromide (80 mmol) in dichloromethane at a temperature of 35°C. Then, the solvent is distilled off and the reaction mixture is heated slowly to boiling point, approx. 175°C. After 18 hours, the mixture is cooled to 0°C, diluted with dichloromethane and stirred with ice-water of pH 1.8. The organic phase is then washed with cold sodium carbonate solution and with 15% sodium chloride solution, dried over magnesium sulfate and concentrated. The residue is ethyl 2-bromo-6- trifluoromethylnicotinate in the form of an oil; 1 H-NMR (CDCI 3 ): 8.20, d, CH, 7.72 d, CH, 4.46, q, CH 2 , 1.42 ppm, t, CH 3 of melting point 164-166°C. 1.0 g (3.4 mmol) of this product, dissolved in a small amount of acetonitrile, is heated for 45 minutes to a temperature of 70°C together with 0.26 g of sodium methanethiolate (3.4 mmol) in the presence of a catalytic amount of 15-crown-5 ether. The solution, which is cooled to room temperature, is then treated with 0.22 g (5.5 mmol) of sodium hydroxide and 5 ml of water, and stirring is continued for 3 hours. The neutral components are subsequently removed with a small amount of diethyl ether, and the aqueous phase is brought to pH 2.5 and extracted twice using ethyl acetate. This gives 2-methylthio-6- trifluoromethylnicotinic acid as crystalline product; 1 H-NMR (CDCI 3 ): 8.46, d, CH, 7.43, d, CH, 2.58 ppm, s, SCH 3 . Example H14: 2-Methanesulfonylamino-6-trifluoromethylnicotinic acid (compound A1203): 0.52 g of methanesulfonamide is introduced into a tetrahydrofuran suspension of 0.24 g of 55% sodium hydride in oil. After the evolution of hydrogen has ceased, 1.5 g (5 mmol) of ethyl 2-bromo-6-trifluoromethylnicotinate, 0.3 g (5.2 mmol) of potassium fluoride and a catalytic amount of crown ether and 5 ml of N-methylpyrrolidone are added and the mixture is heated at the boil for 18 hours. The reaction mixture is then partitioned between ethyl acetate and water and freed from organic neutral constituents. The aqueous phase is brought to pH 2.9, extracted 3 times with fresh ethyl acetate, dried and concentrated. A crystalline product, ethyl 2-methanesulfonylamino-6-trifluoromethyInicotinate, is obtained from ether/hexane; 1 H-NMR (CDCI 3 ): 10.48, s, NH, 8.49, d, CH, 7.38, d, CH, 4.45, q, CH 2 , 3.51 , s, SO 2 CH 3 , 1.42 ppm, t, CH 3 . 0.43 g (1.4 mmol) of the above product is hydrolysed at room temperature using a 1 :1 solution of 0.22 g (3.9 mmol) of potassium hydroxide in dioxane/water. After the solution, which has been acidified to pH 2.5, has been extracted with ethyl acetate, 2-methanesulfonylamino-6-trifluoromethylnicotinic acid is obtained as crystallisate; 1 H-NMR (d 6 -DMSO): 8.62, d, CH, 7.72, d, CH, 3.52 ppm, s, SO 2 CH 3 . Example H15: (3-Methoxycarbonyl-6-trifluoromethylpyridin-2-ylmethyl)triphenylphosphonium bromide: 50 g (0.23 mol) of methyl 2-methyl-6-trifluoromethylnicotinate and 49 g (0.28 mol) of N-bromosuccinimide are heated for 90 minutes at 50°C in 500 ml of carbon tetrachloride in the presence of a catalytic amount of α.α-azaisobutyronitrile with illumination by a 150 watt lamp. Precipitated succinimide is filtered off, and the product methyl 2-bromomethyl-6- trifluoromethylnicotinate is then isolated as main component by means of column chromatography (mobile phase ethyl acetate/hexane 1 :15), 1 H-NMR (CDCI 3 ): 4.01 , s, 3H; 5.03, s, 2H; 7.72, d (J 8.2Hz), 1 H; 8.43 ppm, d, (J 8.2Hz), 1 H. 25.6 g (35 mmol) of the above product are taken up in toluene and treated with 10.6 g (40 mmol) of triphenylphosphine. After the mixture has been heated for 2 hours at boiling point, pure (3-methoxycarbonyl-6- trifluoromethylpyridine-2-ylmethyl)triphenylphosphonium bromide of melting point 215-217°C crystallizes out upon cooling. Example H16: 2-Vinyl-6-trifluoromethylnicotinic acid (compound A21 ) and 2-(2,2-dichloro- cvclopropyl)-6-trifluoromethylnicotinic acid (compound A1092): 5.7 g (10 mmol) of (3-methoxycarbonyl-6-trifluoromethylpyridine-2-ylmethyl)triphenyl- phosphonium bromide are dissolved at room temperature in a 2-phase system of 25 ml of chloroform and 2.1 g (20 mmol) of sodium carbonate and reacted, in 10 ml of water, with a 35% aqueous solution of 1.7 g (20 mmol) of formaldehyde. After 1.5 hours, the organic phase is separated off and filtered through silica gel. Methyl 2-vinyl-6- trifluoromethylnicotinate is obtained as an oil, 1 H-NMR (CDCI 3 ): 8.31 , d, CH, 7.10, dd, CH, 7.09, d, CH, 6.68, dd, CH, 5.68, dd, CH, 3.97 ppm, s, OCH 3 . 0.97 g (4.1 mmol) of this product is again taken up in chloroform and reacted with 6 ml of 50% sodium hydroxide solution with vigorous stirring in the presence of 90 mg of benzyltrimethylammonium bromide. After 20 hours, the organic phase is separated off, concentrated and purified by HPLC (mobile phase: ethyl acetate/hexane 1 :4). This gives pure methyl 2-(2,2-dichlorocyclopropyl)-6-trifluoromethylnicotinate, 1 H-NMR (CDCI 3 ): 8.50, d, CH, 7.70, d, CH, 4.08, s, OCH 3 , 3.68, dd, CH, 2.64, dd, CH, 2.05 ppm, dd, CH. Hydrolysis of the above esters gives, accordingly, the 2-vinyl-6-trifluoromethylnicotinic acid, 1 H-NMR (CDCIg): 8.40, d, CH, 7.22, dd, CH, 7.09, d, CH, 6.68, dd, CH, 5.58 ppm, dd, CH, and 2-(2,2-dichlorocyclopropyl)-6-trifluoromethylnicotinic acid, 1 H-NMR (CDCI 3 ): 8.64, d, CH, 7.23, d, CH, 3.78, dd, CH, 2,67, dd, CH, 2,08 ppm, dd, CH. Example H17: 2-Propa-1 ,2-dienyl-6-trifluoromethylnicotinic acid (A1096) and 2-(3-chloro- propenvD-6-trifluoromethylnicotinic acid (compound A1095). 6.7 g (11 mmol) of ((3-methoxycarbonyl-6-trifluoromethylpyridin-2-yl)methyl)triphenyl- phosphonium bromide are reacted with 2 ml of 45% aqueous chloroacetaldehyde solution (14 mmol) and 1.5 g (14 mmol) of sodium carbonate with vigorous stirring in a 2-phase system of 20 ml of chloroform and 7 ml of water. After 2 hours, the organic solution is separated off and washed with half-saturated sodium chloride solution. The product is separated on silica gel (mobile phase ethyl acetate/hexane 1 :4). As the 1 st fraction, methyl 2-propa-1 ,2-dienyl-6-trifluoromethylnicotinate, 1 H-NMR (CDCI 3 ): 7.62, m, CH, 7.55, d, CH, 7.32, d, CH, 7.04, d, CH, 7.02, m, CH, 3.98 ppm, s, OCH 3) is isolated, and methyl 2-(3- chloropropenyl)-6-trifluoromethylnicotinate, 1 H-NMR (CDCI 3 ): 8.85, d, CH, 7.65, dd, 7.58, d, CH, CH, 7.28, dd, CH, 4.32, d, CH 2 CI, 3.98 ppm, s, OCH 3 is isolated as the 2nd fraction. Hydrolysis of the above esters gives 2-propa-1 ,2-dienyl-6-trifluoromethylnicotinic acid, m.p. 194-196°C, and 2-(3-chloropropenyl)-6-trifluoromethylnicotinic acid, m.p. 137-138°C. Example H18: 2-Chloro-4-methyl-6-trifluoromethylnicotinic acid (compound A1205): In a pressurized vessel, 7.5 g (0.03 mol) of ((3-ethoxycarbonyl)-4-methyl-6-trifluoromethyl)- pyrid-2-one is heated for 3 hours at a temperature of 170°C in the presence of 5.8 ml of phenyl dichlorophosphate. When cold, the reaction solution is filtered directly over a short silica gel column (mobile phase: ethyl acetate/hexane 1 :9), and the 2-chloro-4-methyl-6- trifluoromethylpyridin-3-ylethyl ester is obtained as oily product. The latter is hydrolysed in the presence of aqueous potassium hydroxide solution in dioxane at a temperature of 40°C. After acidification to pH 2.7, extraction with ethyl acetate gives 2-chloro-4-methyl-6- trifluoromethylnicotinic acid as crystalline product: 1 H NMR (CDCI 3 ): 9.55, b, OH, 7.55, s, 1 H; 3.80, s, CH 3 , 2.56 ppm, s, CH 3 . Example H19: 4-Methyl-6-trifluoromethylnicotinic acid (compound A531 ): To a suspension of 0.55 g of 10% Pd/C in 20 ml of methanol there are added 3.0 g (16.8 mmol) of the 2-chloro-4-methyl-6-trifluoromethyIpyridin-3-ylethyl ester and, in 2 portions, a total of 5 g of ammonium formate, and the mixture is stirred for 24 hours at room temperature. The reaction mixture is then filtered through Celite and partitioned between ethyl acetate and sodium chloride solution. Chromatographic purification (mobile phase 1 :9) gives the 4-methyI-6-trifluoromethylpyridin-3-ylethyl ester in the form of an oil: hydrolysis in accordance with the above processes gives 4-methyl-6-trifluoromethylnicotinic acid: 1 H NMR (CDCI 3 ): 9.32, s, 1 H, 7.62, s, 1 H, 2.79 ppm, s, CH 3 . Example H20: 5-Methyl-5-methylsulfanylbicvclo 4.1.0lheptane-2,4-dione (compound H-D113): A 1 -molar solution of 16.7 g (0.1 mol) of lithium bistrimethylsilylamide in tetrahydrofuran is added at a temperature of 0°C to a solution of 13.4 g (0.1 mol) of methyl 2-methylmercaptopropionate in 30 ml of tetrahydrofuran. After the mixture has been stirred for 1 hour, 11.8 g (0.1 mol) of 5-chloropent-3-en-2-one are added dropwise in the course of 20 minutes in such a way that the temperature can be maintained at 0°C. After the mixture has been stirred for a further 30 minutes, ice-water is added, and the mixture is acidified with hydrochloric acid and extracted with diethyl acetate. The crude product is chromatographed with ethyl acetate/hexane 15/85. This gives methyl 2-(2-acetylcyclopropyl)-2- methylsulfanylpropionate, 1 H-NMR (CDCI 3 ): 3.74, s, OCH 3 , 2.19 and 2.14, 2s, SCH 3 , 2.12. and 2.00, 2s, CH 3 , 2.2-1.9, 1 H, 1.3, s, CH 3 , 1.3 to 1.0 ppm, 2H, as a 3:7 isomer mixture. 2.45 g (11 mmol) of the above product, which is enriched in the more polar isomer, is heated with 4.5 g (25 mmol) of 30% sodium ethoxide solution in a mixture of toluene/dimethylformamide 19:1 for 90 minutes at 115°C. The mixture is then taken up in ethyl acetate and washed with dilute hydrochloric acid at pH 3. The residue which has been isolated is purified on silica gel (mobile phase ethyl acetate/hexane 1 :2). This gives the isomer I of 5-methyl-5-methylsulfanylbicyclo[4.1.0]heptane-2,4-dione, 1 H-NMR (CDCI 3 ): 3.48, d, CH, 3.00 d, CH, 2.21 , m, CH, 1.94, m, CH, 1.86, s, CH 3> 1.57, s, CH 3 , 1.44, m, CH, 1.04 ppm, m, CH. The isomer II of 5-methyl-5-methylsulfanylbicyclo[4.1.0]heptane-2,4-dione, 1 H-NMR (CDCI 3 ): 3.78, d, CH, 3.14 d, CH, 2.22, m, CH, 1.93, m, CH, 2.08, s, CH 3 , 1.58, s, CH 3 , 1.6-1.4 ppm, 2H, is obtained from the product which is enriched in apolar isomers. Example H21 : 4-Methylcvclohept-4-ene-1 ,3-dione (compound H-F5): 1.0 g (5.4 mmol) of the 5-methyl-5-methylsulfanylbicyclo[4.1.0]heptane-2,4-dione isomers II is hydrogenated for 90 minutes under atmospheric pressure in 15 ml of methanol in the presence of 5 g Raney nickel. The mixture is concentrated and purified over silica gel (mobile phase ethyl acetate/hexane 1 :1), and 4-methylcyclohept-4-ene-1 ,3-dione, 1 H-NMR (CDCI 3 ): 6.84, m, CH, 3.94, s, CH 2 , 2.77, m, CH 2 , 2,59, m, CH 2 , 1.88 ppm, s, CH 3 , is obtained as an oil. Example H22: 2-OxaspiroF4.5ldecane-1 ,6,8-trione (compound H-E16): A suspension of sodium hydride (55% in oil, 27.5 mmol) in 70 ml of anhydrous tetrahydrofuran is cooled to a temperature of -20°C, and a solution of 2-acylbutyrolactone (2.69 ml, 25 mmol) in 5 ml of tetrahydrofuran is subsequently added dropwise. After the reaction mixture has been stirred for 1 hour at this temperature, it is treated dropwise with a solution of methyl acrylate (4.5 ml, 50 mmol) in tetrahydrofuran at a temperature of -20°C. The reaction mixture is subsequently allowed to warm to room temperature and is stirred for 8 hours. The mixture is then poured into ice-water and acidified with 2 N hydrochloric acid to pH 1. After extraction with ethyl acetate, drying over sodium sulfate and concentration in vacuo, the product is purified by flash chromatography (eluent: ethyl acetate/acetic acid 1 :1). This gives 2-oxaspiro[4.5]decane-1 ,6,8-trione in the form of a white powder of melting point 145-148°C Example H23: Spiror2.51octane-4,6-dione (compound H-C1): 3.4 g of sodium hydride (55% suspension in oil, 78.0 mmol) were introduced into 1 I of tert- butanol and the mixture was stirred for a few minutes at room temperature. Then, 2-acylbutyrolactone (100 g, 0.78 mol) is added and the reaction mixture is treated with methyl acrylate (67.2 g, 0.78 mmol) over a period of 3.5 hours at a temperature of approx. 30°C. The reaction mixture is taken up in diethyl ether and washed in succession with 75 ml of saturated NaH 2 PO 4 solution, water and saturated sodium chloride solution, dried over sodium sulfate and concentrated. This gives 162 g of methyl 3-(3-acetyl-2- oxotetrahydrofuran-3-yl)propionate as colourless oil, which can be reacted further without purification. 2.0 g (9.3 mmol) of the above product and 2.1 g of sodium iodide (14.0 mmol) are dissolved in 10 ml of 1 ,3-dimethyl-2-imidazolidinone and the solution is heated for 3 hours at 210°C. After cooling, the reaction mixture is poured into dilute aqueous saturated NaH 2 PO 4 solution and extracted with diethyl ether, dried over sodium sulfate and concentrated. This gives methyl 3-(1-acetylcyclopropyl)propionate as a colourless oil. 74.5 g of methyl 3-(1-acetylcyclopropyl)propionate (0.32 mol) are dissolved in 1 I of tetrahydrofuran and the solution is treated portionwise with 14.3 g of sodium hydride (55% suspension in oil, 0.32 mol) at room temperature. After 1 hour, the reaction mixture is diluted with 200 ml of dimethylformamide and warmed to 70°C. After 8 hours, tetrahydrofuran is removed in vacuo, and the residue is poured into 2 N hydrochloric acid and extracted with diethyl ether. The organic phase is dried over sodium sulfate and concentrated, and column chromatography over silica gel (methylene chloride:ethanol 9:1 as eluent) gives spiro[2.5]octane-4,6-dione in the form of white crystals of melting point 116-118°C. Example H24: 2-(4.6-Dimethoxypyrimidin-2-ylsulfanylmethyl)-6-trifluoromethylnicotinic acid (compound A1088): 2.0 g (7.89 mmol) of methyl 2-chloromethyl-6-trifluoromethylnicotinate (prepared analogously to Heterocycles, 46, 129 (1997) by heating methyl 4-chloro-3-oxobutyrate and 4-amino- 1 ,1 ,1-trifluorobut-3-en-2-one in toluene in the presence of trifluoroacetic acid) are introduced into 30 ml of acetonitrile and 1.63 g (11.83 mmol) of K 2 CO 3 and reacted with 1.49 g (8.67 mmol) of 4,6-dimethoxypyrimidin-2-thiol at room temperature. After 4 hours, the mixture is poured into ethyl acetate/water, the ethyl acetate phase is removed, and the aqueous phase is reextracted with ethyl acetate. The combined ethyl acetate phases are dried over sodium sulfate, concentrated and purified by recrystallization from ethyl acetate/hexane. This gives methyl 2-(4,6-dimethoxypyrimidin-2-ylsulfanylmethyl)-6- trifluoromethylnicotinate in the form of white crystals of melting point 123-124°C. Hydrolysis of the above esters (analogously to Example H1 ) gives, accordingly, 2-(4,6- dimethoxypyrimidin-2-ylsulfanylmethyl)-6-trifluoromethylnicotinic acid in the form of white crystals of melting point 157-158 °C. 1 H-NMR (CDCI 3 ): 3.96, s, 6H; 3.99,s, 3H; 5.03, s, 2H; 5.72, s, 1 H; 7.66,d (J, 8.1 Hz),1 H; 8.40 ppm, d (J, 8.1 Hz),1 H. Example H25: 2-Cvanomethyl-6-trifluoromethylnicotinic acid (compound A1103): 2.0 g (7.89 mmol) of methyl 2-chloromethyl-6-trifluoromethylnicotinate and 565 mg (8.67 mmol) of potassium cyanide are reacted in 20 ml of acetonitrile/water mixture (1 :1) in the presence of 270 mg of tetrabutylammonium hydrogen sulfate. After the reaction has ended, the mixture is poured into water and extracted with ethyl acetate. After the ethyl acetate phase has been dried over sodium sulfate and concentrated, the crude product is purified by means of HPLC (ethyl acetate: hexane as eluent). This gives 610 mg (32% of theory) of methyl 2-cyanomethyl-6-trifluoromethylnicotinate in the form of an oil. 1 H-NMR (CDCIg): 3.96, s, 3H; 4.38, s, 2H; 7.72,d (J, 8.1Hz),1 H; 8.48 ppm, d (J, 8.1 Hz),1H. Hydrolysis analogous to the methods already mentioned above yields 2-cyanomethyl-6- trifluoromethylnicotinic acid in the form of yellow crystals of melting point 152-153 °C. 1 H- NMR (CDCI 3 ): 4.18, s, 2H; 7.72,d (J, 8.1 Hz),1 H; 8.52 ppm, d (J, 8.1 Hz),1 H. Example H26: 3-(6-Dif luoromethyl-2-methylpyridine-3-carbonyl)-2-hvdroxy-1 -methyl-4- oxocvclohex-2-enecarboxylate (compound A124-B34): 200 mg (0.516 mmol) of methyl 3-[6-(chlorodif luoromethyl)-2-methylpyridine-3-carbonyl]-2- hydroxy-1-methyl-4-oxocyclohex-2-enecarboxylate (compound A94-B34) is heated for 3 hours at a temperature of 120°C in 8 ml of toluene in the presence of 0.18 ml (0.62 mmol) tris(trimethylsilyl)silane. The viscous residue which remains is chromatographed on silica gel. The pale yellow viscous oil which is obtained by eluting with a mixture of toluene, ethyl alcohol, dioxane, triethylamine and water (100:40:20:20:5 by volume) is dissolved in dichloromethane and washed in succession with aqueous hydrochloric acid and water. Evaporation of the organic solution which has been dried with Na 2 SO 4 yields 140 mg (73%) of pure methyl 3-(6-dif luoromethyl-2-methylpyridine-3-carbonyl)-2-hydroxy-1 -methyl-4- oxocyclohex-2-enecarboxylate in the form of a pale yellow oil. 1 H-NMR (CDCI 3 ): 1.28, s, 3H; 1.79-1.97, m, 1 H; 2.39-2.46, m,1 H; 2.43, s, 3H; 2.69, dt (J, 19.2 and 4.8Hz),1 H; 2.82-2.92, m,1 H; 3.67, s, 3H; 6.55, t , (J, 55.5 Hz),1 H; 7.43, d (J, 7.8Hz), 1 H; 7.49, d (J, 7.8Hz), 1 H; 17.20 ppm, br s, 1 H. Example H27:3-Hvdroxy-2-(2-methyl-1 -oxy-6-trifluoromethylpyridine-3-carbonyl)cvclohex-2- enone (compound A1210-B1): 16.1 g (0.054 mol) of 3-hydroxy-2-(2-methyl-6-trifluoromethylpyridine-3-carbonyl)cyclohex-2- enone (Example A2-B1 ) and 10.2 g (0.11 mol) of urea/hydrogen peroxide complex are dissolved in 150 ml of methylene chloride, and 22.1 ml (0.162 mol) of trifluoroacetic anhydride are subsequently added dropwise at a temperature of 25°C. After the reaction mixture has been stirred for 14 hours at a temperature of 25°C, it is poured into ethyl acetate and water, and the organic phase is washed twice with water, dried with sodium sulfate and concentrated. The residue is chromatographed on silica gel (eluent: ethyl acetate/methanol 9/1). This gives 2.4 g (14%) of the desired product in the form of white crystals (m.p. 117- 119°C). 1 H-NMR (d 6 -DMSO): 1.98, m, 2H; 2.30, s, 3H; 2.60, t (J, 7.25Hz), 4H: 7.32, d (J, 9.8Hz), 1 H; 7.92 ppm, d (J, 9.8Hz), 1 H. Example H28: 2-(2-Methyl-6-trifluoromethylpyridine-3-carbonyl)-3-phenylsulfanylcvclohex-2- enone (compound A2-B1102): 4.0 g (0.0134 mol) of 3-hydroxy-2-(2-methyl-6-trifluoromethylpyridine-3-carbonyl)cyclohex-2- enone (compound A2-B1) are suspended in 25 ml of oxalyl chloride, and 0.1 ml of dimethylformamide is subsequently added dropwise. After the vigorous evolution of gas has ceased, the mixture is held for 1.5 hours at a bath temperature of 45°C and subsequently concentrated, and the residue (3-chloro-2-(2-methyl-6-trifluoromethylpyridine-3-carbonyl)- cyclohex-2-enone) is dissolved in 60 ml of methylene chloride. Triethylamine (3.7 ml, 0.0268 mol), dimethylaminopyridine (160 mg, 1.34 mmol) and 1.5 ml (0.0147 mol) of thiophenol are added at a temperature of 0-5°C. After 20 hours at a temperature of 22°C, the reaction mixture is concentrated and purified on silica gel (hexane/ethyl acetate 5:1 ). Trituration in hexane gives pure 2-(2-methyl-6-trifluoromethylpyridine-3-carbonyl)-3- phenylsulfanylcyclohex-2-enone in the form of white crystals of melting point 124-125 °C. 1 H-NMR (CDCI 3 ): 1.99, m, 2H; 2.41 , m 4H; 2.80, s, 3H; 2.60: 7.40-7.60, m, 6H; 7.80 ppm, d (J, 8.2Hz), 1H. Example H29: 3-Benzenesulfonyl-2-(2-methyl-6-trifluoromethylpyridine-3-carbonyl)cvclohex- 2-enone (compound A2-B1104): 0.8 g (0.00204 mol) of the 2-(2-methyl-6-trifluoromethylpyridine-3-carbonyl)-3- phenylsulfanylcycIohex-2-enone obtained above is dissolved in 30 ml of methylene chloride, and 1.39 ml of peracetic acid (39% in acetic acid, 0.00816 mol) are subsequently added dropwise at a temperature of 25°C. After 4 hours at 25°C, the reaction mixture is poured into ethyl acetate and water, the organic phase is washed with water, dried with sodium sulfate and concentrated, and the residue is triturated with a small amount of hexane and ethyl acetate. Filtration gives 0.72 g (84% of theory) of 3-benzenesulfonyl-2-(2-methyl-6- trifluoromethyl-pyridine-3-carbonyl)cyclohex-2-enone in the form of white crystals of melting point 165-167°C. 1 H-NMR (CDCI 3 ): 2.30, m, 2H; 2.55, t (J, 7Hz), 2H; 2.71 , m, 2H; 3.05, s, 3H; : 7.40-7.80, m, 4H; 7.80-8.05 ppm, m, 3H. Example H30: 6-Difluoromethyl-2-methylnicotinic acid (compound A124): 6.1 g (0.026 mol) of methyl 6-(chlorodifluoromethyl)-2-methylnicotinate (prepared analogously to Heterocycles, 46, 129 (1997) by heating methyl 3-oxobutyrate and 4-amino-1-chloro-1 ,1- difluorobut-3-en-2-one in toluene in the presence of trifluoroacetic acid) is heated at a temperature of 120°C in the presence of 430 mg (0.26 mol) of tris(trimethylsilyl)silane in 150 ml of toluene. After 1.5 hours, the reaction mixture is concentrated and purified on silica gel (hexane/ethyl acetate 13:1). This gives 3.8 g (73% of theory) of methyl 6-difluoromethyl- 2-methylnicotinate as colourless oil. Hydrolysis of the above esters (analogously to Example H1) gives, accordingly, 6-difluoromethyl-2-methylnicotinic acid in the form of white crystals of melting point 135-136°C. 1 H-NMR (CDCI 3 ): 2.68, s, 3H; 6.583, t (J, 55.2Hz), 1 H;: 7.54, d (J, 8.1 Hz), 1 H; 7.54 ppm, d (J, 8.1 Hz), 1 H. Example H31 : 6-(Chlorodifluoromethyl)-2-methylnicotinic acid (compound A-94): 5.0 g (18.62 mmol) of methyl 2-methyl-6-trichloromethylnicotinate (prepared analogously to Heterocycles, 46, 129 (1997)) are cooled to a temperature of -40°C in a pressurized container, and 35 g (1 ,75 mol) of distilled hydrofluoric acid are subsequently passed in at this temperature. The mixture is heated for 10 hours at 200°C (pressure approx. 55 bar). After cooling, the pressure is released using a gas-washing system, HF is removed by suction, and the reaction mixture is poured into ethyl acetate/ice. The ethyl acetate phase is separated off, and the aqueous phase is reextracted using ethyl acetate. The combined ethyl acetate phases are washed with water, dried over sodium sulfate and concentrated, and the residue is triturated with a small amount of hexane and ethyl acetate. Filtration gives 2.2 g (53% of theory) of 6-chlorodifluoromethyl-2-methylnicotinic acid as pale green crystals of melting point 134-135°C. 1 H-NMR (CDCI 3 ): 2.987, s, 3H; 7.64,d (J, 8.1 Hz), 1 H; 8.513 ppm, d (J, 8.1 Hz),1 H. Example H32: 2-r2-(4.6-Dimethoxypyrimidine-2-sulfonylmethyl)-6-trifluoromethylpyridine-3- carbonyl]-3-hvdroxycvclohex-2-enone (compound A1090-B1 ): 100 mg of 2-[2-(4,6-dimethoxypyrimidin-2-ylsulfanylmethyl)-6-trif luoromethylpyridine-3- carbonyl]-3-hydroxycyclohex-2-enone (compound A1088-B1 ) are dissolved in methylene chloride, and 0.3 ml of peracetic acid (39% in acetic acid) is subsequently added dropwise at a temperature of 25°C. After 15 hours at 25°C, the reaction mixture is poured into ethyl acetate and water, and the organic phase is washed with water, dried with sodium sulfate and concentrated. This gives 95 mg of 2-[2-(4,6-dimethoxypyrimidine-2-sulfonylmethyl)-6- PH/5-30762A trifluoromethylpyridine-3-carbonyI]-3-hydroxycyclohex-2-enone in the form of a resin. 1 H- NMR (CDCI3): 3.79, s, 6H; 3.91 , s, 3H; 4.99, s, 2H; 6.09, s, 1 H; 7.52, d (J, 9Hz),1 H; 7.68 ppm, d (J, 9Hz),1 H. In the tables which follow, Ph is the phenyl group and CC an ethyne group. Table 1 : Compounds of the formula XVId: Comp. No. R 3 R 4 R 5 A1 H H H CF 3 0 A2 CH 3 H H CF 3 0 A4 (CH 3 ) 2 CH H H CF 3 0 A5 (CH 3 ) 3 C H H CF 3 0 A6 cyclopropyl H H CF 3 0 Comp. No. R 2 R 3 R 4 R 5 P A8 CH 3 OCH 2 H H CF 3 0 A9 CH 3 O(CH 2 ) 2 H H CF 3 0 A10 Ph H H CF 3 0 A11 PhO H H CF 3 0 A12 PhS H H CF 3 0 A13 PhSO H H CF 3 0 A14 PhSO 2 H H CF 3 0 A15 CH 3 S H H CF 3 0 A16 CH 3 SO H H CF 3 0 A17 CF 3 H H CF 3 0 A18 F 2 CH H H CF 3 0 A19 HCC H H CF 3 0 A20 CH 3 CC H H CF 3 0 A21 CH 2 =CH H H CF 3 0 A23 CH 3 SO 2 N(CH 3 ) H H CF 3 0 A24 (CH 3 ) 2 N H H CF 3 0 A25 (CH 3 ) 2 NSO 2 H H CF 3 0 A27 CH 3 SCH 2 H H CF 3 0 A28 CH 3 SOCH 2 H H CF 3 0 A29 CH 3 SO 2 CH 2 H H CF 3 0 A30 [1.2.4]-triazol-1 -ylmethyl H H CF 3 0 A31 CH 3 CF 3 H CH 3 0 A32 CH 3 CH 3 H CF 3 0 A33 H H H CF 3 CF 2 0 A34 CH 3 H H CF 3 CF 2 0 A35 CHsCH 2 H H CF 3 CF 2 0 A36 cyclopropyl H H CF 3 CF 2 0 A37 (CH 3 ) 3 C H H CF 3 CF 2 0 A38 (CH 3 ) 2 CH H H CF 3 CF 2 0 A39 CH3(CH 2 )2 H H CF 3 CF 2 0 A40 CH 3 OCH 2 H H CF 3 CF 2 0 Comp. No. R 2 R 3 R 4 R 5 P A41 CH 3 O(CH 2 ) 2 H H CF 3 CF 2 0 A42 Ph H H CF 3 CF 2 0 A43 PhO H H CF 3 CF 2 0 A44 PhS H H CF 3 CF 2 0 A45 PhSO H H CF 3 CF 2 0 A46 PhSO 2 H H CF 3 CF 2 0 A47 CH 3 S H H CF 3 CF 2 0 A50 F 2 CH H H CF 3 CF 2 0 A51 HCC H H CF 3 CF 2 0 A52 CH 3 CC H H CF 3 CF 2 0 A53 CH 2 =CH H H CF 3 CF 2 0 A54 CH 2 =CHCH 2 H H CF3CF2 0 A55 CH 3 SO 2 N(CH 3 ) H H CF3CF2 0 A56 (CH 3 ) 2 N H H CF 3 CF 2 0 A57 (CH 3 ) 2 NSO 2 H H CF 3 CF 2 0 A60 CH 3 SOCH 2 H H CF 3 CF 2 0 A61 CH 3 SO 2 CH 2 H H CF 3 CF 2 0 A62 [1.2.4]-triazol-1 -ylmethyl H H CF 3 CF 2 0 A63 H H H CF 3 CF 2 CF 2 0 A64 CH 3 H H C F3C F 2 C F 0 A65 CH 3 CH 2 H H C F 3 C 2C F 2 0 A66 cyclopropyl H H CF 3 CF CF 0 A67 (CH 3 ) 3 C H H CF3CF2CF2 0 A68 (CH 3 ) 2 CH H H C F3C F 2 C F2 0 A69 CH 3 (CH 2 ) 2 H H CF 3 CF2CF 2 0 A70 CH 3 OCH 2 H H CF 3 CF 2 CF 2 0 A71 CH 3 O(CH 2 ) 2 H H CF 3 CF 2 CF 2 0 A72 Ph H H C F 3 C F 2 C F 2 0 A73 PhO H H CF 3 CF 2 CF 2 0 Comp. No. R 2 R 3 R 4 Rs P A74 PhS H H CF 3 CF 2 CF 2 0 A75 PhSO H H CF 3 CF 2 CF 2 0 A76 PhSO 2 H H CF 3 CF 2 CF 2 0 A77 CH 3 S H H CF 3 CF 2 CF 2 0 A78 CH 3 SO H H CF 3 CF 2 CF 2 0 A79 CF 3 H H CF 3 CF 2 CF 2 0 A80 F 2 CH H H CF 3 CF 2 CF 2 0 A81 HCC H H CF 3 CF 2 CF 2 0 A82 CH 3 CC H H CF 3 CF 2 CF 2 0 A83 CH 2 =CH H H CF 3 CF 2 CF 2 0 A84 CH 2 =CHCH 2 H H CF 3 CF 2 CF 2 0 A85 CH 3 SO 2 N(CH 3 ) H H CF 3 CF 2 CF 2 0 A86 (CH 3 ) 2 N H H CF 3 CF 2 CF 2 0 A87 (CH 3 ) 2 NSO 2 H H CF 3 CF 2 CF 2 0 A88 CICH 2 H H CF 3 CF 2 CF 2 0 A89 CH 3 SCH0. H H CF 3 CF 2 CF 2 0 A90 CH 3 SOCH 2 H H CF 3 CF 2 CF 2 0 A91 CH3SO 2 CH 2 H H CF 3 CF 2 CF 2 0 A92 [1.2.4]-triazol-1 -ylmethyl H H CF 3 CF 2 CF 2 0 A93 H H H CF 2 CI 0 A94 CH 3 H H CF 2 CI 0 A95 CH 3 CH 2 H H CF 2 CI 0 A96 cyclopropyl H H CF 2 CI 0 A97 (CH 3 ) 3 C H H CF 2 CI 0 A98 (CH 3 ) 2 CH H H CF 2 CI 0 A99 CH 3 (CH 2 ) 2 H H CF 2 CI 0 A100 CH 3 OCH 2 H H CF 2 CI 0 A101 CH 3 O(CH 2 ) 2 H H CF 2 CI 0 A102 Ph H H CF 2 CI 0 A103 PhO H H CF 2 CI 0 A104 PhS H H CF 2 CI 0 A105 PhSO H H CF 2 CI 0 A106 PhSO 2 H H CF 2 CI 0 Comp. No. R 2 R 3 R 4 Rs P A107 CH 3 S H H CF 2 CI 0 A108 CH 3 SO H H CF 2 CI 0 A109 CF 3 H H CF 2 CI 0 A110 F 2 CH H H CF 2 CI 0 A111 HCC H H CF 2 CI 0 A112 CH 3 CC H H CF 2 CI 0 A113 CH 2 =CH H H CF 2 CI 0 A114 CH 2 =CHCH 2 H H CF 2 CI 0 A115 CH 3 SO 2 N(CH 3 ) H H CF 2 CI 0 A116 (CH 3 ) 2 N H H CF 2 CI 0 A117 (CH 3 ) 2 NSO 2 H H CF 2 CI 0 A118 CICH 2 H H CF 2 CI 0 A121 CH 3 SO 2 CH 2 H H CF 2 CI 0 A122 [1 ,2.4]-triazol-1 -ylmethyl H H CF 2 CI 0 A123 H H H CHF 2 0 A124 CH 3 H H CHF 2 0 A125 CH 3 CH 2 H H CHF 2 0 A126 cyclopropyl H H CHF 2 0 A127 (CH 3 ) 3 C H H CHF 2 0 A128 (CH 3 ) 2 CH H H CHF 2 0 A129 CHs(CH 2 ) 2 H H CHF 2 0 A130 CH 3 OCH 2 H H CHF 2 0 A131 CH 3 O(CH 2 ) 2 H H CHF 2 0 A132 Ph H H CHF 2 0 A133 PhO H H CHF 2 0 A134 PhS H H CHF 2 0 A135 PhSO H H CHF 2 0 A136 PhSO 2 H H CHF 2 0 A137 CH 3 S H H CHF 2 0 A139 CF 3 H H CHF 2 0 Comp. No. R 2 R 3 R 4 Rs P A140 F 2 CH H H CHF 2 0 A141 HCC H H CHF 2 0 A142 CH 3 CC H H CHF 2 0 A143 CH 2 =CH H H CHF 2 0 A144 CH 2 =CHCH 2 H H CHF 2 0 A145 CH 3 SO 2 N(CH 3 ) H H CHF 2 0 A146 (CH 3 ) 2 N H H CHF 2 0 A147 (CH 3 ) 2 NSO 2 H H CHF 2 0 A148 CICH 2 H H CHF 2 0 A149 CHsSCH 2 H H CHF 2 0 A150 CH 3 SOCH 2 H H CHF 2 0 A151 CH 3 SO 2 CH 2 H H CHF 2 0 A152 [1.2.4]-triazol-1 -ylmethyl H H CHF 2 0 A156 cyclopropyl H H CCI3 0 A157 (CH 3 ) 3 C H H CCI 3 0 A160 CH 3 OCH 2 H H CCI 3 0 A161 CH 3 O(CH 2 ) 2 H H CCI3 0 A162 Ph H H CCI 3 0 A164 PhS H H CCI 3 0 A165 PhSO H H CCI 3 0 A166 PhSO 2 H H CCI 3 0 A167 CH 3 S H H CCI 3 0 A169 CF 3 H H CCI 3 0 A171 HCC H H CCI 3 0 Comp. No. R 2 R 3 R 4 R 5 P A173 CH 2 =CH H H CCI 3 0 A174 CH 2 =CHCH 2 H H CC 0 A175 CH 3 SO 2 N(CH 3 ) H H CCI3 0 A177 (CH 3 ) 2 NSO 2 H H CCI3 0 A178 CICH 2 H H CCI 3 0 A179 CH 3 SCH 2 H H CCI 3 0 A182 [1.2.4]-triazol-1 -ylmethyl H H CCI3 0 A183 H H CH 3 CF 3 0 A184 CH 3 H CH 3 CF 3 0 A185 CH 3 CH 2 H CH 3 CF 3 0 A186 cyclopropyl H CH 3 CF 3 0 A187 (CH 3 ) 3 C H CH 3 CF 3 0 A188 (CH 3 ) 2 CH H CH 3 CF 3 0 A189 CH 3 (CH 2 ) 2 H CH 3 CF 3 0 A190 CH 3 OCH 2 H CH 3 CF 3 0 A191 CH 3 O(CH 2 ) 2 H CH 3 CF 3 0 A192 Ph H CH 3 CF 3 0 A193 PhO H CH 3 CF 3 0 A194 PhS H CH 3 CF 3 0 A195 PhSO H CH 3 CF 3 0 A196 PhSO 2 H CH 3 CF 3 0 A197 CH 3 S H CH 3 CF 3 0 A198 CH 3 SO H CH 3 CF 3 0 A199 CF 3 H CH 3 CF 3 0 A200 F 2 CH H CH 3 CF 3 0 A201 HCC H CH 3 CF 3 0 A202 CHgCC H CH 3 CF 3 0 A203 CH 2 =CH H CH 3 CF 3 0 A204 CH 2 =CHCH 2 H CH 3 CF 3 0 A205 CH 3 SO 2 N(CH 3 ) H CH 3 CF 3 0 Comp. No. R 2 R 3 R 4 R 5 P A206 (CH 3 ) 2 N H CH 3 CF 3 0 A207 (CH 3 ) 2 NSO 2 H CH 3 CF 3 0 A208 CICH 2 H CH 3 CF 3 0 A210 CH 3 SOCH 2 H CH 3 CF 3 0 A211 CH 3 SO 2 CH 2 H CH 3 CF 3 0 A212 H H CH 3 CF 3 CF 2 0 A213 CH 3 H CH 3 CF 3 CF 2 0 A214 CH 3 CH 2 H CH 3 CF3CF2 0 A215 cyclopropyl H CH 3 CF 3 CF 2 0 A216 (CH 3 ) 3 C H CH 3 CF 3 CF 2 0 A217 (CH 3 ) 2 CH H CH 3 CF 3 CF 2 0 A218 CH 3 (CH 2 ) 2 H CH 3 CF 3 CF 2 0 A219 CH 3 OCH 2 H CH 3 CF 3 CF 2 0 A220 CH 3 O(CH 2 ) 2 H CH 3 CF 3 CF 2 0 A221 Ph H CH 3 CF 3 CF 2 0 A222 PhO H CH 3 CF 3 CF 2 0 A223 PhS H CH 3 CF 3 CF 2 0 A224 PhSO H CH 3 CF 3 CF 2 0 A225 PhSO 2 H CH 3 CF 3 CF 2 0 A226 CH 3 S H CH 3 CF 3 CF 2 0 A227 CH 3 SO H CH 3 CF 3 CF 2 0 A228 CF 3 H CH 3 CF 3 CF 2 0 A229 F 2 CH H CH 3 CF 3 CF 2 0 A230 HCC H CH 3 CF 3 CF 2 0 A231 CH 3 CC H CH 3 CF 3 CF 2 0 A232 CH 2 =CH H CH 3 CF 3 CF 2 0 A233 CH =CHCH 2 H CH 3 CF 3 CF 2 0 A234 CH 3 SO 2 N(CH 3 ) H CH 3 CF 3 CF 2 0 A235 (CH 3 ) 2 N H CH 3 CF 3 CF 2 0 A236 (CH 3 ) 2 NSO 2 H CH 3 CF 3 CF 2 0 A237 CICH 2 H CH 3 CF 3 CF 2 0 A238 CH 3 SCH 2 H CH 3 CF 3 CF 2 0 Comp. No. R 2 R 3 R 4 Rs P A239 CH 3 SOCH 2 H CH 3 CF 3 CF 2 0 A240 CH 3 SO 2 CH 2 H CH 3 CF 3 CF 2 0 A241 H H CH 3 CF 3 CF 2 CF 2 0 A242 CH 3 H CH 3 CF 3 CF 2 CF 2 0 A243 CH 3 CH 2 H CH 3 CF 3 CF 2 CF 2 0 A244 cyclopropyl H CH 3 CF 3 CF 2 CF 2 0 A245 (CH 3 ) 3 C H CH 3 CF 3 CF 2 CF 2 0 A246 (CH 3 ) 2 CH H CH 3 CF 3 CF 2 CF 2 0 A247 CH 3 (CH 2 ) 2 H CH 3 CF 3 CF 2 CF 2 0 A248 CH 3 OCH 2 H CH 3 CF 3 CF 2 CF 2 0 A249 CH 3 O(CH 2 ) 2 H CH 3 CF 3 CF 2 CF 2 0 A250 Ph H CH 3 CF 3 CF 2 CF 2 0 A251 PhO H CH 3 CF 3 CF 2 CF 2 0 A252 PhS H CH 3 CF3CF2CF2 0 A253 PhSO H CH 3 CF 3 CF 2 CF 2 0 A254 PhSO 2 H CH 3 CF 3 CF 2 CF 2 0 A255 CH 3 S H CH 3 CF 3 CF 2 CF 2 0 A256 CH 3 SO H CH 3 CF 3 CF 2 CF 2 0 A257 CF 3 H CH 3 CF 3 CF 2 CF 2 0 A258 F 2 CH H CH 3 CF 3 CF 2 CF 2 0 A259 HCC H CH 3 CF 3 CF 2 CF 2 0 A260 CH 3 CC H CH 3 CF 3 CF 2 CF 2 0 A261 CH 2 =CH H CH 3 CF 3 CF 2 CF 2 0 A262 CH 2 =CHCH2 H CH 3 CF 3 CF 2 CF 2 0 A263 CH 3 SO 2 N(CH 3 ) H CH 3 CF 3 CF 2 CF 2 0 A264 (CH 3 ) 2 N H CH 3 CF 3 CF 2 CF 2 0 A265 (CH 3 ) 2 NSO 2 H CH 3 CF 3 CF 2 CF 2 0 A266 CICH 2 H CH 3 CF 3 CF 2 CF 2 0 A267 CH 3 SCH 2 H CH 3 CF 3 CF 2 CF 2 0 A268 CH 3 SOCH 2 H CH 3 CF 3 CF 2 CF 2 0 A269 CH 3 SO 2 CH 2 H CH 3 CF 3 CF 2 CF 2 0 A270 H H CH 3 CF 2 CI 0 A271 CH 3 H CH 3 CF 2 CI 0 Comp. No. R 2 R 3 R 4 R 5 P A272 CH 3 CH 2 H CH 3 CF 2 CI 0 A273 cyclopropyl H CH 3 CF 2 CI 0 A274 (CH 3 ) 3 C H CH 3 CF 2 CI 0 A275 (CH 3 ) 2 CH H CH 3 CF 2 CI 0 A276 CHs(CH 2 ) 2 H CH 3 CF 2 CI 0 A277 CH 3 OCH 2 H CH 3 CF 2 CI 0 A278 CH 3 O(CH 2 ) 2 H CH 3 CF 2 CI 0 A279 Ph H CH 3 CF 2 CI 0 A280 PhO H CH 3 CF 2 CI 0 A281 PhS H CH 3 CF 2 CI 0 A282 PhSO H CH 3 CF 2 CI 0 A283 PhSO 2 H CH 3 CF 2 CI 0 A284 CH 3 S H CH 3 CF 2 CI 0 A285 CH 3 SO H CH 3 CF 2 CI 0 A286 CF 3 H CH 3 CF 2 CI 0 A287 F 2 CH H CH 3 CF 2 CI 0 A288 HCC H CH 3 CF 2 CI 0 A289 CH 3 CC H CH 3 CF 2 CI 0 A290 CH 2 =CH H CH 3 CF 2 CI 0 A291 CH 2 =CHCH H CH 3 CF 2 CI 0 A292 CH 3 SO 2 N(CH 3 ) H CH 3 CF≥CI 0 A293 (CH 3 ) 2 N H CH 3 CF 2 CI 0 A294 (CH 3 ) 2 NSO 2 H CH 3 CF 2 CI 0 A295 CICH 2 H CH 3 CF 2 CI 0 A296 CH 3 SCH H CH 3 CF 2 CI 0 A297 CH 3 SOCH 2 H CH 3 CF 2 CI 0 A298 CH 3 SO 2 CH 2 H CH 3 CF 2 CI 0 A299 H H CH 3 CHF 2 0 A300 CH 3 H CH 3 CHF 2 0 A302 cyclopropyl H CH 3 CHF 2 0 A303 (CH 3 ) 3 C H CH 3 CHF 2 0 A304 (CH 3 ) 2 CH H CH 3 CHF 2 0 Comp. No. R 2 R 3 R 4 Rs P A305 CH 3 (CH 2 ) 2 H CH 3 CHF 2 0 A306 CH 3 OCH 2 H CH 3 CHF 2 0 A307 CH 3 O(CH 2 ) 2 H CH 3 CHF 2 0 A308 Ph H CH 3 CHF 2 0 A309 PhO H CH 3 CHF 2 0 A310 PhS H CH 3 CHF 2 0 A311 PhSO H CH 3 CHF 2 0 A312 PhSO 2 H CH 3 CHF 2 0 A313 CH 3 S H CH 3 CHF 2 0 A315 CF 3 H CH 3 CHF 2 0 A316 F 2 CH H CH 3 CHF 2 0 A317 HCC H CH 3 CHF 2 0 A318 CH 3 CC H CH 3 CHF 2 0 A319 CH 2 =CH H CH 3 CHF 2 0 A320 CH 2 =CHCH 2 H CH 3 CHF 2 0 A321 CH 3 SO 2 N(CH 3 ) H CH 3 CHF 2 0 A322 (CH 3 ) 2 N H CH 3 CHF 2 0 A323 (CH 3 ) 2 NSO 2 H CH 3 CHF 2 0 A324 CICH 2 H CH 3 CHF 2 0 A325 CH 3 SCH 2 H CH 3 CHF 2 0 A326 CH 3 SOCH 2 H CH 3 CHF 2 0 A327 CH 3 SO 2 CH 2 H CH 3 CHF 2 0 A328 H H CH 3 CCI 3 0 A329 CH 3 H CH 3 CCI 3 0 A330 CH 3 CH 2 H CH 3 CCI 3 0 A332 (CH 3 ) 2 CH H CH 3 CCI3 0 A333 cyclopropyl H CH 3 CCI3 0 A334 CH 3 (CH 2 ) 2 H CH 3 CCI3 0 A336 CH 3 O(CH 2 ) 2 H CH 3 CCI3 0 Comp. No. R 2 R 3 R 4 R 5 P A340 PhSO H CH 3 CCI 3 0 A341 PhSO 2 H CH 3 CC 0 A349 CH 2 =CHCH 2 H CH 3 CCI 3 0 A350 CH 3 SO 2 N(CH 3 ) H CH 3 CCb 0 A352 (CH 3 ) 2 NSO 2 H CH 3 CCI 3 0 A355 CH 3 SOCH 2 H CH 3 CCI 3 0 A356 CH3SO2CH2 H CH 3 CC 0 A360 cyclopropyl H Ph CF 3 0 A361 (CH 3 ) 3 C H Ph CF 3 0 A362 (CH 3 ) 2 CH H Ph CF 3 0 A363 CH 3 (CH 2 ) 2 H Ph CF 3 0 A364 CH 3 OCH 2 H Ph CF 3 0 A365 CH 3 O(CH 2 ) 2 H Ph CF 3 0 A366 Ph H Ph CF 3 0 A367 PhO H Ph CF 3 0 A368 PhS H Ph CF 3 0 A369 PhSO H Ph CF 3 0 A370 PhSO 2 H Ph CF 3 0 Comp. No. R 2 R 3 R 4 Rs P A371 CH 3 S H Ph CF 3 0 A373 CF 3 H Ph CF 3 0 A374 F 2 CH H Ph CF 3 0 A375 HCC H Ph CF 3 0 A376 CH 3 CC H Ph CF 3 0 A377 CH 2 =CH H Ph CF 3 0 A378 CH 2 =CHCH 2 H Ph CF 3 0 A379 CH 3 SO 2 N(CH 3 ) H Ph CF 3 0 A380 (CH 3 ) 2 N H Ph CF 3 0 A381 (CH 3 ) 2 NSO 2 H Ph CF 3 0 A382 CICH 2 H Ph CF 3 0 A383 CH 3 SCH 2 H Ph CF 3 0 A384 CH 3 SOCH 2 H Ph CF 3 0 A385 CH 3 SO 2 CH 2 H Ph CF 3 0 A386 H H Ph CF 3 CF 2 0 A387 CH 3 H Ph CF 3 CF 2 0 A388 CH 3 CH 2 H Ph CF 3 CF 2 0 A389 cyclopropyl H Ph CF 3 CF 2 0 A390 (CH 3 ) 3 C H Ph CF 3 CF 2 0 A391 (CH 3 ) 2 CH H Ph CF 3 CF 2 0 A392 CHs(CH 2 ) 2 H Ph CF 3 CF 2 0 A393 CH 3 OCH 2 H Ph CF 3 CF 2 0 A394 CH 3 O(CH 2 ) 2 H Ph CF 3 CF 2 0 A395 Ph H Ph CF 3 CF 2 0 A396 PhO H Ph CF 3 CF 2 0 A397 PhS H Ph CF 3 CF 2 0 A398 PhSO H Ph CF 3 CF 2 0 A399 PhSO 2 H Ph CF 3 CF 2 0 A400 CH 3 S H Ph CF 3 CF 2 0 A401 CH 3 SO H Ph CF 3 CF 2 0 A402 CF 3 H Ph CF 3 CF 2 0 A403 F 2 CH H Ph CF 3 CF 2 0 Comp. No. R 2 R 3 R 4 Rs P A404 HCC H Ph CF 3 CF 2 0 A405 CH 3 CC H Ph CF 3 CF 2 0 A406 CH 2 =CH H Ph CF 3 CF 2 0 A407 CH 2 =CHCH H Ph CF 3 CF 2 0 A408 CH 3 SO 2 N(CH 3 ) H Ph CF 3 CF 2 0 A409 (CH 3 ) 2 N H Ph CF 3 CF 2 0 A410 (CH 3 ) 2 NSO 2 H Ph CF 3 CF 2 0 A41 1 CICH 2 H Ph CF 3 CF 2 0 A412 CH 3 SCH 2 H Ph CF 3 CF 2 0 A413 CH 3 SOCH 2 H Ph CF 3 CF 2 0 A414 CH 3 SO CH 2 H Ph CF 3 CF 2 0 A415 H H Ph CF 3 CF 2 CF 2 0 A416 CH 3 H Ph CF 3 CF 2 CF 2 0 A417 CHsCH 2 H Ph CF 3 CF2CF2 0 A418 cyclopropyl H Ph CF 3 CF 2 CF 2 0 A419 (CH 3 ) 3 C H Ph CF 3 CF 2 CF 2 0 A420 (CH 3 ) 2 CH H Ph CF 3 CF 2 CF 0 A421 CH 3 (CH 2 ) 2 H Ph CF 3 CF 2 CF 2 0 A422 CH 3 OCH 2 H Ph CF 3 CF 2 CF 2 0 A423 CH 3 O(CH 2 ) 2 H Ph C F 3 C F 2 C r 2 0 A424 Ph H Ph CF 3 CF 2 Cr 2 0 A425 PhO H Ph CFsCF 2 CF 2 0 A426 PhS H Ph C F 3 C F 2 C F 0 A427 PhSO H Ph C F 3 C F 2 C F 2 0 A428 PhSO 2 H Ph C F 3 C 2 C F 2 0 A429 CH 3 S H Ph CF 3 CF 2 CF 2 0 A430 CH 3 SO H Ph C F 3 C F 2 C F 2 0 A431 CF 3 H Ph CF 3 CF 2 CF 2 0 A432 F 2 CH H Ph CF 3 CF 2 CF 2 0 A433 HCC H Ph CFsCF 2 CF 2 0 A434 CH 3 CC H Ph CF 3 CF 2 CF 2 0 A435 CH 2 =CH H Ph C F 3 C F 2 C F 2 0 A436 CH 2 =CHCH 2 H Ph C F 3 C F 2 C F 2 0 Comp. No. R 2 R 3 R 4 Rs P A437 CH 3 SO 2 N(CH 3 ) H Ph CF 3 CF 2 CF 2 0 A438 (CH 3 ) 2 N H Ph C F 3 C F 2 C F 2 0 A439 (CH 3 ) 2 NSO 2 H Ph C F 3 C F C F 2 0 A440 CICH≥ H Ph CF 3 CF 2 CF 2 0 A441 CH 3 SCH 2 H Ph CF 3 CF 2 CF 2 0 A442 CH 3 SOCH 2 H Ph CF 3 CF 2 CF 2 0 A443 CH 3 SO 2 CH2 H Ph CF 3 CF 2 CF 2 0 A444 H H Ph CF 2 CI 0 A445 CH 3 H Ph CF 2 CI 0 A446 CH 3 CH 2 H Ph CF 2 CI 0 A447 cyclopropyl H Ph CF 2 CI 0 A448 (CH 3 ) 3 C H Ph CF 2 CI 0 A449 (CH 3 ) 2 CH H Ph CF 2 CI 0 A450 CH 3 (CH 2 ) 2 H Ph CF 2 CI 0 A451 CH 3 OCH 2 H Ph CF 2 CI 0 A452 CH 3 O(CH 2 ) 2 H Ph CF 2 CI 0 A453 Ph H Ph CF 2 CI 0 A454 PhO H Ph CF 2 CI 0 A455 PhS H Ph CF 2 CI 0 A456 PhSO H Ph CF 2 CI 0 A457 PhSO 2 H Ph CF 2 CI 0 A458 CH 3 S H Ph CF 2 CI 0 A459 CH 3 SO H Ph CF 2 CI 0 A460 CF 3 H Ph CF 2 CI 0 A461 F 2 CH H Ph CF 2 CI 0 A462 HCC H Ph CF 2 CI 0 A463 CH 3 CC H Ph CF 2 CI 0 A464 CH 2 =CH H Ph CF 2 CI 0 A465 CH 2 =CHCH 2 H Ph CF 2 CI 0 A466 CH 3 SO 2 N(CH 3 ) H Ph CF 2 CI 0 A467 (CH 3 ) 2 N H Ph CF 2 CI 0 A468 (CH 3 ) 2 NSO 2 H Ph CF 2 CI 0 A469 CICH 2 H Ph CF 2 CI 0 Comp. No. R 2 R3 R 4 Rs P A470 CH 3 SCH 2 H Ph CF 2 CI 0 A471 CH 3 SOCH 2 H Ph CF 2 CI 0 A472 CH 3 SO 2 CH 2 H Ph CF 2 CI 0 A473 H H Ph CHF 2 0 A474 CH 3 H Ph CHF 2 0 A475 CH 3 CH 2 H Ph CHF 2 0 A476 cyclopropyl H Ph CHF 2 0 A477 (CH 3 ) 3 C H Ph CHF 2 0 A478 (CH 3 ) 2 CH H Ph CHF 2 0 A479 CH 3 (CH 2 ) 2 H Ph CHF 2 0 A480 CH 3 OCH 2 H Ph CHF 2 0 A481 CH 3 O(CH 2 ) 2 H Ph CHF 2 0 A482 Ph H Ph CHF 2 0 A483 PhO H Ph CHF 2 0 A484 PhS H Ph CHF 2 0 A485 PhSO H Ph CHF 2 0 A486 PhSO 2 H Ph CHF 2 0 A487 CH 3 S H Ph CHF 2 0 A488 CH 3 SO H Ph CHF 2 0 A489 CF 3 H Ph CHF 2 0 A490 F 2 CH H Ph CHF 2 0 A491 HCC H Ph CHF 2 0 A492 CH 3 CC H Ph CHF 2 0 A493 CH 2 =CH H Ph CHF 2 0 A494 CH 2 =CHCH 2 H Ph CHF 2 0 A495 CH 3 SO 2 N(CH 3 ) H Ph CHF 2 0 A496 (CH 3 ) 2 N H Ph CHF 2 0 A497 (CH 3 ) 2 NSO 2 H Ph CHF 2 0 A498 CICH 2 H Ph CHF 2 0 A499 CH 3 SCH 2 H Ph CHF 2 0 A500 CH 3 SOCH 2 H Ph CHF 2 0 A501 CH 3 SO CH 2 H Ph CHF 2 0 Comp. No. R 2 R 3 R 4 Rs P A503 CH 3 H Ph CCb 0 A505 cyclopropyl H Ph CCI3 0 A506 (CH 3 ) 3 C H Ph CCI 3 0 A507 (CH 3 ) 2 CH H Ph CCI 3 0 A508 CH3(CH2) 2 H Ph CCI 3 0 A510 CH 3 O(CH 2 ) 2 H Ph CCI 3 0 A511 Ph H Ph CCI 3 0 A512 PhO H Ph CCI 3 0 A513 PhS H Ph CCI 3 0 A514 PhSO H Ph CCI 3 0 A515 PhSO 2 H Ph CCI 3 0 A517 CH 3 SO H Ph CCI 3 0 A518 CF 3 H Ph CCI 3 0 A519 F 2 CH H Ph CCI 3 0 A520 HCC H Ph CCI 3 0 A522 CH 2 =CH H Ph CCI 3 0 A523 CH 2 =CHCH 2 H Ph CCI 3 0 A524 CH 3 SO 2 N(CH 3 ) H Ph CCI 3 0 A526 (CH 3 ) 2 NSO 2 H Ph CCI 3 0 A527 CICH 2 H Ph CCI 3 0 A530 CH 3 SO 2 CH 2 H Ph CCI3 0 A531 H CH 3 H CF 3 0 A532 H CH 3 CH 2 H CF 3 0 A533 H cyclopropyl H CF 3 0 A534 H (CH 3 ) 3 CH H CF 3 0 A535 H (CH 3 ) 2 CH H CF 3 0 Comp. No. R 2 R 3 R 4 Rs P A536 H CH 3 (CH 2 ) 2 H CF 3 0 A537 H CH 3 OCH 2 H CF 3 0 A538 H CH 3 O(CH 2 ) 2 H CF 3 0 A539 H Ph H CF 3 0 A540 H PhO H CF 3 0 A541 H PhS H CF 3 0 A542 H PhSO H CF 3 0 A543 H PhSO 2 H CF 3 0 A544 H CH 3 S H CF 3 0 A546 H CF 3 H CF 3 0 A547 H F 2 CH H CF 3 0 A548 H HCC H CF 3 0 A549 H CH 3 CC H CF 3 0 A550 H CH 2 =CH H CF 3 0 A551 H CH 2 =CHCH H CF 3 0 A552 H CH 3 SO 2 N(CH 3 ) H CF 3 0 A553 H (CH 3 ) 2 N H CF 3 0 A554 H (CH 3 ) 2 NSO 2 H CF 3 0 A555 H CH 3 SCH 2 H CF 3 0 A556 H CH 3 SOCH 2 H CF 3 0 A558 H CH 3 H CF 3 CF 2 0 A559 H CH 3 CH 2 H CF 3 CF 2 0 A560 H cyclopropyl H CF 3 CF 2 0 A561 H (CH 3 ) 3 C H CF 3 CF 2 0 A562 H (CH 3 ) 2 CH H CF 3 CF 2 0 A563 H CH 3 (CH 2 ) 2 H CF 3 CF 2 0 A564 H CH 3 OCH 2 H CF 3 CF 2 0 A565 H CH 3 O(CH 2 ) 2 H CF 3 CF 2 0 A566 H Ph H CF 3 CF 2 0 Comp. No. R 2 R 3 R 4 Rs P A569 H PhSO H CF 3 CF 2 0 A570 H PhSO 2 H CF 3 CF 2 0 A571 H CH 3 S H CF 3 CF 2 0 A572 H CH 3 SO H CF 3 CF 2 0 A573 H CF 3 H CF 3 CF 2 0 A574 H F 2 CH H CF 3 CF 2 0 A575 H HCC H CF 3 CF 2 0 A576 H CH 3 CC H CF 3 CF 2 0 A577 H CH 2 =CH H CF 3 CF 2 0 A578 H CH 2 =CHCH 2 H CF 3 CF 2 0 A579 H CH 3 SO 2 N(CH 3 ) H CF 3 CF 2 0 A581 H (CH 3 ) 2 NSO 2 H CF 3 CF 2 0 A582 H CH 3 SCH 2 H CF 3 CF 2 0 A583 H CH 3 SOCH 2 H CF 3 CF 2 0 A584 H CH 3 SO 2 CH 2 H CF 3 CF 2 0 A585 H CH 3 H CF 3 CF 2 CF 2 0 A586 H CH 3 CH 2 H CF 3 CF 2 CF 2 0 A587 H cyclopropyl H CF 3 CF 2 CF 2 0 A588 H (CH 3 ) 3 C H CF 3 CF 2 CF 2 0 A589 H (CH 3 ) 2 CH H CF 3 CF 2 CF 2 0 A590 H CH 3 (CH 2 ) 2 H CF 3 CF 2 CF 2 0 A591 H CH 3 OCH 2 H CF 3 CF 2 CF 2 0 A592 H CH 3 O(CH 2 ) 2 H CF 3 CF 2 CF 2 0 A593 H Ph H CF 3 CF 2 CF 2 0 A594 H PhO H CF 3 CF 2 CF 2 0 A595 H PhS H CF 3 CF 2 CF 2 0 A596 H PhSO H CF 3 CF 2 CF 2 0 A597 H PhSO 2 H CF 3 CF 2 CF 2 0 A598 H CH 3 S H CF 3 CF 2 CF 2 0 A599 H CH 3 SO H CF 3 CF 2 CF 2 0 A600 H CF 3 H CF 3 CF 2 CF 2 0 A601 H F 2 CH H CF 3 CF 2 CF 2 0 Comp. No. R 2 R 3 R 4 Rs P A602 H HCC H CF 3 CF 2 CF 2 0 A603 H CH 3 CC H C F 3 C F 2 C F 2 0 A604 H CH 2 =CH H C F 3 C F 2 C F 2 0 A606 H CH 3 SO 2 N(CH 3 ) H CF3CF2CF 2 0 A607 H (CH 3 ) 2 N H CF 3 CF2CF 0 A608 H (CH 3 ) 2 NSO 2 H CF 3 CF 2 CF 2 0 A609 H CH 3 SCH2 H CF 3 CF 2 CF 2 0 A610 H CH3SOCH2 H CF3CF 2 CF 2 0 A611 H CH3SO2CH 2 H CF 3 CF 2 CF 2 0 A612 H CH 3 H CF 2 CI 0 A614 H cyclopropyl H CF 2 CI 0 A615 H (CH 3 ) 3 C H CF 2 CI 0 A616 H (CH 3 ) 2 CH H CF 2 CI 0 A617 H CHs(CH 2 ) 2 H CF 2 CI 0 A618 H CH 3 OCH 2 H CF 2 CI 0 A619 H CH 3 O(CH 2 ) 2 H CF 2 CI 0 A620 H Ph H CF 2 CI 0 A621 H PhO H CF 2 CI 0 A622 H PhS H CF 2 CI 0 A623 H PhSO H CF 2 CI 0 A624 H PhSO 2 H CF 2 CI 0 A625 H CH 3 S H CF 2 CI 0 A626 H CH 3 SO H CF 2 CI 0 A627 H CF 3 H CF 2 CI 0 A628 H F 2 CH H CF≥CI 0 A629 H HCC H CF 2 CI 0 A630 H CH 3 CC H CF 2 CI 0 A631 H CH 2 =CH H CF 2 CI 0 A633 H CH 3 SO 2 N(CH 3 ) H CF 2 CI 0 A634 H (CH 3 ) 2 N H CF 2 CI 0 Comp. No. R 2 R 3 R 4 Rs P A635 H (CH 3 ) 2 NSO 2 H CF 2 CI 0 A638 H CH3SO2CH2 H CF 2 CI 0 A639 H CH 3 H CHF 2 0 A641 H cyclopropyl H CHF 2 0 A642 H (CH 3 ) 3 C H CHF 2 0 A643 H (CH 3 ) 2 CH H CHF 2 0 A644 H CH 3 (CH 2 ) 2 H CHF 2 0 A645 H CH 3 OCH 2 H CHF 2 0 A646 H CH 3 O(CH 2 ) 2 H CHF 2 0 A647 H Ph H CHF 2 0 A648 H PhO H CHF 2 0 A649 H PhS H CHF 2 0 A650 H PhSO H CHF 2 0 A651 H PhSO 2 H CHF 2 0 A652 H CH 3 S H CHF 2 0 A653 H CH 3 SO H CHF 2 0 A654 H CF 3 H CHF 2 0 A655 H F 2 CH H CHF 2 0 A656 H HCC H CHF 2 0 A657 H CH 3 CC H CHF 2 0 A658 H CH 2 =CH H CHF 2 0 A659 H CH 2 =CHCH 2 H CHF 2 0 A660 H CH 3 SO 2 N(CH 3 ) H CHF 2 0 A661 H (CH 3 ) 2 N H CHF 2 0 A662 H (CH 3 ) 2 NSO 2 H CHF 2 0 A663 H CH 3 SCH 2 H CHF 2 0 A664 H CH 3 SOCH 2 H CHF 2 0 A665 H CH 3 SO 2 CH 2 H CHF 2 0 A666 H CH 3 H CCI 3 0 A667 H CH 3 CH 2 H CCI 3 0 Comp. No. R 2 R 3 R 4 Rs P A668 H cyclopropyl H CCI3 0 A670 H (CH 3 ) 2 CH H CCI 3 0 A673 H CH 3 O(CH 2 ) 2 H CCI3 0 A677 H PhSO H CCI 3 0 A678 H PhSO 2 H CCI 3 0 A679 H CH 3 S H CCI 3 0 A680 H CHgSO H CCI 3 0 A681 H CF 3 H CCI 3 0 A682 H F 2 CH H CCI 3 0 A683 H HCC H CCI 3 0 A684 H CH 3 CC H CCI 3 0 A685 H CH 2 =CH H CCI 3 0 A687 H CH 3 SO 2 N(CH 3 ) H CCI 3 0 A688 H (CH 3 ) 2 N H CCI 3 0 A689 H (CH 3 ) 2 NSO 2 H CCI3 0 A691 H CH 3 SOCH 2 H CCI 3 0 A695 H cyclopropyl CH 3 CF 3 0 A698 H CH 3 (CH 2 ) 2 CH 3 CF 3 0 A699 H CH 3 OCH 2 CH 3 CF 3 0 A700 H CH 3 O(CH 2 ) 2 CH 3 CF 3 0 Comp. No. R 2 R 3 R 4 Rs P A701 H Ph CH 3 CF 3 0 A702 H PhO CH 3 CF 3 0 A703 H PhS CH 3 CF 3 0 A704 H PhSO CH 3 CF 3 0 A705 H PhSO 2 CH 3 CF 3 0 A706 H CH 3 S CH 3 CF 3 0 A707 H CH 3 SO CH 3 CF 3 0 A708 H CF 3 CH 3 CF 3 0 A709 H F 2 CH CH 3 CF 3 0 A710 H HCC CH 3 CF 3 0 A711 H CH 3 CC CH 3 CF 3 0 A712 H CH 2 =CH CH 3 CF 3 0 A713 H CH 2 = CHCH 2 CH 3 CF 3 0 A714 H CH 3 SO 2 N(CH 3 ) CH 3 CF 3 0 A715 H (CH 3 ) 2 N CH 3 CF 3 0 A716 H (CH 3 ) 2 NSO 2 CH 3 CF 3 0 A717 H CH 3 SCH 2 CH 3 CF 3 0 A718 H CH 3 SOCH 2 CH 3 CF 3 0 A719 H CH 3 SO 2 CH 2 CH 3 CF 3 0 A720 H CH 3 CH 3 CF 3 CF 2 0 A721 H CH 3 CH 2 CH 3 CF 3 CF 2 0 A722 H cyclopropyl CH 3 CF3CF2 0 A723 H (CH 3 ) 3 C CH 3 CF 3 CF 2 0 A724 H (CH 3 ) 2 CH CH 3 CF 3 CF 2 0 A725 H CH 3 (CH 2 )2 CH 3 CF 3 CF 2 0 A726 H CH 3 OCH 2 CH 3 CF3CF2 0 A727 H CH 3 O(CH 2 ) 2 CH 3 CF 3 CF 2 0 A728 H Ph CH 3 CF 3 CF 2 0 A729 H PhO CH 3 CF 3 CF 2 0 A730 H PhS CH 3 CF 3 CF 2 0 A731 H PhSO CH 3 CF 3 CF 2 0 A732 H PhSO 2 CH 3 CF 3 CF 2 0 A733 H CH 3 S CH 3 CF 3 CF 2 0 Comp. No. R 2 R 3 R 4 Rs P A734 H CHgSO CH 3 CF 3 CF 2 0 A735 H CF 3 CH 3 CF 3 CF 2 0 A736 H F 2 CH CH 3 CF 3 CF 2 0 A737 H HCC CH 3 CF 3 CF 2 0 A738 H CH 3 CC CH 3 CF 3 CF 2 0 A739 H CH 2 =CH CH 3 CF 3 CF 2 0 A740 H CH 2 =CHCH 2 CH 3 CF 3 CF 2 0 A741 H CH 3 SO 2 N(CH 3 ) CH 3 CF 3 CF 2 0 A742 H (CH 3 ) 2 N CH 3 CF 3 CF 2 0 A743 H (CH 3 ) 2 NSO 2 CH 3 CF 3 CF 2 0 A744 H CH3SCH 2 CH 3 CF 3 CF 2 0 A745 H CH3SOCH2 CH 3 CF 3 CF 2 0 A746 H CH3SO2CH2 CH 3 CF 3 CF 2 0 A747 H CH 3 CH 3 CF 3 CF 2 CF 2 0 A748 H CH3CH2 CH 3 CF 3 CF 2 CF 2 0 A749 H cyclopropyl CH 3 CF3CF 2 CF 2 0 A750 H (CH 3 ) 3 C CH 3 CF 3 CF 2 CF 2 0 A751 H (CH 3 ) 2 CH CH 3 CF 3 CF 2 CF 2 0 A752 H CH 3 (CH2) 2 CH 3 CF3CF 2 CF 2 0 A753 H CH 3 OCH 2 CH 3 CF 3 CF 2 CF 2 0 A754 H CH 3 O(CH 2 ) 2 CH 3 CF 3 CF 2 CF 2 0 A755 H Ph CH 3 CF 3 CF 2 CF 2 0 A756 H PhO CH 3 CF 3 CF 2 CF 2 0 A757 H PhS CH 3 CF 3 CF 2 CF 2 0 A758 H PhSO CH 3 CF 3 CF 2 CF 2 0 A759 H PhSO 2 CH 3 CF 3 CF 2 CF 2 0 A760 H CH 3 S CH 3 CF 3 CF 2 CF 2 0 A761 H CH 3 SO CH 3 CF 3 CF 2 CF 2 0 A762 H CF 3 CH 3 CF 3 CF 2 CF 2 0 A763 H F 2 CH CH 3 CF3CF 2 CF 2 0 A764 H HCC CH 3 CF3CF 2 CF 2 0 A765 H CH 3 CC CH 3 CF 3 CF 2 CF 2 0 A766 H CH 2 =CH CH 3 CF 3 CF 2 CF 2 0 Comp. No. R 2 R 3 R 4 Rs P A767 H CH 2 =CHCH 2 CH 3 CF 3 CF 2 CF 2 0 A768 H CH 3 SO 2 N(CH 3 ) CH 3 CF 3 CF 2 CF 2 0 A769 H (CH 3 ) 2 N CH 3 CF 3 CF 2 CF 2 0 A770 H (CH 3 ) 2 NSO 2 CH 3 CF 3 CF 2 CF 2 0 A771 H CH 3 SCH 2 CH 3 CF 3 CF 2 CF 2 0 A772 H CH 3 SOCH 2 CH 3 CF 3 CF 2 CF 2 0 A773 H CHsSO 2 CH 2 CH 3 CF 3 CF 2 CF 2 0 A774 H CH 3 CH 3 CF 2 CI 0 A775 H CH 3 CH 2 CH 3 CF 2 CI 0 A776 H cyclopropyl CH 3 CF 2 CI 0 A777 H (CH 3 ) 3 C CH 3 CF 2 CI 0 A778 H (CH 3 ) 2 CH CH 3 CF 2 CI 0 A779 H CH 3 (CH 2 ) 2 CH 3 CF 2 CI 0 A780 H CH 3 OCH 2 CH 3 CF 2 CI 0 A781 H CH 3 O(CH 2 ) 2 CH 3 CF 2 CI 0 A782 H Ph CH 3 CF 2 CI 0 A783 H PhO CH 3 CF 2 CI 0 A784 H PhS CH 3 CF 2 CI 0 A785 H PhSO CH 3 CF 2 CI 0 A786 H PhSO 2 CH 3 CF 2 CI 0 A787 H CH 3 S CH 3 CF 2 CI 0 A788 H CH 3 SO CH 3 CF 2 CI 0 A789 H CF 3 CH 3 CF 2 CI 0 A790 H F 2 CH CH 3 CF 2 CI 0 A791 H HCC CH 3 CF 2 CI 0 A792 H CH 3 CC CH 3 CF 2 CI 0 A793 H CH 2 =CH CH 3 CF 2 CI 0 A794 H CH 2 =CHCH 2 CH 3 CF 2 CI 0 A795 H CH 3 SO 2 N(CH 3 ) CH 3 CF 2 CI 0 A796 H (CH 3 ) 2 N CH 3 CF 2 CI 0 A797 H (CH 3 ) 2 NSO2 CH 3 CF 2 CI 0 A798 H CH3SCH2 CH 3 CF 2 CI 0 A799 H CH 3 SOCH 2 CH 3 CF 2 CI 0 Comp. No. R 2 R 3 R 4 Rs P A800 H CH 3 SO 2 CH 2 CH 3 CF 2 CI 0 A801 H CH 3 CH 3 CHF 2 0 A802 H CH 3 CH 2 CH 3 CHF 2 0 A803 H cyclopropyl CH 3 CHF 2 0 A804 H (CH 3 ) 3 C CH 3 CHF 2 0 A805 H (CH 3 ) 2 CH CH 3 CHF 2 0 A806 H CH 3 (CH 2 ) 2 CH 3 CHF 2 0 A807 H CH 3 OCH 2 CH 3 CHF 2 0 A808 H CH 3 O(CH 2 ) 2 CH 3 CHF 2 0 A809 H Ph CH 3 CHF 2 0 A810 H PhO CH 3 CHF 2 0 A811 H PhS CH 3 CHF 2 0 A812 H PhSO CH 3 CHF 2 0 A813 H PhSO 2 CH 3 CHF 2 0 A814 H CH 3 S CH 3 CHF 2 0 A815 H CH 3 SO CH 3 CHF 2 0 A816 H CF 3 CH 3 CHF 2 0 A817 H F 2 CH CH 3 CHF 2 0 A818 H HCC CH 3 CHF 2 0 A819 H CH 3 CC CH 3 CHF 2 0 A820 H CH 2 =CH CH 3 CHF 2 0 A821 H CH 2 =CHCH 2 CH 3 CHF 2 0 A822 H CH 3 SO 2 N(CH 3 ) CH 3 CHF 2 0 A823 H (CH 3 ) 2 N CH 3 CHF 2 0 A824 H (CH 3 ) 2 NSO 2 CH 3 CHF 2 0 A825 H CH 3 SCH 2 CH 3 CHF 2 0 A826 H CH 3 SOCH 2 CH 3 CHF 2 0 A827 H CH 3 SO 2 CH 2 CH 3 CHF 2 0 A830 H cyclopropyl CH 3 CCI 3 0 A831 H (CH 3 ) 3 C CH 3 CCI 3 0 A832 H (CH 3 ) 2 CH CH 3 CCI 3 0 Comp. No. R 2 R 3 R 4 Rs P A833 H CH 3 (CH 2 ) 2 CH 3 CCb 0 A834 H CH 3 OCH 2 CH 3 CCb 0 A835 H CH 3 O(CH 2 ) 2 CH 3 CCb 0 A836 H Ph CH 3 CCb 0 A837 H PhO CH 3 CCb 0 A838 H PhS CH 3 CCb 0 A839 H PhSO CH 3 CCb 0 A840 H PhSO 2 CH 3 CCb 0 A841 H CH 3 S CH 3 CCb 0 A842 H CH 3 SO CH 3 CCb 0 A843 H CF 3 CH 3 CCb 0 A844 H F 2 CH CH 3 CCb 0 A845 H HCC CH 3 CCb 0 A846 H CH 3 CC CH 3 CCb 0 A847 H CH 2 =CH CH 3 CCb 0 A848 H CH 2 =CHCH 2 CH 3 CCb 0 A849 H CH 3 SO 2 N(CH 3 ) CH 3 CCb 0 A850 H (CH 3 ) 2 N CH 3 CCb 0 A851 H (CH 3 ) 2 NSO 2 CH 3 CCb 0 A852 H CH 3 SCH 2 CH 3 CCb 0 A853 H CH 3 SOCH 2 CH 3 CCb 0 A854 H CHsSO 2 CH 2 CH 3 CCb 0 A855 H CH 3 Ph CF 3 0 A856 H CH 3 CH 2 Ph CF 3 0 A858 H (CH 3 ) 2 CH Ph CF 3 0 A859 H cyclopropyl Ph CF 3 0 A860 H CH 3 (CH 2 ) 2 Ph CF 3 0 A862 H CH 3 O(CH 2 ) 2 Ph CF 3 0 A863 H Ph Ph CF 3 0 A864 H PhO Ph CF 3 0 A865 H PhS Ph CF 3 0 Comp. No. R 2 R 3 R 4 Rs P A866 H PhSO Ph CF 3 0 A867 H PhSO 2 Ph CF 3 0 A868 H CH 3 S Ph CF 3 0 A869 H CH 3 SO Ph CF 3 0 A870 H CF 3 Ph CF 3 0 A871 H F 2 CH Ph CF 3 0 A872 H HCC Ph CF 3 0 A873 H CH 3 CC Ph CF 3 0 A874 H CH 2 =CH Ph CF 3 0 A875 H CH 2 =CHCH Ph CF 3 0 A876 H CH 3 SO 2 N(CH 3 ) Ph CF 3 0 A877 H (CH 3 ) 2 N Ph CF 3 0 A878 H (CH 3 ) 2 NSO 2 Ph CF 3 0 A879 H CH 3 SCH 2 Ph CF 3 0 A880 H CH 3 SOCH 2 Ph CF 3 0 A881 H CH 3 SO 2 CH 2 Ph CF 3 0 A882 H CH 3 Ph CF 3 CF 2 0 A883 H CH 3 CH 2 Ph CF 3 CF 2 0 A884 H cyclopropyl Ph CF3CF2 0 A885 H (CH 3 ) 3 C Ph CF 3 CF 2 0 A886 H (CH 3 ) 2 CH Ph CF 3 CF 2 0 A887 H CH 3 (CH 2 ) 2 Ph CF 3 CF 2 0 A888 H CH 3 OCH 2 Ph CF 3 CF 2 0 A889 H CH 3 O(CH 2 ) 2 Ph CF 3 CF 2 0 A890 H Ph Ph CF 3 CF 2 0 A891 H PhO Ph CF 3 CF 2 0 A892 H PhS Ph CF 3 CF 2 0 A893 H PhSO Ph CF 3 CF 2 0 A894 H PhSO 2 Ph CF 3 CF 2 0 A895 H CH 3 S Ph CF 3 CF 2 0 A896 H CH 3 SO Ph CF 3 CF 2 0 A897 H CF 3 Ph CF 3 CF 2 0 A898 H F 2 CH Ph CF 3 CF 2 0 o o > > > > > > > > > > co co co co co co co co co CO C > _O C>ø C>O C>O >CQ C>O >CO C>O C>O C>O >CO C>O C>O C>O >CO C>O C>ø C>O C>O C>O C>O C>O >CO 3 co co r ro ro r ro ro r ro ro o o o o o o o o o ■ α CO -^ o co oo -sj cn j^ co ) o (o oo Ni o ϋi ^ ω i -' O CO 00 -si Φ en co ro o CO x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x X TJ TJ TJ TJ TJ TJ TJ TJ TJ TJ TJ TJ TJ TJ TJ TJ TJ TJ TJ J TJ TJ TJ TJ TJ TJ T __r __ΓJ T_TJ T_3J- T3J _ _ __r _τ zr __r _τ _τ _ _ IΓ __Γ _T IΓ __Γ _T 3- D- - _ _ zr IT 3- - TZJΓ T__ΓJ *X o o o o o o o o o o o O O O TJ Comp. No. R 2 R 3 R 4 Rs P A932 H (CH 3 ) 2 NSO 2 Ph CF3CF 2 CF 2 0 A933 H CH3SCH2 Ph CF 3 CF 2 CF 2 0 A934 H CH 3 SOCH 2 Ph CF 3 CF 2 CF 2 0 A935 H CH 3 SO 2 CH 2 Ph CF3CF2CF 2 0 A936 H CH 3 Ph CF 2 CI 0 A937 H CHsCH 2 Ph CF 2 CI 0 A938 H cyclopropyl Ph CF 2 CI 0 A939 H (CH 3 ) 3 C Ph CF 2 CI 0 A940 H (CH 3 ) 2 CH Ph CF 2 CI 0 A941 H CH 3 (CH 2 ) 2 Ph CF 2 CI 0 A942 H CH 3 OCH 2 Ph CF 2 CI 0 A943 H CH 3 O(CH 2 ) 2 Ph CF 2 CI 0 A944 H Ph Ph CF 2 CI 0 A945 H PhO Ph CF 2 CI 0 A946 H PhS Ph CF 2 CI 0 A947 H PhSO Ph CF 2 CI 0 A948 H PhSO 2 Ph CF 2 CI 0 A949 H CH 3 S Ph CF 2 CI 0 A951 H CF 3 Ph CF 2 CI 0 A952 H F 2 CH Ph CF 2 CI 0 A953 H HCC Ph CF 2 CI 0 A954 H CH 3 CC Ph CF 2 CI 0 A955 H CH 2 =CH Ph CF 2 CI 0 A956 H CH 2 =CHCH 2 Ph CF 2 CI 0 A957 H CH 3 SO 2 N(CH 3 ) Ph CF 2 CI 0 A958 H (CH 3 ) 2 N Ph CF 2 CI 0 A959 H (CH 3 ) 2 NSO 2 Ph CF 2 CI 0 A960 H CH 3 SCH 2 Ph CF 2 CI 0 A961 H CH 3 SOCH 2 Ph CF 2 CI 0 A962 H CH3SO 2 CH 2 Ph CF 2 CI 0 A963 H CH 3 Ph CHF 2 0 A964 H CHsCH 2 Ph CHF 2 0 omp. No. R 2 R 3 R 4 Rs P A965 H (CH 3 ) 3 C Ph CHF 2 0 A966 H (CH 3 ) 2 CH Ph CHF 2 0 A967 H cyclopropyl Ph CHF 2 0 A968 H CH 3 (CH 2 ) 2 Ph CHF 2 0 A969 H CH 3 OCH 2 Ph CHF 2 0 A970 H CH 3 O(CH 2 ) 2 Ph CHF 2 0 A971 H Ph Ph CHF 2 0 A972 H PhO Ph CHF 2 0 A973 H PhS Ph CHF 2 0 A974 H PhSO Ph CHF 2 0 A975 H PhSO 2 Ph CHF 2 0 A976 H CH 3 S Ph CHF 2 0 A977 H CH 3 SO Ph CHF 2 0 A978 H CF 3 Ph CHF 2 0 A979 H F 2 CH Ph CHF 2 0 A980 H HCC Ph CHF 2 0 A981 H CH 3 CC Ph CHF 2 0 A982 H CH 2 =CH Ph CHF 2 0 A983 H CH 2 =CHCH 2 Ph CHF 2 0 A984 H CH 3 SO 2 N(CH 3 ) Ph CHF 2 0 A985 H (CH 3 ) 2 N Ph CHF 2 0 A986 H (CH 3 ) 2 NSO 2 Ph CHF 2 0 A988 H CH 3 SOCH 2 Ph CHF 2 0 A989 H CH 3 SO 2 CH 2 Ph CHF 2 0 A990 H CH 3 Ph CCb 0 A991 H CH 3 CH 2 Ph CCb 0 A992 H (CH 3 ) 3 C Ph CCb 0 A993 H (CH 3 ) 2 CH Ph CCb 0 A994 H cyclopropyl Ph CCb 0 A995 H CH3(CH2)2 Ph CCI 3 0 A997 H CH 3 O(CH 2 ) 2 Ph CCI 3 0 Comp. No. R 2 R 3 R 4 Rs P A998 H Ph Ph CCI 3 0 A999 H PhO Ph CCI 3 0 A1000 H PhS Ph CCI 3 0 A1001 H PhSO Ph CCI 3 0 A1002 H PhSO 2 Ph CCI 3 0 A1003 H CH 3 S Ph CCb 0 A1004 H CH 3 SO Ph CCb 0 A1005 H CF 3 Ph CCb 0 A1006 H F 2 CH Ph CCb 0 A1007 H HCC Ph CCb 0 A1008 H CH 3 CC Ph CCb 0 A1009 H CH 2 =CH Ph CCb 0 A1010 H CH 2 =CHCH 2 Ph CCb 0 A1011 H CH 3 SO 2 N(CH 3 ) Ph CCb 0 A1012 H (CH 3 ) 2 N Ph CCb 0 A1013 H (CH 3 ) 2 NSO 2 Ph CCb 0 A1014 H CHsSCH 2 Ph CCb 0 A1015 H CH 3 SOCH 2 Ph CCI 3 0 A1016 H CH 3 SO 2 CH 2 Ph CCb 0 A1020 NC H H CF 3 0 A1021 CH 3 SO 2 O H H CF 3 0 A1022 CH 3 O H H CF 3 0 A1023 CH 3 CH 2 O H H CF 3 0 A1024 CH 2 CH=CH 2 O H H CF 3 0 A1025 HCCCH 2 O H H CF 3 0 A1026 PhCH 2 S H H CF 3 0 A1027 PhCH 2 SO 2 H H CF 3 0 A1028 CICH 2 CH 2 H H CF 3 0 A1029 BrCH 2 H H CF 3 0 A1030 FCH 2 H H CF 3 0 Comp. No. R 2 R 3 R Rs P A1031 CHF 2 CH 2 H H CF 3 0 A1033 [1 ,3]-imidazol-1 -ylmethyl H H CF 3 0 A1034 CHCI 2 CH 2 H H CF 3 0 A1035 CICH=CH H H CF 3 0 A1036 CI 2 C=CH H H CF 3 0 A1037 CF 3 CH=CH H H CF 3 0 A1038 CICC H H CF 3 0 A1039 PhCH 2 H H CF 3 0 A1041 CH 3 OH H CF 3 0 A1042 CH 3 F H CF 3 0 A1043 CH 3 Cl H CF 3 0 A1044 F CH 3 H CF 3 0 A1045 Cl CH 3 H CF 3 0 A1046 H F H CF 3 0 A1047 H Cl H CF 3 0 A1048 H Br H CF 3 0 A1049 H OH H CF 3 0 A1051 H OCHF 2 H CF 3 0 A1052 H OSO 2 CH 3 H CF 3 0 A1053 H OSO 2 CF 3 H CF 3 0 A1054 H CICH 2 H CF 3 0 A1055 H BrCH 2 H CF 3 0 A1056 H FCH 2 H CF 3 0 A1057 H CHF 2 CH H CF 3 0 A1059 H triazolylmethyl H CF 3 0 A1061 H CICH=CH H CF 3 0 A1062 H CI 2 C=CH H CF 3 0 A1063 H CF 3 CH=CH H CF 3 0 A1064 H CICC H CF 3 0 A1065 H CH 3 C(O) H CF 3 0 A1066 H Ph H CF 3 0 A1067 H SO 2 CH 3 H CF 3 0 A1068 H SO 2 CF 3 H CF 3 0 A1069 H NC H CF 3 0 A1070 H NO 2 H CF 3 0 A1071 CH 3 H F CF 3 0 A1072 CH 3 H Ci CF 3 0 A1073 CH 3 H Br CF 3 0 A 1074 CH 3 H NC CF 3 0 A1075 CH 3 H CH 3 O CF 3 0 A1076 CH 3 H CH 3 S CF 3 0 A1077 CH 3 H CH 3 SO CF 3 0 A1078 CH 3 H CH 3 SO 2 CF 3 0 A1079 CH 3 CH 2 OCH 2 H H CF 3 0 A1080 PhOCH 2 H H CF 3 0 A1081 ø- ∞B ' H H CF 3 0 A1082 (CH 3 ) 2 CH 2 OCH 2 H H CF 3 0 A1083 BrCH CH 2 H H CF 3 0 A1084 FCH CH 2 H H CF 3 0 Comp. No. R 2 R 3 R 4 Rs P A1091 cyclopropyl-CH 2 H H CF 3 0 A1092 2,2-dichlorocycloprop-1 - H H CF 3 0 yi A1093 CH 3 OC(O)CH=CH H H CF 3 0 A1094 CH 3 CH 2 OC(O)CH=CH H H CF 3 0 A1095 CICH 2 CH=CH H H CF 3 0 A1096 CH=C=CH H H CF 3 0 A1097 (CH 3 ) 2 NCH 2 H H CF 3 0 A1098 HOCH 2 H H CF 3 0 A1099 CH 3 C(O)OCH 2 H H CF 3 0 A1100 PhC(O)OCH 2 H H CF 3 0 A1101 PhCH 2 CH 2 H H CF 3 0 A1102 CH 3 OC(O)CH 2 H H CF 3 0 A1103 NCCH 2 H H CF 3 0 A1104 CH 3 (CH 2 ) 7 SCH 2 H H CF 3 0 A1105 CH 3 (CH 2 ) 7 SOCH 2 H H CF 3 0 A1106 CH 3 (CH 2 ) 7 SO 2 CH 2 H H CF 3 0 A1108 CICH 2 CC H H CF 3 0 A1109 CHF 2 CH 2 CH 2 H H CF 3 0 A1110 CHCI 2 CH 2 CH 2 H H CF 3 0 A1111 CF 3 SO 2 O H H CF 3 0 Comp. No. R 2 R 3 R 4 Rs P A1115 H H CF 3 0 A1116 H H CF 3 A1117 rγ CH - H H CF 3 0 A1118 CH 3 ON=CHCH 2 H H CF 3 0 A1119 O=CHCH 2 H H CF 3 0 A1120 CH 3 CH 2 OCH 2 H H CF 2 CI 0 A1121 PhOCH 2 H H CF 2 CI 0 A1122 ty ™' H H CF 2 CI 0 A1123 (CH 3 ) 2 CH 2 OCH 2 H H CF 2 CI 0 A1124 BrCH 2 H H CF 2 CI 0 A1125 FCH 2 H H CF 2 CI 0 A1132 cyclopropyl-CH 2 H H CF 2 CI 0 A1133 2,2-dichlorocycloprop-1 ■ H H CF 2 CI 0 yi Comp. No. R 2 R 3 R 4 Rs P A1134 CH 3 OC(O)CH=CH H H CF 2 CI 0 A1135 CH 3 CH 2 OC(O)CH=CH H H CF 2 CI 0 A1136 CICH 2 CH=CH H H CF 2 CI 0 A1137 CH=C=CH H H CF 2 CI 0 A1138 (CH 3 ) 2 NCH 2 H H CF 2 CI 0 A1139 HOCH 2 H H CF 2 CI 0 A1140 CH 3 C(O)OCH 2 H H CF 2 CI 0 A1141 PhC(O)OCH 2 H H CF 2 CI 0 A1142 PhCH 2 H H CF 2 CI 0 A1143 CH 3 OC(O)CH 2 H H CF 2 CI 0 A1144 NCCH 2 H H CF 2 CI 0 A1145 CH 3 (CH 2 ) SCH 2 H H CF 2 CI 0 A1146 CH 3 (CH 2 ) 7 SOCH 2 H H CF 2 CI 0 A1147 CH 3 (CH 2 ) 7 SO 2 CH 2 H H CF 2 CI 0 A1149 H H CF 2 CI 0 A1150 H H CF 2 CI 0 A1151 H H CF 2 CI 0 A1152 H H CF 2 CI 0 A1156 r^ .CH 2 H H CF 2 CI 0 A1157 ,^y CH - H H CF 2 CI 0 A1158 ry 0 "- H H CF 2 CI 0 A1159 CH 3 ON=CHCH 2 H H CF 2 CI 0 Comp. No. R 2 R 3 R 4 Rs P A1160 O=CHCH 2 H H CF 2 CI 0 A1161 CH 3 CH 2 OCH 2 H H CF 2 H 0 A1162 PhOCH 2 H H CF 2 H 0 A1164 (CH 3 ) 2 CH 2 OCH 2 H H CF 2 H 0 A1165 BrCH 2 H H CF 2 H 0 A1166 FCH 2 H H CF 2 H 0 A1170 / O- ^N^^SCH, H H CF 2 H 0 A1172 ^° N^S0 2 CH 2 H H CF 2 H 0 A1173 cyclop ropyl-CH 2 H H CF 2 H 0 A1174 2,2-dichlorocycloprop-1 - H H CF 2 H 0 yi A1175 CH 3 OC(O)CH=CH H H CF 2 H 0 A1176 CH 3 CH 2 OC(O)CH=CH H H CF 2 H 0 A1177 CICH 2 CH=CH H H CF 2 H 0 A1178 CH=C=CH H H CF 2 H 0 A1179 (CH 3 ) 2 NCH2 H H CF 2 H 0 A1180 HOCH 2 H H CF 2 H 0 A1181 CH 3 C(O)OCH 2 H H CF 2 H 0 A1182 PhC(O)OCH 2 H H CF 2 H 0 o Q. O O O O O O O O O O O O O O O O O O O O O 0\ P. W X X X X X X X X X X X X X X X X X X LL LL LL LL υ H X __L U_. 1_L L_L _JL U_. __L u_ LL u_ U- LL LL LL LL LL Li- LL o o o o o o o O O O o o o O o O o o o o o o o o o r x x x x x x x X X X X X x x x X x x x x CO CΛ Ct X X X X X X X X X X X X x x x x x g x x x e 6 7* O in CO ^ 00 CΛ O 1- CM CO "* in CD h- 00 <Λ O -— CM O *tf in ca r-~ co 00 00 00 CO 00 CO CO O CΛ CΛ Φ Φ Λ CΛ <Λ φ CΛ o o O O O o o o o o Q. CM CM CM CM CM CM CM CM CM o E o < < < < < < < < < < < < < < < < < < < < < O Comp. No. R 2 R 3 R 4 Rs P A1209 CH 3 OCH 2 OCH 2 H H CF 3 0 A1210 CH 3 H H CF 3 1 A1212 cyclopropyl H H CF 3 1 A1213 CHs(CH 2 ) 2 H H CF 3 1 A1214 CH 3 OCH 2 H H CF 3 1 A1215 CF 3 H H CF 3 1 A1216 F 2 CH H H CF 3 1 A1219 CH 3 CF 3 H CH 3 1 A1220 CH 3 CH 2 OCH 2 H H CF 3 1 A1221 PhOCH 2 H H CF 3 1 A1222 (CH 3 ) 2 CH 2 OCH 2 H H CF 3 1 A1223 BrCH 2 H H CF 3 1 A1224 FCH 2 H H CF 3 1 / °^ ^S0 2 CH 2 A1226 H H CF 3 1 A1227 cyclopropyl-CH 2 H H CF 3 1 A1228 2,2-dichlorocycloprop-1 - H H CF 3 1 yi A1229 (CH 3 ) 2 NCH 2 H H CF 3 1 A1230 HOCH 2 H H CF 3 1 A1231 CH 3 C(O)OCH 2 H H CF 3 1 A1232 PhC(O)OCH 2 H H CF 3 1 A1233 PhCH 2 H H CF 3 1 A1234 CH 3 OC(O)CH 2 H H CF 3 1 A1235 NCCH 2 H H CF 3 1 A1236 CH 3 (CH 2 ) 7 SO 2 CH 2 H H CF 3 1 A1237 Br H H CF 3 1 Comp. No. R 2 R 3 R 4 Rs P A1238 Cl H H CF 3 1 A1239 O=CHCH 2 H H CF 3 1 A1240 CH 3 H H CF 2 CI 1 A1241 CH 3 CH 2 H H CF 2 CI 1 A1242 cyclopropyl H H CF 2 CI 1 A1243 CH 3 (CH 2 ) 2 H H CF 2 CI 1 A1244 CH 3 OCH 2 H H CF 2 CI 1 A1245 CF 3 H H CF 2 CI 1 A1246 F 2 CH H H CF 2 CI 1 A1247 CICH 2 H H CF 2 CI 1 A1248 CH 3 SO 2 CH 2 H H CF 2 CI 1 A1249 CH 3 CF 3 H CF 2 CI 1 A1250 CH3CH 2 OCH2 H H CF 2 CI 1 A1251 PhOCH 2 H H CF 2 CI 1 A1252 (CH 3 ) 2 CH 2 OCH 2 H H CF 2 CI 1 A1253 BrCH 2 H H CF 2 CI 1 A1254 FCH 2 H H CF 2 CI 1 A1257 cyclopropyl-CH 2 H H CF 2 CI 1 A1258 2,2-dichlorocycloprop-1 - H H CF 2 Ci 1 yi A1259 (CH 3 ) 2 NCH 2 H H CF 2 CI 1 A1260 HOCH 2 H H CF 2 CI 1 A1261 CH 3 C(O)OCH 2 H H CF 2 CI 1 A1262 PhC(O)OCH 2 H H CF 2 CI 1 A1263 PhCH 2 H H CF 2 CI 1 A1264 CH 3 OC(O)CH 2 H H CF 2 CI 1 A1265 NCCH 2 H H CF 2 CI 1 A1266 CH 3 (CH 2 ) 7 SO 2 CH 2 H H CF 2 CI 1 Comp. No. R 2 R 3 R 4 Rs P A1267 Br H H CF 2 CI 1 A1268 Cl H H CF 2 CI 1 A1269 O=CHCH 2 H H CF 2 CI 1 A1270 CH 3 H H CF 2 H 1 A1271 CH 3 CH 2 H H CF 2 H 1 A1272 cyclopropyl H H CF 2 H 1 A1273 CH 3 (CH 2 ) 2 H H CF 2 H 1 A1274 CH 3 OCH 2 H H CF 2 H 1 A1275 CF 3 H H CF 2 H 1 A1276 F 2 CH H H CF 2 H 1 A1277 CICH 2 H H CF 2 H 1 A1278 CHsSO 2 CH 2 H H CF 2 H 1 A1279 CH 3 CF 3 H CF 2 H 1 A1280 CH 3 CH 2 OCH 2 H H CF 2 H 1 A1281 PhOCH 2 H H CF 2 H 1 A1282 (CH 3 ) 2 CH 2 OCH 2 H H CF 2 H 1 A1283 BrCH 2 H H CF 2 H 1 A1284 FCH 2 H H CF 2 H 1 A1287 cyclopropyl-CH 2 H H CF 2 H 1 A1288 2,2-dichlorocycloprop-1 - H H CF 2 H 1 yi A1289 (CH 3 ) 2 NCH 2 H H CF 2 H 1 A1290 HOCH 2 H H CF 2 H 1 A1291 CH 3 C(O)OCH 2 H H CF 2 H 1 A1292 PhC(O)OCH 2 H H CF 2 H 1 A1293 PhCH 2 H H CF 2 H 1 A1294 CH 3 OC(O)CH 2 H H CF 2 H 1 A1295 NCCH 2 H H CF 2 H 1 Comp. No. R 2 R 3 R 4 Rs P A1296 CH 3 (CH 2 ) 7 SO 2 CH 2 H H CF 2 H A1297 Br H H CF 2 H A1298 Cl H H CF 2 H A1299 O=CHCH 2 H H CF 2 H A1300 CH 3 H H CF 3 CF 2 A1301 HO H Ph CF 3 0 A1302 CH 3 H CH 2 =CH CF 3 0 A1304 HO CH 3 H CF 3 0 A1305 HO H H CF 3 0 A1306 (CH 3 CH 2 ) 2 N(O)CO H H CF 3 0 A1307 CH 3 H Tosyl-O CF 3 0 A1308 CH 3 H CH 3 CC CF 3 0 A1309 CH 3 H HCC CF 3 0 A1310 CH 3 H CICH 2 CC CF 3 0 A1311 CH 3 H PhCH 2 O CF 3 0 A1312 CH 3 H CF 3 SO 2 O CF 3 0 A1313 CH 3 H (CH 3 ) 2 N CF 3 0 A1314 CH 3 H CH 3 C(O)O CF 3 0 A1315 CH 3 H CH 3 CH 2 C(O)O CF 3 0 A1316 CH 3 H PhC(O)O CF 3 0 A1317 CH 3 H 3-Pyridyl CF 3 0 A1318 CH 3 OCH 2 OCH 2 H H CF 2 CI 0 A1319 CH 3 OCH 2 OCH 2 H H CF 2 H 0 A1320 CH 3 OCH 2 OCH 2 H H CF 2 CF 3 0 A1321 CH 3 OCH 2 OCH 2 H H CF 3 1 A1322 CH 3 O H CH 3 CF 3 0 In Table 2 which follows, Q is Qi and Q 1 the radicals B which follow: Table 2: Radicals B: Radical R fi R 7 s Ra Rio W B1 H H H H OH CH 2 B2 CH 3 H H H OH CH 2 B5 (CH 3 ) 2 CH H H H OH CH 2 B6 (CH 3 ) 3 C H H H OH CH 2 B7 CH 3 S H H H OH CH 2 B8 CH 3 SO H H H OH CH 2 B10 Ph H H H OH CH 2 B12 CH 3 OC(O) H H H OH CH 2 B13 CH 3 CH 2 OC(O) H H H OH CH 2 B14 CH 2 =CHCH 2 H H H OH CH 2 B15 HCCCH 2 H H H OH CH 2 B16 CF 3 H H H OH CH 2 B17 (CH 3 ) 2 NSO 2 H H H OH CH 2 B18 (CH 3 ) 2 N H H H OH CH 2 B19 PhO H H H OH CH 2 B20 PhS H H H OH CH 2 B21 PhSO H H H OH CH 2 B22 PhSO 2 H H H OH CH 2 Radical R 6 R 7 R 8 R 9 R10 W B23 CN H H H OH CH 2 B24 CH 3 CH 3 H H OH CH 2 B25 CHsCH 2 CH 3 H H OH CH 2 B26 CH 3 CH 2 CH 2 CH 3 H H OH CH 2 B27 (CH 3 ) 2 CH CH 3 H H OH CH 2 B28 (CH 3 ) 3 C CH 3 H H OH CH 2 B29 CH 3 S CH 3 H H OH CH 2 B30 CH 3 SO CH 3 H H OH CH 2 B31 CH 3 SO 2 CH 3 H H OH CH 2 B32 Ph CH 3 H H OH CH 2 B33 CH 3 O CH 3 H H OH CH 2 B34 CH 3 OC(O) CH 3 H H OH CH 2 B35 CH 3 CH 2 OC(O) CH 3 H H OH CH 2 B36 CH 2 =CHCH 2 CH 3 H H OH CH 2 B37 HCCCH 2 CH 3 H H OH CH 2 B38 CF 3 CH 3 H H OH CH 2 B39 (CH 3 ) 2 NSO 2 CH 3 H H OH CH 2 B40 (CH 3 ) 2 N CH 3 H H OH CH 2 B41 PhO CH 3 H H OH CH 2 B42 PhS CH 3 H H OH CH 2 B43 PhSO CH 3 H H OH CH 2 B44 PhSO 2 CH 3 H H OH CH 2 B45 CN CH 3 H H OH CH 2 B46 CH 3 H CH 3 H OH CH 2 B47 CH 3 CH 2 H CH 3 H OH CH 2 B48 CH 3 CH 2 CH 2 H CH 3 H OH CH 2 B49 (CH 3 ) 2 CH H CH 3 H OH CH 2 B50 (CH 3 ) 3 C H CH 3 H OH CH 2 B51 CH 3 S H CH 3 H OH CH 2 B53 CH 3 SO 2 H CH 3 H OH CH 2 B54 Ph H CH 3 H OH CH 2 B55 CH 3 O H CH 3 H OH CH 2 Radical Re R 7 R 8 R9 R10 W B56 CH 3 OC(O) H CH 3 H OH CH 2 B57 CH 3 CH 2 OC(O) H CH 3 H OH CH 2 B58 CH 2 =CHCH 2 H CH 3 H OH CH 2 B59 HCCCH 2 H CH 3 H OH CH 2 B60 CF 3 H CH 3 H OH CH 2 B61 (CH 3 ) 2 NSO 2 H CH 3 H OH CH 2 B62 (CH 3 ) 2 N H CH 3 H OH CH 2 B63 PhO H CH 3 H OH CH 2 B64 PhS H CH 3 H OH CH 2 B65 PhSO H CH 3 H OH CH 2 B66 PhSO 2 H CH 3 H OH CH 2 B67 CN H CH 3 H OH CH 2 B68 CH 3 CH 3 CH 3 H OH CH 2 B69 CH 3 CH 2 CH 3 CH 3 H OH CH 2 B70 CH 3 CH 2 CH 2 CH 3 CH 3 H OH CH 2 B71 (CH 3 ) 2 CH CH 3 CH 3 H OH CH 2 B72 (CH 3 ) 3 C CH 3 CH 3 H OH CH 2 B73 CH 3 S CH 3 CH 3 H OH CH 2 B74 CH 3 SO CH 3 CH 3 H OH CH 2 B75 CH 3 SO 2 CH 3 CH 3 H OH CH 2 B76 Ph CH 3 CH 3 H OH CH 2 B77 CH 3 O CH 3 CH 3 H OH CH 2 B78 CH 3 OC(O) CH 3 CH 3 H OH CH 2 B79 CH 3 CH 2 OC(O) CH 3 CH 3 H OH CH 2 B80 CH 2 =CHCH 2 CH 3 CH 3 H OH CH 2 B81 HCCCH 2 CH 3 CH 3 H OH CH 2 B82 CF 3 CH 3 CH 3 H OH CH 2 B83 (CH 3 ) 2 NSO 2 CH 3 CH 3 H OH CH 2 B84 (CH 3 ) 2 N CH 3 CH 3 H OH CH 2 B85 PhO CH 3 CH 3 H OH CH 2 B86 PhS CH 3 CH 3 H OH CH 2 B87 PhSO CH 3 CH 3 H OH CH 2 B88 PhSO 2 CH 3 CH 3 H OH CH 2 X CD CD CD CI) CD CD CD CD CD 2 2 2 2 2 2 2 2 2 2 2 o ro CD » ro to _- -i. -- 2 2 O O o o o o o o CrO CroO CroO CroO CroO CD oCO3 CCOD CCOD CCOD 00 9: -> ■ O CO 00 ^J CΛ en *- eo ro -^ CO 00 -si o Φ en .fc- CO ro o (O ffl ffl ϋl ^ U M -' O CO o X X X X X X X X X X o X ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox o X X X X X X - XT -Xr XT ° X ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox x - Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox Ox sX ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox < ^- Radical Re R 7 RB R 9 R10 W B122 CH 3 CH 2 OC(O) CH 3 CH 2 H H OH CH 2 B124 HCCCH 2 CH 3 CH 2 H H OH CH 2 B125 CF 3 CH 3 CH 2 H H OH CH 2 B126 (CH 3 ) 2 NSO 2 CH 3 CH 2 H H OH CH 2 B127 (CH 3 ) 2 N CH 3 CH H H OH CH 2 B128 PhO CH 3 CH 2 H H OH CH 2 B129 PhS CH 3 CH 2 H H OH CH 2 B130 PhSO CH 3 CH 2 H H OH CH 2 B131 PhSO 2 CH 3 CH 2 H H OH CH 2 B132 CN CH 3 CH H H OH CH 2 B133 H H H H OH CHCH 3 B134 CH 3 H H H OH CHCH 3 B136 CH 3 CH 2 CH 2 H H H OH CHCH 3 B137 (CH 3 ) 2 CH H H H OH CHCH 3 B138 (CH 3 ) 3 C H H H OH CHCH 3 B139 CH 3 S H H H OH CHCH 3 B140 CH 3 SO H H H OH CHCH 3 B141 CH 3 SO 2 H H H OH CHCH 3 B142 Ph H H H OH CHCH 3 B144 CH 3 OC(O) H H H OH CHCH 3 B145 CH 3 CH 2 OC(O) H H H OH CHCH 3 B146 CH 2 =CHCH 2 H H H OH CHCH 3 B147 HCCCH 2 H H H OH CHCH 3 B148 CF 3 H H H OH CHCH 3 B149 (CH 3 ) 2 NSO 2 H H H OH CHCH 3 B150 (CH 3 ) 2 N H H H OH CHCH 3 B151 PhO H H H OH CHCH 3 B152 PhS H H H OH CHCH 3 B153 PhSO H H H OH CHCH 3 B154 PhSO 2 H H H OH CHCH 3 Radical Re R 7 Rs R 9 R10 W B155 CN H H H OH CHCH 3 B156 CH 3 CH 3 H H OH CHCH 3 B157 CH 3 CH 2 CH 3 H H OH CHCH 3 B158 CH 3 CH 2 CH 2 CH 3 H H OH CHCH 3 B159 (CH 3 ) 2 CH CH 3 H H OH CHCH 3 B160 (CH 3 ) 3 C CH 3 H H OH CHCH 3 B161 CH 3 S CH 3 H H OH CHCH 3 B162 CH 3 SO CH 3 H H OH CHCH 3 B163 CH 3 SO 2 CH 3 H H OH CHCHg B164 Ph CH 3 H H OH CHCH 3 B165 CH 3 O CH 3 H H OH CHCH 3 B166 CH 3 OC(O) CH 3 H H OH CHCH 3 B167 CH 3 CH 2 OC(O) CH 3 H H OH CHCH 3 B168 CH 2 =CHCH CH 3 H H OH CHCH 3 B169 HCCCH 2 CH 3 H H OH CHCH 3 B170 CF 3 CH 3 H H OH CHCH 3 B171 (CH 3 ) 2 NSO 2 CH 3 H H OH CHCHg B172 (CH 3 ) 2 N CH 3 H H OH CHCH 3 B173 PhO CH 3 H H OH CHCH 3 B174 PhS CH 3 H H OH CHCH 3 B176 PhSO 2 CH 3 H H OH CHCH 3 B177 CN CH 3 H H OH CHCH 3 B178 CH 3 H CH 3 H OH CHCH 3 B179 CHsCH H CH 3 H OH CHCH 3 B180 CHsCH 2 CH 2 H CH 3 H OH CHCHg B181 (CH 3 ) 2 CH H CH 3 H OH CHCH 3 B182 (CH 3 ) 3 C H CH 3 H OH CHCH 3 B183 CH 3 S H CH 3 H OH CHCH 3 B184 CH 3 SO H CH 3 H OH CHCH 3 B185 CH 3 SO 2 H CH 3 H OH CHCH 3 B186 Ph H CH 3 H OH CHCH 3 Radical Re R 7 R 8 R 9 R10 W B188 CH 3 OC(O) H CH 3 H OH CHCH 3 B189 CH 3 CH 2 OC(O) H CH 3 H OH CHCH 3 B190 CH 2 =CHCH 2 H CH 3 H OH CHCH 3 B191 HCCCH 2 H CH 3 H OH CHCH 3 B192 CF 3 H CH 3 H OH CHCH 3 B193 (CH 3 ) 2 NSO 2 H CH 3 H OH CHCH 3 B194 (CH 3 ) 2 N H CH 3 H OH CHCH 3 B195 PhO H CH 3 H OH CHCH 3 B196 PhS H CH 3 H OH CHCH 3 B197 PhSO H CH 3 H OH CHCH 3 B198 PhSO 2 H CH 3 H OH CHCH 3 B199 CN H CH 3 H OH CHCH 3 B200 CH 3 CH 3 CH 3 H OH CHCH 3 B201 CH 3 CH 2 CH 3 CH 3 H OH CHCH 3 B202 CH3CH 2 CH 2 CH 3 CH 3 H OH CHCH 3 B203 (CH 3 ) 2 CH CH 3 CH 3 H OH CHCH 3 B204 (CH 3 ) 3 C CH 3 CH 3 H OH CHCH 3 B205 CH 3 S CH 3 CH 3 H OH CHCH 3 B206 CH 3 SO CH 3 CH 3 H OH CHCH 3 B207 CH3SO2 CH 3 CH 3 H OH CHCH 3 B208 Ph CH 3 CH 3 H OH CHCH 3 B209 CH 3 O CH 3 CH 3 H OH CHCH3 B210 CH 3 OC(O) CH 3 CH 3 H OH CHCH 3 B211 CH 3 CH 2 OC(O) CH 3 CH 3 H OH CHCH 3 B212 CH 2 =CHCH 2 CH 3 CH 3 H OH CHCH 3 B213 HCCCH 2 CH 3 CH 3 H OH CHCH3 B214 CF 3 CH 3 CH 3 H OH CHCH 3 B215 (CH 3 ) 2 NSO 2 CH 3 CH 3 H OH CHCH 3 B216 (CH 3 ) 2 N CH 3 CH 3 H OH CHCH 3 B217 PhO CH 3 CH 3 H OH CHCH 3 B218 PhS CH 3 CH 3 H OH CHCH 3 B219 PhSO CH 3 CH 3 H OH CHCH 3 B220 PhSO 2 CH 3 CH 3 H OH CHCH 3 Radical Re R 7 R 8 R9 R10 W B221 CN CH 3 CH 3 H OH CHCH 3 B222 CH 3 CH 3 CH 3 CH 3 OH CHCH 3 B223 CH 3 CH;? CH 3 CH 3 CH 3 OH CHCH 3 B224 CH 3 CH 2 CH 2 CH 3 CH 3 CH 3 OH CHCH 3 B225 (CH 3 ) 2 CH CH 3 CH 3 CH 3 OH CHCH 3 B226 (CH 3 ) 3 C CH 3 CH 3 CH 3 OH CHCH 3 B227 CH 3 S CH 3 CH 3 CH 3 OH CHCH 3 B228 CH 3 SO CH 3 CH 3 CH 3 OH CHCH 3 B229 CH 3 SO 2 CH 3 CH 3 CH 3 OH CHCH 3 B230 Ph CH 3 CH 3 CH 3 OH CHCH 3 B231 CH 3 O CH 3 CH 3 CH 3 OH CHCH 3 B232 CH 3 OC(O) CH 3 CH 3 CH 3 OH CHCH 3 B233 CH 3 CH 2 OC(O) CH 3 CH 3 CH 3 OH CHCH 3 B234 CH 2 =CHCH 2 CH 3 CH 3 CH 3 OH CHCH 3 B235 HCCCH 2 CH 3 CH 3 CH 3 OH CHCH 3 B236 CF 3 CH 3 CH 3 CH 3 OH CHCH 3 B237 (CH 3 ) 2 NSO 2 CH 3 CH 3 CH 3 OH CHCH 3 B238 (CH 3 ) 2 N CH 3 CH 3 CH 3 OH CHCH 3 B239 PhO CH 3 CH 3 CH 3 OH CHCH 3 B240 PhS CH 3 CH 3 CH 3 OH CHCH 3 B241 PhSO CH 3 CH 3 CH 3 OH CHCH 3 B242 PhSO 2 CH 3 CH 3 CH 3 OH CHCH 3 B243 CN CH 3 CH 3 CH 3 » OH CHCH 3 B244 CH3CH2 CH 3 CH 2 H H OH CHCH 3 B245 CH 3 CH 2 CH 2 CH 3 CH 2 H H OH CHCH 3 B246 (CH 3 ) 2 CH CHsCH 2 H H OH CHCH 3 B247 (CH 3 ) 3 C CH 3 CH 2 H H OH CHCH 3 B248 CH 3 S CHsCH 2 H H OH CHCH 3 B249 CH 3 SO CH 3 CH 2 H H OH CHCH 3 B250 CH 3 SO 2 CH 3 CH 2 H H OH CHCH 3 B251 Ph CHsCH 2 H H OH CHCH 3 B252 CH 3 O CH 3 CH 2 H H OH CHCH3 B253 CH 3 OC(O) CH 3 CH 2 H H OH CHCH 3 Radical Re R 7 Rs R 9 R10 W B254 CH 3 CH 2 OC(O) CH 3 CH 2 H H OH CHCH3 B255 CH 2 =CHCH 2 CHsCH H H OH CHCH 3 B256 HCCCH 2 CH 3 CH 2 H H OH CHCH 3 B257 CF 3 CHsCH 2 H H OH CHCH 3 B258 (CH 3 ) 2 NSO 2 CHsCH 2 H H OH CHCH 3 B259 (CH 3 ) 2 N CHsCH 2 H H OH CHCH 3 B260 PhO CHsCH 2 H H OH CHCH 3 B261 PhS CHsCH 2 H H OH CHCH 3 B262 PhSO CHsCH 2 H H OH CHCH3 B263 PhSO 2 CHsCH 2 H H OH CHCH 3 B264 CN CH 3 CH 2 H H OH CHCH 3 B265 H H H H OH C=O B266 CH 3 H H H OH C=O B267 CH 3 CH 2 H H H OH C=O B268 CH 3 CH CH 2 H H H OH C=O B269 (CH 3 ) 2 CH H H H OH C=O B270 (CH 3 ) 3 C H H H OH C=O B271 CH 3 S H H H OH C=O B272 CH 3 SO H H H OH C=O B273 CH 3 SO 2 H H H OH C=O B274 Ph H H H OH C=O B275 CH 3 O H H H OH C=O B276 CH 3 OC(O) H H H OH C=O B277 CH 3 CH 2 OC(O) H H H OH C=O B278 CH 2 =CHCH 2 H H H OH C=O B279 HCCCH 2 H H H OH C=O B280 CF 3 H H H OH C=O B281 (CH 3 ) 2 NSO 2 H H H OH C=O B282 (CH 3 ) 2 N H H H OH C=O B283 PhO H H H OH C=O B284 PhS H H H OH C=O B285 PhSO H H H OH C=O B286 PhSO 2 H H H OH C=O Radical Re R 7 Rs R 9 R10 W B287 CN H H H OH C=O B288 CH 3 CH 3 H H OH C=O B289 CH 3 CH 2 CH 3 H H OH C=O B290 CH 3 CH 2 CH2 CH 3 H H OH C=O B291 (CH 3 ) 2 CH CH 3 H H OH C=O B292 (CH 3 ) 3 C CH 3 H H OH C=O B293 CH 3 S CH 3 H H OH C=O B294 CH 3 SO CH 3 H H OH C=O B295 CH 3 SO 2 CH 3 H H OH C=O B296 Ph CH 3 H H OH C=O B297 CH 3 O CH 3 H H OH C=O B298 CH 3 OC(O) CH 3 H H OH C=O B299 CH 3 CH 2 OC(O) CH 3 H H OH C=O B300 CH =CHCH 2 CH 3 H H OH C=O B301 HCCCH 2 CH 3 H H OH C=O B302 CF 3 CH 3 H H OH C=O B303 (CH 3 ) 2 NSO 2 CH 3 H H OH C=O B304 (CH 3 ) 2 N CH 3 H H OH C=O B305 PhO CH 3 H H OH C=O B306 PhS CH 3 H H OH C=O B307 PhSO CH 3 H H OH C=O B308 PhSO 2 CH 3 H H OH C=O B309 CN CH 3 H H OH C=O B310 CH 3 H CH 3 H OH C=O B311 CH 3 CH 2 H CH 3 H OH C=O B312 CH 3 CH 2 CH 2 H CH 3 H OH C=O B313 (CH 3 ) 2 CH H CH 3 H OH C=O B314 (CH 3 ) 3 C H CH 3 H OH C=O B315 CH 3 S H CH 3 H OH C=O B316 CH 3 SO H CH 3 H OH C=O B317 CH 3 SO 2 H CH 3 H OH C=O B318 Ph H CH 3 H OH C=O B319 CH 3 O H CH 3 H OH C=O Radical Re R 7 Rs R 9 R10 W B320 CH 3 OC(O) H CH 3 H OH C=O B321 CH 3 CH 2 OC(O) H CH 3 H OH C=O B322 CH 2 =CHCH 2 H CH 3 H OH C=O B323 HCCCH 2 H CH 3 H OH C=O B324 CF 3 H CH 3 H OH C=O B325 (CH 3 ) 2 NSO 2 H CH 3 H OH C=O B326 (CH 3 ) 2 N H CH 3 H OH C=O B327 PhO H CH 3 H OH C=O B328 PhS H CH 3 H OH C=O B329 PhSO H CH 3 H OH C=O B330 PhSO 2 H CH 3 H OH C=O B331 CN H CH 3 H OH C=O B332 CH 3 CH 3 CH 3 H OH C=O B333 CH3CH2 CH 3 CH 3 H OH C=O B334 CH 3 CH2CH2 CH 3 CH 3 H OH C=O B335 (CH 3 ) 2 CH CH 3 CH 3 H OH C=O B336 (CH 3 ) 3 C CH 3 CH 3 H OH C=O B337 CH 3 S CH 3 CH 3 H OH C=O B338 CH 3 SO CH 3 CH 3 H OH C=O B339 CH 3 SO 2 CH 3 CH 3 H OH C=O B340 Ph CH 3 CH 3 H OH C=O B341 CH 3 O CH 3 CH 3 H OH C=O B342 CH 3 OC(O) CH 3 CH 3 H OH C=O B343 CH 3 CH 2 OC(O) CH 3 CH 3 H OH C=O B344 CH 2 =CHCH CH 3 CH 3 H OH C=O B345 HCCCH 2 CH 3 CH 3 H OH C=O B346 CF 3 CH 3 CH 3 H OH C=O B347 (CH 3 ) 2 NSO 2 CH 3 CH 3 H OH C=O B348 (CH 3 ) 2 N CH 3 CH 3 H OH C=O B349 PhO CH 3 CH 3 H OH C=O B350 PhS CH 3 CH 3 H OH C=O B351 PhSO CH 3 CH 3 H OH C=O B352 PhSO 2 CH 3 CH 3 H OH C=O Radical Re R 7 R 8 R9 R10 W B353 CN CH 3 CH 3 H OH C=O B354 CH 3 CH 3 CH 3 CH 3 OH C=O B355 CH3CH2 CH 3 CH 3 CH 3 OH C=O B356 CH 3 CH 2 CH2 CH 3 CH 3 CH 3 OH C=O B357 (CH 3 ) 2 CH CH 3 CH 3 CH 3 OH C=O B358 (CH 3 ) 3 C CH 3 CH 3 CH 3 OH C=O B359 CH 3 S CH 3 CH 3 CH 3 OH C=O B360 CH3SO CH 3 CH 3 CH 3 OH C=O B361 CH 3 SO 2 CH 3 CH 3 CH 3 OH C=O B362 Ph CH 3 CH 3 CH 3 OH C=O B363 CH 3 O CH 3 CH 3 CH 3 OH C=O B364 CH 3 OC(O) CH 3 CH 3 CH 3 OH C=O B365 CH 3 CH 2 OC(O) CH 3 CH 3 CH 3 OH C=O B367 HCCCH 2 CH 3 CH 3 CH 3 OH C=O B368 CF 3 CH 3 CH 3 CH 3 OH C=O B369 (CH 3 ) 2 NSO 2 CH 3 CH 3 CH 3 OH C=O B370 (CH 3 ) 2 N CH 3 CH 3 CH 3 OH C=O B371 PhO CH 3 CH 3 CH 3 OH C=O B372 PhS CH 3 CH 3 CH 3 OH C=O B373 PhSO CH 3 CH 3 CH 3 OH C=O B374 PhSO 2 CH 3 CH 3 CH 3 OH C=O B375 CN CH 3 CH 3 CH 3 OH C=O B376 CH 3 CH 2 CH3CH2 H H OH C=O B377 CH 3 CH 2 CH 2 CH3CH2 H H OH C=O B378 (CH 3 ) 2 CH CH 3 CH 2 H H OH C=O B379 (CH 3 ) 3 C CH 3 CH 2 H H OH C=O B380 CH 3 S CH 3 CH 2 H H OH C=O B381 CH3SO CH 3 CH 2 H H OH C=O B382 CH 3 SO 2 CH 3 CH 2 H H OH C=O B384 CH3O CH3CH2 H H OH C=O B385 CH 3 OC(O) CH 3 CH2 H H OH C=O Radical Re R 7 Rs R9 R10 W B386 CH 3 CH 2 OC(O) CH 3 CH2 H H OH C=O B387 CH 2 = CHCH 2 CH 3 CH 2 H H OH C=O B388 HCCCH 2 CH 3 CH 2 H H OH C=O B389 CF 3 CH 3 CH 2 H H OH C=O B390 (CH 3 ) 2 NSO 2 CH 3 CH 2 H H OH C=O B391 (CH 3 ) 2 N CH 3 CH 2 H H OH C=O B392 PhO CHsCH 2 H H OH C=O B393 PhS CH 3 CH 2 H H OH C=O B394 PhSO CH 3 CH;? H H OH C=O B395 PhSO 2 CH 3 CH 2 H H OH C=O B396 CN CH 3 CH 2 H H OH C=O B400 CH 3 CH CH 2 H H H OH N-CH 3 B401 (CH 3 ) 2 CH H H H OH N-CH 3 B402 (CH 3 ) 3 C H H H OH N-CH 3 B403 CH 3 S H H H OH N-CH 3 B405 CH 3 SO 2 H H H OH N-CH 3 B406 Ph H H H OH N-CH 3 B407 CH 3 O H H H OH N-CH 3 B408 CH 3 OC(O) H H H OH N-CH 3 B409 CH 3 CH 2 OC(O) H H H OH N-CH 3 B410 CH 2 =CHCH 2 H H H OH N-CH 3 B411 HCCCH 2 H H H OH N-CH 3 B412 CF 3 H H H OH N-CH 3 B413 (CH 3 ) 2 NSO 2 H H H OH N-CH 3 B414 (CH 3 ) 2 N H H H OH N-CH 3 B415 PhO H H H OH N-CH 3 B417 PhSO H H H OH N-CH 3 B418 PhSO 2 H H H OH N-CH 3 Radical Re R 7 Rs R 9 R10 W B419 CN H H H OH N-CH 3 B420 CH 3 CH 3 H H OH N-CH 3 B421 CH 3 CH 2 CH 3 H H OH N-CH 3 B422 CH 3 CH 2 CH 2 CH 3 H H OH N-CH 3 B423 (CH 3 ) 2 CH CH 3 H H OH N-CH 3 B424 (CH 3 ) 3 C CH 3 H H OH N-CH 3 B425 CH 3 S CH 3 H H OH N-CH 3 B426 CH 3 SO CH 3 H H OH N-CH 3 B427 CH 3 SO 2 CH 3 H H OH N-CH 3 B428 Ph CH 3 H H OH N-CH 3 B429 CH 3 O CH 3 H H OH N-CH 3 B430 CH 3 OC(O) CH 3 H H OH N-CH 3 B431 CH 3 CH 2 OC(O) CH 3 H H OH N-CH 3 B432 CH 2 =CHCH 2 CH 3 H H OH N-CH 3 B433 HCCCH 2 CH 3 H H OH N-CH 3 B434 CF 3 CH 3 H H OH N-CH 3 B435 (CH 3 ) 2 NSO 2 CH 3 H H OH N-CH 3 B436 (CH 3 ) 2 N CH 3 H H OH N-CH 3 B437 PhO CH 3 H H OH N-CH 3 B438 PhS CH 3 H H OH N-CH 3 B439 PhSO CH 3 H H OH N-CH 3 B440 PhSO 2 CH 3 H H OH N-CH 3 B441 CN CH 3 H H OH N-CH 3 B442 CH 3 H CH 3 H OH N-CH 3 B443 CHsCH 2 H CH 3 H OH N-CH 3 B444 CH 3 CH 2 CH 2 H CH 3 H OH N-CH 3 B445 (CH 3 ) 2 CH H CH 3 H OH N-CH 3 B446 (CH 3 ) 3 C H CH 3 H OH N-CH 3 B447 CH 3 S H CH 3 H OH N-CH 3 B448 CH 3 SO H CH 3 H OH N-CH 3 B449 CH 3 SO 2 H CH 3 H OH N-CH 3 B450 Ph H CH 3 H OH N-CH 3 B451 CH 3 O H CH 3 H OH N-CH 3 Radical Re R 7 Rs R 9 R10 W B452 CH 3 OC(O) H CH 3 H OH N-CH 3 B453 CH 3 CH 2 OC(O) H CH 3 H OH N-CH 3 B454 CH 2 =CHCH 2 H CH 3 H OH N-CH 3 B455 HCCCH 2 H CH 3 H OH N-CH 3 B456 CF 3 H CH 3 H OH N-CH 3 B457 (CH 3 ) 2 NSO 2 H CH 3 H OH N-CH 3 B458 (CH 3 ) 2 N H CH 3 H OH N-CH 3 B459 PhO H CH 3 H OH N-CH 3 B460 PhS H CH 3 H OH N-CH 3 B461 PhSO H CH 3 H OH N-CH 3 B462 PhSO 2 H CH 3 H OH N-CH 3 B463 CN H CH 3 H OH N-CH 3 B464 CH 3 CH 3 CH 3 H OH N-CH 3 B465 CH 3 CH 2 CH 3 CH 3 H OH N-CH 3 B466 CHsCH CH 2 CH 3 CH 3 H OH N-CH 3 B467 (CH 3 ) 2 CH CH 3 CH 3 H OH N-CH 3 B468 (CH 3 ) 3 C CH 3 CH 3 H OH N-CH 3 B469 CH 3 S CH 3 CH 3 H OH N-CH 3 B470 CHgSO CH 3 CH 3 H OH N-CH 3 B471 CH 3 SO 2 CH 3 CH 3 H OH N-CH 3 B472 Ph CH 3 CH 3 H OH N-CH 3 B473 CH 3 O CH 3 CH 3 H OH N-CH 3 B474 CH 3 OC(O) CH 3 CH 3 H OH N-CH 3 B475 CH 3 CH 2 OC(O) CH 3 CH 3 H OH N-CH 3 B476 CH 2 =CHCH CH 3 CH 3 H OH N-CH 3 B477 HCCCH 2 CH 3 CH 3 H OH N-CH 3 B478 CF 3 CH 3 CH 3 H OH N-CH 3 B479 (CH 3 ) 2 NSO 2 CH 3 CH 3 H OH N-CH 3 B480 (CH 3 ) 2 N CH 3 CH 3 H OH N-CH 3 B481 PhO CH 3 CH 3 H OH N-CH 3 B482 PhS CH 3 CH 3 H OH N-CH 3 B483 PhSO CH 3 CH 3 H OH N-CH 3 B484 PhSO 2 CH 3 CH 3 H OH N-CH 3 Radical Re R 7 Rs R 9 R10 W B485 CN CH 3 CH 3 H OH N-CH 3 B486 CH 3 CH 3 CH 3 CH 3 OH N-CH 3 B487 CH 3 CH 2 CH 3 CH 3 CH 3 OH N-CHg B488 CH 3 CH 2 CH 2 CH 3 CH 3 CH 3 OH N-CH 3 B489 (CH 3 ) 2 CH CH 3 CH 3 CH 3 OH N-CH 3 B490 (CH 3 ) 3 C CH 3 CH 3 CH 3 OH N-CH 3 B491 CH 3 S CH 3 CH 3 CH 3 OH N-CH 3 B492 CH 3 SO CH 3 CH 3 CH 3 OH N-CH 3 B493 CH 3 SO 2 CH 3 CH 3 CH 3 OH N-CH 3 B494 Ph CH 3 CH 3 CH 3 OH N-CH 3 B495 CH 3 O CH 3 CH 3 CH 3 OH N-CH 3 B496 CH 3 OC(O) CH 3 CH 3 CH 3 OH N-CH 3 B497 CH 3 CH 2 OC(O) CH 3 CH 3 CH 3 OH N-CH 3 B498 CH 2 =CHCH 2 CH 3 CH 3 CH 3 OH N-CH 3 B499 HCCCH 2 CH 3 CH 3 CHg OH N-CH 3 B500 CF 3 CH 3 CH 3 CH 3 OH N-CH 3 B501 (CH 3 ) 2 NSO 2 CH 3 CH 3 CH 3 OH N-CH 3 B502 (CH 3 ) 2 N CH 3 CH 3 CH 3 OH N-CH 3 B503 PhO CH 3 CH 3 CH 3 OH N-CH 3 B504 PhS CH 3 CH 3 CH 3 OH N-CH 3 B505 PhSO CH 3 CH 3 CH 3 OH N-CH 3 B506 PhSO 2 CH 3 CH 3 CH 3 OH N-CH 3 B507 CN CH 3 CH 3 CH 3 OH N-CH 3 B508 CHsCH 2 CH 3 CH 2 H H OH N-CH 3 B509 CH 3 CH 2 CH 2 CH 3 CH2 H H OH N-CH 3 B510 (CH 3 ) 2 CH CH3CH2 H H OH N-CH 3 B511 (CH 3 ) 3 C CH 3 CH2 H H OH N-CH 3 B512 CH 3 S CH 3 CH 2 H H OH N-CH 3 B513 CH 3 SO CH 3 CH 2 H H OH N-CH 3 B514 CH 3 SO 2 CH 3 CH 2 H H OH N-CH 3 B515 Ph CHsCH 2 H H OH N-CH 3 B516 CH 3 O CHsCH 2 H H OH N-CH 3 B517 CH 3 OC(O) CH 3 CH 2 H H OH N-CH 3 Radical Re R 7 Rs R 9 R10 W B518 CH 3 CH 2 OC(O) CH 3 CH 2 H H OH N-CH 3 B519 CH 2 =CHCH 2 CH 3 CH 2 H H OH N-CH 3 B520 HCCCH 2 CH 3 CH 2 H H OH N-CH 3 B521 CF 3 CH 3 CH 2 H H OH N-CH 3 B522 (CH 3 ) 2 NSO 2 CH 3 CH 2 H H OH N-CH 3 B523 (CH 3 ) 2 N CH 3 CH 2 H H OH N-CH 3 B524 PhO CHsCH 2 H H OH N-CH 3 B525 PhS CH3CH2 H H OH N-CH 3 B526 PhSO CH3CH2 H H OH N-CH 3 B527 PhSO 2 CH3CH2 H H OH N-CH 3 B528 CN CH3CH2 H H OH N-CH 3 B529 H H H H OH O B530 CH 3 H H H OH O B532 CH 3 CH 2 CH 2 H H H OH O B533 (CH 3 ) 2 CH H H H OH O B534 (CH 3 ) 3 C H H H OH O B535 CH 3 S H H H OH O B537 CH 3 SO 2 H H H OH O B538 Ph H H H OH O B539 CH 3 O H H H OH O B540 CH 3 OC(O) H H H OH O B541 CH 3 CH 2 OC(O) H H H OH O B542 CH 2 =CHCH 2 H H H OH O B543 HCCCH 2 H H H OH O B544 CF 3 H H H OH O B545 (CH 3 ) 2 NSO 2 H H H OH O B546 (CH 3 ) 2 N H H H OH O B547 PhO H H H OH O B548 PhS H H H OH O B549 PhSO H H H OH O B550 PhSO 2 H H H OH O Radical Re R Rs R9 R10 W B551 CN H H H OH O B552 CH 3 CH 3 H H OH O B553 CH 3 CH 2 CH 3 H H OH O B554 CH 3 CH 2 CH 2 CH 3 H H OH O B555 (CH 3 ) 2 CH CH 3 H H OH O B556 (CH 3 ) 3 C CH 3 H H OH O B557 CH 3 S CH 3 H H OH O B558 CH 3 SO CH 3 H H OH O B559 CH 3 SO 2 CH 3 H H OH O B560 Ph CH 3 H H OH O B561 CH 3 O CH 3 H H OH O B562 CHgOC(O) CH 3 H H OH O B563 CH 3 CH 2 OC(O) CH 3 H H OH O B564 CH 2 =CHCH 2 CH 3 H H OH O B565 HCCCH 2 CH 3 H H OH O B566 CF 3 CH 3 H H OH O B567 (CH 3 ) 2 NSO 2 CH 3 H H OH O B568 (CH 3 ) 2 N CH 3 H H OH O B569 PhO CH 3 H H OH O B570 PhS CH 3 H H OH o B571 PhSO CH 3 H H OH O B572 PhSO 2 CH 3 H H OH O B573 CN CH 3 H H OH O B574 CH 3 H CH 3 H OH O B575 CH 3 CH 2 H CH 3 H OH O B576 CH 3 CH 2 CH 2 H CH 3 H OH O B577 (CH 3 ) 2 CH H CH 3 H OH O B578 (CH 3 ) 3 C H CH 3 H OH O B579 CH 3 S H CH 3 H OH O B580 CH 3 SO H CH 3 H OH O B581 CH 3 SO 2 H CH 3 H OH O B582 Ph H CH 3 H OH O B583 CH 3 O H CH 3 H OH O Radical Re R 7 R 8 R 9 R10 W B584 CH 3 OC(O) H CH 3 H OH O B585 CH 3 CH 2 OC(O) H CH 3 H OH O B586 CH 2 =CHCH 2 H CH 3 H OH O B587 HCCCH 2 H CH 3 H OH O B588 CF 3 H CH 3 H OH O B589 (CH 3 ) 2 NSO 2 H CH 3 H OH O B590 (CH 3 ) 2 N H CH 3 H OH O B591 PhO H CH 3 H OH O B592 PhS H CH 3 H OH O B593 PhSO H CH 3 H OH O B594 PhSO 2 H CH 3 H OH O B595 CN H CH 3 H OH O B596 CH 3 CH 3 CH 3 H OH O B597 CH 3 CH 2 CH 3 CH 3 H OH O B598 CH 3 CH 2 CH 2 CH 3 CH 3 H OH O B599 (CH 3 ) 2 CH CH 3 CH 3 H OH O B600 (CH 3 ) 3 C CH 3 CH 3 H OH O B601 CH 3 S CH 3 CH 3 H OH O B602 CH 3 SO CH 3 CH 3 H OH O B603 CH 3 SO 2 CH 3 CH 3 H OH O B604 Ph CH 3 CH 3 H OH O B605 CH 3 O CH 3 CH 3 H OH O B606 CH 3 OC(O) CH 3 CH 3 H OH O B607 CH 3 CH 2 OC(O) CH 3 CHg H OH O B608 CH 2 =CHCH 2 CH 3 CH 3 H OH O B609 HCCCH 2 CH 3 CH 3 H OH O B610 CF 3 CH 3 CH 3 H OH O B611 (CH 3 ) 2 NSO 2 CH 3 CH 3 H OH O B612 (CH 3 ) 2 N CH 3 CH 3 H OH O B613 PhO CH 3 CH 3 H OH O B614 PhS CH 3 CH 3 H OH O B615 PhSO CH 3 CH 3 H OH O B616 PhSO 2 CH 3 CH 3 H OH O Radical Re R 7 Rs R 9 R10 W B619 CH 3 CH 2 CH 3 CH3 CH 3 OH O B620 CH 3 CH 2 CH 2 CH 3 CH3 CH 3 OH O B621 (CH 3 ) 2 CH CH 3 CH3 CH 3 OH O B622 (CH 3 ) 3 C CH 3 CH3 CH 3 OH O B624 CH 3 SO CH 3 CH3 CH 3 OH O B625 CH 3 SO 2 CH 3 CH3 CH 3 OH O B627 CH 3 O CH 3 CH 3 CH 3 OH O B628 CH 3 OC(O) CH 3 CH 3 CH 3 OH O B629 CH 3 CH 2 OC(O) CH 3 CH 3 CH 3 OH O B630 CH 2 =CHCH 2 CH 3 CH 3 CH 3 OH O B631 HCCCH 2 CH 3 CH 3 CH 3 OH O B632 CF 3 CH 3 CH 3 CH 3 OH O B633 (CH 3 ) 2 NSO 2 CH 3 CH 3 CH 3 OH O B634 (CH 3 ) 2 N CH 3 CH 3 CH 3 OH O B635 PhO CH 3 CH 3 CH 3 OH O B636 PhS CH 3 CH 3 CH 3 OH O B637 PhSO CH 3 CH 3 CH 3 OH O B638 PhSO 2 CH 3 CH 3 CH 3 OH O B639 CN CH 3 CH 3 CH 3 OH O B640 CH 3 CH 2 CH 3 CH 2 H H OH O B641 CH 3 CH 2 CH 2 CH 3 CH 2 H H OH O B642 (CH 3 ) 2 CH CH 3 CH 2 H H OH O B643 (CH 3 ) 3 C CH 3 CH 2 H H OH O B644 CH 3 S CHsCH H H OH O B645 CH 3 SO CH 3 CH 2 H H OH O B646 CH 3 SO 2 CHsCH 2 H H OH O B648 CH 3 O CHsCH 2 H H OH O B649 CH 3 OC(O) CH 3 CH 2 H H OH O Radical Re R 7 Rs R9 R.o W B650 CH 3 CH 2 OC(O) CH 3 CH 2 H H OH O B651 CH 2 =CHCH 2 CH 3 CH 2 H H OH O B652 HCCCH 2 CH3CH2 H H OH O B653 CF 3 CH 3 CH 2 H H OH O B654 (CH 3 ) 2 NSO 2 CH 3 CH H H OH O B655 (CH 3 ) 2 N CH 3 CH 2 H H OH O B661 H H H H OH S B662 CH 3 H H H OH S B663 CH 3 CH 2 H H H OH S B664 CH 3 CH 2 CH 2 H H H OH S B665 (CH 3 ) 2 CH H H H OH S B666 (CH 3 ) 3 C H H H OH S B667 CH 3 S H H H OH S B668 CH 3 SO H H H OH S B669 CH 3 SO 2 H H H OH s B670 Ph H H H OH s B671 CH 3 O H H H OH s B672 CH 3 OC(O) H H H OH s B673 CH 3 CH 2 OC(O) H H H OH s B674 CH 2 =CHCH 2 H H H OH s B675 HCCCH 2 H H H OH s B676 CF 3 H H H OH s B677 (CH 3 ) 2 NSO 2 H H H OH s B678 (CH 3 ) 2 N H H H OH s B679 PhO H H H OH s B680 PhS H H H OH s B681 PhSO H H H OH s B682 PhSO 2 H H H OH s Radical Re R 7 Rs R 9 R10 W B683 CN H H H OH S B684 CH 3 CH 3 H H OH S B686 CH 3 CH2CH2 CH 3 H H OH S B687 (CH 3 ) 2 CH CH 3 H H OH S B688 (CH 3 ) 3 C CH 3 H H OH S B689 CH 3 S CH 3 H H OH s B690 CH 3 SO CH 3 H H OH s B692 Ph CH 3 H H OH s B693 CH 3 O CH 3 H H OH s B694 CH 3 OC(O) CH 3 H H OH s B695 CH 3 CH 2 OC(O) CH 3 H H OH s B697 HCCCH≥ CH 3 H H OH s B698 CF 3 CH 3 H H OH s B699 (CH 3 ) 2 NSO 2 CH 3 H H OH s B700 (CH 3 ) 2 N CH 3 H H OH s B701 PhO CH 3 H H OH s B702 PhS CH 3 H H OH s B703 PhSO CH 3 H H OH s B704 PhSO 2 CH 3 H H OH s B705 CN CH 3 H H OH s B706 CH 3 H CH 3 H OH s B707 CH 3 CH 2 H CH 3 H OH s B708 CH 3 CH 2 CH2 H CH 3 H OH s B709 (CH 3 ) 2 CH H CH 3 H OH s B710 (CH 3 ) 3 C H CH 3 H OH s B711 CH 3 S H CH 3 H OH s B712 CH 3 SO H CH 3 H OH s B713 CH 3 SO 2 H CH 3 H OH s B714 Ph H CH 3 H OH s B715 CH 3 O H CH 3 H OH s Radical Re R 7 Rs R 9 R10 W B716 CH 3 OC(O) H CH 3 H OH S B717 CH 3 CH 2 OC(O) H CH 3 H OH S B718 CH 2 =CHCH 2 H CH 3 H OH S B719 HCCCH 2 H CH 3 H OH S B721 (CH 3 ) 2 NSO 2 H CH 3 H OH S B723 PhO H CH 3 H OH S B724 PhS H CH 3 H OH S B725 PhSO H CH 3 H OH S B726 PhSO 2 H CH 3 H OH S B729 CH 3 CH 2 CH 3 CH 3 H OH S B730 CH 3 CH 2 CH 2 CH 3 CHg H OH S B731 (CH 3 ) 2 CH CH 3 CH3 H OH S B732 (CH 3 ) 3 C CH 3 CH3 H OH S B737 CH 3 O CH 3 CH 3 H OH s B738 CH 3 OC(O) CH 3 CHg H OH s B739 CH 3 CH 2 OC(O) CH 3 CH 3 H OH s B740 CH 2 =CHCH 2 CH 3 CH3 H OH s B741 HCCCH 2 CH 3 CH3 H OH s B742 CF 3 CH 3 CH 3 H OH s B743 (CH 3 ) 2 NSO 2 CH 3 CH 3 H OH s B744 (CH 3 ) 2 N CH 3 CH 3 H OH s B745 PhO CH 3 CH 3 H OH s B746 PhS CH 3 CH 3 H OH s B747 PhSO CH 3 CH 3 H OH s B748 PhSO 2 CH 3 CH 3 H OH s Radical Re R 7 Rs R 9 R10 W B751 CH 3 CH 2 CH 3 CH3 CH 3 OH S B752 CHgCH 2 CH 2 CH 3 CH3 CH 3 OH S B753 (CH 3 ) 2 CH CH 3 CH3 CH 3 OH S B754 (CH 3 ) 3 C CH 3 CH 3 CH 3 OH s B756 CH 3 SO CH 3 CH3 CH 3 OH s B757 CH 3 SO 2 CH 3 CHg CH 3 OH s B760 CH 3 OC(O) CH 3 CH3 CH3 OH s B761 CH 3 CH 2 OC(O) CH 3 CHg CHg OH s B762 CH 2 =CHCH 2 CH 3 CHg CHg OH s B763 HCCCH 2 CHg CHg CHg OH s B765 (CH 3 ) 2 NSO 2 CH 3 CH3 CHg OH s B766 (CH 3 ) 2 N CHg CHg CHg OH s B770 PhSO 2 CHg CH3 CH3 OH s B772 CHgCH 2 CH3CH2 H H OH s B773 CHgCH 2 CH 2 CH3CH2 H H OH s B774 (CHg) 2 CH CH3CH2 H H OH s B775 (CH 3 ) 3 C CH3CH2 H H OH s B778 CH 3 SO 2 CH3CH2 H H OH s B781 CH 3 OC(O) CH3CH2 H H OH s Radical Re R 7 Rs R 9 R10 W B782 CH 3 CH 2 OC(O) CHsCH 2 H H OH S B783 CH 2 = CHCH 2 CHsCH 2 H H OH S B784 HCCCH 2 CH 3 CH 2 H H OH S B785 CF 3 CHsCH 2 H H OH S B786 (CH 3 ) 2 NSO 2 CHsCH 2 H H OH S B787 (CH 3 ) 2 N CHsCH 2 H H OH S B788 PhO CHsCH 2 H H OH S B789 PhS CH 3 CH;; H H OH S B790 PhSO CHsCH 2 H H OH S B793 H H H H OH SO 2 B794 CH 3 H H H OH SO 2 B795 CHgCH 2 H H H OH SO 2 B796 CH CH 2 CH2 H H H OH SO 2 B799 CH 3 S H H H OH SO 2 B802 Ph H H H OH SO 2 B803 CH 3 O H H H OH SO 2 B804 CH 3 OC(O) H H H OH SO 2 B805 CH 3 CH 2 OC(O) H H H OH SO 2 B806 CH 2 =CHCH 2 H H H OH SO 2 B807 HCCCH 2 H H H OH SO 2 B808 CF 3 H H H OH SO 2 B809 (CH 3 ) 2 NSO 2 H H H OH SO 2 B810 (CH 3 ) 2 N H H H OH SO 2 B811 PhO H H H OH SO 2 B812 PhS H H H OH SO 2 B813 PhSO H H H OH SO 2 B814 PhSO 2 H H H OH SO 2 Radical Re R 7 R 8 R 9 R10 W B815 CN H H H OH SO 2 B816 CH 3 CH 3 H H OH SO 2 B817 CH 3 CH 2 CH 3 H H OH SO 2 B818 CH 3 CH 2 CH 2 CH 3 H H OH SO 2 B819 (CH 3 ) 2 CH CH 3 H H OH SO 2 B820 (CH 3 ) 3 C CH 3 H H OH SO 2 B821 CH 3 S CH 3 H H OH SO 2 B822 CH 3 SO CH 3 H H OH SO 2 B823 CH 3 SO 2 CH 3 H H OH SO 2 B824 Ph CH 3 H H OH SO 2 B825 CH 3 O CH 3 H H OH SO 2 B826 CH 3 OC(O) CH 3 H H OH SO 2 B827 CH 3 CH 2 OC(O) CH 3 H H OH SO 2 B828 CH 2 =CHCH 2 CH 3 H H OH SO 2 B829 HCCCH 2 CH 3 H H OH SO 2 B830 CF 3 CH 3 H H OH SO 2 B831 (CH 3 ) 2 NSO 2 CH 3 H H OH SO 2 B832 (CH 3 ) 2 N CH 3 H H OH SO 2 B833 PhO CH 3 H H OH SO 2 B834 PhS CH 3 H H OH SO 2 B835 PhSO CH 3 H H OH SO 2 B836 PhSO 2 CH 3 H H OH SO 2 B837 CN CH 3 H H OH SO 2 B838 CH 3 H CH 3 H OH SO 2 B839 CHsCH 2 H CH 3 H OH SO 2 B840 CH 3 CH 2 CH 2 H CH 3 H OH SO 2 B841 (CH 3 ) 2 CH H CH 3 H OH SO 2 B842 (CH 3 ) 3 C H CH 3 H OH SO 2 B843 CH 3 S H CH 3 H OH SO 2 B844 CH 3 SO H CH 3 H OH SO 2 B845 CH 3 SO 2 H CH 3 H OH SO 2 B846 Ph H CH 3 H OH SO 2 B847 CH 3 O H CH 3 H OH SO 2 Radical Re R 7 RB R 9 R10 W B848 CH 3 OC(O) H CH3 H OH SO 2 B849 CH 3 CH 2 OC(O) H CHg H OH SO 2 B850 CH 2 =CHCH 2 H CHg H OH SO 2 B851 HCCCH 2 H CHg H OH SO 2 B853 (CH 3 ) 2 NSO 2 H CHg H OH SO 2 B854 (CH 3 ) 2 N H CHg H OH SO 2 B860 CH 3 CH 3 CH 3 H OH SO 2 B861 CH 3 CH2 CH 3 CHg H OH SO 2 B862 CH 3 CH 2 CH 2 CH 3 CH 3 H OH SO 2 B863 (CHg) 2 CH CH 3 CH 3 H OH SO 2 B864 (CH 3 ) 3 C CH 3 CHg H OH SO 2 B866 CHgSO CH 3 CH 3 H OH SO 2 B867 CH 3 SO 2 CHg CH3 H OH SO 2 B870 CH 3 OC(O) CHg CHg H OH SO 2 B871 CH 3 CH 2 OC(O) CHg CHg H OH SO 2 B873 HCCCH 2 CHg CHg H OH SO 2 B875 (CH 3 ) 2 NSO 2 CHg CHg H OH SO 2 B876 (CH 3 ) 2 N CHg CH 3 H OH SO 2 B880 PhSO 2 CH3 CH3 H OH SO 2 ladical Re R 7 R 8 R 9 R10 W B881 CN CH 3 CH 3 H OH SO 2 B882 CH 3 CH 3 CH 3 CH 3 OH SO 2 B883 CH3CH2 CHg CH 3 CH 3 OH SO 2 B884 CH3CH2CH2 CHg CH 3 CH 3 OH SO 2 B885 (CH 3 ) 2 CH CHg CH 3 CH 3 OH SO 2 B886 (CH 3 ) 3 C CHg CH 3 CH 3 OH SO 2 B887 CH 3 S CHg CH 3 CHg OH SO 2 B888 CH 3 SO CHg CH 3 CHg OH SO 2 B889 CH 3 SO 2 CH3 CHg CHg OH SO 2 B891 CH 3 O CH3 CH3 CHg OH SO 2 B892 CH 3 OC(O) CHg CH3 CH 3 OH SO 2 B893 CH 3 CH 2 OC(O) CHg CH3 CH 3 OH SO 2 B895 HCCCH 2 CH3 CH 3 CH3 OH SO 2 B896 CFg CH3 CH 3 CH3 OH SO 2 B897 (CH 3 ) 2 NSO 2 CHg CH 3 CH3 OH SO 2 B898 (CHg) 2 N CHg CH 3 CH3 OH SO 2 B899 PhO CHg CHg CH3 OH SO 2 B900 PhS CHg CHg CH3 OH SO 2 B901 PhSO CH 3 CHg CH3 OH SO 2 B902 PhSO 2 CH3 CHg CH3 OH SO 2 B904 CHgCH 2 CHgCH 2 H H OH SO 2 B905 CHgCH 2 CH 2 CHgCH 2 H H OH SO 2 B906 (CHg) 2 CH CHgCH 2 H H OH SO 2 B907 (CHg) 3 C CHgCH 2 H H OH SO 2 B908 CH 3 S CHgCH 2 H H OH SO 2 B909 CH 3 SO CHsCH 2 H H OH SO 2 B910 CH 3 SO 2 CH3CH2 H H OH SO 2 B912 CH 3 O CH3CH2 H H OH SO 2 B913 CH 3 OC(O) CH3CH2 H H OH SO 2 Radical Re R 7 Rs R 9 R10 W B914 CH 3 CH 2 OC(O) CH 3 CH 2 H H OH SO 2 B915 CH 2 =CHCH 2 CH 3 CH 2 H H OH SO 2 B916 HCCCH 2 CHsCH 2 H H OH SO 2 B917 CF 3 CHsCH 2 H H OH SO 2 B918 (CH 3 ) 2 NSO 2 CHsCH 2 H H OH SO 2 B919 (CH 3 ) 2 N CH 3 CH 2 H H OH SO 2 B920 PhO CHsCH 2 H H OH SO 2 B921 PhS CH 3 CH 2 H H OH SO 2 B922 PhSO CH3CH2 H H OH SO 2 B923 PhSO 2 CH3CH2 H H OH SO 2 B925 H H H H OH CHC(O)OCH 2 CH 3 B926 CH 3 H H H OH CHC(O)OCH 2 CH 3 B927 CHsCH 2 H H H OH CHC(O)OCH 2 CH 3 B928 CHgCH 2 CH 2 H H H OH CHC(O)OCH 2 CH 3 B929 (CHg) 2 CH H H H OH CHC(O)OCH 2 CH 3 B930 (CHg)gC H H H OH CHC(O)OCH 2 CH 3 B931 CHgS H H H OH CHC(O)OCH 2 CH 3 B932 CHgSO H H H OH CHC(O)OCH 2 CH 3 B933 CHgSO 2 H H H OH CHC(O)OCH 2 CH 3 B934 Ph H H H OH CHC(O)OCH 2 CH 3 B935 CHgO H H H OH CHC(O)OCH 2 CH 3 B936 CH 3 OC(O) H H H OH CHC(O)OCH 2 CH 3 B937 CH 3 CH 2 OC(O) H H H OH CHC(O)OCH 2 CH 3 B938 CH 2 =CHCH 2 H H H OH CHC(O)OCH 2 CH 3 B939 HCCCH 2 H H H OH CHC(O)OCH 2 CH 3 B940 CF 3 H H H OH CHC(O)OCH 2 CH 3 B941 (CH 3 ) 2 NSO 2 H H H OH CHC(O)OCH 2 CH 3 B942 (CH 3 ) 2 N H H H OH CHC(O)OCH 2 CH 3 B943 PhO H H H OH CHC(O)OCH 2 CH 3 B944 PhS H H H OH CHC(O)OCH 2 CH 3 B945 PhSO H H H OH CHC(O)OCH 2 CH 3 B946 PhSO 2 H H H OH CHC(O)OCH 2 CH 3 Radical Re R 7 Rs R 9 R10 W B947 CN H H H OH CHC(O )OCH 2 CH 3 B948 CH 3 CH 3 H H OH CHC(O; )OCH 2 CH 3 B949 CHgCH 2 CH 3 H H OH CHC(O )OCH 2 CH 3 B950 CHgCH 2 CH 2 CH 3 H H OH CHC(O )OCH 2 CH 3 B951 (CHg) 2 CH CH 3 H H OH CHC(O )OCH 2 CH 3 B952 (CH 3 ) 3 C CH 3 H H OH CHC(O )OCH 2 CH 3 B953 CH 3 S CH 3 H H OH CHC(O )OCH 2 CH 3 B954 CH 3 SO CH 3 H H OH CHC(O )OCH 2 CH 3 B955 CH 3 SO 2 CH 3 H H OH CHC(O )OCH 2 CH 3 B956 Ph CH 3 H H OH CHC(O )OCH 2 CH 3 B957 CH 3 O CH 3 H H OH CHC(O )OCH 2 CH 3 B958 CH 3 OC(O) CH 3 H H OH CHC(O )OCH 2 CH 3 B959 CH 3 CH 2 OC(O) CH 3 H H OH CHC(O )OCH 2 CH 3 B960 CH 2 =CHCH 2 CH 3 H H OH CHC(O )OCH 2 CH 3 B961 HCCCH 2 CH 3 H H OH CHC(O )OCH 2 CH 3 B962 CF 3 CH 3 H H OH CHC(O )OCH 2 CH 3 B963 (CH 3 ) 2 NSO 2 CH 3 H H OH CHC(O )OCH 2 CH 3 B964 (CH 3 ) 2 N CH 3 H H OH CHC(O )OCH 2 CH 3 B965 PhO CH 3 H H OH CHC(O )OCH 2 CH 3 B966 PhS CH 3 H H OH CHC(O )OCH 2 CH 3 B967 PhSO CH 3 H H OH CHC(O )OCH 2 CH 3 B968 PhSO 2 CH 3 H H OH CHC(O )OCH 2 CH 3 B969 CN CH 3 H H OH CHC(O )OCH 2 CH 3 B970 CH 3 H CH 3 H OH CHC(O )OCH 2 CH 3 B971 CH3CH2 H CH 3 H OH CHC(O )OCH 2 CH 3 B972 CH3CH2CH2 H CH 3 H OH CHC(O )OCH 2 CH 3 B973 (CH 3 ) 2 CH H CH 3 H OH CHC(O )OCH 2 CH 3 B974 (CH 3 ) 3 C H CH 3 H OH CHC(O )OCH 2 CH 3 B975 CHgS H CH 3 H OH CHC(O )OCH 2 CH 3 B976 CH 3 SO H CH 3 H OH CHC(O )OCH 2 CH 3 B977 CH 3 SO 2 H CH 3 H OH CHC(O )OCH 2 CH 3 B978 Ph H CH 3 H OH CHC(O )OCH 2 CH 3 B979 CH 3 O H CH 3 H OH CHC(O )OCH 2 CH 3 CD CD CD CD CD CD CD CD CD CD CD CD CD X CD ro ro ro ro CD ro ro ro ro ro CD ro ro ro ro ro ro CD ro 03 o o o o o o o CO CO CO CO co CO CO CO CO CO CO CO CO CO CO CO CO CO CO CO Q. - . o o o o o o o o o o o o o o o o CO CO CO CO CO CO CD CD CD CO 00 00 00 00 00 00 00 00 00 00 ro —- O CO 00 -J φ en CO ro —- o C COO 0000 " i φ en -. 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O O . o o o o o o o CO CO CO CO CO CD CO CO CO CO 00 00 00 00 00 00 00 00 00 00 Φ en -To. co ro -»■ o CO 00 -si φ en ■To> CO ro — ^ o CO 00 -M φ en co ro -»■ CO 03 x x x x x x x X X X X X x x x x x x X X -r -xr- -xr- 0 x 0 x 0 x x-τ- -xι- x-π Radical Re R 7 RB R 9 R10 W B1107 CHg CH 3 CH 3 CH 3 CH 3 C(O)O C=O B1108 CH 3 OC(O)CH 2 H H H OH CH 2 B1109 CH 3 OC(O)CH 2 CH 3 H H OH CH 2 B1110 CH 3 OC(O)CH 2 CH 3 CH 3 H OH CH 2 B1111 CH 3 OC(O)CH 2 CH 3 CH 3 CHg OH CH 2 B1112 CH 3 OC(O)CH 2 H CH 3 CHg OH CH 2 B1113 CH 3 OC(O)CH 2 H H H OH CH(CH 3 ) B1114 CH 3 OC(O)CH 2 CHg H H OH CH(CHg) B1115 CH 3 OC(O)CH 2 CHg CH 3 H OH CH(CHg) B1116 CH 3 OC(O)CH 2 CH 3 CHg CHg OH CH(CH 3 ) B1117 CH 3 OC(O)CH 2 H CHg CHg OH CH(CH 3 ) B1118 CH 3 OC(O)CH 2 H H H OH C(CH 3 ) 2 B1119 CH 3 OC(O)CH 2 CH 3 H H OH C(CH 3 ) 2 B1120 CH 3 OC(O)CH 2 CH 3 CHg H OH C(CH 3 ) 2 B1121 CH 3 OC(O)CH 2 CH 3 CHg CHg OH C(CH 3 ) 2 B1122 CH 3 OC(O)CH 2 H CH 3 CHg OH C(CH 3 ) 2 B1123 CH 3 CH 2 OC(O)CH 2 H H H OH CH 2 B1124 CH 3 CH 2 OC(O)CH 2 CH 3 H H OH CH 2 B1125 CH 3 CH 2 OC(O)CH 2 CH 3 CH 3 H OH CH 2 B1126 CH 3 CH 2 OC(O)CH 2 CHg CH 3 CHg OH CH 2 B1127 CH 3 CH 2 OC(O)CH 2 H CH 3 CHg OH CH 2 B1128 CH 3 CH 2 OC(O)CH 2 H H H OH CH(CH 3 ) B1129 CH 3 CH 2 OC(O)CH 2 CHg H H OH CH(CH 3 ) B1130 CH 3 CH 2 OC(O)CH 2 CH 3 CH 3 H OH CH(CH 3 ) B1131 CH 3 CH 2 OC(O)CH 2 CH 3 CH 3 CHg OH CH(CH 3 ) B1132 CH 3 CH 2 OC(O)CH 2 H CH 3 CHg OH CH(CH 3 ) B1133 CH 3 CH 2 OC(O)CH 2 H H H OH C(CH 3 ) 2 B1134 CH 3 CH 2 OC(O)CH 2 CH 3 H H OH C(CH 3 ) 2 B1135 CH 3 CH 2 OC(O)CH 2 CH 3 CH 3 H OH C(CH 3 ) 2 B1136 CH 3 CH 2 OC(O)CH 2 CH 3 CHg CH 3 OH C(CH 3 ) 2 B1137 CH 3 CH 2 OC(O)CH 2 H CHg CH 3 OH C(CH 3 ) 2 ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ? zt ι_l -_! __l __i -_i __! -_i --i ιi ;_i -_i -_i __i __i -_i -i ^ -M CΛ Φ Φ Φ Φ Φ Φ Φ Φ Φ Cn Φ en Φ en Φ Φ en Φ en j?>. j>- j j j5' j . j>. j. j >. co o ' -^ o co oo -si cΛ Φ 4^ ω ro ^ o co c» -M cΛ Φ j>. ω r -^ o cD oo -si cΛ en 4>. eo ro -^ o co 3 O O _ _ O O 0 _ __ r O O O _ _ O O 0 __ _ O 0 O __ _ 0 O O _ _ I _ 0 O O _ ^ - π χ χ X X χ χ χ X X χ χ χ X X χ χ χ X X χ χ χ X X χ χ χ X X χ χ χ χ 3 co co co co co co o ω co co ω co ω ω co ω ω co co co oχ x_ _x oχ ox oχ _x x_ oχ ox oχ _x _x oχ ox oχ x__ r x_ oχ ox oχ _x _x oχ ox oχ _x r _x oχ ox oχ τ x x ^ .<?- π X __ r _X X_ 0χ 0χ X_ _X _X 0χ 0χ _X_ r _X _X 0χ 0χ _X _X X_ 0χ 0χ _X _X X_ 0χ 0χ X_ _X _X 0χ 0χ ^ X. _X r . ^ χ. -3π3 ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox sx 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x 0x Radical Re R 7 Rs R 9 R10 W B1172 CH 3 OCH 2 CH 3 CH 3 CH 3 OH CH 2 B1173 CH 3 OCH 2 H CH 3 CH 3 OH CH 2 B1174 PhCH 2 H H H OH CH 2 B1175 PhCH 2 CH 3 H H OH CH 2 B1176 PhCH 2 CH 3 CH 3 H OH CH 2 B1177 PhCH 2 CH 3 CH 3 CH 3 OH CH 2 B1178 PhCH 2 H CH 3 CH 3 OH CH 2 B1 179 H H H H O-K+ CH 2 B1180 H H H H S(CH 2 ) 7 CH 3 CH 2 B1 181 H H H H S(CH 2 ) 7 CH 3 CH 2 B1182 H H H H SO(CH 2 ) 7 CH 3 CH 2 B1183 H H H H SO 2 (CH 2 ) 7 CH 3 CH 2 B1184 H H H H NHSO 2 CH 3 CH 2 B1185 H H H H NH(CO)S(CH 2 ) 7 CH 3 CH 2 B1 186 H H H H Cl CH 2 B1187 H H H H NH 2 CH 2 B1188 H H H H OC(O)C(CH 3 ) 3 CH 2 B1189 H H H H OC(O)CH 3 CH 2 B1190 H H H H OC(O)Ph CH 2 B1 191 H H H H OC(O)-cyclopropyl CH 2 B1192 H H H H OC(O)CH 2 CH 3 CH 2 B1193 H H H H OC(O)CH=CH 2 CH 2 B1194 H H H H OC(O)CH=CHCH 3 CH 2 B1195 H H H H OC(O)SCH 3 CH 2 B1196 H H H H OC(O)S(CH 2 ) 7 CH 3 CH 2 B1197 H H H H OC(O)OCH 2 CH 3 CH 2 B1198 H H H H OC(O)N(CH 2 CH 3 ) 2 CH 2 B1199 H H H H S-(4-CI-phenyl) CH 2 B1200 H H H H SO-(4-CI-phenyl) CH 2 B1201 H H H H SO 2 -(4-CI-phenyl) CH 2 B1202 H H H H S-(4-CF 3 -phenyl) CH 2 B1203 H H H H SO-(4-CF 3 -phenyl) CH 2 B1204 H H H H SO 2 -(4-CF 3 -phenyl) CH 2 ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro CD ro D ro CD or X 03 ro to ro r o O CO CO CO CO CO co co co co oo oo oo 00 00 oo 00 00 00 —o_ ro ro ro ro ro Q. o o o o o O o CO 00 Φ en J co ro ->■ o co oo -si Φ en co ro -»■ o CD ro o CO 00 -si Φ en 03. ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox x x x x <? ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox X X X X X x x x x x x x x x x x x x x x x x x x x x x X X X X x x x x x x x x x x x x x x x x x x x x x x x x x x x x ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox ox O o o o o o o X o to r Xo to X ro X t Xo ro X to X r Xo Radical Re R 7 Rs R 9 R10 W B1201 CH 3 CH 3 H H SO 2 -(4-CI-phenyl) CH 2 B1202 CH 3 CH 3 H H S-(4-CF 3 -phenyl) CH 2 B1203 CH 3 CH 3 H H SO- ■ (4-CF 3 -phenyl) CH 2 B1204 CH 3 CH 3 H H SO 2 -(4-CFg-phenyl) CH 2 B1205 CH 3 CH 3 H H S-(4-NO 2 -phenyl) CH 2 B1206 CH 3 CH 3 H H SO-(4-NO 2 -phenyl) CH 2 B1207 CHg CH 3 H H SO 2 -(4-NO 2 -phenyl) CH 2 B1213 H H H H OH -CH 2 CH 2 - B1214 CH 3 H H H OH -CH 2 CH 2 ' B1215 CHg CH 3 H H OH -CH 2 CH - B1216 CH 3 CH 3 CH 3 H OH -CH 2 CH 2 - B1217 CH 3 CH 3 CH 3 CH 3 OH -CH 2 CH 2 - In Table 3 which follows, Q is Q 2 and Q 2 the radicals C which follow: Table 3: Radicals C: Radical R 6 R 7 Rl6 R-io p w Radical R 6 R 7 Rι 6 R10 P W C1 H H H OH 1 CH 2 C2 CH 3 H H OH 1 CH 2 C3 CHsCH 2 H H OH 1 CH 2 C4 CH 3 CH 2 CH 2 H H OH 1 CH 2 C5 (CH 3 ) 2 CH H H OH 1 CH 2 C6 (CH 3 ) 3 C H H OH 1 CH 2 C7 CH 3 S H H OH 1 CH 2 C8 CH 3 SO H H OH 1 CH 2 C9 CH 3 SO 2 H H OH 1 CH 2 C10 Ph H H OH 1 CH 2 C11 CH 3 O H H OH 1 CH 2 C12 CH 3 OC(O) H H OH 1 CH 2 C13 CH 3 CH 2 OC(O) H H OH 1 CH 2 C14 CH 2 =CHCH 2 H H OH 1 CH 2 C15 HCCCH 2 H H OH 1 CH 2 C16 CF 3 H H OH 1 CH 2 C17 (CH 3 ) 2 NS02 H H OH 1 CH 2 C18 (CH 3 ) 2 N H H OH 1 CH 2 C19 PhO H H OH 1 CH 2 C20 PhS H H OH 1 CH 2 C21 PhSO H H OH 1 CH 2 C22 PhSO 2 H H OH 1 CH 2 C23 CN H H OH 1 CH 2 C24 CH 3 CH 3 H OH 1 CH 2 C25 CH 3 CH 2 CH 3 H OH 1 CH 2 C26 CH 3 CH 2 CH 2 CH 3 H OH 1 CH 2 C27 (CH 3 ) 2 CH CHg H OH 1 CH 2 C28 (CH 3 ) 3 C CH 3 H OH 1 CH 2 C29 CH 3 S CH 3 H OH 1 CH 2 C30 CH 3 SO CH 3 H OH 1 CH 2 C31 CH 3 SO 2 CH 3 H OH 1 CH 2 C32 Ph CH 3 H OH 1 CH 2 Radical R 6 R 7 Rι 6 R10 P W C33 CH 3 O CH 3 H OH 1 CH 2 C34 CH 3 OC(O) CH 3 H OH 1 CH 2 C35 CH 3 CH 2 OC(O) CH 3 H OH 1 CH 2 C36 CH 2 =CHCH 2 CH 3 H OH 1 CH 2 C37 HCCCH 2 CH 3 H OH 1 CH 2 C38 CF 3 CH 3 H OH 1 CH 2 C39 (CH 3 ) 2 NSO 2 CH 3 H OH 1 CH 2 C40 (CH 3 ) 2 N CH 3 H OH 1 CH 2 C41 PhO CH 3 H OH 1 CH 2 C42 PhS CH 3 H OH 1 CH 2 C43 PhSO CH 3 H OH 1 CH 2 C44 PhSO 2 CH 3 H OH 1 CH 2 C45 CN CH 3 H OH 1 CH 2 C46 H H H OH 4 CH 2 C47 CH 3 H H OH 4 CH 2 C48 CH 3 CH 2 H H OH 4 CH 2 C49 CH 3 CH 2 CH 2 H H OH 4 CH 2 C50 (CH 3 ) 2 CH H H OH 4 CH 2 C51 (CH 3 ) 3 C H H OH 4 CH 2 C52 CH 3 S H H OH 4 CH 2 C53 CH 3 SO H H OH 4 CH 2 C54 CH 3 SO 2 H H OH 4 CH 2 C55 Ph H H OH 4 CH 2 C56 CH 3 O H H OH 4 CH 2 C57 CH 3 OC(O) H H OH 4 CH 2 C58 CH 3 CH 2 OC(O) H H OH 4 CH 2 C59 CH 2 =CHCH 2 H H OH 4 CH 2 C60 HCCCH 2 H H OH 4 CH 2 C61 CF 3 H H OH 4 CH 2 C62 (CH 3 ) 2 NSO 2 H H OH 4 CH 2 C63 (CH 3 ) 2 N H H OH 4 CH 2 C64 PhO H H OH 4 CH 2 C65 PhS H H OH 4 CH 2 Radical Re R 7 Rιe R10 P W C66 PhSO H H OH 4 CH 2 C67 PhSO 2 H H OH 4 CH 2 C68 CN H H OH 4 CH 2 C69 CH 3 CH 3 H OH 4 CH 2 C70 CH 3 CH 2 CH 3 H OH 4 CH 2 C71 CH 3 CH 2 CH 2 CH 3 H OH 4 CH 2 C72 (CH 3 ) 2 CH CH 3 H OH 4 CH 2 C74 CH 3 S CH 3 H OH 4 CH 2 C76 CH 3 SO 2 CH 3 H OH 4 CH 2 C77 Ph CH 3 H OH 4 CH 2 C78 CH 3 O CH 3 H OH 4 CH 2 C79 CH 3 OC(O) CH 3 H OH 4 CH 2 C80 CH 3 CH 2 OC(O) CH 3 H OH 4 CH 2 C81 CH 2 =CHCH 2 CH 3 H OH 4 CH 2 C82 HCCCH 2 CH 3 H OH 4 CH 2 C83 CF 3 CH 3 H OH 4 CH 2 C84 (CH 3 ) 2 NSO 2 CH 3 H OH 4 CH 2 C85 (CH 3 ) 2 N CH 3 H OH 4 CH 2 C86 PhO CH 3 H OH 4 CH 2 C87 PhS CH 3 H OH 4 CH 2 C88 PhSO CH 3 H OH 4 CH 2 C89 PhSO 2 CH 3 H OH 4 CH 2 C90 CN CH 3 H OH 4 CH 2 C91 H H H OH 3 CH 2 C92 CH 3 H H OH 3 CH 2 C93 CH 3 CH 2 H H OH 3 CH 2 C94 CH 3 CH 2 CH 2 H - H OH 3 CH 2 C95 (CH 3 ) 2 CH H H OH 3 CH 2 C96 (CH 3 ) 3 C H H OH 3 CH 2 C97 CH 3 S H H OH 3 CH 2 C98 CH 3 SO H H OH 3 CH 2 Radical R 6 R 7 Rι 6 R10 P W C99 CH 3 SO 2 H H OH 3 CH 2 C100 Ph H H OH 3 CH 2 C101 CH 3 O H H OH 3 CH 2 C102 CH 3 OC(O) H H OH 3 CH 2 C103 CH 3 CH 2 OC(O) H H OH 3 CH 2 C104 CH 2 =CHCH 2 H H OH 3 CH 2 C105 HCCCH 2 H H OH 3 CH 2 C106 CF 3 H H OH 3 CH 2 C107 (CH 3 ) 2 NSO 2 H H OH 3 CH 2 C108 (CH 3 ) 2 N H H OH 3 CH 2 C109 PhO H H OH 3 CH 2 C1 10 PhS H H OH 3 CH 2 C1 1 1 PhSO H H OH 3 CH 2 C1 12 PhSO 2 H H OH 3 CH 2 C1 13 CN H H OH 3 CH 2 C114 CH 3 CH 3 H OH 3 CH 2 C1 15 CH 3 CH 2 CH 3 H OH 3 CH 2 C116 CH 3 CH 2 CH 2 CH 3 H OH 3 CH 2 C1 17 (CH 3 ) 2 CH CH 3 H OH 3 CH 2 C1 18 (CH 3 ) 3 C CH 3 H OH 3 CH 2 C120 CH 3 SO CH 3 H OH 3 CH 2 C121 CH 3 SO 2 CH 3 H OH 3 CH 2 C122 Ph CH 3 H OH 3 CH 2 C124 CH 3 OC(O) CH 3 H OH 3 CH 2 C125 CH 3 CH 2 OC(O) CH 3 H OH 3 CH 2 C126 CH 2 =CHCH 2 CH 3 H OH 3 CH 2 C127 HCCCH 2 CH 3 H OH 3 CH 2 C128 CF 3 CH 3 H OH 3 CH 2 C129 (CH 3 ) 2 NSO 2 CH 3 H OH 3 CH 2 C130 (CH 3 ) 2 N CH 3 H OH 3 CH 2 C131 PhO CH 3 H OH 3 CH 2 Radical Re R 7 R16 R10 P W C136 CHgCH 2 CHgCH 2 H OH 1 CH 2 C139 CH 3 CH 3 H OH 1 CH(CHg) C140 CH 2 CH 3 H H OH 1 CH(CHg) C141 CH 2 CH 3 CH 3 H OH 1 CH(CHg) C142 CHsCH 2 CH3CH2 H OH 1 CH(CH 3 ) C144 CH 3 CH 3 CH 3 OH 1 CH 2 C145 CH3CH2 CH3CH2 CH 3 OH 1 CH 2 C146 H H H OH 2 CH 2 C148 CH3CH2 CHgCH2 H OH 2 CH 2 C149 H H H OH 5 CH 2 C151 CHgCH 2 CHgCH 2 H OH 5 CH 2 In Table 4 which follows, Q is Q 3 and Q 3 the following radicals D: Table 4: Radicals D: Radical R 7 R 8 R12 R10 o Radical Re R 7 R 8 R12 R10 ° D1 H H H H OH 2 D2 CH 3 H H H OH 2 D3 CH 3 CH 2 H H H OH 2 D4 CH 3 CH 2 CH 2 H H H OH 2 D8 CHgSO H H H OH 2 D9 CHgSO 2 H H H OH 2 D10 Ph H H H OH 2 D12 CH 2 =CHCH 2 H H H OH 2 D13 HCCCH 2 H H H OH 2 D15 PhO H H H OH 2 D16 PhS H H H OH 2 D17 PhSO H H H OH 2 D18 PhSO 2 H H H OH 2 D20 CHgCH 2 CH 3 H H OH 2 D21 CHgCH 2 CH 2 CH 3 H H OH 2 D25 CHgSO CH 3 H H OH 2 D26 CH 3 SO 2 CH 3 H H OH 2 D27 Ph CH 3 H H OH 2 D28 CH 3 O CH 3 H H OH 2 D29 CH 2 =CHCH 2 CH 3 H H OH 2 D30 HCCCH≥ CH 3 H H OH 2 D31 CF 3 CH 3 H H OH 2 D32 PhO CH 3 H H OH 2 Radical R 6 R 7 R 8 R12 R10 o D33 PhS CH 3 H H OH 2 D34 PhSO CH 3 H H OH 2 D35 PhSO 2 CH 3 H H OH 2 D36 H H H H OH 3 D37 CH 3 H H H OH 3 D38 CH 3 CH 2 H H H OH 3 D39 CH 3 CH 2 CH 2 H H H OH 3 D40 (CH 3 ) 2 CH H H H OH 3 D41 (CH 3 ) 3 C H H H OH 3 D42 CH 3 S H H H OH 3 D44 CH 3 SO 2 H H H OH 3 D45 Ph H H H OH 3 D46 CH 3 O H H H OH 3 D47 CH 2 =CHCH 2 H H H OH 3 D48 HCCCH 2 H H H OH 3 D49 CF 3 H H H OH 3 D50 PhO H H H OH 3 D51 PhS H H H OH 3 D52 PhSO H H H OH 3 D53 PhSO 2 H H H OH 3 D54 CH 3 CH 3 H H OH 3 D55 CH 3 CH 2 CH 3 H H OH 3 D56 CH 3 CH 2 CH 2 CH 3 H H OH 3 D57 (CH 3 ) 2 CH CH 3 H H OH 3 D58 (CH 3 ) 3 C CH 3 H H OH 3 D59 CH 3 S CH 3 H H OH 3 D60 CH 3 SO CH 3 H H OH 3 D61 CH 3 SO 2 CH 3 H H OH 3 D62 Ph CH 3 H H OH 3 D64 CH 2 =CHCH 2 CH 3 H H OH 3 D65 HCCCH 2 CH 3 H H OH 3 Radical Re R 7 Rs R12 R10 0 D67 PhO CH 3 H H OH 3 D68 PhS CH 3 H H OH 3 D69 PhSO CH 3 H H OH 3 D70 PhSO 2 CH 3 H H OH 3 D71 H H H H OH 4 D73 CHgCH 2 H H H OH 4 D74 CH 3 CH 2 CH 2 H H H OH 4 D75 (CH 3 ) 2 CH H H H OH 4 D76 (CH 3 ) 3 C H H H OH 4 D77 CH 3 S H H H OH 4 D78 CHgSO H H H OH 4 D79 CH 3 SO 2 H H H OH 4 D80 Ph H H H OH 4 D81 CH 3 O H H H OH 4 D82 CH 2 = CHCH2 H H H OH 4 D83 HCCCH 2 H H H OH 4 D84 CF 3 H H H OH 4 D85 PhO H H H OH 4 D86 PhS H H H OH 4 D87 PhSO H H H OH 4 D88 PhSO 2 H H H OH 4 D89 CH 3 CH 3 H H OH 4 D90 CH 3 CH 2 CH 3 H H OH 4 D91 CH 3 CH 2 CH 2 CH 3 H H OH 4 D92 (CH 3 ) 2 CH CH 3 H H OH 4 D93 (CH 3 ) 3 C CH 3 H H OH 4 D94 CH 3 S CH 3 H H OH 4 D96 CH 3 SO 2 CH 3 H H OH 4 D97 Ph CH 3 H H OH 4 D98 CH 3 O CH 3 H H OH 4 o o o o o o σ o o o o o o o o o o o o o o o o o o o o o σ o o o π όT co co ro ' ro ' ro ' ro ' ro ' ro ' ro ' ro ' ro ' ro ' - j ' - - j ' - -^ ' -^ ' -' ' -» ' - '* ' ' _ --^ o, o. ^ o1 o, o_ o. o _Z ^ o1 o, o. Q -^ o co oo i Φ e ^ c ro -^ o co oo ^J Φ en j^ co ro ->• O ffl flf vl Ol ϋl J- C M -' O O o 03 o o o X X X x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x o o x x x x x x x X X X ^ ro o X oX oX oX oX oX oX oX oX oX oX oX oX oX oX oX oX oX oX oX oX oX oX oX o X o X o X o o X o X o X o X o X X X o CO .&> *>. Radical Re R 7 Rs R12 R10 o D132 CH 3 CH 2 OC(O) CH 3 CH 3 H OH 1 D133 CH 3 O CH 3 CH 3 H OH 1 D134 CH 3 S CH 3 CH 3 H OH 1 D135 CH 3 SO CH 3 CH 3 H OH 1 D136 CH 3 SO 2 CH 3 CH 3 H OH 1 D139 H H CH 3 CH 3 OH 1 D140 CH 3 CH 2 OC(O) CH 3 H H OH 4 In Table 5 which follows, Q is Q 4 and Q the following radicals E: Table 5: Radicals E: Radical Re R 7 R10 X Y W q E1 H H OH S CH 2 CH 2 2 E2 CH 3 H OH S CH 2 CH 2 2 E3 CH 3 CH 3 OH S CH 2 CH 2 2 E4 CH 3 OC(O) H OH S CH 2 CH 2 2 E5 CH 3 CH 3 OC(O) OH S CH 2 CH 2 2 E6 H H OH SO CH 2 CH 2 2 E7 CH 3 H OH SO CH 2 CH 2 2 E8 CH 3 CH 3 OH SO CH 2 CH 2 2 E9 CH 3 OC(O) H OH SO CH 2 CH 2 2 E10 CH 3 CH 3 OC(O) OH SO CH 2 CH 2 2 E11 H H OH SO 2 CH 2 CH 2 2 Radical Re R 7 R10 X Y w q E12 CH 3 H OH SO 2 CH 2 CH 2 2 E13 CH 3 CH 3 OH SO 2 CH 2 CH 2 2 E14 CH 3 OC(O) H OH SO 2 CH 2 CH 2 2 E15 CH 3 CH 3 OC(O) OH SO 2 CH 2 CH 2 2 E16 H H OH CO O CH 2 2 E17 CH 3 H OH CO O CH 2 2 E18 CH 3 CH 3 OH CO O CH 2 2 E19 CH 3 OC(O) H OH CO O CH 2 2 E20 CH 3 CH 3 OC(O) OH CO O CH 2 2 E21 H H OH CO O CH 2 2 E22 CH 3 H OH CO O CH 2 2 E23 CH 3 CH 3 OH CO O CH 2 2 E24 CH 3 OC(O) H OH CO O CH 2 2 E25 CH 3 CH 3 OC(O) OH CO O CH 2 2 E26 H H OH CO O CH 2 2 E27 CH 3 H OH CO O CH 2 2 E28 CH 3 CH 3 OH CO O CH 2 2 E29 CH 3 OC(O) H OH CO O CH 2 2 E30 CH 3 CH 3 OC(O) OH CO O CH 2 2 In Table 6 which follows, Q is Q 5 and Q 5 the radicals F which follow: Table 6: Radicals F: Radical Re R 7 Rs Rio F1 H H H OH F2 CH 3 H H OH Radical Re R 7 Rs R 10 F3 CH 3 CH 3 H OH F4 CH 3 CH 3 CH 3 OH F5 H H CH 3 OH F6 H CH 3 CH 3 OH Table 7: Compounds of the formula la Comp. R 2 R 3 R 4 R 5 Qi P No. A5 (CH 3 ) 3 C H H CF 3 B24 0 A6 cyclopropyl H H CF 3 B24 0 A8 CH 3 OCH 2 H H CF 3 B24 0 A9 CH 3 O(CH 2 ) 2 H H CFg B24 0 A11 PhO H H CF 3 B24 0 A12 PhS H H CF 3 B24 0 A13 PhSO H H CF 3 B24 0 A14 PhSO 2 H H CF 3 B24 0 A16 CHgSO H H CF 3 B24 0 Comp. R 2 R 3 R 4 Rs Qi P No. A19 HCC H H CF 3 B24 0 A20 CHgCC H H CF 3 B24 0 A21 CH 2 =CH H H CF 3 B24 0 A22 CH 2 =CHCH 2 H H CF 3 B24 0 A23 CH 3 SO 2 N(CH 3 ) H H CF 3 B24 0 A24 (CH 3 ) 2 N H H CF 3 B24 0 A25 (CH 3 ) 2 NSO 2 H H CF 3 B24 0 A26 CICH 2 H H CF 3 B24 0 A28 CH 3 SOCH 2 H H CF 3 B24 0 A29 CHgSO 2 CH 2 H H CF 3 B24 0 A30 [1.2.4]-triazol-1 - H H CF 3 B24 0 ylmethyl A33 H H H CF 3 CF 2 B24 0 A35 CHgCH 2 H H CF 3 CF 2 B24 0 A36 cyclopropyl H H CF 3 CF 2 B24 0 A37 (CH 3 ) 3 C H H CF 3 CF 2 B24 0 A38 (CHg) 2 CH H H CF 3 CF 2 B24 0 A39 CHg(CH 2 ) 2 H H CF 3 CF 2 B24 0 A40 CH 3 OCH 2 H H CF 3 CF 2 B24 0 A41 CH 3 O(CH 2 ) 2 H H CF 3 CF 2 B24 0 A42 Ph H H CF 3 CF 2 B24 0 A43 PhO H H CF 3 CF 2 B24 0 A44 PhS H H CF 3 CF 2 B24 0 A45 PhSO H H CF 3 CF 2 B24 0 A46 PhSO 2 H H CFgCF 2 B24 0 A47 CH 3 S H H CF 3 CF 2 B24 0 A49 CF 3 H H CF 3 CF 2 B24 0 Comp. R 2 R a Rs Qi P No. A50 F 2 CH H H CF 3 CF 2 B24 0 A51 HCC H H CF 3 CF 2 B24 0 A52 CH 3 CC H H CF 3 CF 2 B24 0 A53 CH 2 =CH H H CF 3 CF 2 B24 0 A54 CH 2 =CHCH 2 H H CF 3 CF 2 B24 0 A55 CH 3 SO 2 N(CH 3 ) H H CF 3 CF 2 B24 0 A56 (CH 3 ) 2 N H H CF 3 CF 2 B24 0 A57 (CH 3 ) 2 NSO 2 H H CF 3 CF 2 B24 0 A58 CICH 2 H H CF 3 CF 2 B24 0 A59 CH 3 SCH 2 H H CF 3 CF 2 B24 0 A60 CH 3 SOCH 2 H H CF 3 CF 2 B24 0 A61 CH 3 SO 2 CH 2 H H CF 3 CF0. B24 0 A62 [1.2.4]-triazol-1- H H CF 3 CF 2 B24 0 ylmethyl A63 H H H CF 3 CF 2 CF 2 B24 0 A64 CH 3 H H CF 3 CF 2 CF 2 B24 0 A65 CH 3 CH 2 H H CF 3 CF 2 CF 2 B24 0 A66 cyclopropyl H H CF 3 CF 2 CF 2 B24 0 A67 (CH 3 ) 3 C H H CF 3 CF 2 CF 2 B24 0 A68 (CH 3 ) 2 CH H H CF 3 CF 2 CF 2 B24 0 A69 CHs(CH 2 ) 2 H H CF 3 CF 2 CF 2 B24 0 A70 CH 3 OCH 2 H H CF 3 CF 2 CF 2 B24 0 A71 CH 3 O(CH 2 ) 2 H H CF 3 CF 2 CF 2 B24 0 A72 Ph H H CF 3 CF 2 CF 2 B24 0 A73 PhO H H CF 3 CF 2 CF 2 B24 0 A74 PhS H H CF 3 CF 2 CF 2 B24 0 A75 PhSO H H CF 3 CF 2 CF 2 B24 0 A76 PhSO 2 H H CF 3 CF 2 CF 2 B24 0 A77 CH 3 S H H CF 3 CF 2 CF 2 B24 0 A78 CHgSO H H CF 3 CF 2 CF 2 B24 0 A79 CFg H H CF 3 CF 2 CF 2 B24 0 A80 F 2 CH H H CF 3 CF 2 CF 2 B24 0 o f © Q. o O O o o O o O o O O o o o o o o o O O 0- W ■ st -sf ■ s ■ st "s ■ s ■ "sf ■ s ■ st ■ st ■ s ■ st "st ■ st ■ st ■ st • st ■ st "st ■ st ■ st "* "st ■ st ■ st H σ ω CM CM m CM CM CM CM CM CM CM CM CM CM CM CM CM CM CM CM CM CM CM CM CM CM CM CM CM CM CM CM CM υ CQ CQ m ω CΩ CQ c Q ω o m Q Q Q ω ω ω Q Q CQ Q m cQ ω a. m CQ CQ CQ LL UL Li. LL LL LL LL LL LL LL LL u_ o o O o O o o o O o O O L LL u_ u_ LL LL LL LL U_ LL o o o o o o o o o o o o o o o o o o o X u_ LL L o O O O o o O O O O o O -_L _i. _i. L L Li. U_. U_. LL LL LL LL LL LL LL L LL U_ LL LL LL LL l_L LL LL LL LL o o o o o o o o o o o o o o o o o o o O O o O o O O o O O o O X x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x _r x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x Comp. R 2 R a Qi P No. A112 CH 3 CC H H CF 2 CI B24 0 A113 CH 2 =CH H H CF 2 CI B24 0 A114 CH 2 =CHCH 2 H H CF 2 CI B24 0 A115 CH 3 SO 2 N(CH 3 ) H H CF 2 CI B24 0 A116 (CH 3 ) 2 N H H CF 2 CI B24 0 A117 (CH 3 ) 2 NSO 2 H H CF 2 CI B24 0 A118 CICH 2 H H CF 2 CI B24 0 A119 CH 3 SCH; ! H H CF 2 CI B24 0 A120 CH 3 SOCH . H H CF 2 CI B24 0 A121 CH 3 SO 2 CH 2 H H CF 2 CI B24 0 A122 [1.2.4]-triazol-1 - H H CF 2 CI B24 0 ylmethyl A123 H H H CHF 2 B24 0 A124 CH 3 H H CHF 2 B24 0 A125 CHsCH 2 H H CHF 2 B24 0 A126 cyclopropyl H H CHF 2 B24 0 A127 (CH 3 ) 3 C H H CHF 2 B24 0 A128 (CH 3 ) 2 CH H H CHF 2 B24 0 A129 CH 3 (CH 2 ) 2 H H CHF 2 B24 0 A130 CH 3 OCH 2 H H CHF 2 B24 0 A131 CH 3 O(CH 2 ) 2 H H CHF 2 B24 0 A132 Ph H H CHF 2 B24 0 A133 PhO H H CHF 2 B24 0 A134 PhS H H CHF 2 B24 0 A135 PhSO H H CHF 2 B24 0 A136 PhSO 2 H H CHF 2 B24 0 A137 CH 3 S H H CHF 2 B24 0 A138 CH 3 SO H H CHF 2 B24 0 A139 CF 3 H H CHF 2 B24 0 A140 F 2 CH H H CHF 2 B24 0 A141 HCC H H CHF 2 B24 0 A142 CH 3 CC H H CHF 2 B24 0 Comp. R 2 R 3 R 4 R 5 Qi P No. A143 CH 2 =CH H H CHF 2 B24 0 A144 CH 2 =CHCH 2 H H CHF 2 B24 0 A145 CH 3 SO 2 N(CH 3 ) H H CHF 2 B24 0 A146 (CH 3 ) 2 N H H CHF 2 B24 0 A147 (CH 3 ) 2 NSO 2 H H CHF 2 B24 0 A148 CICH 2 H H CHF 2 B24 0 A149 CH 3 SCH 2 H H CHF 2 B24 0 A150 CH 3 SOCH 2 H H CHF 2 B24 0 A151 CH 3 SO 2 CH 2 H H CHF 2 B24 0 A152 [1.2.4]-triazol-1 - H H CHF 2 B24 0 ylmethyl A155 CHgCH 2 H H CCI3 B24 0 A156 cyclopropyl H H CCIg B24 0 A157 (CHg)gC H H CCIg B24 0 A158 (CHg) 2 CH H H CCIg B24 0 A159 CHg(CH 2 ) 2 H H CCIg B24 0 A160 CH 3 OCH 2 H H CCIg B24 0 A161 CH 3 O(CH 2 ) 2 H H CCIg B24 0 Comp. R 2 R 3 R 4 R 5 Qi P No. A174 CH 2 =CHCH 2 H H CCI3 B24 0 A175 CHgSO 2 N(CHg) H H CCI3 B24 0 A176 (CHg) 2 N H H CCI3 B24 0 A177 (CH 3 ) 2 NSO 2 H H CCI3 B24 0 A179 CH 3 SCH 2 H H CCI3 B24 0 A180 CH 3 SOCH 2 H H CCI3 B24 0 A181 CH3SO CH2 H H CCI3 B24 0 A182 [1.2.4]-triazol-1 - H H CCIg B24 0 yimethyl A184 CH 3 H CH 3 CF 3 B24 0 A185 CH3CH2 H CH 3 CF 3 B24 0 A186 cyclopropyl H CHg CF 3 B24 0 A187 (CH 3 ) 3 C H CH 3 CF 3 B24 0 A188 (CH 3 ) 2 CH H CHg CFg B24 0 A189 CHg(CH 2 ) 2 H CH 3 CFg B24 0 A190 CH3OCH2 H CH 3 CFg B24 0 A191 CH 3 O(CH 2 ) 2 H CHg CFg B24 0 A192 Ph H CH 3 CF 3 B24 0 A193 PhO H CH 3 CF 3 B24 0 A194 PhS H CH 3 CF 3 B24 0 A195 PhSO H CH 3 CF 3 B24 0 A196 PhSO 2 H CH 3 CF 3 B24 0 A197 CH 3 S H CH 3 CF 3 B24 0 A198 CHgSO H CH 3 CF 3 B24 0 A202 CHgCC H CH3 CF 3 B24 0 A203 CH 2 =CH H CH3 CFg B24 0 A204 CH 2 =CHCH 2 H CH3 CFg B24 0 jomp. π 2 R 4 Qi P No. A205 CHgSO 2 N(CHg) H CHg CF 3 B24 0 A206 (CHg) 2 N H CHg CF 3 B24 0 A207 (CH 3 ) 2 NSO 2 H CHg CF 3 B24 0 A209 CHgSCH 2 H CHg CF 3 B24 0 A210 CH 3 SOCH 2 H CH3 CFg B24 0 A21 1 CHsSO 2 CH 2 H CH3 CF3 B24 0 A213 CH 3 H CH3 CF 3 CF 2 B24 0 A214 CHsCH 2 H CH3 CF 3 CF 2 B24 0 A215 cyclopropyl H CH3 CF 3 CF 2 B24 0 A216 (CH 3 ) 3 C H CH3 CF 3 CF 2 B24 0 A217 (CH 3 ) 2 CH H CHg CFgCF 2 B24 0 A218 CHs(CH 2 ) 2 H CH3 CFgCF 2 B24 0 A219 CH 3 OCH 2 H CHg CFgCF 2 B24 0 A220 CH 3 O(CH 2 ) 2 H CH3 CFgCF 2 B24 0 A222 PhO H CHg CF 3 CF 2 B24 0 A223 PhS H CHg CF 3 CF 2 B24 0 A224 PhSO H CHg CFgCF 2 B24 0 A225 PhSO 2 H CHg CFgCF 2 B24 0 A226 CH 3 S H CH3 CF3CF2 B24 0 A227 CH 3 SO H CH3 CF3CF2 B24 0 A228 CF 3 H CH3 CF 3 CF 2 B24 0 A229 F 2 CH H CH3 CF 3 CF 2 B24 0 A230 HCC H CH3 CF 3 CF 2 B24 0 A231 CH 3 CC H CHg CF 3 CF 2 B24 0 A232 CH 2 =CH H CHg CF 3 CF 2 B24 0 A233 CH 2 =CHCH 2 H CHg CF 3 CF 2 B24 0 A234 CH 3 SO 2 N(CH 3 ) H CH3 CF 3 CF 2 B24 0 A235 (CHg) 2 N H CH3 CF 3 CF 2 B24 0 A236 (CH 3 ) 2 NSO 2 H CH3 CF 3 CF 2 B24 0 Comp. R 2 R 3 R 4 R 5 Qi P No. A237 CICH 2 H CHg CF 3 CF 2 B24 0 A238 CHsSCH 2 H CHg CF 3 CF 2 B24 0 A239 CH 3 SOCH 2 H CH 3 CF 3 CF 2 B24 0 A240 CHgSO 2 CH 2 H CH 3 CF 3 CF 2 B24 0 A241 H H CH 3 CF3CF 2 CF 2 B24 0 A242 CHg H CH 3 CF3CF2CF2 B24 0 A243 CHgCH 2 H CH 3 CFgCF 2 CF 2 B24 0 A244 cyclopropyl H CH 3 CFgCF 2 CF2 B24 0 A245 (CHg)gC H CH 3 CFgCF2C 2 B24 0 A246 (CHg) 2 CH H CH 3 CFgCF CF2 B24 0 A247 CHg(CH 2 ) 2 H CH 3 CFgCF2CF2 B24 0 A248 CH 3 OCH 2 H CH 3 CF CF2CF 2 B24 0 A249 CH 3 O(CH 2 ) 2 H CH 3 C F3C F2C 2 B24 0 A250 Ph H CH 3 CFgCF2CF 2 B24 0 A251 PhO H CH 3 CFgCF CF 2 B24 0 A252 PhS H CH 3 C FgC F 2 C F 2 B24 0 A253 PhSO H CH 3 CFgCF 2 CF B24 0 A254 PhSO 2 H CH 3 CFgCF CF 2 B24 0 A255 CH 3 S H CH 3 C F3C F 2 C F 2 B24 0 A256 CH 3 SO H CHg CF3CF2CF2 B24 0 A257 CF 3 H CH 3 CFgCF 2 CF 2 B24 0 A258 F 2 CH H CH 3 CFgCF 2 CF 2 B24 0 A259 HCC H CH 3 C F3C F C F 2 B24 0 A260 CH 3 CC H CH 3 C F3C F 2 C F 2 B24 0 A261 CH 2 =CH H CH 3 CF3CF 2 CF 2 B24 0 A262 H CH 3 CFsCF 2 CF 2 B24 0 A263 CH 3 SO 2 N(CH 3 ) H CH 3 B24 0 A264 (CH 3 ) 2 N H CH 3 CF3CF 2 CF 2 B24 0 A265 (CH 3 ) 2 NSO 2 H CH 3 CF 3 CF 2 CF 2 B24 0 A266 CICH 2 H CH 3 CF3CF 2 CF 2 B24 0 A267 CH 3 SCH 2 H CH 3 CF3CF 2 CF 2 B24 0 A268 CH 3 SOCH 2 H CHg C 3CF 2 CF 2 B24 0 Comp. R 2 R3 R 4 R 5 Qi P No. A269 CHgSO 2 CH H CHg C FgC C F2 B24 0 A270 H H CH 3 CF 2 CI B24 0 A272 CHgCH 2 H CH 3 CF 2 CI B24 0 A273 cyclopropyl H CH 3 CF 2 CI B24 0 A274 (CH 3 ) 3 C H CH 3 CF 2 CI B24 0 A275 (CHg) 2 CH H CH 3 CF 2 CI B24 0 A276 CH 3 (CH 2 ) 2 H CH 3 CF 2 CI B24 0 A277 CH 3 OCH 2 H CHg CF 2 CI B24 0 A278 CH 3 O(CH 2 ) 2 H CHg CF 2 CI B24 0 A282 PhSO H CH3 CF 2 CI B24 0 A283 PhSO 2 H CH3 CF 2 CI B24 0 A284 CH 3 S H CH3 CF 2 CI B24 0 A285 CH 3 SO H CH3 CF 2 CI B24 0 A287 F 2 CH H CHg CF 2 CI B24 0 A289 CH 3 CC H CHg CF 2 CI B24 0 A290 CH 2 =CH H CHg CF 2 CI B24 0 A291 CH 2 =CHCH 2 H CHg CF 2 CI B24 0 A292 CH 3 SO 2 N(CH 3 ) H CH3 CF 2 CI B24 0 A293 (CH 3 ) 2 N H CH3 CF 2 CI B24 0 A294 (CH 3 ) 2 NSO 2 H CHg CF 2 CI B24 0 A295 CICH 2 H CHg CF 2 CI B24 0 A296 CH 3 SCH 2 H CHg CF 2 CI B24 0 A297 CH3SOCH2 H CHg CF 2 CI B24 0 A298 CH3SO2CH2 H CHg CF 2 CI B24 0 Comp. R 2 R 3 R 4 R 5 Qi P No. A301 CHgCH 2 H CH 3 CHF 2 B24 0 A302 cyclopropyl H CHg CHF 2 B24 0 A303 (CHg)gC H CH 3 CHF 2 B24 0 A304 (CHg) 2 CH H CH 3 CHF 2 B24 0 A305 CHg(CH 2 ) 2 H CH 3 CHF 2 B24 0 A306 CH 3 OCH 2 H CH 3 CHF 2 B24 0 A307 CH 3 O(CH 2 ) 2 H CH 3 CHF 2 B24 0 A308 Ph H CH 3 CHF 2 B24 0 A309 PhO H CH 3 CHF 2 B24 0 A310 PhS H CH 3 CHF 2 B24 0 A311 PhSO H CH 3 CHF 2 B24 0 A312 PhSO 2 H CH 3 CHF 2 B24 0 A314 CHgSO H CH 3 CHF 2 B24 0 A316 F 2 CH H CH 3 CHF 2 B24 0 A317 HCC H CH 3 CHF 2 B24 0 A318 CHgCC H CH 3 CHF 2 B24 0 A319 CH 2 =CH H CH 3 CHF 2 B24 0 A320 CH 2 =CHCH 2 H CH 3 CHF 2 B24 0 A321 CHgSO 2 N(CHg) H CH 3 CHF 2 B24 0 A322 (CH 3 ) 2 N H CH 3 CHF 2 B24 0 A323 (CH 3 ) 2 NSO 2 H CH 3 CHF 2 B24 0 A324 CICH 2 H CH 3 CHF 2 B24 0 A325 CHgSCH 2 H CH 3 CHF 2 B24 0 A326 CH 3 SOCH 2 H CH 3 CHF 2 B24 0 A327 CH 3 SO 2 CH 2 H CH 3 CHF 2 B24 0 A328 H H CH 3 CCI 3 B24 0 A330 CHgCH 2 H CH 3 CCI3 B24 0 A331 (CHg) 3 C H CH 3 CCI3 B24 0 A332 (CH 3 ) 2 CH H CH 3 CCI3 B24 0 Comp. R 2 R 3 R 4 R 5 Qi P No. A333 cyclopropyl H CH 3 CCI3 B24 0 A334 CH 3 (CH 2 )2 H CH 3 CCI3 B24 0 A335 CH 3 OCH 2 H CH 3 CCI3 B24 0 A336 CH 3 O(CH 2 ) 2 H CH 3 CCI3 B24 0 A341 PhSO 2 H CH 3 CCb B24 0 A342 CH 3 S H CH 3 CCb B24 0 A343 CHgSO H CH 3 CCI3 B24 0 A347 CH 3 CC H CH 3 CCb B24 0 A348 CH 2 =CH H CH 3 CCI 3 B24 0 A350 CH 3 SO 2 N(CH 3 ) H CHg CCI 3 B24 0 A351 (CH 3 ) 2 N H CHg CCI 3 B24 0 A352 (CH 3 ) 2 NSO 2 H CHg CCI 3 B24 0 A353 CICH2 H CH 3 CCI 3 B24 0 A354 CH 3 SCH2 H CH 3 CCI3 B24 0 A355 CH 3 SOCH 2 H CH 3 CCI3 B24 0 A356 CH 3 SO2CH2 H CH 3 CCI 3 B24 0 A358 CH 3 H Ph CF 3 B24 0 A360 cyclopropyl H Ph CFg B24 0 A361 (CH 3 ) 3 C H Ph CF 3 B24 0 A362 (CH 3 ) 2 CH H Ph CF 3 B24 0 A363 CH 3 (CH 2 )2 H Ph CF 3 B24 0 A364 CH 3 OCH 2 H Ph CF 3 B24 0 Comp. R 2 R 3 R 4 Rs Qi P No. A365 CH 3 O(CH 2 ) 2 H Ph CF 3 B24 0 A366 Ph H Ph CF 3 B24 0 A367 PhO H Ph CF 3 B24 0 A368 PhS H Ph CF 3 B24 0 A369 PhSO H Ph CF 3 B24 0 A370 PhSO 2 H Ph CF 3 B24 0 A371 CH 3 S H Ph CF 3 B24 0 A372 CH 3 SO H Ph CF 3 B24 0 A373 CF 3 H Ph CF 3 B24 0 A374 F 2 CH H Ph CF 3 B24 0 A375 HCC H Ph CF 3 B24 0 A376 CHgCC H Ph CF 3 B24 0 A377 CH 2 =CH H Ph CF 3 B24 0 A379 CH 3 SO 2 N(CH 3 ) H Ph CF 3 B24 0 A380 (CH 3 ) 2 N H Ph CF 3 B24 0 A381 (CH 3 ) 2 NSO 2 H Ph CF 3 B24 0 A382 CICH 2 H Ph CF 3 B24 0 A383 CH3SCH2 H Ph CF 3 B24 0 A384 CH3SOCH2 H Ph CF 3 B24 0 A385 CH3SO2CH2 H Ph CF 3 B24 0 A388 CH3CH2 H Ph CF3CF2 B24 0 A389 cyclopropyl H Ph CF 3 CF 2 B24 0 A390 (CH 3 ) 3 C H Ph CF 3 CF 2 B24 0 A391 (CH 3 ) 2 CH H Ph CF3CF2 B24 0 A392 CH 3 (CH2)2 H Ph CF3CF2 B24 0 A393 CH 3 OCH 2 H Ph CF3CF2 B24 0 A394 CH 3 O(CH 2 ) 2 H Ph CF3CF 2 B24 0 Comp. R 2 R 3 Qi P No. A397 PhS H Ph CF 3 CF 2 B24 0 A398 PhSO H Ph CF 3 CF 2 B24 0 A399 PhSO 2 H Ph CF 3 CF 2 B24 0 A400 CH 3 S H Ph CF3CF2 B24 0 A401 CH 3 SO H Ph CF 3 CF 2 B24 0 A403 F 2 CH H Ph CF3CF 2 B24 0 A404 HCC H Ph CF 3 CF 2 B24 0 A405 CH 3 CC H Ph CF3CF 2 B24 0 A406 CH 2 =CH H Ph CF3CF 2 B24 0 A407 CH 2 =CHCH 2 H Ph CF3CF 2 B24 0 A408 CH 3 SO 2 N(CH 3 ) H Ph CF3CF2 B24 0 A409 (CH 3 ) 2 N H Ph CF 3 CF 2 B24 0 A410 (CH 3 ) 2 NSO 2 H Ph CF 3 CF 2 B24 0 A411 CICH 2 H Ph CF 3 CF 2 B24 0 A412 CH3SCH2 H Ph CF 3 CF 2 B24 0 A413 CH 3 SOCH 2 H Ph CF 3 CF 2 B24 0 A414 CH3SO2CH2 H Ph CF 3 CF 2 B24 0 A415 H H Ph CF3CF 2 CF 2 B24 0 A416 CH 3 H Ph CF3CF2CF2 B24 0 A417 CH 3 CH2 H Ph CF 3 CF 2 CF 2 B24 0 A418 cyclopropyl H Ph C F 3 C F 2 C F 2 B24 0 A419 (CH 3 ) 3 C H Ph CF 3 CF 2 CF 2 B24 0 A420 (CH 3 ) 2 CH H Ph CF 3 CF 2 CF 2 B24 0 A421 CHs(CH2)2 H Ph CF 3 CF 2 CF 2 B24 0 A422 CH3OCH2 H Ph CF 3 CF 2 CF 2 B24 0 A423 CH 3 O(CH 2 ) 2 H Ph CF 3 CF 2 CF 2 B24 0 A424 Ph H Ph CF 3 CF 2 CF 2 B24 0 A425 PhO H Ph CF 3 CF 2 CF 2 B24 0 A426 PhS H Ph CF 3 CF 2 CF 2 B24 0 A427 PhSO H Ph CF 3 CF 2 CF B24 0 A428 PhSO 2 H Ph CF 3 CF 2 CF 2 B24 0 Comp. R 2 R 3 R 4 Rs Qi P No. A429 CH 3 S H Ph C F 3 C F 2 C F 2 B24 0 A430 CH3SO H Ph CF 3 CF 2 CF 2 B24 0 A431 CF 3 H Ph C F 3 C F 2 C F 2 B24 0 A432 F 2 CH H Ph C F 3 C F C F 2 B24 0 A433 HCC H Ph C F 3 C F 2 C F 2 B24 0 A434 CH 3 CC H Ph CF 3 CF CF 2 B24 0 A435 CH 2 =CH H Ph CF 3 CF 2 CF B24 0 A436 CH 2 -=CHCH 2 H Ph CF 3 CF 2 CF 2 B24 0 A437 CH 3 SO 2 N(CH 3 ) H Ph CF 3 CF 2 CF 2 B24 0 A438 (CH 3 ) 2 N H Ph CF 3 CF 2 CF 2 B24 0 A439 (CH 3 ) 2 NSO 2 H Ph CF 3 CF 2 CF 2 B24 0 A440 CICH2 H Ph CF 3 CF 2 CF 2 B24 0 A441 CH3SCH2 H Ph C F 3 C F 2 C F 2 B24 0 A442 CH 3 SOCH 2 H Ph C F 3 C F 2 C F 2 B24 0 A443 CH 3 SO2CH2 H Ph CF3CF CF 2 B24 0 A444 H H Ph CF 2 CI B24 0 A445 CH 3 H Ph CF 2 CI B24 0 A446 CH3CH2 H Ph CF 2 CI B24 0 A447 cyclopropyl H Ph CF 2 CI B24 0 A448 (CH 3 ) 3 C H Ph CF 2 CI B24 0 A449 (CH 3 ) 2 CH H Ph CF 2 CI B24 0 A450 CH3(CH2) 2 H Ph CF 2 CI B24 0 A451 CH 3 OCH 2 H Ph CF 2 CI B24 0 A452 CH 3 O(CH 2 ) 2 H Ph CF 2 CI B24 0 A453 Ph H Ph CF 2 CI B24 0 A454 PhO H Ph CF 2 CI B24 0 A455 PhS H Ph CF 2 CI B24 0 A456 PhSO H Ph CF 2 CI B24 0 A457 PhSO 2 H Ph CF 2 CI B24 0 A458 CH 3 S H Ph CF 2 CI B24 0 A459 CH 3 SO H Ph CF 2 CI B24 0 A460 CF 3 H Ph CF 2 CI B24 0 Comp. R 2 R 3 R 4 Rs Qi P No. A461 F 2 CH H Ph CF 2 CI B24 0 A462 HCC H Ph CF 2 CI B24 0 A463 CH 3 CC H Ph CF 2 CI B24 0 A464 CH 2 =CH H Ph CF 2 CI B24 0 A465 CH 2 =CHCH 2 H Ph CF 2 CI B24 0 A466 CH 3 SO 2 N(CH 3 ) H Ph CF 2 CI B24 0 A467 (CH 3 ) 2 N H Ph CF 2 CI B24 0 A468 (CH 3 ) 2 NSO 2 H Ph CF 2 CI B24 0 A469 CICH 2 H Ph CF 2 CI B24 0 A470 CH 3 SCH 2 H Ph CF 2 CI B24 0 A471 CH 3 SOCH 2 H Ph CF 2 CI B24 0 A472 CH 3 SO 2 CH 2 H Ph CF 2 CI B24 0 A473 H H Ph CHF 2 B24 0 A474 CH 3 H Ph CHF 2 B24 0 A475 CH 3 CH 2 H Ph CHF 2 B24 0 A476 cyclopropyl H Ph CHF 2 B24 0 A477 (CH 3 ) 3 C H Ph CHF 2 B24 0 A478 (CH 3 ) 2 CH H Ph CHF 2 B24 0 A479 CH 3 (CH 2 ) 2 H Ph CHF 2 B24 0 A480 CH 3 OCH 2 H Ph CHF 2 B24 0 A481 CH 3 O(CH 2 ) 2 H Ph CHF 2 B24 0 A482 Ph H Ph CHF 2 B24 0 A483 PhO H Ph CHF 2 B24 0 A484 PhS H Ph CHF 2 B24 0 A485 PhSO H Ph CHF 2 B24 0 A486 PhSO 2 H Ph CHF 2 B24 0 A487 CH 3 S H Ph CHF 2 B24 0 A488 CH 3 SO H Ph CHF 2 B24 0 A489 CF 3 H Ph CHF 2 B24 0 A490 F 2 CH H Ph CHF 2 B24 0 A491 HCC H Ph CHF 2 B24 0 A492 CH 3 CC H Ph CHF 2 B24 0 Comp. R 2 R 3 R 4 Rs Qi P No. A493 CH 2 =CH H Ph CHF 2 B24 0 A494 CH =CHCH 2 H Ph CHF 2 B24 0 A495 CH 3 SO 2 N(CH 3 ) H Ph CHF 2 B24 0 A496 (CH 3 ) 2 N H Ph CHF 2 B24 0 A497 (CH 3 ) 2 NSO 2 H Ph CHF 2 B24 0 A498 CICH 2 H Ph CHF 2 B24 0 A499 CH 3 SCH 2 H Ph CHF 2 B24 0 A500 CH 3 SOCH 2 H Ph CHF 2 B24 0 A501 CH 3 SO 2 CH 2 H Ph CHF 2 B24 0 A504 CH 3 CH 2 H Ph CCI3 B24 0 A505 cyclopropyl H Ph CCI3 B24 0 A506 (CH 3 ) 3 C H Ph CCI3 B24 0 A507 (CH 3 ) 2 CH H Ph CCI3 B24 0 A508 CH 3 (CH 2 ) 2 H Ph CCI3 B24 0 A509 CH 3 OCH 2 H Ph CCI3 B24 0 A510 CH 3 O(CH 2 ) 2 H Ph CCI3 B24 0 A512 PhO H Ph CCI 3 B24 0 A518 CF 3 H Ph CCI 3 B24 0 A522 CH 2 =CH H Ph CCI3 B24 0 A523 CH 2 =CHCH H Ph CCI 3 B24 0 A524 CH 3 SO 2 N(CH 3 ) H Ph CCI 3 B24 0 Comp. R 2 R 3 R 4 Qi No. A525 (CH 3 ) 2 N H Ph CCI3 B24 0 A526 (CH 3 ) 2 NSO 2 H Ph CCI3 B24 0 A527 CICH 2 H Ph CCI 3 B24 0 A528 CH 3 SCH 2 H Ph CCI3 B24 0 A529 CH 3 SOCH . H Ph CCI3 B24 0 A530 CH 3 SO2CH2 H Ph CCI3 B24 0 A533 H cyclopropyl H CF3 B24 0 A534 H (CH 3 ) 3 CH H CF3 B24 0 A535 H (CH 3 ) 2 CH H CF3 B24 0 A536 H CH 3 (CH 2 ) 2 H CF3 B24 0 A538 H CH 3 O(CH 2 ) 2 H CF 3 B24 0 A539 H Ph H CF 3 B24 0 A540 H PhO H CF 3 B24 0 A541 H PhS H CF 3 B24 0 A542 H PhSO H CF 3 B24 0 A543 H PhSO 2 H CF 3 B24 0 A544 H CH 3 S H CF 3 B24 0 A545 H CH 3 SO H CF 3 B24 0 A546 H CF 3 H CF 3 B24 0 A547 H F 2 CH H CF 3 B24 0 A548 H HCC H CF 3 B24 0 A549 H CH 3 CC H CF 3 B24 0 A550 H CH 2 =CH H CF 3 B24 0 A551 H CH 2 =CHCH 2 H CF 3 B24 0 A552 H CH 3 S0 2 N(CH 3 ) H CF 3 B24 0 A553 H (CH 3 ) 2 N H CF 3 B24 0 A554 H (CH 3 ) NSO2 H CF 3 B24 0 A556 H CH 3 SOCH 2 H CF 3 B24 0 Comp. R 2 R 3 R 4 Rs Qi P No. A557 H CH3SO2CH2 H CF 3 B24 0 A558 H CH 3 H CF 3 CF 2 B24 0 A559 H CH 3 CH2 H CF 3 CF 2 B24 0 A560 H cyclopropyl H CF 3 CF 2 B24 0 A561 H (CH 3 ) 3 C H CF 3 CF 2 B24 0 A562 H (CH 3 ) 2 CH H CF3CF2 B24 0 A563 H CHs(CH 2 ) 2 H CF3CF2 B24 0 A564 H CH 3 OCH 2 H CF3CF2 B24 0 A565 H CH 3 O(CH 2 ) 2 H CF3CF2 B24 0 A566 H Ph H CF 3 CF 2 B24 0 A567 H PhO H CF 3 CF 2 B24 0 A568 H PhS H CF 3 CF 2 B24 0 A569 H PhSO H CF 3 CF 2 B24 0 A570 H PhSO 2 H CF 3 CF 2 B24 0 A571 H CH 3 S H CF 3 CF 2 B24 0 A572 H CH 3 SO H CF 3 CF 2 B24 0 A573 H CF 3 H CF 3 CF 2 B24 0 A574 H F 2 CH H CF 3 CF 2 B24 0 A575 H HCC H CF 3 CF 2 B24 0 A576 H CH 3 CC H CF 3 CF 2 B24 0 A577 H CH 2 =CH H CF 3 CF 2 B24 0 A578 H CH 2 =CHCH 2 H CF 3 CF 2 B24 0 A579 H CH 3 S0 2 N(CH 3 ) H CF 3 CF 2 B24 0 A580 H (CH 3 ) 2 N H CF 3 CF 2 B24 0 A581 H (CH 3 ) 2 NSO 2 H CF 3 CF 2 B24 0 A582 H CHsSCH 2 H CF 3 CF 2 B24 0 A583 H CH 3 SOCH 2 H CF 3 CF 2 B24 0 A584 H CHsSO CH 2 H CF 3 CF 2 B24 0 A585 H CH 3 H CF 3 CF 2 CF 2 B24 0 A586 H CHsCH 2 H CF 3 CF 2 C 2 B24 0 A587 H cyclopropyl H CFsCF 2 CF 2 B24 0 A588 H (CH 3 ) 3 C H CF 3 CF 2 CF 2 B24 0 Comp. R 2 R 3 R 4 Rs Qi P No. A589 H (CH 3 ) 2 CH H CFsCF 2 CF 2 B24 0 A590 H CHs(CH 2 ) 2 H CF3CF 2 CF 2 B24 0 A591 H CH 3 OCH 2 H CF3CF 2 CF B24 0 A592 H CH 3 O(CH 2 ) 2 H C F3C F 2 C F 2 B24 0 A593 H Ph H CF 3 CF 2 CF 2 B24 0 A594 H PhO H CF 3 CF 2 CF 2 B24 0 A595 H PhS H O F 3 C F 2 C F 2 B24 0 A596 H PhSO H C F 3 0 F C F 2 B24 0 A597 H PhSO 2 H CF 3 CF 2 CF B24 0 A598 H CH 3 S H CFsCF 2 CF 2 B24 0 A599 H CH 3 SO H CF 3 CF 2 CF 2 B24 0 A600 H CF 3 H C F 3 C F C F2 B24 0 A601 H F 2 CH H CF 3 CF2CF2 B24 0 A602 H HCC H CF 3 CF CF2 B24 0 A603 H CH 3 CC H CF 3 CF2CF2 B24 0 A604 H CH 2 =CH H CF3CF2CF2 B24 0 A605 H CH 2 =CHCH 2 H C F 3 C F2C F2 B24 0 A606 H CH 3 S0 2 N(CH 3 ) H CF 3 CF2CF 2 B24 0 A607 H (CH 3 ) 2 N H C 3 F C F 2 B24 0 A608 H (CH 3 ) 2 NSO 2 H C F 3 C F 2 C F 2 B24 0 A609 H CHsSCH 2 H C 3CF 2 CF 2 B24 0 A610 H CH 3 SOCH 2 H CF3CF 2 CF 2 B24 0 A611 H CH 3 SO2CH 2 H C F 3 C F 2 C F B24 0 A612 H CH 3 H CF 2 CI B24 0 A613 H CHsCH H CF 2 CI B24 0 A614 H cyclopropyl H CF 2 CI B24 0 A615 H (CH 3 ) 3 C H CF 2 CI B24 0 A616 H (CH 3 ) 2 CH H CF 2 CI B24 0 A617 H CH 3 (CH 2 ) 2 H CF 2 CI B24 0 A618 H CH 3 OCH 2 H CF 2 CI B24 0 A619 H CH 3 O(CH 2 ) 2 H CF 2 CI B24 0 A620 H Ph H CF 2 CI B24 0 Comp. R 2 R 3 R 4 Rs Qi P No. A621 H PhO H CF 2 CI B24 0 A622 H PhS H CF 2 CI B24 0 A623 H PhSO H CF 2 CI B24 0 A624 H PhSO 2 H CF 2 CI B24 0 A625 H CH 3 S H CF 2 CI B24 0 A626 H CH 3 SO H CF 2 CI B24 0 A627 H CF 3 H CF 2 CI B24 0 A628 H F 2 CH H CF 2 CI B24 0 A629 H HCC H CF 2 CI B24 0 A630 H CH 3 CC H CF 2 CI B24 0 A631 H CH 2 =CH H CF 2 CI B24 0 A632 H CH 2 =CHCH 2 H CF 2 CI B24 0 A633 H CH 3 S0 2 N(CH 3 ) H CF 2 CI B24 0 A634 H (CH 3 ) 2 N H CF 2 CI B24 0 A635 H (CH 3 ) 2 NSO 2 H CF 2 CI B24 0 A636 H CH 3 SCH2 H CF 2 CI B24 0 A637 H CH 3 SOCH 2 H CF 2 CI B24 0 A638 H CH 3 Sθ2CH2 H CF 2 CI B24 0 A639 H CH 3 H CHF 2 B24 0 A641 H cyclopropyl H CHF 2 B24 0 A642 H (CH 3 ) 3 C H CHF 2 B24 0 A643 H (CH 3 ) 2 CH H CHF 2 B24 0 A644 H CH 3 (CH2)2 H CHF 2 B24 0 A645 H CH3OCH2 H CHF 2 B24 0 A646 H CH 3 O(CH 2 ) 2 H CHF 2 B24 0 A647 H Ph H CHF 2 B24 0 A648 H PhO H CHF 2 B24 0 A649 H PhS H CHF 2 B24 0 A650 H PhSO H CHF 2 B24 0 A651 H PhSO 2 H CHF 2 B24 0 A652 H CH 3 S H CHF 2 B24 0 Comp. R 2 R 3 R 4 Rs Qi p No. A653 H CHgSO H CHF 2 B24 0 A654 H CF 3 H CHF 2 B24 0 A655 H F 2 CH H CHF 2 B24 0 A656 H HCC H CHF 2 B24 0 A657 H CH 3 CC H CHF 2 B24 0 A658 H CH 2 =CH H CHF 2 B24 0 A659 H CH 2 =CHCH 2 H CHF 2 B24 0 A660 H CH 3 S0 2 N(CH 3 ) H CHF 2 B24 0 A661 H (CH 3 ) 2 N H CHF 2 B24 0 A662 H (CH 3 ) 2 NSO 2 H CHF 2 B24 0 A663 H CH 3 SCH 2 H CHF 2 B24 0 A664 H CH 3 SOCH 2 H CHF 2 B24 0 A665 H CHsSO 2 CH 2 H CHF 2 B24 0 A668 H cyclopropyl H CCI 3 B24 0 A669 H (CH 3 ) 3 C H CCI 3 B24 0 A670 H (CH 3 ) 2 CH H CCI 3 B24 0 A671 H CH 3 (CH 2 ) 2 H CCI 3 B24 0 A672 H CH 3 OCH 2 H CCI 3 B24 0 A673 H CH 3 O(CH 2 ) 2 H CCI 3 B24 0 A676 H PhS H CCI 3 B24 0 A677 H PhSO H CCI 3 B24 0 A678 H PhSO 2 H CCI 3 B24 0 A679 H CH 3 S H CCI 3 B24 0 A681 H CF 3 H CCI 3 B24 0 A682 H F 2 CH H CCI 3 B24 0 A683 H HCC H CCI 3 B24 0 A684 H CH 3 CC H CCI 3 B24 0 Comp. R 2 R 3 R 4 Rs Qi P No. A687 H CH 3 S0 2 N(CH 3 ) H CCIg B24 0 A688 H (CHg) 2 N H CCIg B24 0 A689 H (CH 3 ) 2 NSO 2 H CCIg B24 0 A690 H CH3SCH2 H CCIg B24 0 A691 H CH3SOCH2 H CCIg B24 0 A692 H CH3SO2CH2 H CCIg B24 0 A694 H CH 3 CH 2 CHg CFg B24 0 A695 H cyclopropyl CH 3 CFg B24 0 A696 H (CH 3 ) 3 C CH 3 CFg B24 0 A697 H (CH 3 ) 2 CH CH 3 CFg B24 0 A698 H CH 3 (CH2)2 CH 3 CF 3 B24 0 A699 H CH 3 OCH 2 CH 3 CF 3 B24 0 A700 H CH 3 O(CH 2 ) 2 CH 3 CF 3 B24 0 A701 H Ph CH 3 CF 3 B24 0 A702 H PhO CH 3 CF 3 B24 0 A703 H PhS CH 3 CF 3 B24 0 A704 H PhSO CH 3 CF 3 B24 0 A705 H PhSO 2 CH 3 CF 3 B24 0 A707 H CHgSO CH 3 CFg B24 0 A711 H CHgCC CHg CF3 B24 0 A712 H CH 2 =CH CHg CF 3 B24 0 A714 H CH 3 S0 2 N(CH 3 ) CHg CF 3 B24 0 A715 H (CH 3 ) 2 N CHg CF 3 B24 0 A716 H (CH 3 ) NSO2 CHg CFg B24 0 Comp. R 2 R 3 R 4 Rs Qi P No. A717 H CHgSCH2 CH 3 CF 3 B24 0 A718 H CH3SOCH2 CH 3 CF 3 B24 0 A719 H CH3SO2CH2 CH 3 CF 3 B24 0 A720 H CH3 CH 3 CF 3 CF 2 B24 0 A721 H CH3CH2 CH 3 CF 3 CF 2 B24 0 A722 H cyclopropyl CH 3 CF3CF2 B24 0 A723 H (CHg)gC CH 3 CF3CF 2 B24 0 A724 H (CHg) 2 CH CH 3 CF3CF 2 B24 0 A725 H CH (CH2)2 CHg CF3CF 2 B24 0 A726 H CH3OCH2 CHg CF 3 CF 2 B24 0 A727 H CH 3 O(CH 2 ) 2 CHg CF 3 CF 2 B24 0 A729 H PhO CHg CF 3 CF 2 B24 0 A730 H PhS CHg CF 3 CF 2 B24 0 A731 H PhSO CHg CF 3 CF 2 B24 0 A732 H PhSO 2 CH 3 CF 3 CF 2 B24 0 A733 H CH 3 S CHg CF 3 CF 2 B24 0 A734 H CH 3 SO CHg CF 3 CF 2 B24 0 A735 H CF 3 CHg CF 3 CF 2 B24 0 A736 H F 2 CH CHg CF 3 CF 2 B24 0 A737 H HCC CHg CF 3 CF 2 B24 0 A738 H CH 3 CC CH 3 CF 3 CF 2 B24 0 A739 H CH 2 =CH CH 3 CF 3 CF 2 B24 0 A741 H CH 3 S0 2 N(CH 3 ) CH 3 CF 3 CF 2 B24 0 A742 H (CH 3 ) 2 N CH 3 CF 3 CF 2 B24 0 A743 H (CHg) 2 NSO2 CH 3 CF 3 CF 2 B24 0 A744 H CHgSCH 2 CH 3 CF 3 CF 2 B24 0 A745 H CH3SOCH2 CH 3 CF 3 CF 2 B24 0 A746 H CH3SO2CH2 CH 3 CF 3 CF 2 B24 0 A747 H CH 3 CH 3 CFgCF 2 CF 2 B24 0 A748 H CH3CH2 CH 3 CFgCF 2 CF 2 B24 0 Comp. R 2 R 3 R 4 Rs Qi P No. A749 H cyclopropyl CH 3 CF 3 CF2CF2 B24 0 A750 H (CH 3 ) 3 C CH 3 C F 3 C F 2 C F 2 B24 0 A751 H (CH 3 ) 2 CH CH 3 CF 3 CF 2 CF 2 B24 0 A752 H CH 3 (CH2)2 CH 3 CF 3 CF CF 2 B24 0 A753 H CH 3 OCH 2 CH 3 C F 3 C F 2 C F 2 B24 0 A754 H CH 3 O(CH 2 ) 2 CH 3 CF 3 CF 2 CF2 B24 0 A755 H Ph CH 3 C F3C F 2 C F 2 B24 0 A756 H PhO CH 3 CF 3 CF2CF B24 0 A757 H PhS CH 3 CF 3 CF2CF2 B24 0 A758 H PhSO CH 3 C F 3 C F2C B24 0 A759 H PhSO 2 CH 3 CF3CF2CF2 B24 0 A760 H CH 3 S CH 3 C F3C F 2 C F2 B24 0 A761 H CH 3 SO CH 3 CF3CF2CF2 B24 0 A762 H CF 3 CH 3 CF 3 CF2CF2 B24 0 A763 H F 2 CH CH 3 CF3CF2CF2 B24 0 A764 H HCC CH 3 CF3CF2CF2 B24 0 A765 H CH 3 CC CH 3 CF3CF2CF2 B24 0 A766 H CH 2 =CH CH 3 CF 3 CF2CF2 B24 0 A767 H CH 3 CF3CF2CF2 B24 0 A768 H CH 3 S0 2 N(CH 3 ) CH 3 CF 3 CF2CF2 B24 0 A769 H (CH 3 ) 2 N CH 3 C F 3 C F2C F2 B24 0 A770 H (CH 3 ) 2 NSO 2 CH 3 C F 3 C 2C F2 B24 0 A771 H CH 3 SCH2 CH 3 CF 3 CF2CF2 B24 0 A772 H CH 3 SOCH 2 CH 3 C F 3 C F 2 C F2 B24 0 A773 H CH 3 SO2CH2 CH 3 CF 3 CF2CF2 B24 0 A774 H CH 3 CH 3 CF 2 CI B24 0 A775 H CH3CH2 CH 3 CF 2 CI B24 0 A776 H cyclopropyl CH 3 CF 2 CI B24 0 A777 H (CH 3 ) 3 C CH 3 CF 2 CI B24 0 A778 H (CH 3 ) 2 CH CH 3 CF 2 CI B24 0 A779 H CH3(CH2)2 CH 3 CF 2 CI B24 0 A780 H CH3OCH2 CH 3 CF 2 CI B24 0 Comp. R 2 R 3 R 4 Rs Qi P No. A781 H CH 3 O(CH 2 ) 2 CH 3 CF 2 CI B24 0 A782 H Ph CH 3 CF 2 CI B24 0 A783 H PhO CH 3 CF 2 CI B24 0 A784 H PhS CH 3 CF 2 CI B24 0 A785 H PhSO CH 3 CF 2 CI B24 0 A786 H PhSO 2 CH 3 CF 2 CI B24 0 A787 H CH 3 S CH 3 CF 2 CI B24 0 A788 H CH 3 SO CH 3 CF 2 CI B24 0 A789 H CF 3 CH 3 CF 2 CI B24 0 A790 H F 2 CH CH 3 CF 2 CI B24 0 A791 H HCC CH 3 CF 2 CI B24 0 A792 H CH 3 CC CH 3 CF 2 CI B24 0 A793 H CH 2 =CH CH 3 CF 2 CI B24 0 A794 H CH 2 =CHCH 2 CH 3 CF 2 CI B24 0 A795 H CH 3 S0 2 N(CH 3 ) CH 3 CF 2 CI B24 0 A796 H (CH 3 ) 2 N CH 3 CF 2 CI B24 0 A797 H (CH 3 ) 2 NSO 2 CH 3 CF 2 CI B24 0 A798 H CH 3 SCH CHg CF 2 CI B24 0 A799 H CH 3 SOCH 2 CHg CF 2 CI B24 0 A800 H CH 3 SO2CH2 CHg CF 2 CI B24 0 A801 H CH 3 CH 3 CHF 2 B24 0 A802 H CH 3 CH2 CH 3 CHF 2 B24 0 A803 H cyclopropyl CHg CHF 2 B24 0 A804 H (CH 3 ) 3 C CH 3 CHF 2 B24 0 A805 H (CH 3 ) 2 CH CHg CHF 2 B24 0 A806 H CH 3 (CH2)2 CHg CHF 2 B24 0 A807 H CH 3 OCH 2 CHg CHF 2 B24 0 A808 H CH 3 O(CH 2 ) 2 CHg CHF 2 B24 0 Comp. R 2 R 3 R 4 Rs Qi P No. A813 H PhSO 2 CH 3 CHF 2 B24 0 A814 H CH 3 S CH 3 CHF 2 B24 0 A815 H CH 3 SO CH 3 CHF 2 B24 0 A817 H F 2 CH CH 3 CHF 2 B24 0 A818 H HCC CH 3 CHF 2 B24 0 A819 H CHgCC CHg CHF 2 B24 0 A821 H CH 2 =CHCH 2 CHg CHF 2 B24 0 A822 H CH 3 S0 2 N(CH 3 ) CH 3 CHF 2 B24 0 A823 H (CHg) 2 N CH 3 CHF 2 B24 0 A824 H (CH 3 ) 2 NSO 2 CH 3 CHF 2 B24 0 A825 H CHgSCH 2 CH 3 CHF 2 B24 0 A826 H CH 3 SOCH 2 CHg CHF 2 B24 0 A827 H CH 3 SO CH 2 CHg CHF 2 B24 0 A829 H CH 3 CH 2 CHg CCI 3 B24 0 A830 H cyclopropyl CHg CCI 3 B24 0 A831 H (CHg)gC CH 3 CCI 3 B24 0 A832 H (CH 3 ) 2 CH CH 3 CCI 3 B24 0 A833 H CH 3 (CH 2 ) 2 CH 3 CCI 3 B24 0 A834 H CH 3 OCH 2 CH 3 CCI3 B24 0 A835 H CH 3 O(CH 2 ) 2 CH 3 CCI 3 B24 0 A837 H PhO CH 3 CCI 3 B24 0 A838 H PhS CH 3 CCI 3 B24 0 A839 H PhSO CH 3 CCI 3 B24 0 A840 H PhSO 2 CH 3 CCI 3 B24 0 A841 H CH 3 S CH 3 CCI 3 B24 0 A842 H CH 3 SO CH 3 CCI 3 B24 0 A843 H CF 3 CH 3 CCI 3 B24 0 A844 H F 2 CH CH 3 CCI 3 B24 0 Comp. R 2 R 3 R 4 Rs Qi P No. A846 H CHgCC CH 3 CCI3 B24 0 A847 H CH 2 =CH CH 3 CCI3 B24 0 A849 H CH 3 S0 2 N(CH 3 ) CH 3 CCI 3 B24 0 A850 H (CH 3 ) 2 N CH 3 CCI 3 B24 0 A851 H (CHg) 2 NSO2 CH 3 CCI 3 B24 0 A852 H CH SCH2 CH 3 CCI 3 B24 0 A853 H CH3SOCH2 CH 3 CCI3 B24 0 A854 H CH 3 SO 2 CH 2 CH 3 CCI 3 B24 0 A855 H CH 3 Ph CF 3 B24 0 A857 H (CHg) 2 CH Ph CF 3 B24 0 A858 H (CH 3 ) 2 CH Ph CF 3 B24 0 A859 H cyclopropyl Ph CF 3 B24 0 A860 H CHg(CH2)2 Ph CF 3 B24 0 A861 H CH3OCH2 Ph CF 3 B24 0 A862 H CH 3 O(CH 2 ) 2 Ph CF 3 B24 0 A863 H Ph Ph CF 3 B24 0 A864 H PhO Ph CF 3 B24 0 A865 H PhS Ph CF 3 B24 0 A866 H PhSO Ph CF 3 B24 0 A867 H PhSO 2 Ph CF 3 B24 0 A868 H CH 3 S Ph CF 3 B24 0 A869 H CH 3 SO Ph CF 3 B24 0 A870 H CF 3 Ph CF 3 B24 0 A871 H F 2 CH Ph CF 3 B24 0 A872 H HCC Ph CF 3 B24 0 A873 H CH 3 CC Ph CF 3 B24 0 A874 H CH 2 =CH Ph CF 3 B24 0 A876 H CH 3 S0 2 N(CH 3 ) Ph CF 3 B24 0 Comp. R 2 R 3 R 4 Rs Qi P No. A877 H (CH 3 ) 2 N Ph CFg B24 0 A878 H (CH 3 ) 2 NSO 2 Ph CF 3 B24 0 A879 H CH 3 SCH2 Ph CFg B24 0 A880 H CH 3 SOCH 2 Ph CFg B24 0 A881 H CH 3 SO 2 CH 2 Ph CFg B24 0 A882 H CHg Ph CFgCF 2 B24 0 A883 H CH 3 CH 2 Ph CF 3 CF 2 B24 0 A884 H cyclopropyl Ph CF 3 CF 2 B24 0 A885 H (CH 3 ) 3 C Ph CF 3 CF 2 B24 0 A886 H (CH 3 ) 2 CH Ph CFgCF 2 B24 0 A887 H CH 3 (CH 2 )2 Ph CFgCF 2 B24 0 A888 H CH 3 OCH 2 Ph CFgCF 2 B24 0 A889 H CH 3 O(CH 2 ) Ph CFgCF 2 B24 0 A892 H PhS Ph CF 3 CF 2 B24 0 A893 H PhSO Ph CF 3 CF 2 B24 0 A894 H PhSO 2 Ph CF 3 CF 2 B24 0 A895 H CHgS Ph CF 3 CF2 B24 0 A896 H CH 3 SO Ph CF 3 CF2 B24 0 A898 H F 2 CH Ph CF 3 CF2 B24 0 A900 H CHgCC Ph CF 3 CF2 B24 0 A901 H CH 2 =CH Ph CF 3 CF 2 B24 0 A903 H CH 3 S0 2 N(CH 3 ) Ph CF 3 CF2 B24 0 A904 H (CH 3 ) 2 N Ph CF 3 CF2 B24 0 A905 H (CH 3 ) 2 NSO 2 Ph CF 3 CF 2 B24 0 A906 H CH 3 SCH 2 Ph CF 3 CF 2 B24 0 A907 H CH 3 SOCH 2 Ph CF 3 CF 2 B24 0 A908 H CHgS0 CH 2 Ph CF 3 CF 2 B24 0 CO CO CO CO CO CO CO CO CO CO CO CO CO CO CO CO CO CO CO CO CO CO CO CD CO CO CD CO CO CO CO CD - -5 ^ ω ω ω ω ω ω co ω ω ω ro r ro r ro ro o ro ro ro - j . - j . - » . - i - j . -^ -' -' -^ - j . o 3 o o oo - i θ3 en *>. co ro --»- o co oo -sg Λ en *. co ro -»- θ sθ oo ~i φ en Φ' Cύ ro -^ o co TO x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x x X TJ TJ TJ TJ TJ TJ TJ TJ TJ TJ TJ TJ TJ TJ TJ TJ T TJ TJ TJ TJ TJ TJ TJ TJ TJ TJ TJ TJ __r _x __r __r __r _r :_r zr zr zr zr __r __r zr __r zr zr rx zr zr zr zr IT IX __T _ zr X o o TI oTI oTI oTI o o .oτι oτι oτι o o o o o o o o o o o o O O O O O τι τι τι .TI TI TI TI TI o o o o o ω T| Tl TI Tl Tl O O O O O O O O O O O O O O O O O O O O O I TjI rToI rToI o O TI I o Tl o o o o o r ToI rTI rToI rTo -ToI rToI rToI rToI rToI rToI rToI rToI rToI rToI rTI r-oΠ rTI rToI Tl o TI o o Tl ro ro ro ro ro ro O O O O O O O O O O O O O O O O O O O O O τ o TI o oι fτι rτι rτoι rτoι rτoι rτoι rτoι rτoι rτoι rτoι r-on rτoι rτoι rτoι r-oπ rτoι rτoι rτoι τι o o ro rτoι ro Tl T| o Tl o Tl r τoι ro ro ro ro CD C0 CD O0 CD O3 O3 O0 O0 O0 O0 OT 00 00 O3 O0 O0 00 O0 O0 C_O C0 O0 O0 00 00 CD 00 00 CO 00 00 ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro _fc_. _li. .fc_. _fc> _fc-. -fc_. -fc_. .p_- i. _P_. Ji. ro ro ro ro ro 4-» 45- 4. . 4*. ** *» _tS_ -t _!_- _ . -t- _r-. o 4. *- .&- *. 4*> . o o o o o o o o o o o o o o o o o o o o Comp. R 2 R 3 R 4 Rs Qi P No. A941 H CH 3 (CH 2 ) 2 Ph CF 2 CI B24 0 A942 H CH 3 OCH 2 Ph CF 2 CI B24 0 A943 H CH 3 O(CH 2 ) 2 Ph CF 2 CI B24 0 A944 H Ph Ph CF 2 CI B24 0 A945 H PhO Ph CF 2 CI B24 0 A946 H PhS Ph CF 2 CI B24 0 A947 H PhSO Ph CF 2 CI B24 0 A948 H PhSO 2 Ph CF 2 CI B24 0 A949 H CH 3 S Ph CF 2 CI B24 0 A950 H CH 3 SO Ph CF 2 CI B24 0 A952 H F 2 CH Ph CF 2 CI B24 0 A953 H HCC Ph CF 2 CI B24 0 A954 H CHgCC Ph CF 2 CI B24 0 A955 H CH 2 =CH Ph CF 2 CI B24 0 A956 H CH2=CHCH2 Ph CF 2 CI B24 0 A957 H CH 3 S0 2 N(CH 3 ) Ph CF 2 CI B24 0 A958 H (CH 3 ) 2 N Ph CF 2 CI B24 0 A959 H (CH 3 ) 2 NSO 2 Ph CF 2 CI B24 0 A960 H CHgSCH2 Ph CF 2 CI B24 0 A961 H CH3SOCH2 Ph CF 2 CI B24 0 A962 H CH3SO2CH2 Ph CF 2 CI B24 0 A963 H CH 3 Ph CHF 2 B24 0 A964 H CH 3 CH2 Ph CHF 2 B24 0 A965 H (CH 3 ) 3 C Ph CHF 2 B24 0 A966 H (CH 3 ) 2 CH Ph CHF 2 B24 0 A967 H cyclopropyl Ph CHF 2 B24 0 A968 H CH 3 (CH2)2 Ph CHF 2 B24 0 A969 H CH 3 OCH 2 Ph CHF 2 B24 0 A970 H CH 3 O(CH 2 ) 2 Ph CHF 2 B24 0 A971 H Ph Ph CHF 2 B24 0 A972 H PhO Ph CHF 2 B24 0 Comp. R 2 R 3 R 4 Rs Qi P No. A973 H PhS Ph CHF 2 B24 0 A974 H PhSO Ph CHF 2 B24 0 A975 H PhSO 2 Ph CHF 2 B24 0 A976 H CH 3 S Ph CHF 2 B24 0 A977 H CH 3 SO Ph CHF 2 B24 0 A979 H F 2 CH Ph CHF 2 B24 0 A980 H HCC Ph CHF 2 B24 0 A981 H CHgCC Ph CHF 2 B24 0 A982 H CH 2 =CH Ph CHF 2 B24 0 A984 H CH 3 S0 2 N(CH 3 ) Ph CHF 2 B24 0 A985 H (CH 3 ) 2 N Ph CHF 2 B24 0 A986 H (CH 3 ) 2 NSO 2 Ph CHF 2 B24 0 A987 H CH3SCH2 Ph CHF 2 B24 0 A988 H CH3SOCH2 Ph CHF 2 B24 0 A989 H CH3SO2CH2 Ph CHF 2 B24 0 A991 H CHgCH2 Ph CCIg B24 0 A992 H (CHg)gC Ph CCIg B24 0 A993 H (CHg) 2 CH Ph CCIg B24 0 A994 H cyclopropyl Ph CCIg B24 0 A995 H CHg(CH 2 ) 2 Ph CCIg B24 0 A996 H CH 3 OCH 2 Ph CCI3 B24 0 A997 H CH 3 0(CH 2 ) 2 Ph CCI3 B24 0 A1002 H PhS0 2 Ph CCIg B24 0 A1004 H CHgSO Ph CCI3 B24 0 Comp. R 2 R 3 R 4 R 5 Qi P No. A1005 H CF 3 Ph CCI 3 B24 0 A1006 H F 2 CH Ph CCI 3 B24 0 A1007 H HCC Ph CCI 3 B24 0 A1008 H CH 3 CC Ph CCI 3 B24 0 A1009 H CH 2 =CH Ph CCI 3 B24 0 A1011 H CH 3 S0 2 N(CH 3 ) Ph CCI 3 B24 0 A1012 H (CH 3 ) 2 N Ph CCI 3 B24 0 A1013 H (CH 3 ) 2 NS0 2 Ph CCI 3 B24 0 A1014 H CH 3 SCH2 Ph CCI3 B24 0 A1015 H CH 3 SOCH 2 Ph CCIg B24 0 A1016 H CH 3 Sθ2CH2 Ph CCIg B24 0 A1018 Cl H H CF 3 B24 0 A1020 NC H H CF 3 B24 0 A1021 CH 3 S0 2 0 H H CF 3 B24 0 A1023 CH 3 CH 2 0 H H CFg B24 0 A1024 CH 2 CH=CH 2 0 H H CFg B24 0 A1025 HCCCH 2 0 H H CFg B24 0 A1027 PhCH 2 S0 2 H H CF 3 B24 0 A1028 CICH 2 CH 2 H H CF 3 B24 0 A1029 BrCH 2 H H CF 3 B24 0 A1030 FCH 2 H H CF 3 B24 0 A1031 CHF2CH2 H H CF 3 B24 0 A1032 CF CH2 H H CF 3 B24 0 A1033 [1 ,3]-imidazol-1- H H CF 3 B24 0 ylmethyl A1034 CHCI2CH2 H H CF 3 B24 0 A1035 CICH=CH H H CF 3 B24 0 Comp. R 2 R 3 R 4 Rs Qi P No. A1036 CI 2 C=CH H H CF 3 B24 0 A1037 CF 3 CH=CH H H CF 3 B24 0 A1038 CICC H H CF 3 B24 0 A1040 CH 3 CH 2 CH 3 H CFg B24 0 A1048 H Br H CF 3 B24 0 A1049 H OH H CF 3 B24 0 A1050 H OCH 3 H CF 3 B24 0 A1051 H OCHF 2 H CF 3 B24 0 A1052 H OS0 2 CH 3 H CF 3 B24 0 A1053 H OS0 2 CF 3 H CF 3 B24 0 A1054 H CICH 2 H CF 3 B24 0 A1057 H CHF 2 CH 2 H CFg B24 0 A1059 H triazolylmethyl H CFg B24 0 A1060 H CHCI 2 CH 2 H CFg B24 0 A1061 H CICH=CH H CFg B24 0 A1062 H CI 2 C=CH H CFg B24 0 A1063 H CF 3 CH=CH H CFg B24 0 A1065 H CH 3 C(0) H CFg B24 0 A1066 H Ph H CF 3 B24 0 A1067 H S0 2 CH 3 H CF 3 B24 0 Comp. R 2 R 3 R 4 Rs Qi P No. A1068 H S0 2 CF 3 H CF 3 B24 0 A1075 CH 3 H CH 3 0 CF 3 B24 0 A1077 CH 3 H CH 3 SO CF 3 B24 0 A1078 CH 3 H CH 3 S0 2 CFg B24 0 A1079 CH 3 CH2θCH2 H H CFg B24 0 A1080 PhOCH 2 H H CFg B24 0 A1082 (CH 3 ) 2 CH 2 OCH 2 H H CF 3 B24 0 A1083 BrCH 2 CH 2 H H CFg B24 0 A1084 FCH 2 CH 2 H H CFg B24 0 Comp. R 3 R 5 Qi p No. A1091 cyclopropyl-CH 2 H H CFg B24 0 A1092 2,2-dichlorocycloprop- H H CF 3 B24 0 1-yl A1093 CH 3 OC(0)CH=CH H H CFg B24 0 A1094 CH 3 CH 2 OC(0)CH=CH H H CFg B24 0 A1095 CICH 2 CH=CH H H CFg 0 A1096 CH=C=CH H H CFg B24 0 A1097 (CHg) 2 NCH2 H H CFg B24 0 A1099 CH 3 C(0)OCH 2 H H CFg B24 0 A1100 PhC(0)OCH 2 H H CFg B24 0 A1101 PhCH 2 CH 2 H H CFg B24 0 A1102 CH 3 OC(0)CH 2 H H CFg B24 0 A1104 CH3(CH2) 7 SCH2 H H CFg B24 0 A1105 CH3(CH 2 ) 7 SOCH2 H H CFg B24 0 A1106 CH 3 (CH 2 ) 7 S0 2 CH2 H H CFg B24 0 A1108 CICH 2 CC H H CFg B24 0 A1109 CHF2CH 2 CH2 H H CFg B24 0 A1110 CHCI2CH2CH2 H H CFg B24 0 A1111 CF 3 S0 2 0 H H CFg B24 0 Comp. R 2 R 3 R 4 Rs Qi P No. A1116 " H H CF 3 B24 0 A1117 H H CF 3 B24 0 A1118 CH 3 ON=CHCH 2 H H CF 3 B24 0 A1119 0=CHCH 2 H H CF 3 B24 0 A1120 CH 3 CH 2 0CH 2 H H CF 2 CI B24 0 A1121 PhOCH 2 H H CF 2 CI B24 0 A1122 m' H H CF 2 CI B24 0 A1123 (CH 3 ) 2 CH 2 OCH 2 H H CF 2 CI B24 0 A1124 BrCH 2 H H CF 2 CI B24 0 A1125 FCH 2 H H CF 2 CI B24 0 A1129 ^0-^I^SCH, H H CF 2 CI B24 0 ^. A1132 cyclopropyl-CH 2 H H CF 2 CI B24 0 A1133 2,2-dichlorocycloprop- H H CF 2 CI B24 0 1-yl A1134 CH 3 OC(0)CH=CH H H CF 2 CI B24 0 A1135 CH 3 CH 2 OC(0)CH=CH H H CF 2 CI B24 0 Comp. R 2 R 4 Qi P No. A1136 CICH 2 CH=CH H H CF 2 CI B24 0 A1137 CH=C=CH H H CF 2 CI B24 0 A1138 (CH 3 ) 2 NCH 2 H H CF 2 CI B24 0 A1139 HOCH 2 H H CF 2 CI B24 0 A1140 CH 3 C(0)OCH 2 H H CF 2 CI B24 0 A1141 PhC(0)OCH 2 H H CF 2 CI B24 0 A1142 PhCH 2 H H CF 2 CI B24 0 A1143 CH 3 OC(0)CH 2 H H CF 2 CI B24 0 A1144 NCCH 2 H H CF 2 CI B24 0 A1145 CH 3 (CH2) 7 SCH2 H H CF 2 CI B24 0 A1146 CH 3 (CH 2 ) 7 SOCH 2 H H CF≥CI B24 0 A1147 CH 3 (CH 2 ) 7 S0 2 CH 2 H H CF 2 CI B24 0 A1149 H H CF 2 CI B24 0 A1150 H H CF 2 CI B24 0 A1151 H H CF 2 CI B24 0 A1152 H H CF 2 C! B24 0 A1158 CH- H H CF 2 CI B24 0 A1 159 CH 3 ON=CHCH 2 H H CF 2 CI B24 0 A1 160 0=CHCH 2 H H CF 2 CI B24 0 sO o o o o o o o o o o o o a. ■ st 'st "st 'st "st ■ st ■ st ■ st ■ st ■ st • < ■ « "st ■ st -st 'sf 'st 'st 'st 'st 'st ω σ CM ω CM CM CM CM CM CM CM CM CM CM CM CM CM CM CM CM CM CM CQ CQ CQ ω CQ CO ω CM CQ CQ CQ CQ ω CM ω CM CQ CQ CQ CQ CQ ω CQ CQ υ ft. X X X X X X X X X X X X X X x x x x x x x Li. Li. LL ιT u. LL __£ ■ u. LL LL ti- LL LL LL LL LL U- LL L o o o o o o O O o o o o o o o o o o o X X X X X X X X x x x x x x x CO oo DC X X X X X X X X x x x x x x x x Comp. R 3 R 4 R 5 Qi P No. A1183 PhCH 2 H H CF 2 H B24 0 A1184 CH 3 OC(0)CH 2 H H CF 2 H B24 0 A1185 NCCH 2 H H CF 2 H B24 0 A1186 CH 3 (CH 2 ) 7 SCH 2 H H CF 2 H B24 0 A1187 CH 3 (CH 2 ) 7 SOCH 2 H H CF 2 H B24 0 A1188 CH 3 (CH 2 ) 7 S0 2 CH 2 H H CF 2 H B24 0 A1190 H H CF 2 H B24 0 A1191 H H CF 2 H B24 0 A1192 H H CF 2 H B24 0 A1193 H H CF 2 H B24 0 A1199 ^CH, H H CF 2 H B24 0 A1200 CH 3 ON=CHCH 2 H H CF 2 H B24 0 A1201 0=CHCH 2 H H CF 2 H B24 0 A1202 CH 3 CH=CH H H CF 3 B24 0 A1203 CH 3 S0 2 NH H H CF 3 B24 0 A1204 CH 3 CH 2 CH 2 θ H CH 3 CF 3 B24 0 A1207 CH 3 CH 2 C(0)OCH 2 H H CFg B24 0 Comp. R 2 R 3 R 4 R 5 Qi P No. A1208 CH 3 CH 2 OC(0)OCH 2 H H CFg B24 0 A1209 CH 3 OCH 2 OCH 2 H H CFg B24 0 A1212 cyclopropyl H H CFg B24 1 A1213 CH (CH2)2 H H CFg B24 1 A1214 CH3OCH2 H H CFg B24 1 A1218 CH3SO2CH2 H H CF 3 B24 1 A1220 CHgCH2θCH2 H H CF 3 B24 1 A1221 PhOCH 2 H H CF 3 B24 1 A1222 (CH 3 ) 2 CH 2 OCH 2 H H CF 3 B24 1 A1223 BrCH 2 H H CF 3 B24 1 A1227 cyclopropyl-CH 2 H H CF 3 B24 1 A1228 2,2-dichlorocycloprop- H H CF 3 B24 1 1 -yl A1229 (CH 3 ) 2 NCH 2 H H CF 3 B24 1 A1230 HOCH 2 H H CF 3 B24 1 A1231 CH 3 C(0)OCH 2 H H CF 3 B24 1 A1232 PhC(0)OCH 2 H H CFg B24 1 A1234 CH 3 OC(0)CH 2 H H CFg B24 1 Comp. R 2 R 3 R 4 Rs Qi P No. A1236 CH 3 (CH 2 ) 7 S0 2 CH 2 H H CF 3 B24 1 A1237 Br H H CF 3 B24 1 A1238 Cl H H CF 3 B24 1 A1239 0=CHCH 2 H H CF 3 B24 1 A1241 CHgCH2 H H CF ≥ CI B24 1 A1242 cyclopropyl H H CF 2 CI B24 1 A1243 CHg(CH 2 ) 2 H H CF 2 CI B24 1 A1244 CH 3 OCH 2 H H CF 2 CI B24 1 A1246 F 2 CH H H CF 2 CI B24 1 A1247 CICH 2 H H CF 2 CI B24 1 A1248 CHgS0 2 CH 2 H H CF 2 CI B24 1 A1249 CHg CF 3 H CF 2 CI B24 1 A1250 CHgCH 2 OCH 2 H H CF 2 CI B24 1 A1251 PhOCH 2 H H CF 2 CI B24 1 A1252 (CH 3 ) 2 CH 2 OCH 2 H H CF 2 CI B24 1 A1253 BrCH 2 H H CF 2 CI B24 1 A1254 FCH 2 H H CF 2 CI B24 1 A1256 ^°^' ' S0 * CH * H H CF 2 CI B24 1 A1257 cyclopropyl-CH 2 H H CF 2 CI B24 1 A1258 2,2-dichlorocycloprop- H H CF 2 CI B24 1 1-yl A1259 (CHg) 2 NCH2 H H CF 2 CI B24 1 A1260 HOCH 2 H H CF 2 CI B24 1 A1261 CH 3 C(0)OCH 2 H H CF 2 CI B24 1 A1262 PhC(0)OCH 2 H H CF 2 CI B24 1 A1263 PhCH 2 H H CF 2 CI B24 1 Comp. R 2 R 3 Rs Qi P No. A1264 CH 3 OC(0)CH 2 H H CF 2 CI B24 1 A1265 NCCH 2 H H CF 2 CI B24 1 A1266 CH 3 (CH2)7S0 2 CH2 H H CF 2 CI B24 1 A1267 Br H H CF 2 CI B24 1 A1268 Cl H H CF 2 CI B24 1 A1269 0=CHCH 2 H H CF 2 CI B24 1 A1270 CH 3 H H CF 2 H B24 1 A1271 CH 3 CH2 H H CF 2 H B24 1 A1272 cyclopropyl H H CF 2 H B24 1 A1273 CHg(CH2)2 H H CF 2 H B24 1 A1274 CH30CH2 H H CF 2 H B24 1 A1276 F 2 CH H H CF 2 H B24 1 A1277 CICH 2 H H CF 2 H B24 1 A1278 CH3SO2CH2 H H CF 2 H B24 1 A1280 CHgCH2θCH 2 H H CF 2 H B24 1 A1281 PhOCH 2 H H CF 2 H B24 1 A1282 (CHg) 2 CH2θCH 2 H H CF 2 H B24 1 A1283 BrCH 2 H H CF 2 H B24 1 A1284 FCH 2 H H CF 2 H B24 1 A1287 cyclopropyl-CH 2 H H CF 2 H B24 1 A1288 2,2-dichlorocycloprop- H H CF 2 H B24 1 1-yl A1289 (CHg) 2 NCH 2 H H CF 2 H B24 1 A1290 HOCH 2 H H CF 2 H B24 1 A1291 CH 3 C(0)OCH 2 H H CF 2 H B24 1 > > > > > > > > > > > > > > > > > > > > > > > > > > > > > > > o ω oo co co co ω co CO CO CO CO CO OO CO CO OO ->■ -j. —-. — -. —-. —- —-. O O O ω eo oo ω ω ω CO ro ro ro ro ro ro ro ro ro ro ro -* -* -■• o o o o o o o CD CO CO CO O CO CO CD P ro ->• o co Φ -si CΛ cn 4^ co ro -»- o co oo -si CΛ -t*. co ro ->■ o CO 00 -si CΛ Φ CO ro T 3J X X X X X X X x x x x x x x x x x x x x x x x x x x x x x x 3 x x x x x x x x X o 9 9 o Ω o sj _9_, o -η o -η o -η o -p. o -η o -η o -^ o -y, TI TI 1 ro τι ' " -n o n > n Tl o o o Tl o Tl o o o o o o TI o T| ol o TI O *__ ro ro ro X τι X o τι X X X X X X X X W CD 03 CD CD CO CD 00 O3 00 O3 O3 vO O0 00 O0 0α θ3 00 CO CD Cα σ3 Cπ θ3 O3 CD O. O3 O3 O3 ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro ro _* _!__. _p__ _!_». 4i. t>. -t_. 4-. 4i. 4^ 4o. 4i. 4 *. *. 4*> ■&■ ro ro o 4-s 4_. _f4. _t_. _ 4a. o. 4i. *. s. o o o o o o o O O O O O ln the formulaic representations of the tables (for example Table 7, compound A 1088, substituent R 2 ), the linkage site with the pyridine ring is on the right-hand side of the formulaic representation. Terminal valencies are a methyl group. Table 8: Compounds of the formula lb (p is 0 or 1 ): Qi Qi Qi Qi Oi Qi Qi Qi Oi Qi Oi Oi B1 B2 B3 B4 B5 B6 B7 B8 B9 B10 B11 B12 B13 B14 B15 B16 B17 B18 B19 B20 B21 B22 B23 - B25 B26 B27 B28 B29 B30 B31 B32 B33 B34 B35 B36 B37 B38 B39 B40 B41 B42 B43 B44 B45 B46 B47 B48 B49 B50 B51 B52 B53 B54 B55 B56 B57 B58 B59 B60 B61 B62 B63 B64 B65 B66 B67 B68 B69 B70 B71 B72 B73 B74 B75 B76 B77 B78 B79 B80 B81 B82 B83 B84 B85 B86 B87 B88 B89 B90 B91 B92 B93 B94 B95 B96 B97 B98 B99 B100 B101 B102 B103 B104 B105 B106 B107 B108 B109 B110 B111 B112 B113 B114 B115 B116 B117 B118 B119 B20 B121 B122 B123 B124 B125 B126 B127 B128 B129 B130 B131 B132 B133 B134 B135 B136 B137 B138 B139 B140 B141 B142 B143 B144 B145 B146 B147 B148 B149 B150 B151 B152 B153 B154 B155 B156 B157 B158 B159 B160 B161 B162 B163 B164 B165 B166 B167 B168 B169 B170 B171 B172 B173 B174 B175 B176 B177 B178 B179 B180 B181 B182 B183 B184 B185 B186 B187 B188 B189 B190 B191 B192 B193 B194 B195 B196 B197 B198 B199 B200 B201 B202 B203 B204 B205 B206 B207 B208 B209 B210 B211 B212 B213 B214 B215 B216 B217 B218 B219 B220 B221 B222 B223 B224 B225 B226 B227 B228 B229 B230 B231 B232 B233 B234 B235 B236 B237 B238 B239 B240 B241 B242 B243 B244 B245 B246 B247 B248 B249 B250 B251 B252 B253 B254 B255 B256 B257 B258 B259 B260 B261 B262 B263 B264 B265 B266 B267 B268 B269 B270 B271 B272 B273 B274 B275 B276 B277 B278 B279 B280 B281 B282 B283 B284 B285 B286 B287 B288 B289 B290 B291 B292 B293 B294 B295 B296 B297 B298 B299 B300 Sl Sl dl Sl Sl fil fil fil δl Sl Sl Sl B301 B302 B303 B304 B305 B306 B307 B308 B309 B310 B311 B312 B313 B314 B315 B316 B317 B318 B319 B320 B321 B322 B323 B324 B325 B326 B327 B328 B329 B330 B331 B332 B333 B334 B335 B336 B337 B338 B339 B340 B341 B342 B343 B344 B345 B346 B347 B348 B349 B350 B351 B352 B353 B354 B355 B356 B357 B358 B359 B360 B361 B362 B363 B364 B365 B366 B367 B368 B369 B370 B371 B372 B373 B374 B375 B376 B377 B378 B379 B380 B381 B382 B383 B384 B385 B386 B387 B388 B389 B390 B391 B392 B393 B394 B395 B396 B397 B398 B399 B400 B401 B402 B403 B404 B405 B406 B407 B408 B409 B410 B411 B412 B413 B414 B415 B416 B417 B418 B419 B420 B421 B422 B423 B424 B425 B426 B427 B428 B429 B430 B431 B432 B433 B434 B435 B436 B437 B438 B439 B440 B441 B442 B443 B444 B445 B446 B447 B448 B449 B450 B451 B452 B453 B454 B455 B456 B457 B458 B459 B460 B461 B462 B463 B464 B465 B466 B467 B468 B469 B470 B471 B472 B473 B474 B475 B476 B477 B478 B479 B480 B481 B482 B483 B484 B485 B486 B487 B488 B489 B490 B491 B492 B493 B494 B495 B496 B497 B498 B499 B500 B501 B502 B503 B504 B505 B506 B507 B508 B509 B510 B511 B512 B513 B514 B515 B516 B517 B518 B519 B520 B521 B522 B523 B524 B525 B526 B527 B528 B529 B530 B531 B532 B533 B534 B535 B536 B537 B538 B539 B540 B541 B542 B543 B544 B545 B546 B547 B548 B549 B550 B551 B552 B553 B554 B555 B556 B557 B558 B559 B560 B561 B562 B563 B564 B565 B566 B567 B568 B569 B570 B571 B572 B573 B574 B575 B576 B577 B578 B579 B580 B581 B582 B583 B584 B585 B586 B587 B588 B589 B590 B591 B592 B593 B594 B595 B596 B597 B598 B599 B600 B601 B602 B603 B604 B605 B606 B607 B608 B609 B610 B611 B612 B613 B614 B615 B616 B617 B618 B619 B620 B621 B622 B623 B624 B625 B626 B627 B628 B629 B630 B631 B632 B633 B634 B635 B636 B637 B638 B639 B640 B641 B642 B643 B644 B645 B646 B647 B648 B649 B650 B651 B652 B653 B654 B655 B656 B657 B658 B659 B660 B661 B662 B663 B664 B665 B666 B667 B668 B669 B670 B671 B672 B773 B774 B775 B776 B777 B778 B779 B780 B781 B782 B783 B784 B785 B786 B787 B788 B789 B790 B791 B792 B793 B794 B795 B796 Ql Qi Ql Ql Ql Ql Qi Ql Ql Ql Ql Ql B797 B798 B799 B800 B801 B802 B803 B804 B805 B806 B807 B808 B809 B810 B811 B812 B813 B814 B815 B816 B817 B818 B819 B820 B821 B822 B823 B824 B825 B826 B827 B828 B829 B830 B831 B832 B833 B834 B835 B836 B837 B838 B839 B840 B841 B842 B843 B844 B845 B846 B847 B848 B849 B850 B851 B852 B853 B854 B855 B856 B857 B858 B859 B860 B861 B862 B863 B864 B865 B866 B867 B868 B869 B870 B871 B872 B873 B874 B875 B876 B877 B878 B879 B880 B881 B882 B883 B884 B885 B886 B887 B888 B889 B890 B891 B892 B893 B894 B895 B896 B897 B898 B899 B900 B901 B902 B903 B904 B905 B906 B907 B908 B909 B910 B911 B912 B913 B914 B915 B916 B917 B918 B919 B920 B921 B922 B923 B924 B925 B926 B927 B928 B929 B930 B931 B932 B933 B934 B935 B936 B937 B938 B939 B940 B941 B942 B943 B944 B945 B946 B947 B948 B949 B950 B951 B952 B953 B954 B955 B956 B957 B958 B959 B960 B961 B962 B963 B964 B965 B966 B967 B968 B969 B970 B971 B972 B973 B974 B975 B976 B977 B978 B979 B980 B981 B982 B983 B984 B985 B986 B987 B988 B989 B990 B991 B992 B993 B994 B995 B996 B997 B998 B999 B1000 B1001 B1002 B1003 B1004 B1005 B1006 B1007 B1008 B1009 B1010 B1011 B1012 B1013 B1014 B1015 B1016 B1017 B1018 B1019 B1020 B1021 B1022 B1023 B1024 B1025 B1026 B1027 B1028 B1029 B1030 B1031 B1032 B1033 B1034 B1035 B1036 B1037 B1038 B1039 B1040 B1041 B1042 B1043 B1044 B1045 B1046 B1047 B1048 B1049 B1050 B1051 B1052 B1053 B1054 B1055 B1056 B1057 B1058 B1059 B1060 B1061 B1062 B1063 B1064 B1065 B1066 B1067 B1068 B1069 B1070 B1071 B1072 B1073 B1074 B1075 B1076 B1077 B1078 B1079 B1080 B1081 B1082 B1083 B1084 B1085 B1086 B1087 B1088 B1089 B1090 B1091 B1092 B1093 B1094 B1095 B1096 B1097 B1098 B1099 B1100 B1101 B1102 B1103 B1104 B1105 B1106 B1107 B1108 B1109 B1110 B1111 B1112 B1113 B1114 B1115 B1116 B1117 B1118 B1119 B1120 B1121 B1122 B1123 B1124 B1125 B1126 B1127 B1128 B1129 B1130 B1131 B1132 B1133 B1134 B1135 B1136 B1137 B1138 B1139 B1140 B1141 B1142 B1143 B1144 B1145 B1146 B1147 B1148 B1149 B1150 B1151 B1152 B1153 B1154 B1155 B1156 B1157 B1158 B1159 B1160 B1161 B1162 B1163 B1164 B1165 B1166 B1167 B1168 B1169 B1170 B1171 B1172 B1173 B1174 B1175 B1176 B1177 B1178 B1179 B1180 B1181 B1182 B1183 B1184 B1185 B1186 B1187 B1188 B1189 B1190 B1191 B1192 Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi B1193 B1194 B1195 B1196 B1197 B1198 B1199 B1200 B1201 B1202 B1203 B1204 B1205 B1206 B1207 B1208 B1209 B1210 B1211 B1212 B1213 B1214 B1215 B1216 B1217 Table 9: Compounds of the formula lc (p is 0 or 1): Qi Qi Qi Qi Qi Qi Q i Qi Oi Qi Qi Qi B1 B2 B3 B4 B5 B6 B7 B8 B9 B10 B11 B12 B13 B14 B15 B16 B17 B18 B19 B20 B21 B22 B23 - B25 B26 B27 B28 B29 B30 B31 B32 B33 B34 B35 B36 B37 B38 B39 B40 B41 B42 B43 B44 B45 B46 B47 B48 B49 B50 B51 B52 B53 B54 B55 B56 B57 B58 B59 B60 B61 B62 B63 B64 B65 B66 B67 B68 B69 B70 B71 B72 B73 B74 B75 B76 B77 B78 B79 B80 B81 B82 B83 B84 B85 B86 B87 B88 B89 B90 B91 B92 B93 B94 B95 B96 B97 B98 B99 B100 B101 B102 B103 B104 B105 B106 B107 B108 B109 B110 B111 B112 B113 B114 B115 B116 B117 B118 B119 B120 B121 B122 B123 B124 B125 B126 B127 B128 B129 B130 B131 B132 B133 B134 B135 B136 B137 B138 B139 B140 B141 B142 B143 B144 B145 B146 B147 B148 B149 B150 B151 B152 B153 B154 B155 B156 B157 B158 B159 B160 B161 B162 B163 B164 B165 B166 B167 B168 B169 B170 B171 B172 B173 B174 B175 B176 B177 B178 B179 B180 B181 B182 B183 B184 B185 B186 B187 B188 B189 B190 B191 B192 B193 B194 B195 B196 B197 B198 B199 B200 B201 B202 B203 B204 B205 B206 B207 B208 B209 B210 B211 B212 B213 B214 B215 B216 B217 B218 B219 B220 B221 B222 B223 B224 B225 B226 B227 B228 B229 B230 B231 B232 B233 B234 B235 B236 B237 B238 B239 B240 B241 B242 B243 B244 B245 B246 B247 B248 B249 B250 B251 B252 Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi B253 B254 B255 B256 B257 B258 B259 B260 B261 B262 B263 B264 B265 B266 B267 B268 B269 B270 B271 B272 B273 B274 B275 B276 B277 B278 B279 B280 B281 B282 B283 B284 B285 B286 B287 B288 B289 B290 B291 B292 B293 B294 B295 B296 B297 B298 B299 B300 B301 B302 B303 B304 B305 B306 B307 B308 B309 B310 B311 B312 B313 B314 B315 B316 B317 B318 B319 B320 B321 B322 B323 B324 B325 B326 B327 B328 B329 B330 B331 B332 B333 B334 B335 B336 B337 B338 B339 B340 B341 B342 B343 B344 B345 B346 B347 B348 B349 B350 B351 B352 B353 B354 B355 B356 B357 B358 B359 B360 B361 B362 B363 B364 B365 B366 B367 B368 B369 B370 B371 B372 B373 B374 B375 B376 B377 B378 B379 B380 B381 B382 B383 B384 B385 B386 B387 B388 B389 B390 B391 B392 B393 B394 B395 B396 B397 B398 B399 B400 B401 B402 B403 B404 B405 B406 B407 B408 B409 B410 B411 B412 B413 B414 B415 B416 B417 B418 B419 B420 B421 B422 B423 B424 B425 B426 B427 B428 B429 B430 B431 B432 B433 B434 B435 B436 B437 B438 B439 B440 B441 B442 B443 B444 B445 B446 B447 B448 B449 B450 B451 B452 B453 B454 B455 B456 B457 B458 B459 B460 B461 B462 B463 B464 B465 B466 B467 B468 B469 B470 B471 B472 B473 B474 B475 B476 B477 B478 B479 B480 B481 B482 B483 B484 B485 B486 B487 B488 B489 B490 B491 B492 B493 B494 B495 B496 B497 B498 B499 B500 B501 B502 B503 B504 B505 B506 B507 B508 B509 B510 B511 B512 B513 B514 B515 B516 B517 B518 B519 B520 B521 B522 B523 B524 B525 B526 B527 B528 B529 B530 B531 B532 B533 B534 B535 B536 B537 B538 B539 B540 B541 B542 B543 B544 B545 B546 B547 B548 B549 B550 B551 B552 B553 B554 B555 B556 B557 B558 B559 B560 B561 B562 B563 B564 B565 B566 B567 B568 B569 B570 B571 B572 B573 B574 B575 B576 B577 B578 B579 B580 B581 B582 B583 B584 B585 B586 B587 B588 B589 B590 B591 B592 B593 B594 B595 B596 B597 B598 B599 B600 B601 B602 B603 B604 B605 B606 B607 B608 B609 B610 B611 B612 B613 B614 B615 B616 B617 B618 B619 B620 B621 B622 B623 B624 B625 B626 B627 B628 B629 B630 B631 B632 B633 B634 B635 B636 B637 B638 B639 B640 B641 B642 B643 B644 B645 B646 B647 B648 _9ι _9ι _9ι _9ι _9ι fiι _9ι _9ι _9ι Sι _9ι _9ι B649 B650 B651 B652 B653 B654 B655 B656 B657 B658 B659 B660 B661 B662 B663 B664 B665 B666 B667 B668 B669 B670 B671 B672 B773 B774 B775 B776 B777 B778 B779 B780 B781 B782 B783 B784 B785 B786 B787 B788 B789 B790 B791 B792 B793 B794 B795 B796 B797 B798 B799 B800 B801 B802 B803 B804 B805 B806 B807 B808 B809 B810 B811 B812 B813 B814 B815 B816 B817 B818 B819 B820 B821 B822 B823 B824 B825 B826 B827 B828 B829 B830 B831 B832 B833 B834 B835 B836 B837 B838 B839 B840 B841 B842 B843 B844 B845 B846 B847 B848 B849 B850 B851 B852 B853 B854 B855 B856 B857 B858 B859 B860 B861 B862 B863 B864 B865 B866 B867 B868 B869 B870 B871 B872 B873 B874 B875 B876 B877 B878 B879 B880 B881 B882 B883 B884 B885 B886 B887 B888 B889 B890 B891 B892 B893 B894 B895 B896 B897 B898 B899 B900 B901 B902 B903 B904 B905 B906 B907 B908 B909 B910 B911 B912 B913 B914 B915 B916 B917 B918 B919 B920 B921 B922 B923 B924 B925 B926 B927 B928 B929 B930 B931 B932 B933 B934 B935 B936 B937 B938 B939 B940 B941 B942 B943 B944 B945 B946 B947 B948 B949 B950 B951 B952 B953 B954 B955 B956 B957 B958 B959 B960 B961 B962 B963 B964 B965 B966 B967 B968 B969 B970 B971 B972 B973 B974 B975 B976 B977 B978 B979 B980 B981 B982 B983 B984 B985 B986 B987 B988 B989 B990 B991 B992 B993 B994 B995 B996 B997 B998 B999 B1000 B1001 B1002 B1003 B1004 B1005 B1006 B1007 B1008 B1009 B1010 B1011 B1012 B1013 B1014 B1015 B1016 B1017 B1018 B1019 B1020 B1021 B1022 B1023 B1024 B1025 B1026 B1027 B1028 B1029 B1030 B1031 B1032 B1033 B1034 B1035 B1036 B1037 B1038 B1039 B1040 B1041 B1042 B1043 B1044 B1045 B1046 B1047 B1048 B1049 B1050 B1051 B1052 B1053 B1054 B1055 B1056 B1057 B1058 B1059 B1060 B1061 B1062 B1063 B1064 B1065 B1066 B1067 B1068 B1069 B1070 B1071 B1072 B1073 B1074 B1075 B1076 B1077 B1078 B1079 B1080 B1081 B1082 B1083 B1084 B1085 B1086 B1087 B1088 B1089 B1090 B1091 B1092 B1093 B1094 B1095 B1096 B1097 B1098 B1099 B1100 B1101 B1102 B1103 B1104 B1105 B1106 B1107 B1108 B1109 B1110 B1111 B1112 B1113 B1114 B1115 B1116 B1117 B1118 B1119 B1120 B1121 B1122 B1123 B1124 B1125 B1126 B1127 B1128 B1129 B1130 B1131 B1132 B1133 B1134 B1135 B1136 B1137 B1138 B1139 B1140 B1141 B1142 B1143 B1144 Ql Ql Ql Ql Ql Ql Ql Ql Ql Ql Ql Ql B1145 B1146 B1147 B1148 B1149 B1150 B1151 B1152 B1153 B1154 B1155 B1156 B1157 B1158 B1159 B1160 B1161 B1162 B1163 B1164 B1165 B1166 B1167 B1168 B1169 B1170 B1171 B1172 B1173 B1174 B1175 B1176 B1177 B1178 B1179 B1180 B1181 B1182 B1183 B1184 B1185 B1186 B1187 B1188 B1189 B1190 B1191 B1192 B1193 B1194 B1195 B1196 B1197 B1198 B1199 B1200 B1201 B1202 B1203 B1204 B1205 B1206 B1207 B1208 B1209 B1210 B1211 B1212 B1213 B1214 B1215 B1216 B1217 Table 10: Compounds of the formula Id (p is 0 or 1): Oi Qi Qi Qi Q i Qi Qi Q i Q i Q i Q i Qi B1 B2 B3 B4 B5 B6 B7 B8 B9 BIO B11 B12 B13 B14 B15 B16 B17 B18 B19 B20 B21 B22 B23 - B25 B26 B27 B28 B29 B30 B31 B32 B33 B34 B35 B36 B37 B38 B39 B40 B41 B42 B43 B44 B45 B46 B47 B48 B49 B50 B51 B52 B53 B54 B55 B56 B57 B58 B59 B60 B61 B62 B63 B64 B65 B66 B67 B68 B69 B70 B71 B72 B73 B74 B75 B76 B77 B78 B79 B80 B81 B82 B83 B84 B85 B86 B87 B88 B89 B90 B91 B92 B93 B94 B95 B96 B97 B98 B99 B100 B101 B102 B103 B104 B105 B106 B107 B108 B109 B110 B111 B112 B113 B114 B115 B116 B117 B118 B119 B120 B121 B122 B123 B124 B125 B126 B127 B128 B129 B130 B131 B132 B133 B134 B135 B136 B137 B138 B139 B140 B141 B142 B143 B144 B145 B146 B147 B148 B149 B150 B151 B152 B153 B154 B155 B156 B157 B158 B159 B160 B161 B162 B163 B164 B165 B166 B167 B168 B169 B170 B171 B172 B173 B174 B175 B176 B177 B178 B179 B180 B181 B182 B183 B184 B185 B186 B187 B188 B189 B190 B191 B192 B193 B194 B195 B196 B197 B198 B199 B200 B201 B202 B203 B204 Qι flι 9ι Sι Sι 9ι Sι fiι Sι 9ι 9ι 9ι B205 B206 B207 B208 B209 B210 B211 B212 B213 B214 B215 B216 B217 B218 B219 B220 B221 B222 B223 B224 B225 B226 B227 B228 B229 B230 B231 B232 B233 B234 B235 B236 B237 B238 B239 B240 B241 B242 B243 B244 B245 B246 B247 B248 B249 B250 B251 B252 B253 B254 B255 B256 B257 B258 B259 B260 B261 B262 B263 B264 B265 B266 B267 B268 B269 B270 B271 B272 B273 B274 B275 B276 B277 B278 B279 B280 B281 B282 B283 B284 B285 B286 B287 B288 B289 B290 B291 B292 B293 B294 B295 B296 B297 B298 B299 B300 B301 B302 B303 B304 B305 B306 B307 B308 B309 B310 B311 B312 B313 B314 B315 B316 B317 B318 B319 B320 B321 B322 B323 B324 B325 B326 B327 B328 B329 B330 B331 B332 B333 B334 B335 B336 B337 B338 B339 B340 B341 B342 B343 B344 B345 B346 B347 B348 B349 B350 B351 B352 B353 B354 B355 B356 B357 B358 B359 B360 B361 B362 B363 B364 B365 B366 B367 B368 B369 B370 B371 B372 B373 B374 B375 B376 B377 B378 B379 B380 B381 B382 B383 B384 B385 B386 B387 B388 B389 B390 B391 B392 B393 B394 B395 B396 B397 B398 B399 B400 B401 B402 B403 B404 B405 B406 B407 B408 B409 B410 B411 B412 B413 B414 B415 B416 B417 B418 B419 B420 B421 B422 B423 B424 B425 B426 B427 B428 B429 B430 B431 B432 B433 B434 B435 B436 B437 B438 B439 B440 B441 B442 B443 B444 B445 B446 B447 B448 B449 B450 B451 B452 B453 B454 B455 B456 B457 B458 B459 B460 B461 B462 B463 B464 B465 B466 B467 B468 B469 B470 B471 B472 B473 B474 B475 B476 B477 B478 B479 B480 B481 B482 B483 B484 B485 B486 B487 B488 B489 B490 B491 B492 B493 B494 B495 B496 B497 B498 B499 B500 B501 B502 B503 B504 B505 B506 B507 B508 B509 B510 B511 B512 B513 B514 B515 B516 B517 B518 B519 B520 B521 B522 B523 B524 B525 B526 B527 B528 B529 B530 B531 B532 B533 B534 B535 B536 B537 B538 B539 B540 B541 B542 B543 B544 B545 B546 B547 B548 B549 B550 B551 B552 B553 B554 B555 B556 B557 B558 B559 B560 B561 B562 B563 B564 B565 B566 B567 B568 B569 B570 B571 B572 B573 B574 B575 B576 B577 B578 B579 B580 B581 B582 B583 B584 B585 B586 B587 B588 B589 B590 B591 B592 B593 B594 B595 B596 B597 B598 B599 B600 Qi Ql Ql Qi Ql Ql Qi Qi Ql Ql Ql Ql B601 B602 B603 B604 B605 B606 B607 B608 B609 B610 B611 B612 B613 B614 B615 B616 B617 B618 B619 B620 B621 B622 B623 B624 B625 B626 B627 B628 B629 B630 B631 B632 B633 B634 B635 B636 B637 B638 B639 B640 B641 B642 B643 B644 B645 B646 B647 B648 B649 B650 B651 B652 B653 B654 B655 B656 B657 B658 B659 B660 B661 B662 B663 B664 B665 B666 B667 B668 B669 B670 B671 B672 B773 B774 B775 B776 B777 B778 B779 B780 B781 B782 B783 B784 B785 B786 B787 B788 B789 B790 B791 B792 B793 B794 B795 B796 B797 B798 B799 B800 B801 B802 B803 B804 B805 B806 B807 B808 B809 B810 B811 B812 B813 B814 B815 B816 B817 B818 B819 B820 B821 B822 B823 B824 B825 B826 B827 B828 B829 B830 B831 B832 B833 B834 B835 B836 B837 B838 B839 B840 B841 B842 B843 B844 B845 B846 B847 B848 B849 B850 B851 B852 B853 B854 B855 B856 B857 B858 B859 B860 B861 B862 B863 B864 B865 B866 B867 B868 B869 B870 B871 B872 B873 B874 B875 B876 B877 B878 B879 B880 B881 B882 B883 B884 B885 B886 B887 B888 B889 B890 B891 B892 B893 B894 B895 B896 B897 B898 B899 B900 B901 B902 B903 B904 B905 B906 B907 B908 B909 B910 B911 B912 B913 B914 B915 B916 B917 B918 B919 B920 B921 B922 B923 B924 B925 B926 B927 B928 B929 B930 B931 B932 B933 B934 B935 B936 B937 B938 B939 B940 B941 B942 B943 B944 B945 B946 B947 B948 B949 B950 B951 B952 B953 B954 B955 B956 B957 B958 B959 B960 B961 B962 B963 B964 B965 B966 B967 B968 B969 B970 B971 B972 B973 B974 B975 B976 B977 B978 B979 B980 B981 B982 B983 B984 B985 B986 B987 B988 B989 B990 B991 B992 B993 B994 B995 B996 B997 B998 B999 B1000 B1001 B1002 B1003 B1004 B1005 B1006 B1007 B1008 B1009 B1010 B1011 B1012 B1013 B1014 B1015 B1016 B1017 B1018 B1019 B1020 B1021 B1022 B1023 B1024 B1025 B1026 B1027 B1028 B1029 B1030 B1031 B1032 B1033 B1034 B1035 B1036 B1037 B1038 B1039 B1040 B1041 B1042 B1043 B1044 B1045 B1046 B1047 B1048 B1049 B1050 B1051 B1052 B1053 B1054 B1055 B1056 B1057 B1058 B1059 B1060 B1061 B1062 B1063 B1064 B1065 B1066 B1067 B1068 B1069 B1070 B1071 B1072 B1073 B1074 B1075 B1076 B1077 B1078 B1079 B1080 B1081 B1082 B1083 B1084 B1085 B1086 B1087 B1088 B1089 B1090 B1091 B1092 B1093 B1094 B1095 B1096 QI QI QI QI QI QI QI QI QI Qi Qi Qi B1097 B1098 B1099 B1100 B1101 B1102 B1103 B1104 B1105 B1106 B1107 B1108 B1109 B1110 B1111 B1 112 B1113 B1114 B1115 B1116 B1117 B1118 B1119 B1120 B1121 B1122 B1123 B1124 B1125 B1126 B1127 B1128 B1129 B1130 B1131 B1132 B1133 B1 134 B1 135 B1136 B1137 B1138 B1139 B1140 B1141 B1142 B1143 B1144 B1145 B1146 B1 147 B1148 B1149 B1150 B1151 B1152 B1153 B1154 B1155 B1156 B1157 B1158 B1159 B1160 B1161 B1162 B1163 B1164 B1 165 B1166 B1167 B1168 B1169 B1 170 B1171 B1 172 B1173 B1174 B1175 B1176 B1177 B1178 B1179 B1180 B1 181 B1182 B1183 B1184 B1185 B1186 B1187 B1188 B1189 B1190 B1191 B1192 B1193 B1194 B1195 B1 196 B1197 B1198 B1199 B1200 B1201 B1202 B1203 B1204 B1205 B1206 B1207 B1208 B1209 B1210 B1211 B1212 B1213 B1214 B1215 B1216 B1217 Table 1 1 : Compounds of the formula le (p is 0 or 1 ): Qi Qi Qi Qi Qi Oi Qi Qi Qi Qi Qi Qi B1 B2 B3 B4 B5 B6 B7 B8 B9 B10 B11 B12 B13 B14 B15 B16 B17 B18 B19 B20 B21 B22 B23 - B25 B26 B27 B28 B29 B30 B31 B32 B33 B34 B35 B36 B37 B38 B39 B40 B41 B42 B43 B44 B45 B46 B47 B48 B49 B50 B51 B52 B53 B54 B55 B56 B57 B58 B59 B60 B61 B62 B63 B64 B65 B66 B67 B68 B69 B70 B71 B72 B73 B74 B75 B76 B77 B78 B79 B80 B81 B82 B83 B84 B85 B86 B87 B88 B89 B90 B91 B92 B93 B94 B95 B96 B97 B98 B99 B100 B101 B102 B103 B104 B105 B106 B107 B108 B109 B110 B111 B112 B113 B114 B115 B116 B117 B118 B119 B120 B121 B122 B123 B124 B125 B126 B127 B128 B129 B130 B131 B132 B133 B134 B135 B136 B137 B138 B139 B140 B141 B142 B143 B144 B145 B146 B147 B148 B149 B150 B151 B152 B153 B154 B155 B156 Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi B157 B158 B159 B160 B161 B162 B163 B164 B165 B166 B167 B168 B169 B170 B171 B172 B173 B174 B175 B176 B177 B178 B179 B180 B181 B182 B183 B184 B185 B186 B187 B188 B189 B190 B191 B192 B193 B194 B195 B196 B197 B198 B199 B200 B201 B202 B203 B204 B205 B206 B207 B208 B209 B210 B211 B212 B213 B214 B215 B216 B217 B218 B219 B220 B221 B222 B223 B224 B225 B226 B227 B228 B229 B230 B231 B232 B233 B234 B235 B236 B237 B238 B239 B240 B241 B242 B243 B244 B245 B246 B247 B248 B249 B250 B251 B252 B253 B254 B255 B256 B257 B258 B259 B260 B261 B262 B263 B264 B265 B266 B267 B268 B269 B270 B271 B272 B273 B274 B275 B276 B277 B278 B279 B280 B281 B282 B283 B284 B285 B286 B287 B288 B289 B290 B291 B292 B293 B294 B295 B296 B297 B298 B299 B300 B301 B302 B303 B304 B305 B306 B307 B308 B309 B310 B311 B312 B313 B314 B315 B316 B317 B318 B319 B320 B321 B322 B323 B324 B325 B326 B327 B328 B329 B330 B331 B332 B333 B334 B335 B336 B337 B338 B339 B340 B341 B342 B343 B344 B345 B346 B347 B348 B349 B350 B351 B352 B353 B354 B355 B356 B357 B358 B359 B360 B361 B362 B363 B364 B365 B366 B367 B368 B369 B370 B371 B372 B373 B374 B375 B376 B377 B378 B379 B380 B381 B382 B383 B384 B385 B386 B387 B388 B389 B390 B391 B392 B393 B394 B395 B396 B397 B398 B399 B400 B401 B402 B403 B404 B405 B406 B407 B408 B409 B410 B411 B412 B413 B414 B415 B416 B417 B418 B419 B420 B421 B422 B423 B424 B425 B426 B427 B428 B429 B430 B431 B432 B433 B434 B435 B436 B437 B438 B439 B440 B441 B442 B443 B444 B445 B446 B447 B448 B449 B450 B451 B452 B453 B454 B455 B456 B457 B458 B459 B460 B461 B462 B463 B464 B465 B466 B467 B468 B469 B470 B471 B472 B473 B474 B475 B476 B477 B478 B479 B480 B481 B482 B483 B484 B485 B486 B487 B488 B489 B490 B491 B492 B493 B494 B495 B496 B497 B498 B499 B500 B501 B502 B503 B504 B505 B506 B507 B508 B509 B510 B511 B512 B513 B514 B515 B516 B517 B518 B519 B520 B521 B522 B523 B524 B525 B526 B527 B528 B529 B530 B531 B532 B533 B534 B535 B536 B537 B538 B539 B540 B541 B542 B543 B544 B545 B546 B547 B548 B549 B550 B551 B552 Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi B553 B554 B555 B556 B557 B558 B559 B560 B561 B562 B563 B564 B565 B566 B567 B568 B569 B570 B571 B572 B573 B574 B575 B576 B577 B578 B579 B580 B581 B582 B583 B584 B585 B586 B587 B588 B589 B590 B591 B592 B593 B594 B595 B596 B597 B598 B599 B600 B601 B602 B603 B604 B605 B606 B607 B608 B609 B610 B611 B612 B613 B614 B615 B616 B617 B618 B619 B620 B621 B622 B623 B624 B625 B626 B627 B628 B629 B630 B631 B632 B633 B634 B635 B636 B637 B638 B639 B640 B641 B642 B643 B644 B645 B646 B647 B648 B649 B650 B651 B652 B653 B654 B655 B656 B657 B658 B659 B660 B661 B662 B663 B664 B665 B666 B667 B668 B669 B670 B671 B672 B773 B774 B775 B776 B777 B778 B779 B780 B781 B782 B783 B784 B785 B786 B787 B788 B789 B790 B791 B792 B793 B794 B795 B796 B797 B798 B799 B800 B801 B802 B803 B804 B805 B806 B807 B808 B809 B810 B811 B812 B813 B814 B815 B816 B817 B818 B819 B820 B821 B822 B823 B824 B825 B826 B827 B828 B829 B830 B831 B832 B833 B834 B835 B836 B837 B838 B839 B840 B841 B842 B843 B844 B845 B846 B847 B848 B849 B850 B851 B852 B853 B854 B855 B856 B857 B858 B859 B860 B861 B862 B863 B864 B865 B866 B867 B868 B869 B870 B871 B872 B873 B874 B875 B876 B877 B878 B879 B880 B881 B882 B883 B884 B885 B886 B887 B888 B889 B890 B891 B892 B893 B894 B895 B896 B897 B898 B899 B900 B901 B902 B903 B904 B905 B906 B907 B908 B909 B910 B911 B912 B913 B914 B915 B916 B917 B918 B919 B920 B921 B922 B923 B924 B925 B926 B927 B928 B929 B930 B931 B932 B933 B934 B935 B936 B937 B938 B939 B940 B941 B942 B943 B944 B945 B946 B947 B948 B949 B950 B951 B952 B953 B954 B955 B956 B957 B958 B959 B960 B961 B962 B963 B964 B965 B966 B967 B968 B969 B970 B971 B972 B973 B974 B975 B976 B977 B978 B979 B980 B981 B982 B983 B984 B985 B986 B987 B988 B989 B990 B991 B992 B993 B994 B995 B996 B997 B998 B999 B1000 B1001 B1002 B1003 B1004 B1005 B1006 B1007 B1008 B1009 B1010 B1011 B1012 B1013 B1014 B1015 B1016 B1017 B1018 B1019 B1020 B1021 B1022 B1023 B1024 B1025 B1026 B1027 B1028 B1029 B1030 B1031 B1032 B1033 B1034 B1035 B1036 B1037 B1038 B1039 B1040 B1041 B1042 B1043 B1044 B1045 B1046 B1047 B1048 Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi B1049 B1050 B1051 B1052 B1053 B1054 B1055 B1056 B1057 B1058 B1059 B1060 B1061 B1062 B1063 B1064 B1065 B1066 B1067 B1068 B1069 B1070 B1071 B1072 B1073 B1074 B1075 B1076 B1077 B1078 B1079 B1080 B1081 B1082 B1083 B1084 B1085 B1086 B1087 B1088 B1089 B1090 B1091 B1092 B1093 B1094 B1095 B1096 B1097 B1098 B1099 B1100 B1101 B1102 B1103 B1104 B1105 B1106 B1107 B1108 B1109 B1110 B1111 B1112 B1113 B1114 B1115 B1116 B1117 B1118 B1119 B1120 B1121 B1122 B1123 B1124 B1125 B1126 B1127 B1128 B1129 B1130 B1131 B1132 B1133 B1134 B1135 B1136 B1137 B1138 B1139 B1140 B1141 B1142 B1143 B1144 B1145 B1146 B1147 B1148 B1149 B1150 B1151 B1152 B1153 B1154 B1155 B1156 B1157 B1158 B1159 B1160 B1161 B1162 B1163 B1164 B1165 B1166 B1167 B1168 B1169 B1170 B1171 B1172 B1173 B1174 B1175 B1176 B1177 B1178 B1179 B1180 B1181 B1182 B1183 B1184 B1185 B1186 B1187 B1188 B1189 B1190 B1191 B1192 B1193 B1194 B1195 B1196 B1197 B1198 B1199 B1200 B1201 B1202 B1203 B1204 B1205 B1206 B1207 B1208 B1209 B1210 B1211 B1212 B1213 B1214 B1215 B1216 B1217 Table 12: Compounds of the formula If: Qi Qi Oi Qi Q i Qi Qi Q i Qi Qi Qi Qi B1 B2 B3 B4 B5 B6 B7 B8 B9 B10 B11 B12 B13 B14 B15 B16 B17 B18 B19 B20 B21 B22 B23 - B25 B26 B27 B28 B29 B30 B31 B32 B33 B34 B35 B36 B37 B38 B39 B40 B41 B42 B43 B44 B45 B46 B47 B48 B49 B50 B51 B52 B53 B54 B55 B56 B57 B58 B59 B60 B61 B62 B63 B64 B65 B66 B67 B68 B69 B70 B71 B72 B73 B74 B75 B76 B77 B78 B79 B80 B81 B82 B83 B84 B85 B86 B87 B88 B89 B90 B91 B92 B93 B94 B95 B96 B97 B98 B99 B100 B101 B1 02 B 103 B104 B105 B106 B107 B108 Qi Qi Qi Qi Q Q i Qi Qi Qi Qi Qi Qi B109 B110 B111 B112 B113 B114 B115 B116 B117 B118 B119 B120 B121 B122 B123 B124 B125 B126 B127 B128 B129 B130 B131 B132 B133 B134 B135 B136 B137 B138 B139 B140 B141 B142 B143 B144 B145 B146 B147 B148 B149 B150 B151 B152 B153 B154 B155 B156 B157 B158 B159 B160 B161 B162 B163 B164 B165 B166 B167 B168 B169 B170 B171 B172 B173 B174 B175 B176 B177 B178 B179 B180 B181 B182 B183 B184 B185 B186 B187 B188 B189 B190 B191 B192 B193 B194 B195 B196 B197 B198 B199 B200 B201 B202 B203 B204 B205 B206 B207 B208 B209 B210 B211 B212 B213 B214 B215 B216 B217 B218 B219 B220 B221 B222 B223 B224 B225 B226 B227 B228 B229 B230 B231 B232 B233 B234 B235 B236 B237 B238 B239 B240 B241 B242 B243 B244 B245 B246 B247 B248 B249 B250 B251 B252 B253 B254 B255 B256 B257 B258 B259 B260 B261 B262 B263 B264 B265 B266 B267 B268 B269 B270 B271 B272 B273 B274 B275 B276 B277 B278 B279 B280 B281 B282 B283 B284 B285 B286 B287 B288 B289 B290 B291 B292 B293 B294 B295 B296 B297 B298 B299 B300 B301 B302 B303 B304 B305 B306 B307 B308 B309 B310 B311 B312 B313 B314 B315 B316 B317 B318 B319 B320 B321 B322 B323 B324 B325 B326 B327 B328 B329 B330 B331 B332 B333 B334 B335 B336 B337 B338 B339 B340 B341 B342 B343 B344 B345 B346 B347 B348 B349 B350 B351 B352 B353 B354 B355 B356 B357 B358 B359 B360 B361 B362 B363 B364 B365 B366 B367 B368 B369 B370 B371 B372 B373 B374 B375 B376 B377 B378 B379 B380 B381 B382 B383 B384 B385 B386 B387 B388 B389 B390 B391 B392 B393 B394 B395 B396 B397 B398 B399 B400 B401 B402 B403 B404 B405 B406 B407 B408 B409 B410 B411 B412 B413 B414 B415 B416 B417 B418 B419 B420 B421 B422 B423 B424 B425 B426 B427 B428 B429 B430 B431 B432 B433 B434 B435 B436 B437 B438 B439 B440 B441 B442 B443 B444 B445 B446 B447 B448 B449 B450 B451 B452 B453 B454 B455 B456 B457 B458 B459 B460 B461 B462 B463 B464 B465 B466 B467 B468 B469 B470 B471 B472 B473 B474 B475 B476 B477 B478 B479 B480 B481 B482 B483 B484 B485 B486 B487 B488 B489 B490 B491 B492 B493 B494 B495 B496 B497 B498 B499 B500 B501 B502 B503 B504 Sl fil Sl fil fil fil Sl fil Sl fil Sl fil B505 B506 B507 B508 B509 B510 B511 B512 B513 B514 B515 B516 B517 B518 B519 B520 B521 B522 B523 B524 B525 B526 B527 B528 B529 B530 B531 B532 B533 B534 B535 B536 B537 B538 B539 B540 B541 B542 B543 B544 B545 B546 B547 B548 B549 B550 B551 B552 B553 B554 B555 B556 B557 B558 B559 B560 B561 B562 B563 B564 B565 B566 B567 B568 B569 B570 B571 B572 B573 B574 B575 B576 B577 B578 B579 B580 B581 B582 B583 B584 B585 B586 B587 B588 B589 B590 B591 B592 B593 B594 B595 B596 B597 B598 B599 B600 B601 B602 B603 B604 B605 B606 B607 B608 B609 B610 B611 B612 B613 B614 B615 B616 B617 B618 B619 B620 B621 B622 B623 B624 B625 B626 B627 B628 B629 B630 B631 B632 B633 B634 B635 B636 B637 B638 B639 B640 B641 B642 B643 B644 B645 B646 B647 B648 B649 B650 B651 B652 B653 B654 B655 B656 B657 B658 B659 B660 B661 B662 B663 B664 B665 B666 B667 B668 B669 B670 B671 B672 B773 B774 B775 B776 B777 B778 B779 B780 B781 B782 B783 B784 B785 B786 B787 B788 B789 B790 B791 B792 B793 B794 B795 B796 B797 B798 B799 B800 B801 B802 B803 B804 B805 B806 B807 B808 B809 B810 B811 B812 B813 B814 B815 B816 B817 B818 B819 B820 B821 B822 B823 B824 B825 B826 B827 B828 B829 B830 B831 B832 B833 B834 B835 B836 B837 B838 B839 B840 B841 B842 B843 B844 B845 B846 B847 B848 B849 B850 B851 B852 B853 B854 B855 B856 B857 B858 B859 B860 B861 B862 B863 B864 B865 B866 B867 B868 B869 B870 B871 B872 B873 B874 B875 B876 B877 B878 B879 B880 B881 B882 B883 B884 B885 B886 B887 B888 B889 B890 B891 B892 B893 B894 B895 B896 B897 B898 B899 B900 B901 B902 B903 B904 B905 B906 B907 B908 B909 B910 B911 B912 B913 B914 B915 B916 B917 B918 B919 B920 B921 B922 B923 B924 B925 B926 B927 B928 B929 B930 B931 B932 B933 B934 B935 B936 B937 B938 B939 B940 B941 B942 B943 B944 B945 B946 B947 B948 B949 B950 B951 B952 B953 B954 B955 B956 B957 B958 B959 B960 B961 B962 B963 B964 B965 B966 B967 B968 B969 B970 B971 B972 B973 B974 B975 B976 B977 B978 B979 B980 B981 B982 B983 B984 B985 B986 B987 B988 B989 B990 B991 B992 B993 B994 B995 B996 B997 B998 B999 B1000 Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi B1001 B1002 B1003 B1004 B1005 B1006 B1007 B1008 B1009 B1010 B1011 B1012 B1013 B1014 B1015 B1016 B1017 B1018 B1019 B1020 B1021 B1022 B1023 B1024 B1025 B1026 B1027 B1028 B1029 B1030 B1031 B1032 B1033 B1034 B1035 B1036 B1037 B1038 B1039 B1040 B1041 B1042 B1043 B1044 B1045 B1046 B1047 B1048 B1049 B1050 B1051 B1052 B1053 B1054 B1055 B1056 B1057 B1058 B1059 B1060 B1061 B1062 B1063 B1064 B1065 B1066 B1067 B1068 B1069 B1070 B1071 B1072 B1073 B1074 B1075 B1076 B1077 B1078 B1079 B1080 B1081 B1082 B1083 B1084 B1085 B1086 B1087 B1088 B1089 B1090 B1091 B1092 B1093 B1094 B1095 B1096 B1097 B1098 B1099 B1100 B1101 B1102 B1103 B1104 B1105 B1106 B1107 B1108 B1109 B1110 B1111 B1112 B1113 B1114 B1115 B1116 B1117 B1118 B1119 B1120 B1121 B1122 B1123 B1124 B1125 B1126 B1127 B1128 B1129 B1130 B1131 B1132 B1133 B1134 B1135 B1136 B1137 B1138 B1139 B1140 B1141 B1142 B1143 B1144 B1145 B1146 B1147 B1148 B1149 B1150 B1151 B1152 B1153 B1154 B1155 B1156 B1157 B1158 B1159 B1160 B1161 B1162 B1163 B1164 B1165 B1166 B1167 B1168 B1169 B1170 B1171 B1172 B1173 B1174 B1175 B1176 B1177 B1178 B1179 B1180 B1181 B1182 B1183 B1184 B1185 B1186 B1187 B1188 B1189 B1190 B1191 B1192 B1193 B1194 B1195 B1196 B1197 B1198 B1199 B1200 B1201 B1202 B1203 B1204 B1205 B1206 B1207 B1208 B1209 B1210 B1211 B1212 B1213 B1214 B1215 B1216 B1217 Table 13: Compounds of the formula Iq (p is 0 or 1): Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Oi Qi B1 B2 B3 B4 B5 B6 B7 B8 B9 B10 B11 B12 B13 B14 B15 B16 B17 B18 B19 B20 B21 B22 B23 - B25 B26 B27 B28 B29 B30 B31 B32 B33 B34 B35 B36 B37 B38 B39 B40 B41 B42 B43 B44 B45 B46 B47 B48 B49 B50 B51 B52 B53 B54 B55 B56 B57 B58 B59 B60 B61 B62 B63 B64 B65 B66 B 67 B68 B69 B70 B71 B72 Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi B73 B74 B75 B76 B77 B78 B79 B80 B81 B82 B83 B84 B85 B86 B87 B88 B89 B90 B91 B92 B93 B94 B95 B96 B97 B98 B99 B100 B101 B102 B103 B104 B105 B106 B107 B108 B109 B110 B111 B112 B113 B114 B115 B116 B117 B118 B119 B120 B121 B122 B123 B124 B125 B126 B127 B128 B129 B130 B131 B132 B133 B134 B135 B136 B137 B138 B139 B140 B141 B142 B143 B144 B145 B146 B147 B148 B149 B150 B151 B152 B153 B154 B155 B156 B157 B158 B159 B160 B161 B162 B163 B164 B165 B166 B167 B168 B169 B170 B171 B172 B173 B174 B175 B176 B177 B178 B179 B180 B181 B182 B183 B184 B185 B186 B187 B188 B189 B190 B191 B192 B193 B194 B195 B196 B197 B198 B199 B200 B201 B202 B203 B204 B205 B206 B207 B208 B209 B210 B211 B212 B213 B214 B215 B216 B217 B218 B219 B220 B221 B222 B223 B224 B225 B226 B227 B228 B229 B230 B231 B232 B233 B234 B235 B236 B237 B238 B239 B240 B241 B242 B243 B244 B245 B246 B247 B248 B249 B250 B251 B252 B253 B254 B255 B256 B257 B258 B259 B260 B261 B262 B263 B264 B265 B266 B267 B268 B269 B270 B271 B272 B273 B274 B275 B276 B277 B278 B279 B280 B281 B282 B283 B284 B285 B286 B287 B288 B289 B290 B291 B292 B293 B294 B295 B296 B297 B298 B299 B300 B301 B302 B303 B304 B305 B306 B307 B308 B309 B310 B311 B312 B313 B314 B315 B316 B317 B318 B319 B320 B321 B322 B323 B324 B325 B326 B327 B328 B329 B330 B331 B332 B333 B334 B335 B336 B337 B338 B339 B340 B341 B342 B343 B344 B345 B346 B347 B348 B349 B350 B351 B352 B353 B354 B355 B356 B357 B358 B359 B360 B361 B362 B363 B364 B365 B366 B367 B368 B369 B370 B371 B372 B373 B374 B375 B376 B377 B378 B379 B380 B381 B382 B383 B384 B385 B386 B387 B388 B389 B390 B391 B392 B393 B394 B395 B396 B397 B398 B399 B400 B401 B402 B403 B404 B405 B406 B407 B408 B409 B410 B411 B412 B413 B414 B415 B416 B417 B418 B419 B420 B421 B422 B423 B424 B425 B426 B427 B428 B429 B430 B431 B432 B433 B434 B435 B436 B437 B438 B439 B440 B441 B442 B443 B444 B445 B446 B447 B448 B449 B450 B451 B452 B453 B454 B455 B456 B457 B458 B459 B460 B461 B462 B463 B464 B465 B466 B467 B468 QJ QJ Q I Q I Q I Q I Q I Q I Q I Q I Q I Q I B469 B470 B471 B472 B473 B474 B475 B476 B477 B478 B479 B480 B481 B482 B483 B484 B485 B486 B487 B488 B489 B490 B491 B492 B493 B494 B495 B496 B497 B498 B499 B500 B501 B502 B503 B504 B505 B506 B507 B508 B509 B510 B511 B512 B513 B514 B515 B516 B517 B518 B519 B520 B521 B522 B523 B524 B525 B526 B527 B528 B529 B530 B531 B532 B533 B534 B535 B536 B537 B538 B539 B540 B541 B542 B543 B544 B545 B546 B547 B548 B549 B550 B551 B552 B553 B554 B555 B556 B557 B558 B559 B560 B561 B562 B563 B564 B565 B566 B567 B568 B569 B570 B571 B572 B573 B574 B575 B576 B577 B578 B579 B580 B581 B582 B583 B584 B585 B586 B587 B588 B589 B590 B591 B592 B593 B594 B595 B596 B597 B598 B599 B600 B601 B602 B603 B604 B605 B606 B607 B608 B609 B610 B611 B612 B613 B614 B615 B616 B617 B618 B619 B620 B621 B622 B623 B624 B625 B626 B627 B628 B629 B630 B631 B632 B633 B634 B635 B636 B637 B638 B639 B640 B641 B642 B643 B644 B645 B646 B647 B648 B649 B650 B651 B652 B653 B654 B655 B656 B657 B658 B659 B660 B661 B662 B663 B664 B665 B666 B667 B668 B669 B670 B671 B672 B773 B774 B775 B776 B777 B778 B779 B780 B781 B782 B783 B784 B785 B786 B787 B788 B789 B790 B791 B792 B793 B794 B795 B796 B797 B798 B799 B800 B801 B802 B803 B804 B805 B806 B807 B808 B809 B810 B811 B812 B813 B814 B815 B816 B817 B818 B819 B820 B821 B822 B823 B824 B825 B826 B827 B828 B829 B830 B831 B832 B833 B834 B835 B836 B837 B838 B839 B840 B841 B842 B843 B844 B845 B846 B847 B848 B849 B850 B851 B852 B853 B854 B855 B856 B857 B858 B859 B860 B861 B862 B863 B864 B865 B866 B867 B868 B869 B870 B871 B872 B873 B874 B875 B876 B877 B878 B879 B880 B881 B882 B883 B884 B885 B886 B887 B888 B889 B890 B891 B892 B893 B894 B895 B896 B897 B898 B899 B900 B901 B902 B903 B904 B905 B906 B907 B908 B909 B910 B911 B912 B913 B914 B915 B916 B917 B918 B919 B920 B921 B922 B923 B924 B925 B926 B927 B928 B929 B930 B931 B932 B933 B934 B935 B936 B937 B938 B939 B940 B941 B942 B943 B944 B945 B946 B947 B948 B949 B950 B951 B952 B953 B954 B955 B956 B957 B958 B959 B960 B961 B962 B963 B964 Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi B965 B966 B967 B968 B969 B970 B971 B972 B973 B974 B975 B976 B977 B978 B979 B980 B981 B982 B983 B984 B985 B986 B987 B988 B989 B990 B991 B992 B993 B994 B995 B996 B997 B998 B999 B1000 B1001 B1002 B1003 B1004 B1005 B1006 B1007 B1008 B1009 B1010 B1011 B1012 B1013 B1014 B1015 B1016 B1017 B1018 B1019 B1020 B1021 B1022 B1023 B1024 B1025 B1026 B1027 B1028 B1029 B1030 B1031 B1032 B1033 B1034 B1035 B1036 B1037 B1038 B1039 B1040 B1041 B1042 B1043 B1044 B1045 B1046 B1047 B1048 B1049 B1050 B1051 B1052 B1053 B1054 B1055 B1056 B1057 B1058 B1059 B1060 B1061 B1062 B1063 B1064 B1065 B1066 B1067 B1068 B1069 B1070 B1071 B1072 B1073 B1074 B1075 B1076 B1077 B1078 B1079 B1080 B1081 B1082 B1083 B1084 B1085 B1086 B1087 B1088 B1089 B1090 B1091 B1092 B1093 B1094 B1095 B1096 B1097 B1098 B1099 B1100 B1101 B1102 B1103 B1104 B1105 B1106 B1107 B1108 B1109 B1110 B1111 B1112 B1113 B1114 B1115 B1116 B1117 B1118 B1119 B1120 B1121 B1122 B1123 B1124 B1125 B1126 B1127 B1128 B1129 B1130 B1131 B1132 B1133 B1134 B1135 B1136 B1137 B1138 B1139 B1140 B1141 B1142 B1143 B1144 B1145 B1146 B1147 B1148 B1149 B1150 B1151 B1152 B1153 B1154 B1155 B1156 B1157 B1158 B1159 B1160 B1161 B1162 B1163 B1164 B1165 B1166 B1167 B1168 B1169 B1170 B1171 B1172 B1173 B1174 B1175 B1176 B1177 B1178 B1179 B1180 B1181 B1182 B1183 B1184 B1185 B1186 B1187 B1188 B1189 B1190 B1191 B1192 B1193 B1194 B1195 B1196 B1197 B1198 B1199 B1200 B1201 B1202 B1203 B1204 B1205 B1206 B1207 B1208 B1209 B1210 B1211 B1212 B1213 B1214 B1215 B1216 B1217 Table 14: Compounds of the formula Ih (p is 0 or 1): Q i Qi Qi Q i Q i Qi Qi Qi Qi Qi Qi Qi B1 B2 B3 B4 B5 B6 B7 B8 B9 B10 B11 B12 B13 B14 B15 B16 B17 B18 B19 B20 B21 B22 B23 Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi B25 B26 B27 B28 B29 B30 B31 B32 B33 B34 B35 B36 B37 B38 B39 B40 B41 B42 B43 B44 B45 B46 B47 B48 B49 B50 B51 B52 B53 B54 B55 B56 B57 B58 B59 B60 B61 B62 B63 B64 B65 B66 B67 B68 B69 B70 B71 B72 B73 B74 B75 B76 B77 B78 B79 B80 B81 B82 B83 B84 B85 B86 B87 B88 B89 B90 B91 B92 B93 B94 B95 B96 B97 B98 B99 B100 B101 B102 B103 B104 B105 B106 B107 B108 B109 B110 B111 B112 B113 B114 B115 B116 B117 B118 B119 B120 B121 B122 B123 B124 B125 B126 B127 B128 B129 B130 B131 B132 B133 B134 B135 B136 B137 B138 B139 B140 B141 B142 B143 B144 B145 B146 B147 B148 B149 B150 B151 B152 B153 B154 B155 B156 B157 B158 B159 B160 B161 B162 B163 B164 B165 B166 B167 B168 B169 B170 B171 B172 B173 B174 B175 B176 B177 B178 B179 B180 B181 B182 B183 B184 B185 B186 B187 B188 B189 B190 B191 B192 B193 B194 B195 B196 B197 B198 B199 B200 B201 B202 B203 B204 B205 B206 B207 B208 B209 B210 B211 B212 B213 B214 B215 B216 B217 B218 B219 B220 B221 B222 B223 B224 B225 B226 B227 B228 B229 B230 B231 B232 B233 B234 B235 B236 B237 B238 B239 B240 B241 B242 B243 B244 B245 B246 B247 B248 B249 B250 B251 B252 B253 B254 B255 B256 B257 B258 B259 B260 B261 B262 B263 B264 B265 B266 B267 B268 B269 B270 B271 B272 B273 B274 B275 B276 B277 B278 B279 B280 B281 B282 B283 B284 B285 B286 B287 B288 B289 B290 B291 B292 B293 B294 B295 B296 B297 B298 B299 B300 B301 B302 B303 B304 B305 B306 B307 B308 B309 B310 B311 B312 B313 B314 B315 B316 B317 B318 B319 B320 B321 B322 B323 B324 B325 B326 B327 B328 B329 B330 B331 B332 B333 B334 B335 B336 B337 B338 B339 B340 B341 B342 B343 B344 B345 B346 B347 B348 B349 B350 B351 B352 B353 B354 B355 B356 B357 B358 B359 B360 B361 B362 B363 B364 B365 B366 B367 B368 B369 B370 B371 B372 B373 B374 B375 B376 B377 B378 B379 B380 B381 B382 B383 B384 B385 B386 B387 B388 B389 B390 B391 B392 B393 B394 B395 B396 B397 B398 B399 B400 B401 B402 B403 B404 B405 B406 B407 B408 B409 B410 B411 B412 B413 B414 B415 B416 B417 B418 B419 B420 Q j Q^ Qj Qi Qi Qi Qi αi Qi Qi Qi Qi B421 B422 B423 B424 B425 B426 B427 B428 B429 B430 B431 B432 B433 B434 B435 B436 B437 B438 B439 B440 B441 B442 B443 B444 B445 B446 B447 B448 B449 B450 B451 B452 B453 B454 B455 B456 B457 B458 B459 B460 B461 B462 B463 B464 B465 B466 B467 B468 B469 B470 B471 B472 B473 B474 B475 B476 B477 B478 B479 B480 B481 B482 B483 B484 B485 B486 B487 B488 B489 B490 B491 B492 B493 B494 B495 B496 B497 B498 B499 B500 B501 B502 B503 B504 B505 B506 B507 B508 B509 B510 B511 B512 B513 B514 B515 B516 B517 B518 B519 B520 B521 B522 B523 B524 B525 B526 B527 B528 B529 B530 B531 B532 B533 B534 B535 B536 B537 B538 B539 B540 B541 B542 B543 B544 B545 B546 B547 B548 B549 B550 B551 B552 B553 B554 B555 B556 B557 B558 B559 B560 B561 B562 B563 B564 B565 B566 B567 B568 B569 B570 B571 B572 B573 B574 B575 B576 B577 B578 B579 B580 B581 B582 B583 B584 B585 B586 B587 B588 B589 B590 B591 B592 B593 B594 B595 B596 B597 B598 B599 B600 B601 B602 B603 B604 B605 B606 B607 B608 B609 B610 B611 B612 B613 B614 B615 B616 B617 B618 B619 B620 B621 B622 B623 B624 B625 B626 B627 B628 B629 B630 B631 B632 B633 B634 B635 B636 B637 B638 B639 B640 B641 B642 B643 B644 B645 B646 B647 B648 B649 B650 B651 B652 B653 B654 B655 B656 B657 B658 B659 B660 B661 B662 B663 B664 B665 B666 B667 B668 B669 B670 B671 B672 B773 B774 B775 B776 B777 B778 B779 B780 B781 B782 B783 B784 B785 B786 B787 B788 B789 B790 B791 B792 B793 B794 B795 B796 B797 B798 B799 B800 B801 B802 B803 B804 B805 B806 B807 B808 B809 B810 B811 B812 B813 B814 B815 B816 B817 B818 B819 B820 B821 B822 B823 B824 B825 B826 B827 B828 B829 B830 B831 B832 B833 B834 B835 B836 B837 B838 B839 B840 B841 B842 B843 B844 B845 B846 B847 B848 B849 B850 B851 B852 B853 B854 B855 B856 B857 B858 B859 B860 B861 B862 B863 B864 B865 B866 B867 B868 B869 B870 B871 B872 B873 B874 B875 B876 B877 B878 B879 B880 B881 B882 B883 B884 B885 B886 B887 B888 B889 B890 B891 B892 B893 B894 B895 B896 B897 B898 B899 B900 B901 B902 B903 B904 B905 B906 B907 B908 B909 B910 B911 B912 B913 B914 B915 B916 fiι fiι Sι 9ι £b fiι fii -3ι fiι fiι fiι fiι B917 B918 B919 B920 B921 B922 B923 B924 B925 B926 B927 B928 B929 B930 B931 B932 B933 B934 B935 B936 B937 B938 B939 B940 B941 B942 B943 B944 B945 B946 B947 B948 B949 B950 B951 B952 B953 B954 B955 B956 B957 B958 B959 B960 B961 B962 B963 B964 B965 B966 B967 B968 B969 B970 B971 B972 B973 B974 B975 B976 B977 B978 B979 B980 B981 B982 B983 B984 B985 B986 B987 B988 B989 B990 B991 B992 B993 B994 B995 B996 B997 B998 B999 B1000 B1001 B1002 B1003 B1004 B1005 B1006 B1007 B1008 B1009 B1010 B1011 B1012 B1013 B1014 B1015 B1016 B1017 B1018 B1019 B1020 B1021 B1022 B1023 B1024 B1025 B1026 B1027 B1028 B1029 B1030 B1031 B1032 B1033 B1034 B1035 B1036 B1037 B1038 B1039 B1040 B1041 B1042 B1043 B1044 B1045 B1046 B1047 B1048 B1049 B1050 B1051 B1052 B1053 B1054 B1055 B1056 B1057 B1058 B1059 B1060 B1061 B1062 B1063 B1064 B1065 B1066 B1067 B1068 B1069 B1070 B1071 B1072 B1073 B1074 B1075 B1076 B1077 B1078 B1079 B1080 B1081 B1082 B1083 B1084 B1085 B1086 B1087 B1088 B1089 B1090 B1091 B1092 B1093 B1094 B1095 B1096 B1097 B1098 B1099 B1100 B1101 B1102 B1103 B1104 B1105 B1106 B1107 B1108 B1109 B1110 B1111 B1112 B1113 B1114 B1115 B1116 B1117 B1118 B1119 B1120 B1121 B1122 B1123 B1124 B1125 B1126 B1127 B1128 B1129 B1130 B1131 B1132 B1133 B1134 B1135 B1136 B1137 B1138 B1139 B1140 B1141 B1142 B1143 B1144 B1145 B1146 B1147 B1148 B1149 B1150 B1151 B1152 B1153 B1154 B1155 B1156 B1157 B1158 B1159 B1160 B1161 B1162 B1163 B1164 B1165 B1166 B1167 B1168 B1169 B1170 B1171 B1172 B1173 B1174 B1175 B1176 B1177 B1178 B1179 B1180 B1181 B1182 B1183 B1184 B1185 B1186 B1187 B1188 B1189 B1190 B1191 B1192 B1193 B1194 B1195 B1196 B1197 B1198 B1199 B1200 B1201 B1202 B1203 B1204 B1205 B1206 B1207 B1208 B1209 B1210 B1211 B1212 B1213 B1214 B1215 B1216 B1217 Table 15: Compounds of the formula Ik (p is 0 or 1): Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi B1 B2 B3 B4 B5 B6 B7 B8 B9 B10 B11 B12 B13 B14 B15 B16 B17 B18 B19 B20 B21 B22 B23 - B25 B26 B27 B28 B29 B30 B31 B32 B33 B34 B35 B36 B37 B38 B39 B40 B41 B42 B43 B44 B45 B46 B47 B48 B49 B50 B51 B52 B53 B54 B55 B56 B57 B58 B59 B60 B61 B62 B63 B64 B65 B66 B67 B68 B69 B70 B71 B72 B73 B74 B75 B76 B77 B78 B79 B80 B81 B82 B83 B84 B85 B86 B87 B88 B89 B90 B91 B92 B93 B94 B95 B96 B97 B98 B99 B100 B101 B102 B103 B104 B105 B106 B107 B108 B109 B110 B111 B112 B113 B114 B115 B116 B117 B118 B119 B120 B121 B122 B123 B124 B125 B126 B127 B128 B129 B130 B131 B132 B133 B134 B135 B136 B137 B138 B139 B140 B141 B142 B143 B144 B145 B146 B147 B148 B149 B150 B151 B152 B153 B154 B155 B156 B157 B158 B159 B160 B161 B162 B163 B164 B165 B166 B167 B168 B169 B170 B171 B172 B173 B174 B175 B176 B177 B178 B179 B180 B181 B182 B183 B184 B185 B186 B187 B188 B189 B190 B191 B192 B193 B194 B195 B196 B197 B198 B199 B200 B201 B202 B203 B204 B205 B206 B207 B208 B209 B210 B211 B212 B213 B214 B215 B216 B217 B218 B219 B220 B221 B222 B223 B224 B225 B226 B227 B228 B229 B230 B231 B232 B233 B234 B235 B236 B237 B238 B239 B240 B241 B242 B243 B244 B245 B246 B247 B248 B249 B250 B251 B252 B253 B254 B255 B256 B257 B258 B259 B260 B261 B262 B263 B264 B265 B266 B267 B268 B269 B270 B271 B272 B273 B274 B275 B276 B277 B278 B279 B280 B281 B282 B283 B284 B285 B286 B287 B288 B289 B290 B291 B292 B293 B294 B295 B296 B297 B298 B299 B300 B301 B302 B303 B304 B305 B306 B307 B308 B309 B310 B311 B312 B313 B314 B315 B316 B317 B318 B319 B320 B321 B322 B323 B324 B325 B326 B327 B328 B329 B330 B331 B332 B333 B334 B335 B336 B337 B338 B339 B340 B341 B342 B343 B344 B345 B346 B347 B348 B349 B350 B351 B352 B353 B354 B355 B356 B357 B358 B359 B360 B361 B362 B363 B364 B365 B366 B367 B368 B369 B370 B371 B372 B373 B374 B375 B376 B377 B378 B379 B380 B381 B382 B383 B384 B385 B386 B387 B388 B389 B390 B391 B392 B393 B394 B395 B396 Qi Qi Qi Qi i i Qi Qi Qi Qi Qi Qi B397 B398 B399 B400 B401 B402 B403 B404 B405 B406 B407 B408 B409 B410 B411 B412 B413 B414 B415 B416 B417 B418 B419 B420 B421 B422 B423 B424 B425 B426 B427 B428 B429 B430 B431 B432 B433 B434 B435 B436 B437 B438 B439 B440 B441 B442 B443 B444 B445 B446 B447 B448 B449 B450 B451 B452 B453 B454 B455 B456 B457 B458 B459 B460 B461 B462 B463 B464 B465 B466 B467 B468 B469 B470 B471 B472 B473 B474 B475 B476 B477 B478 B479 B480 B481 B482 B483 B484 B485 B486 B487 B488 B489 B490 B491 B492 B493 B494 B495 B496 B497 B498 B499 B500 B501 B502 B503 B504 B505 B506 B507 B508 B509 B510 B511 B512 B513 B514 B515 B516 B517 B518 B519 B520 B521 B522 B523 B524 B525 B526 B527 B528 B529 B530 B531 B532 B533 B534 B535 B536 B537 B538 B539 B540 B541 B542 B543 B544 B545 B546 B547 B548 B549 B550 B551 B552 B553 B554 B555 B556 B557 B558 B559 B560 B561 B562 B563 B564 B565 B566 B567 B568 B569 B570 B571 B572 B573 B574 B575 B576 B577 B578 B579 B580 B581 B582 B583 B584 B585 B586 B587 B588 B589 B590 B591 B592 B593 B594 B595 B596 B597 B598 B599 B600 B601 B602 B603 B604 B605 B606 B607 B608 B609 B610 B611 B612 B613 B614 B615 B616 B617 B618 B619 B620 B621 B622 B623 B624 B625 B626 B627 B628 B629 B630 B631 B632 B633 B634 B635 B636 B637 B638 B639 B640 B641 B642 B643 B644 B645 B646 B647 B648 B649 B650 B651 B652 B653 B654 B655 B656 B657 B658 B659 B660 B661 B662 B663 B664 B665 B666 B667 B668 B669 B670 B671 B672 B773 B774 B775 B776 B777 B778 B779 B780 B781 B782 B783 B784 B785 B786 B787 B788 B789 B790 B791 B792 B793 B794 B795 B796 B797 B798 B799 B800 B801 B802 B803 B804 B805 B806 B807 B808 B809 B810 B811 B812 B813 B814 B815 B816 B817 B818 B819 B820 B821 B822 B823 B824 B825 B826 B827 B828 B829 B830 B831 B832 B833 B834 B835 B836 B837 B838 B839 B840 B841 B842 B843 B844 B845 B846 B847 B848 B849 B850 B851 B852 B853 B854 B855 B856 B857 B858 B859 B860 B861 B862 B863 B864 B865 B866 B867 B868 B869 B870 B871 B872 B873 B874 B875 B876 B877 B878 B879 B880 B881 B882 B883 B884 B885 B886 B887 B888 B889 B890 B891 B892 Q1 Q1 Q1 Q1 Q1 Q1 Q1 Q1 Q1 1 Q1 Q1 B893 B894 B895 B896 B897 B898 B899 B900 B901 B902 B903 B904 B905 B906 B907 B908 B909 B910 B911 B912 B913 B914 B915 B916 B917 B918 B919 B920 B921 B922 B923 B924 B925 B926 B927 B928 B929 B930 B931 B932 B933 B934 B935 B936 B937 B938 B939 B940 B941 B942 B943 B944 B945 B946 B947 B948 B949 B950 B951 B952 B953 B954 B955 B956 B957 B958 B959 B960 B961 B962 B963 B964 B965 B966 B967 B968 B969 B970 B971 B972 B973 B974 B975 B976 B977 B978 B979 B980 B981 B982 B983 B984 B985 B986 B987 B988 B989 B990 B991 B992 B993 B994 B995 B996 B997 B998 B999 B1000 B1001 B1002 B1003 B1004 B1005 B1006 B1007 B1008 B1009 B1010 B1011 B1012 B1013 B1014 B1015 B1016 B1017 B1018 B1019 B1020 B1021 B1022 B1023 B1024 B1025 B1026 B1027 B1028 B1029 B1030 B1031 B1032 B1033 B1034 B1035 B1036 B1037 B1038 B1039 B1040 B1041 B1042 B1043 B1044 B1045 B1046 B1047 B1048 B1049 B1050 B1051 B1052 B1053 B1054 B1055 B1056 B1057 B1058 B1059 B1060 B1061 B1062 B1063 B1064 B1065 B1066 B1067 B1068 B1069 B1070 B1071 B1072 B1073 B1074 B1075 B1076 B1077 B1078 B1079 B1080 B1081 B1082 B1083 B1084 B1085 B1086 B1087 B1088 B1089 B1090 B1091 B1092 B1093 B1094 B1095 B1096 B1097 B1098 B1099 B1100 B1101 B1102 B1103 B1104 B1105 B1106 B1107 B1108 B1109 B1110 B1111 B1112 B1113 B1114 B1115 B1116 B1117 B1118 B1119 B1120 B1121 B1122 B1123 B1124 B1125 B1126 B1127 B1128 B1129 B1130 B1131 B1132 B1133 B1134 B1135 B1136 B1137 B1138 B1139 B1140 B1141 B1142 B1143 B1144 B1145 B1146 B1147 B1148 B1149 B1150 B1151 B1152 B1153 B1154 B1155 B1156 B1157 B1158 B1159 B1160 B1161 B1162 B1163 B1164 B1165 B1166 B1167 B1168 B1169 B1170 B1171 B1172 B1173 B1174 B1175 B1176 B1177 B1178 B1179 B1180 B1181 B1182 B1183 B1184 B1185 B1186 B1187 B1188 B1189 B1190 B1191 B1192 B1193 B1194 B1195 B1196 B1197 B1198 B1199 B1200 B1201 B1202 B1203 B1204 B1205 B1206 B1207 B1208 B1209 B1210 B1211 B1212 B1213 B1214 B1215 B1216 B1217 Table 16: Compounds of the formula Im (p is 0 or 1): Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi B1 B2 B3 B4 B5 B6 B7 B8 B9 B10 B11 B12 B13 B14 B15 B16 B17 B18 B19 B20 B21 B22 B23 - B25 B26 B27 B28 B29 B30 B31 B32 B33 B34 B35 B36 B37 B38 B39 B40 B41 B42 B43 B44 B45 B46 B47 B48 B49 B50 B51 B52 B53 B54 B55 B56 B57 B58 B59 B60 B61 B62 B63 B64 B65 B66 B67 B68 B69 B70 B71 B72 B73 B74 B75 B76 B77 B78 B79 B80 B81 B82 B83 B84 B85 B86 B87 B88 B89 B90 B91 B92 B93 B94 B95 B96 B97 B98 B99 B100 B101 B102 B103 B104 B105 B106 B107 B108 B109 B110 B111 B112 B113 B114 B115 B116 B117 B118 B119 B120 B121 B122 B123 B124 B125 B126 B127 B128 B129 B130 B131 B132 B133 B134 B135 B136 B137 B138 B139 B140 B141 B142 B143 B144 B145 B146 B147 B148 B149 B150 B151 B152 B153 B154 B155 B156 B157 B158 B159 B160 B161 B162 B163 B164 B165 B166 B167 B168 B169 B170 B171 B172 B173 B174 B175 B176 B177 B178 B179 B180 B181 B182 B183 B184 B185 B186 B187 B188 B189 B190 B191 B192 B193 B194 B195 B196 B197 B198 B199 B200 B201 B202 B203 B204 B205 B206 B207 B208 B209 B210 B211 B212 B213 B214 B215 B216 B217 B218 B219 B220 B221 B222 B223 B224 B225 B226 B227 B228 B229 B230 B231 B232 B233 B234 B235 B236 B237 B238 B239 B240 B241 B242 B243 B244 B245 B246 B247 B248 B249 B250 B251 B252 B253 B254 B255 B256 B257 B258 B259 B260 B261 B262 B263 B264 B265 B266 B267 B268 B269 B270 B271 B272 B273 B274 B275 B276 B277 B278 B279 B280 B281 B282 B283 B284 B285 B286 B287 B288 B289 B290 B291 B292 B293 B294 B295 B296 B297 B298 B299 B300 B301 B302 B303 B304 B305 B306 B307 B308 B309 B310 B311 B312 B313 B314 B315 B316 B317 B318 B319 B320 B321 B322 B323 B324 Q1 Q1 Q1 Q1 Q1 Q1 Q1 Q1 Q1 Q1 Q1 Q1 B325 B326 B327 B328 B329 B330 B331 B332 B333 B334 B335 B336 B337 B338 B339 B340 B341 B342 B343 B344 B345 B346 B347 B348 B349 B350 B351 B352 B353 B354 B355 B356 B357 B358 B359 B360 B361 B362 B363 B364 B365 B366 B367 B368 B369 B370 B371 B372 B373 B374 B375 B376 B377 B378 B379 B380 B381 B382 B383 B384 B385 B386 B387 B388 B389 B390 B391 B392 B393 B394 B395 B396 B397 B398 B399 B400 B401 B402 B403 B404 B405 B406 B407 B408 B409 B410 B411 B412 B413 B414 B415 B416 B417 B418 B419 B420 B421 B422 B423 B424 B425 B426 B427 B428 B429 B430 B431 B432 B433 B434 B435 B436 B437 B438 B439 B440 B441 B442 B443 B444 B445 B446 B447 B448 B449 B450 B451 B452 B453 B454 B455 B456 B457 B458 B459 B460 B461 B462 B463 B464 B465 B466 B467 B468 B469 B470 B471 B472 B473 B474 B475 B476 B477 B478 B479 B480 B481 B482 B483 B484 B485 B486 B487 B488 B489 B490 B491 B492 B493 B494 B495 B496 B497 B498 B499 B500 B501 B502 B503 B504 B505 B506 B507 B508 B509 B510 B511 B512 B513 B514 B515 B516 B517 B518 B519 B520 B521 B522 B523 B524 B525 B526 B527 B528 B529 B530 B531 B532 B533 B534 B535 B536 B537 B538 B539 B540 B541 B542 B543 B544 B545 B546 B547 B548 B549 B550 B551 B552 B553 B554 B555 B556 B557 B558 B559 B560 B561 B562 B563 B564 B565 B566 B567 B568 B569 B570 B571 B572 B573 B574 B575 B576 B577 B578 B579 B580 B581 B582 B583 B584 B585 B586 B587 B588 B589 B590 B591 B592 B593 B594 B595 B596 B597 B598 B599 B600 B601 B602 B603 B604 B605 B606 B607 B608 B609 B610 B611 B612 B613 B614 B615 B616 B617 B618 B619 B620 B621 B622 B623 B624 B625 B626 B627 B628 B629 B630 B631 B632 B633 B634 B635 B636 B637 B638 B639 B640 B641 B642 B643 B644 B645 B646 B647 B648 B649 B650 B651 B652 B653 B654 B655 B656 B657 B658 B659 B660 B661 B662 B663 B664 B665 B666 B667 B668 B669 B670 B671 B672 B773 B774 B775 B776 B777 B778 B779 B780 B781 B782 B783 B784 B785 B786 B787 B788 B789 B790 B791 B792 B793 B794 B795 B796 B797 B798 B799 B800 B801 B802 B803 B804 B805 B806 B807 B808 B809 B810 B811 B812 B813 B814 B815 B816 B817 B818 B819 B820 Ql Qi Qi Ql Ql Ql Ql Ql Qi Qi Qi Ql B821 B822 B823 B824 B825 B826 B827 B828 B829 B830 B831 B832 B833 B834 B835 B836 B837 B838 B839 B840 B841 B842 B843 B844 B845 B846 B847 B848 B849 B850 B851 B852 B853 B854 B855 B856 B857 B858 B859 B860 B861 B862 B863 B864 B865 B866 B867 B868 B869 B870 B871 B872 B873 B874 B875 B876 B877 B878 B879 B880 B881 B882 B883 B884 B885 B886 B887 B888 B889 B890 B891 B892 B893 B894 B895 B896 B897 B898 B899 B900 B901 B902 B903 B904 B905 B906 B907 B908 B909 B910 B911 B912 B913 B914 B915 B916 B917 B918 B919 B920 B921 B922 B923 B924 B925 B926 B927 B928 B929 B930 B931 B932 B933 B934 B935 B936 B937 B938 B939 B940 B941 B942 B943 B944 B945 B946 B947 B948 B949 B950 B951 B952 B953 B954 B955 B956 B957 B958 B959 B960 B961 B962 B963 B964 B965 B966 B967 B968 B969 B970 B971 B972 B973 B974 B975 B976 B977 B978 B979 B980 B981 B982 B983 B984 B985 B986 B987 B988 B989 B990 B991 B992 B993 B994 B995 B996 B997 B998 B999 B1000 B1001 B1002 B1003 B1004 B1005 B1006 B1007 B1008 B1009 B1010 B1011 B1012 B1013 B1014 B1015 B1016 B1017 B1018 B1019 B1020 B1021 B1022 B1023 B1024 B1025 B1026 B1027 B1028 B1029 B1030 B1031 B1032 B1033 B1034 B1035 B1036 B1037 B1038 B1039 B1040 B1041 B1042 B1043 B1044 B1045 B1046 B1047 B1048 B1049 B1050 B1051 B1052 B1053 B1054 B1055 B1056 B1057 B1058 B1059 B1060 B1061 B1062 B1063 B1064 B1065 B1066 B1067 B1068 B1069 B1070 B1071 B1072 B1073 B1074 B1075 B1076 B1077 B1078 B1079 B1080 B1081 B1082 B1083 B1084 B1085 B1086 B1087 B1088 B1089 B1090 B1091 B1092 B1093 B1094 B1095 B1096 B1097 B1098 B1099 B1100 B1101 B1102 B1103 B1104 B1105 B1106 B1107 B1108 B1109 B1110 B1111 B1112 B1113 B1114 B1115 B1116 B1117 B1118 B1119 B1120 B1121 B1122 B1123 B1124 B1125 B1126 B1127 B1128 B1129 B1130 B1131 B1132 B1133 B1134 B1135 B1136 B1137 B1138 B1139 B1140 B1141 B1142 B1143 B1144 B1145 B1146 B1147 B1148 B1149 B1150 B1151 B1152 B1153 B1154 B1155 B1156 B1157 B1158 B1159 B1160 B1161 B1162 B1163 B1164 B1165 B1166 B1167 B1168 B1169 B1170 B1171 B1172 B1173 B1174 B1175 B1176 B1177 B1178 B1179 B1180 B1181 B1182 B1183 B1184 B1185 B1186 B1187 B1188 B1189 B1190 B1191 B1192 B1193 B1194 B1195 B1196 B1197 B1198 B1199 B1200 B1201 B1202 B1203 B1204 B1205 B1206 B1207 B1208 B1209 B1210 B1211 B1212 B1213 B1214 B1215 B1216 Qi Ql Qi Ql Qi Ql Ql Qi Ql Qi Ql Qi B1217 Table 17: Compounds of the formula In (p is 0 or 1): Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi Qi B1 B2 B3 B4 B5 B6 B7 B8 B9 BIO B11 B12 B13 B14 B15 B16 B17 B18 B19 B20 B21 B22 B23 - B25 B26 B27 B28 B29 B30 B31 B32 B33 B34 B35 B36 B37 B38 B39 B40 B41 B42 B43 B44 B45 B46 B47 B48 B49 B50 B51 B52 B53 B54 B55 B56 B57 B58 B59 B60 B61 B62 B63 B64 B65 B66 B67 B68 B69 B70 B71 B72 B73 B74 B75 B76 B77 B78 B79 B80 B81 B82 B83 B84 B85 B86 B87 B88 B89 B90 B91 B92 B93 B94 B95 B96 B97 B98 B99 B100 B101 B102 B103 B104 B105 B106 B107 B108 B109 B110 B111 B112 B113 B114 B115 B116 B117 B118 B119 B120 B121 B122 B123 B124 B125 B126 B127 B128 B129 B130 B131 B132 B133 B134 B135 B136 B137 B138 B139 B140 B141 B142 B143 B144 B145 B146 B147 B148 B149 B150 B151 B152 B153 B154 B155 B156 B157 B158 B159 B160 B161 B162 B163 B164 B165 B166 B167 B168 B169 B170 B171 B172 B173 B174 B175 B176 B177 B178 B179 B180 B181 B182 B183 B184 B185 B186 B187 B188 B189 B190 B191 B192 B193 B194 B195 B196 B197 B198 B199 B200 B201 B202 B203 B204 B205 B206 B207 B208 B209 B210 B211 B212 B213 B214 B215 B216 B217 B218 B219 B220 B221 B222 B223 B224 B225 B226 B227 B228 B229 B230 B231 B232 B233 B234 B235 B236 B237 B238 B239 B240 B241 B242 B243 B244 B245 B246 B247 B248 B249 B250 B251 B252 B253 B254 B255 B256 B257 B258 B259 B260 B261 B262 B263 B264 Ql Ql Qi Ql Qi Qi Ql Qi Qi Ql Ql Ql B265 B266 B267 B268 B269 B270 B271 B272 B273 B274 B275 B276 B277 B278 B279 B280 B281 B282 B283 B284 B285 B286 B287 B288 B289 B290 B291 B292 B293 B294 B295 B296 B297 B298 B299 B300 B301 B302 B303 B304 B305 B306 B307 B308 B309 B310 B311 B312 B313 B314 B315 B316 B317 B318 B319 B320 B321 B322 B323 B324 B325 B326 B327 B328 B329 B330 B331 B332 B333 B334 B335 B336 B337 B338 B339 B340 B341 B342 B343 B344 B345 B346 B347 B348 B349 B350 B351 B352 B353 B354 B355 B356 B357 B358 B359 B360 B361 B362 B363 B364 B365 B366 B367 B368 B369 B370 B371 B372 B373 B374 B375 B376 B377 B378 B379 B380 B381 B382 B383 B384 B385 B386 B387 B388 B389 B390 B391 B392 B393 B394 B395 B396 B397 B398 B399 B400 B401 B402 B403 B404 B405 B406 B407 B408 B409 B410 B411 B412 B413 B414 B415 B416 B417 B418 B419 B420 B421 B422 B423 B424 B425 B426 B427 B428 B429 B430 B431 B432 B433 B434 B435 B436 B437 B438 B439 B440 B441 B442 B443 B444 B445 B446 B447 B448 B449 B450 B451 B452 B453 B454 B455 B456 B457 B458 B459 B460 B461 B462 B463 B464 B465 B466 B467 B468 B469 B470 B471 B472 B473 B474 B475 B476 B477 B478 B479 B480 B481 B482 B483 B484 B485 B486 B487 B488 B489 B490 B491 B492 B493 B494 B495 B496 B497 B498 B499 B500 B501 B502 B503 B504 B505 B506 B507 B508 B509 B510 B511 B512 B513 B514 B515 B516 B517 B518 B519 B520 B521 B522 B523 B524 B525 B526 B527 B528 B529 B530 B531 B532 B533 B534 B535 B536 B537 B538 B539 B540 B541 B542 B543 B544 B545 B546 B547 B548 B549 B550 B551 B552 B553 B554 B555 B556 B557 B558 B559 B560 B561 B562 B563 B564 B565 B566 B567 B568 B569 B570 B571 B572 B573 B574 B575 B576 B577 B578 B579 B580 B581 B582 B583 B584 B585 B586 B587 B588 B589 B590 B591 B592 B593 B594 B595 B596 B597 B598 B599 B600 B601 B602 B603 B604 B605 B606 B607 B608 B609 B610 B611 B612 B613 B614 B615 B616 B617 B618 B619 B620 B621 B622 B623 B624 B625 B626 B627 B628 B629 B630 B631 B632 B633 B634 B635 B636 B637 B638 B639 B640 B641 B642 B643 B644 B645 B646 B647 B648 B649 B650 B651 B652 B653 B654 B655 B656 B657 B658 B659 B660 Qj Qi Qi Qi Qi -3i Q -3i Qj Qj. -i .a_i B661 B662 B663 B664 B665 B666 B667 B668 B669 B670 B671 B672 B773 B774 B775 B776 B777 B778 B779 B780 B781 B782 B783 B784 B785 B786 B787 B788 B789 B790 B791 B792 B793 B794 B795 B796 B797 B798 B799 B800 B801 B802 B803 B804 B805 B806 B807 B808 B809 B810 B811 B812 B813 B814 B815 B816 B817 B818 B819 B820 B821 B822 B823 B824 B825 B826 B827 B828 B829 B830 B831 B832 B833 B834 B835 B836 B837 B838 B839 B840 B841 B842 B843 B844 B845 B846 B847 B848 B849 B850 B851 B852 B853 B854 B855 B856 B857 B858 B859 B860 B861 B862 B863 B864 B865 B866 B867 B868 B869 B870 B871 B872 B873 B874 B875 B876 B877 B878 B879 B880 B881 B882 B883 B884 B885 B886 B887 B888 B889 B890 B891 B892 B893 B894 B895 B896 B897 B898 B899 B900 B901 B902 B903 B904 B905 B906 B907 B908 B909 B910 B911 B912 B913 B914 B915 B916 B917 B918 B919 B920 B921 B922 B923 B924 B925 B926 B927 B928 B929 B930 B931 B932 B933 B934 B935 B936 B937 B938 B939 B940 B941 B942 B943 B944 B945 B946 B947 B948 B949 B950 B951 B952 B953 B954 B955 B956 B957 B958 B959 B960 B961 B962 B963 B964 B965 B966 B967 B968 B969 B970 B971 B972 B973 B974 B975 B976 B977 B978 B979 B980 B981 B982 B983 B984 B985 B986 B987 B988 B989 B990 B991 B992 B993 B994 B995 B996 B997 B998 B999 B1000 B1001 B1002 B1003 B1004 B1005 B1006 B1007 B1008 B1009 B1010 B1011 B1012 B1013 B1014 B1015 B1016 B1017 B1018 B1019 B1020 B1021 B1022 B1023 B1024 B1025 B1026 B1027 B1028 B1029 B1030 B1031 B1032 B1033 B1034 B1035 B1036 B1037 B1038 B1039 B1040 B1041 B1042 B1043 B1044 B1045 B1046 B1047 B1048 B1049 B1050 B1051 B1052 B1053 B1054 B1055 B1056 B1057 B1058 B1059 B1060 B1061 B1062 B1063 B1064 B1065 B1066 B1067 B1068 B1069 B1070 B1071 B1072 B1073 B1074 B1075 B1076 B1077 B1078 B1079 B1080 B1081 B1082 B1083 B1084 B1085 B1086 B1087 B1088 B1089 B1090 B1091 B1092 B1093 B1094 B1095 B1096 B1097 B1098 B1099 B1100 B1101 B1102 B1103 B1104 B1105 B1106 B1107 B1108 B1109 B1110 B1111 B1112 B1113 B1114 B1115 B1116 B1117 B1118 B1119 B1120 B1121 B1122 B1123 B1124 B1125 B1126 B1127 B1128 B1129 B1130 B1131 B1132 B1133 B1134 B1135 B1136 B1137 B1138 B1139 B1140 B1141 B1142 B1143 B1144 B1145 B1146 B1147 B1148 B1149 B1150 B1151 B1152 B1153 B1154 B1155 B1156 Qj Qj Qj Qj Q Q Qj Qj Qi Qi Qi Qi B1157 B1158 B1159 B1160 B1161 B1162 B1163 B1164 B1165 B1166 B1167 B1168 B1169 B1170 B1171 B1172 B1173 B1174 B1175 B1176 B1177 B1178 B1179 B1180 B1181 B1182 B1183 B1184 B1185 B1186 B1187 B1188 B1189 B1190 B1191 B1192 B1193 B1194 B1195 B1196 B1197 B1198 B1199 B1200 B1201 B1202 B1203 B1204 B1205 B1206 B1207 B1208 B1209 B1210 B1211 B1212 B1213 B1214 B1215 B1216 B1217 Table 18: Compounds of the formula lo (p is 0 or 1 : Q2 Q2 Q2 Q2 Q2 Q2 Q2 Q2 Q2 Q2 Q? Q2 C1 C2 C3 C4 C5 C6 C7 C8 C9 C10 C11 C12 C13 C14 C15 C16 C17 C18 C19 C20 C21 C22 C23 C24 C25 C26 C27 C28 C29 C30 C31 C32 C33 C34 C35 C36 C37 C38 C39 C40 C41 C42 C43 C44 C45 C46 C47 C48 C49 C50 C51 C52 C53 C54 C55 C56 C57 C58 C59 C60 C61 C62 C63 C64 C65 C66 C67 C68 C69 C70 C71 C72 C73 C74 C75 C76 C77 C78 C79 C80 C81 C82 C83 C84 C85 C86 C87 C88 C89 C90 C91 C92 C93 C94 C95 C96 C97 C98 C99 C100 C101 C102 C103C104C105 C106C107C108 C109C110 cm C112 C113C114 C115C116C117 C118C119C120 C121 C122 C123C124 C125C126 C127C128C129 C130C131 C132 C133C134 C135C136 C137C138 C139C140C141 C142C143C144 C145C146 C147C148 C149C150 C151 Table 19: Compounds of the formula Ig (p is 0 or 1): 02 02 02 02 02 & Q_2 Q? 02 Qa 02 02 C1 C2 C3 C4 C5 C6 C7 C8 C9 C10 C11 C12 C13 C14 C15 C16 C17 C18 C19 C20 C21 C22 C23 C24 C25 C26 C27 C28 C29 C30 C31 C32 C33 C34 C35 C36 C37 C38 C39 C40 C41 C42 C43 C44 C45 C46 C47 C48 C49 C50 C51 C52 C53 C54 C55 C56 C57 C58 C59 C60 C61 C62 C63 C64 C65 C66 C67 C68 C69 C70 C71 C72 C73 C74 C75 C76 C77 C78 C79 C80 C81 C82 C83 C84 C85 C86 C87 C88 C89 C90 C91 C92 C93 C94 C95 C96 C97 C98 C99 C100 C101 C102 C103 C104 C105 C106 C107 C108 C109 C110 cm C112 C1 13 C114 C115 C116 C117 C118 C119 C120 C121 C122 C123 C124 C125 C126 C127 C128 C129 C130 C131 C132 C133 C134 C135 C136 C137 C138 C139 C140 C141 C142 C143 C144 C145 C146 C147 C148 C149 C150 C151 Table 20: Compounds of the formula Ir (p is 0 or 1 ): D1 D2 D3 D4 D5 D6 D7 D8 D9 D10 D11 D12 D13 D14 D15 D16 D17 D18 D19 D20 D21 D22 D23 D24 D25 D26 D27 D28 D29 D30 D31 D32 D33 D34 D35 D36 D37 D38 D39 D40 D41 D42 D43 D44 D45 D46 D47 D48 Qs Q3 Qg Q3 Q3 Q3 Qg Qg Qg Qg Qs Q 3 D49 D50 D51 D52 D53 D54 D55 D56 D57 D58 D59 D60 D61 D62 D63 D64 D65 D66 D67 D68 D69 D70 D71 D72 D73 D74 D75 D76 D77 D78 D79 D80 D81 D82 D83 D84 D85 D86 D87 D88 D89 D90 D91 D92 D93 D94 D95 D96 D97 D98 D99 D100 D101 D102 D103 D104 D105 D106 D107 D108 D109 D110 D111 D112 D113 D114 D115 D116 D117 D118 D119 D120 D121 D122 D123 D124 D125 D126 D127 D128 D129 D130 D131 D132 D133 D134 D135 D136 D137 D138 D139 D140 Table 21 : Compounds of the formula Is (p is 0 or 1): Q3 Q3 Q3 Q a Qa Qs Q3 Qg Qa Q3 Qa Qs D1 D2 D3 D4 D5 D6 D7 D8 D9 D10 D11 D12 D13 D14 D15 D16 D17 D18 D19 D20 D21 D22 D23 D24 D25 D26 D27 D28 D29 D30 D31 D32 D33 D34 D35 D36 D37 D38 D39 D40 D41 D42 D43 D44 D45 D46 D47 D48 D49 D50 D51 D52 D53 D54 D55 D56 D57 D58 D59 D60 D61 D62 D63 D64 D65 D66 D67 D68 D69 D70 D71 D72 D73 D74 D75 D76 D77 D78 D79 D80 D81 D82 D83 D84 D85 D86 D87 D88 D89 D90 D91 D92 D93 D94 D95 D96 D97 D98 D99 D100 D101 D102 D103 D104 D105 D106 D107 D108 D109 D110 D111 D112 D113 D114 D115 D116 D117 D118 D119 D120 D121 D122 D123 D124 D125 D126 D127 D128 D129 D130 D131 D132 D133 D134 D135 D136 D137 D138 D139 D140 Table 22: Compounds of the formula It (p is 0 or 1): Q Q^ Q Q^ Q Q Q Q^ Q^ Q Qi Q Q Q Qa E1 E2 E3 E4 E5 E6 E7 E8 E9 E10 E11 E12 E13 E14 E15 E16 E17 E18 E19 E20 E21 E22 E23 E24 E25 E26 E27 E28 E29 E30 Table 23: Compounds of the formula lu (p is 0 or 1 ): Q4 Q4 Q QU Q Q4 Q Q Q4 Q4 Q4 Q4 Q4 & Q. E1 E2 E3 E4 E5 E6 E7 E8 E9 E10 E11 E12 E13 E14 E15 E16 E17 E18 E19 E20 E21 E22 E23 E24 E25 E26 E27 E28 E29 E30 Table 24: Compounds of the formula Iv (p is 0 or 1 ): Q§ Qs Q§ Q§ Qs Q§ F1 F2 F3 F4 F5 F6 Table 25: Compounds of the formula Iw (p is 0 or 1): Qs Qs Qs Qs Qs Q§ F1 F2 F3 F4 F5 F6 Table 26: Physical data of the intermediates: Melting points are indicated in °C Compound Phys. dat. Compound Phys. dat. A17 99-100 A1025 crystalline A7 105-106 A1206 94-95 A9 73-74 A1022 oil A6 148-150 A1203 crystalline A26 143-144 A21 amorphous A34 170-171 A1023 1 10-111 A1026 crystalline A1085 188-191 A1304 crystalline A1088 157-158 A1301 crystalline A1092 crystalline A1018 110-111 A1095 136-138 A1 195-197 A1096 194-196 A2 150-151 A124 135-136 A15 164-166 A31 209-210 A27 107-108 H-B1057 166-167 A29 173-174 H-B1058 crystalline A32 145-146 H-B1061 crystalline A30 178-181 H-B1063 crystalline A4 143-144 H-B1065 oil A3 148-149 H-B1066 150-152 A10 166-167 H-B1067 122-123 A8 123-124 H-B1069 117-118 Compound Phys. dat. Compound Phys. dat. A5 81-82 H-B1070 crystalline A154 108-110 H-C1 116-118 A64 134-135 H-C24 172-175 A94 134-135 A1205 crystalline A531 crystalline H-D113 oil A1045 crystalline H-F5 oil A1322 crystalline H-E16 145-148 A184 146-147 A1088 157-158 A358 155-156 A1103 152-153 Table 27: Physical data for the compounds of the formula I indicated in the above tables: (The melting points are indicated in °C) Comp. No. m.p. Phys. state Comp. No. m.p. Phys. state A2-B1 90-92 crystalline A34-B1 53-54 crystalline A2-B1082 - resin A9-B1 - oil A2-B1083 - resin A184-B1 98-99 crystalline A2-B90 - resin A184-B24 101-102 crystalline A2-B68 120-121 crystalline A7-B24 - oil A2-B24 75-76 crystalline A3-B24 - oil A7-B1 - oil A34-B24 51-52 crystalline A2-B73 - resin A2-B1091 - oil A2-B75 - amorphous A2-B1092 - oil A2-B95 106-107 crystalline A8-B24 52-53 crystalline A2-B93 95-96 crystalline A18-B24 - oil A8-B1 97-98 crystalline A2-B552 - resin A2-B925 - oil A2-C152 - oil A3-B1 42-44 crystalline A2-B69 - resin A94-B1 57-58 crystalline A2-D36 - resin A2-B1057 - amorphous A2-B618 - resin A2-B1063 - oil A2-B49 - resin A2-B1061 - oil A2-D71 - resin A2-B133 58-60 crystalline A2-B1093 - resin Comp. No. m.p. Phys. state Comp. No. m.p. Phys. state A2-B1058 89-91 crystalline A2-B26 - oil A64-B24 80-82 crystalline A2-B33 - resin A64-B1 49-51 crystalline A2-B34 - waxy A2-B1089 - oil A2-B35 - waxy A2-B31 151-153 crystalline A2-B1087 - viscous A2-B1090 139-140 crystalline A2-B1094 - viscous A154-B1 94-95 crystalline A2-B1088 108-109 crystalline A2-B46(cis) 61-62 crystalline A531-B24 - viscous A2-B46(trans) 83-84 crystalline A2-B1099 94-96 crystalline A2-B91 - resin A2-B1095 - viscous A2-B2 - resin A2-B1097 - oil A2-B29 87-88 crystalline A2-B1098 92-93 crystalline A2-B1066 - viscous A2-C147 - resin A2-B25 - oil A2-B70 - resin A2-B1067 - resin A2-B49 - resin A2-B1069 - oil A2-C1 - oil A2-B1068 - viscous A2-B1096 - resin A2-B1070 - viscous A2-B1085 176-177 crystalline A2-B5 - resin A1022-B24 - oil A2-C149 - resin A2-C47 107-110 crystalline A2-C146 - oil A2-B1100 128-130 crystalline A2-B112 - resin A8-B2 70-71 crystalline A2-D140 - oil A8-B1064 - resin A2-B354 139-140 crystalline A2-B45 - resin A2-E16 - solid A2-B10 - viscous A6-B1 123-124 crystalline A8-B133 68-69 crystalline A6-B24 - oil A8-B1101 113-114 crystalline A1322-B24 - oil A8-B1106 - oil A2-B1101 124-125 crystalline A2-D111 (trans) - oil A2-B156 - oil A2-D111 (cis) - resin A2-B144 - resin A8-D111 (trans) - oil A2-B145 - resin A8-D109 62-62 amorphous A2-B134 - resin A8-B35 . oil Comp. No. m.p. Phys. state Comp. No. m.p. Phys. state A1210-B354 220 crystalline A1023-B2 - resin A2-C2 - oil A1023-B354 95-97 crystalline A358-B1 - oil A15-B354 - resin A2-D36 - resin A8-B354 - oil A1208-B354 - oil A8-B1067 - oil A2-D113 (lsom. A) - oil A8-C146 - oil A2-D113 (lsom. B) - oil A8-C1 - oil A2-D114 (lsom. A) 159-160 crystalline A94-B34 108-110 crystalline A2-D115 - amorphous A94-B35 82-84 crystalline A1025-B354 - viscous A1210-B354 - amorphous A2-B1102 124-125 crystalline A2-B1105 119 crystalline A2-B1104 165-167 crystalline A1099-B1107 - amorphous A1210-B1 1 17-119 crystalline A2-B1123 - resin A8-B34 - oil A8-B1123 - resin A8-B1103 - oil A2-B1138 - resin A8-B1063 90-92 crystalline A124-B1 60-65 crystalline A8-B29 - oil A1170-B1 106-107 crystalline A2-C24 - oil A124-B34 - oil A8-B552 - oil A124-B35 - oil A8-B156 - resin A94-B2 53-57 crystalline A1210-B1 105 145-146 glassy- A2-B1174 - crystalline amorphous A1206-B354 - amorphous A2-B1213 133-134 crystalline A8-B134 - oil A3-B1213 - oil A8-D36 - oil A4-B1213 - oil A8-B1213 71-72 crystalline A2-B1214 - resin A8-F5 - resin A2-F5 - resin A1029-B1105 94.5-95 crystalline A2-D109 - oil Biological examples Example B1 : Herbicidal action before emergence of the plants (pre-emergence action) Monocotyledonous and dicotyledonous test plants are sown in standard soil in plastic pots. Immediately after sowing, the test substances as aqueous suspensions (prepared with a 25% wettable powder (Example F3, b) in accordance with WO 97/34485) or as emulsions (prepared with a 25% emulsion concentrate (Example F1 , c)) are sprayed on at a rate of 2 kg of a.i./ha or 250 g of a.i./ha (500 I of water/ha). The test plants are then grown in the greenhouse under optimal conditions. After a test period of 3 weeks, the experiment is evaluated with reference to a nine-step scale (1 = complete damage, 9 = no effect). Score figures of 1 to 4 (in particular 1 to 3) mean a good to very good herbicidal action. Table B1 a: pre-emergence action Compound gg//hhaa CCyyppeerruuis Ipomoea Setaria Sinapis Solanum Stellaria A2-B1 2000 2 2 1 2 2 1 A2-B1082 2000 2 2 2 2 1 2 A2-B1083 2000 2 3 3 4 2 3 A2-B90 2000 1 1 1 1 1 A2-B68 2000 1 2 1 2 2 A2-B24 2000 1 1 1 2 1 A2-B73 2000 3 4 2 2 2 A2-B75 2000 2 3 2 2 2 A2-B95 2000 2 4 2 2 2 A2-B93 2000 2 4 2 2 2 A3-B1 2000 2 2 4 2 2 A94-B1 2000 1 2 2 1 2 A2-B1063 2000 1 2 1 2 2 A2-B1061 2000 3 3 2 2 2 A2-B133 2000 1 2 2 2 2 A64-B24 2000 4 4 2 2 2 A2-B1089 2000 1 2 2 2 2 A2-B31 2000 2 3 4 2 2 A2-B46 (cis) 2000 1 2 1 2 2 Compound gg//hhaa CCyyppeerus Ipomoea Setaria Sinapis Solanum Stellaria A2-B46 (trans) 2000 1 2 1 2 2 A2-B91 2000 1 2 1 2 2 A2-B2 2000 1 1 1 1 2 A2-B25 2000 2 3 2 2 2 A2-B1067 2000 2 3 2 2 3 A2-B1068 2000 2 2 2 2 2 A2-B1070 2000 2 3 3 2 2 A2-C146 2000 1 2 2 2 2 A2-B354 2000 1 1 1 1 2 A34-B1 2000 1 2 2 2 3 A9-B1 2000 2 1 2 1 2 A184-B1 2000 2 4 2 2 2 A184-B24 2000 1 3 2 2 2 A3-B24 2000 1 3 2 2 2 A8-B24 2000 1 2 2 2 3 A18-B24 2000 1 1 1 1 2 A2-B552 2000 1 2 2 2 2 A2-C152 2000 1 1 2 2 2 A2-B69 2000 1 4 2 2 1 A2-D36 2000 1 2 2 2 1 A2-B618 2000 1 1 1 2 1 A2-B33 2000 1 3 2 2 3 A2-B34 2000 1 3 2 2 2 A2-B35 2000 2 4 2 2 2 A2-B1095 2000 3 4 2 2 2 A2-C147 2000 2 4 2 2 2 A2-B49 2000 2 4 2 2 2 A2-C1 2000 2 3 1 2 2 A2-B1100 2000 1 3 1 2 2 A8-B2 2000 1 3 2 2 2 A8-B1064 2000 2 4 3 2 3 A8-B1101 2000 2 4 2 2 1 A2-B156 2000 1 2 1 2 2 Compound g/ha Cyperus Ipomoea Setaria Sinapis Solanum i Stell A2-B144 2000 3 4 2 2 2 4 A2-B134 2000 1 2 1 2 1 1 A1210-B354 2000 2 3 2 1 1 2 A2-C2 2000 2 3 1 1 1 1 A2-D36 2000 1 2 1 2 3 1 A2-D1 13 (lsom •A) 2000 4 4 2 1 3 3 A2-D1 15 2000 3 3 2 2 2 3 A8-B34 2000 2 3 2 2 2 2 A8-B1103 2000 1 3 2 1 1 2 A2-C24 2000 1 2 1 1 1 2 Table B1 b: Pre-emergence action: Compound g/ha Panicum Digitaria Echino. Abutilon Amaranthus Chenop. A8-B1 250 2 2 2 1 1 1 A1022-B24 250 2 4 4 3 4 1 A2-B145 250 2 2 4 2 3 1 A1208-B354 250 1 1 1 1 1 1 A8-B1063 250 2 3 3 2 4 1 A8-B552 250 2 3 4 1 4 1 A8-B156 250 3 3 3 3 4 2 A1210-B1105 250 2 3 2 1 4 1 The same results are obtained when the compounds of the formula I are formulated in accordance with Examples F2 and F4 to F8 in accordance with WO 97/34485. Example B2: Post-emergence herbicidal action Monocotyledonous and dicotyledonous test plants are grown in the greenhouse in plastic pots containing standard soil, and, in the 4- to 6-leaf stage, sprayed with an aqueous suspension of the test substances of the formula I prepared with a 25% wettable powder (Example F3, b) in accordance with WO 97/34485) or with an emulsion of the test substances of the formula I prepared with a 25% emulsion concentrate (Example F1 , c) in accordance with WO 97/34485), corresponding to a rate of 2 kg of a.i./ha or 250 g of al/ha (500 I of water/ha). The test plants are subsequently grown on in the greenhouse under optimal conditions. After a test period of approximately 18 days, the test is evaluated with reference to a nine-step scale (1 = complete damage, 9 = no effect). Score figures of 1 to 4 (in particular 1 to 3) mean a good to very good herbicidal action. In this test, the compounds of the formula I show a potent herbicidal action. Table B2a: Post-emergence action: Compound g/ha Ipomoea Lolium Setaria Sinapis Solanum , Btellϊ A2-B1 2000 1 2 1 I 1 2 A2-B1082 2000 1 2 2 I 1 2 A2-B1083 2000 1 4 2 1 2 A2-B90 2000 1 2 2 I 2 2 A2-B68 2000 1 2 2 1 2 A2-B24 2000 1 2 2 I 2 2 A2-B73 2000 1 3 2 1 2 A2-B75 2000 2 2 3 I 2 2 A2-B95 2000 1 2 2 I 2 2 A2-B93 2000 1 2 2 I 2 2 A3-B1 2000 1 3 2 I 1 2 A94-B1 2000 1 2 2 I 1 1 A2-B1063 2000 2 2 4 I 2 2 A2-B1061 2000 2 2 2 I 2 2 A2-B133 2000 1 2 2 I 2 2 A2-B1058 2000 1 2 4 I 2 2 A64-B24 2000 2 2 4 I 2 2 A64-B1 2000 2 3 4 I 1 2 A2-B1089 2000 1 2 2 1 1 2 A2-B31 2000 2 2 2 I 2 2 A2-B1090 2000 2 4 4 _ 2 2 2 A2-B46 (cis) 2000 1 2 3 I 2 2 A2-B46 (trans) 2000 1 2 2 I 1 2 A2-B91 2000 1 2 2 1 2 2 A2-B2 2000 1 2 2 1 2 2 Compound g/ha Ipomoea Lolium Setaria Sinapis Solanum Stell. A2-B29 2000 2 3 2 1 2 2 A2-B1066 2000 1 3 2 1 2 2 A2-B25 2000 1 2 2 2 1 2 A2-B1068 2000 1 2 4 1 1 2 A2-B1070 2000 2 4 2 2 2 2 A2-B5 2000 1 2 2 1 2 2 A2-C149 2000 1 3 2 1 2 2 A2-C146 2000 1 2 2 1 2 2 A2-B112 2000 2 3 2 1 2 2 A2-B354 2000 2 2 2 2 2 2 A2-E16 2000 2 3 2 2 2 2 A6-B24 2000 1 3 2 1 1 2 A34-B1 2000 1 2 2 1 1 2 A9-B1 2000 2 4 2 2 2 2 A184-B1 2000 1 3 2 1 2 2 A184-B24 2000 1 2 2 1 2 2 A7-B24 2000 1 2 2 1 2 2 A3-B24 2000 2 2 2 1 2 2 A34-B24 2000 1 2 2 1 2 2 A8-B24 2000 2 2 2 1 2 2 A18-B24 2000 1 2 2 1 2 2 A2-C152 2000 2 2 3 1 2 2 A2-B69 2000 1 2 2 1 2 2 A2-D36 2000 2 2 2 1 2 2 A2-B618 2000 2 2 2 1 2 2 A2-B49 2000 2 2 2 1 2 2 A2-B1093 2000 2 2 2 1 2 2 A2-B33 2000 2 4 2 1 2 2 A2-B34 2000 1 3 2 1 1 2 A2-B35 2000 1 3 2 1 1 2 A2-B1087 2000 1 4 3 1 2 2 A531 -B24 2000 2 2 2 1 2 2 A2-B1095 2000 1 2 4 1 2 2 Compound g/ha Ipomoea Lolium Setaria Sinapis Solanum . Stel A2-C147 2000 1 2 2 2 2 A2-B70 2000 3 4 3 2 2 A2-B49 2000 2 2 2 2 2 A2-C1 2000 3 2 2 2 2 A2-B1100 2000 2 2 3 1 2 A8-B2 2000 2 2 2 2 2 3 A8-B1064 2000 2 4 2 1 2 A8-B133 2000 2 4 2 2 2 A8-B1101 2000 2 3 2 2 2 A2-B1101 2000 2 2 2 1 3 A2-B156 2000 1 2 2 2 2 A2-B134 2000 2 2 1 1 2 A1210-B354 2000 2 2 2 1 2 A2-C2 2000 2 1 1 1 A2-D36 2000 2 1 1 1 A2-D113 (lsom. A) 2000 2 1 1 2 A2-D113 (lsom. B) 2000 2 2 2 2 1 2 A2-D114 2000 2 1 1 1 A2-D115 2000 1 2 1 1 A8-B34 2000 2 2 2 2 2 2 A8-B1103 2000 1 4 1 1 A2-C24 2000 1 1 1 1 Table B2b: Post-emergence action: Compound Panicum Digitaria Echino. Abutilon Xanth. Ipopur. Chenop. g/ha A8-B1 250 4 3 3 3 3 3 2 A2-B1091 250 4 4 2 3 4 3 3 A2-B1094 250 2 3 2 3 3 3 2 A2-B145 250 2 2 2 3 3 3 1 A1208-B354 250 3 4 2 1 2 2 2 A1210-B1 250 2 2 2 2 2 2 1 A8-B552 250 2 3 3 2 2 2 2 A8-B156 250 2 3 3 1 2 2 1 A1210-B1105 250 1 2 3 2 2 2 1 A8-B134 250 3 3 3 2 3 3 2 A8-D36 250 3 3 2 2 3 3 2 A2-D111 (cis) 250 2 2 4 2 1 2 2 A2-D111 (trans) 250 3 3 3 3 1 3 2 A8-D111 250 3 3 3 3 1 2 3 A8-D109 250 3 3 3 3 1 2 3 A8-F5 250 4 3 4 3 3 3 3 A2-F5 250 3 3 3 3 3 4 3 The same results are obtained when the compounds of the formula I are formulated in accordance with Examples F2 and F4 to F8 in accordance with WO 97/34485.

Claims: WHAT IS CLAIMED IS: 1. A compound of the formula in which p is 0 or 1 ; R 5 is d-Cehaloalkyl; R is hydrogen, Cι-C 6 alkyl, CrC 6 haloalkyl, C 2 -C 6 alkenyl, C 2 -C 6 haloalkenyl, vinyl which is substituted by CrC 2 alkoxycarbonyl or phenyl, or is C 2 -C 6 alkynyl, C 2 -C 6 haloalkynyl, ethynyl which is substituted by trimethylsilyl, hydroxyl, CrC 2 alkoxy, CrC alkoxycarbonyl or phenyl, or is C 3 -C 6 allenyl, C 3 -C 6 cycloalkyl, C 3 -C 6 cycloalkyl which is substituted by halogen, or is CrCβalkoxy, C 3 -C 6 alkenyloxy, C 3 -C 6 -alkynyloxy, CrC 6 haloalkoxy, C 3 -C 6 haloalkenyloxy, cyano-d-C 4 alkoxy, C 1 -C 4 alkoxy-C 1 -C 4 alkoxy, d-C 4 alkylthio-d-C 4 alkoxy, C C 4 alkylsulfinyl- d-C alkoxy, d-C 4 alkylsulfonyl-d-C 4 alkoxy, d-C 4 alkoxycarbonyl-Cι-C 4 alkoxy, Cι-C 6 alkylthio, d-C 6 alkylsulfinyl, CrC 6 alkylsulfonyl, d-C 6 haloalkylthio, d-Cehaloalkylsulfinyl, d-C 6 haloalkylsulfonyl, d-C 4 alkoxycarbonyl-d-C 4 alkylthio, C C 4 - alkoxycarbonyl-d-C 4 alkylsulfinyl, d-C 4 alkoxycarbonyl-Cι-C 4 alkylsulfonyl, benzyl-S(O) n ι-, d- C 6 aIkylamino, C 2 -C 6 dialkylamino, C C 6 alkylaminosulfonyl, di-(CrC 6 alkylamino)sulfonyl, benzyloxy, benzyl, phenyl, phenoxy, phenylthio, phenylsulfinyl or phenylsulfonyl, it being possible for the phenyl-containing groups, in turn, to be substituted by d-C 3 alkyl, d-C 3 haloalkyl, Cι-C 3 alkoxy, C C 3 haloalkoxy, halogen, cyano or nitro or R 2 is OS(O) n2 -R 2 i . N(R 2 3)-S(O) n3 -R2 2 , cyano, carbamoyl, d-C 4 alkoxycarbonyl, formyl, halogen, thiocyanato, amino, hydroxy-d-C 4 alkyl, Cι-C 4 alkoxy-Cι-C 4 alkyl, C C alkyl-S(O) n4 -Cι-C 4 alkyl, cyano- C 1 -C 4 alkyl, d-Cealkylcarbonyloxy-d-dalkyl, d-C 4 alkoxycarbonyl-Cι-C 4 alkyl, C C 4 alkoxycarbonyloxy-Cι-C 4 alkyl, CrC 4 thiocyanato-d-C 4 alkyl, benzoyloxy-CrC 4 alkyl, C 2 -C 6 oxiranyl, Cι-C 4 alkylamino-Cι-C 4 alkyl, di-(C 1 -C 4 -alkyl)amino-C 1 -C 4 alkyl, d-C^alkylthiocarbonyl-Ci-dalkyl or formyl-Cι-C 4 alkyl, or R 2 is a five- to ten-membered monocyclic or fused bicyclic ring system which can be aromatic or partially saturated and can contain 1 to 4 hetero atoms selected from the group consisting of nitrogen, oxygen and sulfur, the ring system being bonded to the pyridine ring via a Cι-C alkylene, -CH=CH-, -CsC-, -CH2O-, -CH 2 N(Cι-C 4 alkyl)-, -CH 2 SO-, or -CH 2 SO 2 group and it not being possible for each ring system to contain more than 2 oxygen atoms and more than 2 sulfur atoms, and it being possible for the ring system itself to be mono-, di- or trisubstituted by d-C 6 alkyl, Cι- C 6 haloalkyl, C 3 -C 6 alkenyl, C 3 -C 6 haloaIkenyl, C 3 -C 6 alkynyl, C 3 -C 6 haloalkynyl, d-C 6 alkoxy, C C 6 haIoalkoxy, C 3 -C 6 alkenyloxy, C 3 -C 6 alkynyloxy, mercapto, d-Cβalkylthio, d-C 6 haloalkylthio, C 3 -C 6 alkenylthio, C 3 -C 6 haloalkenylthio, C 3 -C 6 alkynylthio, C 2 -C 5 alkoxyalkylthio, C 3 -C 5 acetylalkylthio, C 3 -C 6 alkoxycarbonylalkylthio, C 2 -C 4 cyanoalkylthio, CrC 6 alkylsulfinyl, d-C 6 haloalkylsulfinyl, CrC 6 alkylsulfonyl, d-C 6 haloalkylsulfonyl, aminosulfonyl, d-C alkylaminosulfonyl, di-(d-C 2 alkyl)aminosulfonyl, di-(Cι-C alkyl)amino, halogen, cyano, nitro, phenyl and benzylthio, it being possible for phenyl and benzylthio, in turn, to be substituted on the phenyl ring by Cι-C 3 alkyl, d-C 3 haloalkyl, Cι-C 3 alkoxy, d-C 3 haloalkoxy, halogen, cyano or nitro, and where substituents on the nitrogen in the heterocyclic ring are other than halogen; R 3 is hydrogen, d-C 6 alkyl, d-C 6 haloalkyl, C 2 -C 6 alkenyl, C 2 -C 6 haloalkenyl, C 2 -C 6 alkynyl, C 2 -C 6 haloalkynyl, C 3 -C 6 cycloalkyl, d-C 6 alkoxy, CrC 6 haloalkoxy, CrC 6 alkylthio, d-C 6 alkylsulfinyl, d-C 6 alkylsulfonyl, d-C 6 haloalkylthio, d-C 6 haloalkylsulfinyl, CrC 6 haloalkylsulfonyl, d-C 6 alkylamino, C -C 6 dialkylamino, d-C 6 alkylaminosulfonyl, C 2 -C 6 dialkylaminosulfonyl, phenyl, phenylthio, phenylsulfinyl, phenylsulfonyl or phenoxy, it being possible for phenyl, in turn, to be substituted by d-C 3 alkyl, d-C 3 haloalkyl, d-C 3 alkoxy, d-C 3 haloalkoxy, halogen, cyano or nitro, or R 3 is -N(R 23 )-S(O) n -R 2 2, cyano, halogen, amino, d-C 4 alkoxy-Cι-C 4 alkyl or C 1 -C 4 alkyl-S(O) n -C 1 -C 4 .alkyl; R 4 is hydrogen, d-C 6 alkyl, hydroxyl, C C 6 alkoxy, C C 6 haloalkoxy, C 3 -C 6 alkenyloxy, C 3 -C 6 haloalkenyloxy, C 3 -C 6 alkynyloxy, Cι-C 4 alkylcarbonyloxy, d-C 4 alkylsulfonyloxy, tosyloxy, Cι-C 4 alkylthio, C 1 -C alkylsulfinyl, C C 4 alkylsulfonyl, Cι-C 4 alkylamino, CrC dialkylamino, d-C 4 alkoxycarbonyl, d-C 4 haloalkyl, formyl, cyano, halogen, phenyl or phenoxy, it being possible for phenyl, in turn, to be substituted by d-C 3 alkyl, Cι-C 3 haloalkyl, d-C 3 alkoxy, d-C 3 haloalkoxy, halogen, cyano or nitro; or R 4 is a five to ten-membered monocyclic or R 3 -fused bicyclic ring system which can contain 1 to 4 hetero atoms selected from the group consisting of nitrogen, oxygen and sulfur, the ring system, unless fused, being bonded to the pyridine ring directly or via a d-C 4 alkylene, -CH=CH-, -C≡C-, -CH 2 O- , -CH 2 N(d-C 4 alkyl)-, -CH 2 S-, -CH 2 SO-, or -CH 2 SO 2 - group and it not being possible for the ring system to contain more than 2 oxygen atoms and more than two sulfur atoms, and it being possible for the ring system itself to be mono-, di- or trisubstituted by CrCealkyl, d-C 6 haloalkyl, C 2 -C 6 alkenyl, C 2 -C 6 haloalkenyl, C 2 -C 6 alkynyl, C 2 -C 6 haloalkynyl, d-C 6 alkoxy, Ci-dhaloalkoxy, C 3 -C 6 alkenyloxy, C 3 -C 6 alkynyloxy, d-C 6 alkylthio, C C 6 haloalkylthio, C 3 -C 6 alkenylthio, C 3 -C 6 haloalkenylthio, C 3 -C 6 alkynylthio, d-C 4 alkoxy-C 1 -C 2 alkylthio, C1-dalkylcarbonyl-d-C 2 alky.tr.io, Cι-C alkoxycarbonyl-Cι-C 2 alkylthio, cyano-Cι-C 4 alkylthio, d-C 6 alkylsulfinyl, Cι-C 6 haloalkyIsulfinyl, d-C 6 alkylsulfonyl, CrC 6 haloalkylsulfonyl, aminosulfonyl, Cι-C 2 alkylaminosulfonyl, di-(d-C 2 alkyl)aminosulfonyl, di-(d-C 4 alkyl)amino, halogen, cyano, nitro, phenyl and benzylthio, it being possible for phenyl and benzylthio, in turn, to be substituted on the phenyl ring by d-C 3 alkyl, d-C 3 haloalkyl, d-C 3 alkoxy, C C 3 haloalkoxy, halogen, cyano or nitro, and where substituents on the nitrogen in the heterocyclic ring are other than halogen; R 21 is d-C 4 alkyl or C C haloalkyl; R 22 is Cι-C alkyl, d-C haloalkyl or di-(d-C 4 alkyl)amino; R 2 3, R 24 , R 2 5 independently of one another are hydrogen or d-C 4 alkyl; n, ni, n 2) n 3 and n 4 independently of one another are 0, 1 or 2; Q is Q ! in which R 6 , R , R 8 and R 9 independently of one another are hydrogen, Cι-C 6 alkyl, d-C 6 haloalkyl, C 2 -C 6 alkenyl, C 2 -C 6 alkynyl, d-C 6 alkoxycarbonyl, d-C 6 alkylcarbonyl, Cι-C 6 alkyl-S(O) n ι , Cι-C 6 alkyl-NHS(O) 2 , Cι-C 6 alkylamino, di-(d-C 6 alkyl)amino, hydroxyl, d-C 6 alkoxy, C 3 -C 6 alkenyloxy, C 3 -C 6 alkynyloxy, hydroxy-d-C 6 alkyl, CrC alkylsulfonyloxy-Cι-C 6 alkyl, tosyloxy-Cι-C 6 alkyl, Cι-C 6 alkoxy-Cι-C 6 alkyl, C 1 -C 6 alkyl-S(O) n4 -Cι-C 6 alkyl, cyano-d-C 6 alkyl, Ci-Cβalkoxy-CrCβalkoxy, benzyloxy-Cι-C 6 alkyl, Cι-C 6 alkoxycarbonyl-d-C 6 alkyl, Cι-C 6 alkoxycarbonyloxy-Cι-C 6 alkyl, thiocyanato-d-C 6 alkyl, oxiranyl, d-C 6 alkylamino- Cι-C 6 alkyl, di(d-C 6 alkyl)amino-Cι-C 6 alkyl, formyl-d-C 6 alkyI, Cι-C 6 alkyloximo, halogen, cyano, nitro, phenyl or phenyl which is substituted by C C alkyl, Cι-C 4 haloalkyl, Cι-C 4 alkoxy, CrC 4 haloalkoxy, Cι-C alkylcarbonyl, CrC 4 alkoxycarbonyl, amino, Cι-C alkylamino, di- d-C 4 alkylamino, Cι-C 4 alkyl-S(O)ni8, Cι-C 4 alkyl-S(O) 2 O, d-C 4 haloalkyl-S(O) n5 , d-C 4 haloalkyl-S(O) 2 O, d-C 4 alkyl-S(O) 2 NH, Cι-C 4 alkyl-S(O) n ι 9 N(Cι-C 4 alkyl) 2 , halogen, nitro, COOH or cyano; or adjacent R 6 and R 7 or R 8 and R 9 together are -(CH 2 ) m - , C(O)O(CH ) n2 o- or n 5 , n 17 , nιs, nig and n 2 ι independently of one another are 0, 1 or 2; n 2 o is 2 or 3; n 22 is 2, 3 or 4; m is 2, 3, 4, 5, or 6; W is oxygen, S(O)nβ,-CRιιRi2, -C(O)- or -NR 13 ; Rβ3. R^, Res and R 6 e independently of one another are hydrogen or C Cealkyl, or R 65 together with R 7 or R 9 forms a direct bond; n 6 is 0, 1 or 2; Rn is hydrogen, d-C 4 alkyl, d-C 4 haloalkyl, CrC 4 alkoxy-d-C 4 alkyl, d-C 4 alkylthio-Cr C 4 alkyl, CrC alkylthio-C 3 -C 6 cycloalkyl, CrC 4 alkycarbonyloxy-Cι-C 4 alkyl, d- C 4 alkysulfonyloxy-d-C 4 alkyl, tosyloxy-d-C 4 alkyl, di-(CrC 3 alkoxyalkyl)methyl, di-(C C 3 alkthioalkyl)methyl, (CrC 3 alkoxyalkyl)-(CrC 3 alkthioalkyl)methyl, C 3 -C 5 oxacycloalkyl, C 3 - C 5 thiacycloalkyl, C 3 -C 4 dioxacycloalkyl, C 3 -C 4 dithiacycloalkyl, C 3 -C 4 oxathiacycloalkyl, formyl, CrC 4 alkoxycarbonyl, carbamoyl, CrC 4 alkylaminocarbonyl, di-(CrC alkyl)aminocarbonyl, phenylaminocarbonyl, benzylaminocarbonyl or phenyl which, in turn, can be substituted by Crdalkyl, d-C haloalkyl, CrC alkoxy, d-C haloalkoxy, CrC 4 alkylcarbonyl, CrC 4 alkoxycarbonyl, amino, d-C 4 alkylamino, di-d-C 4 alkylamino, CrC 4 alkyl-S(O) n2 ι, CrC 4 alkyl-S(O) 2 O, CrC 4 haloalkyl-S(O) n7 , CrC 4 haloalkyl-S(O) 2 O, d-C 4 alkyl-S(O) 2 NH, CrC 4 alkyl-S(O) n2 oN(CrC 4 alkyl), halogen, nitro, COOH or cyano; n 7 , n 2 o and n 2 ι independently of one another are 0, 1 or 2; or R12 together with R 6 or R 9 is a group -(CH 2 ) 0 -; o is 1 , 2, 3, 4 or 5; R 12 is hydrogen, Crdalkyl or d-C 4 haloalkyl; or R12 together with Rn is a group -(CH 2 )π.ι. Rio is hydroxyl, O " M + , halogen, cyano, SCN, OCN, C,-C 12 alkoxy, C C 4 alkoxycarbonyl- C^dalkoxy, CrCι 2 alkylthio, d-Cι 2 alkylsulfinyl, d-C^alkylsulfonyl, CrC 12 haloalkylthio, CrC 12 haloalkylsulfinyl, d-C 12 haloalkylsulfonyl, CrCealkoxy-d-Cealkylthio, d-C 6 alkoxy- CrC 6 alkylsulfinyl, CrC 6 alkoxy-Cι-C6alkylsulfonyl, C 2 -Ci 2 alkenylthio, C 2 -Cι 2 alkenylsulfinyl, C 2 -C 12 alkenylsulfonyl, C 2 -C 12 alkynylthio, C 2 -Cι 2 alkynylsulfinyl, C 2 -Cι 2 alkynylsulfonyl, C 2 -Cι haloalkenylthio, C 2 -Cι 2 haloalkenylsulfinyl, C 2 -C 2 haloalkenylsulfonyl, C C 4 - alkoxycarbonyl-CrC 4 alkylthio, d-C 4 alkoxycarbonyl-CrC 4 alkylsulfinyl, d-C alkoxycarbonyl- d-C 4 alkylsulfonyl, (C 1 -C 4 alkoxy) 2 P(O)O ) CrC 4 alkyl-(CrC 4 alkoxy)P(O)O, H(d-C 4 alkoxy)P(O)O, Rι 4 Rι 5 N, R 14 Rι 5 NNH, R 16 R 17 NC(O)O-, Rι 6 Rι 7 NC(O)NH-, Crd 2 alkyl- S(O) 2 NR 18 , CrC 4 haloalkyl-S(O) 2 NR 19 , CrCι 2 alkyl-S(O) 2 O, d-C 4 haloalkyl-S(O) 2 O, d-Cisalkylcarbonyloxy, it being possible for the alkyl group to be substituted by halogen, d-dalkoxy, CrC 6 alkylthio or cyano, or is C 2 -Cι 8 alkenylcarbonyloxy, C 2 -C 8 alkynylcarbonyloxy, C 3 -C 6 cycloalkylcarbonyloxy, CrCι 2 alkoxycarbonyloxy, d-C^alkylthiocarbonyloxy, CrCι 2 alkylthiocarbamoyl, Cι-C 6 alkyl-NH(CS)N(CrC 6 alkyl)-NH-, di-CrC 6 alkyl-N(CS)N(CrC6alkyl)-NH-, benzyloxy, benzylthio, benzylsulfinyl, benzylsulfonyl, phenoxy, phenylthio, phenylsulfinyl, phenylsulfonyl, phenylsulfonylamino, phenylsulfonyloxy or benzoyloxy, it being possible for the phenyl groups, in turn, to be substituted by Crdalkyl, Crdhaloalkyl, d-dalkoxy, d-C 4 haloalkoxy, C C 4 alkylcarbonyl, d-dalkoxycarbonyl, d-C 4 alkylamino, di-d-C 4 alkyIamino, C C 4 alkylthio, d-C 4 alkylsulfinyl, d-C 4 alkyIsulfonyl, CrC 4 alkyl-S(O) 2 O, d-C 4 haloalkylthio, d-dhaloalkylsulfinyl, d-C 4 haloalkylsulfonyl, d-C 4 haloalkyl-S(O) 2 O, CrC 4 alkyl-S(O) 2 NH, d-dalkyl- S(O) 2 N(CrC 4 alkyl), halogen, nitro or cyano; or R 10 is a group An-thio, Ar 2 -sulfinyl, Ar 3 -sulfonyl, -OCO-Ar or NH-Ar 5 in which Ar^ Ar 2 , Ar 3 , Ar 4 and Ar 5 independently of one another are a five- to ten-membered monocyclic or fused bicyclic ring system which can be aromatic or partially saturated and can contain 1 to 4 hetero atoms selected from the group consisting of nitrogen, oxygen and sulfur, and it not being possible for each ring system to contain more than 2 oxygen atoms and more than two sulfur atoms, and it being possible for the ring system itself to be mono-, di- or trisubstituted by d-C 6 alkyl, d-dhaloalkyl, C 3 -C 6 alkenyl, C 3 -C 6 haloalkenyl, C 3 -C 6 alkynyl, C 3 -C 6 haloalkynyl, d-dalkoxy, d-C 6 haloalkoxy, C 3 -C 6 alkenyloxy, C 3 -C 6 alkynyloxy, mercapto, d-C 6 alkylthio, d-dhaloalkylthio, C 3 -C 6 alkenylthio, C 3 -C 6 haloalkenylthio, C 3 -C 6 alkynylthio, C 2 -C 5 alkoxyalkylthio, C 3 -C 5 acetylalkylthio, C 3 -C 6 alkoxycarbonylalkylthio, C 2 -C 4 -cyanoaIkylthio, d-dalkylsulfinyl, d-dhaloalkylsulfinyl, d-dalkylsulfonyl, d-C 6 - haloalkylsulfonyl, aminosulfonyl, C C 2 alkylaminosulfonyl, di-(CrC 2 alkyl)aminosulfonyl, di- (Cι-C 4 alkyl)amino, halogen, cyano, nitro, phenyl and benzylthio, it being possible for phenyl and benzylthio, in turn, to be substituted on the phenyl ring by d-dalkyl, d-dhaloalkyl, d-dalkoxy, d-dhaloalkoxy, halogen, cyano or nitro, and where substituents on the nitrogen in the heterocyclic rings are other than halogen; R i4 , R 15 , R 16 , Rι and R 18 independently of one another are hydrogen or d-dalkyl; n 8> n 9 , nio, nu, nι 2 , n 13 and n 14 independently of one another are 0, 1 or 2; Rι 3 is hydrogen, d-dalkyl, Crdalkythio-d-dcarbonyl, CrC 4 alkylsulfinyl-Cι-C 4 carbonyl, d-dalkylsulfonyl-Crdcarbonyl, d-C 4 -alkoxycarbonyl, d-C alkylcarbonyl, phenylcarbonyl, or is phenyl which, in turn, can be substituted by d-dalkyl, d-dhaloalkyl, d-C 4 alkoxy, d-dhaloalkoxy, CrC alkylcarbonyl, CrC 4 alkoxycarbonyl, d-C 4 alkylamino, di-d-C - alkylamino, CrC 4 alkyl-S(O) n i5, CrC 4 alkyl-S(O) 2 O, d-C 4 haloalkyl-S(O) n i6, d-dhaloalkyl- S(O) 2 O, CrC 4 alkyl-S(O) 2 NH, CrC 4 alkyl-S(O) 2 N(CrC 4 alkyl), halogen, nitro, or cyano; and nis and nι 6 independently of one another are 0, 1 or 2; or an agrochemically tolerated salt M + or a stereoisomer or tautomer of a compound of the formula I. 2. A compound according to claim 1 , wherein p is 0; R 5 is d-dhaloalkyl; R 2 is hydrogen, d-dalkyl, d-dhaloalkyl, C 2 -C 6 alkenyl, C 2 -C 6 haloalkenyl, C -C 6 alkynyl, C 2 -C 6 haloalkynyl, C 3 -C 6 cycloalkyl, d-dalkoxy, d-dhaloalkoxy, d-dalkylthio, d-C 6 - alkylsulfinyl, CrC 6 alkylsulfonyl, d-dhaloalkylthio, CrC 6 haloalkylsulfinyl, C C 6 - haloalkylsulfonyl, benzyl-S(O) n r, d-dalkylamino, C 2 -C 6 dialkylamino, d-C 6 - alkylaminosulfonyl, C 2 -C 6 -dialkylaminosulfonyl, phenyl, phenoxy, phenylthio, phenylsulfinyl or phenylsulfonyl, it being possible for the phenyl group, in turn, to be substituted by d-dalkyl, d-dhaloalkyl, d-dalkoxy, d-C 3 haloalkoxy, halogen, cyano or nitro, or is OS(O) n2 -R 2 i, N(R 2 3)-S(O)n 3 -R 22 , cyano, halogen, amino, Cι-C 4 alkoxy-d-C 4 alkyl, C C 4 alkyl- S(O) n -CrC alkyl, cyano-Crdalkyl or d-dalkoxy-d-dalkoxy; R 3 is hydrogen, d-C 6 alkyl, d-dhaloalkyl, C 2 -C 6 alkenyl, C 2 -C 6 haloalkenyl, C 2 -C 6 alkynyl, C 2 -C 6 haloalkynyl, C 3 -C 6 cycloalkyl, d-C 6 alkoxy, CrC 6 haloalkoxy, d-C 6 alkylthio, d-C 6 - alkylsulfinyl, d-C 6 alkylsulfonyl, d-C 6 haloalkylthio, d-C 6 haloalkylsulfinyl, Crd- haloalkylsulfonyl, CrC 6 alkylamino, C 2 -C 6 dialkylamino, d-C 6 -alkylaminosulfonyl, C 2 -C 6 - dialkylaminosulfonyl, phenyl, phenylthio, phenylsulfinyl, phenylsulfonyl or phenoxy, it being possible for phenyl, in turn, to be substituted by d-C 3 alkyl, d-C 3 haloalkyl, d-dalkoxy, d-dhaloalkoxy, halogen, cyano or nitro, or is -N(R 23 )-S(O) n -R 22> cyano, halogen, amino, d-dalkoxy-Crdalkyl or CrC 4 alkyl-S(O) n -CrC 4 alkyl; R 4 is hydrogen, d-dalkyl, d-C 4 alkoxy, d-C 4 haloalkoxy, d-C 4 alkylcarbonyloxy, C C - Alkylthio, d-C 4 alkylsulfinyl, d-dalkylsulfonyl, d-C 4 haloalkyl, formyl, cyano, halogen, phenyl or phenoxy, it being possible for phenyl, in turn, to be substituted by d-dalkyl, d-dhaloalkyl, d-dalkoxy, d-dhaloalkoxy, halogen, cyano or nitro; or R 4 is a five- to ten-membered monocyclic or R 3 -fused bicyclic ring system which can contain 1 to 4 hetero atoms selected from the group consisting of nitrogen, oxygen and sulfur, the ring system being bonded to the pyridine ring via a d-C 4 alkylene group and it not being possible for the ring system to contain more than 2 oxygen atoms and more than two sulfur atoms, and it being possible for the ring system itself to be mono-, di- or trisubstituted by d-dalkyl, d-dhaloalkyl, C -C 6 alkenyl, C 2 -C 6 haloalkenyl, C 2 -C 6 alkynyl, C 2 -C 6 haloalkynyl, d-dalkoxy, d-C 6 haloalkoxy, C 3 -C 6 alkenyloxy, C 3 -C 6 alkynyloxy, d-C 6 - Alkylthio, d-C 6 haloalkylthio, C 3 -C 6 alkenylthio, C 3 -C 6 haloalkenylthio, C 3 -C 6 alkynylthio, C C 4 - alkoxy-d-dalkylthio, d-dalkylcarbonyl-d-dalkylthio, d-dalkoxycarbonyl-d-dalkylthio, cyano-d-dalkylthio, d-dalkylsulfinyl, d-dhaloalkylsulfinyl, d-dalkylsulfonyl, d-C 6 - haloalkylsulfonyl, aminosulfonyl, d-C 2 alkylaminosulfonyl, C 2 -C dialkylaminosulfonyl, halogen, cyano, nitro, phenyl and benzylthio, it being possible for phenyl and benzylthio, in turn, to be substituted on the phenyl ring by d-dalkyl, d-C 3 haloalkyl, d-dalkoxy, d-dhaloalkoxy, halogen, cyano or nitro, and where substituents on the nitrogen in the heterocyclic ring are other than halogen; R 21 and R 22 independently of one another are d-dalkyl or d-dhaloalkyl; R 23 , R 24 and R 25 independently of one another are hydrogen or d-dalkyl; n, ni, n 2 , n 3 and n 4 independently of one another are 0, 1 or 2; Q is Qi in which Re, R 7 , Rs and R 9 independently of one another are hydrogen, Crdalkyl, d-C 6 -haloalkyl, d-dalkenyl, C 2 -C 6 alkynyl, d-C 6 alkoxycarbonyl, CrC 6 alkyl-S(O) n i7. CrC 6 alkyl-NHS(O) 2 , CrC 6 alkylamino, di-(CrC 6 alkyl)amino, hydroxyl, d-dalkoxy, C 3 .C 6 alkenyloxy, C 3 -C 6 - alkynyloxy, hydroxy-d-C 6 alkyl, d-dalkylsulfonyloxy-d-dalkyl, tosyloxy-d-C 6 alkyl, halogen, cyano, nitro, phenyl or phenyl which is substituted by d-C 4 a!kyl, d-dhaloalkyl, d- dalkoxy, d-C 4 haloalkoxy, d-C 4 alkylcarbonyl, d-C 4 alkoxycarbonyl, amino, C C 4 - alkylamino, di-d-C 4 alkylamino, Cι-C 4 alkyl-S(O)ni8, C C 4 alkyl-S(O) 2 O, CrC 4 haloalkyl-S(O) n5 , d-C 4 haloalkyl-S(O) 2 O, d-C 4 alkyl-S(O) 2 NH, CrC 4 alkyl-S(O) n ι 9 N(CrC 4 alkyl), halogen, nitro, COOH or cyano; or adjacent R 6 and R 7 or R 8 and R 9 together are -(CH 2 ) m -; n 5 nι 7 , n 18 and n 19 independently of one another are 0, 1 or 2; m is 2, 3, 4, 5, or 6; W is oxygen, S(O) n6 , -CRn R12-, -C(O)- or -NR13-; n 6 is 0, 1 or 2; Rn is hydrogen, d-C 4 alkyl, C C 4 haloalkyl, CrC 4 alkoxy-d-C 4 alkyl, d-C 4 alkylthio-Cr C 4 alkyl, d-C 4 alkylcarbonyloxy-CrC 4 alkyl, d-dalkylsulfonyloxy-d-dalkyl, tosyloxy-d- dalkyl, di-(d-C 3 alkoxyalkyl)methyl, di-(CrC 3 alkylthioalkyl)methyl, (CrC 3 alkoxyalkyl)-(d- C 3 alkylthioalkyl)methyl, C 3 -C 5 oxacycloalkyl, C 3 -C 5 thiacycloalkyl, C 3 -C 4 dioxacycloalkyl, C 3 -C 4 - dithiacycloalkyl, C 3 -C 4 oxathiacycloalkyl, formyl, C C 4 alkoxycarbonyl or phenyl which, in turn, can be substituted by d-dalkyl, d-C 4 haloalkyl, d-C alkoxy, d-C 4 haloalkoxy, CrC - alkylcarbonyl, d-C 4 alkoxycarbonyl, amino, d-C 4 alkylamino, di-d-C 4 alkylamino, d-C alkyl- S(O)n2i, CrC 4 alkyl-S(O) 2 O, d-C 4 haloalkyl-S(O) n7 , CrC 4 haloalkyl-S(O) 2 O, d-dalkyl- S(O) 2 NH, Cι-C 4 alkyl-S(O) n2 oN(Cι-C 4 alkyl), halogen, nitro, COOH or cyano; n 7 , n 2 o and n 2 ι independently of one another are 0, 1 or 2; or R1 2 together with R 9 is a group -(CH 2 )cr. o is 1 , 2, 3, 4 or 5; R 12 is hydrogen, d-C 4 alkyl or C C 4 haloalkyl; or R12 together with Rn is a group -(CH 2 ) ι; Rio is hydroxyl, O " M + , halogen, d-C^alkoxy, d-C^alkylcarbonyloxy, C 2 -C 4 - alkenylcarbonyloxy, C 3 -C 6 cycloalkylcarbonyloxy, CrCι 2 alkoxycarbonyloxy, CrC 1 - alkylcarbonyloxy, R 23 R2 4 N-C(O)O, CrCι 2 alkylS(O)n 8 -, C C 4 haloalkyl-S(O) n9 -, C 2 -C 12 - alkenylS(O) n ιo-, C 2 -Ci2haloalkenylS(O) n ιr, C 2 -C 1 2alkynylS(O) n ι 2 -; benzyloxy, phenoxy, phenylthio, phenylsulfinyl or phenylsulfonyl, where the phenyl group, in turn, can be substituted by d-C 4 alkyl, C C 4 haloalkyl, C C 4 alkoxy, d-C 4 haloalkoxy, CrC 4 alkylcarbonyl, d-dalkoxycarbonyl, CrC 4 alkylamino, di-CrC 4 alkylamino, d-C alkyl-S(O) n i 3 , d-C 4 alkyl- S(O) 2 O, C 1 -C 4 haloalkyl-S(O)ni4, CrC 4 haloalkyl-S(O) 2 O, d-C 4 alkyl-S(O) 2 NH, d-dalkyl- S(O) 2 N(CrC 4 alkyl), halogen, nitro or cyano, or is CrC 4 alkyl-S(O) 2 O, phenyl-S(O) 2 O, (d-C 4 - alkoxy) 2 P(O)O, CrC 4 alkyl(d-C 4 alkoxy)P(O)O, or H(C C 4 alkoxy)P(O)O; n 8 , n 9 , n 10 , nn, nι 2 , nι 3 and n 14 independently of one another are 0, 1 or 2; Rι 3 is hydrogen, d-dalkyl, d-C alkoxycarbonyl or phenyl which, in turn, can be substituted by d-dalkyl, d-dhaloalkyl, d-dalkoxy, C C 4 haloalkoxy, d-C 4 alkylcarbonyl, C C 4 alkoxycarbonyl, Cι-C alkylamino, di-d-C 4 alkylamino, CrC alkyl-S(O) n ι 5 , Crdalkyl- S(O) 2 O, d-C 4 haloalkyl-S(O)ni6, d-C 4 haloalkyl-S(O) 2 O, d-C 4 alkyl-S(O) 2 NH, C C 4 alkyl- S(O) 2 N(d-C 4 alkyI), halogen, nitro or cyano; n i5 and n i6 independently of one another are 0, 1 or 2; or an agrochemically tolerated salt M + or a stereoisomer or tautomer of a compound of the formula I. 3. A compound according to claim 1 , in which Rι 0 is hydroxyl or O " M + . 4. A compound according to claim 1 , in which W is oxygen, -CRnRι 2 - or -C(O)-. 5. A compound according to claim 1 , in which W is oxygen and R 6 , R 7 , R 8 and R 9 independently of one another are hydrogen or d-C 3 alkyl. 6. A compound according to claim 1 , in which W is -C(O)- and R 6 , R 7 , R 8 and R 9 independently of one another are d-dalkyl. 7. A compound according to claim 1 , in which R is hydrogen and R 3 is methyl. 8. A compound according to claim 1 , in which R 2 is methyl, ethyl, n-propyl, i-propyl, vinyl, methoxymethyl, methoxycarbonyloxymethyl, ethoxycarbonyloxymethyl, acetoxymethyl, propionyloxymethyl, chloromethyl, bromomethyl, fluoromethyl, difluoromethyl, trifluoromethyl or cyanomethyl. 9. A compound according to claim 1 , in which R 4 is hydrogen or methyl. 10. A compound according to claim 1 , in which R 5 is trifluoromethyl, difluorochloromethyl, pentafluoroethyl, heptafluoropropyl or difluoromethyl. 11. A compound according to claim 1 , in which R 3 is hydrogen and R 2 is d-dalkyl, d-dhaloalkyl, cyclopropyl, C 2 -C 3 alkenyl, C 2 -C 3 haloalkenyl, C 2 -C 3 alkynyl, allenyl, d-C 2 - alkoxy-d-dalkyl, d-dalkylthio-d-dalkyl, cyano-d-C 2 alkyl, d-dalkoxycarbonyl-d-d- alkyl, d-dalkylcarbonyloxy-d-dalkyl, C C 3 alkoxy, d-C 3 haloalkoxy, allyloxy, propargyloxy, d-dalkylthio, d-C 3 alkylsulfinyl or cyano. 12. A compound of the formula Ilia in which R 501 is Cι-C 6 haloalkyl; R 30 ι is hydrogen; R 40 ι is hydrogen or d-dalkyl; and R 201 is CrC 6 alkyl, Crdhaloalkyl-Crdalkyl, C 2 -C 6 alkenyl, C 2 -C 6 haloalkenyl, or d-C 2 - alkoxycarbonyl- or phenyl-substituted vinyl, C 2 -C 6 alkynyl or C 2 -C 6 haloalkynyl; or trimethylsilyl-, hydroxyl-, d-C 2 alkoxy-, CrC 2 alkoxycarbonyl- or phenyl-substituted ethynyl or C 3 -C 6 allenyl; or C 3 -C 6 cycloalkyl, halogen-substituted C 3 -C 6 cycloalkyl, d-dalkoxy-d-d- alkyl, Cι-C 4 alkyl-S(O) n -CrC 4 alkyl, cyano-C C 4 alkyl, d-dalkoxycarbonyl-d-dalkyl, d-C 4 - thiocyanato, oxiranyl, CrC 4 alkylamino-CrC 4 alkyl, CrC 4 dialkylamino-CrC 4 alkyl, hydroxy- d-C alkyl, Cι-C 12 alkylthiocarbonyl-CrC 4 alkyl or formyl-d-C 4 alkyl, or R 20 ι is a five- to ten- membered monocyclic or fused bicyclic ring system which can be aromatic or partially saturated and can contain 1 to 4 hetero atoms selected from the group consisting of nitrogen, oxygen and sulfur, the ring system being bonded to the pyridine ring via a d-C 4 - alkylene, -CH=CH-, -C≡C-, -CH 2 O- , -CH 2 N(C C 4 alkyl)-, -CH 2 S-, -CH 2 SO- or -CH 2 SO 2 - group and it not being possible for each ring system to contain more than 2 oxygen atoms and more than two sulfur atoms, and it being possible for the ring system itself to be mono-, di- or trisubstituted by Crdalkyl, d-dhaloalkyl, C 3 -C 6 alkenyl, C 3 -C 8 haloalkenyl, C 3 - dalkynyl, C 3 -C 6 haloalkynyl, d-dalkoxy, d-dhaloalkoxy, C 3 -C 6 alkenyloxy, C 3 - dalkynyloxy, mercapto, d-dalkylthio, d-dhaloalkylthio, C 3 -C 6 alkenylthio, C 3 - dhaloalkenylthio, C 3 -C 6 -alkynylthio, C 2 -C 5 alkoxyalkylthio, C 3 -C 5 acetylalkylthio, C 3 - C 6 alkoxycarbonylalkylthio, C 2 -C -cyanoalkylthio, CrC 6 alkylsulfinyl, d-dhaloalkylsulfinyl, d- C 6 alkylsulfonyl, CrC 6 -haloalkyIsulfonyl, aminosulfonyl, d-dalkylaminosulfonyl, di-(C C 2 alkyl)aminosulfonyl, di-(CrC 4 alkyl)amino, halogen, cyano, nitro, phenyl and benzylthio, it being possible for phenyl and benzylthio, in turn, to be substituted on the phenyl ring by d- dalkyl, d-dhaloalkyl, d-C 3 alkoxy, CrC 3 -haloalkoxy, halogen, cyano or nitro, and where the substituents on the nitrogen in the heterocyclic ring are other than halogen; and X is halogen or cyano. 13. A compound of the formula XVIa in which R 50 i is d-dhaloalkyl; R 30 ι is hydrogen; R 40 ι is hydrogen or Crdalkyl; and R 201 is CrC 6 alkyl, d-dhaloalkyl-Crdalkyl, C -C 6 alkenyl, C 2 -C 6 haloalkenyl, or d-C 2 - alkoxycarbonyl- or phenyl-substituted vinyl, C 2 -C 6 alkynyl or C -C 6 haloalkynyl; or trimethylsilyl-, hydroxyl-, d-dalkoxy-, d-dalkoxycarbonyl- or phenyl-substituted ethynyl or C 3 -C 6 allenyl; or C 3 -C 6 cycloalkyl, halogen-substituted C 3 -C 6 cycloalkyl, d-dalkoxy-d-d- alkyl, C 1 -C 4 alkyl-S(O) n4 -C 1 -C 4 alkyl, cyano-d-C 4 alkyl, CrC 4 alkoxycarbonyl-d-C 4 alkyl, C C 4 - thiocyanato, oxiranyl, CrC alkylamino-CrC alkyl, Cι-C 4 dialkylamino-Cι-C 4 alkyl, hydroxy- d-C 4 alkyl, CrCι 2 alkylthiocarbonyl-CrC 4 alkyl or formyl-d-dalkyl, or R 20 ι is a five- to ten- membered monocyclic or fused bicyclic ring system which can be aromatic or partially saturated and can contain 1 to 4 hetero atoms selected from the group consisting of nitrogen, oxygen and sulfur, the ring system being bonded to the pyridine ring via a C 1 -C 4 - alkylene, -CH=CH-, -C≡C-, -CH 2 O- , -CH 2 N(d-C 4 alkyl)-, -CH 2 S-, -CH 2 SO- or -CH 2 SO 2 - group and it not being possible for each ring system to contain more than 2 oxygen atoms and more than two sulfur atoms, and it being possible for the ring system itself to be mono-, di- or trisubstituted by d-dalkyl, d-dhaloalkyl, C 3 -C 6 alkenyl, C 3 -C 6 haloalkenyl, C 3 - dalkynyl, C 3 -C 6 haloalkynyl, d-dalkoxy, d-dhaloalkoxy, C 3 -C 6 alkenyloxy, C 3 - dalkynyloxy, mercapto, d-dalkylthio, d-dhaloalkylthio, C 3 -C 6 alkenylthio, C 3 - dhaloalkenylthio, C 3 -C 6 -alkynylthio, C 2 -C 5 alkoxyalkylthio, C 3 -C 5 acetylalkylthio, C 3 - C 6 alkoxycarbonylalkylthio, C 2 -C 4 -cyanoalkylthio, CrC 6 alkylsulfinyl, d-dhaloalkylsulfinyl, d- C 6 alkyIsulfonyl, CrC 6 -haloalkylsulfonyl, aminosulfonyl, d-dalkylaminosuifonyl, di-(d- C 2 alkyl)aminosulfonyl, di-(CrC 4 alkyl)amino, halogen, cyano, nitro, phenyl and benzylthio, it being possible for phenyl and benzylthio, in turn, to be substituted on the phenyl ring by C dalkyl, d-dhaloalkyl, d-dalkoxy, d-d-haloalkoxy, halogen, cyano or nitro, and where the substituents on the nitrogen in the heterocyclic ring are other than halogen; and X is halogen or cyano, with the proviso that, when R 50 ι is trifluoromethyl and, simultaneously, R 30 ι and R. 401 are hydrogen, then R 20 ι is other than d-dalkyl. 14. Herbicidal and plant-growth-inhibitory composition, which has a herbicidally active content of a compound of the formula I on an inert carrier. 15. A method of controlling undesired vegetation, in which a herbicidally active amount of an active ingredient of the formula I or of a composition comprising this active ingredient is applied to the plants or their environment. 16. A method of inhibiting plant growth, in which a herbicidally active amount of an active ingredient of the formula I or of a composition comprising this active ingredient is applied to the plants or their environment. 17. The use of a composition according to claim 14 for controlling undesired plant growth.

Inventors: DE MESMAEKER ALAIN, EDMUNDS ANDREW, KUNZ WALTER, LUETHY CHRISTOPH, SCHAETZER JUERGEN, SECKINGER KARL, DE MESMAEKER, ALAIN, EDMUNDS, ANDREW, KUNZ, WALTER, LUETHY, CHRISTOPH, SCHAETZER, JUERGEN, SECKINGER, KARL
Applicants: EDMUNDS ANDREW, KUNZ WALTER, LUETHY CHRISTOPH, MESMAEKER ALAIN DE, NOVARTIS AG, NOVARTIS ERFIND VERWALT GMBH, SCHAETZER JUERGEN, SECKINGER KARL, DE MESMAEKER, ALAIN, EDMUNDS, ANDREW, KUNZ, WALTER, LUETHY, CHRISTOPH, NOVARTIS-ERFINDUNGEN VERWALTUNGSGESELLSCHAFT M.B.H., SCHAETZER, JUERGEN, SECKINGER, KARL
Application year: 1999
Main classification: C07D213
IPC codes: A01N43, C07D213, C07D401, C07D405, C07D409