# Patent

## Title
3-phenylisoxazolin derivatives with herbicidal action

## Abstract

3-Phenylisoxazoline derivatives of the formula (I), and the use thereof as herbicides, are described.




In this formula (I), X2 to X6 and R1 to R3 are radicals such as hydrogen, halogen, and organic radicals such as substituted alkyl. W* is carboxyl, cyano or CHO.

## Background
CROSS REFERENCE TO RELATED APPLICATIONS
This application is a §371 National Stage Application of PCT/EP2013/069453, filed Sep. 19, 2013, which claims priority to EP 12185768.4, filed Sep. 25, 2012.
BACKGROUND
Field of the Invention
The invention relates to the technical field of herbicides, especially that of herbicides for selective control of broad-leaved weeds and weed grasses in crops of useful plants.
Description of Related Art
WO1999/05130 A1 discloses herbicidally active 3-phenylisoxazolines substituted in the 5 position by a hydroxyl and trifluoromethyl group inter alia. WO2005/021516 A1, WO1995/014680 A1, WO 2008/035315 A1, WO2005/051931 A1 and WO2005/021515 A1 each describe, inter alia, 3-phenylisoxazoline-5-carboxylic acids, -carboxylic esters and -carbaldehydes substituted on the phenyl ring in the 3 and 4 positions by alkoxy radicals. These compounds are described as precursors for preparation of pharmacologically active 3-arylisoxazoline-5-carboxamides. J. Med. Chem. 42 (1999) 2760 described the compounds methyl 3-(3-cyanophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate, ethyl 3-(3-cyanophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate, 3-(3-cyanophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylic acid and methyl 3-(3-cyanophenyl)-5-(methoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate as pharmacologically active. Indian Journal of Chemistry, Section B: Organic Chemistry Including Medicinal Chemistry (1993), 32B(9), 938-41 discloses the compound methyl 5-methyl-3-(3-nitrophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate. Izvestiya Akademii Nauk, Seriya Khimicheskaya (1996), (2), 426-429 mentions the compound methyl 3-(3,5-di-tert-butyl-4-hydroxyphenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate. Under the following CAS numbers, the compounds which follow each one are known:

    1326815-55-7: 3-(3-bromophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylic acid,
    1326814-80-5: 3-(5-bromo-2-fluorophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylic acid,
    1326811-51-1: 3-(5-bromo-2-methoxyphenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylic acid,
    1326813-57-3: 3-(3-bromo-4-methoxyphenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylic acid,
    1326814-71-4: ethyl 3-(3-chlorophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate,
    1326810-45-0: 3-(3,4-dichlorophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylic acid,
    1326815-81-9: 3-(2,5-dichlorophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylic acid,
    1326813-44-8: 3-(4-chloro-3-nitrophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylic acid,
    1326810-59-6: 3-(2-chloro-5-nitrophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylic acid,
    1326814-16-7: 3-(3-chloro-4-fluorophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylic acid,
    1326815-03-5: 3-(3-fluorophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylic acid,
    1326810-73-4: 3-(3,4-difluorophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylic acid,
    1326811-86-2: 3-(2,5-difluorophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylic acid,
    1326811-50-0: 3-(2,3-difluorophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylic acid,
    1326813-45-9: 3-(4-fluoro-3-methoxyphenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylic acid,
    1326813-37-9: 3-[2-fluoro-5-(trifluoromethyl)phenyl]-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylic acid,
    1326811-79-3: 3-(3-methoxyphenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylic acid
    1326811-74-8: 3-(2,5-dimethoxyphenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylic acid,
    1326814-78-1: 3-(3-methylphenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylic acid
    1326813-55-1: 3-(2,5-dimethylphenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylic acid,
    1326815-05-7: 5-methyl-3-(3-nitrophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylic acid,
    1326812-83-2: 5-methyl-3-[3-(trifluoromethyl)phenyl]-4,5-dihydro-1,2-oxazole-5-carboxylic acid,
    1027426-25-0: methyl 3-(3-cyanophenyl)-5-(ethoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate,
    1026410-22-9: methyl 3-(3-cyanophenyl)-5-(isopropoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate,
    1027205-06-6: methyl 5-(butoxymethyl)-3-(3-cyanophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate,
    231300-28-0: methyl 3-(3-cyanophenyl)-5-(2-methoxyethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, and
    1026948-50-4: 3-(3-cyanophenyl)-5-(trifluoromethyl)-4,5-dihydro-1,2-oxazole-5-carboxylic acid.


No herbicidal effect of the compounds known by their CAS numbers has been disclosed.
SUMMARY
It is an object of the present invention to provide herbicidally active compounds which are additionally also suitable as precursors for preparation of further herbicidally active compounds.
It has been found that particular 3-phenylisoxazoline derivatives are of particularly good suitability for this purpose. The present invention provides 3-phenylisoxazoline derivatives, or salts thereof, of the formula (I)




in which

R1 and R2 are each independently hydrogen, fluorine, chlorine, bromine, iodine, cyano, or (C1-C4)-alkyl or (C1-C4)-alkoxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine and cyano,

or

R1 and R2 together with the carbon atom to which they are bonded form a saturated or partly or fully unsaturated three-, four- or five-membered ring formed from q carbon atoms and p oxygen atoms;

R3 is fluorine, chlorine, cyano, (C1-C3)-alkylcarbonyloxy or S(O)nR5,

or (C1-C6)-alkyl, (C3-C6)-cycloalkyl, (C2-C6)-alkenyl or (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano, (C1-C4)-alkoxy and hydroxyl,

or (C1-C6)-alkylcarbonyl, (C2-C6)-alkenylcarbonyl or (C3-C6)-cycloalkylcarbonyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C6)-alkoxy;

R5 is (C1-C6)-alkyl or (C3-C6)-cycloalkyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and hydroxyl;

R6 is hydrogen or R5;

R7 is hydrogen or (C1-C6)-alkyl, (C3-C6)-cycloalkyl, (C2-C4)-alkenyl or (C2-C4)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano and (C1-C2)-alkoxy;

R8 is R7;

W* is COOH, COOY, CN or CHO;

Y is (C1-C8)-alkyl which is substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano, hydroxyl and COO—(C1-C8)-alkyl and which is interrupted by n heteroatoms from the group consisting of oxygen, sulfur and nitrogen, or

a radical from the group consisting of (cyclohex-2-en-1-one)-3-yl, (propan-1-ol)-3-yl, (2,2-dimethylpropan-1-ol)-3-yl, (methyl 2,2-dimethylpropanoate)-3-yl, (methyl propanoate)-3-yl, (ethyl propanoate)-3-yl, (ethyl butanoate)-3-yl, (ethyl (3R)-4,4,4-trifluorobutanoate)-3-yl, (butan-2-one)-4-yl, (3-methylbutan-2-one)-4-yl, (pent-3-en-2-one)-4-yl, ((2S)-dimethyl butanedioate)-2-yl, (dimethyl pentanedioate)-3-yl, (methyl (2R)-2-methylpropanoate)-3-yl, 4-methoxycarbonylbenzyl, 3,5-difluorobenzyl, 3,4-difluorobenzyl, 2,6-difluorobenzyl, 5-methylpyridin-3-ylmethyl, tetrahydrofuran-3-yl and (butan-1-ol)-4-yl;

X2, X4 and X6 are each independently hydrogen, fluorine, chlorine, bromine, iodine, cyano, nitro,

or (C1-C4)-alkyl, (C3-C5)-cycloalkyl, (C2-C4)-alkenyl, (C2-C4)-alkynyl, (C1-C4)-alkoxy, (C2-C4)-alkenyloxy, (C2-C4)-alkynyloxy or (C1-C4)-alkylcarbonyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C4)-alkoxy;

X3 is fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8SO2R5, CONR6R8, COR6, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)nR5, SO2NR6R8, OSO2NR6R8,

or (C1-C6)-alkyl, (C3-C5)-cycloalkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano,

or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy, (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy;

X5 is hydrogen, fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8SO2R5, CONR6R8, COR6, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)nR5, SO2NR6R8, OSO2NR6R8,

or (C1-C6)-alkyl, (C3-C5)-cycloalkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano,

or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy, (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy;

m is 0, 1, 2, 3, 4 or 5;

n is 0, 1 or 2;

p is 0 or 1;

q is 3, 4 or 5;

with the proviso that

a) X3 and X4 are not both substituted or unsubstituted alkoxy,

b) in the compounds in which R3 is methyl and W* is COOH, X5 is not hydrogen, and

c) the compounds

    methyl 3-(3-cyanophenyl)-5-(isopropoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate,
    methyl 5-(butoxymethyl)-3-(3-cyanophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate,
    methyl 3-(3-cyanophenyl)-5-(methoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate,
    methyl 3-(3-cyanophenyl)-5-(2-methoxyethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate,
    3-(3-cyanophenyl)-5-(trifluoromethyl)-4,5-dihydro-1,2-oxazole-5-carboxylic acid,
    methyl 3-(3-cyanophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate,
    ethyl 3-(3-cyanophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate,
    methyl 5-methyl-3-(3-nitrophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate,
    methyl 3-(3,5-di-tert-butyl-4-hydroxyphenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate and ethyl 3-(3-chlorophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate

are excluded.





DETAILED DESCRIPTION OF A PREFERRED EMBODIMENT
Alkyl means saturated straight-chain or branched hydrocarbyl radicals having the number of carbon atoms specified in each case, e.g. C1-C6-alkyl such as methyl, ethyl, propyl, 1-methylethyl, butyl, 1-methylpropyl, 2-methylpropyl, 1,1-dimethylethyl, pentyl, 1-methylbutyl, 2-methylbutyl, 3-methylbutyl, 2,2-dimethylpropyl, 1-ethylpropyl, hexyl, 1,1-dimethylpropyl, 1,2-dimethylpropyl, 1-methylpentyl, 2-methylpentyl, 3-methylpentyl, 4-methylpentyl, 1,1-dimethylbutyl, 1,2-dimethylbutyl, 1,3-dimethylbutyl, 2,2-dimethylbutyl, 2,3-dimethylbutyl, 3,3-dimethylbutyl, 1-ethylbutyl, 2-ethylbutyl, 1,1,2-trimethylpropyl, 1,2,2-trimethylpropyl, 1-ethyl-1-methylpropyl and 1-ethyl-2-methylpropyl.
Halogen-substituted alkyl means straight-chain or branched alkyl groups where some or all of the hydrogen atoms in these groups may be replaced by halogen atoms, e.g. C1-C2-haloalkyl such as chloromethyl, bromomethyl, dichloromethyl, trichloromethyl, fluoromethyl, difluoromethyl, trifluoromethyl, chlorofluoromethyl, dichlorofluoromethyl, chlorodifluoromethyl, 1-chloroethyl, 1-bromoethyl, 1-fluoroethyl, 2-fluoroethyl, 2,2-difluoroethyl, 2,2,2-trifluoroethyl, 2-chloro-2-fluoroethyl, 2-chloro-1,2-difluoroethyl, 2,2-dichloro-2-fluoroethyl, 2,2,2-trichloroethyl, pentafluoroethyl and 1,1,1-trifluoroprop-2-yl.
Alkenyl means unsaturated straight-chain or branched hydrocarbyl radicals having the number of carbon atoms specified in each case and one double bond in any position, e.g. C2-C6-alkenyl such as ethenyl, 1-propenyl, 2-propenyl, 1-methylethenyl, 1-butenyl, 2-butenyl, 3-butenyl, 1-methyl-1-propenyl, 2-methyl-1-propenyl, 1-methyl-2-propenyl, 2-methyl-2-propenyl, 1-pentenyl, 2-pentenyl, 3-pentenyl, 4-pentenyl, 1-methyl-1-butenyl, 2-methyl-1-butenyl, 3-methyl-1-butenyl, 1-methyl-2-butenyl, 2-methyl-2-butenyl, 3-methyl-2-butenyl, 1-methyl-3-butenyl, 2-methyl-3-butenyl, 3-methyl-3-butenyl, 1,1-dimethyl-2-propenyl, 1,2-dimethyl-1-propenyl, 1,2-dimethyl-2-propenyl, 1-ethyl-1-propenyl, 1-ethyl-2-propenyl, 1-hexenyl, 2-hexenyl, 3-hexenyl, 4-hexenyl, 5-hexenyl, 1-methyl-1-pentenyl, 2-methyl-1-pentenyl, 3-methyl-1-pentenyl, 4-methyl-1-pentenyl, 1-methyl-2-pentenyl, 2-methyl-2-pentenyl, 3-methyl-2-pentenyl, 4-methyl-2-pentenyl, 1-methyl-3-pentenyl, 2-methyl-3-pentenyl, 3-methyl-3-pentenyl, 4-methyl-3-pentenyl, 1-methyl-4-pentenyl, 2-methyl-4-pentenyl, 3-methyl-4-pentenyl, 4-methyl-4-pentenyl, 1,1-dimethyl-2-butenyl, 1,1-dimethyl-3-butenyl, 1,2-dimethyl-1-butenyl, 1,2-dimethyl-2-butenyl, 1,2-dimethyl-3-butenyl, 1,3-dimethyl-1-butenyl, 1,3-dimethyl-2-butenyl, 1,3-dimethyl-3-butenyl, 2,2-dimethyl-3-butenyl, 2,3-dimethyl-1-butenyl, 2,3-dimethyl-2-butenyl, 2,3-dimethyl-3-butenyl, 3,3-dimethyl-1-butenyl, 3,3-dimethyl-2-butenyl, 1-ethyl-1-butenyl, 1-ethyl-2-butenyl, 1-ethyl-3-butenyl, 2-ethyl-1-butenyl, 2-ethyl-2-butenyl, 2-ethyl-3-butenyl, 1,1,2-trimethyl-2-propenyl, 1-ethyl-1-methyl-2-propenyl, 1-ethyl-2-methyl-1-propenyl and 1-ethyl-2-methyl-2-propenyl.
Alkynyl means straight-chain or branched hydrocarbyl radicals having the number of carbon atoms specified in each case and one triple bond in any position, e.g. C2-C6-alkynyl such as ethynyl, 1-propynyl, 2-propynyl (or propargyl), 1-butynyl, 2-butynyl, 3-butynyl, 1-methyl-2-propynyl, 1-pentynyl, 2-pentynyl, 3-pentynyl, 4-pentynyl, 3-methyl-1-butynyl, 1-methyl-2-butynyl, 1-methyl-3-butynyl, 2-methyl-3-butynyl, 1,1-dimethyl-2-propynyl, 1-ethyl-2-propynyl, 1-hexynyl, 2-hexynyl, 3-hexynyl, 4-hexynyl, 5-hexynyl, 3-methyl-1-pentynyl, 4-methyl-1-pentynyl, 1-methyl-2-pentynyl, 4-methyl-2-pentynyl, 1-methyl-3-pentynyl, 2-methyl-3-pentynyl, 1-methyl-4-pentynyl, 2-methyl-4-pentynyl, 3-methyl-4-pentynyl, 1,1-dimethyl-2-butynyl, 1,1-dimethyl-3-butynyl, 1,2-dimethyl-3-butynyl, 2,2-dimethyl-3-butynyl, 3,3-dimethyl-1-butynyl, 1-ethyl-2-butynyl, 1-ethyl-3-butynyl, 2-ethyl-3-butynyl and 1-ethyl-1-methyl-2-propynyl.
Alkoxy means saturated straight-chain or branched alkoxy radicals having the number of carbon atoms stated in each case, for example C1-C6-alkoxy such as methoxy, ethoxy, propoxy, 1-methylethoxy, butoxy, 1-methylpropoxy, 2-methylpropoxy, 1,1-dimethylethoxy, pentoxy, 1-methylbutoxy, 2-methylbutoxy, 3-methylbutoxy, 2,2-dimethylpropoxy, 1-ethylpropoxy, hexoxy, 1,1-dimethylpropoxy, 1,2-dimethylpropoxy, 1-methylpentoxy, 2-methylpentoxy, 3-methylpentoxy, 4-methylpentoxy, 1,1-dimethylbutoxy, 1,2-dimethylbutoxy, 1,3-dimethylbutoxy, 2,2-dimethylbutoxy, 2,3-dimethylbutoxy, 3,3-dimethylbutoxy, 1-ethylbutoxy, 2-ethylbutoxy, 1,1,2-trimethylpropoxy, 1,2,2-trimethylpropoxy, 1-ethyl-1-methylpropoxy and 1-ethyl-2-methylpropoxy. Halogen-substituted alkoxy means straight-chain or branched alkoxy radicals having the number of carbon atoms specified in each case, where some or all of the hydrogen atoms in these groups may be replaced by halogen atoms as specified above, e.g. C1-C2-haloalkoxy such as chloromethoxy, bromomethoxy, dichloromethoxy, trichloromethoxy, fluoromethoxy, difluoromethoxy, trifluoromethoxy, chlorofluoromethoxy, dichlorofluoromethoxy, chlorodifluoromethoxy, 1-chloroethoxy, 1-bromoethoxy, 1-fluoroethoxy, 2-fluoroethoxy, 2,2-difluoroethoxy, 2,2,2-trifluoroethoxy, 2-chloro-2-fluoroethoxy, 2-chloro-1,2-difluoroethoxy, 2,2-dichloro-2-fluoroethoxy, 2,2,2-trichloroethoxy, pentafluoroethoxy and 1,1,1-trifluoroprop-2-oxy.
According to the nature of the substituents and the way in which they are joined, the compounds of the formula (I) may be present as stereoisomers. If, for example, one or more asymmetrically substituted carbon atoms and/or sulfoxides are present, enantiomers and diastereomers may occur. Stereoisomers can be obtained from the mixtures obtained in the preparation by customary separation methods, for example by chromatographic separation processes. It is likewise possible to selectively prepare stereoisomers by using stereoselective reactions with use of optically active starting materials and/or assistants. The invention also relates to all stereoisomers and mixtures thereof which are encompassed by the formula (I) but not defined specifically. For the sake of simplicity, however, reference is always made hereinafter to compounds of the formula (I), even though this means both the pure compounds and, if appropriate, mixtures having different proportions of isomeric compounds.
According to the nature of the substituents defined above, the compounds of the formula (I) have acidic properties and can form salts, and if appropriate also internal salts, or adducts with inorganic or organic bases or with metal ions.
If the compounds of the formula (I) bear hydroxyl, carboxyl or other groups which induce acidic properties, these compounds can be reacted with bases to give salts. Suitable bases are, for example, hydroxides, carbonates, hydrogencarbonates of the alkali metals and alkaline earth metals, especially those of sodium, potassium, magnesium and calcium, and also ammonia, primary, secondary and tertiary amines having C1-C4-alkyl groups, mono-, di- and trialkanolamines of C1-C4-alkanols, choline and chlorocholine.
If a group is polysubstituted by radicals, this means that this group is substituted by one or more identical or different radicals from those mentioned.
In all the formulae specified hereinafter, the substituents and symbols have the same definition as in formula (I), unless defined differently. Arrows in a chemical formula denote the points at which it is joined to the rest of the molecule.
Preference is given to 3-phenylisoxazoline derivatives of the formula (I) in which
R1 and R2 are each hydrogen,
R3 is (C1-C6)-alkyl, (C1-C4)-alkoxy-(C1-C4)-alkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl halo-(C1-C6)-alkyl or halo-(C2-C6)-alkenyl;
R5 is (C1-C6)-alkyl or (C3-C6)-cycloalkyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and hydroxyl;
R6 is hydrogen or R5;
R7 is hydrogen or (C1-C6)-alkyl, (C3-C6)-cycloalkyl, (C2-C4)-alkenyl or (C2-C4)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano and (C1-C2)-alkoxy;
R8 is R7;
W* is COOH or COOY;
Y is (C1-C6)-alkyl which is substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano, hydroxyl and COO—(C1-C4)-alkyl and which is interrupted by n oxygen atoms, or
a radical from the group consisting of (cyclohex-2-en-1-one)-3-yl, (propan-1-ol)-3-yl, (2,2-dimethylpropan-1-ol)-3-yl, (methyl 2,2-dimethylpropanoate)-3-yl, (methyl propanoate)-3-yl, (ethyl propanoate)-3-yl, (ethyl butanoate)-3-yl, (ethyl (3R)-4,4,4-trifluorobutanoate)-3-yl, (butan-2-one)-4-yl, (3-methylbutan-2-one)-4-yl, (pent-3-en-2-one)-4-yl, ((2S)-dimethyl butanedioate)-2-yl, (dimethyl pentanedioate)-3-yl, (methyl (2R)-2-methylpropanoate)-3-yl, 4-methoxycarbonylbenzyl, 3,5-difluorobenzyl, 3,4-difluorobenzyl, 2,6-difluorobenzyl, 5-methylpyridin-3-ylmethyl, tetrahydrofuran-3-yl and (butan-1-ol)-4-yl;

X2, X4 and X6 are each independently hydrogen, fluorine, chlorine, bromine, iodine, cyano, nitro,

or (C1-C4)-alkyl, (C3-C5)-cycloalkyl, (C2-C4)-alkenyl, (C2-C4)-alkynyl, (C1-C4)-alkoxy, (C2-C4)-alkenyloxy, (C2-C4)-alkynyloxy or (C1-C4)-alkylcarbonyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C4)-alkoxy;

X3 is fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8SO2R5, CONR6R8, CORE, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)nR5, SO2NR6R8, OSO2NR6R8,

or (C1-C6)-alkyl, (C3-C5)-cycloalkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano,

or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy, (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy;

X5 is hydrogen, fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8SO2R5, CONR6R8, CORE, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)nR5, SO2NR6R8, OSO2NR6R8,

or (C1-C6)-alkyl, (C3-C5)-cycloalkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano,

or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy, (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy;

m is 0, 1, 2, 3, 4 or 5;

n is 0, 1 or 2;

with the proviso that

a) X3 and X4 are not both substituted or unsubstituted alkoxy,

b) in the compounds in which R3 is methyl and W* is COOH, X5 is not hydrogen, and

c) the compounds

    methyl 3-(3-cyanophenyl)-5-(isopropoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 5-(butoxymethyl)-3-(3-cyanophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 3-(3-cyanophenyl)-5-(methoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 3-(3-cyanophenyl)-5-(2-methoxyethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate,
    3-(3-cyanophenyl)-5-(trifluoromethyl)-4,5-dihydro-1,2-oxazole-5-carboxylic acid,
    methyl 3-(3-cyanophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate,
    ethyl 3-(3-cyanophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate,
    methyl 5-methyl-3-(3-nitrophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate,
    methyl 3-(3,5-di-tert-butyl-4-hydroxyphenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate and ethyl 3-(3-chlorophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate

are excluded.



Particular preference is given to 3-phenylisoxazoline derivatives of the formula (I) in which
R1 and R2 are each hydrogen,
R3 is (C1-C4)-alkyl, (C1-C4)-alkoxy-(C1-C4)-alkyl, vinyl, (C2-C4)-alkynyl, halo-(C1-C4)-alkyl or halo-(C2-C4)-alkenyl;
R5 is methyl or ethyl;
R6 is hydrogen or R5;
R7 is hydrogen or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine;
R8 is R7;
W* is COOH or COOY;
Y is (C1-C6)-alkyl which is substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano, hydroxyl and COO—(C1-C4)-alkyl and which is interrupted by n oxygen atoms, or
a radical from the group consisting of (cyclohex-2-en-1-one)-3-yl, (propan-1-ol)-3-yl, (2,2-dimethylpropan-1-ol)-3-yl, (methyl 2,2-dimethylpropanoate)-3-yl, (methyl propanoate)-3-yl, (ethyl propanoate)-3-yl, (ethyl butanoate)-3-yl, (ethyl (3R)-4,4,4-trifluorobutanoate)-3-yl, (butan-2-one)-4-yl, (3-methylbutan-2-one)-4-yl, (pent-3-en-2-one)-4-yl, ((2S)-dimethyl butanedioate)-2-yl, (dimethyl pentanedioate)-3-yl, (methyl (2R)-2-methylpropanoate)-3-yl, 4-methoxycarbonylbenzyl, 3,5-difluorobenzyl, 3,4-difluorobenzyl, 2,6-difluorobenzyl, 5-methylpyridin-3-ylmethyl, tetrahydrofuran-3-yl and (butan-1-ol)-4-yl;

X2, X4 and X6 are each independently hydrogen, fluorine, or chlorine,

or (C1-C4)-alkyl or (C1-C4)-alkoxy each substituted by m radicals from the group consisting of fluorine, chlorine, cyano and (C1-C4)-alkoxy;

X3 is fluorine, chlorine, bromine, cyano,

or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine,

or (C1-C6)-alkoxy substituted by m radicals from the group consisting of fluorine and chlorine;

X5 is hydrogen, fluorine, chlorine, bromine, cyano,

or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine,

or (C1-C6)-alkoxy substituted by m radicals from the group consisting of fluorine and chlorine;

m is 0, 1, 2 or 3;

n is 0, 1 or 2;

with the proviso that

a) X3 and X4 are not both substituted or unsubstituted alkoxy,

b) in the compounds in which R3 is methyl and W* is COOH, X5 is not hydrogen, and

c) the compounds

    methyl 3-(3-cyanophenyl)-5-(isopropoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate,
    methyl 5-(butoxymethyl)-3-(3-cyanophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate,
    methyl 3-(3-cyanophenyl)-5-(methoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate,
    methyl 3-(3-cyanophenyl)-5-(2-methoxyethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate,
    3-(3-cyanophenyl)-5-(trifluoromethyl)-4,5-dihydro-1,2-oxazole-5-carboxylic acid,
    methyl 3-(3-cyanophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate,
    ethyl 3-(3-cyanophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate,
    methyl 5-methyl-3-(3-nitrophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate,
    methyl 3-(3,5-di-tert-butyl-4-hydroxyphenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate and ethyl 3-(3-chlorophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate

are excluded.



Very particular preference is given to 3-phenylisoxazoline derivatives of the formula (I) in which
R1 and R2 are each hydrogen,
R3 is (C1-C4)-alkyl, (C1-C4)-alkoxy-(C1-C4)-alkyl, vinyl, (C2-C4)-alkynyl, halo-(C1-C4)-alkyl or halo-(C2-C4)-alkenyl;
R5 is methyl or ethyl;
R6 is hydrogen or R5;
R7 is hydrogen or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine;
R8 is R7;
W* is COOH or COOY;
Y is (C1-C6)-alkyl which is substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano, hydroxyl and COO—(C1-C4)-alkyl and which is interrupted by n oxygen atoms, or
a radical from the group consisting of (cyclohex-2-en-1-one)-3-yl, (propan-1-ol)-3-yl, (2,2-dimethylpropan-1-ol)-3-yl, (methyl 2,2-dimethylpropanoate)-3-yl, (methyl propanoate)-3-yl, (ethyl propanoate)-3-yl, (ethyl butanoate)-3-yl, (ethyl (3R)-4,4,4-trifluorobutanoate)-3-yl, (butan-2-one)-4-yl, (3-methylbutan-2-one)-4-yl, (pent-3-en-2-one)-4-yl, ((2S)-dimethyl butanedioate)-2-yl, (dimethyl pentanedioate)-3-yl, (methyl (2R)-2-methylpropanoate)-3-yl, 4-methoxycarbonylbenzyl, 3,5-difluorobenzyl, 3,4-difluorobenzyl, 2,6-difluorobenzyl, 5-methylpyridin-3-ylmethyl, tetrahydrofuran-3-yl and (butan-1-ol)-4-yl;

X2, X4 and X6 are each independently hydrogen, fluorine, or chlorine,

or (C1-C4)-alkyl or (C1-C4)-alkoxy each substituted by m radicals from the group consisting of fluorine, chlorine, cyano and C1-C4)-alkoxy;

X3 is fluorine, chlorine, bromine, cyano,

or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine,

or (C1-C6)-alkoxy substituted by m radicals from the group consisting of fluorine and chlorine;

X5 is fluorine, chlorine, bromine, cyano,

or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine,

or (C1-C6)-alkoxy substituted by m radicals from the group consisting of fluorine and chlorine;

m is 0, 1, 2 or 3;

n is 0, 1 or 2;

with the proviso that

a) X3 and X4 are not both substituted or unsubstituted alkoxy,

b) in the compounds in which R3 is methyl and W* is COOH, X5 is not hydrogen, and

c) the compounds

    methyl 3-(3-cyanophenyl)-5-(isopropoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate,
    methyl 5-(butoxymethyl)-3-(3-cyanophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate,
    methyl 3-(3-cyanophenyl)-5-(methoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate,
    methyl 3-(3-cyanophenyl)-5-(2-methoxyethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate,
    3-(3-cyanophenyl)-5-(trifluoromethyl)-4,5-dihydro-1,2-oxazole-5-carboxylic acid,
    methyl 3-(3-cyanophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate,
    ethyl 3-(3-cyanophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate,
    methyl 5-methyl-3-(3-nitrophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate,
    methyl 3-(3,5-di-tert-butyl-4-hydroxyphenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate and ethyl 3-(3-chlorophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate

are excluded.



The compounds described in the documents cited above have not only pharmacological action but also, surprisingly, herbicidal action. Furthermore, they are outstandingly suitable as intermediates for preparation of herbicidally active 3-phenylisoxazoline-5-carboxamides and 3-phenylisoxazoline-5-thioamides. The present invention therefore further provides for the use of 3-phenylisoxazoline derivatives of the formula (Ia) as herbicides. The present invention therefore further provides for the use of 3-phenylisoxazoline derivatives of the formula (Ia) as intermediates for preparation of herbicidally active 3-phenylisoxazoline-5-carboxamides and 3-phenylisoxazoline-5-thioamides.




In formula (Ia), the radicals and indices are defined as follows:
R1 and R2 are each independently hydrogen, fluorine, chlorine, bromine, iodine, cyano, or (C1-C4)-alkyl or (C1-C4)-alkoxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine and cyano,
or
R1 and R2 together with the carbon atom to which they are bonded form a saturated or partly or fully unsaturated three-, four- or five-membered ring formed from q carbon atoms and p oxygen atoms;
R3 is fluorine, chlorine, cyano, (C1-C3)-alkylcarbonyloxy or S(O)nR5,
or (C1-C6)-alkyl, (C3-C6)-cycloalkyl, (C2-C6)-alkenyl or (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano, (C1-C4)-alkoxy and hydroxyl,
or (C1-C6)-alkylcarbonyl, (C2-C6)-alkenylcarbonyl or (C3-C6)-cycloalkylcarbonyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C6)-alkoxy;
R5 is (C1-C6)-alkyl or (C3-C6)-cycloalkyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and hydroxyl;
R6 is hydrogen or R5;
R7 is hydrogen or (C1-C6)-alkyl, (C3-C6)-cycloalkyl, (C2-C4)-alkenyl or (C2-C4)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano and (C1-C2)-alkoxy;
R8 is R7;
W* is COOH, COOY, CN or CHO;
Y is (C1-C8)-alkyl which is substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano, hydroxyl and COO—(C1-C8)-alkyl and which is interrupted by n heteroatoms from the group consisting of oxygen, sulfur and nitrogen, or
a radical from the group consisting of (cyclohex-2-en-1-one)-3-yl, (propan-1-ol)-3-yl, (2,2-dimethylpropan-1-ol)-3-yl, (methyl 2,2-dimethylpropanoate)-3-yl, (methyl propanoate)-3-yl, (ethyl propanoate)-3-yl, (ethyl butanoate)-3-yl, (ethyl (3R)-4,4,4-trifluorobutanoate)-3-yl, (butan-2-one)-4-yl, (3-methylbutan-2-one)-4-yl, (pent-3-en-2-one)-4-yl, ((2S)-dimethyl butanedioate)-2-yl, (dimethyl pentanedioate)-3-yl, (methyl (2R)-2-methylpropanoate)-3-yl, 4-methoxycarbonylbenzyl, 3,5-difluorobenzyl, 3,4-difluorobenzyl, 2,6-difluorobenzyl, 5-methylpyridin-3-ylmethyl, tetrahydrofuran-3-yl and (butan-1-ol)-4-yl;

X2, X4 and X6 are each independently hydrogen, fluorine, chlorine, bromine, iodine, cyano, nitro,

or (C1-C4)-alkyl, (C3-C5)-cycloalkyl, (C2-C4)-alkenyl, (C2-C4)-alkynyl, (C1-C4)-alkoxy, (C2-C4)-alkenyloxy, (C2-C4)-alkynyloxy or (C1-C4)-alkylcarbonyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C4)-alkoxy;

X3 is fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8SO2R5, CONR6R8, COR6, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)nR5, SO2NR6R8, OSO2NR6R8,

or (C1-C6)-alkyl, (C3-C5)-cycloalkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano,

or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy, (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy;

X5 is hydrogen, fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8SO2R5, CONR6R8, COR6, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)nR5, SO2NR6R8, OSO2NR6R8,

or (C1-C6)-alkyl, (C3-C5)-cycloalkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano,

or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy, (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy;

m is 0, 1, 2, 3, 4 or 5;

n is 0, 1 or 2;

p is 0 or 1;

q is 3, 4 or 5.

Preferentially suitable as herbicides and intermediates are 3-phenylisoxazoline derivatives of the formula (Ia) in which
R1 and R2 are each hydrogen,
R3 is (C1-C6)-alkyl, (C1-C4)-alkoxy-(C1-C4)-alkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl, halo-(C1-C6)-alkyl or halo-(C2-C6)-alkenyl;
R5 is (C1-C6)-alkyl or (C3-C6)-cycloalkyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and hydroxyl;
R6 is hydrogen or R5;
R7 is hydrogen or (C1-C6)-alkyl, (C3-C6)-cycloalkyl, (C2-C4)-alkenyl or (C2-C4)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano and (C1-C2)-alkoxy;
R8 is R7;
W* is COOH or COOY;
Y is (C1-C6)-alkyl which is substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano, hydroxyl and COO—(C1-C4)-alkyl and which is interrupted by n oxygen atoms, or
a radical from the group consisting of (cyclohex-2-en-1-one)-3-yl, (propan-1-ol)-3-yl, (2,2-dimethylpropan-1-ol)-3-yl, (methyl 2,2-dimethylpropanoate)-3-yl, (methyl propanoate)-3-yl, (ethyl propanoate)-3-yl, (ethyl butanoate)-3-yl, (ethyl (3R)-4,4,4-trifluorobutanoate)-3-yl, (butan-2-one)-4-yl, (3-methylbutan-2-one)-4-yl, (pent-3-en-2-one)-4-yl, ((2S)-dimethyl butanedioate)-2-yl, (dimethyl pentanedioate)-3-yl, (methyl (2R)-2-methylpropanoate)-3-yl, 4-methoxycarbonylbenzyl, 3,5-difluorobenzyl, 3,4-difluorobenzyl, 2,6-difluorobenzyl, 5-methylpyridin-3-ylmethyl, tetrahydrofuran-3-yl and (butan-1-ol)-4-yl;

X2, X4 and X6 are each independently hydrogen, fluorine, chlorine, bromine, iodine, cyano, nitro,

or (C1-C4)-alkyl, (C3-C5)-cycloalkyl, (C2-C4)-alkenyl, (C2-C4)-alkynyl, (C1-C4)-alkoxy, (C2-C4)-alkenyloxy, (C2-C4)-alkynyloxy or (C1-C4)-alkylcarbonyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C4)-alkoxy;

X3 is fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8SO2R5, CONR6R8, COR6, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)nR5, SO2NR6R8, OSO2NR6R8,

or (C1-C6)-alkyl, (C3-C5)-cycloalkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by

m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano,

or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy, (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy;

X5 is hydrogen, fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8SO2R5, CONR6R8, COR6, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)nR5, SO2NR6R8, OSO2NR6R8,

or (C1-C6)-alkyl, (C3-C5)-cycloalkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano,

or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy, (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy;

m is 0, 1, 2, 3, 4 or 5;

n is 0, 1 or 2.

More preferentially suitable as herbicides and intermediates are 3-phenylisoxazoline derivatives of the formula (Ia) in which
R1 and R2 are each hydrogen,
R3 is (C1-C4)-alkyl, (C1-C4)-alkoxy-(C1-C4)-alkyl, vinyl, (C2-C4)-alkynyl, halo-(C1-C6)-alkyl or halo-(C2-C6)-alkenyl;
R5 is methyl or ethyl;
R6 is hydrogen or R5;
R7 is hydrogen or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine;
R8 is R7;
W* is COOH or COOY;
Y is (C1-C6)-alkyl which is substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano, hydroxyl and COO—(C1-C4)-alkyl and which is interrupted by n oxygen atoms, or
a radical from the group consisting of (cyclohex-2-en-1-one)-3-yl, (propan-1-ol)-3-yl, (2,2-dimethylpropan-1-ol)-3-yl, (methyl 2,2-dimethylpropanoate)-3-yl, (methyl propanoate)-3-yl, (ethyl propanoate)-3-yl, (ethyl butanoate)-3-yl, (ethyl (3R)-4,4,4-trifluorobutanoate)-3-yl, (butan-2-one)-4-yl, (3-methylbutan-2-one)-4-yl, (pent-3-en-2-one)-4-yl, ((2S)-dimethyl butanedioate)-2-yl, (dimethyl pentanedioate)-3-yl, (methyl (2R)-2-methylpropanoate)-3-yl, 4-methoxycarbonylbenzyl, 3,5-difluorobenzyl, 3,4-difluorobenzyl, 2,6-difluorobenzyl, 5-methylpyridin-3-ylmethyl, tetrahydrofuran-3-yl and (butan-1-ol)-4-yl;

X2, X4 and X6 are each independently hydrogen, fluorine, or chlorine,

or (C1-C4)-alkyl or (C1-C4)-alkoxy each substituted by m radicals from the group consisting of fluorine, chlorine, cyano and (C1-C4)-alkoxy;

X3 is fluorine, chlorine, bromine, cyano,

or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine,

or (C1-C6)-alkoxy substituted by m radicals from the group consisting of fluorine and chlorine;

X5 is hydrogen, fluorine, chlorine, bromine, cyano,

or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine,

or (C1-C6)-alkoxy substituted by m radicals from the group consisting of fluorine and chlorine;

m is 0, 1, 2 or 3;

n is 0, 1 or 2.

Most preferentially suitable as herbicides and intermediates are 3-phenylisoxazoline derivatives of the formula (Ia) in which
R1 and R2 are each hydrogen,
R3 is (C1-C4)-alkyl, (C1-C4)-alkoxy-(C1-C4)-alkyl, vinyl, (C2-C4)-alkynyl, halo-(C1-C6)-alkyl or halo-(C2-C6)-alkenyl;
R5 is methyl or ethyl;
R6 is hydrogen or R5;
R7 is hydrogen or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine;
R8 is R7;
W* is COOH or COOY;
Y is (C1-C6)-alkyl which is substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano, hydroxyl and COO—(C1-C4)-alkyl and which is interrupted by n oxygen atoms, or
a radical from the group consisting of (cyclohex-2-en-1-one)-3-yl, (propan-1-ol)-3-yl, (2,2-dimethylpropan-1-ol)-3-yl, (methyl 2,2-dimethylpropanoate)-3-yl, (methyl propanoate)-3-yl, (ethyl propanoate)-3-yl, (ethyl butanoate)-3-yl, (ethyl (3R)-4,4,4-trifluorobutanoate)-3-yl, (butan-2-one)-4-yl, (3-methylbutan-2-one)-4-yl, (pent-3-en-2-one)-4-yl, ((2S)-dimethyl butanedioate)-2-yl, (dimethyl pentanedioate)-3-yl, (methyl (2R)-2-methylpropanoate)-3-yl, 4-methoxycarbonylbenzyl, 3,5-difluorobenzyl, 3,4-difluorobenzyl, 2,6-difluorobenzyl, 5-methylpyridin-3-ylmethyl, tetrahydrofuran-3-yl and (butan-1-ol)-4-yl;

X2, X4 and X6 are each independently hydrogen, fluorine, or chlorine,

or (C1-C4)-alkyl or (C1-C4)-alkoxy each substituted by m radicals from the group consisting of fluorine, chlorine, cyano and (C1-C4)-alkoxy;

X3 is fluorine, chlorine, bromine, cyano,

or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine,

or (C1-C6)-alkoxy substituted by m radicals from the group consisting of fluorine and chlorine;

X5 is hydrogen, fluorine, chlorine, bromine, cyano,

or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine,

or (C1-C6)-alkoxy substituted by m radicals from the group consisting of fluorine and chlorine;

m is 0, 1, 2 or 3;

n is 0, 1 or 2.

Inventive compounds in which W* is COOH can be prepared by reactions known per se to those skilled in the art, for example by the reaction sequence shown in scheme 1.




In scheme 1 and the schemes which follow, (X)n represents the substituents X2, X3, X4, X5 and X6. Such 1,3-dipolar cycloadditions of nitrile oxides with suitable dipolarophiles are described, for example, in reviews: 1,3 dipolar Cycloaddition Chemistry, Padwa (editor), Wiley, New York, 1984; Kanemasa and Tsuge, Heterocycles 1990, 30, 719 and H. Feurer, Nitrones and Nitronates in Organic Synthesis, Second Edition, 1-129, Hoboken, N.J. 2008.
The cycloadditions can be performed in a one-pot reaction without isolation of the dipole precursor or with isolation of the dipole precursor.
Inventive compounds substituted in the 4 and 5 positions of the isoxazoline ring system can likewise be prepared by 1,3-dipolar cycloaddition by using suitably 1,2-disubstituted olefins as dipolarophiles. Usually, this reaction gives diastereomer mixtures which can be separated by column chromatography. Optically active isoxazolines can be obtained by chiral HPLC of suitable precursors or end products, and likewise by enantioselective reactions, for example enzymatic ester or amide cleavage or through the use of chiral auxiliaries on the dipolarophile, as described by Olssen (J. Org. Chem. 1988, 53, 2468). As well as the inventive acids (W*═COOH), salts thereof are also claimed, these being preparable by the customary route through reaction with an inorganic or organic base (scheme 2). In this scheme, Me+ represents a metal cation.




Inventive compounds in which W* is COOH can also be prepared by the methods specified in scheme 3a, by hydrolysis of anhydrides or hydrolysis of nitriles, or by the methods specified in scheme 3ba, by oxidation of alcohols or aldehydes.











Inventive compounds in which W* is COOY can be prepared, for example, according to scheme 4, by conversion of inventive compounds in which W* is COOH with addition of mineral acids and an appropriate alcohol, or by reaction of the particular acid halide with the respective alcohol or by coupling of the particular acid with coupling reagents.




Inventive compounds in which W* is CN can be prepared, for example, according to scheme 5 by cycloaddition or with dehydrating agents from a carboxamide or an aldoxime (The Chemistry of the Cyano Group, pp. 92-96, pp. 1345-1390, Interscience, New York, 1970).




Inventive compounds in which W* is CHO can be prepared, for example, according to scheme 6 by selective reduction of carboxylic acids, carboxylic esters, carbonyl halides, or of Weinreb amides, or by oxidation of alcohols or hydrolysis of




A general synthesis option for preparation of the inventive compounds 1 is the cycloaddition described in scheme 7 with dihaloformoximes (dichloroformoxime: Wade, Peter A.; Singh, Shankar M.; Pillay, M. Krishna, Tetrahedron (1984), 40(3), 601-11 and dibromoformoxime: DE 3612278) and subsequent introduction of the phenyl ring by means of Suzuki coupling (EP 0 792 870 A1) or Stille reaction (WO 2004/029066 A1).




Transformations of the functional group R3 are possible either at the alkene stage or at the isoxazoline stage. Scheme 8 describes preparation methods for different inventive 3-phenyl isoxazoline derivatives.




Commercially available methyl 2-bromomethylacrylate can be reacted under basic conditions with alcohols to give methyl 2-alkoxymethylacrylates, which then react with chloroximes via the nitrile oxides to give 3-phenyl-5-methoxymethylisoxazolines. Various 2-alkylacrylic esters can be prepared proceeding from methyl 2-bromomethylacrylate, for example by reaction with organometallic reagents. Such methods are described, for example, in Metzger, Albrecht; Piller, Fabian M.; Knochel, Paul; Chemical Communications, 2008, 44, pp. 5824-5826, and are also known from WO2006/33551.

    Chem. Ber., 1963, 96, 1373; Tanoury, G. J.; Chen, M.; Dong, Y.; Forslund, R. E.; Magdziak, D.; Organic Letters, 2008, 10, 185.


Collections of compounds of the formula (I) and/or salts thereof which can be synthesized by the abovementioned reactions can also be prepared in a parallelized manner, in which case this may be accomplished in a manual, partly automated or fully automated manner. It is possible, for example, to automate the conduct of the reaction, the workup or the purification of the products and/or intermediates. Overall, this is understood to mean a procedure as described, for example, by D. Tiebes in Combinatorial Chemistry—Synthesis, Analysis, Screening (editor: Gunther Jung), Wiley, 1999, on pages 1 to 34.
For the parallelized conduct of the reaction and workup, it is possible to use a number of commercially available instruments, for example Calypso reaction blocks from Barnstead International, Dubuque, Iowa 52004-0797, USA or reaction stations from Radleys, Shirehill, Saffron Walden, Essex, CB11 3AZ, England, or MultiPROBE Automated Workstations from PerkinElmer, Waltham, Mass. 02451, USA. For the parallelized purification of compounds of the formula (I) and salts thereof or of intermediates which occur in the course of preparation, available apparatuses include chromatography apparatuses, for example from ISCO, Inc., 4700 Superior Street, Lincoln, Nebr. 68504, USA.
The apparatuses detailed lead to a modular procedure in which the individual working steps are automated, but manual operations have to be carried out between the working steps. This can be circumvented by using partly or fully integrated automation systems in which the respective automation modules are operated, for example, by robots. Automation systems of this type can be purchased, for example, from Caliper, Hopkinton, Mass. 01748, USA.
The implementation of single or multiple synthesis steps can be supported by the use of polymer-supported reagents/scavenger resins. The specialist literature describes a series of experimental protocols, for example in ChemFiles, Vol. 4, No. 1, Polymer-Supported Scavengers and Reagents for Solution-Phase Synthesis (Sigma-Aldrich).
Aside from the methods described here, the compounds of the formula (I) and salts thereof can be prepared completely or partially by solid-phase supported methods. For this purpose, individual intermediates or all intermediates in the synthesis or a synthesis adapted for the corresponding procedure are bound to a synthesis resin. Solid phase-supported synthesis methods are described adequately in the technical literature, for example Barry A. Bunin in “The Combinatorial Index”, Academic Press, 1998 and Combinatorial Chemistry—Synthesis, Analysis, Screening (editor: Gunther Jung), Wiley, 1999. The use of solid phase-supported synthesis methods permits a number of protocols known from the literature, and these may again be executed manually or in an automated manner. The reactions can be performed, for example, by means of IRORI technology in microreactors from Nexus Biosystems, 12140 Community Road, Poway, Calif. 92064, USA.
Either on a solid phase or in the liquid phase, the performance of single or multiple synthesis steps can be supported by the use of microwave technology. The technical literature describes a number of experimental protocols, for example in Microwaves in Organic and Medicinal Chemistry (editors: C. O. Kappe and A. Stadler), Wiley, 2005.
The preparation by the processes described here gives compounds of the formula (I) and salts thereof in the form of substance collections, which are called libraries. The present invention also provides libraries comprising at least two compounds of the formula (I) and salts thereof.
The inventive compounds of the formula (I) (and/or salts thereof), collectively referred to hereinafter as “inventive compounds”, have excellent herbicidal efficacy against a broad spectrum of economically important monocotyledonous and dicotyledonous annual harmful plants. The active ingredients also have good control over perennial harmful plants which are difficult to control and produce shoots from rhizomes, root stocks or other perennial organs.
The present invention therefore also provides a method for controlling unwanted plants or for regulating the growth of plants, preferably in plant crops, in which one or more inventive compound(s) is/are applied to the plants (for example harmful plants such as monocotyledonous or dicotyledonous weeds or unwanted crop plants), to the seeds (for example grains, seeds or vegetative propagules such as tubers or shoot parts with buds) or to the area on which the plants grow (for example the area under cultivation). The inventive compounds can be deployed, for example, prior to sowing (if appropriate also by incorporation into the soil), prior to emergence or after emergence. Specific examples of some representatives of the monocotyledonous and dicotyledonous weed flora which can be controlled by the inventive compounds are as follows, though the enumeration is not intended to impose a restriction to particular species:
Monocotyledonous harmful plants of the genera: Aegilops, Agropyron, Agrostis, Alopecurus, Apera, Avena, Brachiaria, Bromus, Cenchrus, Commelina, Cynodon, Cyperus, Dactyloctenium, Digitaria, Echinochloa, Eleocharis, Eleusine, Eragrostis, Eriochloa, Festuca, Fimbristylis, Heteranthera, Imperata, Ischaemum, Leptochloa, Lolium, Monochoria, Panicum, Paspalum, Phalaris, Phleum, Poa, Rottboellia, Sagittaria, Scirpus, Setaria, Sorghum. 
Dicotyledonous weeds of the genera: Abutilon, Amaranthus, Ambrosia, Anoda, Anthemis, Aphanes, Artemisia, Atriplex, Bellis, Bidens, Capsella, Carduus, Cassia, Centaurea, Chenopodium, Cirsium, Convolvulus, Datura, Desmodium, Emex, Erysimum, Euphorbia, Galeopsis, Galinsoga, Galium, Hibiscus, Ipomoea, Kochia, Lamium, Lepidium, Lindernia, Matricaria, Mentha, Mercurialis, Mullugo, Myosotis, Papaver, Pharbitis, Plantago, Polygonum, Portulaca, Ranunculus, Raphanus, Rorippa, Rotala, Rumex, Salsola, Senecio, Sesbania, Sida, Sinapis, Solanum, Sonchus, Sphenoclea, Stellaria, Taraxacum, Thlaspi, Trifolium, Urtica, Veronica, Viola, Xanthium. 
When the inventive compounds are applied to the soil surface before germination, either the weed seedlings are prevented completely from emerging or the weeds grow until they have reached the cotyledon stage, but then stop growing and eventually, after three to four weeks have elapsed, die completely.
If the active ingredients are applied post-emergence to the green parts of the plants, growth stops after the treatment, and the harmful plants remain at the growth stage of the time of application, or die completely after a certain time, such that competition by the weeds, which is harmful to the crop plants, is thus eliminated very early and in a lasting manner.
Although the inventive compounds have excellent herbicidal activity against monocotyledonous and dicotyledonous weeds, crop plants of economically important crops, for example dicotyledonous crops of the genera Arachis, Beta, Brassica, Cucumis, Cucurbita, Helianthus, Daucus, Glycine, Gossypium, Ipomoea, Lactuca, Linum, Lycopersicon, Nicotiana, Phaseolus, Pisum, Solanum, Vicia, or monocotyledonous crops of the genera Allium, Ananas, Asparagus, Avena, Hordeum, Oryza, Panicum, Saccharum, Secale, Sorghum, Triticale, Triticum, Zea, especially Zea and Triticum, are damaged only to an insignificant extent, if at all, depending on the structure of the respective inventive compound and the application rate thereof. For these reasons, the present compounds are very suitable for selective control of unwanted plant growth in plant crops such as agriculturally useful plants or ornamentals.
Furthermore, the inventive compounds (depending on their particular structure and the application rate applied) have outstanding growth-regulating properties in crop plants. They intervene to regulate the plant's metabolism and can thus be used for controlled influence on plant constituents and to facilitate harvesting, for example by triggering desiccation and stunted growth. In addition, they are also suitable for general control and inhibition of unwanted vegetative growth without killing the plants. Inhibiting vegetative growth plays a major role for many monocotyledonous and dicotyledonous crops, since, for example, this can reduce or completely prevent lodging.
Because of their herbicidal and plant growth-regulating properties, the active ingredients can also be used to control harmful plants in crops of known genetically modified plants or of those yet to be developed. In general, transgenic plants are notable for special advantageous properties, for example for resistances to certain pesticides, in particular certain herbicides, resistances to plant diseases or organisms that cause plant diseases, such as certain insects or microorganisms such as fungi, bacteria or viruses. Other special properties relate, for example, to the harvested material with regard to quantity, quality, storability, composition and specific constituents. Thus, transgenic plants are known whose starch content is increased, or whose starch quality is altered, or those where the harvested material has a different fatty acid composition. Further special properties may be tolerance or resistance to abiotic stress factors, for example heat, cold, drought, salinity and ultraviolet radiation.
Preference is given to the use of the inventive compounds of the formula (I) or salts thereof in economically important transgenic crops of useful plants and ornamental plants, for example of cereals such as wheat, barley, rye, oats, sorghum and millet, rice, cassava and corn, or else crops of sugar beet, cotton, soybean, oilseed rape, potatoes, tomatoes, peas and other vegetables.
The compounds of the formula (I) can preferably be used as herbicides in crops of useful plants which are resistant, or have been made resistant by recombinant means, to the phytotoxic effects of the herbicides.
Conventional ways of producing novel plants which have modified properties in comparison to plants which have occurred to date consist, for example, in traditional breeding methods and the generation of mutants. Alternatively, novel plants with altered properties can be generated with the aid of recombinant methods (see, for example, EP 0221044, EP 0131624). For example, there have been descriptions of several cases of genetic modifications of crop plants for the purpose of modifying the starch synthesized in the plants (e.g. WO 92/011376 A, WO 92/014827 A, WO 91/019806 A),
transgenic crop plants resistant to particular herbicides of the glufosinate type (cf., for example, EP 0242236 A, EP 0242246 A) or of the glyphosate type (WO 92/000377A) or of the sulfonylurea type (EP 0257993 A, U.S. Pat. No. 5,013,659) or to combinations or mixtures of these herbicides through “gene stacking”, such as transgenic crop plants, for example corn or soybean with the tradename or the designation OptimumTM GATTM (Glyphosate ALS Tolerant),

    
    
        transgenic crop plants, for example cotton, capable of producing Bacillus thuringiensis toxins (Bt toxins), which make the plants resistant to particular pests (EP-A-0142924, EP-A-0193259),
        transgenic crop plants having a modified fatty acid composition (WO 91/013972 A),
        genetically modified crop plants having novel constituents or secondary metabolites, for example novel phytoalexins, which cause an increase in disease resistance (EP 0309862 A, EP 0464461 A),
        genetically modified plants having reduced photorespiration, which have higher yields and higher stress tolerance (EP 0305398 A),
        transgenic crop plants which produce pharmaceutically or diagnostically important proteins (“molecular pharming”),
        transgenic crop plants which are notable for higher yields or better quality, transgenic crop plants which are notable for a combination, for example, of the abovementioned novel properties (“gene stacking”).
    
    


Numerous molecular biology techniques which can be used to produce novel transgenic plants with modified properties are known in principle; see, for example, I. Potrykus and G. Spangenberg (eds.), Gene Transfer to Plants, Springer Lab Manual (1995), Springer Verlag Berlin, Heidelberg or Christou, “Trends in Plant Science” 1 (1996) 423-431).
For such recombinant manipulations, nucleic acid molecules which allow mutagenesis or a sequence change by recombination of DNA sequences can be introduced into plasmids. With the aid of standard methods, it is possible, for example, to undertake base exchanges, remove parts of sequences or add natural or synthetic sequences. For the connection of the DNA fragments to one another, it is possible to add adapters or linkers to the fragments; see, for example, Sambrook et al., 1989, Molecular Cloning, A Laboratory Manual, 2nd ed., Cold Spring Harbor Laboratory Press, Cold Spring Harbor, N.Y.; or Winnacker “Gene and Klone”, VCH Weinheim, 2nd edition, 1996.
The production of plant cells with a reduced activity of a gene product can be achieved, for example, by the expression of at least one appropriate antisense RNA, or of a sense RNA for achievement of a cosuppression effect, or the expression of at least one appropriately constructed ribozyme which specifically cleaves transcripts of the abovementioned gene product. For this purpose, it is firstly possible to use DNA molecules which comprise the entire coding sequence of a gene product including any flanking sequences present, or else DNA molecules which comprise only parts of the coding sequence, in which case these parts must be long enough to bring about an antisense effect in the cells. It is also possible to use DNA sequences which have a high degree of homology to the coding sequences of a gene product, but are not completely identical.
When expressing nucleic acid molecules in plants, the protein synthesized may be localized in any desired compartment of the plant cell. However, to achieve localization in a particular compartment, it is possible, for example, to link the coding region with DNA sequences which ensure localization in a particular compartment. Such sequences are known to those skilled in the art (see, for example, Braun et al., EMBO J. 11 (1992), 3219-3227; Wolter et al., Proc. Natl. Acad. Sci. USA 85 (1988), 846-850; Sonnewald et al., Plant J. 1 (1991), 95-106). The nucleic acid molecules can also be expressed in the organelles of the plant cells.
The transgenic plant cells can be regenerated by known techniques to give whole plants. In principle, the transgenic plants may be plants of any desired plant species, i.e. both monocotyledonous and dicotyledonous plants. Thus, it is possible to obtain transgenic plants whose properties are altered by overexpression, suppression or inhibition of homologous (=natural) genes or gene sequences, or expression of heterologous (=foreign) genes or gene sequences.
The inventive compounds (I) can be used with preference in transgenic crops which are resistant to growth regulators, for example 2,4-D, dicamba, or to herbicides which inhibit essential plant enzymes, for example acetolactate synthases (ALS), EPSP synthases, glutamine synthases (GS) or hydroxyphenylpyruvate dioxygenases (HPPD), or to herbicides from the group of the sulfonylureas, the glyphosates, glufosinates or benzoylisoxazoles and analogous active ingredients, or to any desired combinations of these active ingredients.
The inventive compounds can be used with particular preference in transgenic crop plants which are resistant to a combination of glyphosates and glufosinates, glyphosates and sulfonylureas or imidazolinones. The inventive compounds can be used with very particular preference in transgenic crop plants, for example corn or soybeans with the trade name or the designation OptimumTM GATTM (Glyphosate ALS Tolerant).
On employment of the inventive active ingredients in transgenic crops, not only do the effects toward harmful plants observed in other crops occur, but often also effects which are specific to application in the particular transgenic crop, for example an altered or specifically widened spectrum of weeds which can be controlled, altered application rates which can be used for the application, preferably good combinability with the herbicides to which the transgenic crop is resistant, and influencing of growth and yield of the transgenic crop plants.
The invention therefore also provides for the use of the inventive compounds of the formula (I) and of the compounds of the formula (Ia) as herbicides for control of harmful plants in transgenic crop plants.
The inventive compounds can be applied in the form of wettable powders, emulsifiable concentrates, sprayable solutions, dusting products or granules in the customary formulations. The invention therefore also provides herbicidal and plant growth-regulating compositions which comprise the inventive compounds.
The inventive compounds can be formulated in various ways, according to the biological and/or physicochemical parameters required. Possible formulations include, for example: wettable powders (WP), water-soluble powders (SP), water-soluble concentrates, emulsifiable concentrates (EC), emulsions (EW), such as oil-in-water and water-in-oil emulsions, sprayable solutions, suspension concentrates (SC), oil- or water-based dispersions, oil-miscible solutions, capsule suspensions (CS), dusting products (DP), seed-dressing products, granules for broadcasting and soil application, granules (GR) in the form of microgranules, sprayable granules, coated granules and adsorption granules, water-dispersible granules (WG), water-soluble granules (SG), ULV formulations, microcapsules and waxes. These individual formulation types are known in principle and are described, for example, in: Winnacker-Küchler, “Chemische Technologie” [Chemical Technology], Volume 7, C. Hanser Verlag Munich, 4th Ed. 1986, Wade van Valkenburg, “Pesticide Formulations”, Marcel Dekker, N.Y., 1973; K. Martens, “Spray Drying” Handbook, 3rd Ed. 1979, G. Goodwin Ltd. London.
The necessary formulation assistants, such as inert materials, surfactants, solvents and further additives, are likewise known and are described, for example, in: Watkins, “Handbook of Insecticide Dust Diluents and Carriers”, 2nd ed., Darland Books, Caldwell N.J., H.v. Olphen, “Introduction to Clay Colloid Chemistry”, 2nd ed., J. Wiley & Sons, N.Y., C. Marsden, “Solvents Guide”, 2nd ed., Interscience, N.Y. 1963, McCutcheon's “Detergents and Emulsifiers Annual”, MC Publ. Corp., Ridgewood N.J., Sisley and Wood, “Encyclopedia of Surface Active Agents”, Chem. Publ. Co. Inc., N.Y. 1964, Schonfeldt, “Grenzflächenaktive Äthylenoxidaddukte” [Interface-active Ethylene Oxide Adducts], Wiss. Verlagsgesell., Stuttgart 1976, Winnacker-Kuchler, “Chemische Technologie”, Volume 7, C. Hanser Verlag Munich, 4th ed. 1986.
On the basis of these formulations, it is also possible to produce combinations with other active ingredients, for example insecticides, acaricides, herbicides, fungicides, and also with safeners, fertilizers and/or growth regulators, for example in the form of a finished formulation or as a tank mix. Suitable safeners are, for example, mefenpyr-diethyl, cyprosulfamide, isoxadifen-ethyl, cloquintocet-mexyl, benoxacor and dichlormid.
Wettable powders are preparations which can be dispersed uniformly in water and, in addition to the active ingredient, apart from a diluent or inert substance, also comprise surfactants of the ionic and/or nonionic type (wetting agents, dispersants), for example polyoxyethylated alkylphenols, polyoxyethylated fatty alcohols, polyoxyethylated fatty amines, fatty alcohol polyglycol ether sulfates, alkanesulfonates, alkylbenzenesulfonates, sodium lignosulfonate, sodium 2,2′ dinaphthylmethane-6,6′-disulfonate, sodium dibutylnaphthalenesulfonate or else sodium oleoylmethyltaurinate. To produce the wettable powders, the herbicidal active ingredients are ground finely, for example in customary apparatus such as hammer mills, blower mills and air-jet mills, and simultaneously or subsequently mixed with the formulation auxiliaries.
Emulsifiable concentrates are produced by dissolving the active ingredient in an organic solvent, for example butanol, cyclohexanone, dimethylformamide, xylene or else relatively high-boiling aromatics or hydrocarbons or mixtures of the organic solvents, with addition of one or more surfactants of the ionic and/or nonionic type (emulsifiers). The emulsifiers used may, for example, be: calcium alkylarylsulfonates such as calcium dodecylbenzenesulfonate, or nonionic emulsifiers such as fatty acid polyglycol esters, alkylaryl polyglycol ethers, fatty alcohol polyglycol ethers, propylene oxide-ethylene oxide condensation products, alkyl polyethers, sorbitan esters, for example sorbitan fatty acid esters, or polyoxyethylene sorbitan esters, for example polyoxyethylene sorbitan fatty acid esters.
Dusting products are obtained by grinding the active ingredient with finely distributed solid substances, for example talc, natural clays, such as kaolin, bentonite and pyrophyllite, or diatomaceous earth.
Suspension concentrates may be water- or oil-based. They can be produced, for example, by wet grinding by means of commercial bead mills with optional addition of surfactants as already listed above, for example, for the other formulation types.
Emulsions, for example oil-in-water emulsions (EW), can be produced, for example, by means of stirrers, colloid mills and/or static mixers using aqueous organic solvents and optionally surfactants as already listed above, for example, for the other formulation types.
Granules can be produced either by spraying the active ingredient onto adsorptive granulated inert material or by applying active ingredient concentrates by means of adhesives, for example polyvinyl alcohol, sodium polyacrylate or mineral oils, to the surface of carrier substances, such as sand, kaolinites or granulated inert material. Suitable active ingredients can also be granulated in the manner customary for the production of fertilizer granules—if desired as a mixture with fertilizers.
Water-dispersible granules are produced generally by the customary processes such as spray-drying, fluidized bed granulation, pan granulation, mixing with high-speed mixers and extrusion without solid inert material.
For the production of pan granules, fluidized bed granules, extruder granules and spray granules, see, for example, processes in “Spray-Drying Handbook” 3rd ed. 1979, G. Goodwin Ltd., London; J. E. Browning, “Agglomeration”, Chemical and Engineering 1967, pages 147 ff.; “Perry's Chemical Engineer's Handbook”, 5th ed., McGraw-Hill, New York 1973, pp. 8-57.
For further details regarding the formulation of crop protection compositions, see, for example, G. C. Klingman, “Weed Control as a Science”, John Wiley and Sons, Inc., New York, 1961, pages 81-96 and J. D. Freyer, S. A. Evans, “Weed Control Handbook”, 5th Ed., Blackwell Scientific Publications, Oxford, 1968, pages 101-103.
The agrochemical formulations contain generally 0.1 to 99% by weight, especially 0.1 to 95% by weight, of inventive compounds. In wettable powders, the active compound concentration is, for example, from about 10 to 90% by weight, the remainder to 100% by weight consisting of customary formulation components. In emulsifiable concentrates, the active ingredient concentration may be about 1 to 90% and preferably 5 to 80% by weight. Dust-type formulations contain 1 to 30% by weight of active ingredient, preferably usually 5 to 20% by weight of active ingredient; sprayable solutions contain about 0.05 to 80% by weight, preferably from 2 to 50% by weight, of active ingredient. In the case of water-dispersible granules, the active ingredient content depends partly on whether the active compound is present in liquid or solid form and on which granulation assistants, fillers, etc., are used. In the water-dispersible granules, the content of active ingredient is, for example, between 1 and 95% by weight, preferably between 10 and 80% by weight.
In addition, the active ingredient formulations mentioned optionally comprise the respective customary tackifiers, wetting agents, dispersants, emulsifiers, penetrants, preservatives, antifreeze agents and solvents, fillers, carriers and dyes, defoamers, evaporation inhibitors and agents which influence the pH and the viscosity.
Usable combination partners for the inventive compounds in mixture formulations or in a tankmix are, for example, known active ingredients based on inhibition of, for example, acetolactate synthase, acetyl-CoA carboxylase, cellulose synthase, enolpyruvylshikimate-3-phosphate synthase, glutamine synthetase, p-hydroxyphenylpyruvate dioxygenase, phytoendesaturase, photosystem I, photosystem II, protoporphyrinogen oxidase, as described, for example, in Weed Research 26 (1986) 441-445 or “The Pesticide Manual”, 15th edition, The British Crop Protection Council and the Royal Soc. of Chemistry, 2009 and literature cited therein. Examples of known herbicides or plant growth regulators which can be combined with the inventive compounds include the active ingredients which follow (the compounds are designated either by the “common name” according to the International Organization for Standardization (ISO) or by the chemical name or by the code number) and always encompass all use forms, such as acids, salts, esters and isomers, such as stereoisomers and optical isomers.
For application, the formulations in commercial form are, if appropriate, diluted in a customary manner, for example in the case of wettable powders, emulsifiable concentrates, dispersions and water-dispersible granules with water. Dust-type formulations, granules for soil application or granules for broadcasting and sprayable solutions are not normally diluted further with other inert substances prior to application.
The required application rate of the compounds of the formula (I) varies with the external conditions, including temperature, humidity and the type of herbicide used. It may vary within wide limits, for example between 0.001 and 1.0 kg/ha or more of active substance; however, preferably it is between 0.005 and 750 g/ha.
The inventive compositions may additionally comprise further components, for example surfactants. Useful surfactants are emulsifiers and/or foam formers, dispersants or wetting agents having ionic or nonionic properties, or mixtures of these surfactants. Examples thereof are salts of polyacrylic acid, salts of lignosulphonic acid, salts of phenolsulphonic acid or naphthalenesulphonic acid, polycondensates of ethylene oxide with fatty alcohols or with fatty acids or with fatty amines, substituted phenols (preferably alkylphenols or arylphenols), salts of sulphosuccinic esters, taurine derivatives (preferably alkyl taurates), phosphoric esters of polyethoxylated alcohols or phenols, fatty esters of polyols, and derivatives of the compounds containing sulphates, sulphonates and phosphates, for example alkylaryl polyglycol ethers, alkylsulphonates, alkyl sulphates, arylsulphonates, protein hydrolysates, lignosulphite waste liquors and methylcellulose. The presence of a surfactant is necessary if one of the active ingredients and/or one of the inert carriers is insoluble in water and when application is effected in water. The proportion of surfactants is between 5 and 40 per cent by weight of the inventive composition. It is possible to use dyes such as inorganic pigments, for example iron oxide, titanium oxide and Prussian Blue, and organic dyes such as alizarin dyes, azo dyes and metal phthalocyanine dyes, and trace nutrients such as salts of iron, manganese, boron, copper, cobalt, molybdenum and zinc.
If appropriate, it is also possible for other additional components to be present, for example protective colloids, binders, adhesives, thickeners, thixotropic substances, penetrants, stabilizers, sequestrants, complexing agents. In general, the active ingredients can be combined with any solid or liquid additive commonly used for formulation purposes. In general, the inventive compositions and formulations contain between 0.05 and 99% by weight, 0.01 and 98% by weight, preferably between 0.1 and 95% by weight and more preferably between 0.5 and 90% active ingredient, most preferably between 10 and 70 percent by weight. The inventive active ingredients or compositions can be used as such or, depending on their respective physical and/or chemical properties, in the form of the formulations thereof or the use forms prepared therefrom, such as aerosols, capsule suspensions, cold-fogging concentrates, warm-fogging concentrates, encapsulated granules, fine granules, free-flowing concentrates for the treatment of seed, ready-to-use solutions, dustable powders, emulsifiable concentrates, oil-in-water emulsions, water-in-oil emulsions, macrogranules, microgranules, oil-dispersible powders, oil-miscible free-flowing concentrates, oil-miscible liquids, foams, pastes, pesticide-coated seed, suspension concentrates, suspoemulsion concentrates, soluble concentrates, suspensions, spray powders, soluble powders, dusts and granules, water-soluble granules or tablets, water-soluble powders for seed treatment, wettable powders, active ingredient-impregnated natural products and synthetic substances, and also microencapsulations in polymeric substances and in coating materials for seed, and also ULV cold-fogging and warm-fogging formulations.
The formulations mentioned can be produced in a manner known per se, for example by mixing the active ingredients with at least one customary extender, solvent or diluent, emulsifier, dispersant and/or binder or fixative, wetting agent, water repellent, optionally siccatives and UV stabilizers and optionally dyes and pigments, antifoams, preservatives, secondary thickeners, tackifiers, gibberellins and other processing auxiliaries.
The inventive compositions include not only formulations which are already ready for use and can be deployed with a suitable apparatus onto the plant or the seed, but also commercial concentrates which have to be diluted with water prior to use. The inventive active ingredients may be present as such or in their (commercial standard) formulations, or else in the use forms prepared from these formulations as a mixture with other (known) active ingredients, such as insecticides, attractants, sterilants, bactericides, acaricides, nematicides, fungicides, growth regulators, herbicides, fertilizers, safeners or semiochemicals.
The inventive treatment of the plants and plant parts with the active ingredients or compositions is effected directly or by action on their surroundings, habitat or storage space by the customary treatment methods, for example by dipping, spraying, atomizing, irrigating, evaporating, dusting, fogging, broadcasting, foaming, painting, spreading-on, watering (drenching), drip irrigating and, in the case of propagation material, especially in the case of seeds, also by dry seed treatment, wet seed treatment, slurry treatment, incrustation, coating with one or more coats, etc. It is also possible to deploy the active ingredients by the ultra-low volume method or to inject the active ingredient preparation/the active ingredient itself into the soil.
The examples which follow illustrate the invention in detail.
A. CHEMICAL EXAMPLES
1. Preparation of ethyl 3-(2,3-difluorophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate
Example No. 2.1.056
To this end, 3.320 g (21.13 mmol) of 2,3-difluorobenzaldehyde oxime are initially charged in 25 ml of dimethylformamide, and 2.822 g (21.13 mmol) of N-chlorosuccinimide are added thereto, in the course of which the temperature rises to 79° C. Subsequently, the mixture is heated to 40° C. for 1 h, another spatula-tip of N-chlorosuccinimide is added, 15 minutes later the mixture is cooled to room temperature (RT), then 3.618 g (31.70 mmol) of ethyl methacrylate and 4.097 g (31.70 mmol) of N,N-diisopropylethylamine are added dropwise. After cooling to RT, the mixture is stirred for another 15 minutes, the flask contents are added to 50 ml of water, and the mixture is acidified with 1 M sulfuric acid and extracted repeatedly with methyl t-butyl ether. The combined organic phases are washed once with water and with sodium chloride solution, dried over sodium sulfate and filtered off, and the filtrate is concentrated under reduced pressure. This gives 6.06 g of yellow oil, which was chromatographed on silica gel using an ethyl acetate/heptane gradient. This gives 5.140 g (90%) of colorless oil.
1H NMR [CDCl3]: δ=1.31 (t, 3H); 1.72 (s, 3H); 3.33 (d, 1H); 3.95 (d, 1H); 4.36 (q, 2H); 7.12 (m, 1H); 7.23 (m, 1H); 7.53 (m, 1H).
2. Preparation of isopropyl 5-cyano-3-(3,5-difluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate
Example No. 2.2.475
1.00 g (6.37 mmol) of 3,5-difluorobenzaldehyde oxime is dissolved in 25 ml of dichloromethane and cooled to 0° C., and 1.195 g (9.55 mmol) of ethyl 2-cyanoacrylate are added. Then 2.050 g (6.37 mmol) of iodosobenzene are added and the mixture is warmed to RT. After the reaction has ended, the solution is admixed with thiosulfate solution, extracted with ethyl acetate and dried over sodium sulfate. After purification by chromatography using silica gel, this gives 1.010 g (54%) of the desired product.
1H NMR [DMSO]: δ=1.30 (t, 3H); 4.11 (d, 1H); 4.32 (q, 2H); 4.48 (d, 1H); 7.48 (m, 3H).
3. Preparation of ethyl 3-(3,5-difluorophenyl)-5-ethyl-4,5-dihydro-1,2-oxazole-5-carboxylate
Example No. 2.1.471
Intermediate: 3,5-difluoro-N-hydroxybenzenecarboximidoyl chloride
19.000 g (259.94 mmol) of 3,5-difluorobenzaldehyde oxime are initially charged in 20 ml of dry DMF under nitrogen, and 510 mg (3.81 mmol) of N-chlorosuccinimide are added first. Subsequently, gaseous hydrochloric acid is introduced into the reaction solution until the reaction temperature has risen to 35° C. Then the remaining 1.990 g (15.28 mmol) of N-chlorosuccinimide are metered in, such that the internal temperature of 40° C. is not exceeded. After cooling to RT, ice-water is added, the mixture is diluted with diethyl ether, and the organic phase is extracted twice with ice-water. After drying over sodium sulfate, the solvent is removed under reduced pressure. This gives 3.177 g (87%) of colorless solid.
2.000 g (10.44 mmol) of 3,5-difluoro-N-hydroxybenzenecarboximidoyl chloride are dissolved in 117 g of isopropanol. Then 1.606 g (9.39 mmol) of 75% ethyl 2-methylenebutanoate are added thereto, and the mixture is admixed with 4.385 g (52.20 mmol) of sodium hydrogencarbonate and stirred at RT. After 12 h, undissolved material is filtered off, and the mother liquor is concentrated and separated on silica gel with ethyl acetate/heptane. This gives 1.900 g (61%) of the desired product.
1H NMR [CDCl3]: δ=1.00 (t, 3H); 1.32 (t, 3H); 2.06 (q, 2H); 3.18 (d, 1H); 3.88 (d, 1H); 4.27 (M, 2H); 6.85 (m, 1H), 7.18 (m, 2H).
4. Preparation of 3-[3-chloro-5-(trifluoromethoxy)phenyl]-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylic acid
Example No. 1.1.554
3.878 g (11.03 mmol) of ethyl 3-[3-chloro-5-(trifluoromethoxy)phenyl]-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate are initially charged in 50 ml of THF and stirred with 33.1 ml (33.079 mmol) of 1 M sodium hydroxide solution at RT for 16 h. Subsequently, the mixture is acidified with dilute sulfuric acid, sodium chloride solution is added and the mixture is extracted repeatedly with ethyl acetate. This gives 2.323 g (65%) of the above compound after chromatographic purification on silica gel with ethyl acetate/heptane mixtures.
1H NMR [DMSO]: δ=1.58 (s, 3H); 3.3 (OH); 3.32 (d, 1H); 3.84 (d; 1H); 7.61 (m, 1H); 7.70 (s, 1H); 7.78 (m, 1H).
5. Preparation of 3-methoxy-3-oxopropyl-3-(3,5-difluorophenyl)-5-ethyl-4,5-dihydro-1,2-oxazole-5-carboxylate
Example No. 2.6.486
Intermediate: 3-(3,5-difluorophenyl)-5-ethyl-4,5-dihydro-1,2-oxazole-5-carbonyl chloride
2.000 g (7.84 mmol) of 3-(3,5-difluorophenyl)-5-ethyl-4,5-dihydro-1,2-oxazole-5-carboxylic acid are dissolved in 50 ml of dichloromethane, and 29.0 mg (73.10 mmol) of dimethylformamide are added thereto. Then the reaction solution is admixed with 1.492 g (11.76 mmol) of oxalyl chloride and stirred at RT. After 1 h, the reaction mixture is concentrated by rotary evaporation, and twice more admixed with toluene and concentrated by rotary evaporation. This gives 2.30 g (97%) of the above carbonyl chloride, which is reacted without further purification.
200.0 mg (0.73 mmol) of 3-(3,5-difluorophenyl)-5-ethyl-4,5-dihydro-1,2-oxazole-5-carbonyl chloride are initially charged in 5 ml of dichloromethane, then 221.86 mg (2.19 mmol) of triethylamine are added thereto, and finally 91.3 mg (0.88 mmol) of methyl 3-hydroxypropanoate in 5 ml of dichloromethane are added thereto. After 1 h, the reaction solution is concentrated by rotary evaporation and separated on silica gel with a heptane/ethyl acetate mixture. This gives 134 mg (51%) of the above compound as a colorless oil.
1H NMR [CDCl3]: δ=0.99 (t, 3H); 2.01-2.07 (m, 2H); 2.72 (t, 2H), 3.17 (d, 1H); 3.68 (s, 3H); 3.75 (d, 1H); 4.41-4.53 (m, 2H); 6.86 (t, 1H); 7.18 (d, 2H).
6. Preparation of 3-(3,5-dichlorophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carbonitrile
Example No. 3.417
0.700 g (3.68 mmol) of 3,5-dichlorobenzaldehyde oxime is initially charged in 50 ml of DMF, then 0.516 g (3.87 mmol) of N-chlorosuccinimide is added thereto and the mixture is left to stir at RT for 4 h. Subsequently, 0.371 g (5.53 mmol) of methacrylonitrile and 0.559 g (5.53 mmol) of triethylamine are added thereto and the mixture is left to stir at RT for another 18 h. The mixture is concentrated by rotary evaporation under reduced pressure and separated on preparative HPLC (RP phase). This gives 110 mg (12%) of the desired product as a colorless oil.
1H NMR [CDCl3]: δ=[CDCl3] 1.91 (s, 3H); 3.38 (d, 1H); 3.80 (d, 1H); 7.45 (s, 1H); 7.52 (s, 1H).
7. Preparation of methyl 4-bromo-3-(3,5-difluorophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate
Example No. 2.1.470
1.000 g (5.22 mmol) of 3,5-difluoro-N-hydroxybenzenecarboximidoyl chloride is dissolved in 20 ml of isopropanol, then 1121 mg (6.26 mmol) of methyl 3-bromo-2-methylacrylate are added thereto, and 1754.1 mg (20.88 mmol) of solid sodium hydrogencarbonate. The mixture is left to stir at RT for 2 d and the crude mixture obtained is purified using silica gel with ethyl acetate/heptane. This gives 540 mg (31%) of a yellow oil.
1H NMR [CDCl3]: δ=D1=1.58 (s, 3H); 3.82 (s, 3H); 5.50 (s, 1H); D2=1.85 (s, 3H); 3.72 (s, 3H); 5.78 (s, 1H); 6.8-7.5 (m, 3H).
8. Preparation of methyl 3-(3,5-difluorophenyl)-5-fluoro-4,5-dihydro-1,2-oxazole-5-carboxylate
Example No. 2.2.468
1.000 g (5.22 mmol) of 3,5-difluoro-N-hydroxybenzenecarboximidoyl chloride is dissolved in 23 ml of isopropanol, then 1086.6 mg (10.44 mmol) of methyl 2-fluoroacrylate are added thereto, and then the mixture is admixed with 2.192 g (26.10 mmol) of sodium hydrogencarbonate. The mixture is left to stir at 40° C. for 1 h, taken up in water and extracted with ethyl acetate to obtain 1.230 g (91%) of the above compound in solid form.
1H NMR [CDCl3]: δ=3.65 (dd, 1H); 3.96 (s, 3H); 4.12 (dd, 1H); 6.96 (t, 1H); 7.22 (d, 2H).
9. Preparation of 5-(fluoromethyl)-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylic acid
Example No. 1.2.001
3.00 g (11.14 mmol) of ethyl 5-(fluoromethyl)-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate are dissolved in 150 ml of THF, and 0.543 g (22.28 mmol) of lithium hydroxide is added at RT. After 20 h, the mixture is concentrated by rotary evaporation under reduced pressure, and the residue is taken up with dichloromethane and extracted with saturated sodium hydrogencarbonate solution. The aqueous phase is subsequently adjusted to pH 1-2 and the mixture is extracted with ethyl acetate. This gives 2.530 g (89%) of the carboxylic acid.
1H NMR [CDCl3]: δ=3.56 (d, 1H); 3.80 (d, 1H); 4.71 (d, 1H); 4.83 (d, 1H); 7.18 (m, 1H); 7.41 (m, 3H).
10. Preparation of methyl 3-(3-chloro-4-fluorophenyl)-5-(trifluoromethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate
Example No. 2.2.1208
1.500 g (8.64 mmol) of 3-chloro-4-fluorobenzaldehyde oxime are initially charged in 47.5 g of DMF and cyclized with 1.212 g (9.07 mmol) of N-chlorosuccinimide, 1.312 g (12.96 mmol) and 2.179 g (12.96 mmol) of methyl 2-(trifluoromethyl)acrylate. After purification on silica gel with ethyl acetate/heptane as a solvent mixture, 1.300 g (43%) of the above product are obtained.
1H NMR [CDCl3]: δ=1.52 8s, 3H); 3.74 (d, 1H); 3.94 (s, 3H); 4.03 (d, 1H); 7.22 (m, 1H); 7.58 (m, 1H); 7.72 (m, 1H).
11. Preparation of 3-(3-chloro-4-fluorophenyl)-5-(trifluoromethyl)-4,5-dihydro-1,2-oxazole-5-carboxylic acid
Example No. 1.2.1205
2.000 g (6.14 mmol) of the ester methyl 3-(3-chloro-4-fluorophenyl)-5-(trifluoromethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate are dissolved in 20 ml of THF, 0.295 g (7.37 mmol) of sodium hydroxide in water are added and the mixture is stirred at RT. After 18 h, the solvent is removed by rotary evaporation, water is added, the mixture is washed once with dichloromethane and the water phase is acidified with dilute hydrochloric acid. The latter is extracted twice more with dichloromethane. The mixture is dried over magnesium sulfate to obtain 1.740 g (85%) of the carboxylic acid.
1H NMR [CDCl3]: δ=3.81 (d, 1H); 4.00 (d, 1H); 7.22 (m, 1H); 7.58 (m, 1H); 7.74 (m, 1H).
12. Preparation of methyl 3-(3,5-dichlorophenyl)-5-(methoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate
Example No. 2.5.544
1.156 g (6.08 mmol) of 3,5-dichlorobenzaldehyde oxime are cyclized with 0.950 g (7.30 mmol) of methyl 2-(methoxymethyl)acrylate, 0.853 g (6.39 mmol) of N-chlorosuccinimide and 0.923 g (9.13 mmol) of triethylamine in 47.5 g of dimethylformamide. After chromatographic purification on silica gel, 0.150 g (7.34%) of the above compound is obtained as a yellowish oil.
1H NMR [CDCl3]: δ=3.43 (s, 3H); 3.50 (d, 1H); 3.72 (d, 1H); 3.80 (mc, 2H); 3.82 (s, 3H); 7.41 (m, 1H); 7.55 (s, 2H).
13. Preparation of 3-(3,5-dichlorophenyl)-5-(methoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylic acid
Example No. 1.5.544
100.0 mg (0.31 mmol) of methyl 3-(3,5-dichlorophenyl)-5-(methoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate are dissolved in 5 ml of THF, 40.0 mg (0.47 mmol) of sodium hydroxide in 2 ml of water are added and the mixture is stirred at RT for 18 h.
After removing the solvent, the mixture is diluted with water, the water phase is washed with dichloromethane, then the water phase is acidified with dilute hydrochloric acid and washed once again with dichloromethane. The latter dichloromethane phase is dried. This gives 100 mg (100%) of the above acid as a colorless oil.
1H NMR [CDCl3]: δ=3.48 (s, 3H); 3.50 (d, 1H); 3.72 8d, 1H); 3.85 (q, 2H); 7.42 (m, 1H); 7.55 (m, 2H).
14. Preparation of methyl 3-(3-fluoro-5-methylphenyl)-5-(1-hydroxyethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate
Example No. 2.5.498
10.0 g (53.31 mmol) of 3-fluoro-N-hydroxy-5-methylbenzenecarboximidoyl chloride are reacted with 7.631 g (58.64 mmol) of methyl 3-hydroxy-2-methylenebutanoate and 22.390 g (22.54 mmol) of sodium hydrogencarbonate according to method C overnight. After filtration of the reaction solution, it is chromatographed on silica gel. This gives 15.00 g (95%) of the above compound as an oil.
1H NMR [CDCl3]: δ=D1 1.20 (d, 3H); 2.37 (d, 1H); 2.38 (s, 3H); 3.54 (d, 1H), 3.69 (d, 1H); 3.83 (s, 3H); 4.33 (m, 1H); 6.96 (s, 1H); 7.23 (s, 1H); 7.25 (s, 1H). D2 1.26 (d, 3H); 2.18 (d, 1H); 2.38 (s, 3H); 3.60 (d, 1H); 3.72 (d, 1H); 3.83 (s, 3H); 4.22 (m, 1H); 6.93 (s, 1H); 7.21 (s, 1H); 7.25 (s, 1H)
15. Preparation of 3-(3,5-difluorophenyl)-5-(1-hydroxyethyl)-4,5-dihydro-1,2-oxazole-5-carboxylic acid
Example No. 1.5.479
1.5 g (5.26 mmol) of methyl 3-(3,5-difluorophenyl)-5-(1-hydroxyethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate in 75 ml THF are hydrolyzed with 0.151 g (6.31 mmol) of LiOH at RT. After 1 h, the solvent is removed under reduced pressure, the pH is brought to 1-2 with hydrochloric acid and extraction is effected with ethyl acetate. This gives 1.50 g (99%) of the above acid.
1H NMR [CDCl3]: δ=D1 1.25 (d, 3H); 1.36 (d, 1H); 3.60 (d, 1H); 3.70 (d, 1H); 4.29 (m, 1H); 6.91 (t, 1H); 7.20 (d, 2H). D2 1.29 (d, 3H); 1.42 (d, 1H); 3.60 (d, 1H); 3.69 (d, 1H); 4.22 (m, 1H); 6.91 (t, 1H); 7.20 (d, 2H).
16. Preparation of methyl 5-acetyl-3-(3,5-difluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate
Example No. 2.4.462
To this end, 2.000 g (7.01 mmol) of methyl 3-(3,5-difluorophenyl)-5-(1-hydroxyethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate are stirred with 6.048 g (28.05 mmol) of pyridinium chlorochromate and molecular sieve in 75 ml of dichloromethane at RT for 5 h. The reaction solution is filtered with diethyl ether through an SPE cartridge and concentrated by rotary evaporation. This gives 2.000 g (96%) of the above compound in solid form.
1H NMR [CDCl3]: δ=2.44 (s, 3H); 3.80 (d, 1H); 3.86 (s, 3H); 3.89 (d, 1H); 6.90 (m, 1H); 7.19 (d, 2H).
17. Preparation of methyl 3-(3-chloro-5-fluorophenyl)-5-vinyl-4,5-dihydro-1,2-oxazole-5-carboxylate
Example No. 2.3.572
4.400 g (15.76 mmol) of methyl 3-(3-bromo-5-methylphenyl)-5-(1-{[(trifluoromethyl)-sulfonyl]oxy}ethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, prepared from the corresponding alcohol, trifluoromethanesulfonic anhydride and pyridine (62% yield), are converted together with 600.29 mg (3.94 mmol) of DBU. After 2 days, the reaction mixture is diluted with water, acidified with dilute hydrochloric acid up to pH 4-5 and finally extracted with dichloromethane. Subsequently, the mixture is chromatographed on silica gel with ethyl acetate/heptane. This gives 450 mg (57%) of the above compound as a colorless oil.
1H NMR [CDCl3]: δ=2.35 (s, 3H), 3.35 (d, 1H); 3.83 (s, 3H); 3.93 (d, 1H); 5.35 (d, 1H), 5.55 (d, 1H); 6.13 (dd, 1H); 7.38 (s, 1H), 7.42 (s, 1H); 7.58 (s, 1H).
18. Preparation of methyl 5-(1-chlorovinyl)-3-(3,5-difluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate
Example No. 2.3.473
730 mg (2.58 mmol) of methyl 5-acetyl-3-(3,5-difluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate are dissolved in 20 ml of dichloromethane, one drop of DMF is added and the mixture is heated with 590 mg (2.84 mmol) of phosphorus pentachloride at 100° C. in a microwave for 6 h. Subsequently, the reaction mixture is added to a mixture of warm water (about 35° C.) and dichloromethane and stirred at the temperature for 1 h. The water phase (pH 2) is removed. The dichloromethane phase is washed with saturated sodium carbonate solution and dried over sodium sulfate. Subsequently, the mixture is chromatographed using silica gel (ethyl acetate/heptane). This gives 230 mg (25%) of the above compound in solid form.
1H NMR [CDCl3]: δ=3.53 (d, 1H); 3.88 (s, 3H); 4.22 (d, 1H); 5.55 (s, 1H); 5.93 (s, 1H); 6.90 (m, 1H); 7.20 (d, 2H).
In analogy to the preparation of the abovementioned compounds and in accordance with the general details of the preparation, the compounds specified in the following tables are obtainable. The NMR data of the examples disclosed in these tables are given either in conventional form (δ values, number of hydrogen atoms, multiplet splitting) or as NMR peak lists. In the NMR peak list method, the NMR data of selected examples are stated in the form of NMR peak lists, giving, for each signal peak, first the δ value in ppm and then the signal intensity separated by a space. The δ value/signal intensity number pairs for different signal peaks are listed separated from one another by semicolons.
The abbreviations used mean:



















Ac
acetoxy
Bu
butyl
Et
ethyl
Me
methyl


Pr
propyl
Pen
pentyl
Hex
hexyl
Ph
phenyl


c
cyclo
s
secondary
i
iso
t
tertiary


THF
tetrahydrofuran









D1, D2 denote diastereomers of a diastereomer pair present as a racemate of two enantiomers.







TABLE 1.1







Inventive compounds of the general formula (I) in which W* is COOH, R1


is hydrogen, and aryl is the radical.








 


1








 











No.
Aryl
R2
R3
Physical data





1.1.1
3-fluorophenyl
H
methyl
[CDCl3] 1.78 (s, 3H); 3.29 (d, 1H);






3.85 (d, 1H); 7.12 (m, 1H); 7.40 (m,






2H).


1.1.2
3-fluorophenyl
H
ethyl
[CDCl3] 1.08 (t, 3H); 2.14 (mc; 2H);






3.32 (d, 1H); 3.30 (d, 1H); 7.15 (m,






1H); 7.40 (m, 2H).


1.1.3
3-fluorophenyl
H
propyl



1.1.4
3-fluorophenyl
H
cyclopropyl



1.1.5
3-chlorophenyl
H
methyl
[CDCl3] 1.78 (s, 3H); 3.28 (d, 1H);






3.86 (d, 1H); 7.35 (m, 1H); 7.42 (m,






1H); 7.51 (m, 1H); 7.65 (m, 1H).


1.1.6
3-chlorophenyl
H
ethyl



1.1.7
3-chlorophenyl
H
propyl



1.1.8
3-chlorophenyl
H
cyclopropyl



1.1.9
3-bromophenyl
H
methyl
[CDCl3] 1.72 (s, 3H); 3.19 (d, 1H);






3.82 (s, 3H); 3.86 (d, 1H); 7.28 (t,






1H); 7.55 (m, 1H); 7.59 (m, 1H);






7.80 (t, 1 H).


1.1.10
3-bromophenyl
H
ethyl



1.1.11
3-iodophenyl
H
methyl



1.1.12
3-iodophenyl
H
ethyl



1.1.13
3-methylphenyl
H
methyl
[DMSO] 1.55 (s, 3H); 2.32 (s, 3H);






3.35 (d, 1H); 3.76 (d, 1H); 7.20-






7.50 (m, 4H).


1.1.14
3-methylphenyl
H
ethyl



1.1.15
3-ethylphenyl
H
methyl
[DMSO] 1.20 (t, 3H); 1.55 (s, 3H);






2.65 (q, 2H); 3.38 (d, 1H); 3.80 (d,






1H); 7.28-7.50 (m, 4H).


1.1.16
3-propylphenyl
H
methyl



1.1.17
3-isopropylphenyl
H
methyl
[DMSO] 1.20 (d, 6H); 1.55 (s, 3H);






2.94 (m, 1H); 3.40 (d, 1H); 3.80 (d,






1H); 7.35 (m, 2H); 7.48 (m, 1H);






7.55 (s, 1H).


1.1.18
3-n-butylphenyl
H
methyl



1.1.19
3-i-butylphenyl
H
methyl



1.1.20
3-tert-butylphenyl
H
methyl



1.1.21
3-cyclopropylphenyl
H
methyl



1.1.22
3-cyclobutylphenyl
H
methyl



1.1.23
3-cyclopentylphenyl
H
methyl



1.1.24
3-vinylphenyl
H
methyl



1.1.25
3-ethynylphenyl
H
methyl
[CDCl3] 1.78 (s, 1H); 3.10 (s, 1H);






3.30 (d, 1H); 3.87 (d, 1H); 7.35 (m,






1H); 7.52 (m, 1H); 7.68 (m, 1H);






7.75 (s, 1H).


1.1.26
3-cyanophenyl
H
methyl
[CDCl3] 1.80 (s, 3H); 3.29 (d, 1H);






3.89 (d, 1H); 7.55 (m, 1H); 7.72 (m,






1H); 7.90 (m, 2H).


1.1.27
3-trifluoromethyl-
H
methyl
[CDCl3] 1.80 (s, 3H); 3.32 (d, 1H);



phenyl


3.91 (d, 1H); 7.56 (m, 1H); 7.69 (m,






1H); 7.88 (m, 2H).


1.1.28
3-difluoromethyl-
H
methyl




phenyl





1.1.29
3-(hydroxycarbonyl)-
H
methyl
[DMSO] 1.58 (s, 3H); 3.42 (d,



phenyl


1H);3.82 (d, 1H); 7.60 (t, 1H); 7.90






(d, 1H); 8.03 (d, 1H); 8.20 (s,






1H). 13.2 (bs, 1H)


1.1.30
3-(methoxycarbonyl)-
H
methyl




phenyl





1.1.31
3-(ethoxycarbonyl)-
H
methyl




phenyl





1.1.32
3-hydroxymethyl-
H
methyl




phenyl





1.1.33
3-carbamoylphenyl
H
methyl
[DMSO] 1.58 (s, 3H); 3.40 (d, 1H);






3.85 (d, 1H); 7.43 (bs, 1H); 7.53 t,






1H); 7.85 (d, 1H); 7.95 (d, 1H); 8.08






(bs, 1H); 8.11 (s, 1H).


1.1.34
3-hydroxyphenyl
H
methyl
[DMSO] 1.52 (s, 3H); 3.32 (d, 1H);






3.71 (d, 1H); 6.85 (d, 1H); 7.08 (m,






2H); 7.24 /t, 1H); 9.65 (s, 1H); 13.2






(bs, 1H).


1.1.35
3-methoxyphenyl
H
methyl
[CDCl3] 1.75 (s, 3H); 3.30 (d, 1H);






3.85 (s, 3H); 3.89 (d, 1H); 7.00 (m,






1H); 7.16 (m, 1H); 7.25 (m, 1H);






7.35 (m, 1H).


1.1.36
3-ethoxyphenyl
H
methyl
[CDCl3] 1.41 (t, 1H), 1.75 (s, 1H);






3.25 (d, 1H); 3.83 (d, 1H); 4.05 (q,






2H); 6.95 (m, 1H); 7.15 (m, 1H);






7.20-7.32 (m, 2H).


1.1.37
3-propyloxyphenyl
H
methyl



1.1.38
3-isopropyloxyphenyl
H
methyl



1.1.39
3-n-butyloxyphenyl
H
methyl



1.1.40
3-i-butyloxyphenyl
H
methyl



1.1.41
3-t-butyloxyphenyl
H
methyl



1.1.42
3-difluoromethoxy-
H
methyl
[CDCl3] 1.78 (s, 3H); 3.38 (d, 1H);



phenyl


3.86 (d, 1H); 6.52 (t, 1H); 7.21 (m,






1H); 7.43 (m, 2H).


1.1.43
3-trifluoromethoxy-
H
methyl
[CDCl3] 1.80 (s, 3H); 3.30 (d, 1H);



phenyl


3.88 (d, 1H); 7.25 (m, 1H); 7.45 (m,






1H); 7.55 (m, 2H).


1.1.44
3-(2,2,2-trifluoro-
H
methyl




ethoxy)phenyl





1.1.45
3-(2-chloroethoxy)-
H
methyl




phenyl





1.1.46
3-(2-hydroxyethoxy)-
H
methyl




phenyl





1.1.47
3-(2-methoxyethoxy)-
H
methyl
[CDCl3] 1.75 (s, 3H); 3.35 (d, 1H);



phenyl


3.43 (s, 3H); 3.75 (dd, 2H); 3.85 (d,






1H); 4.14 (dd, 2H); 7.04 (d, 1H);






7.15 (d, 1H); 7.25-7.40 (m, 2H).


1.1.48
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]phenyl





1.1.49
3-nitrophenyl
H
methyl
[DMSO] 1.52 (s, 3H); 3.40 (d, 1H);






3.85 (d, 1H); 7.75 (t, 1H); 8.08 (d,






1H); 8.29 (d, 1H); 8.4 (s, 1H).


1.1.50
3-acetoxyphenyl
H
methyl



1.1.51
{3-[(tert-
H
methyl
[CDCl3] 1.50 (s, 9H); 1.75 (s, 3H);



butoxycarbonyl)-


3.30 (d, 1H); 3.90 (d, 1H); 6.70 (bs,



amino]phenyl}


1H); 7.30 (s, 2H), 7.40 (s, 1H), 7.70






(s, 1H). 


1.1.52
3-methylsulfanyl-
H
methyl




phenyl





1.1.53
3-ethylsulfanylphenyl
H
methyl



1.1.54
3-(pentafluoro-
H
methyl
[CDCl3] 1.80 (s, 3H); 3.30 (d, 1H);



lambda6-sulfanyl)-


3.90 (d, 1H); 7.51 (t, 1H); 7.80 (2d,



phenyl


2H); 8.00 (s, 1H).


1.1.55
2,3-difluorophenyl
H
methyl
[CDCl3] 1.78 (s, 3H); 3.40 (dd, 1H);






3.95 (dd, 1H); 7.13 (m, 1H); 7.22






(m, 2H); 7.61 (t, 1H).


1.1.56
2,3-difluorophenyl
H
ethyl



1.1.57
2,3-difluorophenyl
H
propyl



1.1.58
2,3-difluorophenyl
H
cyclopropyl



1.1.59
2-chloro-3-
H
methyl




fluorophenyl





1.1.60
2-bromo-3-
H
methyl




fluorophenyl





1.1.61
2-methy1-3-
H
methyl




fluorophenyl





1.1.62
2-ethyl-3-
H
methyl




fluorophenyl





1.1.63
2-cyclopropyl-3-
H
methyl




fluorophenyl





1.1.64
2-vinyl-3-
H
methyl




fluorophenyl





1.1.65
2-ethyny1-3-
H
methyl




fluorophenyl





1.1.66
2-cyano-3-
H
methyl




fluorophenyl





1.1.67
2-methoxy-3-
H
methyl




fluorophenyl





1.1.68
2-ethoxy-3-
H
methyl




fluorophenyl





1.1.69
2-trifluoromethoxy-3-
H
methyl




fluorophenyl





1.1.70
2-nitro-3-fluorophenyl
H
methyl



1.1.71
2-fluoro-3-
H
methyl




chlorophenyl





1.1.72
2,3-dichlorophenyl
H
methyl
[CDCl3] 1.80 (s, 3H); 3.50 (d, 1H);






3.95 (d, 1H); 7.25 (m, 1 H); 7.26 (m,






1H); 7.50 (m, 1H); 7.58 (m, 1H).


1.1.73
2,3-dichlorophenyl
H
ethyl



1.1.74
2,3-dichlorophenyl
H
propyl



1.1.75
2,3-dichlorophenyl
H
cyclopropyl



1.1.76
2-bromo-3-
H
methyl




chlorophenyl





1.1.77
2-methy1-3-
H
methyl




chlorophenyl





1.1.78
2-ethyl-3-
H
methyl




chlorophenyl





1.1.79
2-cyclopropyl-3-
H
methyl




chlorophenyl





1.1.80
2-vinyl-3-
H
methyl




chlorophenyl





1.1.81
2-ethyny1-3-
H
methyl




chlorophenyl





1.1.82
2-cyano-3-
H
methyl




chlorophenyl





1.1.83
2-trifluoromethyl-2-
H
methyl




chlorophenyl





1.1.84
2-methoxy-3-
H
methyl




chlorophenyl





1.1.85
2-ethoxy-3-
H
methyl




chlorophenyl





1.1.86
2-trifluoromethoxy-3-
H
methyl




chlorophenyl





1.1.87
2-nitro-3-
H
methyl




chlorophenyl





1.1.88
2-fluoro-3-
H
methyl




bromophenyl





1.1.89
2-chloro-3-
H
methyl




bromophenyl





1.1.90
2,3-dibromophenyl
H
methyl



1.1.91
2-methyl-3-
H
methyl




bromophenyl





1.1.92
2-ethyl-3-
H
methyl




bromophenyl





1.1.93
2-cyclopropyl-3-
H
methyl




bromophenyl





1.1.94
2-vinyl-3-
H
methyl




bromophenyl





1.1.95
2-ethynyl-3-
H
methyl




bromophenyl





1.1.96
2-cyano-3-
H
methyl




bromophenyl





1.1.97
2-trifluoromethyl-3-
H
methyl




bromophenyl





1.1.98
2-methoxy-3-phenyl
H
methyl



1.1.99
2-ethoxy-3-
H
methyl




bromophenyl





1.1.100
2-trifluoromethoxy-3-
H
methyl




bromophenyl





1.1.101
2-nitro-3-
H
methyl




bromophenyl





1.1.102
2-fluoro-3-iodophenyl
H
methyl



1.1.103
2-chloro-3-
H
methyl




iodophenyl





1.1.104
2-bromo-3-
H
methyl




iodophenyl





1.1.105
2-methyl-3-
H
methyl




iodophenyl





1.1.106
2-ethyl-3-iodophenyl
H
methyl



1.1.107
2-cyclopropyl-3-
H
methyl




iodophenyl





1.1.108
2-vinyl-3-iodophenyl
H
methyl



1.1.109
2-ethynyl-3-
H
methyl




iodophenyl





1.1.110
2-cyano-3-
H
methyl




iodophenyl





1.1.111
2-trifluoromethyl-3-
H
methyl




iodophenyl





1.1.112
2-methoxy-3-
H
methyl




iodophenyl





1.1.113
2-ethoxy-3-
H
methyl




iodophenyl





1.1.114
2-trifluoromethoxy-3-
H
methyl




iodophenyl





1.1.115
2-nitro-3-iodophenyl
H
methyl



1.1.116
2-fluoro-3-
H
methyl
[CDCl3] 1.56 (s, 3H); 2.25 (s, 3H);



methylphenyl


3.35 (d, 1H); 3.80 (d, 1H); 7.15 (t,






1H); 7.40 (t, 1H); 7.51 (t, 1H).


1.1.117
2-fluoro-3-
H
ethyl




methylphenyl





1.1.118
2-fluoro-3-
H
propyl




methylphenyl





1.1.119
2-fluoro-3-
H
cyclopropyl




methylphenyl





1.1.120
2-chloro-3-
H
methyl




methylphenyl





1.1.121
2-chloro-3-
H
ethyl




methylphenyl





1.1.122
2-chloro-3-
H
propyl




methylphenyl





1.1.123
2-chloro-3-
H
cyclopropyl




methylphenyl





1.1.124
2-bromo-3-
H
methyl




methylphenyl





1.1.125
2,3-dimethylphenyl
H
methyl



1.1.126
2,3-dimethylphenyl
H
ethyl



1.1.127
2,3-dimethylphenyl
H
propyl



1.1.128
2,3-dimethylphenyl
H
cyclopropyl



1.1.129
2-ethyl-3-
H
methyl




methylphenyl





1.1.130
2-cyclopropyl-3-
H
methyl




methylphenyl





1.1.131
2-vinyl-3-
H
methyl




methylphenyl





1.1.132
2-ethynyl-3-
H
methyl




methylphenyl





1.1.133
2-cyano-3-
H
methyl




methylphenyl





1.1.134
2-trifluoromethyl-3-
H
methyl




methylphenyl





1.1.135
2-methoxy-3-
H
methyl




methylphenyl





1.1.136
2-ethoxy-3-
H
methyl




methylphenyl





1.1.137
2-trifluoromethoxy-3-
H
methyl




methylphenyl





1.1.138
2-nitro-3-
H
methyl




methylphenyl





1.1.139
2-fluoro-3-
H
methyl




ethylphenyl





1.1.140
2-chloro-3-
H
methyl




ethylphenyl





1.1.141
2-bromo-3-
H
methyl




ethylphenyl





1.1.142
2-methyl-3-
H
methyl




ethylphenyl





1.1.143
2,3-diethylphenyl
H
methyl



1.1.144
2-cyclopropyl-3-
H
methyl




ethylphenyl





1.1.145
2-vinyl-3-ethylphenyl
H
methyl



1.1.146
2-ethynyl-3-
H
methyl




ethylphenyl





1.1.147
2-cyano-3-
H
methyl




ethylphenyl





1.1.148
2-trifluoromethyl-3-
H
methyl




ethylphenyl





1.1.149
2-methoxy-3-
H
methyl




ethylphenyl





1.1.150
2-ethoxy-3-
H
methyl




ethylphenyl





1.1.151
2-trifluoromethoxy-3-
H
methyl




ethylphenyl





1.1.152
2-nitro-3-ethylphenyl
H
methyl



1.1.153
2-fluoro-3-
H
methyl




propylphenyl





1.1.154
2-chloro-3-
H
methyl




propylphenyl





1.1.155
2-bromo-3-
H
methyl




propylphenyl





1.1.156
2-methyl-3-
H
methyl




propylphenyl





1.1.157
2-methyl-3-
H
methyl




propylphenyl





1.1.158
2-cyclopropyl-3-
H
methyl




propylphenyl





1.1.159
2-vinyl-3-
H
methyl




propylphenyl





1.1.160
2-ethynyl-
H
methyl




3propylphenyl





1.1.161
2-cyano-3-
H
methyl




propylphenyl





1.1.162
2-trifluoromethyl-3-
H
methyl




propylphenyl





1.1.163
2-methoxy-3-
H
methyl




propylphenyl





1.1.164
2-ethoxy-3-
H
methyl




propylphenyl





1.1.165
2-trifluoromethoxy-3-
H
methyl




propylphenyl





1.1.166
2-nitro-3-
H
methyl




propylphenyl





1.1.167
2-fluoro-3-
H
methyl




isopropylphenyl





1.1.168
2-chloro-3-
H
methyl




isopropylphenyl





1.1.169
2-bromo-3-
H
methyl




isopropylphenyl





1.1.170
2-methyl-3-
H
methyl




isopropylphenyl





1.1.171
2-ethyl-3-
H
methyl




isopropylphenyl





1.1.172
2-cyclopropyl-3-
H
methyl




isopropylphenyl





1.1.173
2-vinyl-3-
H
methyl




isopropylphenyl





1.1.174
2-ethynyl-3-
H
methyl




isopropylphenyl





1.1.175
2-cyano-3-
H
methyl




isopropylphenyl





1.1.176
2-trifluoromethyl-3-
H
methyl




isopropylphenyl





1.1.177
2-methoxy-3-
H
methyl




isopropylphenyl





1.1.178
2-thoxy-3-
H
methyl




isopreopylphenyl





1.1.179
2-trifluoromethoxy-3-
H
methyl




isopropylphenyl





1.1.180
2-nitro-3-
H
methyl




isopropylphenyl





1.1.181
2-fluoro-3-tert-
H
methyl




butylphenyl





1.1.182
2-chloro-3-tert-
H
methyl




butylphenyl





1.1.183
2-bromo-3-tert-
H
methyl




butylphenyl





1.1.184
2-methyl-3-tert-
H
methyl




butylphenyl





1.1.185
2-ethyl-3-tert-
H
methyl




butylphenyl





1.1.186
2-cyclopropyl-3-tert-
H
methyl




butylphenyl





1.1.187
2-vinyl-3-tert-
H
methyl




butylphenyl





1.1.188
2-ethynyl-3-tert-
H
methyl




butylphenyl





1.1.189
2-cyano-3-tert-
H
methyl




butylphenyl





1.1.190
2-trifluoromethyl-3-
H
methyl




tert-butylphenyl





1.1.191
2-methoxy-3-tert-
H
methyl




butylphenyl





1.1.192
2-ethoxy-3-tert-
H
methyl




butylphenyl





1.1.193
2-trifluoromethoxy-3-
H
methyl




tert-butylphenyl





1.1.194
2-nitro-3-tert-
H
methyl




butylphenyl





1.1.195
2-fluoro-3-
H
methyl




hydroxymethylphenyl





1.1.196
2-chloro-3-
H
methyl




hydroxymethylphenyl





1.1.197
2-bromo-3-
H
methyl




hydroxymethylphenyl





1.1.198
2-methyl-3-
H
methyl




hydroxymethylphenyl





1.1.199
2-ethyl-3-
H
methyl




hydroxymethylphenyl





1.1.200
2-cyclopropy1-3-
H
methyl




hydroxymethylphenyl





1.1.201
2-vinyl-3-
H
methyl




hydroxymethylphenyl





1.1.202
2-ethyny1-3-
H
methyl




hydroxymethylphenyl





1.1.203
2-cyano-3-
H
methyl




hydroxymethylphenyl





1.1.204
2-trifluoromethyl-3-
H
methyl




hydroxymethylphenyl





1.1.205
2-methoxy-3-
H
methyl




hydroxymethylphenyl





1.1.206
2-ethoxy-3-
H
methyl




hydroxymethylphenyl





1.1.207
2-trifluoromethoxy-3-
H
methyl




hydroxymethylphenyl





1.1.208
2-nitro-3-
H
methyl




hydroxymethylphenyl





1.1.209
2-fluoro-3-
H
methyl




cyclopropylphenyl





1.1.210
2-chloro-3-
H
methyl




cyclopropylphenyl





1.1.211
2-bromo-3-
H
methyl




cyclopropylphenyl





1.1.212
2-methyl-3-
H
methyl




cyclopropylphenyl





1.1.213
2-ethyl-3-
H
methyl




cyclopropylphenyl





1.1.214
2-cyclopropyl-3-
H
methyl




cyclopropylphenyl





1.1.215
2-vinyl-3-
H
methyl




cyclopropylphenyl





1.1.216
2-ethynyl-3-
H
methyl




cyclopropylphenyl





1.1.217
2-cyano-3-
H
methyl




cyclopropylphenyl





1.1.218
2-trifluoromethyl-3-
H
methyl




cyclopropylphenyl





1.1.219
2-methoxy-3-
H
methyl




cyclopropylphenyl





1.1.220
2-ethoxy-3-
H
methyl




cyclopropylphenyl





1.1.221
2-trifluoromethoxy-3-
H
methyl




cyclopropylphenyl





1.1.222
2-fluoro-3-methoxy-
H
methyl




carbonylphenyl





1.1.223
2-chloro-3-methoxy-
H
methyl




carbonylphenyl





1.1.224
2-bromo-3-methoxy-
H
methyl




carbonylphenyl





1.1.225
2-methyl-3-methoxy-
H
methyl




carbonylphenyl





1.1.226
2-ethyl-3-methoxy-
H
methyl




carbonylphenyl





1.1.227
2-cyclopropyl-3-
H
methyl




methoxycarbonyl-






phenyl





1.1.228
2-vinyl-3-methoxy-
H
methyl




carbonylphenyl





1.1.229
2-ethynyl-3-methoxy-
H
methyl




carbonylphenyl





1.1.230
2-cyano-3-methoxy-
H
methyl




carbonylphenyl





1.1.231
2-trifluoromethyl-3-
H
methyl




methoxycarbonyl-






phenyl





1.1.232
2-methoxy-3-
H
methyl




methoxycarbonyl-






phenyl





1.1.233
2-ethoxy-3-methoxy-
H
methyl




carbonylphenyl





1.1.234
2-trifluoromethoxy-3-
H
methyl




methoxycarbonyl-






phenyl





1.1.235
2-nitro-3-methoxy-
H
methyl




carbonylphenyl





1.1.236
2-fluoro-3-
H
methyl




vinylphenyl





1.1.237
2-chloro-3-
H
methyl




vinylphenyl





1.1.238
2-bromo-3-
H
methyl




vinylphenyl





1.1.239
2-methyl-3-
H
methyl




vinylphenyl





1.1.240
2-ethyl-3-vinylphenyl
H
methyl



1.1.241
2-cyclopropyl-3-
H
methyl




vinylphenyl





1.1.242
2-vinyl-3-vinylphenyl 
H
methyl



1.1.243
2-ethynyl-3-
H
methyl




vinylphenyl





1.1.244
2-cyano-3-
H
methyl




vinylphenyl





1.1.245
2-trifluoromethyl-3-
H
methyl




vinylphenyl





1.1.246
2-methoxy-3-
H
methyl




vinylphenyl





1.1.247
2-ethoxy-3-
H
methyl




vinylphenyl





1.1.248
2-trifluoromethoxy-3-
H
methyl




vinylphenyl





1.1.249
2-nitro-3-vinylphenyl
H
methyl



1.1.250
2-fluoro-3-
H
methyl




ethynylphenyl





1.1.251
2-chloro-3-
H
methyl




ethynylphenyl





1.1.252
2-bromo-3-
H
methyl




ethynylphenyl





1.1.253
2-methyl-3-
H
methyl




ethynylphenyl





1.1.254
2-ethyl-3-
H
methyl




ethynylphenyl





1.1.255
2-cyclopropyl-3-
H
methyl




ethynylphenyl





1.1.256
2-vinyl-3-
H
methyl




ethynylphenyl





1.1.257
2-cyano-3-
H
methyl




ethynylphenyl





1.1.258
2-trifluoromethyl-3-
H
methyl




ethynylphenyl





1.1.259
2-methoxy-3-
H
methyl




ethynylphenyl





1.1.260
2-ethoxy-3-
H
methyl




ethynylphenyl





1.1.261
2-trifluoromethoxy-3-
H
methyl




ethynylphenyl





1.1.262
2-nitro-3-
H
methyl




ethynylphenyl





1.1.263
2-fluoro-3-
H
methyl




ethynylphenyl





1.1.264
2-fluoro-3-
H
methyl




cyanophenyl





1.1.265
2-chloro-3-
H
methyl




cyanophenyl





1.1.266
2-bromo-3-
H
methyl




cyanophenyl





1.1.267
2-methyl-3-
H
methyl




cyanophenyl





1.1.268
2-ethyl-3-
H
methyl




cyanophenyl





1.1.269
2-ethyl-3-
H
ethyl




cyanophenyl





1.1.270
2-ethyl-3-
H
propyl




cyanophenyl





1.1.271
2-ethyl-3 -
H
cyclopropyl




cyanophenyl





1.1.272
2-cyclopropyl-3-
H
methyl




cyanophenyl





1.1.273
2-vinyl-3-
H
methyl




cyanophenyl





1.1.274
2-ethynyl-3-
H
methyl




cyanophenyl





1.1.275
2-cyano-3-
H
methyl




cyanophenyl





1.1.276
2-trifluoromethyl-3-
H
methyl




cyanophenyl





1.1.277
2-methoxy-3-
H
methyl




cyanophenyl





1.1.278
2-ethoxy-3-
H
methyl




cyanophenyl





1.1.279
2-trifluoromethoxy-3-
H
methyl




cyanophenyl





1.1.280
2-nitro-3-
H
methyl




cyanophenyl





1.1.281
2-fluoro-3-
H
methyl




hydroxyphenyl





1.1.282
2-chloro-3-
H
methyl




hydroxyphenyl





1.1.283
2-bromo-3-
H
methyl




hydroxyphenyl





1.1.284
2-methyl-3-
H
methyl




hydroxyphenyl





1.1.285
2-ethyl-3-
H
methyl




hydroxyphenyl





1.1.286
2-cyclopropyl-3-
H
methyl




hydroxyphenyl





1.1.287
2-vinyl-3-
H
methyl




hydroxyphenyl





1.1.288
2-ethynyl-3-
H
methyl




hydroxyphenyl





1.1.289
2-cyano-3-
H
methyl




hydroxyphenyl





1.1.290
2-trifluoromethyl-3-
H
methyl




hydroxyphenyl





1.1.291
2-methoxy-3-
H
methyl




hydroxyphenyl





1.1.292
2-ethoxy-3-
H
methyl




hydroxyphenyl





1.1.293
2-trifluoromethoxy-3-
H
methyl




hydroxyphenyl





1.1.294
2-nitro-3-
H
methyl




hydroxyphenyl





1.1.295
2-fluoro-3-
H
methyl




methoxyphenyl





1.1.296
2-chloro-3-
H
methyl




methoxyphenyl





1.1.297
2-bromo-3-
H
methyl




methoxyphenyl





1.1.298
2-methyl-3-
H
methyl




methoxyphenyl





1.1.299
2-ethyl-3-
H
methyl




methoxyphenyl





1.1.300
2-cyclopropyl-3-
H
methyl




methoxyphenyl





1.1.301
2-vinyl-3-
H
methyl




methoxyphenyl





1.1.302
2-ethynyl-3-
H
methyl




methoxyphenyl





1.1.303
2-cyano-3-
H
methyl




methoxyphenyl





1.1.304
2-trifluoromethyl-3-
H
methyl




methoxyphenyl





1.1.305
2,3-dimethoxy-
H
methyl




phenyl





1.1.306
2-ethoxy-3-
H
methyl




methoxyphenyl





1.1.307
2-trifluoromethoxy-3-
H
methyl




methoxyphenyl





1.1.308
2-nitro-3-
H
methyl




methoxyphenyl





1.1.309
2-fluoro-3-
H
methyl




ethoxyphenyl





1.1.310
2-chloro-3-
H
methyl




ethoxyphenyl





1.1.311
2-bromo-3-
H
methyl




ethoxyphenyl





1.1.312
2-methyl-3-
H
methyl




ethoxyphenyl





1.1.313
2-ethyl-3-
H
methyl




ethoxyphenyl





1.1.314
2-cyclopropyl-3-
H
methyl




ethoxyphenyl





1.1.315
2-vinyl-3-
H
methyl




ethoxyphenyl





1.1.316
2-ethynyl-3-
H
methyl




ethoxyphenyl





1.1.317
2-cyano-3-
H
methyl




ethoxyphenyl





1.1.318
2-trifluoromethyl-3-
H
methyl




ethoxyphenyl





1.1.319
2-methoxy-3-
H
methyl




ethoxyphenyl





1.1.320
2,3-diethoxyphenyl
H
methyl



1.1.321
2-trifluoromethoxy-3-
H
methyl




ethoxyphenyl





1.1.322
2-nitro-3-
H
methyl




ethoxyphenyl





1.1.323
2-fluoro-3-
H
methyl




propoxyphenyl





1.1.324
2-chloro-3-
H
methyl




propoxyphenyl





1.1.325
2-bromo-3-
H
methyl




propoxyphenyl





1.1.326
2-methyl-3-
H
methyl




propoxyphenyl





1.1.327
2-ethyl-3-
H
methyl




propoxyphenyl





1.1.328
2-cyclopropyl-3-
H
methyl




propoxyphenyl





1.1.329
2-vinyl-3-
H
methyl




propoxyphenyl





1.1.330
2-ethynyl-3-
H
methyl




propoxyphenyl





1.1.331
2-cyano-3-
H
methyl




propoxyphenyl





1.1.332
2-trifluoromethyl-3-
H
methyl




propoxyphenyl





1.1.333
2-methoxy-3-
H
methyl




propoxyphenyl





1.1.334
2-ethoxy-3-
H
methyl




propoxyphenyl





1.1.335
2-trifluoromethoxy-3-
H
methyl




propoxyphenyl





1.1.336
2-nitro-3-
H
methyl




propoxyphenyl





1.1.337
2-fluoro-3-
H
methyl




isopropoxyphenyl





1.1.338
2-chloro-3-
H
methyl




isopropoxyphenyl





1.1.339
2-bromo-3-
H
methyl




isopropoxyphenyl





1.1.340
2-methy1-3-
H
methyl




isopropoxyphenyl





1.1.341
2-ethyl-3-
H
methyl




isopropoxyphenyl





1.1.342
2-cyclopropyl-3-
H
methyl




isopropoxyphenyl





1.1.343
2-vinyl-3-
H
methyl




isopropoxyphenyl





1.1.344
2-ethynyl-3-
H
methyl




isopropoxyphenyl





1.1.345
2-cyano-3-
H
methyl




isopropoxyphenyl





1.1.346
2-trifluoromethyl-3-
H
methyl




isopropoxyphenyl





1.1.347
2-methoxy-3-
H
methyl




isopropoxyphenyl





1.1.348
2-ethoxy-3-
H
methyl




isopropoxyphenyl





1.1.349
2-trifluoromethoxy-3-
H
methyl




isopropoxyphenyl





1.1.350
2-nitro-3-isopropoxy-
H
methyl




phenyl





1.1.351
2-fluoro-3-tert-
H
methyl




butoxyphenyl





1.1.352
2-chloro-3-tert-
H
methyl




butoxyphenyl





1.1.353
2-bromo-3-tert-
H
methyl




butoxyphenyl





1.1.354
2-methyl-3-tert-
H
methyl




butoxyphenyl





1.1.355
2-ethyl-3-tert-
H
methyl




butoxyphenyl





1.1.356
2-cyclopropyl-3-tert-
H
methyl




butoxyphenyl





1.1.357
2-vinyl-3-tert-
H
methyl




butoxyphenyl





1.1.358
2-ethynyl-3-tert-
H
methyl




butoxyphenyl





1.1.359
2-cyano-3-tert-
H
methyl




butoxyphenyl





1.1.360
2-trifluoromethyl-3-
H
methyl




tert-butoxyphenyl





1.1.361
2-methoxy-3-tert-
H
methyl




butoxyphenyl





1.1.362
2-ethoxy-3-tert-
H
methyl




butoxyphenyl





1.1.363
2-trifluoromethoxy-3-
H
methyl




tert-butoxyphenyl





1.1.364
2-nitro-3-tert-
H
methyl




butoxyphenyl





1.1.365
2-fluoro-3-trifluoro-
H
methyl




methoxyphenyl





1.1.366
2-chloro-3-trifluoro-
H
methyl




methoxyphenyl





1.1.367
2-bromo-3-trifluoro-
H
methyl




methoxyphenyl





1.1.368
2-methy1-3-trifluoro-
H
methyl




methoxyphenyl





1.1.369
2-ethyl-3-trifluoro-
H
methyl




methoxyphenyl





1.1.370
2-cyclopropyl-3-
H
methyl




trifluoromethoxy-






phenyl





1.1.371
2-viny1-3-trifluoro-
H
methyl




methoxyphenyl





1.1.372
2-ethynyl-3-trifluoro-
H
methyl




methoxyphenyl





1.1.373
2-cyano-3-trifluoro-
H
methyl




methoxyphenyl





1.1.374
2-trifluoromethyl-3-
H
methyl




trifluoromethoxy-






phenyl





1.1.375
2-methoxy-3-
H
methyl




trifluoromethoxy-






phenyl





1.1.376
2-ethoxy-3-trifluoro-
H
methyl




methoxyphenyl





1.1.377
2,3-bis(trifluoro-
H
methyl




methoxy)phenyl





1.1.378
2-nitro-3-trifluoro-
H
methyl




methoxyphenyl





1.1.379
2-fluoro-3-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.380
2-chloro-3-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.381
2-bromo-3-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.382
2-methyl-3-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.383
2-ethyl-3-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.384
2-cyclopropy1-3-
H
methyl




(2,2,2-trifluoro-






ethoxy)phenyl





1.1.385
2-vinyl-3-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.386
2-ethynyl-3-(2,2,2-
H
methyl




trifluoroethoxyphenyl





1.1.387
2-cyano-3-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.388
2-trifluoromethyl-3-
H
methyl




(2,2,2-trifluoro-






ethoxy)phenyl





1.1.389
2-methoxy-3-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.390
2-ethoxy-3-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.391
2-trifluoromethoxy-3-
H
methyl




(2,2,2-trifluoro-






ethoxy)phenyl





1.1.392
2-nitro-3-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.393
2-fluoro-3-
H
methyl




difluoromethoxy-






phenyl





1.1.394
2-chloro-3-
H
methyl




difluoromethoxy-






phenyl





1.1.395
2-bromo-3-
H
methyl




difluoromethoxy-






phenyl





1.1.396
2-methyl-3-
H
methyl




difluoromethoxy-






phenyl





1.1.397
2-ethyl-3-
H
methyl




difluoromethoxy-






phenyl





1.1.398
2-cyclopropyl-3-
H
methyl




difluoromethoxy-






phenyl





1.1.399
2-vinyl-3-
H
methyl




difluoromethoxy-






phenyl





1.1.400
2-ethynyl-3-
H
methyl




difluoromethoxy-






phenyl





1.1.401
2-cyano-3-difluoro-
H
methyl




methoxyphenyl





1.1.402
2-trifluoromethyl-3-
H
methyl




difluoromethoxy-






phenyl





1.1.403
2-methoxy-3-difluoro-
H
methyl




methoxyphenyl





1.1.404
2-ethoxy-3-difluoro-
H
methyl




methoxyphenyl





1.1.405
2-trifluoromethoxy-3-
H
methyl




difluoromethoxy-






phenyl





1.1.406
2-nitro-3-difluoro-
H
methyl




methoxyphenyl





1.1.407
2-fluoro-3-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.408
2-chloro-3-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.409
2-bromo-3-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.410
2-methyl-3-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.411
2-ethyl-3-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.412
2-cyclopropyl-3-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.413
2-vinyl-3-(2-methoxy-
H
methyl




ethoxy)phenyl





1.1.414
2-ethynyl-3-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.415
2-cyano-3-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.416
2-trifluoromethy1-3-
H
methyl




(2-methoxyethoxy)-






phenyl





1.1.417
2-methoxy-3-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.418
2-ethoxy-3-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.419
2-trifluoromethoxy-
H
methyl




(2-methoxyethoxy)-






phenyl





1.1.420
2-nitro-3-(2-methoxy-
H
methyl




ethoxy)phenyl





1.1.421
2-fluoro-3-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.422
2-chloro-3-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.423
2-bromo-3-(tert-
H
methyl




butoxycarbonyl-






oxy)phenyl





1.1.424
2-methyl-3-(tert-
H
methyl




butoxycarbonyl-






oxy)phenyl





1.1.425
2-ethyl-3-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.426
2-cyclopropyl-3-(tert-
H
methyl




butoxycarbonyl-






oxy)phenyl





1.1.427
2-vinyl-3-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.428
2-ethynyl-3-(tert-
H
methyl




butoxycarbonyl-






oxy)phenyl





1.1.429
2-cyano-3-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.430
2-trifluoromethyl-3-
H
methyl




(tert-butoxycarbonyl-






oxy)phenyl





1.1.431
2-methoxy-3-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.432
2-ethoxy-3-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.433
2-trifluoromethoxy-3-
H
methyl




(tert-butoxycarbonyl-






oxy)phenyl





1.1.434
2-nitro-3-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.435
2-fluoro-3-nitrophenyl
H
methyl



1.1.436
2-chloro-3-
H
methyl




nitrophenyl





1.1.437
2-bromo-3-
H
methyl




nitrophenyl





1.1.438
2-methyl-3-
H
methyl




nitrophenyl





1.1.439
2-ethyl-3-nitrophenyl
H
methyl



1.1.440
2-cyclopropyl-3-
H
methyl




nitrophenyl





1.1.441
2-vinyl-3-nitrophenyl
H
methyl



1.1.442
2-ethynyl-3-
H
methyl




nitrophenyl





1.1.443
2-cyano-3-
H
methyl




nitrophenyl





1.1.444
2-trifluoromethyl-3-
H
methyl




nitrophenyl





1.1.445
2-methoxy-3-
H
methyl




nitrophenyl





1.1.446
2-ethoxy-3-
H
methyl




nitrophenyl





1.1.447
2-trifluoromethoxy-3-
H
methyl




nitrophenyl





1.1.448
2-fluoro-3-
H
methyl




methylsulfanylphenyl





1.1.449
2-chloro-3-
H
methyl




methylsulfanylphenyl





1.1.450
2-bromo-3-
H
methyl




methylsulfanylphenyl





1.1.451
2-methy1-3-
H
methyl




methylsulfanylphenyl





1.1.452
2-ethyl-3-
H
methyl




methylsulfanylphenyl





1.1.453
2-cyclopropyl-3-
H
methyl




methylsulfanylphenyl





1.1.454
2-vinyl-3-
H
methyl




methylsulfanylphenyl





1.1.455
2-ethynyl-3-
H
methyl




methylsulfanylphenyl





1.1.456
2-cyano-3-
H
methyl




methylsulfanylphenyl





1.1.457
2-trifluoromethy1-3-
H
methyl




methylsulfanylphenyl





1.1.458
2-methoxy-3-
H
methyl




methylsulfanylphenyl





1.1.459
2-ethoxy-3-
H
methyl




methylsulfanylphenyl





1.1.460
2-trifluoromethoxy-3-
H
methyl




methylsulfanylphenyl





1.1.461
2-nitro-3-
H
methyl




methylsulfanylphenyl





1.1.462
3,5-difluorophenyl
H
methyl
[CDCl3] 1.80 (s, 3H); 3.25 (d, 1H);






3.83 (d, 1H); 6.90 (m, 1H); 7.15 (m,






2H).


1.1.463
(R)-3,5-
H
methyl
[CDCl3] 1.79 (s, 3H); 1.90 (s br, 1H);



difluorophenyl


3.26 (d, 1H); 3.84 (d, 1H), 6.90






(t, 1H); 7.18 (d, 2H).


1.1.464
(S)-3,5-
H
methyl
[CDCl3] 1.79 (s, 3H); 3.25 (d, 1H);



difluorophenyl


3.83 (d, 1H), 6.89 (t, 1H); 7.18






(d, 2H).


1.1.465
rel-(4R,5R)-3,5-
methyl
methyl




difluorophenyl





1.1.466
rel-(4R,5R)-3,5-
ethyl
methyl
[CDCl3] 0.93 (t, 3H); 1.61 (s, 3H);



difluorophenyl


1.75 (m, 2H); 3.84 (dd, 1H); 6.90






(m, 1H); 7.21 (m, 2H).


1.1.467
3,5-difluorophenyl
Br
methyl



1.1.468
3,5-difluorophenyl
H
ethyl
[CDCl3] 1.09 (t, 3H); 2.12 (mc, 2H);






3.30 (d, 1H); 3.75 (d, 1H); 6.90 (m,






1H); 7.18 (m, 2H).


1.1.469
3,5-difluorophenyl
H
isopropyl
[CDCl3] 1.06 (m, 6H); 2.40 (m, 1H);






3.30 (d, 1H); 3.70 (d, 1H); 6.90






(m, 1H); 7.19 (m, 2H).


1.1.470
3,5-difluorophenyl
H
cyclopropyl



1.1.471
3-chloro-5-
H
methyl
[CDCl3] 1.76 (s, 3H); 3.25 (d, 1H);



fluorophenyl


3.82 (d, 1H); 7.16 (m, 1H); 7.30 (m,






1H); 7.4 (bs, 1H).


1.1.472
3-chloro-5-
H
ethyl
[CDCl3] 1.05 (t, 3H); 2.11 (mc, 2H);



fluorophenyl


3.28 (d, 1H); 3.75 (d, 1H); 7.18 (m,






1H); 7.28 (m, 1H); 7.40 (1H).


1.1.473
3-chloro-5-
H
isopropyl




fluorophenyl





1.1.474
3-chloro-5-
H
cyclopropyl




fluorophenyl





1.1.475
3-bromo-5-
H
methyl
[CDCl3] 1.70 (s, 3H); 3.25 (d, 1H);



fluorophenyl


3.85 (d, 1H); 7.35 (m, 2H); 7.56 (m,






1H).


1.1.476
3-bromo-5-
H
ethyl




fluorophenyl





1.1.477
3-bromo-5-
H
isopropyl




fluorophenyl





1.1.478
3-bromo-5-
H
cyclopropyl




fluorophenyl





1.1.479
3-iodo-5-fluorophenyl
H
methyl



1.1.480
3-methyl-5-
H
methyl
[DMSO] 1.51 (s, 3H); 2.35 (s, 3H);



fluorophenyl


3.31 (d, 1H); 3.76 (d, 1H); 7.14 (d,






1H); 7.25 (d, 1H); 7.35 (s, 1H).


1.1.481
3-methyl-5-
H
ethyl




fluorophenyl





1.1.482
3-methyl-5-
H
propyl




fluorophenyl





1.1.483
3-methyl-5-
H
cyclopropyl




fluorophenyl





1.1.484
3-ethyl-5-
H
methyl
[DMSO] 1.20 (t, 3H); 1.55 (s, 3H);



fluorophenyl


2.65 (q, 2H); 3.38 (d, 1H); 3.80 (d,






1H); 7.15 (d, 1H); 7.38 (d, 1H); 7.39






(s, 1H).


1.1.485
3-propyl-5-
H
methyl




fluorophenyl





1.1.486
3-i-propyl-5-
H
methyl




fluorophenyl





1.1.487
3-n-butyl-5-
H
methyl




fluorophenyl





1.1.488
3-isobutyl-5-
H
methyl




fluorophenyl





1.1.489
3-tert-butyl-5-
H
methyl




fluorophenyl





1.1.490
3-cyclopropyl-5-
H
methyl
[CDCl3] 0.71 (m, 2H); 1.03 (m, 2H);



fluorophenyl


1.75 (s, 3H); 1.91 (m, 1H); 3.26 (d,






1H); 3.85 (d, 1H); 6.81 (dd, 1H);






7.13 (dd, 2H).


1.1.491
3-vinyl-5-
H
methyl
[CDCl3] 1.80 (s, 3H); 3.27 (d, 1H);



fluorophenyl


3.86 (d, 1H); 5.39 (d, 1H); 5.8 (d,






1H); 6.69 (dd, 1H); 7.19 (m, 1H);






7.25 (m, 1H); 7.40 (bs, 1H).


1.1.492
3-ethynyl-5-
H
methyl




fluorophenyl





1.1.493
3-cyano-5-
H
methyl




fluorophenyl





1.1.494
3-trifluoromethyl-5-
H
methyl
[CDCl3] 1.80 (s, 3H); 3.29 (d, 1H);



fluorophenyl


3.90 (d, 1H); 7.40 (m, 1H); 7.59 (m,






1H); 7.66 (s, 1H).


1.1.495
3-trifluoromethyl-5-
H
ethyl




fluorophenyl





1.1.496
3-trifluoromethyl-5-
H
propyl




fluorophenyl





1.1.497
3-trifluoromethyl-5-
H
cyclopropyl




fluorophenyl





1.1.498
3-(methoxycarbonyl)-
H
methyl




5-fluorophenyl





1.1.499
3-hydroxymethyl-5-
H
methyl




fluorophenyl





1.1.500
3-carbamoyl-5-
H
methyl




fluorophenyl





1.1.501
3-hydroxy-5-
H
methyl




fluorophenyl





1.1.502
3-methoxy-5-
H
methyl
[CDCl3] 1.78 (s, 3H); 3.25 (d, 1H);



fluorophenyl


3.82 (s, 3H); 3.88 (d, 1H); 6.7 (dd,






1H); 6.92 (dd, 1H); 7.05 (bs, 1H).


1.1.503
3-ethoxy-5-
H
methyl




fluorophenyl





1.1.504
3-n-propoxy-5-
H
methyl




fluorophenyl





1.1.505
3-isopropoxy-5-
H
methyl




fluorophenyl





1.1.506
3-n-butoxy-5-
H
methyl




fluorophenyl





1.1.507
3-isobutoxy-5-
H
methyl




fluorophenyl





1.1.508
3-tert-butoxy-5-
H
methyl




fluorophenyl





1.1.509
3-difluoromethoxy-5-
H
methyl




fluorophenyl





1.1.510
3-trifluoromethoxy-5-
H
methyl




fluorophenyl





1.1.511
3-(2,2,2-
H
methyl




trifluoroethoxy)-5-






fluorophenyl





1.1.512
3-(2-chloroethoxy)-5-
H
methyl




fluorophenyl





1.1.513
3-(2-hydroxyethoxy)-
H
methyl




5-fluorophenyl





1.1.514
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






fluorophenyl





1.1.515
3-nitro-5-fluorophenyl
H
methyl



1.1.516
3-acetoxy-5-
H
methyl




fluorophenyl





1.1.517
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






fluorophenyl}





1.1.518
3-methylsulfanyl-5-
H
methyl




fluorophenyl





1.1.519
3,5-dichlorophenyl
H
methyl
[CDCl3] 1.79 (s, 3H); 3.25 (d, 1H),






3.83 (d, 1H); 7.41 (s, 1H); 7.53






(s, 2H).


1.1.520
(R)-3,5-
H
methyl
[CDCl3] 1.78 (s, 3H); 3.25 (d, 1H);



dichlorophenyl


3.83 (d, 1H); 5.3 (s br, 1H); 7.42






(s, 1H); 7.52 (s, 2H).


1.1.521
(S)-3,5-
H
methyl
[CDCl3] 1.78 (s, 3H); 3.25 (d, 1H),



dichlorophenyl


3.83 (d, 1H); 5.3 (s br, 1H); 7.42






(s, 1H); 7.52 (s, 2H).


1.1.522
rel-(4R,5S)-3,5-
methyl
methyl
[CDCl3] 1.30 (d, 3H); 1.70 (s, 3H);



dichlorophenyl


3.55 (q, 1H); 7.44 (m, 1H); 7.55 (m,






2H).


1.1.523
rel-(4R,5R)-3,5-
methyl
methyl
[CDCl3] 1.25 (d, 3H); 1.70 (s, 3H);



dichlorophenyl


3.95 (q, 2H); 7.42 (m, 1H); 7.58 (m,






2H).


1.1.524
3,5-dichlorophenyl
H
ethyl
[CDCl3] 1.18 (dq, 3H); 2.11 (m, 2H);






3.30 (d, 1H); 3.75 (d, 1H); 7.42 (s,






1H), 7.72 (s, 1H).


1.1.525
3,5-dichlorophenyl
H
isopropyl
[CDCl3] 1.18 (dd, 6H); 2.40 (dq,






1H); 3.32 (d, 1H); 3.70 (d, 1H); 7.41






(bs, 1H); 7.55 (bs, 2H).


1.1.526
3,5-dichlorophenyl
H
cyclopropyl
[CDCl3] 0.45-0.80 (m, 4H); 1.51 (m,






1H); 3.39 (d, 1H); 3.82 (d, 1H); 7.42






(m, 1H); 7.50 (m, m, 2H).


1.1.527
3-bromo-5-
H
methyl
[CDCl3] 1.79 (s, 3H); 3.25 (d, 1H);



chlorophenyl


3.85 (d, 1H); 7.60 (s, 2H); 7.70 (s,






1H).


1.1.528
3-iodo-5-
H
methyl




chlorophenyl





1.1.529
3-methyl-5-
H
methyl
[DMSO] 1.55 (s, 3H); 2.35 (s, 3H);



chlorophenyl


3.38 (d, 1H); 3.77 (d, 1H); 7.38 (s,






1H); 7.50 (d, 1H).


1.1.530
3-ethyl-5-
H
methyl
[CDCl3] 1.25 (7. 3H); 1.80 (s, 3H);



chlorophenyl


2.68 (q, 2H); 3.27 (d, 1H); 3.85 (d,






1H); 7.28 (m, 1H); 3.38 (s, 1H);






7.43 (s, 1H).


1.1.531
3-propy1-5-
H
methyl




chlorophenyl





1.1.532
3-isopropyl-5-
H
methyl




chlorophenyl





1.1.533
3-n-butyl-5-
H
methyl




chlorophenyl





1.1.534
3-isobutyl-5-
H
methyl




chlorophenyl





1.1.535
3-tert-butyl-5-
H
methyl




chlorophenyl





1.1.536
3-cyclopropyl-5-
H
methyl




chlorophenyl





1.1.537
3-vinyl-5-
H
methyl




chlorophenyl





1.1.538
3-ethynyl-5-
H
methyl




chlorophenyl





1.1.539
3-cyano-5-
H
methyl




chlorophenyl





1.1.540
3-trifluoromethyl-5-
H
methyl
[CDCl3] 1.80 (s, 3H); 3.30 (d, 1H);



chlorophenyl


3.89 (d, 1H); 7.69 (s, 1H); 7.78 (s,






1 H); 7.82 (s, 1 H).


1.1.541
3-(hydroxycarbonyl)-
H
methyl




5-chlorophenyl





1.1.542
3-(methoxycarbonyl)-
H
methyl




5-chlorophenyl





1.1.543
3-hydroxymethyl-5-
H
methyl




chlorophenyl





1.1.544
3-carbamoyl-5-
H
methyl




chlorophenyl





1.1.545
3-hydroxy-5-
H
methyl




chlorophenyl





1.1.546
3-methoxy-5-
H
methyl
[CDCl3] 1.77 (s, 3H); 3.25 (d, 1H);



chlorophenyl


3.71 (s, 3H); 3.82 (d, 1H); 6.95-






7.18 (m, Ar, 3H)


1.1.547
3-ethoxy-5-
H
methyl




chlorophenyl





1.1.548
3-n-propoxy-5-
H
methyl




chlorophenyl





1.1.549
3-isopropoxy-5-
H
methyl




chlorophenyl





1.1.550
3-n-butoxy-5-
H
methyl




chlorophenyl





1.1.551
3-isobutoxy-5-
H
methyl




chlorophenyl





1.1.552
3-tert-butoxy-5-
H
methyl




chlorophenyl





1.1.553
3-difluoromethoxy-5-
H
methyl




chlorophenyl





1.1.554
3-trifluoromethoxy-5-
H
methyl
[DMSO] 1.59 (s, 3H); 3.43 (d, 1H);



chlorophenyl


3.85 (d, 1H); 7.63 (s, 1H); 7.69 (s,






1H); 6.78 (s, 1H).


1.1.555
3-(2,2,2-
H
methyl




trifluoroethoxy)-5-






chlorophenyl





1.1.556
3-(2-chloroethoxy)-5-
H
methyl




chlorophenyl





1.1.557
3-(2-hydroxyethoxy)-
H
methyl




5-chlorophenyl





1.1.558
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






chlorophenyl





1.1.559
3-nitro-5-
H
methyl




chlorophenyl





1.1.560
3-acetoxy-5-
H
methyl




chlorophenyl





1.1.561
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






chlorophenyl}





1.1.562
3-methylsulfanyl-5-
H
methyl




chlorophenyl





1.1.563
3,5-dibromophenyl
H
methyl
[CDCl3] 1.80 (s, 3H); 3.25 (d, 1H);






3.85 (d, 1H); 7.73 (s, 3H).


1.1.564
3,5-dibromophenyl
H
ethyl
[CDCl3] 1.08 (t, 3H); 2.10 (m, 2H);






3.25 (d, 1H); 3.75 (d, 1H); 7.72 (s,






3H).


1.1.565
3-iodo-5-
H
methyl




bromophenyl





1.1.566
3-methyl-5-
H
methyl
[CDCl3] 1.78 (s, 3H); 2.36 (s, 3H);



bromophenyl


3.27 (d, 1H); 3.84 (d, 1H); 7.40






(s, 2H); 7.57 (s, 1H).


1.1.567
3-methyl-5-
H
ethyl




bromophenyl





1.1.568
3-methyl-5-
H
isopropyl




bromophenyl





1.1.569
3-methyl-5-
H
cyclopropyl



1.1.570
3-ethyl-5-
H
methyl




bromophenyl





1.1.571
3-propyl-5-
H
methyl




bromophenyl





1.1.572
3-isopropyl-5-
H
methyl




bromophenyl





1.1.573
3-n-butyl-5-
H
methyl




bromophenyl





1.1.574
3-isobutyl-5-
H
methyl




bromophenyl





1.1.575
3-tert-butyl-5-
H
methyl




bromophenyl





1.1.576
3-cyclopropyl-5-
H
methyl




bromophenyl





1.1.577
3-vinyl-5-
H
methyl




bromophenyl





1.1.578
3-ethynyl-5-
H
methyl




bromophenyl





1.1.579
3-cyano-5-
H
methyl




bromophenyl





1.1.580
3-trifluoromethyl-5-
H
methyl
[CDCl3] 1.80 (s, 3H); 3.30 (d, 1H);



bromophenyl


3.90 (d, 1H); 7.81 (s, 2H); 8.0 (s,






1H).


1.1.581
3-(hydroxycarbonyl)-
H
methyl




5-bromophenyl





1.1.582
3-(methoxycarbonyl)-
H
methyl




5-bromophenyl





1.1.583
3-hydroxymethyl-5-
H
methyl




bromophenyl





1.1.584
3-carbamoyl-5-
H
methyl




bromophenyl





1.1.585
3-hydroxy -5-
H
methyl




bromophenyl





1.1.586
3-methoxy-5-
H
methyl




bromophenyl





1.1.587
3-ethoxy-5-
H
methyl




bromophenyl





1.1.588
3-n-propoxy-5-
H
methyl




bromophenyl





1.1.589
3-isopropoxy-5-
H
methyl




bromophenyl





1.1.590
3-n-butoxy-5-
H
methyl




bromophenyl





1.1.591
3-isobutoxy-5-
H
methyl




bromophenyl





1.1.592
3-tert-butoxy-5-
H
methyl




bromophenyl





1.1.593
3-difluoromethoxy-5-
H
methyl




bromophenyl





1.1.594
3-trifluoromethoxy-5-
H
methyl




bromophenyl





1.1.595
3-(2,2,2-
H
methyl




trifluoroethoxy)-5-






bromophenyl





1.1.596
3-(2-chloroethoxy)-5-
H
methyl




bromophenyl





1.1.597
3-(2-hydroxyethoxy)-
H
methyl




5-bromophenyl





1.1.598
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






bromophenyl





1.1.599
3-nitro-5-
H
methyl




bromophenyl





1.1.600
3-acetoxy-5-
H
methyl




bromophenyl





1.1.601
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






bromophenyl}





1.1.602
3-methylsulfanyl-5-
H
methyl




bromophenyl





1.1.603
3,5-diiodophenyl
H
methyl
[CDCl3] 1.75 (s, 3H); 3.23 (d; 1H);






3.80 (d, 1H); 7.91 (s, 2H); 8.10 (s,






1H):


1.1.604
3-methyl-5-
H
methyl




iodophenyl





1.1.605
3-ethyl-5-iodophenyl
H
methyl



1.1.606
3-propy1-5-
H
methyl




iodophenyl





1.1.607
3-isopropyl-5-
H
methyl




iodophenyl





1.1.608
3-n-butyl-5-
H
methyl




iodophenyl





1.1.609
3-isobutyl-5-
H
methyl




iodophenyl





1.1.610
3-tert-butyl-5-
H
methyl




iodophenyl





1.1.611
3-cyclopropyl-5-
H
methyl




iodophenyl





1.1.612
3-vinyl-5-iodophenyl
H
methyl



1.1.613
3-ethynyl-5-
H
methyl




iodophenyl





1.1.614
3-cyano-5-
H
methyl




iodophenyl





1.1.615
3-trifluoromethyl-5-
H
methyl




iodophenyl





1.1.616
3-(hydroxycarbonyl)-
H
methyl




5-iodophenyl





1.1.617
3-(methoxycarbonyl)-
H
methyl




5-iodophenyl





1.1.618
3-hydroxymethyl-5-
H
methyl




iodophenyl





1.1.619
3-carbamoyl-5-
H
methyl




iodophenyl





1.1.620
3-hydroxy -5-
H
methyl




iodophenyl





1.1.621
3-methoxy-5-
H
methyl




iodophenyl





1.1.622
3-ethoxy-5-
H
methyl




iodophenyl





1.1.623
3-n-propoxy-5-
H
methyl




iodophenyl





1.1.624
3-isopropoxy-5-
H
methyl




iodophenyl





1.1.625
3-n-butoxy-5-
H
methyl




iodophenyl





1.1.626
3-isobutoxy-5-
H
methyl




iodophenyl





1.1.627
3-tert-butoxy-5-
H
methyl




iodophenyl





1.1.628
3-difluoromethoxy-5-
H
methyl




iodophenyl





1.1.629
3-trifluoromethoxy-5-
H
methyl




iodophenyl





1.1.630
3-(2,2,2-
H
methyl




trifluoroethoxy)-5-






iodophenyl





1.1.631
3-(2-chloroethoxy)-5-
H
methyl




iodophenyl





1.1.632
3-(2-hydroxyethoxy)-
H
methyl




5-iodophenyl





1.1.633
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






iodophenyl





1.1.634
3-nitro-5-iodophenyl
H
methyl



1.1.635
3-acetoxy-5-
H
methyl




iodophenyl





1.1.636
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






iodophenyl}





1.1.637
3-methylsulfanyl-5-
H
methyl




iodophenyl





1.1.638
3,5-dimethylphenyl
H
methyl
[CDCl3] 1.75 (s, 3H);, 2.32 (s, 6H);






3.3 (d, 1H); 3.85 (d. 1H); 7.09 (s,






1H); 7.35 (s, 2H).


1.1.639
3-ethyl-5-
H
methyl




methylphenyl





1.1.640
3-propyl-5-
H
methyl




methylphenyl





1.1.641
3-isopropyl-5-
H
methyl




methylphenyl





1.1.642
3-n-butyl-5-
H
methyl




methylphenyl





1.1.643
3-isobutyl-5-
H
methyl




methylphenyl





1.1.644
3-tert-butyl-5-
H
methyl




methylphenyl





1.1.645
3-cyclopropyl-5-
H
methyl




methylphenyl





1.1.646
3-vinyl-5-
H
methyl




methylphenyl





1.1.647
3-ethynyl-5-
H
methyl




methylphenyl





1.1.648
3-cyano-5-
H
methyl




methylphenyl





1.1.649
3-trifluoromethyl-5-
H
methyl




methylphenyl





1.1.650
3-(hydroxycarbonyl)-
H
methyl




5-methylphenyl





1.1.651
3-(methoxycarbonyl)-
H
methyl




5-methylphenyl





1.1.652
3-hydroxymethyl-5-
H
methyl




methylphenyl





1.1.653
3-carbamoyl-5-
H
methyl




methylphenyl





1.1.654
3-hydroxy-5-
H
methyl




methylphenyl





1.1.655
3-methoxy-5-
H
methyl




methylphenyl





1.1.656
3-ethoxy-5-
H
methyl




methylphenyl





1.1.657
3-n-propoxy-5-
H
methyl




methylphenyl





1.1.658
3-n-butoxy-5-
H
methyl




methylphenyl





1.1.659
3-isobutoxy-5-
H
methyl




methylphenyl





1.1.660
3-tert-butoxy-5-
H
methyl




methylphenyl





1.1.661
3-difluoromethoxy-5-
H
methyl




methylphenyl





1.1.662
3-trifluoromethoxy-5-
H
methyl




methylphenyl





1.1.663
3-(2,2,2-
H
methyl




trifluoroethoxy)-5-






methylphenyl





1.1.664
3-(2-chloroethoxy)-5-
H
methyl




methylphenyl





1.1.665
3-(2-hydroxyethoxy)-
H
methyl




5-methylphenyl





1.1.666
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






methylphenyl





1.1.667
3-nitro-5-
H
methyl




methylphenyl





1.1.668
3-acetoxy-5-
H
methyl




methylphenyl





1.1.669
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






methylphenyl}





1.1.670
3-methylsulfanyl-5-
H
methyl




methylphenyl





1.1.671
3,5-diethylphenyl
H
methyl



1.1.672
3-propyl-5-
H
methyl




ethylphenyl





1.1.673
3-isopropyl-5-
H
methyl




ethylphenyl





1.1.674
3-n-butyl-5-
H
methyl




ethylphenyl





1.1.675
3-isobutyl-5-
H
methyl




ethylphenyl





1.1.676
3-tert-butyl-5-
H
methyl




ethylphenyl





1.1.677
3-cyclopropyl-5-
H
methyl




ethylphenyl





1.1.678
3-vinyl-5-ethylphenyl
H
methyl



1.1.679
3-ethynyl-5-
H
methyl




ethylphenyl





1.1.680
3-cyano-5-
H
methyl




ethylphenyl





1.1.681
3-trifluoromethyl-5-
H
methyl




ethylphenyl





1.1.682
3-(hydroxycarbonyl)-
H
methyl




5-ethylphenyl





1.1.683
3-(methoxycarbonyl)-
H
methyl




5-ethylphenyl





1.1.684
3-hydroxymethyl-5-
H
methyl




ethylphenyl





1.1.685
3-carbamoyl-5-
H
methyl




ethylphenyl





1.1.686
3-hydroxy-5-
H
methyl




ethylphenyl





1.1.687
3-methoxy-5-
H
methyl




ethylphenyl





1.1.688
3-ethoxy-5-
H
methyl




ethylphenyl





1.1.689
3-n-propoxy-5-
H
methyl




ethylphenyl





1.1.690
3-n-butoxy-5-
H
methyl




ethylphenyl





1.1.691
3-isobutoxy-5-
H
methyl




ethylphenyl





1.1.692
3-tert-butoxy-5-
H
methyl




ethylphenyl





1.1.693
3-difluoromethoxy-5-
H
methyl




ethylphenyl





1.1.694
3-trifluoromethoxy-5-
H
methyl




ethylphenyl





1.1.695
3-(2,2,2-
H
methyl




trifluoroethoxy)-5-






ethylphenyl





1.1.696
3-(2-chloroethoxy)-5-
H
methyl




ethylphenyl





1.1.697
3-(2-hydroxyethoxy)-
H
methyl




5-ethylphenyl





1.1.698
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






ethylphenyl





1.1.699
3-nitro-5-ethylphenyl
H
methyl



1.1.700
3-acetoxy-5-
H
methyl




ethylphenyl





1.1.701
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






ethylphenyl}





1.1.702
3-methylsulfanyl-5-
H
methyl




ethylphenyl





1.1.703
3,5-dipropylphenyl
H
methyl



1.1.704
3-isopropyl-5-
H
methyl




propylphenyl





1.1.705
3-n-butyl-5-
H
methyl




propylphenyl





1.1.706
3-isobutyl-5-
H
methyl




propylphenyl





1.1.707
3-tert-butyl-5-
H
methyl




propylphenyl





1.1.708
3-cyclopropyl-5-
H
methyl




propylphenyl





1.1.709
3-viny1-5-
H
methyl




propylphenyl





1.1.710
3-ethynyl-5-
H
methyl




propylphenyl





1.1.711
3-cyano-5-
H
methyl




propylphenyl





1.1.712
3-trifluoromethyl-5-
H
methyl




propylphenyl





1.1.713
3-(hydroxycarbonyl)-
H
methyl




5-propylphenyl





1.1.714
3-(methoxycarbonyl)-
H
methyl




5-propylphenyl





1.1.715
3-hydroxymethyl-5-
H
methyl




propylphenyl





1.1.716
3-carbamoyl-5-
H
methyl




propylphenyl





1.1.717
3-hydroxy-5-
H
methyl




propylphenyl





1.1.718
3-methoxy-5-
H
methyl




propylphenyl





1.1.719
3-ethoxy-5-
H
methyl




propylphenyl





1.1.720
3-n-propoxy-5-
H
methyl




propylphenyl





1.1.721
3-n-butoxy-5-
H
methyl




propylphenyl





1.1.722
3-isobutoxy-5-
H
methyl




propylphenyl





1.1.723
3-tert-butoxy-5-
H
methyl




propylphenyl





1.1.724
3-difluoromethoxy-5-
H
methyl




propylphenyl





1.1.725
3-trifluoromethoxy-5-
H
methyl




ethylphenyl





1.1.726
3-(2,2,2-
H
methyl




trifluoroethoxy)-5-






propylphenyl





1.1.727
3-(2-chloroethoxy)-5-
H
methyl




propylphenyl





1.1.728
3-(2-hydroxyethoxy)-
H
methyl




5-propylphenyl





1.1.729
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






propylphenyl





1.1.730
3-nitro-5-
H
methyl




propylphenyl





1.1.731
3-acetoxy-5-
H
methyl




propylphenyl





1.1.732
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






propylphenyl}





1.1.733
3-methylsulfanyl-5-
H
methyl




propylphenyl





1.1.734
3,5-diisopropylphenyl
H
methyl



1.1.735
3-n-butyl-5-
H
methyl




isopropylphenyl





1.1.736
3-isobutyl-5-
H
methyl




isopropylphenyl





1.1.737
3-tert-butyl-5-
H
methyl




isopropylphenyl





1.1.738
3-cyclopropyl-5-
H
methyl




isopropylphenyl





1.1.739
3-vinyl-5-
H
methyl




isopropylphenyl





1.1.740
3-thynyl-5-
H
methyl




isopreopylphenyl





1.1.741
3-cyano-5-
H
methyl




isopropylphenyl





1.1.742
3-trifluoromethyl-5-
H
methyl




isopropylphenyl





1.1.743
3-(hydroxycarbonyl)-
H
methyl




5-isopropylphenyl





1.1.744
3-(methoxycarbonyl)-
H
methyl




5-isopropylphenyl





1.1.745
3-hydroxymethyl-5-
H
methyl




isopropylphenyl





1.1.746
3-carbamoyl-5-
H
methyl




isopropylphenyl





1.1.747
3-hydroxy-5-
H
methyl




isopropylphenyl





1.1.748
3-methoxy-5-
H
methyl




isopropylphenyl





1.1.749
3-thoxy-5-
H
methyl




isopropylphenyl





1.1.750
3-n-propoxy-5-
H
methyl




isopropylphenyl





1.1.751
3-n-butoxy-5-
H
methyl




isopropylphenyl





1.1.752
3-isobutoxy-5-
H
methyl




isopropylphenyl





1.1.753
3-tert-butoxy-5-
H
methyl




isopropylphenyl





1.1.754
3-difluoromethoxy-5-
H
methyl




isopropylphenyl





1.1.755
3-trifluoromethoxy-5-
H
methyl




isopropylphenyl





1.1.756
3-(2,2,2-
H
methyl




trifluoroethoxy)-5-






isopropylphenyl





1.1.757
3-(2-chloroethoxy)-5-
H
methyl




isopropylphenyl





1.1.758
3-(2-hydroxyethoxy)-
H
methyl




5-propylphenyl





1.1.759
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






isopropylphenyl





1.1.760
3-nitro-5-
H
methyl




isopropylphenyl





1.1.761
3-acetoxy-5-
H
methyl




isopropylphenyl





1.1.762
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






isopropylphenyl}





1.1.763
3-methylsulfanyl-5-
H
methyl




isopropylphenyl





1.1.764
3,5-dibutylphenyl
H
methyl



1.1.765
3-isobutyl-5-
H
methyl




butylphenyl





1.1.766
3-tert-butyl-5-
H
methyl




butylphenyl





1.1.767
3-cyclopropyl-5-
H
methyl




butylphenyl





1.1.768
3-vinyl-5-butylphenyl
H
methyl



1.1.769
3-ethynyl-5-
H
methyl




butylphenyl





1.1.770
3-cyano-5-
H
methyl




butylphenyl





1.1.771
3-trifluoromethyl-5-
H
methyl




butylphenyl





1.1.772
3-(hydroxycarbonyl)-
H
methyl




5-butylphenyl





1.1.773
3-(methoxycarbonyl)-
H
methyl




5-butylphenyl





1.1.774
3-hydroxymethyl-5-
H
methyl




butylphenyl





1.1.775
3-carbamoyl-5-
H
methyl




butylphenyl





1.1.776
3-hydroxy-5-
H
methyl




butylphenyl





1.1.777
3-methoxy-5-
H
methyl




butylphenyl





1.1.778
3-ethoxy-5-
H
methyl




butylphenyl





1.1.779
3-n-propoxy-5-
H
methyl




butylphenyl





1.1.780
3-n-butoxy-5-
H
methyl




butylphenyl





1.1.781
3-isobutoxy-5-
H
methyl




butylphenyl





1.1.782
3-tert-butoxy-5-
H
methyl




butylphenyl





1.1.783
3-difluoromethoxy-5-
H
methyl




butylphenyl





1.1.784
3-trifluoromethoxy-5-
H
methyl




butylphenyl





1.1.785
3-(2,2,2-
H
methyl




trifluoroethoxy)-5-






butylphenyl





1.1.786
3-(2-chloroethoxy)-5-
H
methyl




butylphenyl





1.1.787
3-(2-hydroxyethoxy)-
H
methyl




5-butylphenyl





1.1.788
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






butylphenyl





1.1.789
3-nitro-5-butylphenyl
H
methyl



1.1.790
3-acetoxy-5-
H
methyl




butylphenyl





1.1.791
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






butylphenyl}





1.1.792
3-methylsulfanyl-5-
H
methyl




butylphenyl





1.1.793
3,5-diisobutylphenyl
H
methyl



1.1.794
3-tert-butyl-5-
H
methyl




isobutylphenyl





1.1.795
3-cyclopropyl-5-
H
methyl




isobutylphenyl





1.1.796
3-vinyl-5-
H
methyl




isobutylphenyl





1.1.797
3-ethynyl-5-
H
methyl




isobutylphenyl





1.1.798
3-cyano-5-
H
methyl




isobutylphenyl





1.1.799
3-trifluoromethyl-5-
H
methyl




isobutylphenyl





1.1.800
3-(hydroxycarbonyl)-
H
methyl




5-isobutylphenyl





1.1.801
3-(methoxycarbonyl)-
H
methyl




5-isobutylphenyl





1.1.802
3-hydroxymethyl-5-
H
methyl




isobutylphenyl





1.1.803
3-carbamoyl-5-
H
methyl




isobutylphenyl





1.1.804
3-hydroxy-5-
H
methyl




isobutylphenyl





1.1.805
3-methoxy-5-
H
methyl




isobutylphenyl





1.1.806
3-ethoxy-5-
H
methyl




isobutylphenyl





1.1.807
3-n-propoxy-5-
H
methyl




isobutylphenyl





1.1.808
3-n-butoxy-5-
H
methyl




isobutylphenyl





1.1.809
3-isobutoxy-5-
H
methyl




isobutylphenyl





1.1.810
3-tert-butoxy-5-
H
methyl




isobutylphenyl





1.1.811
3-difluoromethoxy-5-
H
methyl




isobutylphenyl





1.1.812
3-trifluoromethoxy-5-
H
methyl




isobutylphenyl





1.1.813
3-(2,2,2-
H
methyl




trifluoroethoxy)-5-






isobutylphenyl





1.1.814
3-(2-chloroethoxy)-5-
H
methyl




isobutylphenyl





1.1.815
3-(2-hydroxyethoxy)-
H
methyl




5-isobutylphenyl





1.1.816
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






isobutylphenyl





1.1.817
3-nitro-5-
H
methyl




isobutylphenyl





1.1.818
3-acetoxy-5-
H
methyl




isobutylphenyl





1.1.819
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






isobutylphenyl}





1.1.820
3-methylsulfanyl-5-
H
methyl




isobutylphenyl





1.1.821
3,5-di(tert-
H
methyl
[DMSO] 1.30 (s, 9H); 1.56 (s, 3H);



butylphenyl


3.41 (d, 1H); 3.82 (d, 1H); 7.48 (s,






2H); 7.5 (s, 1H).


1.1.822
3-cyclopropyl-5-tert-
H
methyl




butylphenyl





1.1.823
3-vinyl-5-tert-
H
methyl




butylphenyl





1.1.824
3-ethynyl-5-tert-
H
methyl




butylphenyl





1.1.825
3-cyano-5-tert-
H
methyl




butylphenyl





1.1.826
3-trifluoromethyl-5-
H
methyl




tert-butylphenyl





1.1.827
3-(hydroxycarbonyl)-
H
methyl




5-tert-butylphenyl





1.1.828
3-(methoxycarbonyl)-
H
methyl




5-tert-butylphenyl





1.1.829
3-hydroxymethyl-5-
H
methyl




tert-butylphenyl





1.1.830
3-carbamoyl-5-tert-
H
methyl




butylphenyl





1.1.831
3-hydroxy-5-tert-
H
methyl




butylphenyl





1.1.832
3-methoxy-5-tert-
H
methyl




butylphenyl





1.1.833
3-ethoxy-5-tert-
H
methyl




butylphenyl





1.1.834
3-n-propoxy-5-tert-
H
methyl




butylphenyl





1.1.835
3-n-butoxy-5-tert-
H
methyl




butylphenyl





1.1.836
3-isobutoxy-5-tert-
H
methyl




butylphenyl





1.1.837
3-tert-butoxy-5-tert-
H
methyl




butylphenyl





1.1.838
3-difluoromethoxy-5-
H
methyl




tert-butylphenyl





1.1.839
3-trifluoromethoxy-5-
H
methyl




tert-butylphenyl





1.1.840
3-(2,2,2-
H
methyl




trifluoroethoxy)-5-






tert-butylphenyl





1.1.841
3-(2-chloroethoxy)-5-
H
methyl




tert-butylphenyl





1.1.842
3-(2-hydroxyethoxy)-
H
methyl




5-tert-butylphenyl





1.1.843
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-tert-






butylphenyl





1.1.844
3-nitro-5-tert-
H
methyl




butylphenyl





1.1.845
3-acetoxy-5-tert-
H
methyl




butylphenyl





1.1.846
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






tert-butylphenyl}





1.1.847
3-methylsulfanyl-5-
H
methyl




tert-butylphenyl





1.1.848
3-tert-butyl-5-
H
methyl




cyclopropylphenyl





1.1.849
3,5-dicyclopropyl-
H
methyl




phenyl





1.1.850
3-vinyl-5-
H
methyl




cyclopropylphenyl





1.1.851
3-ethynyl-5-
H
methyl




cyclopropylphenyl





1.1.852
3-cyano-5-
H
methyl




cyclopropylphenyl





1.1.853
3-trifluoromethyl-5-
H
methyl




cyclopropylphenyl





1.1.854
3-(hydroxycarbonyl)-
H
methyl




5-cyclopropylphenyl





1.1.855
3-(methoxycarbonyl)-
H
methyl




5-cyclopropylphenyl





1.1.856
3-hydroxymethyl-5-
H
methyl




cyclopropylphenyl





1.1.857
3-carbamoyl-5-
H
methyl




cyclopropylphenyl





1.1.858
3-hydroxy-5-
H
methyl




cyclopropylphenyl





1.1.859
3-methoxy-5-
H
methyl




cyclopropylphenyl





1.1.860
3-ethoxy-5-
H
methyl




cyclopropylphenyl





1.1.861
3-n-propoxy-5-
H
methyl




cyclopropylphenyl





1.1.862
3-n-butoxy-5-
H
methyl




cyclopropylphenyl





1.1.863
3-isobutoxy-5-
H
methyl




cyclopropylphenyl





1.1.864
3-tert-butoxy-5-
H
methyl




cyclopropylphenyl





1.1.865
3-difluoromethoxy-5-
H
methyl




cyclopropylphenyl





1.1.866
3-trifluoromethoxy-5-
H
methyl




cyclopropylphenyl





1.1.867
3-(2,2,2-
H
methyl




trifluoroethoxy)-5-






cyclopropylphenyl





1.1.868
3-(2-chloroethoxy)-5-
H
methyl




cyclopropylphenyl





1.1.869
3-(2-hydroxyethoxy)-
H
methyl




5-cyclopropylphenyl





1.1.870
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






cyclopropylphenyl





1.1.871
3-nitro-5-
H
methyl




cyclopropylphenyl





1.1.872
3-acetoxy-5-
H
methyl




cyclopropylphenyl





1.1.873
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






cyclopropylphenyl}





1.1.874
3-methylsulfanyl-5-
H
methyl




cyclopropylphenyl





1.1.875
3,5-divinylphenyl
H
methyl



1.1.876
3-ethynyl-5-
H
methyl




vinylphenyl





1.1.877
3-cyano-5-
H
methyl




vinylphenyl





1.1.878
3-trifluoromethyl-5-
H
methyl




vinylphenyl





1.1.879
3-(hydroxycarbonyl)-
H
methyl




5-vinylphenyl





1.1.880
3-(methoxycarbonyl)-
H
methyl




5-vinylphenyl





1.1.881
3-hydroxymethyl-5-
H
methyl




vinylphenyl





1.1.882
3-carbamoyl-5-
H
methyl




vinylphenyl





1.1.883
3-hydroxy-5-
H
methyl




vinylphenyl





1.1.884
3-methoxy-5-
H
methyl




vinylphenyl





1.1.885
3-ethoxy-5-
H
methyl




vinylphenyl





1.1.886
3-n-propoxy-5-
H
methyl




vinylphenyl





1.1.887
3-n-butoxy-5-
H
methyl




vinylphenyl





1.1.888
3-isobutoxy-5-
H
methyl




vinylphenyl





1.1.889
3-tert-butoxy-5-
H
methyl




vinylphenyl





1.1.890
3-difluoromethoxy-5-
H
methyl




vinylphenyl





1.1.891
3-trifluoromethoxy-5-
H
methyl




vinylphenyl





1.1.892
3-(2,2,2-
H
methyl




trifluoroethoxy)-5-






vinylphenyl





1.1.893
3-(2-chloroethoxy)-5-
H
methyl




vinylphenyl





1.1.894
3-(2-hydroxyethoxy)-
H
methyl




5-vinylphenyl





1.1.895
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






vinylphenyl





1.1.896
3-nitro-5-vinylphenyl
H
methyl



1.1.897
3-acetoxy-5-
H
methyl




vinylphenyl





1.1.898
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






vinylphenyl}





1.1.899
3-methylsulfanyl-5-
H
methyl




vinylphenyl





1.1.900
3,5-diethynylphenyl
H
methyl



1.1.901
3-cyano-5-
H
methyl




ethynylphenyl





1.1.902
3-trifluoromethyl-5-
H
methyl




ethynylphenyl





1.1.903
3-(hydroxycarbonyl)-
H
methyl




5-ethynylphenyl





1.1.904
3-(methoxycarbonyl)-
H
methyl




5-ethynylphenyl





1.1.905
3-hydroxymethyl-5-
H
methyl




ethynylphenyl





1.1.906
3-carbamoyl-5-
H
methyl




ethynylphenyl





1.1.907
3-hydroxy-5-
H
methyl




ethynylphenyl





1.1.908
3-methoxy-5-
H
methyl




ethynylphenyl





1.1.909
3-ethoxy-5-
H
methyl




ethynylphenyl





1.1.910
3-n-propoxy-5-
H
methyl




ethynylphenyl





1.1.911
3-n-butoxy-5-
H
methyl




ethynylphenyl





1.1.912
3-isobutoxy-5-
H
methyl




ethynylphenyl





1.1.913
3-tert-butoxy-5-
H
methyl




ethynylphenyl





1.1.914
3-difluoromethoxy-5-
H
methyl




ethynylphenyl





1.1.915
3-trifluoromethoxy-5-
H
methyl




ethynylphenyl





1.1.916
3-(2,2,2-
H
methyl




trifluoroethoxy)-5-






ethynylphenyl





1.1.917
3-(2-chloroethoxy)-5-
H
methyl




ethynylphenyl





1.1.918
3-(2-hydroxyethoxy)-
H
methyl




5-ethynylphenyl





1.1.919
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






ethynylphenyl





1.1.920
3-nitro-5-
H
methyl




ethynylphenyl





1.1.921
3-acetoxy-5-
H
methyl




ethynylphenyl





1.1.922
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






ethynylphenyl}





1.1.923
3-methylsulfanyl-5-
H
methyl




ethynylphenyl





1.1.924
3,5-dicyanophenyl
H
methyl
[CDCl3] 1.80 (s, 3H); 3.28 (d, 1H);






3.90 (d, 1H); 7.98 (s, 1H); 8.15 (s,






2H).


1.1.925
3-trifluoromethyl-5-
H
methyl
[CDCl3] 1.81 (s, 3H); 3.30 (d, 1H);



cyanophenyl


3.91 (d, 1H); 7.92 (s, 1H); 8.11 (d,






2H).


1.1.926
3-(hydroxycarbonyl)-
H
methyl




5-cyanophenyl





1.1.927
3-(methoxycarbonyl)-
H
methyl




5-cyanophenyl





1.1.928
3-hydroxymethyl-5-
H
methyl




cyanophenyl





1.1.929
3-carbamoyl-5-
H
methyl




cyanophenyl





1.1.930
3-hydroxy -5-
H
methyl




cyanophenyl





1.1.931
3-methoxy-5-
H
methyl




cyanophenyl





1.1.932
3-ethoxy-5-
H
methyl




cyanophenyl





1.1.933
3-n-propoxy-5-
H
methyl




cyanophenyl





1.1.934
3-n-butoxy-5-
H
methyl




cyanophenyl





1.1.935
3-isobutoxy-5-
H
methyl




cyanophenyl





1.1.936
3-tert-butoxy-5-
H
methyl




cyanophenyl





1.1.937
3-difluoromethoxy-5-
H
methyl




cyanophenyl





1.1.938
3-trifluoromethoxy-5-
H
methyl




cyanophenyl





1.1.939
3-(2,2,2-
H
methyl




trifluoroethoxy)-5-






cyanophenyl





1.1.940
3-(2-chloroethoxy)-5-
H
methyl




cyanophenyl





1.1.941
3-(2-hydroxyethoxy)-
H
methyl




5-cyanophenyl





1.1.942
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






cyanophenyl





1.1.943
3-nitro-5-
H
methyl




cyanophenyl





1.1.944
3-acetoxy-5-
H
methyl




cyanophenyl





1.1.945
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






cyanophenyl}





1.1.946
3-methylsulfanyl-5-
H
methyl




cyanophenyl





1.1.947
3,5-
H
methyl
[CDCl3] 1.81 (s, 3H); 3.35 (d, 1H);



di(trifluoromethyl)-


3.95 (d, 1H); 7.92 (s, 1H); 8.08 (s,



phenyl


2H).


1.1.948
3-(hydroxycarbonyl)-
H
methyl




5-trifluoromethyl-






phenyl





1.1.949
3-(methoxycarbonyl)-
H
methyl




5-trifluoromethyl-






phenyl





1.1.950
3-hydroxymethyl-5-
H
methyl




trifluoromethylphenyl





1.1.951
3-carbamoyl-5-
H
methyl




trifluoromethylphenyl





1.1.952
3-hydroxy-5-
H
methyl




trifluoromethylphenyl





1.1.953
3-methoxy-5-
H
methyl




trifluoromethylphenyl





1.1.954
3-ethoxy-5-
H
methyl




trifluoromethylphenyl





1.1.955
3-n-propoxy-5-
H
methyl




trifluoromethylphenyl





1.1.956
3-n-butoxy-5-
H
methyl




trifluoromethylphenyl





1.1.957
3-isobutoxy-5-
H
methyl




trifluoromethylphenyl





1.1.958
3-tert-butoxy-5-
H
methyl




trifluoromethylphenyl





1.1.959
3-difluoromethoxy-5-
H
methyl




trifluoromethylphenyl





1.1.960
3-trifluoromethoxy-5-
H
methyl




trifluoromethylphenyl





1.1.961
3-(2,2,2-trifluoro-
H
methyl




ethoxy)-5-trifluoro-






methylphenyl





1.1.962
3-(2-chloroethoxy)-5-
H
methyl




trifluoromethyl-






phenyl





1.1.963
3-(2-hydroxyethoxy)-
H
methyl




5-trifluoromethyl-






phenyl





1.1.964
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






trifluoromethylphenyl





1.1.965
3-nitro-5-
H
methyl




trifluoromethylphenyl





1.1.966
3-acetoxy-5-
H
methyl




trifluoromethylphenyl





1.1.967
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






trifluoromethyl-






phenyl}





1.1.968
3-methylsulfanyl-5-
H
methyl




trifluoromethylphenyl





1.1.969
3,5-bis(hydroxy-
H
methyl




carbonyl)phenyl





1.1.970
3-(methoxycarbonyl)-
H
methyl




5-(hydroxycarbonyl)-






phenyl





1.1.971
3-hydroxymethyl-5-
H
methyl




(hydroxycarbonyl)-






phenyl





1.1.972
3-carbamoyl-5-
H
methyl




(hydroxycarbonyl)-






phenyl





1.1.973
3-hydroxy-5-
H
methyl




(hydroxycarbonyl)-






phenyl





1.1.974
3-methoxy-5-
H
methyl




(hydroxycarbonyl)-






phenyl





1.1.975
3-ethoxy-5-
H
methyl




(hydroxycarbonyl)-






phenyl





1.1.976
3-n-propoxy-5-
H
methyl




(hydroxycarbonyl)-






phenyl





1.1.977
3-n-butoxy-5-
H
methyl




(hydroxycarbonyl)-






phenyl





1.1.978
3-isobutoxy-5-
H
methyl




(hydroxycarbonyl)-






phenyl





1.1.979
3-tert-butoxy-5-
H
methyl




(hydroxycarbonyl)-






phenyl





1.1.980
3-difluoromethoxy-5-
H
methyl




(hydroxycarbonyl)-






phenyl





1.1.981
3-trifluoromethoxy-5-
H
methyl




(hydroxycarbonyl)-






phenyl





1.1.982
3-(2,2,2-trifluoro-
H
methyl




ethoxy)-5-(hydroxy-






carbonyl)phenyl





1.1.983
3-(2-chloroethoxy)-5-
H
methyl




(hydroxycarbonyl)-






phenyl





1.1.984
3-(2-hydroxyethoxy)-
H
methyl




5-(hydroxycarbonyl)-






phenyl





1.1.985
3-[(tert-butoxy-
H
methyl




(hydroxycarbonyl)-






phenyl





1.1.986
3-nitro-5-
H
methyl




(hydroxycarbonyl)-






phenyl





1.1.987
3-acetoxy-5-
H
methyl




(hydroxycarbonyl)-






phenyl





1.1.988
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






(hydroxycarbonyl)-






phenyl)





1.1.989
3-methylsulfanyl-5-
H
methyl




(hydroxycarbonyl)-






phenyl





1.1.990
3,5-di(methoxy-
H
methyl




carbonyl)phenyl





1.1.991
3-hydroxymethyl-5-
H
methyl




(methoxycarbonyl)-






phenyl





1.1.992
3-carbamoyl-5-
H
methyl




(methoxycarbonyl)-






phenyl





1.1.993
3-hydroxy-5-
H
methyl




(methoxycarbonyl)-






phenyl





1.1.994
3-methoxy-5-
H
methyl




(methoxycarbonyl)-






phenyl





1.1.995
3-ethoxy-5-
H
methyl




(methoxycarbonyl)-






phenyl





1.1.996
3-n-propoxy-5-
H
methyl




(methoxycarbonyl)-






phenyl





1.1.997
3-n-butoxy-5-
H
methyl




(methoxycarbonyl)-






phenyl





1.1.998
3-isobutoxy-5-
H
methyl




(methoxycarbonyl)-






phenyl





1.1.999
3-tert-butoxy-5-
H
methyl




(methoxycarbonyl)-






phenyl





1.1.1000
3-difluoromethoxy-5-
H
methyl




(methoxycarbonyl)-






phenyl





1.1.1001
3-trifluoromethoxy-5-
H
methyl




(methoxycarbonyl)-






phenyl





1.1.1002
3-(2,2,2-trifluoro-
H
methyl




ethoxy)-5-(methoxy-






carbonyl)phenyl





1.1.1003
3-(2-chloroethoxy)-5-
H
methyl




(methoxycarbonyl)-






phenyl





1.1.1004
3-(2-hydroxyethoxy)-
H
methyl




5-(methoxycarbonyl)-






phenyl





1.1.1005
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






methoxycarbonyl)-






phenyl





1.1.1006
3-nitro-5-(methoxy-
H
methyl




carbonyl)phenyl





1.1.1007
3-acetoxy-5-
H
methyl




(methoxycarbonyl)-






phenyl





1.1.1008
(3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






(methoxycarbonyl)-






phenyl)





1.1.1009
3-methylsulfanyl-5-
H
methyl




(methoxycarbonyl)-






phenyl





1.1.1010
3,5-di(hydroxy-
H
methyl




methyl)phenyl





1.1.1011
3-carbamoyl-5-
H
methyl




hydroxymethylphenyl





1.1.1012
3-hydroxy-5-
H
methyl




hydroxymethylphenyl





1.1.1013
3-methoxy-5-
H
methyl




hydroxymethylphenyl





1.1.1014
3-ethoxy-5-
H
methyl




hydroxymethylphenyl





1.1.1015
3-n-propoxy-5-
H
methyl




hydroxymethylphenyl





1.1.1016
3-n-butoxy-5-
H
methyl




hydroxymethylphenyl





1.1.1017
3-isobutoxy-5-
H
methyl




hydroxymethylphenyl





1.1.1018
3-tert-butoxy-5-
H
methyl




hydroxymethylphenyl





1.1.1019
3-difluoromethoxy-5-
H
methyl




hydroxymethylphenyl





1.1.1020
3-trifluoromethoxy-5-
H
methyl




hydroxymethylphenyl





1.1.1021
3-(2,2,2-
H
methyl




trifluoroethoxy)-5-






hydroxymethylphenyl





1.1.1022
3-(2-chloroethoxy)-5-
H
methyl




hydroxymethylphenyl





1.1.1023
3-(2-hydroxyethoxy)-
H
methyl




5-hydroxymethyl-






phenyl





1.1.1024
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






hydroxymethylphenyl





1.1.1025
3-nitro-5-
H
methyl




hydroxymethylphenyl





1.1.1026
3-acetoxy-5-
H
methyl




hydroxymethylphenyl





1.1.1027
(3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






hydroxymethyl-






phenyl}





1.1.1028
3-methylsulfanyl-5-
H
methyl




hydroxymethylphenyl





1.1.1029
3,5-dicarbamoyl-5-
H
methyl




carbamoylphenyl





1.1.1030
3-hydroxy-5-
H
methyl




carbamoylphenyl





1.1.1031
3-methoxy-5-
H
methyl




carbamoylphenyl





1.1.1032
3-ethoxy-5-
H
methyl




carbamoylphenyl





1.1.1033
3-n-propoxy-5-
H
methyl




carbamoylphenyl





1.1.1034
3-n-butoxy-5-
H
methyl




carbamoylphenyl





1.1.1035
3-isobutoxy-5-
H
methyl




arbamoylphenyl





1.1.1036
3-tert-butoxy-5-
H
methyl




carbamoylphenyl





1.1.1037
3-difluoromethoxy-5-
H
methyl




carbamoylphenyl





1.1.1038
3-trifluoromethoxy-5-
H
methyl




carbamoylphenyl





1.1.1039
3-(2,2,2-
H
methyl




trifluoroethoxy)-5-






carbamoylphenyl





1.1.1040
3-(2-chloroethoxy)-5-
H
methyl




carbamoylphenyl





1.1.1041
3-(2-hydroxyethoxy)-
H
methyl




5-carbamoylphenyl





1.1.1042
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






carbamoylphenyl





1.1.1043
3-nitro-5-
H
methyl




carbamoylphenyl





1.1.1044
3-acetoxy-5-
H
methyl




carbamoylphenyl





1.1.1045
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






carbamoylphenyl}





1.1.1046
3-methylsulfanyl-5-
H
methyl




carbamoylphenyl





1.1.1047
3,5-dihydroxyphenyl
H
methyl



1.1.1048
3-methoxy-5-
H
methyl




hydroxyphenyl





1.1.1049
3-ethoxy-5-
H
methyl




hydroxyphenyl





1.1.1050
3-n-propoxy-5-
H
methyl




hydroxyphenyl





1.1.1051
3-n-butoxy-5-
H
methyl




hydroxyphenyl





1.1.1052
3-isobutoxy-5-
H
methyl




hydroxyphenyl





1.1.1053
3-tert-butoxy-5-
H
methyl




hydroxyphenyl





1.1.1054
3-difluoromethoxy-5-
H
methyl




hydroxyphenyl





1.1.1055
3-trifluoromethoxy-5-
H
methyl




hydroxyphenyl





1.1.1056
3-(2,2,2-
H
methyl




trifluoroethoxy)-5-






hydroxyphenyl





1.1.1057
3-(2-chloroethoxy)-5-
H
methyl




hydroxyphenyl





1.1.1058
3-(2-hydroxyethoxy)-
H
methyl




5-hydroxyphenyl





1.1.1059
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






hydroxyphenyl





1.1.1060
3-nitro-5-
H
methyl




hydroxyphenyl





1.1.1061
3-acetoxy-5-
H
methyl




hydroxyphenyl





1.1.1062
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






hydroxyphenyl}





1.1.1063
3-methylsulfanyl-5-
H
methyl




hydroxyphenyl





1.1.1064
3,5-dimethoxyphenyl
H
methyl



1.1.1065
3-ethoxy-5-
H
methyl




methoxyphenyl





1.1.1066
3-n-propoxy-5-
H
methyl




methoxyphenyl





1.1.1067
3-n-butoxy-5-
H
methyl




methoxyphenyl





1.1.1068
3-isobutoxy-5-
H
methyl




methoxyphenyl





1.1.1069
3-tert-butoxy-5-
H
methyl




methoxyphenyl





1.1.1070
3-difluoromethoxy-5-
H
methyl




methoxyphenyl





1.1.1071
3-trifluoromethoxy-5-
H
methyl




methoxyphenyl





1.1.1072
3-(2,2,2-
H
methyl




trifluoroethoxy)-5-






methoxyphenyl





1.1.1073
3-(2-chloroethoxy)-5-
H
methyl




methoxyphenyl





1.1.1074
3-(2-hydroxyethoxy)-
H
methyl




5-methoxyphenyl





1.1.1075
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






methoxyphenyl





1.1.1076
3-nitro-5-
H
methyl




methoxyphenyl





1.1.1077
3-acetoxy-5-
H
methyl




methoxyphenyl





1.1.1078
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






methoxyphenyl}





1.1.1079
3-methylsulfanyl-5-
H
methyl




methoxyphenyl





1.1.1080
3,5-diethoxyphenyl
H
methyl



1.1.1081
3-n-propoxy-5-
H
methyl




ethoxyphenyl





1.1.1082
3-n-butoxy-5-
H
methyl




ethoxyphenyl





1.1.1083
3-isobutoxy-5-
H
methyl




ethoxyphenyl





1.1.1084
3-tert-butoxy-5-
H
methyl




ethoxyphenyl





1.1.1085
3-difluoromethoxy-5-
H
methyl




ethoxyphenyl





1.1.1086
3-trifluoromethoxy-5-
H
methyl




ethoxyphenyl





1.1.1087
3-(2,2,2-
H
methyl




trifluoroethoxy)-5-






ethoxyphenyl





1.1.1088
3-(2-chloroethoxy)-5-
H
methyl




ethoxyphenyl





1.1.1089
3-(2-hydroxyethoxy)-
H
methyl




5-ethoxyphenyl





1.1.1090
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






ethoxyphenyl





1.1.1091
3-nitro-5-
H
methyl




ethoxyphenyl





1.1.1092
3-acetoxy-5-
H
methyl




ethoxyphenyl





1.1.1093
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






ethoxyphenyl}





1.1.1094
3-methylsulfanyl-5-
H
methyl




ethoxyphenyl





1.1.1095
3,5-dipropoxyphenyl
H
methyl



1.1.1096
3-n-butoxy-5-
H
methyl




propoxyphenyl





1.1.1097
3-isobutoxy-5-
H
methyl




propoxyphenyl





1.1.1098
3-tert-butoxy-5-
H
methyl




propoxyphenyl





1.1.1099
3-difluoromethoxy-5-
H
methyl




propoxyphenyl





1.1.1100
3-trifluoromethoxy-5-
H
methyl




propoxyphenyl





1.1.1101
3-(2,2,2-
H
methyl




trifluoroethoxy)-5-






propoxyphenyl





1.1.1102
3-(2-chloroethoxy)-5-
H
methyl




propoxyphenyl





1.1.1103
3-(2-hydroxyethoxy)-
H
methyl




5-propoxyphenyl





1.1.1104
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






propoxyphenyl





1.1.1105
3-nitro-5-
H
methyl




propoxyphenyl





1.1.1106
3-acetoxy-5-
H
methyl




propoxyphenyl





1.1.1107
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






propoxyphenyl}





1.1.1108
3-methylsulfanyl-5-
H
methyl




propoxyphenyl





1.1.1109
3,5-
H
methyl




di(isopropoxy)phenyl





1.1.1110
3-n-butoxy-5-
H
methyl




isopropoxyphenyl





1.1.1111
3-isobutoxy-5-
H
methyl




isopropoxyphenyl





1.1.1112
3-tert-butoxy-5-
H
methyl




isopropoxyphenyl





1.1.1113
3-difluoromethoxy-5-
H
methyl




isopropoxyphenyl





1.1.1114
3-trifluoromethoxy-5-
H
methyl




isopropoxyphenyl





1.1.1115
3-(2,2,2-
H
methyl




trifluoroethoxy)-5-






isopropoxyphenyl





1.1.1116
3-(2-chloroethoxy)-5-
H
methyl




isopropoxyphenyl





1.1.1117
3-(2-hydroxyethoxy)-
H
methyl




5-isopropoxyphenyl





1.1.1118
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






isopropoxyphenyl





1.1.1119
3-nitro-5-
H
methyl




isopropoxyphenyl





1.1.1120
3-acetoxy-5-
H
methyl




isopropoxyphenyl





1.1.1121
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






isopropoxyphenyl}





1.1.1122
3-methylsulfanyl-5-
H
methyl




isopropoxyphenyl





1.1.1123
3,5-di(tert-butoxy)-
H
methyl




phenyl





1.1.1124
3-difluoromethoxy-5-
H
methyl




tert-butoxyphenyl





1.1.1125
3-trifluoromethoxy-5-
H
methyl




tert-butoxyphenyl





1.1.1126
3-(2,2,2-
H
methyl




trifluoroethoxy)-5-






tert-butoxyphenyl





1.1.1127
3-(2-chloroethoxy)-5-
H
methyl




tert-butoxylphenyl





1.1.1128
3-(2-hydroxyethoxy)-
H
methyl




5-tert-butoxyphenyl





1.1.1129
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-tert-






butoxyphenyl





1.1.1130
3-nitro-5-tert-
H
methyl




butoxyphenyl





1.1.1131
3-acetoxy-5-tert-
H
methyl




butoxyphenyl





1.1.1132
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






tert-butoxyphenyl}





1.1.1133
3-methylsulfanyl-5-
H
methyl




tert-butoxyphenyl





1.1.1134
3,5-di(trifluoro-
H
methyl




methoxy)phenyl





1.1.1135
3-(2,2,2-trifluoro-
H
methyl




ethoxy)-5-trifluoro-






methoxyphenyl





1.1.1136
3-(2-chloroethoxy)-5-
H
methyl




trifluoromethoxy-






phenyl





1.1.1137
3-(2-hydroxyethoxy)-
H
methyl




5-trifluoromethoxy-






phenyl





1.1.1138
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






trifluoromethoxy-






phenyl





1.1.1139
3-nitro-5-trifluoro-
H
methyl




methoxyphenyl





1.1.1140
3-acetoxy-5-tert-
H
methyl




butoxyphenyl





1.1.1141
(3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






trifluoromethoxy-






phenyl}





1.1.1142
3-methylsulfanyl-5-
H
methyl




trifluoromethoxy-






phenyl





1.1.1143
3,5-bis(difluoro-
H
methyl




methoxy)phenyl





1.1.1144
3,5-bis(difluoro-
H
ethyl




methoxy)phenyl





1.1.1145
3,5-bis(difluoro-
H
isopropyl




methoxy)phenyl





1.1.1146
3,5-bis(difluoro-
H
cyclopropyl




methoxy)phenyl





1.1.1147
3-trifluoromethoxy-5-
H
methyl




difluoromethoxy-






phenyl





1.1.1148
3-(2,2,2-trifluoro-
H
methyl




ethoxy)-5-difluoro-






methoxyphenyl





1.1.1149
3-(2-chloroethoxy)-5-






difluoromethoxy-
H
methyl




phenyl





1.1.1150
3-(2-hydroxyethoxy)-
H
methyl




5-difluoromethoxy-






phenyl





1.1.1151
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






difluoromethoxy-






phenyl





1.1.1152
3-nitro-5-difluoro-
H
methyl




methoxyphenyl





1.1.1153
3-acetoxy-5-difluoro-
H
methyl




methoxyphenyl





1.1.1154
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






difluoromethoxy-






phenyl}





1.1.1155
3-methylsulfanyl-5-
H
methyl




difluoromethoxy-






phenyl





1.1.1156
3,5-bis(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.1157
3-(2-chloroethoxy)-5-
H
methyl




(2,2,2-trifluoro-






ethoxy)phenyl





1.1.1158
3-(2-hydroxyethoxy)-
H
methyl




5-(2,2,2-trifluoro-






ethoxy)phenyl





1.1.1159
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-






(2,2,2-trifluoro-






ethoxy)phenyl





1.1.1160
3-nitro-5-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.1161
3-acetoxy-5-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.1162
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






(2,2,2-trifluoro-






ethoxy)phenyl}





1.1.1163
3-methylsulfanyl-5-
H
methyl




(2,2,2-trifluoro-






ethoxy)phenyl





1.1.1164
3,5-bis(2-
H
methyl




chloroethoxy)phenyl





1.1.1165
3-(2-hydroxyethoxy)-
H
methyl




5-(2-chloroethoxy)-






phenyl





1.1.1166
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-(2-






chloroethoxy)phenyl





1.1.1167
3-nitro-5-(2-
H
methyl




chloroethoxy)phenyl





1.1.1168
3-acetoxy-5-(2-
H
methyl




chloroethoxy)phenyl





1.1.1169
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






(2-chloroethoxy)-






phenyl}





1.1.1170
3-methylsulfanyl-5-
H
methyl




(2-chloroethoxy)-






phenyl





1.1.1171
3,5-bis(2-hydroxy-
H
methyl




ethoxy)phenyl





1.1.1172
3-[(tert-butoxy-
H
methyl




carbonyl)oxy]-5-(2-






hydroxyethoxy)-






phenyl





1.1.1173
3-nitro-5-(2-hydroxy-
H
methyl




ethoxy)phenyl






3-acetoxy-5-(2-





1.1.1174
hydroxyethoxy)-
H
methyl




phenyl





1.1.1175
3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






(2-hydroxyethoxy)-






phenyl





1.1.1176
3-methylsulfanyl-5-
H
methyl




(2-hydroxyethoxy)-






phenyl





1.1.1177
3,5-bis[(tert-butoxy-
H
methyl




carbonyl)oxy]phenyl





1.1.1178
3-nitro-5-[(tert-
H
methyl




butoxycarbonyl)-






oxy]phenyl





1.1.1179
3-acetoxy-5-[(tert-
H
methyl




butoxycarbonyl)oxy]-






phenyl





1.1.1180
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






[(tert-butoxy-






carbonyl)oxy]phenyl}





1.1.1181
3,5-
H
methyl




bis(acetoxy)phenyl





1.1.1182
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






acetoxyphenyl}





1.1.1183
3-methylsulfanyl-5-
H
methyl




acetoxyphenyl





1.1.1184
3,5-dinitrophenyl
H
methyl



1.1.1185
3-acetoxy-5-
H
methyl




nitrophenyl





1.1.1186
{3-[(tert-butoxy-
H
methyl




carbonyl)amino]-5-






nitrophenyl}





1.1.1187
3-methylsulfanyl-5-
H
methyl




nitrophenyl





1.1.1188
3,5-bis[(tert-
H
methyl




butoxycarbonyl)-






amino]phenyl





1.1.1189
3-methylsulfanyl-5-
H
methyl




[(tert-butoxy-






carbonyl)amino]phenyl





1.1.1190
3,5-
H
methyl




di(methylsulfanyl)phenyl





1.1.1191
3,4-difluorophenyl
H
methyl
[CDCl3] 1.80 (s, 3H); 3.25 (d, 1H);






3.85 (d, 1H); 7.22 (m, 1H); 7.30 (m,






1H); 7.55 (m, 1H).


1.1.1192
3,4-difluorophenyl
H
ethyl
[CDCl3] 1.09 (t, 3H); 2.12 (mc, 2H);






3.29 (d, 1H); 3.25 (d, 1H); 7.22 (m,






1H); 7.35 (m, 1H); 7.55 (m, 1H).


1.1.1193
3,4-difluorophenyl
H
isopropyl



1.1.1194
3,4-difluorophenyl
H
cyclopropyl



1.1.1195
3-chloro-4-
H
methyl
[CDCl3] 1.81 (s, 3H); 3.28 (d, 1H);



fluorophenyl


3.85 (d, 1H), 7.21 (m, 1H); 7.52 (m,






1H); 7.72 (m, 1H).


1.1.1196
3-chloro-4-
H
ethyl




fluorophenyl





1.1.1197
3-chloro-4-
H
isopropyl




fluorophenyl





1.1.1198
3-chloro-4-
H
cyclopropyl




fluorophenyl





1.1.1199
3-bromo-4-
H
methyl




fluorophenyl





1.1.1200
3-methyl-4-
H
methyl




fluorophenyl





1.1.1201
3-methy1-4-
H
ethyl




fluorophenyl





1.1.1202
3-ethyl-4-
H
methyl




fluorophenyl





1.1.1203
3-cyclopropyl-4-
H
methyl




fluorophenyl





1.1.1204
3-vinyl-4-
H
methyl




fluorophenyl





1.1.1205
3-ethynyl-4-
H
methyl




fluorophenyl





1.1.1206
3-cyano-4-
H
methyl




fluorophenyl





1.1.1207
3-methoxy-4-
H
methyl




fluorophenyl





1.1.1208
3-ethoxy-4-
H
methyl




fluorophenyl





1.1.1209
3-trifluoromethoxy-4-
H
methyl




fluorophenyl





1.1.1210
3-nitro-4-fluorophenyl
H
methyl



1.1.1211
3-fluoro-4-
H
methyl
[CDCl3] 1.71 (s, 3H); 3.25 (d, 1H);



chlorophenyl


3.82 (d, 1H); 7.35 (m, 1H); 7.48 (m,






1H).


1.1.1212
3,4-dichlorophenyl
H
methyl
[CDCl3] 1.8 (s, 3H); 3.25 (d, 1H);






3.83 (d, 1H); 7.5 (s, 2H); 7.72 (s,






1H).


1.1.1213
3-bromo-4-
H
methyl




chlorophenyl





1.1.1214
3-methyl-4-
H
methyl




chlorophenyl





1.1.1215
3-ethyl-4-
H
methyl




chlorophenyl





1.1.1216
3-cyclopropyl-4-
H
methyl




chlorophenyl





1.1.1217
3-vinyl-4-
H
methyl




chlorophenyl





1.1.1218
3-ethynyl-4-
H
methyl




chlorophenyl





1.1.1219
3-cyano-4-
H
methyl




chlorophenyl





1.1.1220
3-trifluoromethyl-4-
H
methyl




chlorophenyl





1.1.1221
3-methoxy-4-
H
methyl




chlorophenyl





1.1.1222
3-ethoxy-4-
H
methyl




chlorophenyl





1.1.1223
3-trifluoromethoxy-4-
H
methyl




chlorophenyl





1.1.1224
3-nitro-4-
H
methyl




chlorophenyl





1.1.1225
3-fluoro-4-
H
methyl




bromophenyl





1.1.1226
3-chloro-4-
H
methyl




bromophenyl





1.1.1227
3,4-dibromophenyl
H
methyl



1.1.1228
3-methyl-4-
H
methyl




bromophenyl





1.1.1229
3-ethyl-4-
H
methyl




bromophenyl





1.1.1230
3-cyclopropyl-4-
H
methyl




bromophenyl





1.1.1231
3-vinyl-4-
H
methyl




bromophenyl





1.1.1232
3-ethynyl-4-
H
methyl




bromophenyl





1.1.1233
3-cyano-4-
H
methyl




bromophenyl





1.1.1234
3-trifluoromethyl-4-
H
methyl




bromophenyl





1.1.1235
3-methoxy-4-phenyl
H
methyl



1.1.1236
3-ethoxy-4-
H
methyl




bromophenyl





1.1.1237
3-trifluoromethoxy-4-
H
methyl




bromophenyl





1.1.1238
3-nitro-4-
H
methyl




bromophenyl





1.1.1239
3-fluoro-4-iodophenyl
H
methyl



1.1.1240
3-chloro-4-
H
methyl




iodophenyl





1.1.1241
3-bromo-4-
H
methyl




iodophenyl





1.1.1242
3-methyl-4-
H
methyl




iodophenyl





1.1.1243
3-ethyl-4-iodophenyl
H
methyl



1.1.1244
3-cyclopropyl-4-
H
methyl




iodophenyl





1.1.1245
3-vinyl-4-iodophenyl
H
methyl



1.1.1246
3-ethynyl-4-
H
methyl




iodophenyl





1.1.1247
3-cyano-4-
H
methyl




iodophenyl





1.1.1248
3-trifluoromethyl-4-
H
methyl




iodophenyl





1.1.1249
3-methoxy-4-
H
methyl




iodophenyl





1.1.1250
3-ethoxy-4-
H
methyl




iodophenyl





1.1.1251
3-trifluoromethoxy-4-
H
methyl




iodophenyl





1.1.1252
3-nitro-4-iodophenyl
H
methyl



1.1.1253
3-fluoro-4-
H
methyl




methylphenyl





1.1.1254
3-chloro-4-
H
methyl
[CDCl3] 1.75 (s, 3H); 2.42 (s, 3H);



methylphenyl


3.29 (d, 1H); 3.85 (d, 1H); 7.25 (m,






1H); 7.41 (m, 1H); 7.51 (m, 1H).


1.1.1255
3-bromo-4-
H
methyl




methylphenyl





1.1.1256
3,4-dimethylphenyl
H
methyl



1.1.1257
3,4-dimethylphenyl
H
ethyl



1.1.1258
3,4-dimethylphenyl
H
isopropyl



1.1.1259
3,4-dimethylphenyl
H
cyclopropyl



1.1.1260
3-ethyl-4-
H
methyl




methylphenyl





1.1.1261
3-cyclopropyl-4-
H
methyl




methylphenyl





1.1.1262
3-vinyl-4-
H
methyl




methylphenyl





1.1.1263
3-ethyny1-4-
H
methyl




methylphenyl





1.1.1264
3-cyano-4-
H
methyl




methylphenyl





1.1.1265
3-trifluoromethyl-4-
H
methyl




methylphenyl





1.1.1266
3-methoxy-4-
H
methyl




methylphenyl





1.1.1267
3-ethoxy-4-
H
methyl




methylphenyl





1.1.1268
3-trifluoromethoxy-4-
H
methyl




methylphenyl





1.1.1269
3-nitro-4-
H
methyl




methylphenyl





1.1.1270
3-fluoro-4-
H
methyl




ethylphenyl





1.1.1271
3-chloro-4-
H
methyl




ethylphenyl





1.1.1272
3-bromo-4-
H
methyl




ethylphenyl





1.1.1273
3-methyl-4-
H
methyl




ethylphenyl





1.1.1274
3,4-diethylphenyl
H
methyl



1.1.1275
3-cyclopropyl-4-
H
methyl




ethylphenyl





1.1.1276
3-vinyl-4-ethylphenyl
H
methyl



1.1.1277
3-ethynyl-4-
H
methyl




ethylphenyl





1.1.1278
3-cyano-4-
H
methyl




ethylphenyl





1.1.1279
3-trifluoromethyl-4-
H
methyl




ethylphenyl





1.1.1280
3-methoxy-4-
H
methyl




ethylphenyl





1.1.1281
3-ethoxy-4-
H
methyl




ethylphenyl





1.1.1282
3-trifluoromethoxy-4-
H
methyl




ethylphenyl





1.1.1283
3-nitro-4-ethylphenyl
H
methyl



1.1.1284
3-fluoro-4-
H
methyl




propylphenyl





1.1.1285
3-chloro-4-
H
methyl




propylphenyl





1.1.1286
3-bromo-4-
H
methyl




propylphenyl





1.1.1287
3-methyl-4-
H
methyl




propylphenyl





1.1.1288
3-methyl-4-
H
methyl




propylphenyl





1.1.1289
3-cyclopropyl-4-
H
methyl




propylphenyl





1.1.1290
3-vinyl-4-
H
methyl




propylphenyl





1.1.1291
3-ethynyl-4-
H
methyl




propylphenyl





1.1.1292
3-cyano-4-
H
methyl




propylphenyl





1.1.1293
3-trifluoromethyl-4-
H
methyl




propylphenyl





1.1.1294
3-methoxy-4-
H
methyl




propylphenyl





1.1.1295
3-ethoxy-4-
H
methyl




propylphenyl





1.1.1296
3-trifluoromethoxy-4-
H
methyl




propylphenyl





1.1.1297
3-nitro-4-
H
methyl




propylphenyl





1.1.1298
3-fluoro-4-
H
methyl




isopropylphenyl





1.1.1299
3-chloro-4-
H
methyl




isopropylphenyl





1.1.1300
3-bromo-4-
H
methyl




isopropylphenyl





1.1.1301
3-methyl-4-
H
methyl




isopropylphenyl





1.1.1302
3-ethyl-4-
H
methyl




isopropylphenyl





1.1.1303
3-cyclopropyl-4-
H
methyl




isopropylphenyl





1.1.1304
3-vinyl-4-
H
methyl




isopropylphenyl





1.1.1305
3-thynyl-4-
H
methyl




isopreopylphenyl





1.1.1306
3-cyano-4-
H
methyl




isopropylphenyl





1.1.1307
3-trifluoromethyl-4-
H
methyl




isopropylphenyl





1.1.1308
3-methoxy-4-
H
methyl




isopropylphenyl





1.1.1309
3-ethoxy-4-
H
methyl




isopropylphenyl





1.1.1310
3-trifluoromethoxy-4-
H
methyl




isopropylphenyl





1.1.1311
3-nitro-4-
H
methyl




isopropylphenyl





1.1.1312
3-fluoro-4-tert-
H
methyl




butylphenyl





1.1.1313
3-chloro-4-tert-
H
methyl




butylphenyl





1.1.1314
3-bromo-4-tert-
H
methyl




butylphenyl





1.1.1315
3-methyl-4-tert-
H
methyl




butylphenyl





1.1.1316
3-ethyl-4-tert-
H
methyl




butylphenyl





1.1.1317
3-cyclopropyl-4-tert-
H
methyl




butylphenyl





1.1.1318
3-vinyl-4-tert-
H
methyl




butylphenyl





1.1.1319
3-ethynyl-4-tert-
H
methyl




butylphenyl





1.1.1320
3-cyano-4-tert-
H
methyl




butylphenyl





1.1.1321
3-trifluoromethyl-4-
H
methyl




tert-butylphenyl





1.1.1322
3-trifluoromethyl-4-
H
ethyl




tert-butylphenyl





1.1.1323
3-trifluoromethyl-4-
H
isopropyl




tert-butylphenyl





1.1.1324
3-trifluoromethyl-4-
H
cyclopropyl




tert-butylphenyl





1.1.1325
3-methoxy-4-tert-
H
methyl




butylphenyl





1.1.1326
3-ethoxy-4-tert-
H
methyl




butylphenyl





1.1.1327
3-trifluoromethoxy-4-
H
methyl




tert-butylphenyl





1.1.1328
3-nitro-4-tert-
H
methyl




butylphenyl





1.1.1329
3-fluoro-4-
H
methyl




hydroxymethylphenyl





1.1.1330
3-chloro-4-
H
methyl




hydroxymethylphenyl





1.1.1331
3-bromo-4-
H
methyl




hydroxymethylphenyl





1.1.1332
3-methyl-4-
H
methyl




hydroxymethylphenyl





1.1.1333
3-ethyl-4-
H
methyl




hydroxymethylphenyl





1.1.1334
3-cyclopropyl-4-
H
methyl




hydroxymethylphenyl





1.1.1335
3-vinyl-4-
H
methyl




hydroxymethylphenyl





1.1.1336
3-ethynyl-4-
H
methyl




hydroxymethylphenyl





1.1.1337
3-cyano-4-
H
methyl




hydroxymethylphenyl





1.1.1338
3-trifluoromethyl-4-
H
methyl




hydroxymethylphenyl





1.1.1339
3-methoxy-4-
H
methyl




hydroxymethylphenyl





1.1.1340
3-ethoxy-4-
H
methyl




hydroxymethylphenyl





1.1.1341
3-trifluoromethoxy-4-
H
methyl




hydroxymethylphenyl





1.1.1342
3-nitro-4-
H
methyl




hydroxymethylphenyl





1.1.1343
3-fluoro-4-
H
methyl




cyclopropylphenyl





1.1.1344
3-chloro-4-
H
methyl




cyclopropylphenyl





1.1.1345
3-bromo-4-
H
methyl




cyclopropylphenyl





1.1.1346
3-methyl-4-
H
methyl




cyclopropylphenyl





1.1.1347
3-ethyl-4-
H
methyl




cyclopropylphenyl





1.1.1348
3-cyclopropyl-4-
H
methyl




cyclopropylphenyl





1.1.1349
3-vinyl-4-
H
methyl




cyclopropylphenyl





1.1.1350
3-ethyny1-4-
H
methyl




cyclopropylphenyl





1.1.1351
3-cyano-4-
H
methyl




cyclopropylphenyl





1.1.1352
3-trifluoromethyl-4-
H
methyl




cyclopropylphenyl





1.1.1353
3-methoxy-4-
H
methyl




cyclopropylphenyl





1.1.1354
3-ethoxy-4-
H
methyl




cyclopropylphenyl





1.1.1355
3-trifluoromethoxy-4-
H
methyl




cyclopropylphenyl





1.1.1356
3-fluoro-4-
H
methyl




methoxycarbonyl-






phenyl





1.1.1357
3-chloro-4-methoxy-
H
methyl




carbonylphenyl





1.1.1358
3-bromo-4-methoxy-
H
methyl




carbonylphenyl





1.1.1359
3-methyl-4-methoxy-
H
methyl




carbonylphenyl





1.1.1360
3-ethyl-4-methoxy-
H
methyl




carbonylphenyl





1.1.1361
3-cyclopropyl-4-
H
methyl




methoxycarbonyl-






phenyl





1.1.1362
3-vinyl-4-methoxy-
H
methyl




carbonylphenyl





1.1.1363
3-ethynyl-4-methoxy-
H
methyl




carbonylphenyl





1.1.1364
3-cyano-4-
H
methyl




methoxycarbonylphenyl





1.1.1365
3-trifluoromethyl-4-
H
methyl




methoxycarbonyl-






phenyl





1.1.1366
3-methoxy-4-
H
methyl




methoxycarbonyl-






phenyl





1.1.1367
3-ethoxy-4-
H
methyl




methoxycarbonyl-






phenyl





1.1.1368
3-trifluoromethoxy-4-
H
methyl




methoxycarbonyl-






phenyl





1.1.1369
3-nitro-4-methoxy-
H
methyl




carbonylphenyl





1.1.1370
3-fluoro-4-
H
methyl




vinylphenyl





1.1.1371
3-chloro-4-
H
methyl




vinylphenyl





1.1.1372
3-bromo-4-
H
methyl




vinylphenyl





1.1.1373
3-methyl-4-
H
methyl




vinylphenyl





1.1.1374
3-ethyl-4-vinylphenyl
H
methyl



1.1.1375
3-cyclopropyl-4-
H
methyl




vinylphenyl





1.1.1376
3,4-divinylphenyl
H
methyl



1.1.1377
3-ethynyl-4-
H
methyl




vinylphenyl





1.1.1378
3-cyano-4-
H
methyl




vinylphenyl





1.1.1379
3-trifluoromethyl-4-
H
methyl




vinylphenyl





1.1.1380
3-methoxy-4-
H
methyl




vinylphenyl





1.1.1381
3-ethoxy-4-
H
methyl




vinylphenyl





1.1.1382
3-trifluoromethoxy-4-
H
methyl




vinylphenyl





1.1.1383
3-nitro-4-vinylphenyl
H
methyl



1.1.1384
3-fluoro-4-
H
methyl




ethynylphenyl





1.1.1385
3-chloro-4-
H
methyl




ethynylphenyl





1.1.1386
3-bromo-4-
H
methyl




ethynylphenyl





1.1.1387
3-methyl-4-
H
methyl




ethynylphenyl





1.1.1388
3-ethyl-4-
H
methyl




ethynylphenyl





1.1.1389
3-cyclopropyl-4-
H
methyl




ethynylphenyl





1.1.1390
3-vinyl-4-
H
methyl




ethynylphenyl





1.1.1391
3-cyano-4-
H
methyl




ethynylphenyl





1.1.1392
3-trifluoromethyl-4-
H
methyl




ethynylphenyl





1.1.1393
3-methoxy-4-
H
methyl




ethynylphenyl





1.1.1394
3-ethoxy-4-
H
methyl




ethynylphenyl





1.1.1395
3-trifluoromethoxy-4-
H
methyl




ethynylphenyl





1.1.1396
3-nitro-4-
H
methyl




ethynylphenyl





1.1.1397
3-fluoro-4-
H
methyl




ethynylphenyl





1.1.1398
3-fluoro-4-
H
methyl




cyanophenyl





1.1.1399
3-chloro-4-
H
methyl




cyanophenyl





1.1.1400
3-bromo-4-
H
methyl




cyanophenyl





1.1.1401
3-methyl-4-
H
methyl




cyanophenyl





1.1.1402
3-ethyl-4-
H
methyl




cyanophenyl





1.1.1403
3-cyclopropyl-4-
H
methyl




cyanophenyl





1.1.1404
3-vinyl-4-
H
methyl




cyanophenyl





1.1.1405
3-ethynyl-4-
H
methyl




cyanophenyl





1.1.1406
3,4-dicyanophenyl
H
methyl



1.1.1407
3-trifluoromethyl-4-
H
methyl




cyanophenyl





1.1.1408
3-trifluoromethyl-4-
H
ethyl




cyanophenyl





1.1.1409
3-trifluoromethyl-4-
H
isopropyl




cyanophenyl





1.1.1410
3-trifluoromethyl-4-
H
cyclopropyl




cyanophenyl





1.1.1411
3-methoxy-4-
H
methyl




cyanophenyl





1.1.1412
3-ethoxy-4-
H
methyl




cyanophenyl





1.1.1413
3-trifluoromethoxy-4-
H
methyl




cyanophenyl





1.1.1414
3-nitro-4-
H
methyl




cyanophenyl





1.1.1415
3-fluoro-4-
H
methyl




hydroxyphenyl





1.1.1416
3-chloro-4-
H
methyl




hydroxyphenyl





1.1.1417
3-bromo-4-
H
methyl




hydroxyphenyl





1.1.1418
3-methy1-4-
H
methyl




hydroxyphenyl





1.1.1419
3-ethyl-4-
H
methyl




hydroxyphenyl





1.1.1420
3-cyclopropyl-4-
H
methyl




hydroxyphenyl





1.1.1421
3-vinyl-4-
H
methyl




hydroxyphenyl





1.1.1422
3-ethynyl-4-
H
methyl




hydroxyphenyl





1.1.1423
3-cyano-4-
H
methyl




hydroxyphenyl





1.1.1424
3-trifluoromethyl-4-
H
methyl




hydroxyphenyl





1.1.1425
3-methoxy-4-
H
methyl




hydroxyphenyl





1.1.1426
3-ethoxy-4-
H
methyl




hydroxyphenyl





1.1.1427
3-trifluoromethoxy-4-
H
methyl




hydroxyphenyl





1.1.1428
3-nitro-4-
H
methyl




hydroxyphenyl





1.1.1429
3-fluoro-4-
H
methyl




methoxyphenyl





1.1.1430
3-chloro-4-
H
methyl




methoxyphenyl





1.1.1431
3-bromo-4-
H
methyl




methoxyphenyl





1.1.1432
3-methyl-4-
H
methyl




methoxyphenyl





1.1.1433
3-ethyl-4-
H
methyl




methoxyphenyl





1.1.1434
3-cyclopropyl-4-
H
methyl




methoxyphenyl





1.1.1435
3-vinyl-4-
H
methyl




methoxyphenyl





1.1.1436
3-ethynyl-4-
H
methyl




methoxyphenyl





1.1.1437
3-cyano-4-
H
methyl




methoxyphenyl





1.1.1438
3-trifluoromethyl-4-
H
methyl




methoxyphenyl





1.1.1439
3,4-dimethoxyphenyl
H
methyl



1.1.1440
3-ethoxy-4-
H
methyl




methoxyphenyl





1.1.1441
3-trifluoromethoxy-4-
H
methyl




methoxyphenyl





1.1.1442
3-nitro-4-
H
methyl




methoxyphenyl





1.1.1443
3-fluoro-4-
H
methyl




ethoxyphenyl





1.1.1444
3-chloro-4-
H
methyl




ethoxyphenyl





1.1.1445
3-chloro-4-
H
ethyl




ethoxyphenyl





1.1.1446
3-chloro-4-
H
isopropyl




ethoxyphenyl





1.1.1447
3-chloro-4-
H
cyclopropyl




ethoxyphenyl





1.1.1448
3-bromo-4-
H
methyl




ethoxyphenyl





1.1.1449
3-methyl-4-
H
methyl




ethoxyphenyl





1.1.1450
3-ethyl-4-
H
methyl




ethoxyphenyl





1.1.1451
3-cyclopropyl-4-
H
methyl




ethoxyphenyl





1.1.1452
3-vinyl-4-
H
methyl




ethoxyphenyl





1.1.1453
3-ethynyl-4-
H
methyl




ethoxyphenyl





1.1.1454
3-cyano-4-
H
methyl




ethoxyphenyl





1.1.1455
3-trifluoromethyl-4-
H
methyl




ethoxyphenyl





1.1.1456
3-methoxy-4-
H
methyl




ethoxyphenyl





1.1.1457
2,4-diethoxyphenyl
H
methyl



1.1.1458
3-trifluoromethoxy-4-
H
methyl




ethoxyphenyl





1.1.1459
3-nitro-4-
H
methyl




ethoxyphenyl





1.1.1460
3-fluoro-4-
H
methyl




propoxyphenyl





1.1.1461
3-chloro-4-
H
methyl




propoxyphenyl





1.1.1462
3-bromo-4-
H
methyl




propoxyphenyl





1.1.1463
3-methyl-4-
H
methyl




propoxyphenyl





1.1.1464
3-ethyl-4-
H
methyl




propoxyphenyl





1.1.1465
3-cyclopropyl-4-
H
methyl




propoxyphenyl





1.1.1466
3-vinyl-4-
H
methyl




propoxyphenyl





1.1.1467
3-ethynyl-4-
H
methyl




propoxyphenyl





1.1.1468
3-cyano-4-
H
methyl




propoxyphenyl





1.1.1469
3-trifluoromethyl-4-
H
methyl




propoxyphenyl





1.1.1470
3-methoxy-4-propoxy-
H
methyl




phenyl





1.1.1471
3-ethoxy-4-
H
methyl




propoxyphenyl





1.1.1472
3-trifluoromethoxy-4-
H
methyl




propoxyphenyl





1.1.1473
3-nitro-4-
H
methyl




propoxyphenyl





1.1.1474
3-fluoro-4-
H
methyl




isopropoxyphenyl





1.1.1475
3-chloro-4-
H
methyl




isopropoxyphenyl





1.1.1476
3-bromo-4-
H
methyl




isopropoxyphenyl





1.1.1477
3-methyl-4-
H
methyl




isopropoxyphenyl





1.1.1478
3-ethyl-4-
H
methyl




isopropoxyphenyl





1.1.1479
3-cyclopropy1-4-
H
methyl




isopropoxyphenyl





1.1.1480
3-vinyl-4-
H
methyl




isopropoxyphenyl





1.1.1481
3-ethynyl-4-
H
methyl




isopropoxyphenyl





1.1.1482
3-cyano-4-
H
methyl




isopropoxyphenyl





1.1.1483
3-trifluoromethyl-4-
H
methyl




isopropoxyphenyl





1.1.1484
3-methoxy-4-
H
methyl




isopropoxyphenyl





1.1.1485
3-ethoxy-4-
H
methyl




isopropoxyphenyl





1.1.1486
3-trifluoromethoxy-4-
H
methyl




isopropoxyphenyl





1.1.1487
3-nitro-4-
H
methyl




isopropoxyphenyl





1.1.1488
3-fluoro-4-tert-
H
methyl




butoxyphenyl





1.1.1489
3-chloro-4-tert-
H
methyl




butoxyphenyl





1.1.1490
3-bromo-4-tert-
H
methyl




butoxyphenyl





1.1.1491
3-methyl-4-tert-
H
methyl




butoxyphenyl





1.1.1492
3-ethyl-4-tert-
H
methyl




butoxyphenyl





1.1.1493
3-cyclopropyl-4-tert-
H
methyl




butoxyphenyl





1.1.1494
3-vinyl-4-tert-
H
methyl




butoxyphenyl





1.1.1495
3-ethynyl-4-tert-
H
methyl




butoxyphenyl





1.1.1496
3-cyano-4-tert-
H
methyl




butoxyphenyl





1.1.1497
3-trifluoromethyl-4-
H
methyl




tert-butoxyphenyl





1.1.1498
3-methoxy-4-tert-
H
methyl




butoxyphenyl





1.1.1499
3-ethoxy-4-tert-
H
methyl




butoxyphenyl





1.1.1500
3-trifluoromethoxy-4-
H
methyl




tert-butoxyphenyl





1.1.1501
3-nitro-4-tert-
H
methyl




butoxyphenyl





1.1.1502
3-fluoro-4-trifluoro-
H
methyl




methoxyphenyl





1.1.1503
3-chloro-4-trifluoro-
H
methyl




methoxyphenyl





1.1.1504
3-bromo-4-trifluoro-
H
methyl




methoxyphenyl





1.1.1505
3-methyl-4-trifluoro-
H
methyl




methoxyphenyl





1.1.1506
3-ethyl-4-trifluoro-
H
methyl




methoxyphenyl





1.1.1507
3-cyclopropyl-4-
H
methyl




trifluoromethoxy-






phenyl





1.1.1508
3-vinyl-4-trifluoro-
H
methyl




methoxyphenyl





1.1.1509
3-ethynyl-4-trifluoro-
H
methyl




methoxyphenyl





1.1.1510
3-cyano-4-trifluoro-
H
methyl




methoxyphenyl





1.1.1511
3-trifluoromethyl-4-
H
methyl




trifluoromethoxy-






phenyl





1.1.1512
3-methoxy-4-
H
methyl




trifluoromethoxy-






phenyl





1.1.1513
3-ethoxy-4-trifluoro-
H
methyl




methoxyphenyl





1.1.1514
3,4-bis(trifluoro-
H
methyl




methoxy)phenyl





1.1.1515
3-nitro-4-trifluoro-
H
methyl




methoxyphenyl





1.1.1516
3-fluoro-4-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.1517
3-chloro-4-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.1518
3-bromo-4-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.1519
3-methyl-4-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.1520
3-ethyl-4-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.1521
3-cyclopropyl-4-
H
methyl




(2,2,2-trifluoro-






ethoxy)phenyl





1.1.1522
3-vinyl-4-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.1523
3-ethynyl-4-(2,2,2-
H
methyl




trifluoroethoxyphenyl





1.1.1524
3-cyano-4-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.1525
3-trifluoromethyl-4-
H
methyl




(2,2,2-trifluoro-






ethoxy)phenyl





1.1.1526
3-methoxy-4-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.1527
3-ethoxy-4-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.1528
3-trifluoromethoxy-4-
H
methyl




(2,2,2-trifluoro-






ethoxy)phenyl





1.1.1529
3-nitro-4-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.1530
3-fluoro-4-difluoro-
H
methyl




methoxyphenyl





1.1.1531
3-chloro-4-difluoro-
H
methyl




methoxyphenyl





1.1.1532
3-bromo-4-difluoro-
H
methyl




methoxyphenyl





1.1.1533
3-methyl-4-difluoro-
H
methyl




methoxyphenyl





1.1.1534
3-ethyl-4-difluoro-
H
methyl




methoxyphenyl





1.1.1535
3-cyclopropyl-4-
H
methyl




difluoromethoxy-






phenyl





1.1.1536
3-vinyl-4-difluoro-
H
methyl




methoxyphenyl





1.1.1537
3-ethynyl-4-difluoro-
H
methyl




methoxyphenyl





1.1.1538
3-cyano-4-difluoro-
H
methyl




methoxyphenyl





1.1.1539
3-trifluoromethyl-4-
H
methyl




difluoromethoxy-






phenyl





1.1.1540
3-methoxy-4-difluoro-
H
methyl




methoxyphenyl





1.1.1541
3-ethoxy-4-difluoro-
H
methyl




methoxyphenyl





1.1.1542
3-trifluoromethoxy-4-
H
methyl




difluoromethoxy-






phenyl





1.1.1543
3-nitro-4-difluoro-
H
methyl




methoxyphenyl





1.1.1544
3-fluoro-4-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.1545
3-chloro-4-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.1546
3-bromo-4-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.1547
3-methyl-4-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.1548
3-ethyl-4-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.1549
3-cyclopropyl-4-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.1550
3-vinyl-4-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.1551
3-ethynyl-4-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.1552
3-cyano-4-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.1553
3-trifluoromethyl-4-
H
methyl




(2-methoxyethoxy)-






phenyl





1.1.1554
3-methoxy-4-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.1555
3-ethoxy-4-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.1556
3-trifluoromethoxy-
H
methyl




(2-methoxyethoxy)-






phenyl





1.1.1557
3-nitro-4-(2-methoxy-
H
methyl




ethoxy)phenyl





1.1.1558
3-fluoro-4-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1559
3-chloro-4-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1560
3-bromo-4-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1561
3-methyl-4-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1562
3-ethy1-4-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1563
3-cyclopropyl-4-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1564
3-viny1-4-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1565
3-ethynyl-4-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1566
3-cyano-4-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1567
3-trifluoromethyl-4-
H
methyl




(tert-butoxycarbonyl-






oxy)phenyl





1.1.1568
3-methoxy-4-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1569
3-ethoxy-4-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1570
3-trifluoromethoxy-4-
H
methyl




(tert-butoxycarbonyl-






oxy)phenyl





1.1.1571
2-nitro-4-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1572
3-fluoro-4-nitrophenyl
H
methyl



1.1.1573
3-chloro-4-
H
methyl




nitrophenyl





1.1.1574
3-bromo-4-
H
methyl




nitrophenyl





1.1.1575
3-methyl-4-
H
methyl




nitrophenyl





1.1.1576
3-ethyl-4-nitrophenyl
H
methyl



1.1.1577
3-cyclopropyl-4-
H
methyl




nitrophenyl





1.1.1578
3-vinyl-4-nitrophenyl
H
methyl



1.1.1579
3-ethynyl-4-
H
methyl




nitrophenyl





1.1.1580
3-cyano-4-
H
methyl




nitrophenyl





1.1.1581
3-trifluoromethyl-4-
H
methyl




nitrophenyl





1.1.1582
3-methoxy-4-
H
methyl




nitrophenyl





1.1.1583
3-ethoxy-4-
H
methyl




nitrophenyl





1.1.1584
3-trifluoromethoxy-4-
H
methyl




nitrophenyl





1.1.1585
3-fluoro-4-
H
methyl




methylsulfanylphenyl





1.1.1586
3-chloro-4-
H
methyl




methylsulfanylphenyl





1.1.1587
3-bromo-4-
H
methyl




methylsulfanylphenyl





1.1.1588
3-methyl-4-
H
methyl




methylsulfanylphenyl





1.1.1589
3-ethyl-4-
H
methyl




methylsulfanylphenyl





1.1.1590
3-cyclopropyl-4-
H
methyl




methylsulfanylphenyl





1.1.1591
3-vinyl-4-
H
methyl




methylsulfanylphenyl





1.1.1592
3-ethynyl-4-
H
methyl




methylsulfanylphenyl





1.1.1593
3-cyano-4-
H
methyl




methylsulfanylphenyl





1.1.1594
3-trifluoromethyl-4-
H
methyl




methylsulfanylphenyl





1.1.1595
3-methoxy-4-
H
methyl




methylsulfanylphenyl





1.1.1596
3-ethoxy-4-
H
methyl




methylsulfanylphenyl





1.1.1597
3-trifluoromethoxy-4-
H
methyl




methylsulfanylphenyl





1.1.1598
3-nitro-4-
H
methyl




methylsulfanylphenyl





1.1.1599
3,6-difluorophenyl
H
methyl
[CDCl3] 1.78 (s, 3H); 3.39 (d, 1H);






3.91 (dd, 1H); 7.09 (m, 2H); 7.59






(m, 1H).


1.1.1600
3,6-difluorophenyl
H
ethyl



1.1.1601
3,6-difluorophenyl
H
isopropyl



1.1.1602
3,6-difluorophenyl
H
cyclopropyl



1.1.1603
3-chloro-6-
H
methyl




fluorophenyl





1.1.1604
3-bromo-6-
H
methyl
[CDCl3] 1.75 (s, 3H); 3.35 (d, 1H);



fluorophenyl


3.90 (d, 1H); 7.00 (t, 3H); 7.51 (m,






1H); 8.0 (m, 1H).


1.1.1605
3-methyl-6-
H
methyl




fluorophenyl





1.1.1606
3-ethyl-6-
H
methyl




fluorophenyl





1.1.1607
3-cyclopropyl-6-
H
methyl




fluorophenyl





1.1.1608
3-vinyl-6-
H
methyl




fluorophenyl





1.1.1609
3-ethynyl-6-
H
methyl




fluorophenyl





1.1.1610
3-cyano-6-
H
methyl




fluorophenyl





1.1.1611
3-methoxy-6-
H
methyl
[DMSO] 1.53 (s, 3H); 3.39 (d, 1H);



fluorophenyl


3.75 (s, 3H); 3.81 (d, 1H); 7.06 (m,






1H); 7.18 (m, 1H); 7.38 (t, 1H).


1.1.1612
3-ethoxy-6-
H
methyl




fluorophenyl





1.1.1613
3-trifluoromethoxy-6-
H
methyl




fluorophenyl





1.1.1614
3-nitro-6-fluorophenyl
H
methyl



1.1.1615
3-fluoro-6-
H
methyl
[CDCl3] 1.80 (s, 3H); 3.50 (d, 1H);



chlorophenyl


4.02 (d, 1H); 7.10 (m, 1H); 7.40 (m,






2H).


1.1.1616
3-fluoro-6-
H
ethyl




chlorophenyl





1.1.1617
3-fluoro-6-
H
isopropyl




chlorophenyl





1.1.1618
3-fluoro-6-
H
cyclopropyl




chlorophenyl





1.1.1619
3,6-dichlorophenyl
H
methyl
[CDCl3] 1.78 (s, 3H); 3.48 (d, 1H);






3.97 (d, 1H); 7.35 (m, 2H); 7.67 (m,






1H).


1.1.1620
3,6-dichlorophenyl
H
ethyl



1.1.1621
3,6-dichlorophenyl
H
isopropyl



1.1.1622
3,6-dichlorophenyl
H
cyclopropyl



1.1.1623
3-bromo-6-
H
methyl




chlorophenyl





1.1.1624
3-methy1-6-
H
methyl




chlorophenyl





1.1.1625
3-ethyl-6-
H
methyl




chlorophenyl





1.1.1626
3-cyclopropyl-6-
H
methyl




chlorophenyl





1.1.1627
3-vinyl-6-
H
methyl




chlorophenyl





1.1.1628
3-ethyny1-6-
H
methyl




chlorophenyl





1.1.1629
3-cyano-6-
H
methyl




chlorophenyl





1.1.1630
3-trifluoromethyl-6-
H
methyl




chlorophenyl





1.1.1631
3-methoxy-6-
H
methyl




chlorophenyl





1.1.1632
3-ethoxy-6-
H
methyl




chlorophenyl





1.1.1633
3-trifluoromethoxy-6-
H
methyl




chlorophenyl





1.1.1634
3-nitro-6-
H
methyl




chlorophenyl





1.1.1635
3-fluoro-6-
H
methyl




bromophenyl





1.1.1636
3-chloro-6-
H
methyl




bromophenyl





1.1.1637
3,6-dibromophenyl
H
methyl



1.1.1638
3-methyl-6-
H
methyl




bromophenyl





1.1.1639
3-ethyl-6-
H
methyl




bromophenyl





1.1.1640
3-cyclopropyl-6-
H
methyl




bromophenyl





1.1.1641
3-vinyl-6-
H
methyl




bromophenyl





1.1.1642
3-ethynyl-6-
H
methyl




bromophenyl





1.1.1643
3-cyano-6-
H
methyl




bromophenyl





1.1.1644
3-trifluoromethyl-6-
H
methyl




bromophenyl





1.1.1645
3-methoxy-6-phenyl
H
methyl



1.1.1646
3-ethoxy-6-
H
methyl




bromophenyl





1.1.1647
3-trifluoromethoxy-6-
H
methyl




bromophenyl





1.1.1648
3-nitro-6-
H
methyl




bromophenyl





1.1.1649
3-fluoro-6-iodophenyl
H
methyl



1.1.1650
3-chloro-6-
H
methyl




iodophenyl





1.1.1651
3-bromo-6-
H
methyl




iodophenyl





1.1.1652
3-methyl-6-
H
methyl




iodophenyl





1.1.1653
3-ethyl-6-iodophenyl
H
methyl



1.1.1654
3-cyclopropyl-6-
H
methyl




iodophenyl





1.1.1655
3-vinyl-6-iodophenyl
H
methyl



1.1.1656
3-ethynyl-6-
H
methyl




iodophenyl





1.1.1657
3-cyano-6-
H
methyl




iodophenyl





1.1.1658
3-trifluoromethyl-6-
H
methyl




iodophenyl





1.1.1659
3-methoxy-6-
H
methyl




iodophenyl





1.1.1660
3-ethoxy-6-
H
methyl




iodophenyl





1.1.1661
3-trifluoromethoxy-6-
H
methyl




iodophenyl





1.1.1662
3-nitro-6-iodophenyl
H
methyl



1.1.1663
3-fluoro-6-
H
methyl




methylphenyl





1.1.1664
3-chloro-6-
H
methyl




methylphenyl





1.1.1665
3-bromo-6-
H
methyl




methylphenyl





1.1.1666
3,6-dimethylphenyl
H
methyl
[DMSO] 1.56 (s, 3H); 2.28 (s, 3H);






2.40 (s, 3H); 3.38 (d, 1H); 3.80 (d,






1H); 7.15 (m, 2H); 7.25 (d, 1H).


1.1.1667
3-ethyl-6-
H
methyl




methylphenyl





1.1.1668
3-cyclopropyl-6-
H
methyl




methylphenyl





1.1.1669
3-vinyl-6-
H
methyl




methylphenyl





1.1.1670
3-ethynyl-6-
H
methyl




methylphenyl





1.1.1671
3-cyano-6-
H
methyl




methylphenyl





1.1.1672
3-trifluoromethyl-6-
H
methyl




methylphenyl





1.1.1673
3-methoxy-6-
H
methyl




methylphenyl





1.1.1674
3-ethoxy-6-
H
methyl




methylphenyl





1.1.1675
3-trifluoromethoxy-6-
H
methyl




methylphenyl





1.1.1676
3-nitro-6-
H
methyl




methylphenyl





1.1.1677
3-fluoro-6-
H
methyl




ethylphenyl





1.1.1678
3-chloro-6-
H
methyl




ethylphenyl





1.1.1679
3-bromo-6-
H
methyl




ethylphenyl





1.1.1680
3-methyl-6-
H
methyl




ethylphenyl





1.1.1681
3,6-diethylphenyl
H
methyl



1.1.1682
3-cyclopropyl-6-
H
methyl




ethylphenyl





1.1.1683
3-vinyl-6-ethylphenyl
H
methyl



1.1.1684
3-ethynyl-6-
H
methyl




ethylphenyl





1.1.1685
3-cyano-6-
H
methyl




ethylphenyl





1.1.1686
3-trifluoromethyl-6-
H
methyl




ethylphenyl





1.1.1687
3-methoxy-6-
H
methyl




ethylphenyl





1.1.1688
3-ethoxy-6-
H
methyl




ethylphenyl





1.1.1689
3-trifluoromethoxy-6-
H
methyl




ethylphenyl





1.1.1690
3-nitro-6-ethylphenyl
H
methyl



1.1.1691
3-fluoro-6-
H
methyl




propylphenyl





1.1.1692
3-chloro-6-
H
methyl




propylphenyl





1.1.1693
3-bromo-6-
H
methyl




propylphenyl





1.1.1694
3-methyl-6-
H
methyl




propylphenyl





1.1.1695
3-methyl-6-
H
methyl




propylphenyl





1.1.1696
3-cyclopropyl-6-
H
methyl




propylphenyl





1.1.1697
3-vinyl-6-
H
methyl




propylphenyl





1.1.1698
3-ethynyl-6-
H
methyl




propylphenyl





1.1.1699
3-cyano-6-
H
methyl




propylphenyl





1.1.1700
3-trifluoromethyl-6-
H
methyl




propylphenyl





1.1.1701
3-methoxy-6-
H
methyl




propylphenyl





1.1.1702
3-ethoxy-6-
H
methyl




propylphenyl





1.1.1703
3-trifluoromethoxy-6-
H
methyl




propylphenyl





1.1.1704
3-nitro-6-
H
methyl




propylphenyl





1.1.1705
3-fluoro-6-
H
methyl




isopropylphenyl





1.1.1706
3-chloro-6-
H
methyl




isopropylphenyl





1.1.1707
3-bromo-6-
H
methyl




isopropylphenyl





1.1.1708
3-methyl-6-
H
methyl




isopropylphenyl





1.1.1709
3-ethyl-6-
H
methyl




isopropylphenyl





1.1.1710
3-cyclopropyl-6-
H
methyl




isopropylphenyl





1.1.1711
3-vinyl-6-
H
methyl




isopropylphenyl





1.1.1712
3-ethynyl-6-
H
methyl




isopropylphenyl





1.1.1713
3-cyano-6-
H
methyl




isopropylphenyl





1.1.1714
3-trifluoromethyl-6-
H
methyl




isopropylphenyl





1.1.1715
3-methoxy-6-
H
methyl




isopropylphenyl





1.1.1716
3-ethoxy-6-
H
methyl




isopropylphenyl





1.1.1717
3-trifluoromethoxy-6-
H
methyl




isopropylphenyl





1.1.1718
3-nitro-6-
H
methyl




isopropylphenyl





1.1.1719
3-fluoro-6-tert-
H
methyl




butylphenyl





1.1.1720
3-chloro-6-tert-
H
methyl




butylphenyl





1.1.1721
3-bromo-6-tert-
H
methyl




butylphenyl





1.1.1722
3-methyl-6-tert-
H
methyl




butylphenyl





1.1.1723
3-ethyl-6-tert-
H
methyl




butylphenyl





1.1.1724
3-cyclopropyl-6-tert-
H
methyl




butylphenyl





1.1.1725
3-vinyl-6-tert-
H
methyl




butylphenyl





1.1.1726
3-ethynyl-6-tert-
H
methyl




butylphenyl





1.1.1727
3-cyano-6-tert-
H
methyl




butylphenyl





1.1.1728
3-trifluoromethyl-6-
H
methyl




tert-butylphenyl





1.1.1729
3-methoxy-6-tert-
H
methyl




butylphenyl





1.1.1730
3-ethoxy-6-tert-
H
methyl




butylphenyl





1.1.1731
3-trifluoromethoxy-6-
H
methyl




tert-butylphenyl





1.1.1732
3-nitro-6-tert-
H
methyl




butylphenyl





1.1.1733
3-fluoro-6-
H
methyl




hydroxymethylphenyl





1.1.1734
3-chloro-6-
H
methyl




hydroxymethylphenyl





1.1.1735
3-bromo-6-
H
methyl




hydroxymethylphenyl





1.1.1736
3-methyl-6-
H
methyl




hydroxymethylphenyl





1.1.1737
3-ethyl-6-
H
methyl




hydroxymethylphenyl





1.1.1738
3-cyclopropy1-6-
H
methyl




hydroxymethylphenyl





1.1.1739
3-vinyl-6-
H
methyl




hydroxymethylphenyl





1.1.1740
3-ethynyl-6-
H
methyl




hydroxymethylphenyl





1.1.1741
3-cyano-6-
H
methyl




hydroxymethylphenyl





1.1.1742
3-trifluoromethyl-6-
H
methyl




hydroxymethylphenyl





1.1.1743
3-methoxy-6-
H
methyl




hydroxymethylphenyl





1.1.1744
3-ethoxy-6-
H
methyl




hydroxymethylphenyl





1.1.1745
3-trifluoromethoxy-6-
H
methyl




hydroxymethylphenyl





1.1.1746
3-nitro-6-
H
methyl




hydroxymethylphenyl





1.1.1747
3-fluoro-6-
H
methyl




cyclopropylphenyl





1.1.1748
3-chloro-6-
H
methyl




cyclopropylphenyl





1.1.1749
3-bromo-6-
H
methyl




cyclopropylphenyl





1.1.1750
3-methyl-6-
H
methyl




cyclopropylphenyl





1.1.1751
3-ethyl-6-
H
methyl




cyclopropylphenyl





1.1.1752
3-cyclopropyl-6-
H
methyl




cyclopropylphenyl





1.1.1753
3-vinyl-6-
H
methyl




cyclopropylphenyl





1.1.1754
3-ethynyl-6-
H
methyl




cyclopropylphenyl





1.1.1755
3-cyano-6-
H
methyl




cyclopropylphenyl





1.1.1756
3-trifluoromethyl-6-
H
methyl




cyclopropylphenyl





1.1.1757
3-methoxy-6-
H
methyl




cyclopropylphenyl





1.1.1758
3-ethoxy-6-
H
methyl




cyclopropylphenyl





1.1.1759
3-trifluoromethoxy-6-
H
methyl




cyclopropylphenyl





1.1.1760
3-fluoro-6-methoxy-
H
methyl




carbonylphenyl





1.1.1761
3-chloro-6-methoxy-
H
methyl




carbonylphenyl





1.1.1762
3-bromo-6-methoxy-
H
methyl




carbonylphenyl





1.1.1763
3-methyl-6-methoxy-
H
methyl




carbonylphenyl





1.1.1764
3-ethyl-6-methoxy-
H
methyl




carbonylphenyl





1.1.1765
3-cyclopropy1-6-
H
methyl




methoxycarbonyl-






phenyl





1.1.1766
3-vinyl-6-methoxy-
H
methyl




carbonylphenyl





1.1.1767
3-ethynyl-6-methoxy-
H
methyl




carbonylphenyl





1.1.1768
3-cyano-6-methoxy-
H
methyl




carbonylphenyl





1.1.1769
3-trifluoromethyl-6-
H
methyl




methoxycarbonyl-






phenyl





1.1.1770
3-methoxy-6-
H
methyl




methoxycarbonyl-






phenyl





1.1.1771
3-ethoxy-6-
H
methyl




methoxycarbonyl-






phenyl





1.1.1772
3-trifluoromethoxy-6-
H
methyl




methoxycarbonyl-






phenyl





1.1.1773
3-nitro-6-methoxy-
H
methyl




carbonylphenyl





1.1.1774
3-fluoro-6-
H
methyl




vinylphenyl





1.1.1775
3-chloro-6-
H
methyl




vinylphenyl





1.1.1776
3-bromo-6-
H
methyl




vinylphenyl





1.1.1777
3-methy1-6-
H
methyl




vinylphenyl





1.1.1778
3-ethyl-6-vinylphenyl
H
methyl



1.1.1779
3-cyclopropyl-6-
H
methyl




vinylphenyl





1.1.1780
3,6-divinylphenyl
H
methyl



1.1.1781
3-ethynyl-6-
H
methyl




vinylphenyl





1.1.1782
3-cyano-6-
H
methyl




vinylphenyl





1.1.1783
3-trifluoromethyl-6-
H
methyl




vinylphenyl





1.1.1784
3-methoxy-6-
H
methyl




vinylphenyl





1.1.1785
3-ethoxy-6-
H
methyl




vinylphenyl





1.1.1786
3-trifluoromethoxy-6-
H
methyl




vinylphenyl





1.1.1787
3-nitro-6-vinylphenyl
H
methyl



1.1.1788
3-fluoro-6-
H
methyl




ethynylphenyl





1.1.1789
3-chloro-6-
H
methyl




ethynylphenyl





1.1.1790
3-bromo-6-
H
methyl




ethynylphenyl





1.1.1791
3-methy-6-
H
methyl




ethynylphenyl





1.1.1792
3-ethyl-6-
H
methyl




ethynylphenyl





1.1.1793
3-cyclopropyl-6-
H
methyl




ethynylphenyl





1.1.1794
3-vinyl-6-
H
methyl




ethynylphenyl





1.1.1795
3-cyano-6-
H
methyl




ethynylphenyl





1.1.1796
3-trifluoromethyl-6-
H
methyl




ethynylphenyl





1.1.1797
3-methoxy-6-
H
methyl




ethynylphenyl





1.1.1798
3-ethoxy-6-
H
methyl




ethynylphenyl





1.1.1799
3-trifluoromethoxy-6-
H
methyl




ethynylphenyl





1.1.1800
3-nitro-6-
H
methyl




ethynylphenyl





1.1.1801
3-fluoro-6-
H
methyl




ethynylphenyl





1.1.1802
3-fluoro-6-
H
methyl




cyanophenyl





1.1.1803
3-chloro-6-
H
methyl




cyanophenyl





1.1.1804
3-bromo-6-
H
methyl




cyanophenyl





1.1.1805
3-methyl-6-
H
methyl




cyanophenyl





1.1.1806
3-ethyl-6-
H
methyl




cyanophenyl





1.1.1807
3-cyclopropyl-6-
H
methyl




cyanophenyl





1.1.1808
3-vinyl-6-
H
methyl




cyanophenyl





1.1.1809
3-ethynyl-6-
H
methyl




cyanophenyl





1.1.1810
3-cyano-6-
H
methyl




cyanophenyl





1.1.1811
3-trifluoromethyl-6-
H
methyl




cyanophenyl





1.1.1812
3-methoxy-6-
H
methyl




cyanophenyl





1.1.1813
3-ethoxy-6-
H
methyl




cyanophenyl





1.1.1814
3-trifluoromethoxy-6-
H
methyl




cyanophenyl





1.1.1815
3-nitro-6-
H
methyl




cyanophenyl





1.1.1816
3-fluoro-6-
H
methyl




hydroxyphenyl





1.1.1817
3-chloro-6-
H
methyl




hydroxyphenyl





1.1.1818
3-bromo-6-
H
methyl




hydroxyphenyl





1.1.1819
3-methyl-6-
H
methyl




hydroxyphenyl





1.1.1820
3-ethyl-6-
H
methyl




hydroxyphenyl





1.1.1821
3-cyclopropyl-6-
H
methyl




hydroxyphenyl





1.1.1822
3-vinyl-6-
H
methyl




hydroxyphenyl





1.1.1823
3-ethynyl-6-
H
methyl




hydroxyphenyl





1.1.1824
3-cyano-6-
H
methyl




hydroxyphenyl





1.1.1825
3-trifluoromethyl-6-
H
methyl




hydroxyphenyl





1.1.1826
3-methoxy-6-
H
methyl




hydroxyphenyl





1.1.1827
3-ethoxy-6-
H
methyl




hydroxyphenyl





1.1.1828
3-trifluoromethoxy-6-
H
methyl




hydroxyphenyl





1.1.1829
3-nitro-6-
H
methyl




hydroxyphenyl





1.1.1830
3-fluoro-6-
H
methyl




methoxyphenyl





1.1.1831
3-chloro-6-
H
methyl




methoxyphenyl





1.1.1832
3-bromo-6-
H
methyl




methoxyphenyl





1.1.1833
3-methyl-6-
H
methyl




methoxyphenyl





1.1.1834
3-ethyl-6-
H
methyl




methoxyphenyl





1.1.1835
3-cyclopropyl-6-
H
methyl




methoxyphenyl





1.1.1836
3-vinyl-6-
H
methyl




methoxyphenyl





1.1.1837
3-ethynyl-6-
H
methyl




methoxyphenyl





1.1.1838
3-cyano-6-
H
methyl




methoxyphenyl





1.1.1839
3-trifluoromethyl-6-
H
methyl




methoxyphenyl





1.1.1840
3,6-dimethoxy--
H
methyl




phenyl





1.1.1841
3-ethoxy-6-
H
methyl




methoxyphenyl





1.1.1842
3-trifluoromethoxy-6-
H
methyl




methoxyphenyl





1.1.1843
3-nitro-6-
H
methyl




methoxyphenyl





1.1.1844
3-fluoro-6-
H
methyl




ethoxyphenyl





1.1.1845
3-chloro-6-
H
methyl




ethoxyphenyl





1.1.1846
3-bromo-6-
H
methyl




ethoxyphenyl





1.1.1847
3-methyl-6-
H
methyl




ethoxyphenyl





1.1.1848
3-ethyl-6-
H
methyl




ethoxyphenyl





1.1.1849
3-cyclopropyl-6-
H
methyl




ethoxyphenyl





1.1.1850
3-vinyl-6-
H
methyl




ethoxyphenyl





1.1.1851
3-ethynyl-6-
H
methyl




ethoxyphenyl





1.1.1852
3-cyano-6-
H
methyl




ethoxyphenyl





1.1.1853
3-trifluoromethyl-6-
H
methyl




ethoxyphenyl





1.1.1854
3-methoxy-6-
H
methyl




ethoxyphenyl





1.1.1855
2,6-diethoxyphenyl
H
methyl



1.1.1856
3-trifluoromethoxy-6-
H
methyl




ethoxyphenyl





1.1.1857
3-nitro-6-
H
methyl




ethoxyphenyl





1.1.1858
3-fluoro-6-
H
methyl




propoxyphenyl





1.1.1859
3-chloro-6-
H
methyl




propoxyphenyl





1.1.1860
3-bromo-6-
H
methyl




propoxyphenyl





1.1.1861
3-methyl-6-
H
methyl




propoxyphenyl





1.1.1862
3-ethyl-6-
H
methyl




propoxyphenyl





1.1.1863
3-cyclopropyl-6-
H
methyl




propoxyphenyl





1.1.1864
3-vinyl-6-
H
methyl




propoxyphenyl





1.1.1865
3-ethynyl-6-
H
methyl




propoxyphenyl





1.1.1866
3-cyano-6-
H
methyl




propoxyphenyl





1.1.1867
3-trifluoromethyl-6-
H
methyl




propoxyphenyl





1.1.1868
3-methoxy-6-propoxy-
H
methyl




phenyl





1.1.1869
3-ethoxy-6-
H
methyl




propoxyphenyl





1.1.1870
3-trifluoromethoxy-6-
H
methyl




propoxyphenyl





1.1.1871
3-nitro-6-
H
methyl




propoxyphenyl





1.1.1872
3-fluoro-6-
H
methyl




isopropoxyphenyl





1.1.1873
3-chloro-6-
H
methyl




isopropoxyphenyl





1.1.1874
3-bromo-6-
H
methyl




isopropoxyphenyl





1.1.1875
3-methy1-6-
H
methyl




isopropoxyphenyl





1.1.1876
3-ethy1-6-
H
methyl




isopropoxyphenyl





1.1.1877
3-cyclopropy1-6-
H
methyl




isopropoxyphenyl





1.1.1878
3-viny1-6-
H
methyl




isopropoxyphenyl





1.1.1879
3-ethyny1-6-
H
methyl




isopropoxyphenyl





1.1.1880
3-cyano-6-
H
methyl




isopropoxyphenyl





1.1.1881
3-trifluoromethy1-6-
H
methyl




isopropoxyphenyl





1.1.1882
3-methoxy-6-
H
methyl




isopropoxyphenyl





1.1.1883
3-ethoxy-6-
H
methyl




isopropoxyphenyl





1.1.1884
3-trifluoromethoxy-6-
H
methyl




isopropoxyphenyl





1.1.1885
3-nitro-6-
H
methyl




isopropoxyphenyl





1.1.1886
3-fluoro-6-tert-
H
methyl




butoxyphenyl





1.1.1887
3-chloro-6-tert-
H
methyl




butoxyphenyl





1.1.1888
3-bromo-6-tert-
H
methyl




butoxyphenyl





1.1.1889
3-methyl-6-tert-
H
methyl




butoxyphenyl





1.1.1890
3-ethyl-6-tert-
H
methyl




butoxyphenyl





1.1.1891
3-cyclopropyl-6-tert-
H
methyl




butoxyphenyl





1.1.1892
3-vinyl-6-tert-
H
methyl




butoxyphenyl





1.1.1893
3-ethynyl-6-tert-
H
methyl




butoxyphenyl





1.1.1894
3-cyano-6-tert-
H
methyl




butoxyphenyl





1.1.1895
3-trifluoromethyl-6-
H
methyl




tert-butoxyphenyl





1.1.1896
3-methoxy-6-tert-
H
methyl




butoxyphenyl





1.1.1897
3-ethoxy-6-tert-
H
methyl




butoxyphenyl





1.1.1898
3-trifluoromethoxy-6-
H
methyl




tert-butoxyphenyl





1.1.1899
3-nitro-6-tert-
H
methyl




butoxyphenyl





1.1.1900
3-fluoro-6-trifluoro-
H
methyl




methoxyphenyl





1.1.1901
3-chloro-6-trifluoro-
H
methyl




methoxyphenyl





1.1.1902
3-bromo-6-trifluoro-
H
methyl




methoxyphenyl





1.1.1903
3-methyl-6-trifluoro-
H
methyl




methoxyphenyl





1.1.1904
3-ethyl-6-trifluoro-
H
methyl




methoxyphenyl





1.1.1905
3-cyclopropyl-6-
H
methyl




trifluoromethoxy-






phenyl





1.1.1906
3-vinyl-6-trifluoro-
H
methyl




methoxyphenyl





1.1.1907
3-ethynyl-6-trifluoro-
H
methyl




methoxyphenyl





1.1.1908
3-cyano-6-trifluoro-
H
methyl




methoxyphenyl





1.1.1909
3-trifluoromethyl-6-
H
methyl




trifluoromethoxy-






phenyl





1.1.1910
3-methoxy-6-
H
methyl




trifluoromethoxy-






phenyl





1.1.1911
3-ethoxy-6-trifluoro-
H
methyl




methoxyphenyl





1.1.1912
3,6-bis(trifluoro-
H
methyl




methoxy)phenyl





1.1.1913
3-nitro-6-trifluoro-
H
methyl




methoxyphenyl





1.1.1914
3-fluoro-6-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.1915
3-chloro-6-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.1916
3-bromo-6-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.1917
3-methyl-6-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.1918
3-ethyl-6-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.1919
3-cyclopropyl-6-
H
methyl




(2,2,2-trifluoro-






ethoxy)phenyl





1.1.1920
3-vinyl-6-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.1921
3-ethynyl-6-(2,2,2-
H
methyl




trifluoroethoxyphenyl





1.1.1922
3-cyano-6-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.1923
3-trifluoromethyl-6-
H
methyl




(2,2,2-trifluoro-






ethoxy)phenyl





1.1.1924
3-methoxy-6-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.1925
3-ethoxy-6-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.1926
3-trifluoromethoxy-6-
H
methyl




(2,2,2-trifluoro-






ethoxy)phenyl





1.1.1927
3-nitro-6-(2,2,2-
H
methyl




trifluoroethoxy)-






phenyl





1.1.1928
3-fluoro-6-difluoro-
H
methyl




methoxyphenyl





1.1.1929
3-chloro-6-difluoro-
H
methyl




methoxyphenyl





1.1.1930
3-bromo-6-difluoro-
H
methyl




methoxyphenyl





1.1.1931
3-methyl-6-difluoro-
H
methyl




methoxyphenyl





1.1.1932
3-ethyl-6-difluoro-
H
methyl




methoxyphenyl





1.1.1933
3-cyclopropyl-6-
H
methyl




difluoromethoxy-






phenyl





1.1.1934
3-vinyl-6-difluoro-
H
methyl




methoxyphenyl





1.1.1935
3-ethynyl-6-difluoro-
H
methyl




methoxyphenyl





1.1.1936
3-cyano-6-difluoro-
H
methyl




methoxyphenyl





1.1.1937
3-trifluoromethyl-6-
H
methyl




difluoromethoxy-






phenyl





1.1.1938
3-methoxy-6-difluoro-
H
methyl




methoxyphenyl





1.1.1939
3-ethoxy-6-difluoro-
H
methyl




methoxyphenyl





1.1.1940
3-trifluoromethoxy-6-
H
methyl




difluoromethoxy-






phenyl





1.1.1941
3-nitro-6-difluoro-
H
methyl




methoxyphenyl





1.1.1942
3-fluoro-6-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.1943
3-chloro-6-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.1944
3-bromo-6-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.1945
3-methyl-6-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.1946
3-ethyl-6-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.1947
3-cyclopropyl-6-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.1948
3-vinyl-6-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.1949
3-ethynyl-6-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.1950
3-cyano-6-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.1951
3-trifluoromethyl-6-
H
methyl




(2-methoxyethoxy)-






phenyl





1.1.1952
3-methoxy-6-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.1953
3-ethoxy-6-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.1954
3-trifluoromethoxy-
H
methyl




(2-methoxyethoxy)-






phenyl





1.1.1955
3-nitro-6-(2-
H
methyl




methoxyethoxy)-






phenyl





1.1.1956
3-fluoro-6-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1957
3-chloro-6-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1958
3-bromo-6-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1959
3-methyl-6-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1960
3-ethyl-6-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1961
3-cyclopropyl-6-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1962
3-vinyl-6-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1963
3-ethynyl-6-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1964
3-cyano-6-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1965
3-trifluoromethyl-6-
H
methyl




(tert-






butoxycarbonyloxy)-






phenyl





1.1.1966
3-methoxy-6-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1967
3-ethoxy-6-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1968
3-trifluoromethoxy-6-
H
methyl




(tert-butoxycarbonyl-






oxy)phenyl





1.1.1969
2-nitro-6-(tert-
H
methyl




butoxycarbonyloxy)-






phenyl





1.1.1970
3-fluoro-6-nitrophenyl
H
methyl



1.1.1971
3-chloro-6-
H
methyl




nitrophenyl





1.1.1972
3-bromo-6-
H
methyl




nitrophenyl





1.1.1973
3-methyl-6-
H
methyl




nitrophenyl





1.1.1974
3-ethyl-6-nitrophenyl
H
methyl



1.1.1975
3-cyclopropyl-6-
H
methyl




nitrophenyl





1.1.1976
3-vinyl-6-nitrophenyl
H
methyl



1.1.1977
3-ethynyl-6-
H
methyl




nitrophenyl





1.1.1978
3-cyano-6-
H
methyl




nitrophenyl





1.1.1979
3-trifluoromethyl-6-
H
methyl




nitrophenyl





1.1.1980
3-methoxy-6-
H
methyl




nitrophenyl





1.1.1981
3-ethoxy-6-
H
methyl




nitrophenyl





1.1.1982
3-trifluoromethoxy-6-
H
methyl




nitrophenyl





1.1.1983
3-fluoro-6-
H
methyl




methylsulfanylphenyl





1.1.1984
3-chloro-6-
H
methyl




methylsulfanylphenyl





1.1.1985
3-bromo-6-
H
methyl




methylsulfanylphenyl





1.1.1986
3-methyl-6-
H
methyl




methylsulfanylphenyl





1.1.1987
3-ethyl-6-
H
methyl




methylsulfanylphenyl





1.1.1988
3-cyclopropyl-6-
H
methyl




methylsulfanylphenyl





1.1.1989
3-vinyl-6-
H
methyl




methylsulfanylphenyl





1.1.1990
3-ethynyl-6-
H
methyl




methylsulfanylphenyl





1.1.1991
3-cyano-6-
H
methyl




methylsulfanylphenyl





1.1.1992
3-trifluoromethyl-6-
H
methyl




methylsulfanylphenyl





1.1.1993
3-methoxy-6-
H
methyl




methylsulfanylphenyl





1.1.1994
3-ethoxy-6-
H
methyl




methylsulfanylphenyl





1.1.1995
3-trifluoromethoxy-6-
H
methyl




methylsulfanylphenyl





1.1.1996
3-nitro-6-
H
methyl




methylsulfanylphenyl





1.1.1997
2,3,4-trifluorophenyl
H
methyl
[CDCl3] 1.78 (s, 3H); 3.35 (dd, 1H);






3.90 (dd, 1H); 7.03 (m, 1H); 7.60






(m, 1H).


1.1.1998
2,3,4-trichlorophenyl
H
methyl



1.1.1999
2,3,4-trimethylphenyl
H
methyl



1.1.2000
2-fluoro-2-chloro-5-
H
methyl




trifluoromethylphenyl





1.1.2001
2,3,5-trifluorophenyl
H
methyl
[DMSO] 1.58 (s, 3H); 3.41 (d, 1H);






3.71 (d, 1H); 7.41 (m, 1H); 7.71 (m,






1H).


1.1.2002
2,3,5-trichlorophenyl
H
methyl



1.1.2003
2,3,5-trimethylphenyl
H
methyl



1.1.2004
2,3-dichloro-5-
H
methyl
[CDCl3] 1.7.(s, 3H); 3,5 (d, 1H); 3.7



methoxyphenyl


(s, 3H); 3,95 (d, 1H); 7.02-7.13 (m,






2H).


1.1.2005
2,3,6-trifluorophenyl
H
methyl



1.1.2006
2,3,6-trichlorophenyl
H
methyl
[CDCl3] 1.85 (s, 3H); 3.26 (d, 1H);






3.78 (d, 1H); 7.33 (d, 1H); 7.49 (d,






1H).


1.1.2007
2,3,6-trimethylphenyl
H
methyl



1.1.2008
3,4,5-trifluorophenyl
H
methyl
[CDCl3] 1.80 (s, 3H); 3.22 (d, 1H);






3.80 (d, 1H); 7.30 (m, 2H).


1.1.2009
3,4,5-trichlorophenyl
H
methyl
[CDCl3] 1.80 (s, 3H); 3.25 (d, 1H);






3.85 (d, 1H); 7.65 (, 2H).


1.1.2010
3,4,5-trimethylphenyl
H
methyl



1.1.2011
3,5-dimethy1-4-
H
methyl




fluorophenyl





1.1.2012
3,5-dichloro-4-
H
methyl
[CDCl3] 1.81 (s, 3H); 3.25 (d, 1H);



methoxyphenyl


3.82 (d, 1H); 3.95 (s, 3H); 7.60 (s,






2H).


1.1.2013
3,5-difluoro-4-
H
methyl
[CDCl3] 1.81 (s, 3H); 3.24 (d, 1H);



chlorophenyl


3.83 (d, 1H); 7.27 (m, 3H).


1.1.2014
3,5-dichloro-4-
H
methyl
[CDCl3] 1.79 (s, 3H); 3.25 (d, 1H);



hydroxyphenyl


3.80 (d, 1H); 7.59 (s, 2H).


1.1.2015
3,5-trifluoromethyl-4-
H
methyl




chlorophenyl





1.1.2016
3,4,6-trifluorophenyl
H
methyl



1.1.2017
3,4,6-trichlorophenyl
H
methyl



1.1.2018
3,4,6-trimethylphenyl
H
methyl



1.1.2019
pentafluorophenyl
H
methyl
[CDCl3] 1.80 (s, 3H); 3.34 (d, 1H);






3.9 (d, 1H).
















TABLE 1.2







Inventive compounds of the general formula (I) in which W* is COOH, R1


and R2 are each hydrogen, and aryl is the radical.








 








 










No.
Aryl
R3
Physical data





1.2.1
3-fluorophenyl
fluoromethyl
[CDCl3] 3.56 (d,1H); 3.80





(d,1H); 4.71 (d,1H); 4.83





(d,1H); 7.18 (m,1H); 7.41





(m,3H).


1.2.2
3-fluorophenyl
chloromethyl
[CDCl3] 3.62 (d,1H); 3.90





(m,2H); 4.03 (d,1H); 7.17





(m,1H); 7.41 (m,3H).


1.2.3
3-fluorophenyl
bromomethyl



1.2.4
3-fluorophenyl
difluoromethyl



1.2.5
3-fluorophenyl
trifluoromethyl



1.2.6
3-fluorophenyl
cyano



1.2.7
3-chlorophenyl
fluoromethyl



1.2.8
3-chlorophenyl
chloromethyl



1.2.9
3-chlorophenyl
bromomethyl



1.2.10
3-chlorophenyl
difluoromethyl



1.2.11
3-chlorophenyl
trifluoromethyl



1.2.12
3-chlorophenyl
cyano



1.2.13
3-bromophenyl
fluoromethyl



1.2.14
3-bromophenyl
chloromethyl



1.2.15
3-iodophenyl
fluoromethyl



1.2.16
3-iodophenyl
chloromethyl



1.2.17
3-methylphenyl
fluoromethyl



1.2.18
3-methylphenyl
chloromethyl



1.2.19
3-ethylphenyl
fluoromethyl



1.2.20
3-propylphenyl
fluoromethyl



1.2.21
3-isopropylphenyl
fluoromethyl



1.2.22
3-n-butylphenyl
fluoromethyl



1.2.23
3-i-butylphenyl
fluoromethyl



1.2.24
3-tert-butylphenyl
fluoromethyl



1.2.25
3-cyclopropylphenyl
fluoromethyl



1.2.26
3-cyclobutylphenyl
fluoromethyl



1.2.27
3-cyclopentylphenyl
fluoromethyl



1.2.28
3-vinylphenyl
fluoromethyl



1.2.29
3-ethynylphenyl
fluoromethyl



1.2.30
3-cyanophenyl
fluoromethyl



1.2.31
3-trifluoromethylphenyl
fluoromethyl



1.2.32
3-difluoromethylphenyl
fluoromethyl



1.2.33
3-(hydroxycarbonyl)phenyl
fluoromethyl



1.2.34
3-(methoxycarbonyl)phenyl
fluoromethyl



1.2.35
3-(ethoxycarbonyl)phenyl
fluoromethyl



1.2.36
3-hydroxymethylphenyl
fluoromethyl



1.2.37
3-carbamoylphenyl
fluoromethyl



1.2.38
3-hydroxyphenyl
fluoromethyl



1.2.39
3-methoxyphenyl
fluoromethyl



1.2.40
3-ethoxyphenyl
fluoromethyl



1.2.41
3-propyloxyphenyl
fluoromethyl



1.2.42
3-isopropyloxyphenyl
fluoromethyl



1.2.43
3-n-butyloxyphenyl
fluoromethyl



1.2.44
3-i-butyloxyphenyl
fluoromethyl



1.2.45
3-t-butyloxyphenyl
fluoromethyl



1.2.46
3-difluoromethoxyphenyl
fluoromethyl



1.2.47
3-trifluoromethoxyphenyl
fluoromethyl



1.2.48
3-(2,2,2-trifluoroethoxy)-phenyl
fluoromethyl



1.2.49
3-(2-chloroethoxy)-phenyl
fluoromethyl



1.2.50
3-(2-hydroxyethoxy)-phenyl
fluoromethyl



1.2.51
3-(2-methoxyethoxy)-phenyl
fluoromethyl



1.2.52
3-[(tert-butoxycarbonyl)oxy]phenyl
fluoromethyl



1.2.53
3-nitrophenyl
fluoromethyl



1.2.54
3-acetoxyphenyl
fluoromethyl



1.2.55
{3-[(tert-
fluoromethyl




butoxycarbonyl)amino]phenyl}




1.2.56
3-methylsulfanylphenyl
fluoromethyl



1.2.57
3-ethylsulfanylphenyl
fluoromethyl



1.2.58
3-(pentafluoro-lambda6-sulfanyl)-
fluoromethyl




phenyl




1.2.59
2,3-difluorophenyl
fluoromethyl



1.2.60
2,3-difluorophenyl
chloromethyl



1.2.61
2,3-difluorophenyl
bromomethyl



1.2.62
2,3-difluorophenyl
difluoromethyl



1.2.63
2,3-difluorophenyl
trifluoromethyl



1.2.64
2,3-difluorophenyl
cyano



1.2.65
2-chloro-3-fluorophenyl
fluoromethyl



1.2.66
2-bromo-3-fluorophenyl
fluoromethyl



1.2.67
2-methyl-3-fluorophenyl
fluoromethyl



1.2.68
2-ethyl-3-fluorophenyl
fluoromethyl



1.2.69
2-cyclopropyl-3-fluorophenyl
fluoromethyl



1.2.70
2-vinyl-3-fluorophenyl
fluoromethyl



1.2.71
2-ethynyl-3-fluorophenyl
fluoromethyl



1.2.72
2-cyano-3-fluorophenyl
fluoromethyl



1.2.73
2-methoxy-3-fluorophenyl
fluoromethyl



1.2.74
2-ethoxy-3-fluorophenyl
fluoromethyl



1.2.75
2-trifluoromethoxy-3-fluorophenyl
fluoromethyl



1.2.76
2-nitro-3-fluorophenyl
fluoromethyl



1.2.77
2-fluoro-3-chlorophenyl
fluoromethyl



1.2.78
2,3-dichlorophenyl
fluoromethyl



1.2.79
2,3-dichlorophenyl
chloromethyl



1.2.80
2,3-dichlorophenyl
bromomethyl



1.2.81
2,3-dichlorophenyl
difluoromethyl



1.2.82
2-bromo-3-chlorophenyl
fluoromethyl



1.2.83
2-methyl-3-chlorophenyl
fluoromethyl



1.2.84
2-ethyl-3-chlorophenyl
fluoromethyl



1.2.85
2-cyclopropyl-3-chlorophenyl
fluoromethyl



1.2.86
2-vinyl-3-chlorophenyl
fluoromethyl



1.2.87
2-ethynyl-3-chlorophenyl
fluoromethyl



1.2.88
2-cyano-3-chlorophenyl
fluoromethyl



1.2.89
2-trifluoromethyl-2-chlorophenyl
fluoromethyl



1.2.90
2-methoxy-3-chlorophenyl
fluoromethyl



1.2.91
2-ethoxy-3-chlorophenyl
fluoromethyl



1.2.92
2-trifluoromethoxy-3-chlorophenyl
fluoromethyl



1.2.93
2-nitro-3-chlorophenyl
fluoromethyl



1.2.94
2-fluoro-3-bromophenyl
fluoromethyl



1.2.95
2-chloro-3-bromophenyl
fluoromethyl



1.2.96
2,3-dibromophenyl
fluoromethyl



1.2.97
2-methyl-3-bromophenyl
fluoromethyl



1.2.98
2-ethyl-3-bromophenyl
fluoromethyl



1.2.99
2-cyclopropyl-3-bromophenyl
fluoromethyl



1.2.100
2-vinyl-3-bromophenyl
fluoromethyl



1.2.101
2-ethynyl-3-bromophenyl
fluoromethyl



1.2.102
2-cyano-3-bromophenyl
fluoromethyl



1.2.103
2-trifluoromethyl-3-bromophenyl
fluoromethyl



1.2.104
2-methoxy-3-phenyl
fluoromethyl



1.2.105
2-ethoxy-3-bromophenyl
fluoromethyl



1.2.106
2-trifluoromethoxy-3-bromophenyl
fluoromethyl



1.2.107
2-nitro-3-bromophenyl
fluoromethyl



1.2.108
2-fluoro-3-iodophenyl
fluoromethyl



1.2.109
2-chloro-3-iodophenyl
fluoromethyl



1.2.110
2-bromo-3-iodophenyl
fluoromethyl



1.2.111
2-methyl-3-iodophenyl
fluoromethyl



1.2.112
2-ethyl-3-iodophenyl
fluoromethyl



1.2.113
2-cyclopropyl-3-iodophenyl
fluoromethyl



1.2.114
2-vinyl-3-iodophenyl
fluoromethyl



1.2.115
2-ethynyl-3-iodophenyl
fluoromethyl



1.2.116
2-cyano-3-iodophenyl
fluoromethyl



1.2.117
2-trifluoromethyl-3-iodophenyl
fluoromethyl



1.2.118
2-methoxy-3-iodophenyl
fluoromethyl



1.2.119
2-ethoxy-3-iodophenyl
fluoromethyl



1.2.120
2-trifluoromethoxy-3-iodophenyl
fluoromethyl



1.2.121
2-nitro-3-iodophenyl
fluoromethyl



1.2.122
2-fluoro-3-methylphenyl
fluoromethyl



1.2.123
2-fluoro-3-methylphenyl
chloromethyl



1.2.124
2-fluoro-3-methylphenyl
bromomethyl



1.2.125
2-fluoro-3-methylphenyl
difluoromethyl



1.2.126
2-chloro-3-methylphenyl
fluoromethyl



1.2.127
2-chloro-3-methylphenyl
chloromethyl



1.2.128
2-chloro-3-methylphenyl
bromomethyl



1.2.129
2-chloro-3-methylphenyl
difluoromethyl



1.2.130
2-bromo-3-methylphenyl
fluoromethyl



1.2.131
2,3-dimethylphenyl
fluoromethyl



1.2.132
2,3-dimethylphenyl
chloromethyl



1.2.133
2,3-dimethylphenyl
bromomethyl



1.2.134
2,3-dimethylphenyl
difluoromethyl



1.2.135
2-ethyl-3-methylphenyl
fluoromethyl



1.2.136
2-cyclopropyl-3-methylphenyl
fluoromethyl



1.2.137
2-vinyl-3-methylphenyl
fluoromethyl



1.2.138
2-ethynyl-3-methylphenyl
fluoromethyl



1.2.139
2-cyano-3-methylphenyl
fluoromethyl



1.2.140
2-trifluoromethyl-3-methylphenyl
fluoromethyl



1.2.141
2-methoxy-3-methylphenyl
fluoromethyl



1.2.142
2-ethoxy-3-methylphenyl
fluoromethyl



1.2.143
2-trifluoromethoxy-3-methylphenyl
fluoromethyl



1.2.144
2-nitro-3-methylphenyl
fluoromethyl



1.2.145
2-fluoro-3-ethylphenyl
fluoromethyl



1.2.146
2-chloro-3-ethylphenyl
fluoromethyl



1.2.147
2-bromo-3-ethylphenyl
fluoromethyl



1.2.148
2-methyl-3-ethylphenyl
fluoromethyl



1.2.149
2,3-diethylphenyl
fluoromethyl



1.2.150
2-cyclopropyl-3-ethylphenyl
fluoromethyl



1.2.151
2-vinyl-3-ethylphenyl
fluoromethyl



1.2.152
2-ethynyl-3-ethylphenyl
fluoromethyl



1.2.153
2-cyano-3-ethylphenyl
fluoromethyl



1.2.154
2-trifluoromethyl-3-ethylphenyl
fluoromethyl



1.2.155
2-methoxy-3-ethylphenyl
fluoromethyl



1.2.156
2-ethoxy-3-ethylphenyl
fluoromethyl



1.2.157
2-trifluoromethoxy-3-ethylphenyl
fluoromethyl



1.2.158
2-nitro-3-ethylphenyl
fluoromethyl



1.2.159
2-fluoro-3-propylphenyl
fluoromethyl



1.2.160
2-chloro-3-propylphenyl
fluoromethyl



1.2.161
2-bromo-3-propylphenyl
fluoromethyl



1.2.162
2-methyl-3-propylphenyl
fluoromethyl



1.2.163
2-methyl-3-propylphenyl
fluoromethyl



1.2.164
2-cyclopropyl-3-propylphenyl
fluoromethyl



1.2.165
2-vinyl-3-propylphenyl
fluoromethyl



1.2.166
2-ethynyl-3propylphenyl
fluoromethyl



1.2.167
2-cyano-3-propylphenyl
fluoromethyl



1.2.168
2-trifluoromethyl-3-propylphenyl
fluoromethyl



1.2.169
2-methoxy-3-propylphenyl
fluoromethyl



1.2.170
2-ethoxy-3-propylphenyl
fluoromethyl



1.2.171
2-trifluoromethoxy-3-propylphenyl
fluoromethyl



1.2.172
2-nitro-3-propylphenyl
fluoromethyl



1.2.173
2-fluoro-3-isopropylphenyl
fluoromethyl



1.2.174
2-chloro-3-isopropylphenyl
fluoromethyl



1.2.175
2-bromo-3-isopropylphenyl
fluoromethyl



1.2.176
2-methyl-3-isopropylphenyl
fluoromethyl



1.2.177
2-ethyl-3-isopropylphenyl
fluoromethyl



1.2.178
2-cyclopropyl-3-isopropylphenyl
fluoromethyl



1.2.179
2-vinyl-3-isopropylphenyl
fluoromethyl



1.2.180
2-ethynyl-3-isopropylphenyl
fluoromethyl



1.2.181
2-cyano-3-isopropylphenyl
fluoromethyl



1.2.182
2-trifluoromethyl-3-isopropylphenyl
fluoromethyl



1.2.183
2-methoxy-3-isopropylphenyl
fluoromethyl



1.2.184
2-ethoxy-3-isopropylphenyl
fluoromethyl



1.2.185
2-trifluoromethoxy-3-
fluoromethyl




isopropylphenyl




1.2.186
2-nitro-3-isopropylphenyl
fluoromethyl



1.2.187
2-fluoro-3-tert-butylphenyl
fluoromethyl



1.2.188
2-chloro-3-tert-butylphenyl
fluoromethyl



1.2.189
2-bromo-3-tert-butylphenyl
fluoromethyl



1.2.190
2-methyl-3-tert-butylphenyl
fluoromethyl



1.2.191
2-ethyl-3-tert-butylphenyl
fluoromethyl



1.2.192
2-cyclopropyl-3-tert-butylphenyl
fluoromethyl



1.2.193
2-vinyl-3-tert-butylphenyl
fluoromethyl



1.2.194
2-ethynyl-3-tert-butylphenyl
fluoromethyl



1.2.195
2-cyano-3-tert-butylphenyl
fluoromethyl



1.2.196
2-trifluoromethyl-3-tert-butylphenyl
fluoromethyl



1.2.197
2-methoxy-3-tert-butylphenyl
fluoromethyl



1.2.198
2-ethoxy-3-tert-butylphenyl
fluoromethyl



1.2.199
2-trifluoromethoxy-3-tert-
fluoromethyl




butylphenyl




1.2.200
2-nitro-3-tert-butylphenyl
fluoromethyl



1.2.201
2-fluoro-3-hydroxymethylphenyl
fluoromethyl



1.2.202
2-chloro-3-hydroxymethylphenyl
fluoromethyl



1.2.203
2-bromo-3-hydroxymethylphenyl
fluoromethyl



1.2.204
2-methyl-3-hydroxymethylphenyl
fluoromethyl



1.2.205
2-ethyl-3-hydroxymethylphenyl
fluoromethyl



1.2.206
2-cyclopropyl-3-
fluoromethyl




hydroxymethylphenyl




1.2.207
2-vinyl-3-hydroxymethylphenyl
fluoromethyl



1.2.208
2-ethynyl-3-hydroxymethylphenyl
fluoromethyl



1.2.209
2-cyano-3-hydroxymethylphenyl
fluoromethyl



1.2.210
2-trifluoromethyl-3-
fluoromethyl




hydroxymethylphenyl




1.2.211
2-methoxy-3-hydroxymethylphenyl
fluoromethyl



1.2.212
2-ethoxy-3-hydroxymethylphenyl
fluoromethyl



1.2.213
2-trifluoromethoxy-3-
fluoromethyl




hydroxymethylphenyl




1.2.214
2-nitro-3-hydroxymethylphenyl
fluoromethyl



1.2.215
2-fluoro-3-cyclopropylphenyl
fluoromethyl



1.2.216
2-chloro-3-cyclopropylphenyl
fluoromethyl



1.2.217
2-bromo-3-cyclopropylphenyl
fluoromethyl



1.2.218
2-methyl-3-cyclopropylphenyl
fluoromethyl



1.2.219
2-ethyl-3-cyclopropylphenyl
fluoromethyl



1.2.220
2-cyclopropyl-3-cyclopropylphenyl
fluoromethyl



1.2.221
2-vinyl-3-cyclopropylphenyl
fluoromethyl



1.2.222
2-ethynyl-3-cyclopropylphenyl
fluoromethyl



1.2.223
2-cyano-3-cyclopropylphenyl
fluoromethyl



1.2.224
2-trifluoromethyl-3-
fluoromethyl




cyclopropylphenyl




1.2.225
2-methoxy-3-cyclopropylphenyl
fluoromethyl



1.2.226
2-ethoxy-3-cyclopropylphenyl
fluoromethyl



1.2.227
2-trifluoromethoxy-3-
fluoromethyl




cyclopropylphenyl




1.2.228
2-fluoro-3-methoxycarbonylphenyl
fluoromethyl



1.2.229
2-chloro-3-methoxycarbonylphenyl
fluoromethyl



1.2.230
2-bromo-3-methoxycarbonylphenyl
fluoromethyl



1.2.231
2-methyl-3-methoxycarbonylphenyl
fluoromethyl



1.2.232
2-ethyl-3-methoxycarbonylphenyl
fluoromethyl



1.2.233
2-cyclopropyl-3-methoxycarbonyl-
fluoromethyl




phenyl




1.2.234
2-vinyl-3-methoxycarbonylphenyl
fluoromethyl



1.2.235
2-ethynyl-3-methoxycarbonyl-
fluoromethyl




phenyl




1.2.236
2-cyano-3-methoxycarbonylphenyl
fluoromethyl



1.2.237
2-trifluoromethyl-3-
fluoromethyl




methoxycarbonylphenyl




1.2.238
2-methoxy-3-methoxycarbonyl-
fluoromethyl




phenyl




1.2.239
2-ethoxy-3-methoxycarbonylphenyl
fluoromethyl



1.2.240
2-trifluoromethoxy-3-
fluoromethyl




methoxycarbonylphenyl




1.2.241
2-nitro-3-methoxycarbonylphenyl
fluoromethyl



1.2.242
2-fluoro-3-vinylphenyl
fluoromethyl



1.2.243
2-chloro-3-vinylphenyl
fluoromethyl



1.2.244
2-bromo-3-vinylphenyl
fluoromethyl



1.2.245
2-methyl-3-vinylphenyl
fluoromethyl



1.2.246
2-ethyl-3-vinylphenyl
fluoromethyl



1.2.247
2-cyclopropyl-3-vinylphenyl
fluoromethyl



1.2.248
2-vinyl-3-vinylphenyl
fluoromethyl



1.2.249
2-ethynyl-3-vinylphenyl
fluoromethyl



1.2.250
2-cyano-3-vinylphenyl
fluoromethyl



1.2.251
2-trifluoromethyl-3-vinylphenyl
fluoromethyl



1.2.252
2-methoxy-3-vinylphenyl
fluoromethyl



1.2.253
2-ethoxy-3-vinylphenyl
fluoromethyl



1.2.254
2-trifluoromethoxy-3-vinylphenyl
fluoromethyl



1.2.255
2-nitro-3-vinylphenyl
fluoromethyl



1.2.256
2-fluoro-3-ethynylphenyl
fluoromethyl



1.2.257
2-chloro-3-ethynylphenyl
fluoromethyl



1.2.258
2-bromo-3-ethynylphenyl
fluoromethyl



1.2.259
2-methyl-3-ethynylphenyl
fluoromethyl



1.2.260
2-ethyl-3-ethynylphenyl
fluoromethyl



1.2.261
2-cyclopropyl-3-ethynylphenyl
fluoromethyl



1.2.262
2-vinyl-3-ethynylphenyl
fluoromethyl



1.2.263
2-cyano-3-ethynylphenyl
fluoromethyl



1.2.264
2-trifluoromethyl-3-ethynylphenyl
fluoromethyl



1.2.265
2-methoxy-3-ethynylphenyl
fluoromethyl



1.2.266
2-ethoxy-3-ethynylphenyl
fluoromethyl



1.2.267
2-trifluoromethoxy-3-ethynylphenyl
fluoromethyl



1.2.268
2-nitro-3-ethynylphenyl
fluoromethyl



1.2.269
2-fluoro-3-ethynylphenyl
fluoromethyl



1.2.270
2-fluoro-3-cyanophenyl
fluoromethyl



1.2.271
2-chloro-3-cyanophenyl
fluoromethyl



1.2.272
2-bromo-3-cyanophenyl
fluoromethyl



1.2.273
2-methyl-3-cyanophenyl
fluoromethyl



1.2.274
2-ethyl-3-cyanophenyl
fluoromethyl



1.2.275
2-ethyl-3-cyanophenyl
chloromethyl



1.2.276
2-ethyl-3-cyanophenyl
bromomethyl



1.2.277
2-ethyl-3-cyanophenyl
difluoromethyl



1.2.278
2-cyclopropyl-3-cyanophenyl
fluoromethyl



1.2.279
2-vinyl-3-cyanophenyl
fluoromethyl



1.2.280
2-ethynyl-3-cyanophenyl
fluoromethyl



1.2.281
2-cyano-3-cyanophenyl
fluoromethyl



1.2.282
2-trifluoromethyl-3-cyanophenyl
fluoromethyl



1.2.283
2-methoxy-3-cyanophenyl
fluoromethyl



1.2.284
2-ethoxy-3-cyanophenyl
fluoromethyl



1.2.285
2-trifluoromethoxy-3-cyanophenyl
fluoromethyl



1.2.286
2-nitro-3-cyanophenyl
fluoromethyl



1.2.287
2-fluoro-3-hydroxyphenyl
fluoromethyl



1.2.288
2-chloro-3-hydroxyphenyl
fluoromethyl



1.2.289
2-bromo-3-hydroxyphenyl
fluoromethyl



1.2.290
2-methyl-3-hydroxyphenyl
fluoromethyl



1.2.291
2-ethyl-3-hydroxyphenyl
fluoromethyl



1.2.292
2-cyclopropyl-3-hydroxyphenyl
fluoromethyl



1.2.293
2-vinyl-3-hydroxyphenyl
fluoromethyl



1.2.294
2-ethynyl-3-hydroxyphenyl
fluoromethyl



1.2.295
2-cyano-3-hydroxyphenyl
fluoromethyl



1.2.296
2-trifluoromethyl-3-hydroxyphenyl
fluoromethyl



1.2.297
2-methoxy-3-hydroxyphenyl
fluoromethyl



1.2.298
2-ethoxy-3-hydroxyphenyl
fluoromethyl



1.2.299
2-trifluoromethoxy-3-hydroxyphenyl
fluoromethyl



1.2.300
2-nitro-3-hydroxyphenyl
fluoromethyl



1.2.301
2-fluoro-3-methoxyphenyl
fluoromethyl



1.2.302
2-chloro-3-methoxyphenyl
fluoromethyl



1.2.303
2-bromo-3-methoxyphenyl
fluoromethyl



1.2.304
2-methyl-3-methoxyphenyl
fluoromethyl



1.2.305
2-ethyl-3-methoxyphenyl
fluoromethyl



1.2.306
2-cyclopropyl-3-methoxyphenyl
fluoromethyl



1.2.307
2-vinyl-3-methoxyphenyl
fluoromethyl



1.2.308
2-ethynyl-3-methoxyphenyl
fluoromethyl



1.2.309
2-cyano-3-methoxyphenyl
fluoromethyl



1.2.310
2-trifluoromethyl-3-methoxyphenyl
fluoromethyl



1.2.311
2,3-dimethoxy--phenyl
fluoromethyl



1.2.312
2-ethoxy-3-methoxyphenyl
fluoromethyl



1.2.313
2-trifluoromethoxy-3-
fluoromethyl




methoxyphenyl




1.2.314
2-nitro-3-methoxyphenyl
fluoromethyl



1.2.315
2-fluoro-3-ethoxyphenyl
fluoromethyl



1.2.316
2-chloro-3-ethoxyphenyl
fluoromethyl



1.2.317
2-bromo-3-ethoxyphenyl
fluoromethyl



1.2.318
2-methyl-3-ethoxyphenyl
fluoromethyl



1.2.319
2-ethyl-3-ethoxyphenyl
fluoromethyl



1.2.320
2-cyclopropyl-3-ethoxyphenyl
fluoromethyl



1.2.321
2-vinyl-3-ethoxyphenyl
fluoromethyl



1.2.322
2-ethynyl-3-ethoxyphenyl
fluoromethyl



1.2.323
2-cyano-3-ethoxyphenyl
fluoromethyl



1.2.324
2-trifluoromethyl-3-ethoxyphenyl
fluoromethyl



1.2.325
2-methoxy-3-ethoxyphenyl
fluoromethyl



1.2.326
2,3-diethoxy--phenyl
fluoromethyl



1.2.327
2-trifluoromethoxy-3-ethoxyphenyl
fluoromethyl



1.2.328
2-nitro-3-ethoxyphenyl
fluoromethyl



1.2.329
2-fluoro-3-propoxyphenyl
fluoromethyl



1.2.330
2-chloro-3-propoxyphenyl
fluoromethyl



1.2.331
2-bromo-3-propoxyphenyl
fluoromethyl



1.2.332
2-methyl-3-propoxyphenyl
fluoromethyl



1.2.333
2-ethyl-3-propoxyphenyl
fluoromethyl



1.2.334
2-cyclopropyl-3-propoxyphenyl
fluoromethyl



1.2.335
2-vinyl-3-propoxyphenyl
fluoromethyl



1.2.336
2-ethynyl-3-propoxyphenyl
fluoromethyl



1.2.337
2-cyano-3-propoxyphenyl
fluoromethyl



1.2.338
2-trifluoromethyl-3-propoxyphenyl
fluoromethyl



1.2.339
2-methoxy-3-propoxyphenyl
fluoromethyl



1.2.340
2-ethoxy-3-propoxyphenyl
fluoromethyl



1.2.341
2-trifluoromethoxy-3-propoxyphenyl
fluoromethyl



1.2.342
2-nitro-3-propoxyphenyl
fluoromethyl



1.2.343
2-fluoro-3-isopropoxyphenyl
fluoromethyl



1.2.344
2-chloro-3-isopropoxyphenyl
fluoromethyl



1.2.345
2-bromo-3-isopropoxyphenyl
fluoromethyl



1.2.346
2-methyl-3-isopropoxyphenyl
fluoromethyl



1.2.347
2-ethyl-3-isopropoxyphenyl
fluoromethyl



1.2.348
2-cyclopropyl-3-isopropoxyphenyl
fluoromethyl



1.2.349
2-vinyl-3-isopropoxyphenyl
fluoromethyl



1.2.350
2-ethynyl-3-isopropoxyphenyl
fluoromethyl



1.2.351
2-cyano-3-isopropoxyphenyl
fluoromethyl



1.2.352
2-trifluoromethyl-3-
fluoromethyl




isopropoxyphenyl




1.2.353
2-methoxy-3-isopropoxyphenyl
fluoromethyl



1.2.354
2-ethoxy-3-isopropoxyphenyl
fluoromethyl



1.2.355
2-trifluoromethoxy-3-
fluoromethyl




isopropoxyphenyl




1.2.356
2-nitro-3-isopropoxyphenyl
fluoromethyl



1.2.357
2-fluoro-3-tert-butoxyphenyl
fluoromethyl



1.2.358
2-chloro-3-tert-butoxyphenyl
fluoromethyl



1.2.359
2-bromo-3-tert-butoxyphenyl
fluoromethyl



1.2.360
2-methyl-3-tert-butoxyphenyl
fluoromethyl



1.2.361
2-ethyl-3-tert-butoxyphenyl
fluoromethyl



1.2.362
2-cyclopropyl-3-tert-butoxyphenyl
fluoromethyl



1.2.363
2-vinyl-3-tert-butoxyphenyl
fluoromethyl



1.2.364
2-ethynyl-3-tert-butoxyphenyl
fluoromethyl



1.2.365
2-cyano-3-tert-butoxyphenyl
fluoromethyl



1.2.366
2-trifluoromethyl-3-tert-
fluoromethyl




butoxyphenyl




1.2.367
2-methoxy-3-tert-butoxyphenyl
fluoromethyl



1.2.368
2-ethoxy-3-tert-butoxyphenyl
fluoromethyl



1.2.369
2-trifluoromethoxy-3-tert-
fluoromethyl




butoxyphenyl




1.2.370
2-nitro-3-tert-butoxyphenyl
fluoromethyl



1.2.371
2-fluoro-3-trifluoromethoxyphenyl
fluoromethyl



1.2.372
2-chloro-3-trifluoromethoxyphenyl
fluoromethyl



1.2.373
2-bromo-3-trifluoromethoxyphenyl
fluoromethyl



1.2.374
2-methyl-3-trifluoromethoxyphenyl
fluoromethyl



1.2.375
2-ethyl-3-trifluoromethoxyphenyl
fluoromethyl



1.2.376
2-cyclopropyl-3-trifluoromethoxy-
fluoromethyl




phenyl




1.2.377
2-vinyl-3-trifluoromethoxyphenyl
fluoromethyl



1.2.378
2-ethynyl-3-trifluoromethoxyphenyl
fluoromethyl



1.2.379
2-cyano-3-trifluoromethoxyphenyl
fluoromethyl



1.2.380
2-trifluoromethyl-3-trifluoromethoxy-
fluoromethyl




phenyl




1.2.381
2-methoxy-3-trifluoromethoxy-
fluoromethyl




phenyl




1.2.382
2-ethoxy-3-trifluoromethoxyphenyl
fluoromethyl



1.2.383
2,3-bis(trifluoromethoxy)phenyl
fluoromethyl



1.2.384
2-nitro-3-trifluoromethoxyphenyl
fluoromethyl



1.2.385
2-fluoro-3-(2,2,2-trifluoroethoxy)-
fluoromethyl




phenyl




1.2.386
2-chloro-3-(2,2,2-trifluoroethoxy)-
fluoromethyl




phenyl




1.2.387
2-bromo-3-(2,2,2-trifluoroethoxy)-
fluoromethyl




phenyl




1.2.388
2-methyl-3-(2,2,2-trifluoroethoxy)-
fluoromethyl




phenyl




1.2.389
2-ethyl-3-(2,2,2(2,2,2-trifluoroethoxy)-
fluoromethyl




phenyl




1.2.390
2-cyclopropyl-3-(2,2,2-trifluoro-
fluoromethyl




ethoxy)phenyl




1.2.391
2-vinyl-3-(2,2,2-trifluoroethoxy)-
fluoromethyl




phenyl




1.2.392
2-ethynyl-3-(2,2,2-
fluoromethyl




trifluoroethoxyphenyl




1.2.393
2-cyano-3-(2,2,2-trifluoroethoxy)-
fluoromethyl




phenyl




1.2.394
2-trifluoromethyl-3-(2,2,2-trifluoro-
fluoromethyl




ethoxy)phenyl




1.2.395
2-methoxy-3-(2,2,2-trifluoroethoxy)-
fluoromethyl




phenyl




1.2.396
2-ethoxy-3-(2,2,2-trifluoroethoxy)-
fluoromethyl




phenyl




1.2.397
2-trifluoromethoxy-3-(2,2,2-trifluoro-
fluoromethyl




ethoxy)phenyl




1.2.398
2-nitro-3-(2,2,2-trifluoroethoxy)-
fluoromethyl




phenyl




1.2.399
2-fluoro-3-difluoromethoxyphenyl
fluoromethyl



1.2.400
2-chloro-3-difluoromethoxyphenyl
fluoromethyl



1.2.401
2-bromo-3-difluoromethoxyphenyl
fluoromethyl



1.2.402
2-methyl-3-difluoromethoxyphenyl
fluoromethyl



1.2.403
2-ethyl-3-difluoromethoxyphenyl
fluoromethyl



1.2.404
2-cyclopropyl-3-difluoromethoxy-
fluoromethyl




phenyl




1.2.405
2-vinyl-3-difluoromethoxyphenyl
fluoromethyl



1.2.406
2-ethynyl-3-difluoromethoxyphenyl
fluoromethyl



1.2.407
2-cyano-3-difluoromethoxyphenyl
fluoromethyl



1.2.408
2-trifluoromethyl-3-difluoromethoxy-
fluoromethyl




phenyl




1.2.409
2-methoxy-3-difluoromethoxy-
fluoromethyl




phenyl




1.2.410
2-ethoxy-3-difluoromethoxyphenyl
fluoromethyl



1.2.411
2-trifluoromethoxy-3-
fluoromethyl




difluoromethoxyphenyl




1.2.412
2-nitro-3-difluoromethoxyphenyl
fluoromethyl



1.2.413
2-fluoro-3-(2-methoxyethoxy)-
fluoromethyl




phenyl




1.2.414
2-chloro-3-(2-methoxyethoxy)-
fluoromethyl




phenyl




1.2.415
2-bromo-3-(2-methoxyethoxy)-
fluoromethyl




phenyl




1.2.416
2-methyl-3-(2-methoxyethoxy)-
fluoromethyl




phenyl




1.2.417
2-ethyl-3-(2-methoxyethoxy)phenyl
fluoromethyl



1.2.418
2-cyclopropyl-3-(2-methoxyethoxy)-
fluoromethyl




phenyl




1.2.419
2-vinyl-3-(2-methoxyethoxy)phenyl
fluoromethyl



1.2.420
2-ethynyl-3-(2-methoxyethoxy)-
fluoromethyl




phenyl




1.2.421
2-cyano-3-(2-methoxyethoxy)-
fluoromethyl




phenyl




1.2.422
2-trifluoromethyl-3-(2-
fluoromethyl




methoxyethoxy)-phenyl




1.2.423
2-methoxy-3-(2-methoxyethoxy)-
fluoromethyl




phenyl




1.2.424
2-ethoxy-3-(2-methoxyethoxy)-
fluoromethyl




phenyl




1.2.425
2-trifluoromethoxy-(2-
fluoromethyl




methoxyethoxy)-phenyl




1.2.426
2-nitro-3-(2-methoxyethoxy)phenyl
fluoromethyl



1.2.427
2-fluoro-3-(tert-butoxycarbonyloxy)-
fluoromethyl




phenyl




1.2.428
2-chloro-3-(tert-butoxycarbonyloxy)-
fluoromethyl




phenyl




1.2.429
2-bromo-3-(tert-butoxycarbonyl-
fluoromethyl




oxy)phenyl




1.2.430
2-methyl-3-(tert-butoxycarbonyl-
fluoromethyl




oxy)phenyl




1.2.431
2-ethyl-3-(tert-butoxycarbonyloxy)-
fluoromethyl




phenyl




1.2.432
2-cyclopropyl-3-(tert-butoxy-
fluoromethyl




carbonyloxy)phenyl




1.2.433
2-vinyl-3-(tert-butoxycarbonyloxy)-
fluoromethyl




phenyl




1.2.434
2-ethynyl-3-(tert-butoxycarbonyl-
fluoromethyl




oxy)phenyl




1.2.435
2-cyano-3-(tert-butoxycarbonyloxy)-
fluoromethyl




phenyl




1.2.436
2-trifluoromethyl-3-(tert-butoxy-
fluoromethyl




carbonyloxy)phenyl




1.2.437
2-methoxy-3-(tert-butoxycarbonyl-
fluoromethyl




oxy)phenyl




1.2.438
2-ethoxy-3-(tert-butoxycarbonyl-
fluoromethyl




oxy)phenyl




1.2.439
2-trifluoromethoxy-3-(tert-
fluoromethyl




butoxycarbonyl-oxy)phenyl




1.2.440
2-nitro-3-(tert-butoxycarbonyloxy)-
fluoromethyl




phenyl




1.2.441
2-fluoro-3-nitrophenyl
fluoromethyl



1.2.442
2-chloro-3-nitrophenyl
fluoromethyl



1.2.443
2-bromo-3-nitrophenyl
fluoromethyl



1.2.444
2-methyl-3-nitrophenyl
fluoromethyl



1.2.445
2-ethyl-3-nitrophenyl
fluoromethyl



1.2.446
2-cyclopropyl-3-nitrophenyl
fluoromethyl



1.2.447
2-vinyl-3-nitrophenyl
fluoromethyl



1.2.448
2-ethynyl-3-nitrophenyl
fluoromethyl



1.2.449
2-cyano-3-nitrophenyl
fluoromethyl



1.2.450
2-trifluoromethyl-3-nitrophenyl
fluoromethyl



1.2.451
2-methoxy-3-nitrophenyl
fluoromethyl



1.2.452
2-ethoxy-3-nitrophenyl
fluoromethyl



1.2.453
2-trifluoromethoxy-3-nitrophenyl
fluoromethyl



1.2.454
2-fluoro-3-methylsulfanylphenyl
fluoromethyl



1.2.455
2-chloro-3-methylsulfanylphenyl
fluoromethyl



1.2.456
2-bromo-3-methylsulfanylphenyl
fluoromethyl



1.2.457
2-methyl-3-methylsulfanylphenyl
fluoromethyl



1.2.458
2-ethyl-3-methylsulfanylphenyl
fluoromethyl



1.2.459
2-cyclopropyl-3-
fluoromethyl




methylsulfanylphenyl




1.2.460
2-vinyl-3-methylsulfanylphenyl
fluoromethyl



1.2.461
2-ethynyl-3-methylsulfanylphenyl
fluoromethyl



1.2.462
2-cyano-3-methylsulfanylphenyl
fluoromethyl



1.2.463
2-trifluoromethyl-3-
fluoromethyl




methylsulfanylphenyl




1.2.464
2-methoxy-3-methylsulfanylphenyl
fluoromethyl



1.2.465
2-ethoxy-3-methylsulfanylphenyl
fluoromethyl



1.2.466
2-trifluoromethoxy-3-
fluoromethyl




methylsulfanylphenyl




1.2.467
2-nitro-3-methylsulfanylphenyl
fluoromethyl



1.2.468
3,5-difluorophenyl
fluoromethyl
[CDCl3] 3.56 (d,1H); 3.80





(d,1H); 4.72 (s, 1H); 4.84





(s,1H); 6.0 (s br, 1H); 6.92





(t,1H); 7.19 (d,2H).


1.2.469
3,5-difluorophenyl
chloromethyl
[CDCl3] 3.57 (d,1H); 3.88





( s,1H), 3.92 (d, 1H); 4.03





(d,1H), 6.93 (t,1H); 7.21





(d,2H).


1.2.470
3,5-difluorophenyl
bromomethyl
[CDCl3] 3.56 (d,1H); 3.71





(d,1H); 3.91 (d,1H); 3.96





(d,1H); 6.91 (t,1H); 7.18





(d,2H).


1.2.471
3,5-difluorophenyl
difluoromethyl
[CDCl3] 3.69 (d,1H); 3.91





(d,1H); 6.10-6.40 (s,1H);





6.92 (m,1H); 7.22 (m,2H).


1.2.472
3,5-difluorophenyl
trifluoromethyl



1.2.473
3,5-difluorophenyl
1,1-
[CDCl3] 2.40 (s,3H); 3.93




dichloroethyl
(d,1H, 4.00 (d,1H); 6.94





(t,1H) 7.21 (d,2H).


1.2.474
3,5-difluorophenyl
CN
[CDCl3] 3.97 (d,1H); 4.14





(d,1H); 6.97 (m,1H); 7.21





(m,2H).


1.2.475
3-chloro-5-fluorophenyl
fluoromethyl



1.2.476
3-chloro-5-fluorophenyl
chloromethyl



1.2.477
3-chloro-5-fluorophenyl
bromomethyl



1.2.478
3-chloro-5-fluorophenyl
difluoromethyl



1.2.479
3-bromo-5-fluorophenyl
fluoromethyl



1.2.480
3-bromo-5-fluorophenyl
chloromethyl



1.2.481
3-bromo-5-fluorophenyl
bromomethyl



1.2.482
3-bromo-5-fluorophenyl
difluoromethyl



1.2.483
3-iodo-5-fluorophenyl
fluoromethyl



1.2.484
3-methyl-5-fluorophenyl
fluoromethyl



1.2.485
3-methyl-5-fluorophenyl
chloromethyl



1.2.486
3-methyl-5-fluorophenyl
bromomethyl



1.2.487
3-methyl-5-fluorophenyl
difluoromethyl



1.2.488
3-ethyl-5-fluorophenyl
fluoromethyl



1.2.489
3-propyl-5-fluorophenyl
fluoromethyl



1.2.490
3-i-propyl-5-fluorophenyl
fluoromethyl



1.2.491
3-n-butyl-5-fluorophenyl
fluoromethyl



1.2.492
3-isobutyl-5-fluorophenyl
fluoromethyl



1.2.493
3-tert-butyl-5-fluorophenyl
fluoromethyl



1.2.494
3-cyclopropyl-5-fluorophenyl
fluoromethyl



1.2.495
3-vinyl-5-fluorophenyl
fluoromethyl



1.2.496
3-ethynyl-5-fluorophenyl
fluoromethyl



1.2.497
3-cyano-5-fluorophenyl
fluoromethyl



1.2.498
3-trifluoromethyl-5-fluorophenyl
fluoromethyl



1.2.499
3-trifluoromethyl-5-fluorophenyl
chloromethyl



1.2.500
3-trifluoromethyl-5-fluorophenyl
bromomethyl



1.2.501
3-trifluoromethyl-5-fluorophenyl
difluoromethyl



1.2.502
3-(methoxycarbonyl)-5-fluorophenyl
fluoromethyl



1.2.503
3-hydroxymethyl-5-fluorophenyl
fluoromethyl



1.2.504
3-carbamoyl-5-fluorophenyl
fluoromethyl



1.2.505
3-hydroxy-5-fluorophenyl
fluoromethyl



1.2.506
3-methoxy-5-fluorophenyl
fluoromethyl



1.2.507
3-ethoxy-5-fluorophenyl
fluoromethyl



1.2.508
3-n-propoxy-5-fluorophenyl
fluoromethyl



1.2.509
3-isopropoxy-5-fluorophenyl
fluoromethyl



1.2.510
3-n-butoxy-5-fluorophenyl
fluoromethyl



1.2.511
3-isobutoxy-5-fluorophenyl
fluoromethyl



1.2.512
3-tert-butoxy-5-fluorophenyl
fluoromethyl



1.2.513
3-difluoromethoxy-5-fluorophenyl
fluoromethyl



1.2.514
3-trifluoromethoxy-5-fluorophenyl
fluoromethyl



1.2.515
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl




fluorophenyl




1.2.516
3-(2-chloroethoxy)-5-fluorophenyl
fluoromethyl



1.2.517
3-(2-hydroxyethoxy)-5-fluorophenyl
fluoromethyl



1.2.518
3-[(tert-butoxycarbonyl)oxy]-5-
fluoromethyl




fluorophenyl




1.2.519
3-nitro-5-fluorophenyl
fluoromethyl



1.2.520
3-acetoxy-5-fluorophenyl
fluoromethyl



1.2.521
{3-[(tert-butoxycarbonyl)amino]-5-
fluoromethyl




fluorophenyl}




1.2.522
3-methylsulfanyl-5-fluorophenyl
fluoromethyl



1.2.523
3,5-dichlorophenyl
fluoromethyl



1.2.524
3,5-dichlorophenyl
chloromethyl
[CDCl3] 3.59 (d, 1H); 3.88 (d,





1H); 3.91 (d, 1H); 4.03 (d,





1H); 7.45 (m, 1H); 7.58 (m,





1H).


1.2.525
3,5-dichlorophenyl
bromomethyl
[CDCl3] 3.55 (d, 1H); 3.71 (d,





1H); 3.90 (d, 1H); 3.96 (d,





1H); 7.45 (s, 1H); 7.55 (s,





2H).


1.2.526
3,5-dichlorophenyl
difluoromethyl



1.2.527
3,5-dichlorophenyl
trifluoromethyl
[CDCl3] 3.8 (d, 1H); 4.0 (d,





1H); 7.45 (m, 1H); 7.55 (m,





1H).


1.2.528
3,5-dichlorophenyl
cyano
[DMSO] 3.87 (d, 1H); 4.02





(d, 1H); 7.74 (m, 3H).


1.2.529
3-bromo-5-chlorophenyl
fluoromethyl



1.2.530
3-iodo-5-chlorophenyl
fluoromethyl



1.2.531
3-methyl-5-chlorophenyl
fluoromethyl



1.2.532
3-ethyl-5-chlorophenyl
fluoromethyl



1.2.533
3-propyl-5-chlorophenyl
fluoromethyl



1.2.534
3-isopropyl-5-chlorophenyl
fluoromethyl



1.2.535
3-n-butyl-5-chlorophenyl
fluoromethyl



1.2.536
3-isobutyl-5-chlorophenyl
fluoromethyl



1.2.537
3-tert-butyl-5-chlorophenyl
fluoromethyl



1.2.538
3-cyclopropyl-5-chlorophenyl
fluoromethyl



1.2.539
3-vinyl-5-chlorophenyl
fluoromethyl



1.2.540
3-ethynyl-5-chlorophenyl
fluoromethyl



1.2.541
3-cyano-5-chlorophenyl
fluoromethyl



1.2.542
3-trifluoromethyl-5-chlorophenyl
fluoromethyl



1.2.543
3-(hydroxycarbonyl)-5-chlorophenyl
fluoromethyl



1.2.544
3-(methoxycarbonyl)-5-
fluoromethyl




chlorophenyl




1.2.545
3-hydroxymethyl-5-chlorophenyl
fluoromethyl



1.2.546
3-carbamoyl-5-chlorophenyl
fluoromethyl



1.2.547
3-hydroxy-5-chlorophenyl
fluoromethyl



1.2.548
3-methoxy-5-chlorophenyl
fluoromethyl



1.2.549
3-ethoxy-5-chlorophenyl
fluoromethyl



1.2.550
3-n-propoxy-5-chlorophenyl
fluoromethyl



1.2.551
3-isopropoxy-5-chlorophenyl
fluoromethyl



1.2.552
3-n-butoxy-5-chlorophenyl
fluoromethyl



1.2.553
3-isobutoxy-5-chlorophenyl
fluoromethyl



1.2.554
3-tert-butoxy-5-chlorophenyl
fluoromethyl



1.2.555
3-difluoromethoxy-5-chlorophenyl
fluoromethyl



1.2.556
3-trifluoromethoxy-5-chlorophenyl
fluoromethyl



1.2.557
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl




chlorophenyl




1.2.558
3-(2-chloroethoxy)-5-chlorophenyl
fluoromethyl



1.2.559
3-(2-hydroxyethoxy)-5-chlorophenyl
fluoromethyl



1.2.560
3-[(tert-butoxycarbonyl)oxy]-5-
fluoromethyl




chlorophenyl




1.2.561
3-nitro-5-chlorophenyl
fluoromethyl



1.2.562
3-acetoxy-5-chlorophenyl
fluoromethyl



1.2.563
{3-[(tert-butoxycarbonyl)amino]-5-
fluoromethyl




chlorophenyl}




1.2.564
3-methylsulfanyl-5-chlorophenyl
fluoromethyl



1.2.565
3,5-dibromophenyl
fluoromethyl



1.2.566
3,5-dibromophenyl
chloromethyl



1.2.567
3-iodo-5-bromophenyl
fluoromethyl



1.2.568
3-methyl-5-bromophenyl
fluoromethyl



1.2.569
3-methyl-5-bromophenyl
chloromethyl



1.2.570
3-methyl-5-bromophenyl
bromomethyl



1.2.571
3-methyl-5-bromophenyl
difluoromethyl



1.2.572
3-methyl-5-bromophenyl
trifluoromethyl



1.2.573
3-methyl-5-bromophenyl
cyano



1.2.574
3-ethyl-5-bromophenyl
fluoromethyl



1.2.575
3-propyl-5-bromophenyl
fluoromethyl



1.2.576
3-isopropyl-5-bromophenyl
fluoromethyl



1.2.577
3-n-butyl-5-bromophenyl
fluoromethyl



1.2.578
3-isobutyl-5-bromophenyl
fluoromethyl



1.2.579
3-tert-butyl-5-bromophenyl
fluoromethyl



1.2.580
3-cyclopropyl-5-bromophenyl
fluoromethyl



1.2.581
3-vinyl-5-bromophenyl
fluoromethyl



1.2.582
3-ethynyl-5-bromophenyl
fluoromethyl



1.2.583
3-cyano-5-bromophenyl
fluoromethyl



1.2.584
3-trifluoromethyl-5-bromophenyl
fluoromethyl



1.2.585
3-(hydroxycarbonyl)-5-bromophenyl
fluoromethyl



1.2.586
3-(methoxycarbonyl)-5-
fluoromethyl




bromophenyl




1.2.587
3-hydroxymethyl-5-bromophenyl
fluoromethyl



1.2.588
3-carbamoyl-5-bromophenyl
fluoromethyl



1.2.589
3-hydroxy-5-bromophenyl
fluoromethyl



1.2.590
3-methoxy-5-bromophenyl
fluoromethyl



1.2.591
3-ethoxy-5-bromophenyl
fluoromethyl



1.2.592
3-n-propoxy-5-bromophenyl
fluoromethyl



1.2.593
3-isopropoxy-5-bromophenyl
fluoromethyl



1.2.594
3-n-butoxy-5-bromophenyl
fluoromethyl



1.2.595
3-isobutoxy-5-bromophenyl
fluoromethyl



1.2.596
3-tert-butoxy-5-bromophenyl
fluoromethyl



1.2.597
3-difluoromethoxy-5-bromophenyl
fluoromethyl



1.2.598
3-trifluoromethoxy-5-bromophenyl
fluoromethyl



1.2.599
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl




bromophenyl




1.2.600
3-(2-chloroethoxy)-5-bromophenyl
fluoromethyl



1.2.601
3-(2-hydroxyethoxy)-5-bromophenyl
fluoromethyl



1.2.602
3-[(tert-butoxycarbonyl)oxy]-5-
fluoromethyl




bromophenyl




1.2.603
3-nitro-5-bromophenyl
fluoromethyl



1.2.604
3-acetoxy-5-bromophenyl
fluoromethyl



1.2.605
{3-[(tert-butoxy-carbonyl)amino]-5-
fluoromethyl




bromophenyl}




1.2.606
3-methylsulfanyl-5-bromophenyl
fluoromethyl



1.2.607
3,5-diiodophenyl
fluoromethyl



1.2.608
3-methyl-5-iodophenyl
fluoromethyl



1.2.609
3-ethyl-5-iodophenyl
fluoromethyl



1.2.610
3-propyl-5-iodophenyl
fluoromethyl



1.2.611
3-isopropyl-5-iodophenyl
fluoromethyl



1.2.612
3-n-butyl-5-iodophenyl
fluoromethyl



1.2.613
3-isobutyl-5-iodophenyl
fluoromethyl



1.2.614
3-tert-butyl-5-iodophenyl
fluoromethyl



1.2.615
3-cyclopropyl-5-iodophenyl
fluoromethyl



1.2.616
3-vinyl-5-iodophenyl
fluoromethyl



1.2.617
3-ethynyl-5-iodophenyl
fluoromethyl



1.2.618
3-cyano-5-iodophenyl
fluoromethyl



1.2.619
3-trifluoromethyl-5-iodophenyl
fluoromethyl



1.2.620
3-(hydroxycarbonyl)-5-iodophenyl
fluoromethyl



1.2.621
3-(methoxycarbonyl)-5-iodophenyl
fluoromethyl



1.2.622
3-hydroxymethyl-5-iodophenyl
fluoromethyl



1.2.623
3-carbamoyl-5-iodophenyl
fluoromethyl



1.2.624
3-hydroxy-5-iodophenyl
fluoromethyl



1.2.625
3-methoxy-5-iodophenyl
fluoromethyl



1.2.626
3-ethoxy-5-iodophenyl
fluoromethyl



1.2.627
3-n-propoxy-5-iodophenyl
fluoromethyl



1.2.628
3-isopropoxy-5-iodophenyl
fluoromethyl



1.2.629
3-n-butoxy-5-iodophenyl
fluoromethyl



1.2.630
3-isobutoxy-5-iodophenyl
fluoromethyl



1.2.631
3-tert-butoxy-5-iodophenyl
fluoromethyl



1.2.632
3-difluoromethoxy-5-iodophenyl
fluoromethyl



1.2.633
3-trifluoromethoxy-5-iodophenyl
fluoromethyl



1.2.634
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl




iodophenyl




1.2.635
3-(2-chloroethoxy)-5-iodophenyl
fluoromethyl



1.2.636
3-(2-hydroxyethoxy)-5-iodophenyl
fluoromethyl



1.2.637
3-[tert-butoxycarbonyl)oxy]-5-
fluoromethyl




iodophenyl




1.2.638
3-nitro-5-iodophenyl
fluoromethyl



1.2.639
3-acetoxy-5-iodophenyl
fluoromethyl



1.2.640
(3-[(tert-butoxy-carbonyl)amino]-5-
fluoromethyl




iodophenyl}




1.2.641
3-methylsulfanyl-5-iodophenyl
fluoromethyl



1.2.642
3,5-dimethylphenyl
fluoromethyl



1.2.643
3-ethyl-5-methylphenyl
fluoromethyl



1.2.644
3-propyl-5-methylphenyl
fluoromethyl



1.2.645
3-isopropyl-5-methylphenyl
fluoromethyl



1.2.646
3-n-butyl-5-methylphenyl
fluoromethyl



1.2.647
3-isobutyl-5-methylphenyl
fluoromethyl



1.2.648
3-tert-butyl-5-methylphenyl
fluoromethyl



1.2.649
3-cyclopropyl-5-methylphenyl
fluoromethyl



1.2.650
3-vinyl-5-methylphenyl
fluoromethyl



1.2.651
3-ethynyl-5-methylphenyl
fluoromethyl



1.2.652
3-cyano-5-methylphenyl
fluoromethyl



1.2.653
3-trifluoromethyl-5-methylphenyl
fluoromethyl



1.2.654
3-(hydroxycarbonyl)-5-
fluoromethyl




methylphenyl




1.2.655
3-(methoxycarbonyl)-5-
fluoromethyl




methylphenyl




1.2.656
3-hydroxymethyl-5-methylphenyl
fluoromethyl



1.2.657
3-carbamoyl-5-methylphenyl
fluoromethyl



1.2.658
3-hydroxy-5-methylphenyl
fluoromethyl



1.2.659
3-methoxy-5-methylphenyl
fluoromethyl



1.2.660
3-ethoxy-5-methylphenyl
fluoromethyl



1.2.661
3-n-propoxy-5-methylphenyl
fluoromethyl



1.2.662
3-n-butoxy-5-methylphenyl
fluoromethyl



1.2.663
3-isobutoxy-5-methylphenyl
fluoromethyl



1.2.664
3-tert-butoxy-5-methylphenyl
fluoromethyl



1.2.665
3-difluoromethoxy-5-methylphenyl
fluoromethyl



1.2.666
3-trifluoromethoxy-5-methylphenyl
fluoromethyl



1.2.667
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl




methylphenyl




1.2.668
3-(2-chloroethoxy)-5-methylphenyl
fluoromethyl



1.2.669
3-(2-hydroxyethoxy)-5-
fluoromethyl




methylphenyl




1.2.670
3-[tert-butoxycarbonyl)oxy]-5-
fluoromethyl




methylphenyl




1.2.671
3-nitro-5-methylphenyl
fluoromethyl



1.2.672
3-acetoxy-5-methylphenyl
fluoromethyl



1.2.673
{3-[(tert-butoxycarbonyl)amino]-5-
fluoromethyl




methylphenyl}




1.2.674
3-methylsulfanyl-5-methylphenyl
fluoromethyl



1.2.675
3,5-diethylphenyl
fluoromethyl



1.2.676
3-propyl-5-ethylphenyl
fluoromethyl



1.2.677
3-isopropyl-5-ethylphenyl
fluoromethyl



1.2.678
3-n-butyl-5-ethylphenyl
fluoromethyl



1.2.679
3-isobutyl-5-ethylphenyl
fluoromethyl



1.2.680
3-tert-butyl-5-ethylphenyl
fluoromethyl



1.2.681
3-cyclopropyl-5-ethylphenyl
fluoromethyl



1.2.682
3-vinyl-5-ethylphenyl
fluoromethyl



1.2.683
3-ethynyl-5-ethylphenyl
fluoromethyl



1.2.684
3-cyano-5-ethylphenyl
fluoromethyl



1.2.685
3-trifluoromethyl-5-ethylphenyl
fluoromethyl



1.2.686
3-(hydroxycarbonyl)-5-ethylphenyl
fluoromethyl



1.2.687
3-(methoxycarbonyl)-5-ethylphenyl
fluoromethyl



1.2.688
3-hydroxymethyl-5-ethylphenyl
fluoromethyl



1.2.689
3-carbamoyl-5-ethylphenyl
fluoromethyl



1.2.690
3-hydroxy-5-ethylphenyl
fluoromethyl



1.2.691
3-methoxy-5-ethylphenyl
fluoromethyl



1.2.692
3-ethoxy-5-ethylphenyl
fluoromethyl



1.2.693
3-n-propoxy-5-ethylphenyl
fluoromethyl



1.2.694
3-n-butoxy-5-ethylphenyl
fluoromethyl



1.2.695
3-isobutoxy-5-ethylphenyl
fluoromethyl



1.2.696
3-tert-butoxy-5-ethylphenyl
fluoromethyl



1.2.697
3-difluoromethoxy-5-ethylphenyl
fluoromethyl



1.2.698
3-trifluoromethoxy-5-ethylphenyl
fluoromethyl



1.2.699
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl




ethylphenyl




1.2.700
3-(2-chloroethoxy)-5-ethylphenyl
fluoromethyl



1.2.701
3-(2-hydroxyethoxy)-5-ethylphenyl
fluoromethyl



1.2.702
3-[tert-butoxycarbonyl)oxy]-5-
fluoromethyl




ethylphenyl




1.2.703
3-nitro-5-ethylphenyl
fluoromethyl



1.2.704
3-acetoxy-5-ethylphenyl
fluoromethyl



1.2.705
(3-[(tert-butoxy-carbonyl)amino]-5-
fluoromethyl




ethylphenyl}




1.2.706
3-methylsulfanyl-5-ethylphenyl
fluoromethyl



1.2.707
3,5-dipropylphenyl
fluoromethyl



1.2.708
3-isopropyl-5-propylphenyl
fluoromethyl



1.2.709
3-n-butyl-5-propylphenyl
fluoromethyl



1.2.710
3-isobutyl-5-propylphenyl
fluoromethyl



1.2.711
3-tert-butyl-5-propylphenyl
fluoromethyl



1.2.712
3-cyclopropyl-5-propylphenyl
fluoromethyl



1.2.713
3-vinyl-5-propylphenyl
fluoromethyl



1.2.714
3-ethynyl-5-propylphenyl
fluoromethyl



1.2.715
3-cyano-5-propylphenyl
fluoromethyl



1.2.716
3-trifluoromethyl-5-propylphenyl
fluoromethyl



1.2.717
3-(hydroxycarbonyl)-5-propylphenyl
fluoromethyl



1.2.718
3-(methoxycarbonyl)-5-
fluoromethyl




propylphenyl




1.2.719
3-hydroxymethyl-5-propylphenyl
fluoromethyl



1.2.720
3-carbamoyl-5-propylphenyl
fluoromethyl



1.2.721
3-hydroxy-5-propylphenyl
fluoromethyl



1.2.722
3-methoxy-5-propylphenyl
fluoromethyl



1.2.723
3-ethoxy-5-propylphenyl
fluoromethyl



1.2.724
3-n-propoxy-5-propylphenyl
fluoromethyl



1.2.725
3-n-butoxy-5-propylphenyl
fluoromethyl



1.2.726
3-isobutoxy-5-propylphenyl
fluoromethyl



1.2.727
3-tert-butoxy-5-propylphenyl
fluoromethyl



1.2.728
3-difluoromethoxy-5-propylphenyl
fluoromethyl



1.2.729
3-trifluoromethoxy-5-ethylphenyl
fluoromethyl



1.2.730
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl




propylphenyl




1.2.731
3-(2-chloroethoxy)-5-propylphenyl
fluoromethyl



1.2.732
3-(2-hydroxyethoxy)-5-propylphenyl
fluoromethyl



1.2.733
3-[tert-butoxycarbonyl)oxy]-5-
fluoromethyl




propylphenyl




1.2.734
3-nitro-5-propylphenyl
fluoromethyl



1.2.735
3-acetoxy-5-propylphenyl
fluoromethyl



1.2.736
{3-[(tert-butoxy-carbonyl)amino]-5-
fluoromethyl




propylphenyl}




1.2.737
3-methylsulfanyl-5-propylphenyl
fluoromethyl



1.2.738
3,5-diisopropylphenyl
fluoromethyl



1.2.739
3-n-butyl-5-isopropylphenyl
fluoromethyl



1.2.740
3-isobutyl-5-isopropylphenyl
fluoromethyl



1.2.741
3-tert-butyl-5-isopropylphenyl
fluoromethyl



1.2.742
3-cyclopropyl-5-isopropylphenyl
fluoromethyl



1.2.743
3-vinyl-5-isopropylphenyl
fluoromethyl



1.2.744
3-ethynyl-5-isopropylphenyl
fluoromethyl



1.2.745
3-cyano-5-isopropylphenyl
fluoromethyl



1.2.746
3-trifluoromethyl-5-isopropylphenyl
fluoromethyl



1.2.747
3-(hydroxycarbonyl)-5-
fluoromethyl




isopropylphenyl




1.2.748
3-(methoxycarbonyl)-5-
fluoromethyl




isopropylphenyl




1.2.749
3-hydroxymethyl-5-isopropylphenyl
fluoromethyl



1.2.750
3-carbamoyl-5-isopropylphenyl
fluoromethyl



1.2.751
3-hydroxy-5-isopropylphenyl
fluoromethyl



1.2.752
3-methoxy-5-isopropylphenyl
fluoromethyl



1.2.753
3-ethoxy-5-isopropylphenyl
fluoromethyl



1.2.754
3-n-propoxy-5-isopropylphenyl
fluoromethyl



1.2.755
3-n-butoxy-5-isopropylphenyl
fluoromethyl



1.2.756
3-isobutoxy-5-isopropylphenyl
fluoromethyl



1.2.757
3-tert-butoxy-5-isopropylphenyl
fluoromethyl



1.2.758
3-difluoromethoxy-5-
fluoromethyl




isopropylphenyl




1.2.759
3-trifluoromethoxy-5-
fluoromethyl




isopropylphenyl




1.2.760
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl




isopropylphenyl




1.2.761
3-(2-chloroethoxy)-5-
fluoromethyl




isopropylphenyl




1.2.762
3-(2-hydroxyethoxy)-5-propylphenyl
fluoromethyl



1.2.763
3-[tert-butoxycarbonyl)oxy]-5-
fluoromethyl




isopropylphenyl




1.2.764
3-nitro-5-isopropylphenyl
fluoromethyl



1.2.765
3-acetoxy-5-isopropylphenyl
fluoromethyl



1.2.766
{3-[tert-butoxy-carbonyl)amino]-5-
fluoromethyl




isopropylphenyl}




1.2.767
3-methylsulfanyl-5-isopropylphenyl
fluoromethyl



1.2.768
3,5-dibutylphenyl
fluoromethyl



1.2.769
3-isobutyl-5-butylphenyl
fluoromethyl



1.2.770
3-tert-butyl-5-butylphenyl
fluoromethyl



1.2.771
3-cyclopropyl-5-butylphenyl
fluoromethyl



1.2.772
3-vinyl-5-butylphenyl
fluoromethyl



1.2.773
3-ethynyl-5-butylphenyl
fluoromethyl



1.2.774
3-cyano-5-butylphenyl
fluoromethyl



1.2.775
3-trifluoromethyl-5-butylphenyl
fluoromethyl



1.2.776
3-(hydroxycarbonyl)-5-butylphenyl
fluoromethyl



1.2.777
3-(methoxycarbonyl)-5-butylphenyl
fluoromethyl



1.2.778
3-hydroxymethyl-5-butylphenyl
fluoromethyl



1.2.779
3-carbamoyl-5-butylphenyl
fluoromethyl



1.2.780
3-hydroxy-5-butylphenyl
fluoromethyl



1.2.781
3-methoxy-5-butylphenyl
fluoromethyl



1.2.782
3-ethoxy-5-butylphenyl
fluoromethyl



1.2.783
3-n-propoxy-5-butylphenyl
fluoromethyl



1.2.784
3-n-butoxy-5-butylphenyl
fluoromethyl



1.2.785
3-isobutoxy-5-butylphenyl
fluoromethyl



1.2.786
3-tert-butoxy-5-butylphenyl
fluoromethyl



1.2.787
3-difluoromethoxy-5-butylphenyl
fluoromethyl



1.2.788
3-trifluoromethoxy-5-butylphenyl
fluoromethyl



1.2.789
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl




butylphenyl




1.2.790
3-(2-chloroethoxy)-5-butylphenyl
fluoromethyl



1.2.791
3-(2-hydroxyethoxy)-5-butylphenyl
fluoromethyl



1.2.792
3-[tert-butoxycarbonyl)oxy]-5-
fluoromethyl




butylphenyl




1.2.793
3-nitro-5-butylphenyl
fluoromethyl



1.2.794
3-acetoxy-5-butylphenyl
fluoromethyl



1.2.795
(3-[(tert-butoxy-carbonyl)amino]-5-
fluoromethyl




butylphenyl}




1.2.796
3-methylsulfanyl-5-butylphenyl
fluoromethyl



1.2.797
3,5-diisobutylphenyl
fluoromethyl



1.2.798
3-tert-butyl-5-isobutylphenyl
fluoromethyl



1.2.799
3-cyclopropyl-5-isobutylphenyl
fluoromethyl



1.2.800
3-vinyl-5-isobutylphenyl
fluoromethyl



1.2.801
3-ethynyl-5-isobutylphenyl
fluoromethyl



1.2.802
3-cyano-5-isobutylphenyl
fluoromethyl



1.2.803
3-trifluoromethyl-5-isobutylphenyl
fluoromethyl



1.2.804
3-(hydroxycarbonyl)-5-
fluoromethyl




isobutylphenyl




1.2.805
3-(methoxycarbonyl)-5-
fluoromethyl




isobutylphenyl




1.2.806
3-hydroxymethyl-5-isobutylphenyl
fluoromethyl



1.2.807
3-carbamoyl-5-isobutylphenyl
fluoromethyl



1.2.808
3-hydroxy-5-isobutylphenyl
fluoromethyl



1.2.809
3-methoxy-5-isobutylphenyl
fluoromethyl



1.2.810
3-ethoxy-5-isobutylphenyl
fluoromethyl



1.2.811
3-n-propoxy-5-isobutylphenyl
fluoromethyl



1.2.812
3-n-butoxy-5-isobutylphenyl
fluoromethyl



1.2.813
3-isobutoxy-5-isobutylphenyl
fluoromethyl



1.2.814
3-tert-butoxy-5-isobutylphenyl
fluoromethyl



1.2.815
3-difluoromethoxy-5-isobutylphenyl
fluoromethyl



1.2.816
3-trifluoromethoxy-5-isobutylphenyl
fluoromethyl



1.2.817
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl




isobutylphenyl




1.2.818
3-(2-chloroethoxy)-5-isobutylphenyl
fluoromethyl



1.2.819
3-(2-hydroxyethoxy)-5-
fluoromethyl




isobutylphenyl




1.2.820
3-[(tert-butoxycarbonyl)oxy]-5-
fluoromethyl




isobutylphenyl




1.2.821
3-nitro-5-isobutylphenyl
fluoromethyl



1.2.822
3-acetoxy-5-isobutylphenyl
fluoromethyl



1.2.823
{3-[tert-butoxycarbonyl)amino]-5-
fluoromethyl




isobutylphenyl}




1.2.824
3-methylsulfanyl-5-isobutylphenyl
fluoromethyl



1.2.825
3,5-di(tert-butyl)phenyl
fluoromethyl



1.2.826
3-cyclopropyl-5-tert-butylphenyl
fluoromethyl



1.2.827
3-vinyl-5-tert-butylphenyl
fluoromethyl



1.2.828
3-ethynyl-5-tert-butylphenyl
fluoromethyl



1.2.829
3-cyano-5-tert-butylphenyl
fluoromethyl



1.2.830
3-trifluoromethyl-5-tert-butylphenyl
fluoromethyl



1.2.831
3-(hydroxycarbonyl)-5-tert-
fluoromethyl




butylphenyl




1.2.832
3-(methoxycarbonyl)-5-tert-
fluoromethyl




butylphenyl




1.2.833
3-hydroxymethyl-5-tert-butylphenyl
fluoromethyl



1.2.834
3-carbamoyl-5-tert-butylphenyl
fluoromethyl



1.2.835
3-hydroxy-5-tert-butylphenyl
fluoromethyl



1.2.836
3-methoxy-5-tert-butylphenyl
fluoromethyl



1.2.837
3-ethoxy-5-tert-butylphenyl
fluoromethyl



1.2.838
3-n-propoxy-5-tert-butylphenyl
fluoromethyl



1.2.839
3-n-butoxy-5-tert-butylphenyl
fluoromethyl



1.2.840
3-isobutoxy-5-tert-butylphenyl
fluoromethyl



1.2.841
3-tert-butoxy-5-tert-butylphenyl
fluoromethyl



1.2.842
3-difluoromethoxy-5-tert-
fluoromethyl




butylphenyl




1.2.843
3-trifluoromethoxy-5-tert-
fluoromethyl




butylphenyl




1.2.844
3-(2,2,2-trifluoroethoxy)-5-tert-fluoromethyl





butylphenyl




1.2.845
3-(2-chloroethoxy)-5-tert-
fluoromethyl




butylphenyl




1.2.846
3-(2-hydroxyethoxy)-5-tert-
fluoromethyl




butylphenyl




1.2.847
3-[tert-butoxycarbonyl)oxy]-5-tert-
fluoromethyl




butylphenyl




1.2.848
3-nitro-5-tert-butylphenyl
fluoromethyl



1.2.849
3-acetoxy-5-tert-butylphenyl
fluoromethyl



1.2.850
{3-[tert-butoxy-carbonyl)amino]-5-
fluoromethyl




tert-butylphenyl}




1.2.851
3-methylsulfanyl-5-tert-butylphenyl
fluoromethyl



1.2.852
3-tert-butyl-5-cyclopropylphenyl
fluoromethyl



1.2.853
3,5-dicyclopropyl-phenyl
fluoromethyl



1.2.854
3-vinyl-5-cyclopropylphenyl
fluoromethyl



1.2.855
3-ethynyl-5-cyclopropylphenyl
fluoromethyl



1.2.856
3-cyano-5-cyclopropylphenyl
fluoromethyl



1.2.857
3-trifluoromethyl-5-
fluoromethyl




cyclopropylphenyl




1.2.858
3-(hydroxycarbonyl)-5-
fluoromethyl




cyclopropylphenyl




1.2.859
3-(methoxycarbonyl)-5-
fluoromethyl




cyclopropylphenyl




1.2.860
3-hydroxymethyl-5-
fluoromethyl




cyclopropylphenyl




1.2.861
3-carbamoyl-5-cyclopropylphenyl
fluoromethyl



1.2.862
3-hydroxy-5-cyclopropylphenyl
fluoromethyl



1.2.863
3-methoxy-5-cyclopropylphenyl
fluoromethyl



1.2.864
3-ethoxy-5-cyclopropylphenyl
fluoromethyl



1.2.865
3-n-propoxy-5-cyclopropylphenyl
fluoromethyl



1.2.866
3-n-butoxy-5-cyclopropylphenyl
fluoromethyl



1.2.867
3-isobutoxy-5-cyclopropylphenyl
fluoromethyl



1.2.868
3-tert-butoxy-5-cyclopropylphenyl
fluoromethyl



1.2.869
3-difluoromethoxy-5-
fluoromethyl




cyclopropylphenyl




1.2.870
3-trifluoromethoxy-5-
fluoromethyl




cyclopropylphenyl




1.2.871
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl




cyclopropylphenyl




1.2.872
3-(2-chloroethoxy)-5-
fluoromethyl




cyclopropylphenyl




1.2.873
3-(2-hydroxyethoxy)-5-
fluoromethyl




cyclopropylphenyl




1.2.874
3-[tert-butoxycarbonyl)oxy]-5-
fluoromethyl




cyclopropylphenyl




1.2.875
3-nitro-5-cyclopropylphenyl
fluoromethyl



1.2.876
3-acetoxy-5-cyclopropylphenyl
fluoromethyl



1.2.877
{3-[(tert-butoxycarbonyl)amino]-5-
fluoromethyl




cyclopropylphenyl}




1.2.878
3-methylsulfanyl-5-
fluoromethyl




cyclopropylphenyl




1.2.879
3,5-divinylphenyl
fluoromethyl



1.2.880
3-ethynyl-5-vinylphenyl
fluoromethyl



1.2.881
3-cyano-5-vinylphenyl
fluoromethyl



1.2.882
3-trifluoromethyl-5-vinylphenyl
fluoromethyl



1.2.883
3-(hydroxycarbonyl)-5-vinylphenyl
fluoromethyl



1.2.884
3-(methoxycarbonyl)-5-vinylphenyl
fluoromethyl



1.2.885
3-hydroxymethyl-5-vinylphenyl
fluoromethyl



1.2.886
3-carbamoyl-5-vinylphenyl
fluoromethyl



1.2.887
3-hydroxy-5-vinylphenyl
fluoromethyl



1.2.888
3-methoxy-5-vinylphenyl
fluoromethyl



1.2.889
3-ethoxy-5-vinylphenyl
fluoromethyl



1.2.890
3-n-propoxy-5-vinylphenyl
fluoromethyl



1.2.891
3-n-butoxy-5-vinylphenyl
fluoromethyl



1.2.892
3-isobutoxy-5-vinylphenyl
fluoromethyl



1.2.893
3-tert-butoxy-5-vinylphenyl
fluoromethyl



1.2.894
3-difluoromethoxy-5-vinylphenyl
fluoromethyl



1.2.895
3-trifluoromethoxy-5-vinylphenyl
fluoromethyl



1.2.896
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl




vinylphenyl




1.2.897
3-(2-chloroethoxy)-5-vinylphenyl
fluoromethyl



1.2.898
3-(2-hydroxyethoxy)-5-vinylphenyl
fluoromethyl



1.2.899
3-[tert-butoxycarbonyl)oxy]-5-
fluoromethyl




vinylphenyl




1.2.900
3-nitro-5-vinylphenyl
fluoromethyl



1.2.901
3-acetoxy-5-vinylphenyl
fluoromethyl



1.2.902
(3-[(tert-butoxy-carbonyl)amino]-5-
fluoromethyl




vinylphenyl}




1.2.903
3-methylsulfanyl-5-vinylphenyl
fluoromethyl



1.2.904
3,5-diethynylphenyl
fluoromethyl



1.2.905
3-cyano-5-ethynylphenyl
fluoromethyl



1.2.906
3-trifluoromethyl-5-ethynylphenyl
fluoromethyl



1.2.907
3-(hydroxycarbonyl)-5-
fluoromethyl




ethynylphenyl




1.2.908
3-(methoxycarbonyl)-5-
fluoromethyl




ethynylphenyl




1.2.909
3-hydroxymethyl-5-ethynylphenyl
fluoromethyl



1.2.910
3-carbamoyl-5-ethynylphenyl
fluoromethyl



1.2.911
3-hydroxy-5-ethynylphenyl
fluoromethyl



1.2.912
3-methoxy-5-ethynylphenyl
fluoromethyl



1.2.913
3-ethoxy-5-ethynylphenyl
fluoromethyl



1.2.914
3-n-propoxy-5-ethynylphenyl
fluoromethyl



1.2.915
3-n-butoxy-5-ethynylphenyl
fluoromethyl



1.2.916
3-isobutoxy-5-ethynylphenyl
fluoromethyl



1.2.917
3-tert-butoxy-5-ethynylphenyl
fluoromethyl



1.2.918
3-difluoromethoxy-5-ethynylphenyl
fluoromethyl



1.2.919
3-trifluoromethoxy-5-ethynylphenyl
fluoromethyl



1.2.920
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl




ethynylphenyl




1.2.921
3-(2-chloroethoxy)-5-ethynylphenyl
fluoromethyl



1.2.922
3-(2-hydroxyethoxy)-5-
fluoromethyl




ethynylphenyl




1.2.923
3-[tert-butoxycarbonyl)oxy]-5-
fluoromethyl




ethynylphenyl




1.2.924
3-nitro-5-ethynylphenyl
fluoromethyl



1.2.925
3-acetoxy-5-ethynylphenyl
fluoromethyl



1.2.926
(3-[(tert-butoxy-carbonyl)amino]-5-
fluoromethyl




ethynylphenyl}




1.2.927
3-methylsulfanyl-5-ethynylphenyl
fluoromethyl



1.2.928
3,5-dicyanophenyl
fluoromethyl



1.2.929
3-trifluoromethyl-5-cyanophenyl
fluoromethyl



1.2.930
3-(hydroxycarbonyl)-5-cyanophenyl
fluoromethyl



1.2.931
3-(methoxycarbonyl)-5-
fluoromethyl




cyanophenyl




1.2.932
3-hydroxymethyl-5-cyanophenyl
fluoromethyl



1.2.933
3-carbamoyl-5-cyanophenyl
fluoromethyl



1.2.934
3-hydroxy-5-cyanophenyl
fluoromethyl



1.2.935
3-methoxy-5-cyanophenyl
fluoromethyl



1.2.936
3-ethoxy-5-cyanophenyl
fluoromethyl



1.2.937
3-n-propoxy-5-cyanophenyl
fluoromethyl



1.2.938
3-n-butoxy-5-cyanophenyl
fluoromethyl



1.2.939
3-isobutoxy-5-cyanophenyl
fluoromethyl



1.2.940
3-tert-butoxy-5-cyanophenyl
fluoromethyl



1.2.941
3-difluoromethoxy-5-cyanophenyl
fluoromethyl



1.2.942
3-trifluoromethoxy-5-cyanophenyl
fluoromethyl



1.2.943
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl




cyanophenyl




1.2.944
3-(2-chloroethoxy)-5-cyanophenyl
fluoromethyl



1.2.945
3-(2-hydroxyethoxy)-5-cyanophenyl
fluoromethyl



1.2.946
3-[tert-butoxycarbonyl)oxy]-5-
fluoromethyl




cyanophenyl




1.2.947
3-nitro-5-cyanophenyl
fluoromethyl



1.2.948
3-acetoxy-5-cyanophenyl
fluoromethyl



1.2.949
(3-[(tert-butoxy-carbonyl)amino]-5-
fluoromethyl




cyanophenyl}




1.2.950
3-methylsulfanyl-5-cyanophenyl
fluoromethyl



1.2.951
3,5-di(trifluoromethyl)-phenyl
fluoromethyl



1.2.952
3-(hydroxycarbonyl)-5-
fluoromethyl




trifluoromethyl-phenyl




1.2.953
3-(methoxycarbonyl)-5-
fluoromethyl




trifluoromethyl-phenyl




1.2.954
3-hydroxymethyl-5-
fluoromethyl




trifluoromethylphenyl




1.2.955
3-carbamoyl-5-
fluoromethyl




trifluoromethylphenyl




1.2.956
3-hydroxy-5-trifluoromethylphenyl
fluoromethyl



1.2.957
3-methoxy-5-trifluoromethylphenyl
fluoromethyl



1.2.958
3-ethoxy-5-trifluoromethylphenyl
fluoromethyl



1.2.959
3-n-propoxy-5-trifluoromethylphenyl
fluoromethyl



1.2.960
3-n-butoxy-5-trifluoromethylphenyl
fluoromethyl



1.2.961
3-isobutoxy-5-trifluoromethylphenyl
fluoromethyl



1.2.962
3-tert-butoxy-5-
fluoromethyl




trifluoromethylphenyl




1.2.963
3-difluoromethoxy-5-
fluoromethyl




trifluoromethylphenyl




1.2.964
3-trifluoromethoxy-5-
fluoromethyl




trifluoromethylphenyl




1.2.965
3-(2,2,2-trifluoroethoxy)-5-trifluoro-
fluoromethyl




methylphenyl




1.2.966
3-(2-chloroethoxy)-5-
fluoromethyl




trifluoromethyl-phenyl




1.2.967
3-(2-hydroxyethoxy)-5-
fluoromethyl




trifluoromethyl-phenyl




1.2.968
3-[tert-butoxycarbonyl)oxy]-5-
fluoromethyl




trifluoromethylphenyl




1.2.969
3-nitro-5-trifluoromethylphenyl
fluoromethyl



1.2.970
3-acetoxy-5-trifluoromethylphenyl
fluoromethyl



1.2.971
(3-[tert-butoxy-carbonyl)amino]-5-
fluoromethyl




trifluoromethylphenyl}




1.2.972
3-methylsulfanyl-5-
fluoromethyl




trifluoromethylphenyl




1.2.973
3,5-bis(hydroxy-carbonyl)phenyl
fluoromethyl



1.2.974
3-(methoxycarbonyl)-5-
fluoromethyl




(hydroxycarbonyl)phenyl




1.2.975
3-hydroxymethyl-5-
fluoromethyl




(hydroxycarbonyl)phenyl




1.2.976
3-carbamoyl-5-(hydroxycarbonyl)-
fluoromethyl




phenyl




1.2.977
3-hydroxy-5-(hydroxycarbonyl)-
fluoromethyl




phenyl




1.2.978
3-methoxy-5-(hydroxycarbonyl)-
fluoromethyl




phenyl




1.2.979
3-ethoxy-5-(hydroxycarbonyl)-
fluoromethyl




phenyl




1.2.980
3-n-propoxy-5-(hydroxycarbonyl)-
fluoromethyl




phenyl




1.2.981
3-n-butoxy-5-(hydroxycarbonyl)-
fluoromethyl




phenyl




1.2.982
3-isobutoxy-5-(hydroxycarbonyl)-
fluoromethyl




phenyl




1.2.983
3-tert-butoxy-5-(hydroxycarbonyl)-
fluoromethyl




phenyl




1.2.984
3-difluoromethoxy-5-
fluoromethyl




(hydroxycarbonyl)phenyl




1.2.985
3-trifluoromethoxy-5-
fluoromethyl




(hydroxycarbonyl)phenyl




1.2.986
3-(2,2,2-trifluoroethoxy)-5-(hydroxy-
fluoromethyl




carbonyl)phenyl




1.2.987
3-(2-chloroethoxy)-5-
fluoromethyl




(hydroxycarbonyl)phenyl




1.2.988
3-(2-hydroxyethoxy)-5-
fluoromethyl




(hydroxycarbonyl)phenyl




1.2.989
3-[tert-butoxycarbonyl)oxy]-5-
fluoromethyl




(hydroxycarbonyl)phenyl




1.2.990
3-nitro-5-(hydroxycarbonyl)phenyl
fluoromethyl



1.2.991
3-acetoxy-5-(hydroxycarbonyl)-
fluoromethyl




phenyl




1.2.992
(3-[tert-butoxy-carbonyl)amino]-5-
fluoromethyl




(hydroxycarbonyl)phenyl)




1.2.993
3-methylsulfanyl-5-
fluoromethyl




(hydroxycarbonyl)phenyl




1.2.994
3,5-di(methoxy-carbonyl)phenyl
fluoromethyl



1.2.995
3-hydroxymethyl-5-
fluoromethyl




(methoxycarbonyl)phenyl




1.2.996
3-carbamoyl-5-(methoxycarbonyl)-
fluoromethyl




phenyl




1.2.997
3-hydroxy-5-(methoxycarbonyl)-
fluoromethyl




phenyl




1.2.998
3-methoxy-5-(methoxycarbonyl)-
fluoromethyl




phenyl




1.2.999
3-ethoxy-5-(methoxycarbonyl)-
fluoromethyl




phenyl




1.2.1000
3-n-propoxy-5-(methoxycarbonyl)-
fluoromethyl




phenyl




1.2.1001
3-n-butoxy-5-(methoxycarbonyl)-
fluoromethyl




phenyl




1.2.1002
3-isobutoxy-5-(methoxycarbonyl)-
fluoromethyl




phenyl




1.2.1003
3-tert-butoxy-5-(methoxycarbonyl)-
fluoromethyl




phenyl




1.2.1004
3-difluoromethoxy-5-
fluoromethyl




(methoxycarbonyl)-phenyl




1.2.1005
3-trifluoromethoxy-5-
fluoromethyl




(methoxycarbonyl)phenyl




1.2.1006
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl




(methoxy-carbonyl)phenyl




1.2.1007
3-(2-chloroethoxy)-5-
fluoromethyl




(methoxycarbonyl)phenyl




1.2.1008
3-(2-hydroxyethoxy)-5-
fluoromethyl




(methoxycarbonyl)phenyl




1.2.1009
3-[tert-butoxycarbonyl)oxy]-5-
fluoromethyl




(methoxycarbonyl)phenyl




1.2.1010
3-nitro-5-(methoxycarbonyl)phenyl
fluoromethyl



1.2.1011
3-acetoxy-5-(methoxycarbonyl)-
fluoromethyl




phenyl




1.2.1012
{3-[tert-butoxycarbonyl)amino]-5-
fluoromethyl




(methoxycarbonyl)phenyl}




1.2.1013
3-methylsulfanyl-5-
fluoromethyl




(methoxycarbonyl)phenyl




1.2.1014
3,5-di(hydroxymethyl)phenyl
fluoromethyl



1.2.1015
3-carbamoyl-5-
fluoromethyl




hydroxymethylphenyl




1.2.1016
3-hydroxy-5-hydroxymethylphenyl
fluoromethyl



1.2.1017
3-methoxy-5-hydroxymethylphenyl
fluoromethyl



1.2.1018
3-ethoxy-5-hydroxymethylphenyl
fluoromethyl



1.2.1019
3-n-propoxy-5-
fluoromethyl




hydroxymethylphenyl




1.2.1020
3-n-butoxy-5-hydroxymethylphenyl
fluoromethyl



1.2.1021
3-isobutoxy-5-hydroxymethylphenyl
fluoromethyl



1.2.1022
3-tert-butoxy-5-
fluoromethyl




hydroxymethylphenyl




1.2.1023
3-difluoromethoxy-5-
fluoromethyl




hydroxymethylphenyl




1.2.1024
3-trifluoromethoxy-5-
fluoromethyl




hydroxymethylphenyl




1.2.1025
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl




hydroxymethylphenyl




1.2.1026
3-(2-chloroethoxy)-5-
fluoromethyl




hydroxymethylphenyl




1.2.1027
3-(2-hydroxyethoxy)-5-
fluoromethyl




hydroxymethyl-phenyl




1.2.1028
3-[tert-butoxycarbonyl)oxy]-5-
fluoromethyl




hydroxymethylphenyl




1.2.1029
3-nitro-5-hydroxymethylphenyl
fluoromethyl



1.2.1030
3-acetoxy-5-hydroxymethylphenyl
fluoromethyl



1.2.1031
(3-[tert-butoxycarbonyl)amino]-5-
fluoromethyl




hydroxymethyl-phenyl}




1.2.1032
3-methylsulfanyl-5-
fluoromethyl




hydroxymethylphenyl




1.2.1033
3,5-dicarbamoyl-5-carbamoylphenyl
fluoromethyl



1.2.1034
3-hydroxy-5-carbamoylphenyl
fluoromethyl



1.2.1035
3-methoxy-5-carbamoylphenyl
fluoromethyl



1.2.1036
3-ethoxy-5-carbamoylphenyl
fluoromethyl



1.2.1037
3-n-propoxy-5-carbamoylphenyl
fluoromethyl



1.2.1038
3-n-butoxy-5-carbamoylphenyl
fluoromethyl



1.2.1039
3-isobutoxy-5-carbamoylphenyl
fluoromethyl



1.2.1040
3-tert-butoxy-5-carbamoylphenyl
fluoromethyl



1.2.1041
3-difluoromethoxy-5-
fluoromethyl




carbamoylphenyl




1.2.1042
3-trifluoromethoxy-5-
fluoromethyl




carbamoylphenyl




1.2.1043
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl




carbamoylphenyl




1.2.1044
3-(2-chloroethoxy)-5-
fluoromethyl




carbamoylphenyl




1.2.1045
3-(2-hydroxyethoxy)-5-
fluoromethyl




carbamoylphenyl




1.2.1046
3-[tert-butoxycarbonyl)oxy]-5-
fluoromethyl




carbamoylphenyl




1.2.1047
3-nitro-5-carbamoylphenyl
fluoromethyl



1.2.1048
3-acetoxy-5-carbamoylphenyl
fluoromethyl



1.2.1049
{3-[(tert-butoxycarbonyl)amino]-5-
fluoromethyl




carbamoylphenyl}




1.2.1050
3-methylsulfanyl-5-
fluoromethyl




carbamoylphenyl




1.2.1051
3,5-dihydroxyphenyl
fluoromethyl



1.2.1052
3-methoxy-5-hydroxyphenyl
fluoromethyl



1.2.1053
3-ethoxy-5-hydroxyphenyl
fluoromethyl



1.2.1054
3-n-propoxy-5-hydroxyphenyl
fluoromethyl



1.2.1055
3-n-butoxy-5-hydroxyphenyl
fluoromethyl



1.2.1056
3-isobutoxy-5-hydroxyphenyl
fluoromethyl



1.2.1057
3-tert-butoxy-5-hydroxyphenyl
fluoromethyl



1.2.1058
3-difluoromethoxy-5-hydroxyphenyl
fluoromethyl



1.2.1059
3-trifluoromethoxy-5-hydroxyphenyl
fluoromethyl



1.2.1060
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl




hydroxyphenyl




1.2.1061
3-(2-chloroethoxy)-5-hydroxyphenyl
fluoromethyl



1.2.1062
3-(2-hydroxyethoxy)-5-
fluoromethyl




hydroxyphenyl




1.2.1063
3-[tert-butoxycarbonyl)oxy]-5-
fluoromethyl




hydroxyphenyl




1.2.1064
3-nitro-5-hydroxyphenyl
fluoromethyl



1.2.1065
3-acetoxy-5-hydroxyphenyl
fluoromethyl



1.2.1066
{3-[(tert-butoxycarbonyl)amino]-5-
fluoromethyl




hydroxyphenyl}




1.2.1067
3-methylsulfanyl-5-hydroxyphenyl
fluoromethyl



1.2.1068
3,5-dimethoxyphenyl
fluoromethyl



1.2.1069
3-ethoxy-5-methoxyphenyl
fluoromethyl



1.2.1070
3-n-propoxy-5-methoxyphenyl
fluoromethyl



1.2.1071
3-n-butoxy-5-methoxyphenyl
fluoromethyl



1.2.1072
3-isobutoxy-5-methoxyphenyl
fluoromethyl



1.2.1073
3-tert-butoxy-5-methoxyphenyl
fluoromethyl



1.2.1074
3-difluoromethoxy-5-methoxyphenyl
fluoromethyl



1.2.1075
3-trifluoromethoxy-5-
fluoromethyl




methoxyphenyl




1.2.1076
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl




methoxyphenyl




1.2.1077
3-(2-chloroethoxy)-5-
fluoromethyl




methoxyphenyl




1.2.1078
3-(2-hydroxyethoxy)-5-
fluoromethyl




methoxyphenyl




1.2.1079
3-[tert-butoxycarbonyl)oxy]-5-
fluoromethyl




methoxyphenyl




1.2.1080
3-nitro-5-methoxyphenyl
fluoromethyl



1.2.1081
3-acetoxy-5-methoxyphenyl
fluoromethyl



1.2.1082
{3-[(tert-butoxycarbonyl)amino]-5-
fluoromethyl




methoxyphenyl}




1.2.1083
3-methylsulfanyl-5-methoxyphenyl
fluoromethyl



1.2.1084
3,5-diethoxyphenyl
fluoromethyl



1.2.1085
3-n-propoxy-5-ethoxyphenyl
fluoromethyl



1.2.1086
3-n-butoxy-5-ethoxyphenyl
fluoromethyl



1.2.1087
3-isobutoxy-5-ethoxyphenyl
fluoromethyl



1.2.1088
3-tert-butoxy-5-ethoxyphenyl
fluoromethyl



1.2.1089
3-difluoromethoxy-5-ethoxyphenyl
fluoromethyl



1.2.1090
3-trifluoromethoxy-5-ethoxyphenyl
fluoromethyl



1.2.1091
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl




ethoxyphenyl




1.2.1092
3-(2-chloroethoxy)-5-ethoxyphenyl
fluoromethyl



1.2.1093
3-(2-hydroxyethoxy)-5-
fluoromethyl




ethoxyphenyl




1.2.1094
3-[tert-butoxycarbonyl)oxy]-5-
fluoromethyl




ethoxyphenyl




1.2.1095
3-nitro-5-ethoxyphenyl
fluoromethyl



1.2.1096
3-acetoxy-5-ethoxyphenyl
fluoromethyl



1.2.1097
{3-[(tert-butoxycarbonyl)amino]-5-
fluoromethyl




ethoxyphenyl}




1.2.1098
3-methylsulfanyl-5-ethoxyphenyl
fluoromethyl



1.2.1099
3,5-dipropoxyphenyl
fluoromethyl



1.2.1100
3-n-butoxy-5-propoxyphenyl
fluoromethyl



1.2.1101
3-isobutoxy-5-propoxyphenyl
fluoromethyl



1.2.1102
3-tert-butoxy-5-propoxyphenyl
fluoromethyl



1.2.1103
3-difluoromethoxy-5-propoxyphenyl
fluoromethyl



1.2.1104
3-trifluoromethoxy-5-propoxyphenyl
fluoromethyl



1.2.1105
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl




propoxyphenyl




1.2.1106
3-(2-chloroethoxy)-5-propoxyphenyl
fluoromethyl



1.2.1107
3-(2-hydroxyethoxy)-5-
fluoromethyl




propoxyphenyl




1.2.1108
3-[tert-butoxycarbonyl)oxy]-5-
fluoromethyl




propoxyphenyl




1.2.1109
3-nitro-5-propoxyphenyl
fluoromethyl



1.2.1110
3-acetoxy-5-propoxyphenyl
fluoromethyl



1.2.1111
{3-[(tert-butoxycarbonyl)amino]-5-
fluoromethyl




propoxyphenyl}




1.2.1112
3-methylsulfanyl-5-propoxyphenyl
fluoromethyl



1.2.1113
3,5-di(isopropoxy)phenyl
fluoromethyl



1.2.1114
3-n-butoxy-5-isopropoxyphenyl
fluoromethyl



1.2.1115
3-isobutoxy-5-isopropoxyphenyl
fluoromethyl



1.2.1116
3-tert-butoxy-5-isopropoxyphenyl
fluoromethyl



1.2.1117
3-difluoromethoxy-5-
fluoromethyl




isopropoxyphenyl




1.2.1118
3-trifluoromethoxy-5-
fluoromethyl




isopropoxyphenyl




1.2.1119
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl




isopropoxyphenyl




1.2.1120
3-(2-chloroethoxy)-5-
fluoromethyl




isopropoxyphenyl




1.2.1121
3-(2-hydroxyethoxy)-5-
fluoromethyl




isopropoxyphenyl




1.2.1122
3-[tert-butoxycarbonyl)oxy]-5-
fluoromethyl




isopropoxyphenyl




1.2.1123
3-nitro-5-isopropoxyphenyl
fluoromethyl



1.2.1124
3-acetoxy-5-isopropoxyphenyl
fluoromethyl



1.2.1125
{3-[tert-butoxycarbonyl)amino]-5-
fluoromethyl




isopropoxyphenyl}




1.2.1126
3-methylsulfanyl-5-
fluoromethyl




isopropoxyphenyl




1.2.1127
3,5-di(tert-butoxy)-phenyl
fluoromethyl



1.2.1128
3-difluoromethoxy-5-tert-
fluoromethyl




butoxyphenyl




1.2.1129
3-trifluoromethoxy-5-tert-
fluoromethyl




butoxyphenyl




1.2.1130
3-(2,2,2-trifluoroethoxy)-5-tert-
fluoromethyl




butoxyphenyl




1.2.1131
3-(2-chloroethoxy)-5-tert-
fluoromethyl




butoxylphenyl




1.2.1132
3-(2-hydroxyethoxy)-5-tert-
fluoromethyl




butoxyphenyl




1.2.1133
3-[tert-butoxycarbonyl)oxy]-5-tert-
fluoromethyl




butoxyphenyl




1.2.1134
3-nitro-5-tert-butoxyphenyl
fluoromethyl



1.2.1135
3-acetoxy-5-tert-butoxyphenyl
fluoromethyl



1.2.1136
{3-[tert-butoxycarbonyl)amino]-5-
fluoromethyl




tert-butoxyphenyl}




1.2.1137
3-methylsulfanyl-5-tert-
fluoromethyl




butoxyphenyl




1.2.1138
3,5-di(trifluoromethoxy)phenyl
fluoromethyl



1.2.1139
3-(2,2,2-trifluoroethoxy)-5-trifluoro-
fluoromethyl




methoxyphenyl




1.2.1140
3-(2-chloroethoxy)-5-
fluoromethyl




trifluoromethoxyphenyl




1.2.1141
3-(2-hydroxyethoxy)-5-
fluoromethyl




trifluoromethoxyphenyl




1.2.1142
3-[tert-butoxycarbonyl)oxy]-5-
fluoromethyl




trifluoromethoxyphenyl




1.2.1143
3-nitro-5-trifluoromethoxyphenyl
fluoromethyl



1.2.1144
3-acetoxy-5-tert-butoxyphenyl
fluoromethyl



1.2.1145
{3-[(tert-butoxycarbonyl)amino]-5-
fluoromethyl




trifluoromethoxyphenyl}




1.2.1146
3-methylsulfanyl-5-trifluoromethoxy-
fluoromethyl




phenyl




1.2.1147
3,5-bis(difluoromethoxy)phenyl
fluoromethyl



1.2.1148
3,5-bis(difluoromethoxy)phenyl
chloromethyl



1.2.1149
3,5-bis(difluoromethoxy)phenyl
bromomethyl



1.2.1150
3,5-bis(difluoromethoxy)phenyl
fluoromethyl



1.2.1151
3-trifluoromethoxy-5-
fluoromethyl




difluoromethoxyphenyl




1.2.1152
3-(2,2,2-trifluoroethoxy)-5-difluoro-
fluoromethyl




methoxyphenyl




1.2.1153
3-(2-chloroethoxy)-5-
fluoromethyl




difluoromethoxyphenyl




1.2.1154
3-(2-hydroxyethoxy)-5-
fluoromethyl




difluoromethoxyphenyl




1.2.1155
3-[tert-butoxycarbonyl)oxy]-5-
fluoromethyl




difluoromethoxyphenyl




1.2.1156
3-nitro-5-difluoromethoxyphenyl
fluoromethyl



1.2.1157
3-acetoxy-5-difluoromethoxyphenyl
fluoromethyl



1.2.1158
{3-[tert-butoxycarbonyl)amino]-5-
fluoromethyl




difluoromethoxyphenyl}




1.2.1159
3-methylsulfanyl-5-
fluoromethyl




difluoromethoxyphenyl




1.2.1160
3,5-bis(2,2,2-trifluoroethoxy)-phenyl
fluoromethyl



1.2.1161
3-(2-chloroethoxy)-5-(2,2,2-trifluoro-
fluoromethyl




ethoxy)phenyl




1.2.1162
3-(2-hydroxyethoxy)-5-(2,2,2-
fluoromethyl




trifluoroethoxy)phenyl




1.2.1163
3-[tert-butoxycarbonyl)oxy]-5-
fluoromethyl




(2,2,2-trifluoroethoxy)-phenyl




1.2.1164
3-nitro-5-(2,2,2-trifluoroethoxy)-
fluoromethyl




phenyl




1.2.1165
3-acetoxy-5-(2,2,2-trifluoroethoxy)-
fluoromethyl




phenyl




1.2.1166
{3-[tert-butoxycarbonyl)amino]-5-
fluoromethyl




(2,2,2-trifluoroethoxy)phenyl}




1.2.1167
3-methylsulfanyl-5-(2,2,2-trifluoro-
fluoromethyl




ethoxy)phenyl




1.2.1168
3,5-bis(2-chloroethoxy)phenyl
fluoromethyl



1.2.1169
3-(2-hydroxyethoxy)-5-(2-
fluoromethyl




chloroethoxy)phenyl




1.2.1170
3-[tert-butoxycarbonyl)oxy]-5-(2-
fluoromethyl




chloroethoxy)phenyl




1.2.1171
3-nitro-5-(2-chloroethoxy)-phenyl
fluoromethyl



1.2.1172
3-acetoxy-5-(2-chloroethoxy)-
fluoromethyl




phenyl




1.2.1173
{3-[tert-butoxycarbonyl)amino]-5-
fluoromethyl




(2-chloroethoxy)phenyl}




1.2.1174
3-methylsulfanyl-5-(2-
fluoromethyl




chloroethoxy)phenyl




1.2.1175
3,5-bis(2-hydroxyethoxy)phenyl
fluoromethyl



1.2.1176
3-[tert-butoxycarbonyl)oxy]-5-(2-
fluoromethyl




hydroxyethoxy)phenyl




1.2.1177
3-nitro-5-(2-hydroxy-ethoxy)phenyl
fluoromethyl



1.2.1178
3-acetoxy-5-(2-hydroxyethoxy)-
fluoromethyl




phenyl




1.2.1179
3-[tert-butoxycarbonyl)amino]-5-(2-
fluoromethyl




hydroxyethoxy)phenyl




1.2.1180
3-methylsulfanyl-5-(2-
fluoromethyl




hydroxyethoxy)phenyl




1.2.1181
3,5-bis[(tert-butoxy-
fluoromethyl




carbonyl)oxy]phenyl




1.2.1182
3-nitro-5-[(tert-butoxy-
fluoromethyl




carbonyl)oxy]phenyl




1.2.1183
3-acetoxy-5-[(tert-butoxy-
fluoromethyl




carbonyl)oxy]phenyl




1.2.1184
{3-[tert-butoxycarbonyl)amino]-5-
fluoromethyl




[(tert-butoxycarbonyl)oxy]phenyl)




1.2.1185
3,5-bis(acetoxy)phenyl
fluoromethyl



1.2.1186
{3-[tert-butoxycarbonyl)amino]-5-
fluoromethyl




acetoxyphenyl}




1.2.1187
3-methylsulfanyl-5-acetoxyphenyl
fluoromethyl



1.2.1188
3,5-dinitrophenyl
fluoromethyl



1.2.1189
3-acetoxy-5-nitrophenyl
fluoromethyl



1.2.1190
{3-[tert-butoxycarbonyl)amino]-5-
fluoromethyl




nitrophenyl}




1.2.1191
3-methylsulfanyl-5-nitrophenyl
fluoromethyl



1.2.1192
3,5-bis[(tert-butoxycarbonyl)-
fluoromethyl




amino]phenyl




1.2.1193
3-methylsulfanyl-5-[(tert-butoxy-
fluoromethyl




carbonyl)amino]phenyl




1.2.1194
3,5-di(methylsulfanyl)phenyl
fluoromethyl



1.2.1195
3,4-difluorophenyl
fluoromethyl



1.2.1196
3,4-difluorophenyl
chloromethyl



1.2.1197
3,4-difluorophenyl
bromomethyl



1.2.1198
3,4-difluorophenyl
difluoromethyll



1.2.1199
3,4-difluorophenyl
trifluoromethyl



1.2.1200
3,4-difluorophenyl
cyano



1.2.1201
3-chloro-4-fluorophenyl
fluoromethyl



1.2.1202
3-chloro-4-fluorophenyl
chloromethyl



1.2.1203
3-chloro-4-fluorophenyl
bromomethyl



1.2.1204
3-chloro-4-fluorophenyl
difluoromethyl



1.2.1205
3-chloro-4-fluorophenyl
trifluoromethyl
[CDCl3] 3.81 (d, 1H); 4.00 (d,





1H); 7.22 (m, 1H); 7.58 (m,





1H); 7.74 (m, 1H).


1.2.1206
3-chloro-4-fluorophenyl
cyano



1.2.1207
3-bromo-4-fluorophenyl
fluoromethyl



1.2.1208
3-methyl-4-fluorophenyl
fluoromethyl



1.2.1209
3-methyl-4-fluorophenyl
chloromethyl



1.2.1210
3-ethyl-4-fluorophenyl
fluoromethyl



1.2.1211
3-cyclopropyl-4-fluorophenyl
fluoromethyl



1.2.1212
3-cyano-4-fluorophenyl
fluoromethyl



1.2.1213
3-methoxy-4-fluorophenyl
fluoromethyl



1.2.1214
3-ethoxy-4-fluorophenyl
fluoromethyl



1.2.1215
3-trifluoromethoxy-4-fluorophenyl
fluoromethyl



1.2.1216
3-nitro-4-fluorophenyl
fluoromethyl



1.2.1217
3-fluoro-4-chlorophenyl
fluoromethyl



1.2.1218
3,4-dichlorophenyl
fluoromethyl



1.2.1219
3-bromo-4-chlorophenyl
fluoromethyl



1.2.1220
3-methyl-4-chlorophenyl
fluoromethyl



1.2.1221
3-cyclopropyl-4-chlorophenyl
fluoromethyl



1.2.1222
3-cyano-4-chlorophenyl
fluoromethyl



1.2.1223
3-trifluoromethyl-4-chlorophenyl
fluoromethyl



1.2.1224
3-methoxy-4-chlorophenyl
fluoromethyl



1.2.1225
3-ethoxy-4-chlorophenyl
fluoromethyl



1.2.1226
3-trifluoromethoxy-4-chlorophenyl
fluoromethyl



1.2.1227
3-nitro-4-chlorophenyl
fluoromethyl



1.2.1228
3-fluoro-4-bromophenyl
fluoromethyl



1.2.1229
3-chloro-4-bromophenyl
fluoromethyl



1.2.1230
3,4-dibromophenyl
fluoromethyl



1.2.1231
3-methyl-4-bromophenyl
fluoromethyl



1.2.1232
3-ethyl-4-bromophenyl
fluoromethyl



1.2.1233
3-cyclopropyl-4-bromophenyl
fluoromethyl



1.2.1234
3-cyano-4-bromophenyl
fluoromethyl



1.2.1235
3-trifluoromethyl-4-bromophenyl
fluoromethyl



1.2.1236
3-methoxy-4-phenyl
fluoromethyl



1.2.1237
3-ethoxy-4-bromophenyl
fluoromethyl



1.2.1238
3-trifluoromethoxy-4-bromophenyl
fluoromethyl



1.2.1239
3-nitro-4-bromophenyl
fluoromethyl



1.2.1240
3-fluoro-4-iodophenyl
fluoromethyl



1.2.1241
3-chloro-4-iodophenyl
fluoromethyl



1.2.1242
3-bromo-4-iodophenyl
fluoromethyl



1.2.1243
3-methyl-4-iodophenyl
fluoromethyl



1.2.1244
3-ethyl-4-iodophenyl
fluoromethyl



1.2.1245
3-cyclopropyl-4-iodophenyl
fluoromethyl



1.2.1246
3-cyano-4-iodophenyl
fluoromethyl



1.2.1247
3-trifluoromethyl-4-iodophenyl
fluoromethyl



1.2.1248
3-methoxy-4-iodophenyl
fluoromethyl



1.2.1249
3-ethoxy-4-iodophenyl
fluoromethyl



1.2.1250
3-trifluoromethoxy-4-iodophenyl
fluoromethyl



1.2.1251
3-nitro-4-iodophenyl
fluoromethyl



1.2.1252
3-fluoro-4-methylphenyl
fluoromethyl



1.2.1253
3-chloro-4-methylphenyl
fluoromethyl



1.2.1254
3-bromo-4-methylphenyl
fluoromethyl



1.2.1255
3,4-dimethylphenyl
fluoromethyl



1.2.1256
3,4-dimethylphenyl
chloromethyl



1.2.1257
3,4-dimethylphenyl
bromomethyl



1.2.1258
3,4-dimethylphenyl
difluoromethyl



1.2.1259
3,4-dimethylphenyl
trifluoromethyl



1.2.1260
3,4-dimethylphenyl
cyano



1.2.1261
3-ethyl-4-methylphenyl
fluoromethyl



1.2.1262
3-cyclopropyl-4-methylphenyl
fluoromethyl



1.2.1263
3-cyano-4-methylphenyl
fluoromethyl



1.2.1264
3-trifluoromethyl-4-methylphenyl
fluoromethyl



1.2.1265
3-methoxy-4-methylphenyl
fluoromethyl



1.2.1266
3-ethoxy-4-methylphenyl
fluoromethyl



1.2.1267
3-trifluoromethoxy-4-methylphenyl
fluoromethyl



1.2.1268
3-nitro-4-methylphenyl
fluoromethyl



1.2.1269
3-fluoro-4-ethylphenyl
fluoromethyl



1.2.1270
3-chloro-4-ethylphenyl
fluoromethyl



1.2.1271
3-bromo-4-ethylphenyl
fluoromethyl



1.2.1272
3-methyl-4-ethylphenyl
fluoromethyl



1.2.1273
3,4-diethylphenyl
fluoromethyl



1.2.1274
3-cyclopropyl-4-ethylphenyl
fluoromethyl



1.2.1275
3-cyano-4-ethylphenyl
fluoromethyl



1.2.1276
3-trifluoromethyl-4-ethylphenyl
fluoromethyl



1.2.1277
3-methoxy-4-ethylphenyl
fluoromethyl



1.2.1278
3-ethoxy-4-ethylphenyl
fluoromethyl



1.2.1279
3-trifluoromethoxy-4-ethylphenyl
fluoromethyl



1.2.1280
3-nitro-4-ethylphenyl
fluoromethyl



1.2.1281
3-fluoro-4-propylphenyl
fluoromethyl



1.2.1282
3-chloro-4-propylphenyl
fluoromethyl



1.2.1283
3-bromo-4-propylphenyl
fluoromethyl



1.2.1284
3-methyl-4-propylphenyl
fluoromethyl



1.2.1285
3-cyclopropyl-4-propylphenyl
fluoromethyl



1.2.1286
3-cyano-4-propylphenyl
fluoromethyl



1.2.1287
3-trifluoromethyl-4-propylphenyl
fluoromethyl



1.2.1288
3-methoxy-4-propylphenyl
fluoromethyl



1.2.1289
3-ethoxy-4-propylphenyl
fluoromethyl



1.2.1290
3-trifluoromethoxy-4-propylphenyl
fluoromethyl



1.2.1291
3-nitro-4-propylphenyl
fluoromethyl



1.2.1292
3-fluoro-4-isopropylphenyl
fluoromethyl



1.2.1293
3-chloro-4-isopropylphenyl
fluoromethyl



1.2.1294
3-bromo-4-isopropylphenyl
fluoromethyl



1.2.1295
3-methyl-4-isopropylphenyl
fluoromethyl



1.2.1296
3-ethyl-4-isopropylphenyl
fluoromethyl



1.2.1297
3-cyclopropyl-4-isopropylphenyl
fluoromethyl



1.2.1298
3-cyano-4-isopropylphenyl
fluoromethyl



1.2.1299
3-trifluoromethyl-4-isopropylphenyl
fluoromethyl



1.2.1300
3-methoxy-4-isopropylphenyl
fluoromethyl



1.2.1301
3-ethoxy-4-isopropylphenyl
fluoromethyl



1.2.1302
3-trifluoromethoxy-4-
fluoromethyl




isopropylphenyl




1.2.1303
3-nitro-4-isopropylphenyl
fluoromethyl



1.2.1304
3-fluoro-4-tert-butylphenyl
fluoromethyl



1.2.1305
3-chloro-4-tert-butylphenyl
fluoromethyl



1.2.1306
3-bromo-4-tert-butylphenyl
fluoromethyl



1.2.1307
3-methyl-4-tert-butylphenyl
fluoromethyl



1.2.1308
3-cyclopropyl-4-tert-butylphenyl
fluoromethyl



1.2.1309
3-cyano-4-tert-butylphenyl
fluoromethyl



1.2.1310
3-trifluoromethyl-4-tert-butylphenyl
fluoromethyl



1.2.1311
3-trifluoromethyl-4-tert-butylphenyl
chloromethyl



1.2.1312
3-trifluoromethyl-4-tert-butylphenyl
bromomethyl



1.2.1313
3-trifluoromethyl-4-tert-butylphenyl
difluoromethyl



1.2.1314
3-methoxy-4-tert-butylphenyl
fluoromethyl



1.2.1315
3-ethoxy-4-tert-butylphenyl
fluoromethyl



1.2.1316
3-trifluoromethoxy-4-tert-
fluoromethyl




butylphenyl




1.2.1317
3-nitro-4-tert-butylphenyl
fluoromethyl



1.2.1318
3-fluoro-4-cyclopropylphenyl
fluoromethyl



1.2.1319
3-chloro-4-cyclopropylphenyl
fluoromethyl



1.2.1320
3-bromo-4-cyclopropylphenyl
fluoromethyl



1.2.1321
3-methyl-4-cyclopropylphenyl
fluoromethyl



1.2.1322
3-ethyl-4-cyclopropylphenyl
fluoromethyl



1.2.1323
3-cyclopropyl-4-cyclopropylphenyl
fluoromethyl



1.2.1324
3-cyano-4-cyclopropylphenyl
fluoromethyl



1.2.1325
3-trifluoromethyl-4-
fluoromethyl




cyclopropylphenyl




1.2.1326
3-methoxy-4-cyclopropylphenyl
fluoromethyl



1.2.1327
3-ethoxy-4-cyclopropylphenyl
fluoromethyl



1.2.1328
3-trifluoromethoxy-4-
fluoromethyl




cyclopropylphenyl




1.2.1329
3-fluoro-4-methoxycarbonyl-phenyl
fluoromethyl



1.2.1330
3-chloro-4-methoxycarbonylphenyl
fluoromethyl



1.2.1331
3-bromo-4-methoxycarbonylphenyl
fluoromethyl



1.2.1332
3-methyl-4-methoxycarbonylphenyl
fluoromethyl



1.2.1333
3-cyclopropyl-4-methoxycarbonyl-
fluoromethyl




phenyl




1.2.1334
3-cyano-4-methoxycarbonylphenyl
fluoromethyl



1.2.1335
3-trifluoromethyl-4-
fluoromethyl




methoxycarbonyl-phenyl




1.2.1336
3-methoxy-4-methoxycarbonyl-
fluoromethyl




phenyl




1.2.1337
3-ethoxy-4-methoxycarbonyl-phenyl
fluoromethyl



1.2.1338
3-trifluoromethoxy-4-
fluoromethyl




methoxycarbonyl-phenyl




1.2.1339
3-nitro-4-methoxycarbonylphenyl
fluoromethyl



1.2.1340
3-fluoro-4-cyanophenyl
fluoromethyl



1.2.1341
3-chloro-4-cyanophenyl
fluoromethyl



1.2.1342
3-bromo-4-cyanophenyl
fluoromethyl



1.2.1343
3-methyl-4-cyanophenyl
fluoromethyl



1.2.1344
3-cyclopropyl-4-cyanophenyl
fluoromethyl



1.2.1345
3,4-dicyanophenyl
fluoromethyl



1.2.1346
3-trifluoromethyl-4-cyanophenyl
fluoromethyl



1.2.1347
3-trifluoromethyl-4-cyanophenyl
chloromethyl



1.2.1348
3-trifluoromethyl-4-cyanophenyl
bromomethyl



1.2.1349
3-trifluoromethyl-4-cyanophenyl
difluoromethyl



1.2.1350
3-methoxy-4-cyanophenyl
fluoromethyl



1.2.1351
3-ethoxy-4-cyanophenyl
fluoromethyl



1.2.1352
3-trifluoromethoxy-4-cyanophenyl
fluoromethyl



1.2.1353
3-nitro-4-cyanophenyl
fluoromethyl



1.2.1354
3-fluoro-4-methoxyphenyl
fluoromethyl



1.2.1355
3-chloro-4-methoxyphenyl
fluoromethyl



1.2.1356
3-bromo-4-methoxyphenyl
fluoromethyl



1.2.1357
3-methyl-4-methoxyphenyl
fluoromethyl



1.2.1358
3-cyclopropyl-4-methoxyphenyl
fluoromethyl



1.2.1359
3-cyano-4-methoxyphenyl
fluoromethyl



1.2.1360
3-trifluoromethyl-4-methoxyphenyl
fluoromethyl



1.2.1361
3,4-dimethoxyphenyl
fluoromethyl



1.2.1362
3-ethoxy-4-methoxyphenyl
fluoromethyl



1.2.1363
3-trifluoromethoxy-4-
fluoromethyl




methoxyphenyl




1.2.1364
3-nitro-4-methoxyphenyl
fluoromethyl



1.2.1365
3-fluoro-4-ethoxyphenyl
fluoromethyl



1.2.1366
3-chloro-4-ethoxyphenyl
fluoromethyl



1.2.1367
3-chloro-4-ethoxyphenyl
chloromethyl



1.2.1368
3-chloro-4-ethoxyphenyl
bromomethyl



1.2.1369
3-chloro-4-ethoxyphenyl
difluoromethyl



1.2.1370
3-bromo-4-ethoxyphenyl
fluoromethyl



1.2.1371
3-methyl-4-ethoxyphenyl
fluoromethyl



1.2.1372
3-ethyl-4-ethoxyphenyl
fluoromethyl



1.2.1373
3-cyclopropyl-4-ethoxyphenyl
fluoromethyl



1.2.1374
3-cyano-4-ethoxyphenyl
fluoromethyl



1.2.1375
3-trifluoromethyl-4-ethoxyphenyl
fluoromethyl



1.2.1376
3-methoxy-4-ethoxyphenyl
fluoromethyl



1.2.1377
2,4-diethoxyphenyl
fluoromethyl



1.2.1378
3-trifluoromethoxy-4-ethoxyphenyl
fluoromethyl



1.2.1379
3-nitro-4-ethoxyphenyl
fluoromethyl



1.2.1380
3-fluoro-4-isopropoxyphenyl
fluoromethyl



1.2.1381
3-chloro-4-isopropoxyphenyl
fluoromethyl



1.2.1382
3-bromo-4-isopropoxyphenyl
fluoromethyl



1.2.1383
3-methyl-4-isopropoxyphenyl
fluoromethyl



1.2.1384
3-cyclopropyl-4-isopropoxyphenyl
fluoromethyl



1.2.1385
3-cyano-4-isopropoxyphenyl
fluoromethyl



1.2.1386
3-trifluoromethyl-4-
fluoromethyl




isopropoxyphenyl




1.2.1387
3-methoxy-4-isopropoxyphenyl
fluoromethyl



1.2.1388
3-ethoxy-4-isopropoxyphenyl
fluoromethyl



1.2.1389
3-trifluoromethoxy-4-
fluoromethyl




isopropoxyphenyl




1.2.1390
3-nitro-4-isopropoxyphenyl
fluoromethyl



1.2.1391
3-fluoro-4-trifluoromethoxyphenyl
fluoromethyl



1.2.1392
3-chloro-4-trifluoromethoxyphenyl
fluoromethyl



1.2.1393
3-bromo-4-trifluoromethoxyphenyl
fluoromethyl



1.2.1394
3-methyl-4-trifluoromethoxyphenyl
fluoromethyl



1.2.1395
3-cyclopropyl-4-trifluoromethoxy-
fluoromethyl




phenyl




1.2.1396
3-cyano-4-trifluoromethoxyphenyl
fluoromethyl



1.2.1397
3-trifluoromethyl-4-trifluoromethoxy-
fluoromethyl




phenyl




1.2.1398
3-methoxy-4-trifluoromethoxy-
fluoromethyl




phenyl




1.2.1399
3-ethoxy-4-trifluoromethoxyphenyl
fluoromethyl



1.2.1400
3,4-bis(trifluoromethoxy)phenyl
fluoromethyl



1.2.1401
3-nitro-4-trifluoromethoxyphenyl
fluoromethyl



1.2.1402
3-fluoro-4-difluoromethoxyphenyl
fluoromethyl



1.2.1403
3-chloro-4-difluoromethoxyphenyl
fluoromethyl



1.2.1404
3-bromo-4-difluoromethoxyphenyl
fluoromethyl



1.2.1405
3-methyl-4-difluoromethoxyphenyl
fluoromethyl



1.2.1406
3-cyclopropyl-4-difluoromethoxy-
fluoromethyl




phenyl




1.2.1407
3-cyano-4-difluoromethoxyphenyl
fluoromethyl



1.2.1408
3-trifluoromethyl-4-difluoromethoxy-
fluoromethyl




phenyl




1.2.1409
3-methoxy-4-difluoromethoxy-
fluoromethyl




phenyl




1.2.1410
3-ethoxy-4-difluoromethoxyphenyl
fluoromethyl



1.2.1411
3-trifluoromethoxy-4-
fluoromethyl




difluoromethoxyphenyl




1.2.1412
3-nitro-4-difluoromethoxyphenyl
fluoromethyl



1.2.1413
3-fluoro-4-nitrophenyl
fluoromethyl



1.2.1414
3-chloro-4-nitrophenyl
fluoromethyl



1.2.1415
3-bromo-4-nitrophenyl
fluoromethyl



1.2.1416
3-methyl-4-nitrophenyl
fluoromethyl



1.2.1417
3-ethyl-4-nitrophenyl
fluoromethyl



1.2.1418
3-cyclopropyl-4-nitrophenyl
fluoromethyl



1.2.1419
3-cyano-4-nitrophenyl
fluoromethyl



1.2.1420
3-trifluoromethyl-4-nitrophenyl
fluoromethyl



1.2.1421
3-methoxy-4-nitrophenyl
fluoromethyl



1.2.1422
3-ethoxy-4-nitrophenyl
fluoromethyl



1.2.1423
3-trifluoromethoxy-4-nitrophenyl
fluoromethyl



1.2.1424
3-fluoro-4-methylsulfanylphenyl
fluoromethyl



1.2.1425
3-chloro-4-methylsulfanylphenyl
fluoromethyl



1.2.1426
3-bromo-4-methylsulfanylphenyl
fluoromethyl



1.2.1427
3-methyl-4-methylsulfanylphenyl
fluoromethyl



1.2.1428
3-ethyl-4-methylsulfanylphenyl
fluoromethyl



1.2.1429
3-cyclopropyl-4-
fluoromethyl




methylsulfanylphenyl




1.2.1430
3-cyano-4-methylsulfanylphenyl
fluoromethyl



1.2.1431
3-trifluoromethyl-4-
fluoromethyl




methylsulfanylphenyl




1.2.1432
3-methoxy-4-methylsulfanylphenyl
fluoromethyl



1.2.1433
3-ethoxy-4-methylsulfanylphenyl
fluoromethyl



1.2.1434
3-trifluoromethoxy-4-
fluoromethyl




methylsulfanylphenyl




1.2.1435
3-nitro-4-methylsulfanylphenyl
fluoromethyl



1.2.1436
3,6-difluorophenyl
fluoromethyl



1.2.1437
3,6-difluorophenyl
chloromethyl



1.2.1438
3,6-difluorophenyl
bromomethyl



1.2.1439
3,6-difluorophenyl
difluoromethyl



1.2.1440
3,6-difluorophenyl
trifluoromethyl



1.2.1441
3,6-difluorophenyl
cyano



1.2.1442
3-chloro-6-fluorophenyl
fluoromethyl



1.2.1443
3-bromo-6-fluorophenyl
fluoromethyl



1.2.1444
3-methyl-6-fluorophenyl
fluoromethyl



1.2.1445
3-cyclopropyl-6-fluorophenyl
fluoromethyl



1.2.1446
3-cyano-6-fluorophenyl
fluoromethyl



1.2.1447
3-methoxy-6-fluorophenyl
fluoromethyl



1.2.1448
3-ethoxy-6-fluorophenyl
fluoromethyl



1.2.1449
3-trifluoromethoxy-6-fluorophenyl
fluoromethyl



1.2.1450
3-nitro-6-fluorophenyl
fluoromethyl



1.2.1451
3-fluoro-6-chlorophenyl
fluoromethyl



1.2.1452
3-fluoro-6-chlorophenyl
chloromethyl



1.2.1453
3-fluoro-6-chlorophenyl
bromomethyl



1.2.1454
3-fluoro-6-chlorophenyl
difluoromethyl



1.2.1455
3,6-dichlorophenyl
fluoromethyl



1.2.1456
3,6-dichlorophenyl
chloromethyl



1.2.1457
3,6-dichlorophenyl
bromomethyl



1.2.1458
3,6-dichlorophenyl
difluoromethyl



1.2.1459
3,6-dichlorophenyl
trifluoromethyl



1.2.1460
3,6-dichlorophenyl
cyano



1.2.1461
3-bromo-6-chlorophenyl
fluoromethyl



1.2.1462
3-methyl-6-chlorophenyl
fluoromethyl



1.2.1463
3-cyclopropyl-6-chlorophenyl
fluoromethyl



1.2.1464
3-cyano-6-chlorophenyl
fluoromethyl



1.2.1465
3-trifluoromethyl-6-chlorophenyl
fluoromethyl



1.2.1466
3-methoxy-6-chlorophenyl
fluoromethyl



1.2.1467
3-ethoxy-6-chlorophenyl
fluoromethyl



1.2.1468
3-trifluoromethoxy-6-chlorophenyl
fluoromethyl



1.2.1469
3-nitro-6-chlorophenyl
fluoromethyl



1.2.1470
3-fluoro-6-bromophenyl
fluoromethyl



1.2.1471
3-chloro-6-bromophenyl
fluoromethyl



1.2.1472
3,6-dibromophenyl
fluoromethyl



1.2.1473
3-methyl-6-bromophenyl
fluoromethyl



1.2.1474
3-cyclopropyl-6-bromophenyl
fluoromethyl



1.2.1475
3-cyano-6-bromophenyl
fluoromethyl



1.2.1476
3-trifluoromethyl-6-bromophenyl
fluoromethyl



1.2.1477
3-methoxy-6-phenyl
fluoromethyl



1.2.1478
3-ethoxy-6-bromophenyl
fluoromethyl



1.2.1479
3-trifluoromethoxy-6-bromophenyl
fluoromethyl



1.2.1480
3-nitro-6-bromophenyl
fluoromethyl



1.2.1481
3-fluoro-6-iodophenyl
fluoromethyl



1.2.1482
3-chloro-6-iodophenyl
fluoromethyl



1.2.1483
3-bromo-6-iodophenyl
fluoromethyl



1.2.1484
3-methyl-6-iodophenyl
fluoromethyl



1.2.1485
3-cyclopropyl-6-iodophenyl
fluoromethyl



1.2.1486
3-cyano-6-iodophenyl
fluoromethyl



1.2.1487
3-trifluoromethyl-6-iodophenyl
fluoromethyl



1.2.1488
3-methoxy-6-iodophenyl
fluoromethyl



1.2.1489
3-ethoxy-6-iodophenyl
fluoromethyl



1.2.1490
3-trifluoromethoxy-6-iodophenyl
fluoromethyl



1.2.1491
3-nitro-6-iodophenyl
fluoromethyl



1.2.1492
3-fluoro-6-methylphenyl
fluoromethyl



1.2.1493
3-chloro-6-methylphenyl
fluoromethyl



1.2.1494
3-bromo-6-methylphenyl
fluoromethyl



1.2.1495
3,6-dimethylphenyl
fluoromethyl



1.2.1496
3-ethyl-6-methylphenyl
fluoromethyl



1.2.1497
3-cyclopropyl-6-methylphenyl
fluoromethyl



1.2.1498
3-cyano-6-methylphenyl
fluoromethyl



1.2.1499
3-trifluoromethyl-6-methylphenyl
fluoromethyl



1.2.1500
3-methoxy-6-methylphenyl
fluoromethyl



1.2.1501
3-ethoxy-6-methylphenyl
fluoromethyl



1.2.1502
3-trifluoromethoxy-6-methylphenyl
fluoromethyl



1.2.1503
3-nitro-6-methylphenyl
fluoromethyl



1.2.1504
3-fluoro-6-ethylphenyl
fluoromethyl



1.2.1505
3-chloro-6-ethylphenyl
fluoromethyl



1.2.1506
3-bromo-6-ethylphenyl
fluoromethyl



1.2.1507
3-methyl-6-ethylphenyl
fluoromethyl



1.2.1508
3,6-diethylphenyl
fluoromethyl



1.2.1509
3-cyclopropyl-6-ethylphenyl
fluoromethyl



1.2.1510
3-cyano-6-ethylphenyl
fluoromethyl



1.2.1511
3-trifluoromethyl-6-ethylphenyl
fluoromethyl



1.2.1512
3-methoxy-6-ethylphenyl
fluoromethyl



1.2.1513
3-ethoxy-6-ethylphenyl
fluoromethyl



1.2.1514
3-trifluoromethoxy-6-ethylphenyl
fluoromethyl



1.2.1515
3-nitro-6-ethylphenyl
fluoromethyl



1.2.1516
3-fluoro-6-propylphenyl
fluoromethyl



1.2.1517
3-chloro-6-propylphenyl
fluoromethyl



1.2.1518
3-bromo-6-propylphenyl
fluoromethyl



1.2.1519
3-methyl-6-propylphenyl
fluoromethyl



1.2.1520
3-cyclopropyl-6-propylphenyl
fluoromethyl



1.2.1521
3-cyano-6-propylphenyl
fluoromethyl



1.2.1522
3-trifluoromethyl-6-propylphenyl
fluoromethyl



1.2.1523
3-methoxy-6-propylphenyl
fluoromethyl



1.2.1524
3-ethoxy-6-propylphenyl
fluoromethyl



1.2.1525
3-trifluoromethoxy-6-propylphenyl
fluoromethyl



1.2.1526
3-nitro-6-propylphenyl
fluoromethyl



1.2.1527
3-fluoro-6-isopropylphenyl
fluoromethyl



1.2.1528
3-chloro-6-isopropylphenyl
fluoromethyl



1.2.1529
3-bromo-6-isopropylphenyl
fluoromethyl



1.2.1530
3-methyl-6-isopropylphenyl
fluoromethyl



1.2.1531
3-cyclopropyl-6-isopropylphenyl
fluoromethyl



1.2.1532
3-cyano-6-isopropylphenyl
fluoromethyl



1.2.1533
3-trifluoromethyl-6-isopropylphenyl
fluoromethyl



1.2.1534
3-methoxy-6-isopropylphenyl
fluoromethyl



1.2.1535
3-trifluoromethoxy-6-
fluoromethyl




isopropylphenyl




1.2.1536
3-nitro-6-isopropylphenyl
fluoromethyl



1.2.1537
3-fluoro-6-tert-butylphenyl
fluoromethyl



1.2.1538
3-chloro-6-tert-butylphenyl
fluoromethyl



1.2.1539
3-bromo-6-tert-butylphenyl
fluoromethyl



1.2.1540
3-methyl-6-tert-butylphenyl
fluoromethyl



1.2.1541
3-cyclopropyl-6-tert-butylphenyl
fluoromethyl



1.2.1542
3-cyano-6-tert-butylphenyl
fluoromethyl



1.2.1543
3-trifluoromethyl-6-tert-butylphenyl
fluoromethyl



1.2.1544
3-methoxy-6-tert-butylphenyl
fluoromethyl



1.2.1545
3-ethoxy-6-tert-butylphenyl
fluoromethyl



1.2.1546
3-trifluoromethoxy-6-tert-
fluoromethyl




butylphenyl




1.2.1547
3-nitro-6-tert-butylphenyl
fluoromethyl



1.2.1548
3-fluoro-6-cyclopropylphenyl
fluoromethyl



1.2.1549
3-chloro-6-cyclopropylphenyl
fluoromethyl



1.2.1550
3-bromo-6-cyclopropylphenyl
fluoromethyl



1.2.1551
3-methyl-6-cyclopropylphenyl
fluoromethyl



1.2.1552
3-cyclopropyl-6-cyclopropylphenyl
fluoromethyl



1.2.1553
3-cyano-6-cyclopropylphenyl
fluoromethyl



1.2.1554
3-trifluoromethyl-6-
fluoromethyl




cyclopropylphenyl




1.2.1555
3-methoxy-6-cyclopropylphenyl
fluoromethyl



1.2.1556
3-ethoxy-6-cyclopropylphenyl
fluoromethyl



1.2.1557
3-trifluoromethoxy-6-
fluoromethyl




cyclopropylphenyl




1.2.1558
3-fluoro-6-methoxycarbonyl-phenyl
fluoromethyl



1.2.1559
3-chloro-6-methoxycarbonyl-phenyl
fluoromethyl



1.2.1560
3-bromo-6-methoxycarbonyl-phenyl
fluoromethyl



1.2.1561
3-methyl-6-methoxycarbonyl-phenyl
fluoromethyl



1.2.1562
3-cyclopropyl-6-methoxycarbonyl-
fluoromethyl




phenyl




1.2.1563
3-cyano-6-methoxycarbonyl-phenyl
fluoromethyl



1.2.1564
3-trifluoromethyl-6-
fluoromethyl




methoxycarbonyl-phenyl




1.2.1565
3-methoxy-6-methoxycarbonyl-
fluoromethyl




phenyl




1.2.1566
3-ethoxy-6-methoxycarbonyl-phenyl
fluoromethyl



1.2.1567
3-trifluoromethoxy-6-
fluoromethyl




methoxycarbonyl-phenyl




1.2.1568
3-nitro-6-methoxycarbonyl-phenyl
fluoromethyl



1.2.1569
3-fluoro-6-cyanophenyl
fluoromethyl



1.2.1570
3-chloro-6-cyanophenyl
fluoromethyl



1.2.1571
3-bromo-6-cyanophenyl
fluoromethyl



1.2.1572
3-methyl-6-cyanophenyl
fluoromethyl



1.2.1573
3-cyclopropyl-6-cyanophenyl
fluoromethyl



1.2.1574
3-cyano-6-cyanophenyl
fluoromethyl



1.2.1575
3-trifluoromethyl-6-cyanophenyl
fluoromethyl



1.2.1576
3-methoxy-6-cyanophenyl
fluoromethyl



1.2.1577
3-ethoxy-6-cyanophenyl
fluoromethyl



1.2.1578
3-trifluoromethoxy-6-cyanophenyl
fluoromethyl



1.2.1579
3-nitro-6-cyanophenyl
fluoromethyl



1.2.1580
3-fluoro-6-methoxyphenyl
fluoromethyl



1.2.1581
3-chloro-6-methoxyphenyl
fluoromethyl



1.2.1582
3-bromo-6-methoxyphenyl
fluoromethyl



1.2.1583
3-methyl-6-methoxyphenyl
fluoromethyl



1.2.1584
3-cyclopropyl-6-methoxyphenyl
fluoromethyl



1.2.1585
3-cyano-6-methoxyphenyl
fluoromethyl



1.2.1586
3-trifluoromethyl-6-methoxyphenyl
fluoromethyl



1.2.1587
3,6-dimethoxyphenyl
fluoromethyl



1.2.1588
3-ethoxy-6-methoxyphenyl
fluoromethyl



1.2.1589
3-trifluoromethoxy-6-
fluoromethyl




methoxyphenyl




1.2.1590
3-nitro-6-methoxyphenyl
fluoromethyl



1.2.1591
3-fluoro-6-ethoxyphenyl
fluoromethyl



1.2.1592
3-chloro-6-ethoxyphenyl
fluoromethyl



1.2.1593
3-bromo-6-ethoxyphenyl
fluoromethyl



1.2.1594
3-methyl-6-ethoxyphenyl
fluoromethyl



1.2.1595
3-ethyl-6-ethoxyphenyl
fluoromethyl



1.2.1596
3-cyclopropyl-6-ethoxyphenyl
fluoromethyl



1.2.1597
3-cyano-6-ethoxyphenyl
fluoromethyl



1.2.1598
3-trifluoromethyl-6-ethoxyphenyl
fluoromethyl



1.2.1599
3-methoxy-6-ethoxyphenyl
fluoromethyl



1.2.1600
2,6-diethoxyphenyl
fluoromethyl



1.2.1601
3-trifluoromethoxy-6-ethoxyphenyl
fluoromethyl



1.2.1602
3-nitro-6-ethoxyphenyl
fluoromethyl



1.2.1603
3-fluoro-6-isopropoxyphenyl
fluoromethyl



1.2.1604
3-chloro-6-isopropoxyphenyl
fluoromethyl



1.2.1605
3-bromo-6-isopropoxyphenyl
fluoromethyl



1.2.1606
3-methyl-6-isopropoxyphenyl
fluoromethyl



1.2.1607
3-cyclopropyl-6-isopropoxyphenyl
fluoromethyl



1.2.1608
3-cyano-6-isopropoxyphenyl
fluoromethyl



1.2.1609
3-trifluoromethyl-6-
fluoromethyl




isopropoxyphenyl




1.2.1610
3-methoxy-6-isopropoxyphenyl
fluoromethyl



1.2.1611
3-ethoxy-6-isopropoxyphenyl
fluoromethyl



1.2.1612
3-trifluoromethoxy-6-
fluoromethyl




isopropoxyphenyl




1.2.1613
3-nitro-6-isopropoxyphenyl
fluoromethyl



1.2.1614
3-fluoro-6-trifluoromethoxyphenyl
fluoromethyl



1.2.1615
3-chloro-6-trifluoromethoxyphenyl
fluoromethyl



1.2.1616
3-bromo-6-trifluoromethoxyphenyl
fluoromethyl



1.2.1617
3-methyl-6-trifluoromethoxyphenyl
fluoromethyl



1.2.1618
3-cyclopropyl-6-trifluoromethoxy-
fluoromethyl




phenyl




1.2.1619
3-cyano-6-trifluoromethoxyphenyl
fluoromethyl



1.2.1620
3-trifluoromethyl-6-trifluoromethoxy-
fluoromethyl




phenyl




1.2.1621
3-methoxy-6-trifluoromethoxy-
fluoromethyl




phenyl




1.2.1622
3-ethoxy-6-trifluoromethoxyphenyl
fluoromethyl



1.2.1623
3,6-bis(trifluoromethoxy)phenyl
fluoromethyl



1.2.1624
3-nitro-6-trifluoromethoxyphenyl
fluoromethyl



1.2.1625
3-fluoro-6-difluoromethoxyphenyl
fluoromethyl



1.2.1626
3-chloro-6-difluoromethoxyphenyl
fluoromethyl



1.2.1627
3-bromo-6-difluoromethoxyphenyl
fluoromethyl



1.2.1628
3-methyl-6-difluoromethoxyphenyl
fluoromethyl



1.2.1629
3-cyclopropyl-6-difluoromethoxy-
fluoromethyl




phenyl




1.2.1630
3-cyano-6-difluoromethoxyphenyl
fluoromethyl



1.2.1631
3-trifluoromethyl-6-difluoromethoxy-
fluoromethyl




phenyl




1.2.1632
3-methoxy-6-difluoromethoxy-
fluoromethyl




phenyl




1.2.1633
3-ethoxy-6-difluoromethoxyphenyl
fluoromethyl



1.2.1634
3-trifluoromethoxy-6-
fluoromethyl




difluoromethoxyphenyl




1.2.1635
3-nitro-6-difluoromethoxyphenyl
fluoromethyl



1.2.1636
3-fluoro-6-nitrophenyl
fluoromethyl



1.2.1637
3-chloro-6-nitrophenyl
fluoromethyl



1.2.1638
3-bromo-6-nitrophenyl
fluoromethyl



1.2.1639
3-methyl-6-nitrophenyl
fluoromethyl



1.2.1640
3-cyclopropyl-6-nitrophenyl
fluoromethyl



1.2.1641
3-cyano-6-nitrophenyl
fluoromethyl



1.2.1642
3-trifluoromethyl-6-nitrophenyl
fluoromethyl



1.2.1643
3-methoxy-6-nitrophenyl
fluoromethyl



1.2.1644
3-ethoxy-6-nitrophenyl
fluoromethyl



1.2.1645
3-trifluoromethoxy-6-nitrophenyl
fluoromethyl



1.2.1646
3-fluoro-6-methylsulfanylphenyl
fluoromethyl



1.2.1647
3-chloro-6-methylsulfanylphenyl
fluoromethyl



1.2.1648
3-bromo-6-methylsulfanylphenyl
fluoromethyl



1.2.1649
3-methyl-6-methylsulfanylphenyl
fluoromethyl



1.2.1650
3-cyclopropyl-6-
fluoromethyl




methylsulfanylphenyl




1.2.1651
3-cyano-6-methylsulfanylphenyl
fluoromethyl



1.2.1652
3-trifluoromethyl-6-
fluoromethyl




methylsulfanylphenyl




1.2.1653
3-methoxy-6-methylsulfanylphenyl
fluoromethyl



1.2.1654
3-ethoxy-6-methylsulfanylphenyl
fluoromethyl



1.2.1655
3-trifluoromethoxy-6-
fluoromethyl




methylsulfanylphenyl




1.2.1656
3-nitro-6-methylsulfanylphenyl
fluoromethyl



1.2.1657
2,3,4-trifluorophenyl
fluoromethyl



1.2.1658
2,3,4-trichlorophenyl
fluoromethyl



1.2.1659
2,3,4-trimethylphenyl
fluoromethyl



1.2.1660
2-fluoro-2-chloro-5-
fluoromethyl




trifluoromethylphenyl




1.2.1661
2,3,5-trifluorophenyl
fluoromethyl



1.2.1662
2,3,5-trichlorophenyl
fluoromethyl



1.2.1663
2,3,5-trimethylphenyl
fluoromethyl



1.2.1664
2,3-dichloro-5-methoxyphenyl
fluoromethyl



1.2.1665
2,3,6-trifluorophenyl
fluoromethyl



1.2.1666
2,3,6-trichlorophenyl
fluoromethyl



1.2.1667
2,3,6-trimethylphenyl
fluoromethyl



1.2.1668
3,4,5-trifluorophenyl
fluoromethyl



1.2.1669
3,4,5-trichlorophenyl
fluoromethyl



1.2.1670
3,4,5-trimethylphenyl
fluoromethyl



1.2.1671
3,5-dimethyl-4-fluorophenyl
fluoromethyl



1.2.1672
3,5-dichloro-4-methoxyphenyl
fluoromethyl



1.2.1673
3,5-difluoro-4-chlorophenyl
fluoromethyl



1.2.1674
3,5-dichloro-4-hydroxyphenyl
fluoromethyl



1.2.1675
3,5-trifluoromethyl-4-chlorophenyl
fluoromethyl



1.2.1676
3,4,6-trifluorophenyl
fluoromethyl



1.2.1677
3,4,6-trichlorophenyl
fluoromethyl



1.2.1678
3,4,6-trimethylphenyl
fluoromethyl



1.2.1679
pentafluorophenyl
fluoromethyl
















TABLE 1.3







Inventive compounds of the general formula (I) in which W* is COOH, R1


and R2 are each hydrogen, and aryl is the radical.








 








 










No.
Aryl
R3
Physical data





1.3.1
3-fluorophenyl
vinyl
[CDCl3] 3.44 (d, 1H);





3.96 (d, 1H); 5.44





(d, 1H); 5.63 (d, 1H);





6.16 (dd, 1H); 7.10-





7.20 (m, 1H); 7.37-





7.45 (m, 2H).


1.3.2
3-fluorophenyl
1-methylvinyl



1.3.3
3-fluorophenyl
allyl



1.3.4
3-fluorophenyl
1-chlorovinyl
[CDCl3] 3.66 (d, 1H);





4.16 (d, 1H); 5.61





(s, 1H); 5.95 (s, 1H);





7.13-7.20 (m, 1H);





7.39-7.45 (m, 2H).


1.3.5
3-fluorophenyl
ethynyl



1.3.6
3-chlorophenyl
vinyl



1.3.7
3-chlorophenyl
1-methylvinyl



1.3.8
3-chlorophenyl
allyl



1.3.9
3-chlorophenyl
1-chlorovinyl



1.3.10
3-chlorophenyl
ethynyl



1.3.11
3-bromophenyl
vinyl



1.3.12
3-bromophenyl
1-methylvinyl



1.3.13
3-iodophenyl
vinyl



1.3.14
3-iodophenyl
1-methylvinyl



1.3.15
3-methylphenyl
vinyl



1.3.16
3-methylphenyl
1-methylvinyl



1.3.17
3-ethylphenyl
vinyl



1.3.18
3-propylphenyl
vinyl



1.3.19
3-isopropylphenyl
vinyl



1.3.20
3-n-butylphenyl
vinyl



1.3.21
3-i-butylphenyl
vinyl



1.3.22
3-tert-butylphenyl
vinyl



1.3.23
3-cyclopropylphenyl
vinyl



1.3.24
3-cyclobutylphenyl
vinyl



1.3.25
3-cyclopentylphenyl
vinyl



1.3.26
3-vinylphenyl
vinyl



1.3.27
3-ethynylphenyl
vinyl



1.3.28
3-cyanophenyl
vinyl



1.3.29
3-trifluoromethylphenyl
vinyl



1.3.30
3-difluoromethylphenyl
vinyl



1.3.31
3-(hydroxycarbonyl)phenyl
vinyl



1.3.32
3-(methoxycarbonyl)phenyl
vinyl



1.3.33
3-(ethoxycarbonyl)phenyl
vinyl



1.3.34
3-hydroxymethylphenyl
vinyl



1.3.35
3-carbamoylphenyl
vinyl



1.3.36
3-hydroxyphenyl
vinyl



1.3.37
3-methoxyphenyl
vinyl



1.3.38
3-ethoxyphenyl
vinyl



1.3.39
3-propyloxyphenyl
vinyl



1.3.40
3-isopropyloxyphenyl
vinyl



1.3.41
3-n-butyloxyphenyl
vinyl



1.3.42
3-i-butyloxyphenyl
vinyl



1.3.43
3-t-butyloxyphenyl
vinyl



1.3.44
3-difluoromethoxyphenyl
vinyl



1.3.45
3-trifluoromethoxyphenyl
vinyl



1.3.46
3-(2,2,2-trifluoroethoxy)phenyl
vinyl



1.3.47
3-(2-chloroethoxy)phenyl
vinyl



1.3.48
3-(2-hydroxyethoxy)phenyl
vinyl



1.3.49
3-(2-methoxyethoxy)phenyl
vinyl



1.3.50
3-[(tert-butoxycarbonyl)oxy]phenyl
vinyl



1.3.51
3-nitrophenyl
vinyl



1.3.52
3-acetoxyphenyl
vinyl



1.3.53
{3-[(tert-butoxycarbonyl)amino]phenyl)
vinyl



1.3.54
3-methylsulfanylphenyl
vinyl



1.3.55
3-ethylsulfanylphenyl
vinyl



1.3.56
3-(pentafluoro-lambda6-sulfanyl)phenyl
vinyl



1.3.57
2,3-difluorophenyl
vinyl



1.3.58
2,3-difluorophenyl
1-methylvinyl



1.3.59
2,3-difluorophenyl
allyl



1.3.60
2,3-difluorophenyl
1-chlorovinyl



1.3.61
2,3-difluorophenyl
ethynyl



1.3.62
2-chloro-3-fluorophenyl
vinyl



1.3.63
2-bromo-3-fluorophenyl
vinyl



1.3.64
2-methyl-3-fluorophenyl
vinyl



1.3.65
2-ethyl-3-fluorophenyl
vinyl



1.3.66
2-cyclopropyl-3-fluorophenyl
vinyl



1.3.67
2-vinyl-3-fluorophenyl
vinyl



1.3.68
2-ethynyl-3-fluorophenyl
vinyl



1.3.69
2-cyano-3-fluorophenyl
vinyl



1.3.70
2-methoxy-3-fluorophenyl
vinyl



1.3.71
2-ethoxy-3-fluorophenyl
vinyl



1.3.72
2-trifluoromethoxy-3-fluorophenyl
vinyl



1.3.73
2-nitro-3-fluorophenyl
vinyl



1.3.74
2-fluoro-3-chlorophenyl
vinyl



1.3.75
2,3-dichlorophenyl
vinyl



1.3.76
2,3-dichlorophenyl
1-methylvinyl



1.3.77
2,3-dichlorophenyl
allyl



1.3.78
2,3-dichlorophenyl
1-chlorovinyl



1.3.79
2,3-dichlorophenyl
ethynyl



1.3.80
2-bromo-3-chlorophenyl
vinyl



1.3.81
2-methyl-3-chlorophenyl
vinyl



1.3.82
2-ethyl-3-chlorophenyl
vinyl



1.3.83
2-cyclopropyl-3-chlorophenyl
vinyl



1.3.84
2-vinyl-3-chlorophenyl
vinyl



1.3.85
2-ethynyl-3-chlorophenyl
vinyl



1.3.86
2-cyano-3-chlorophenyl
vinyl



1.3.87
2-trifluoromethyl-2-chlorophenyl
vinyl



1.3.88
2-methoxy-3-chlorophenyl
vinyl



1.3.89
2-ethoxy-3-chlorophenyl
vinyl



1.3.90
2-trifluoromethoxy-3-chlorophenyl
vinyl



1.3.91
2-nitro-3-chlorophenyl
vinyl



1.3.92
2-fluoro-3-bromophenyl
vinyl



1.3.93
2-chloro-3-bromophenyl
vinyl



1.3.94
2,3-dibromophenyl
vinyl



1.3.95
2-methyl-3-bromophenyl
vinyl



1.3.96
2-ethyl-3-bromophenyl
vinyl



1.3.97
2-cyclopropyl-3-bromophenyl
vinyl



1.3.98
2-vinyl-3-bromophenyl
vinyl



1.3.99
2-ethynyl-3-bromophenyl
vinyl



1.3.100
2-cyano-3-bromophenyl
vinyl



1.3.101
2-trifluoromethyl-3-bromophenyl
vinyl



1.3.102
2-methoxy-3-phenyl
vinyl



1.3.103
2-ethoxy-3-bromophenyl
vinyl



1.3.104
2-trifluoromethoxy-3-bromophenyl
vinyl



1.3.105
2-nitro-3-bromophenyl
vinyl



1.3.106
2-fluoro-3-iodophenyl
vinyl



1.3.107
2-chloro-3-iodophenyl
vinyl



1.3.108
2-bromo-3-iodophenyl
vinyl



1.3.109
2-methyl-3-iodophenyl
vinyl



1.3.110
2-ethyl-3-iodophenyl
vinyl



1.3.111
2-cyclopropyl-3-iodophenyl
vinyl



1.3.112
2-vinyl-3-iodophenyl
vinyl



1.3.113
2-ethynyl-3-iodophenyl
vinyl



1.3.114
2-cyano-3-iodophenyl
vinyl



1.3.115
2-trifluoromethyl-3-iodophenyl
vinyl



1.3.116
2-methoxy-3-iodophenyl
vinyl



1.3.117
2-ethoxy-3-iodophenyl
vinyl



1.3.118
2-trifluoromethoxy-3-iodophenyl
vinyl



1.3.119
2-nitro-3-iodophenyl
vinyl



1.3.120
2-fluoro-3-methylphenyl
vinyl



1.3.121
2-fluoro-3-methylphenyl
1-methylvinyl



1.3.122
2-fluoro-3-methylphenyl
allyl



1.3.123
2-fluoro-3-methylphenyl
1-chlorovinyl



1.3.124
2-fluoro-3-methylphenyl
ethynyl



1.3.125
2-chloro-3-methylphenyl
vinyl



1.3.126
2-chloro-3-methylphenyl
1-methylvinyl



1.3.127
2-chloro-3-methylphenyl
allyl



1.3.128
2-chloro-3-methylphenyl
1-chlorovinyl



1.3.129
2-chloro-3-methylphenyl
ethynyl



1.3.130
2-bromo-3-methylphenyl
vinyl



1.3.131
2,3-dimethylphenyl
vinyl



1.3.132
2,3-dimethylphenyl
1-methylvinyl



1.3.133
2,3-dimethylphenyl
allyl



1.3.134
2,3-dimethylphenyl
1-chlorovinyl



1.3.135
2,3-dimethylphenyl
ethynyl



1.3.136
2-ethyl-3-methylphenyl
vinyl



1.3.137
2-cyclopropyl-3-methylphenyl
vinyl



1.3.138
2-vinyl-3-methylphenyl
vinyl



1.3.139
2-ethynyl-3-methylphenyl
vinyl



1.3.140
2-cyano-3-methylphenyl
vinyl



1.3.141
2-trifluoromethyl-3-methylphenyl
vinyl



1.3.142
2-methoxy-3-methylphenyl
vinyl



1.3.143
2-ethoxy-3-methylphenyl
vinyl



1.3.144
2-trifluoromethoxy-3-methylphenyl
vinyl



1.3.145
2-nitro-3-methylphenyl
vinyl



1.3.146
2-fluoro-3-ethylphenyl
vinyl



1.3.147
2-chloro-3-ethylphenyl
vinyl



1.3.148
2-bromo-3-ethylphenyl
vinyl



1.3.149
2-methyl-3-ethylphenyl
vinyl



1.3.150
2,3-diethylphenyl
vinyl



1.3.151
2-cyclopropyl-3-ethylphenyl
vinyl



1.3.152
2-vinyl-3-ethylphenyl
vinyl



1.3.153
2-ethynyl-3-ethylphenyl
vinyl



1.3.154
2-cyano-3-ethylphenyl
vinyl



1.3.155
2-trifluoromethyl-3-ethylphenyl
vinyl



1.3.156
2-methoxy-3-ethylphenyl
vinyl



1.3.157
2-ethoxy-3-ethylphenyl
vinyl



1.3.158
2-trifluoromethoxy-3-ethylphenyl
vinyl



1.3.159
2-nitro-3-ethylphenyl
vinyl



1.3.160
2-fluoro-3-propylphenyl
vinyl



1.3.161
2-chloro-3-propylphenyl
vinyl



1.3.162
2-bromo-3-propylphenyl
vinyl



1.3.163
2-methyl-3-propylphenyl
vinyl



1.3.164
2-methyl-3-propylphenyl
vinyl



1.3.165
2-cyclopropyl-3-propylphenyl
vinyl



1.3.166
2-vinyl-3-propylphenyl
vinyl



1.3.167
2-ethynyl-3propylphenyl
vinyl



1.3.168
2-cyano-3-propylphenyl
vinyl



1.3.169
2-trifluoromethyl-3-propylphenyl
vinyl



1.3.170
2- methoxy-3-propylphenyl
vinyl



1.3.171
2-ethoxy-3-propylphenyl
vinyl



1.3.172
2-trifluoromethoxy-3-propyl phenyl
vinyl



1.3.173
2-nitro-3-propylphenyl
vinyl



1.3.174
2-fluoro-3-isopropylphenyl
vinyl



1.3.175
2-chloro-3-isopropylphenyl
vinyl



1.3.176
2-bromo-3- isopropylphenyl
vinyl



1.3.177
2-methyl-3-isopropylphenyl
vinyl



1.3.178
2-ethyl-3-isopropylphenyl
vinyl



1.3.179
2-cyclopropyl-3-isopropylphenyl
vinyl



1.3.180
2-vinyl-3-isopropylphenyl
vinyl



1.3.181
2-ethynyl-3-isopropylphenyl
vinyl



1.3.182
2-cyano-3-isopropylphenyl
vinyl



1.3.183
2-trifluoromethyl-3-isopropylphenyl
vinyl



1.3.184
2-methoxy-3-isopropylphenyl
vinyl



1.3.185
2-ethoxy-3-isopropylphenyl
vinyl



1.3.186
2-trifluoromethoxy-3-isopropylphenyl
vinyl



1.3.187
2-n itro-3-isopropylphenyl
vinyl



1.3.188
2-fluoro-3-tert-butylphenyl
vinyl



1.3.189
2-chloro-3-tert-butylphenyl
vinyl



1.3.190
2-bromo-3-tert-butylphenyl
vinyl



1.3.191
2-methyl-3-tert-butylphenyl
vinyl



1.3.192
2-ethyl-3-tert-butylphenyl
vinyl



1.3.193
2-cyclopropyl-3-tert-butylphenyl
vinyl



1.3.194
2-vinyl-3-tert-butylphenyl
vinyl



1.3.195
2-ethynyl-3-tert-butylphenyl
vinyl



1.3.196
2-cyano-3-tert-butylphenyl
vinyl



1.3.197
2-trifluoromethyl-3-tert-butylphenyl
vinyl



1.3.198
2- methoxy-3-tert-butylphenyl
vinyl



1.3.199
2-ethoxy-3-tert-butylphenyl
vinyl



1.3.200
2-trifluoromethoxy-3-tert-butylphenyl 
vinyl



1.3.201
2-nitro-3-tert-butylphenyl
vinyl



1.3.202
2-fluoro-3-hydroxymethylphenyl
vinyl



1.3.203
2-chloro-3-hydroxymethylphenyl
vinyl



1.3.204
2-bromo-3- hydroxymethylphenyl
vinyl



1.3.205
2-methyl-3-hydroxymethylphenyl
vinyl



1.3.206
2-ethyl-3-hydroxymethylphenyl
vinyl



1.3.207
2-cyclopropyl-3-hydroxymethylphenyl
vinyl



1.3.208
2-vinyl-3-hydroxymethylphenyl
vinyl



1.3.209
2-ethynyl-3-hydroxymethylphenyl
vinyl



1.3.210
2-cyano-3-hydroxymethylphenyl
vinyl



1.3.211
2-trifluoromethyl-3-hydroxymethylphenyl
vinyl



1.3.212
2-methoxy-3-hydroxymethylphenyl
vinyl



1.3.213
2-ethoxy-3-hydroxymethylphenyl
vinyl



1.3.214
2-trifluoromethoxy-3-hydroxymethylphenyl
vinyl



1.3.215
2-nitro-3-hydroxymethylphenyl
vinyl



1.3.216
2-fluoro-3-cyclopropylphenyl
vinyl



1.3.217
2-chloro-3-cyclopropylphenyl
vinyl



1.3.218
2-bromo-3-cyclopropylphenyl
vinyl



1.3.219
2-methyl-3-cyclopropylphenyl
vinyl



1.3.220
2-ethyl-3-cyclopropylphenyl
vinyl



1.3.221
2-cyclopropyl-3-cyclopropylphenyl
vinyl



1.3.222
2-vinyl-3-cyclopropylphenyl
vinyl



1.3.223
2-ethynyl-3-cyclopropylphenyl
vinyl



1.3.224
2-cyano-3-cyclopropylphenyl
vinyl



1.3.225
2-trifluoromethyl-3-cyclopropylphenyl
vinyl



1.3.226
2-methoxy-3-cyclopropylphenyl
vinyl



1.3.227
2-ethoxy-3-cyclopropylphenyl
vinyl



1.3.228
2-trifluoromethoxy-3-cyclopropylphenyl
vinyl



1.3.229
2-fluoro-3-methoxycarbonylphenyl
vinyl



1.3.230
2-chloro-3-methoxycarbonylphenyl
vinyl



1.3.231
2-bromo-3-methoxycarbonylphenyl
vinyl



1.3.232
2-methyl-3-methoxycarbonylphenyl
vinyl



1.3.233
2-ethyl-3-methoxycarbonylphenyl
vinyl



1.3.234
2-cyclopropyl-3-methoxycarbonylphenyl
vinyl



1.3.235
2-vinyl-3-methoxycarbonylphenyl
vinyl



1.3.236
2-ethynyl-3-methoxycarbonylphenyl
vinyl



1.3.237
2-cyano-3-methoxycarbonylphenyl
vinyl



1.3.238
2-trifluoromethyl-3-
vinyl




methoxycarbonylphenyl




1.3.239
2-methoxy-3-methoxycarbonylphenyl
vinyl



1.3.240
2-ethoxy-3-methoxycarbonylphenyl
vinyl



1.3.241
2-trifluoromethoxy-3-
vinyl




methoxycarbonylphenyl




1.3.242
2-nitro-3-methoxycarbonylphenyl
vinyl



1.3.243
2-fluoro-3-vinylphenyl
vinyl



1.3.244
2-chloro-3-vinylphenyl
vinyl



1.3.245
2-bromo-3-vinylphenyl
vinyl



1.3.246
2-methyl-3-vinylphenyl
vinyl



1.3.247
2-ethyl-3-vinylphenyl
vinyl



1.3.248
2-cyclopropyl-3-vinylphenyl
vinyl



1.3.249
2-vinyl-3-vinylphenyl
vinyl



1.3.250
2-ethynyl-3-vinylphenyl
vinyl



1.3.251
2-cyano-3-vinylphenyl
vinyl



1.3.252
2-trifluoromethyl-3-vinylphenyl
vinyl



1.3.253
2-methoxy-3-vinylphenyl
vinyl



1.3.254
2-ethoxy-3-vinylphenyl
vinyl



1.3.255
2-trifluoromethoxy-3-vinylphenyl
vinyl



1.3.256
2-nitro-3-vinylphenyl
vinyl



1.3.257
2-fluoro-3-ethynylphenyl
vinyl



1.3.258
2-chloro-3-ethynylphenyl
vinyl



1.3.259
2-bromo-3-ethynylphenyl
vinyl



1.3.260
2-methyl-3-ethynylphenyl
vinyl



1.3.261
2-ethyl-3-ethynylphenyl
vinyl



1.3.262
2-cyclopropyl-3-ethynylphenyl
vinyl



1.3.263
2-vinyl-3-ethynylphenyl
vinyl



1.3.264
2-cyano-3-ethynylphenyl
vinyl



1.3.265
2-trifluoromethyl-3-ethynylphenyl
vinyl



1.3.266
2-methoxy-3-ethynylphenyl
vinyl



1.3.267
2-ethoxy-3-ethynylphenyl
vinyl



1.3.268
2-trifluoromethoxy-3-ethynylphenyl
vinyl



1.3.269
2-nitro-3-ethynylphenyl
vinyl



1.3.270
2-fluoro-3-ethynylphenyl
vinyl



1.3.271
2-fluoro-3-cyanophenyl
vinyl



1.3.272
2-chloro-3-cyanophenyl
vinyl



1.3.273
2-bromo-3-cyanophenyl
vinyl



1.3.274
2-methyl-3-cyanophenyl
vinyl



1.3.275
2-ethyl-3-cyanophenyl
vinyl



1.3.276
2-ethyl-3-cyanophenyl
1-methylvinyl



1.3.277
2-ethyl-3-cyanophenyl
allyl



1.3.278
2-ethyl-3-cyanophenyl
1-chlorovinyl



1.3.279
2-ethyl-3-cyanophenyl
ethynyl



1.3.280
2-cyclopropyl-3-cyanophenyl
vinyl



1.3.281
2-vinyl-3-cyanophenyl
vinyl



1.3.282
2-ethynyl-3-cyanophenyl
vinyl



1.3.283
2-cyano-3-cyanophenyl
vinyl



1.3.284
2-trifluoromethyl-3-cyanophenyl
vinyl



1.3.285
2- methoxy-3-cyanophenyl
vinyl



1.3.286
2-ethoxy-3-cyanophenyl
vinyl



1.3.287
2-trifluoromethoxy-3-cyanophenyl
vinyl



1.3.288
2-nitro-3-cyanophenyl
vinyl



1.3.289
2-fluoro-3-hydroxyphenyl
vinyl



1.3.290
2-chloro-3-hydroxyphenyl
vinyl



1.3.291
2-bromo-3-hydroxyphenyl
vinyl



1.3.292
2- methyl-3-hydroxyphenyl
vinyl



1.3.293
2-ethyl-3-hydroxyphenyl
vinyl



1.3.294
2-cyclopropyl-3-hydroxyphenyl
vinyl



1.3.295
2-vinyl-3-hydroxyphenyl
vinyl



1.3.296
2-ethynyl-3-hydroxyphenyl
vinyl



1.3.297
2-cyano-3-hydroxyphenyl
vinyl



1.3.298
2-trifluoromethyl-3-hydroxyphenyl
vinyl



1.3.299
2-methoxy-3-hydroxyphenyl
vinyl



1.3.300
2-ethoxy-3-hydroxyphenyl
vinyl



1.3.301
2-trifluoromethoxy-3-hydroxyphenyl
vinyl



1.3.302
2-nitro-3-hydroxyphenyl
vinyl



1.3.303
2-fluoro-3-methoxyphenyl
vinyl



1.3.304
2-chloro-3-methoxyphenyl
vinyl



1.3.305
2-bromo-3-methoxyphenyl
vinyl



1.3.306
2-methyl-3-methoxyphenyl
vinyl



1.3.307
2-ethyl-3-methoxyphenyl
vinyl



1.3.308
2-cyclopropyl-3-methoxyphenyl
vinyl



1.3.309
2-vinyl-3-methoxyphenyl
vinyl



1.3.310
2-ethynyl-3-methoxyphenyl
vinyl



1.3.311
2-cyano-3-methoxyphenyl
vinyl



1.3.312
2-trifluoromethyl-3-methoxyphenyl
vinyl



1.3.313
2,3-dimethoxyphenyl
vinyl



1.3.314
2-ethoxy-3-methoxyphenyl
vinyl



1.3.315
2-trifluoromethoxy-3-methoxyphenyl
vinyl



1.3.316
2-nitro-3-methoxyphenyl
vinyl



1.3.317
2-fluoro-3-ethoxyphenyl
vinyl



1.3.318
2-chloro-3-ethoxyphenyl
vinyl



1.3.319
2-bromo-3-ethoxyphenyl
vinyl



1.3.320
2-methyl-3-ethoxyphenyl
vinyl



1.3.321
2-ethyl-3-ethoxyphenyl
vinyl



1.3.322
2-cyclopropyl-3-ethoxyphenyl
vinyl



1.3.323
2-vinyl-3-ethoxyphenyl
vinyl



1.3.324
2-ethynyl-3-ethoxyphenyl
vinyl



1.3.325
2-cyano-3-ethoxyphenyl
vinyl



1.3.326
2-trifluoromethyl-3-ethoxyphenyl
vinyl



1.3.327
2-methoxy-3-ethoxyphenyl
vinyl



1.3.328
2,3-diethoxy--phenyl
vinyl



1.3.329
2-trifluoromethoxy-3-ethoxyphenyl
vinyl



1.3.330
2-nitro-3-ethoxyphenyl
vinyl



1.3.331
2-fluoro-3-propoxyphenyl
vinyl



1.3.332
2-chloro-3-propoxyphenyl
vinyl



1.3.333
2-bromo-3-propoxyphenyl
vinyl



1.3.334
2-methyl-3-propoxyphenyl
vinyl



1.3.335
2-ethyl-3-propoxyphenyl
vinyl



1.3.336
2-cyclopropyl-3-propoxyphenyl
vinyl



1.3.337
2-vinyl-3-propoxyphenyl
vinyl



1.3.338
2-ethynyl-3-propoxyphenyl
vinyl



1.3.339
2-cyano-3-propoxyphenyl
vinyl



1.3.340
2-trifluoromethyl-3-propoxyphenyl
vinyl



1.3.341
2-methoxy-3-propoxyphenyl
vinyl



1.3.342
2-ethoxy-3-propoxyphenyl
vinyl



1.3.343
2-trifluoromethoxy-3-propoxyphenyl
vinyl



1.3.344
2-nitro-3-propoxyphenyl
vinyl



1.3.345
2-fluoro-3-isopropoxyphenyl
vinyl



1.3.346
2-chloro-3-isopropoxyphenyl
vinyl



1.3.347
2-bromo-3-isopropoxyphenyl
vinyl



1.3.348
2-methyl-3-isopropoxyphenyl
vinyl



1.3.349
2-ethyl-3-isopropoxyphenyl
vinyl



1.3.350
2-cyclopropyl-3-isopropoxyphenyl
vinyl



1.3.351
2-vinyl-3-isopropoxyphenyl
vinyl



1.3.352
2-ethynyl-3-isopropoxyphenyl
vinyl



1.3.353
2-cyano-3-isopropoxyphenyl
vinyl



1.3.354
2-trifluoromethyl-3-isopropoxyphenyl
vinyl



1.3.355
2-methoxy-3-isopropoxyphenyl
vinyl



1.3.356
2-ethoxy-3-isopropoxyphenyl
vinyl



1.3.357
2-trifluoromethoxy-3-isopropoxyphenyl
vinyl



1.3.358
2-nitro-3-isopropoxyphenyl
vinyl



1.3.359
2-fluoro-3-tert-butoxyphenyl
vinyl



1.3.360
2-chloro-3-tert-butoxyphenyl
vinyl



1.3.361
2-bromo-3-tert-butoxyphenyl
vinyl



1.3.362
2-methyl-3-tert-butoxyphenyl
vinyl



1.3.363
2-ethyl-3-tert-butoxyphenyl
vinyl



1.3.364
2-cyclopropyl-3-tert-butoxyphenyl
vinyl



1.3.365
2-vinyl-3-tert-butoxyphenyl
vinyl



1.3.366
2-ethynyl-3-tert-butoxyphenyl
vinyl



1.3.367
2-cyano-3-tert-butoxyphenyl
vinyl



1.3.368
2-trifluoromethyl-3-tert-butoxyphenyl
vinyl



1.3.369
2-methoxy-3-tert-butoxyphenyl
vinyl



1.3.370
2-ethoxy-3-tert-butoxyphenyl
vinyl



1.3.371
2-trifluoromethoxy-3-tert-butoxyphenyl
vinyl



1.3.372
2-nitro-3-tert-butoxyphenyl
vinyl



1.3.373
2-fluoro-3-trifluoromethoxyphenyl
vinyl



1.3.374
2-chloro-3-trifluoromethoxyphenyl
vinyl



1.3.375
2-bromo-3-trifluoromethoxyphenyl
vinyl



1.3.376
2-methyl-3-trifluoromethoxyphenyl
vinyl



1.3.377
2-ethyl-3-trifluoromethoxyphenyl
vinyl



1.3.378
2-cyclopropyl-3-trifluoromethoxyphenyl
vinyl



1.3.379
2-vinyl-3-trifluoromethoxyphenyl
vinyl



1.3.380
2-ethynyl-3-trifluoromethoxyphenyl
vinyl



1.3.381
2-cyano-3-trifluoromethoxyphenyl
vinyl



1.3.382
2-trifluoromethyl-3-trifluoromethoxy-
vinyl




phenyl




1.3.383
2-methoxy-3-trifluoromethoxyphenyl
vinyl



1.3.384
2-ethoxy-3-trifluoromethoxyphenyl
vinyl



1.3.385
2,3-bis(trifluoromethoxy)phenyl
vinyl



1.3.386
2-nitro-3-trifluoromethoxyphenyl
vinyl



1.3.387
2-fluoro-3-(2,2,2-trifluoroethoxy)phenyl
vinyl



1.3.388
2-chloro-3-(2,2,2-trifluoroethoxy)phenyl
vinyl



1.3.389
2-bromo-3-(2,2,2-trifluoroethoxy)phenyl
vinyl



1.3.390
2-methyl-3-(2,2,2-trifluoroethoxy)phenyl
vinyl



1.3.391
2-ethyl-3-(2,2,2-trifluoroethoxy)phenyl
vinyl



1.3.392
2-cyclopropyl-3-(2,2,2-trifluoro-
vinyl




ethoxy)phenyl




1.3.393
2-vinyl-3-(2,2,2-trifluoroethoxy)phenyl
vinyl



1.3.394
2-ethynyl-3-(2,2,2-trifluoroethoxyphenyl
vinyl



1.3.395
2-cyano-3-(2,2,2-trifluoroethoxy)phenyl
vinyl



1.3.396
2-trifluoromethyl-3-(2,2,2-trifluoro-
vinyl




ethoxy)phenyl




1.3.397
2-methoxy-3-(2,2,2-trifluoroethoxy)phenyl
vinyl



1.3.398
2-ethoxy-3-(2,2,2-trifluoroethoxy)phenyl
vinyl



1.3.399
2-trifluoromethoxy-3-(2,2,2-trifluoro-
vinyl




ethoxy)phenyl




1.3.400
2-nitro-3-(2,2,2-trifluoroethoxy)phenyl
vinyl



1.3.401
2-fluoro-3-difluoromethoxyphenyl
vinyl



1.3.402
2-chloro-3-difluoromethoxyphenyl
vinyl



1.3.403
2-bromo-3-difluoromethoxyphenyl
vinyl



1.3.404
2-methyl-3-difluoromethoxyphenyl
vinyl



1.3.405
2-ethyl-3-difluoromethoxyphenyl
vinyl



1.3.406
2-cyclopropyl-3-difluoromethoxyphenyl
vinyl



1.3.407
2-vinyl-3-difluoromethoxyphenyl
vinyl



1.3.408
2-ethynyl-3-difluoromethoxyphenyl
vinyl



1.3.409
2-cyano-3-difluoromethoxyphenyl
vinyl



1.3.410
2-trifluoromethyl-3-difluoromethoxyphenyl
vinyl



1.3.411
2-methoxy-3-difluoromethoxyphenyl
vinyl



1.3.412
2-ethoxy-3-difluoromethoxyphenyl
vinyl



1.3.413
2-trifluoromethoxy-3-difluoromethoxy-
vinyl




phenyl




1.3.414
2-nitro-3-difluoromethoxyphenyl
vinyl



1.3.415
2-fluoro-3-(2-methoxyethoxy)phenyl
vinyl



1.3.416
2-chloro-3-(2-methoxyethoxy)phenyl
vinyl



1.3.417
2-bromo-3-(2-methoxyethoxy)phenyl
vinyl



1.3.418
2-methyl-3-(2-methoxyethoxy)phenyl
vinyl



1.3.419
2-ethyl-3-(2-methoxyethoxy)phenyl
vinyl



1.3.420 
2-cyclopropyl-3-(2-methoxyethoxy)phenyl
vinyl



1.3.421
2-vinyl-3-(2-methoxyethoxy)phenyl
vinyl



1.3.422
2-ethynyl-3-(2-methoxyethoxy)phenyl
vinyl



1.3.423
2-cyano-3-(2-methoxyethoxy)phenyl
vinyl



1.3.424
2-trifluoromethyl-3-(2-methoxyethoxy)-
vinyl




phenyl




1.3.425
2-methoxy-3-(2-methoxyethoxy)phenyl
vinyl



1.3.426
2-ethoxy-3-(2-methoxyethoxy)phenyl
vinyl



1.3.427
2-trifluoromethoxy-(2-methoxyethoxy)-
vinyl




phenyl




1.3.428
2-nitro-3-(2-methoxyethoxy)phenyl
vinyl



1.3.429 
2-fluoro-3-(tert-butoxycarbonyloxy)phenyl
vinyl



1.3.430
2-chloro-3-(tert-butoxycarbonyloxy)-
vinyl




phenyl




1.3.431
2-bromo-3-(tert-butoxycarbonyl-
vinyl




oxy)phenyl




1.3.432
2-methyl-3-(tert-butoxycarbonyl-
vinyl




oxy)phenyl




1.3.433
2-ethyl-3-(tert-butoxycarbonyloxy)phenyl
vinyl



1.3.434
2-cyclopropyl-3-(tert-butoxycarbonyl-
vinyl




oxy)phenyl




1.3.435
2-vinyl-3-(tert-butoxycarbonyloxy)phenyl
vinyl



1.3.436
2-ethynyl-3-(tert-butoxycarbonyl-
vinyl




oxy)phenyl




1.3.437
2-cyano-3-(tert-butoxycarbonyloxy)-
vinyl




phenyl




1.3.438
2-trifluoromethyl-3-(tert-butoxycarbonyl-
vinyl




oxy)phenyl




1.3.439
2-methoxy-3-(tert-butoxycarbonyloxy)-
vinyl




phenyl




1.3.440
2-ethoxy-3-(tert-butoxycarbonyloxy)-
vinyl




phenyl




1.3.441
2-trifluoromethoxy-3-(tert-butoxycarbonyl-
vinyl




oxy)phenyl




1.3.442
2-nitro-3-(tert-butoxycarbonyloxy)phenyl
vinyl



1.3.443
2-fluoro-3-nitrophenyl
vinyl



1.3.444
2-chloro-3-nitrophenyl
vinyl



1.3.445
2-bromo-3-nitrophenyl
vinyl



1.3.446
2-methyl-3-nitrophenyl
vinyl



1.3.447
2-ethyl-3-nitrophenyl
vinyl



1.3.448
2-cyclopropyl-3-nitrophenyl
vinyl



1.3.449
2-vinyl-3-nitrophenyl
vinyl



1.3.450
2-ethynyl-3-nitrophenyl
vinyl



1.3.451
2-cyano-3-nitrophenyl
vinyl



1.3.452
2-trifluoromethyl-3-nitrophenyl
vinyl



1.3.453
2-methoxy-3-nitrophenyl
vinyl



1.3.454
2-ethoxy-3-nitrophenyl
vinyl



1.3.455
2-trifluoromethoxy-3-nitrophenyl
vinyl



1.3.456
2-fluoro-3-methylsulfanylphenyl
vinyl



1.3.457
2-chloro-3-methylsulfanylphenyl
vinyl



1.3.458
2-bromo-3-methylsulfanylphenyl
vinyl



1.3.459
2-methyl-3-methylsulfanylphenyl
vinyl



1.3.460
2-ethyl-3-methylsulfanylphenyl
vinyl



1.3.461
2-cyclopropyl-3-methylsulfanylphenyl
vinyl



1.3.462
2-vinyl-3-methylsulfanylphenyl
vinyl



1.3.463
2-ethynyl-3-methylsulfanylphenyl
vinyl



1.3.464
2-cyano-3-methylsulfanylphenyl
vinyl



1.3.465
2-trifluoromethyl-3-methylsulfanylphenyl
vinyl



1.3.466
2-methoxy-3-methylsulfanylphenyl
vinyl



1.3.467
2-ethoxy-3-methylsulfanylphenyl
vinyl



1.3.468
(R)- or (S)-3,5-difluorophenyl
vinyl
One unassigned





enantiomer [CDCl3]





3.41 (d, 1H); 3.93





(d, 1H); 5.45 (d, 1H);





5.63 (d, 1H); 6.16





(dd, 1H); 6.91 (t, 1H);





7.17 (d, 2H).


1.3.469
(S)- or (R)-3,5-difluorophenyl
vinyl
One unassigned





enantiomer





[CDCl3] 3.41 (d, 1H);





3.93 (d, 1H); 5.45





(d, 1H); 5.63 (d, 1H);





6.16 (dd, 1H); 6.91





(t, 1H); 7.17 (d, 2H).


1.3.470
3,5-difluorophenyl
vinyl
[CDCl3] 3.40 (d, 1H);





3.93 (d, 1H); 5.45





(d, 1H); 5.63 (d, 1H);





6.15 (dd, 1H); 6.90





(t, 1H); 7.18 (d, 2H).


1.3.471
3,5-difluorophenyl
1-methylvinyl



1.3.472
3,5-difluorophenyl
2,2-difluorovinyl
[CDCl3] 3.54 (d, 1H);





4.01 (d, 1H); 4.90





(d, 1H); 6.91 (t, 1H);





7.18 (d, 2H).


1.3.473
3,5-difluorophenyl
1-chlorovinyl
[CDCl3] 3.62 (d, 1H);





4.14 (d, 1H); 5.61





(d, 1H); 5.96 (d, 1H);





6.91 (t, 1H); 7.20





(d, 2H).


1.3.474
3,5-difluorophenyl
ethynyl
[CDCl3] 2.1 (s





br, 1H); 2.86 (s, 1H),





3.76 (d, 1H); 4.08





(d, 1H); 6.82 (t, 1H);





7.19 (d, 2H).


1.3.475
3-chloro-5-fluorophenyl
vinyl



1.3.476
3-chloro-5-fluorophenyl
1-methylvinyl
[CDCl3] 1.91 (s, 3H);





3.40 (d, 1H); 4.00





(d, 1H); 5.17 (s, 1H);





5.35 (s, 1H); 7.17





(d, 1H); 7.32 (d, 1H);





7.42 (s, 1H), 8.9 (s





br, 1H).


1.3.477
3-chloro-5-fluorophenyl
allyl



1.3.478
3-chloro-5-fluorophenyl
1-chlorovinyl



1.3.479
3-chloro-5-fluorophenyl
ethynyl



1.3.480
3-bromo-5-fluorophenyl
vinyl



1.3.481
3-bromo-5-fluorophenyl
1-methylvinyl



1.3.482
3-bromo-5-fluorophenyl
allyl



1.3.483
3-bromo-5-fluorophenyl
1-chlorovinyl



1.3.484
3-bromo-5-fluorophenyl
ethynyl



1.3.485
3-iodo-5-fluorophenyl
vinyl



1.3.486
3-methyl-5-fluorophenyl
vinyl
[CDCl3] 2.38 (s, 3H);





3.42 (d, 1H); 3.94





(d, 1H); 5.43 (d, 1H);





5.65 (d, 1H); 6.15





(dd, 1H); 6.98 (d, 1H);





7.18 (d, 1H); 7.22





(s, 1H).


1.3.487
3-methyl-5-fluorophenyl
1-methylvinyl
[CDCl3] 1.91 (s, 3H),





2.38 (s, 3H); 3.42





(d, 1H), 4.00 (d, 1H);





5.15 (s, 1H); 5.35





(s, 1H); 6.3 (s br, 1H),





6.98 (d, 1H); 7.17





(d, 1H); 7.21 (s, 1H).


1.3.488
3-methyl-5-fluorophenyl
allyl



1.3.489
3-methyl-5-fluorophenyl
1-chlorovinyl



1.3.490
3-methyl-5-fluorophenyl
ethynyl



1.3.491
3-ethyl-5-fluorophenyl
vinyl



1.3.492
3-propyl-5-fluorophenyl
vinyl



1.3.493
3-i-propyl-5-fluorophenyl
vinyl



1.3.494
3-n-butyl-5-fluorophenyl
vinyl



1.3.495
3-isobutyl-5-fluorophenyl
vinyl



1.3.496
3-tert-butyl-5-fluorophenyl
vinyl



1.3.497
3-cyclopropyl-5-fluorophenyl
vinyl



1.3.498
3-vinyl-5-fluorophenyl
vinyl



1.3.499
3-ethynyl-5-fluorophenyl
vinyl



1.3.500
3-cyano-5-fluorophenyl
vinyl



1.3.501
3-trifluoromethyl-5-fluorophenyl
vinyl



1.3.502
3-trifluoromethyl-5-fluorophenyl
1-methylvinyl



1.3.503
3-trifluoromethyl-5-fluorophenyl
allyl



1.3.504
3-trifluoromethyl-5-fluorophenyl
1-chlorovinyl



1.3.505
3-trifluoromethyl-5-fluorophenyl
ethynyl



1.3.506
3-(methoxycarbonyI)-5-fluorophenyl
vinyl



1.3.507
3-hydroxymethyl-5-fluorophenyl
vinyl



1.3.508
3-carbamoyl-5-fluorophenyl
vinyl



1.3.509
3-hydroxy-5-fluorophenyl
vinyl



1.3.510
3-methoxy-5-fluorophenyl
vinyl



1.3.511
3-ethoxy-5-fluorophenyl
vinyl



1.3.512
3-n-propoxy-5-fluorophenyl
vinyl



1.3.513
3-isopropoxy-5-fluorophenyl
vinyl



1.3.514
3-n-butoxy-5-fluorophenyl
vinyl



1.3.515
3-isobutoxy-5-fluorophenyl
vinyl



1.3.516
3-tert-butoxy-5-fluorophenyl
vinyl



1.3.517
3-difluoromethoxy-5-fluorophenyl
vinyl



1.3.518
3-trifluoromethoxy-5-fluorophenyl
vinyl



1.3.519
3-(2,2,2-trifluoroethoxy)-5-fluorophenyl
vinyl



1.3.520
3-(2-chloroethoxy)-5-fluorophenyl
vinyl



1.3.521
3-(2-hydroxyethoxy)-5-fluorophenyl
vinyl



1.3.522
3-[(tert-butoxycarbonyl)oxy]-5-
vinyl




fluorophenyl




1.3.523
3-nitro-5-fluorophenyl
vinyl



1.3.524
3-acetoxy-5-fluorophenyl
vinyl



1.3.525
{3-[(tert-butoxycarbonyl)amino]-5-
vinyl




fluorophenyl}




1.3.526
3-methylsulfanyl-5-fluorophenyl
vinyl



1.3.527
3,5-dichlorophenyl
vinyl
[CDCl3] 3.41 (d, 1H);





3.93 (d, 1H); 5.45





(d, 1H); 5.62 (d, 1H);





6.15 (dd, 1H); 7.44





(s, 1H); 7.54 (s, 2H).


1.3.528
3,5-dichlorophenyl
1-methylvinyl
[CDCl3] 1.91 (s, 3H);





3.40 (d, 1H); 3.99





(d, 1H); 5.16 (s, 1H),





5.35 (s, 1H); 5.9 (s





br, 1H), 7.42 (s, 1H);





7.54 (s, 2H).


1.3.529
3,5-dichlorophenyl
allyl



1.3.530
3,5-dichlorophenyl
1-chlorovinyl



1.3.531
3,5-dichlorophenyl
ethynyl



1.3.532
3-bromo-5-chlorophenyl
vinyl



1.3.533
3-iodo-5-chlorophenyl
vinyl



1.3.534
3-methyl-5-chlorophenyl
vinyl



1.3.535
3-methyl-5-chlorophenyl
1-methylvinyl
[CDCl3] 1.91 (s, 3H);





2.36 (s, 3H); 3.42





(d, 1H); 4.00 (d, 1H);





5.15 (s, 1H); 5.35





(s, 1H); 6.6 (s br, 1H);





7.24 (s, 1H); 7.36





(s, 1H); 7.45 (s, 1H).


1.3.536
3-ethyl-5-chlorophenyl
vinyl
[CDC13] 1.25 (t, 3H);





2.65 (q, 2H); 3.43





(d, 1H); 3.95 (d, 1H);





5.43 (d, 1H); 5.63





(d, 1H); 6.16 (dd, 1H);





7.27 (s, 1H); 7.38





(s, 1H); 7.43 (s, 1H).


1.3.537
3-propyl-5-chlorophenyl
vinyl



1.3.538
3-n-butyl-5-chlorophenyl
vinyl



1.3.539
3-isobutyl-5-chlorophenyl
vinyl



1.3.540
3-tert-butyl-5-chlorophenyl
vinyl



1.3.541
3-cyclopropyl-5-chlorophenyl
vinyl



1.3.542
3-vinyl-5-chlorophenyl
vinyl



1.3.543
3-ethynyl-5-chlorophenyl
vinyl



1.3.544
3-cyano-5-chlorophenyl
vinyl



1.3.545
3-trifluoromethyl-5-chlorophenyl
vinyl



1.3.546
3-(hydroxycarbonyl)-5-chlorophenyl
vinyl



1.3.547
3-(methoxycarbonyl)-5-chlorophenyl
vinyl



1.3.548
3-hydroxymethyl-5-chlorophenyl
vinyl



1.3.549
3-carbamoyl-5-chlorophenyl
vinyl



1.3.550
3-hydroxy-5-chlorophenyl
vinyl



1.3.551
3-methoxy-5-chlorophenyl
vinyl



1.3.552
3-ethoxy-5-chlorophenyl
vinyl



1.3.553
3-n-propoxy-5-chlorophenyl
vinyl



1.3.554
3-isopropoxy-5-chlorophenyl
vinyl



1.3.555
3-n-butoxy-5-chlorophenyl
vinyl



1.3.556
3-isobutoxy-5-chlorophenyl
vinyl



1.3.557
3-tert-butoxy-5-chlorophenyl
vinyl



1.3.558
3-difluoromethoxy-5-chlorophenyl
vinyl



1.3.559
3-trifluoromethoxy-5-chlorophenyl
vinyl



1.3.560
3-(2,2,2-trifluoroethoxy)-5-chlorophenyl
vinyl



1.3.561
3-(2-chloroethoxy)-5-chlorophenyl
vinyl



1.3.562
3-(2-hydroxyethoxy)-5-chlorophenyl
vinyl



1.3.563
3-[(tert-butoxycarbonyl)oxy]-5-
vinyl




chlorophenyl




1.3.564
3-nitro-5-chlorophenyl
vinyl



1.3.565
3-acetoxy-5-chlorophenyl
vinyl



1.3.566
(3-[(tert-butoxycarbonyl)amino]-5-
vinyl




chlorophenyl}




1.3.567
3-methylsulfanyl-5-chlorophenyl
vinyl



1.3.568
3,5-dibromophenyl
vinyl



1.3.569
3,5-dibromophenyl
1-methylvinyl



1.3.570
3-iodo-5-bromophenyl
vinyl



1.3.571
3-methyl-5-bromophenyl
vinyl
[CDCl3] 2.36 (s, 3H);





3.42 (d, 1H); 3.94





(d, 1H); 5.43 (d, 1H);





5.63 (d, 1H); 6.15





(dd, 1H); 7.40 (d, 2H);





7.58 (s, 1H).


1.3.572
3-methyl-5-bromophenyl
1-methylvinyl



1.3.573
3-methyl-5-bromophenyl
allyl



1.3.574
3-methyl-5-bromophenyl
1-chlorovinyl



1.3.575
3-methyl-5-bromophenyl
ethynyl



1.3.576
3-ethyl-5-bromophenyl
vinyl



1.3.577
3-propyl-5-bromophenyl
vinyl



1.3.578
3-isopropyl-5-bromophenyl
vinyl



1.3.579
3-n-butyl-5-bromophenyl
vinyl



1.3.580
3-isobutyl-5-bromophenyl
vinyl



1.3.581
3-tert-butyl-5-bromophenyl
vinyl



1.3.582
3-cyclopropyl-5-bromophenyl
vinyl



1.3.583
3-vinyl-5-bromophenyl
vinyl



1.3.584
3-ethynyl-5-bromophenyl
vinyl



1.3.585
3-cyano-5-bromophenyl
vinyl



1.3.586
3-trifluoromethyl-5-bromophenyl
vinyl



1.3.587
3-(hydroxycarbonyI)-5-bromophenyl
vinyl



1.3.588
3-(methoxycarbonyI)-5-bromophenyl
vinyl



1.3.589
3-hydroxymethyl-5-bromophenyl
vinyl



1.3.590
3-carbamoyl-5-bromophenyl
vinyl



1.3.591
3-hydroxy-5-bromophenyl
vinyl



1.3.592
3-methoxy-5-bromophenyl
vinyl



1.3.593
3-ethoxy-5-bromophenyl
vinyl



1.3.594
3-n-propoxy-5-bromophenyl
vinyl



1.3.595
3-isopropoxy-5-bromophenyl
vinyl



1.3.596
3-n-butoxy-5-bromophenyl
vinyl



1.3.597
3-isobutoxy-5-bromophenyl
vinyl



1.3.598
3-tert-butoxy-5-bromophenyl
vinyl



1.3.599
3-difluoromethoxy-5-bromophenyl
vinyl



1.3.600
3-trifluoromethoxy-5-bromophenyl
vinyl



1.3.601
3-(2,2,2-trifluoroethoxy)-5-bromophenyl
vinyl



1.3.602
3-(2-chloroethoxy)-5-bromophenyl
vinyl



1.3.603
3-(2-hydroxyethoxy)-5-bromophenyl
vinyl



1.3.604
3-[(tert-butoxycarbonyl)oxy]-5-
vinyl




bromophenyl




1.3.605
3-nitro-5-bromophenyl
vinyl



1.3.606
3-acetoxy-5-bromophenyl
vinyl



1.3.607
(3-[(tert-butoxycarbonyl)amino]-5-
vinyl




bromophenyl}




1.3.608
3-methylsulfanyl-5-bromophenyl
vinyl



1.3.609
3,5-diiodophenyl
vinyl



1.3.610
3-methyl-5-iodophenyl
vinyl



1.3.611
3-ethyl-5-iodophenyl
vinyl



1.3.612
3-propyl-5-iodophenyl
vinyl



1.3.613
3-isopropyl-5-iodophenyl
vinyl



1.3.614
3-n-butyl-5-iodophenyl
vinyl



1.3.615
3-isobutyl-5-iodophenyl
vinyl



1.3.616
3-tert-butyl-5-iodophenyl
vinyl



1.3.617
3-cyclopropyl-5-iodophenyl
vinyl



1.3.618
3-vinyl-5-iodophenyl
vinyl



1.3.619
3-ethynyl-5-iodophenyl
vinyl



1.3.620
3-cyano-5-iodophenyl
vinyl



1.3.621
3-trifluoromethyl-5-iodophenyl
vinyl



1.3.622
3-(hydroxycarbony1)-5-iodophenyl
vinyl



1.3.623
3-(methoxycarbony1)-5-iodophenyl
vinyl



1.3.624
3-hydroxymethyl-5-iodophenyl
vinyl



1.3.625
3-carbamoyl-5-iodophenyl
vinyl



1.3.626
3-hydroxy-5-iodophenyl
vinyl



1.3.627
3-methoxy-5-iodophenyl
vinyl



1.3.628
3-ethoxy-5-iodophenyl
vinyl



1.3.629
3-n-propoxy-5-iodophenyl
vinyl



1.3.630
3-isopropoxy-5-iodophenyl
vinyl



1.3.631
3-n-butoxy-5-iodophenyl
vinyl



1.3.632
3-isobutoxy-5-iodophenyl
vinyl



1.3.633
3-tert-butoxy-5-iodophenyl
vinyl



1.3.634
3-difluoromethoxy-5-iodophenyl
vinyl



1.3.635
3-trifluoromethoxy-5-iodophenyl
vinyl



1.3.636
3-(2,2,2-trifluoroethoxy)-5-iodophenyl
vinyl



1.3.637
3-(2-chloroethoxy)-5-iodophenyl
vinyl



1.3.638
3-(2-hydroxyethoxy)-5-iodophenyl
vinyl



1.3.639 
3-[(tert-butoxycarbonyl)oxy]-5-iodophenyl
vinyl



1.3.640
3-nitro-5-iodophenyl
vinyl



1.3.641
3-acetoxy-5-iodophenyl
vinyl



1.3.642
(3-[(tert-butoxycarbonyl)amino]-5-
vinyl




iodophenyl}




1.3.643
3-methylsulfanyl-5-iodophenyl
vinyl



1.3.644
3,5-dimethylphenyl
vinyl
[CDCl3] 2.34 (s, 6H);





3.45 (d, 1H); 3.97





(d, 1H); 5.42 (d, 1H);





5.62 (d, 1H); 6.15





(dd, 1H); 7.09 (s, 1H);





7.26 (s, 2H).


1.3.645
3-ethyl-5-methylphenyl
vinyl



1.3.646
3-propyl-5-methylphenyl
vinyl



1.3.647
3-isopropyl-5-methylphenyl
vinyl



1.3.648
3-n-butyl-5-methylphenyl
vinyl



1.3.649
3-isobutyl-5-methylphenyl
vinyl



1.3.650
3-tert-butyl-5-methylphenyl
vinyl



1.3.651
3-cyclopropyl-5-methylphenyl
vinyl



1.3.652
3-cyano-5-methylphenyl
vinyl



1.3.653
3-trifluoromethyl-5-methylphenyl
vinyl



1.3.654
3-(methoxycarbonyl)-5-methylphenyl
vinyl



1.3.655
3-methoxy-5-methylphenyl
vinyl



1.3.656
3-ethoxy-5-methylphenyl
vinyl



1.3.657
3-n-propoxy-5-methylphenyl
vinyl



1.3.658
3-n-butoxy-5-methylphenyl
vinyl



1.3.659
3-isobutoxy-5-methylphenyl
vinyl



1.3.660
3-difluoromethoxy-5-methylphenyl
vinyl



1.3.661
3-trifluoromethoxy-5-methylphenyl
vinyl



1.3.662
3-nitro-5-methylphenyl
vinyl



1.3.663
3-acetoxy-5-methylphenyl
vinyl



1.3.664
3-methylsulfanyl-5-methylphenyl
vinyl



1.3.665
3,5-diethylphenyl
vinyl



1.3.666
3-propyl-5-ethylphenyl
vinyl



1.3.667
3-isopropyl-5-ethylphenyl
vinyl



1.3.668
3-n-butyl-5-ethylphenyl
vinyl



1.3.669
3-isobutyl-5-ethylphenyl
vinyl



1.3.670
3-tert-butyl-5-ethylphenyl
vinyl



1.3.671
3-cyclopropyl-5-ethylphenyl
vinyl



1.3.672
3-cyano-5-ethylphenyl
vinyl



1.3.673
3-trifluoromethyl-5-ethylphenyl
vinyl



1.3.674
3-(methoxycarbonyI)-5-ethylphenyl
vinyl



1.3.675
3-methoxy-5-ethylphenyl
vinyl



1.3.676
3-ethoxy-5-ethylphenyl
vinyl



1.3.677
3-n-propoxy-5-ethylphenyl
vinyl



1.3.678
3-n-butoxy-5-ethylphenyl
vinyl



1.3.679
3-isobutoxy-5-ethylphenyl
vinyl



1.3.680
3-difluoromethoxy-5-ethylphenyl
vinyl



1.3.681
3-trifluoromethoxy-5-ethylphenyl
vinyl



1.3.682
3-nitro-5-ethylphenyl
vinyl



1.3.683
3-acetoxy-5-ethylphenyl
vinyl



1.3.684
3-methylsulfanyl-5-ethylphenyl
vinyl



1.3.685
3,5-dipropylphenyl
vinyl



1.3.686
3-isopropyl-5-propylphenyl
vinyl



1.3.687
3-n-butyl-5-propylphenyl
vinyl



1.3.688
3-isobutyl-5-propylphenyl
vinyl



1.3.689
3-tert-butyl-5-propylphenyl
vinyl



1.3.690
3-cyclopropyl-5-propylphenyl
vinyl



1.3.691
3-cyano-5-propylphenyl
vinyl



1.3.692
3-trifluoromethyl-5-propylphenyl
vinyl



1.3.693
3-(methoxycarbonyl)-5-propylphenyl
vinyl



1.3.694
3-methoxy-5-propylphenyl
vinyl



1.3.695
3-ethoxy-5-propylphenyl
vinyl



1.3.696
3-n-propoxy-5-propylphenyl
vinyl



1.3.697
3-n-butoxy-5-propylphenyl
vinyl



1.3.698
3-isobutoxy-5-propylphenyl
vinyl



1.3.699
3-tert-butoxy-5-propylphenyl
vinyl



1.3.700
3-difluoromethoxy-5-propylphenyl
vinyl



1.3.701
3-trifluoromethoxy-5-ethylphenyl
vinyl



1.3.702
3-nitro-5-propylphenyl
vinyl



1.3.703
3-acetoxy-5-propylphenyl
vinyl



1.3.704
3-methylsulfanyl-5-propylphenyl
vinyl



1.3.705
3,5-diisopropylphenyl
vinyl



1.3.706
3-n-butyl-5-isopropylphenyl
vinyl



1.3.707
3-isobutyl-5-isopropylphenyl
vinyl



1.3.708
3-tert-butyl-5-isopropylphenyl
vinyl



1.3.709
3-cyclopropyl-5-isopropylphenyl
vinyl



1.3.710
3-cyano-5-isopropylphenyl
vinyl



1.3.711
3-trifluoromethyl-5-isopropylphenyl
vinyl



1.3.712
3-(methoxycarbonyI)-5-isopropylphenyl
vinyl



1.3.713
3-methoxy-5-isopropylphenyl
vinyl



1.3.714
3-ethoxy-5-isopropylphenyl
vinyl



1.3.715
3-n-propoxy-5-isopropylphenyl
vinyl



1.3.716
3-n-butoxy-5-isopropylphenyl
vinyl



1.3.717
3-isobutoxy-5-isopropylphenyl
vinyl



1.3.718
3-difluoromethoxy-5-isopropylphenyl
vinyl



1.3.719
3-trifluoromethoxy-5-isopropylphenyl
vinyl



1.3.720
3-nitro-5-isopropylphenyl
vinyl



1.3.721
3-acetoxy-5-isopropylphenyl
vinyl



1.3.722
3-methylsulfanyl-5-isopropylphenyl
vinyl



1.3.723
3,5-dibutylphenyl
vinyl



1.3.724
3-isobutyl-5-butylphenyl
vinyl



1.3.725
3-tert-butyl-5-butylphenyl
vinyl



1.3.726
3-cyclopropyl-5-butylphenyl
vinyl



1.3.727
3-cyano-5-butylphenyl
vinyl



1.3.728
3-trifluoromethyl-5-butylphenyl
vinyl



1.3.729
3-(methoxycarbonyl)-5-butylphenyl
vinyl



1.3.730
3-methoxy-5-butylphenyl
vinyl



1.3.731
3-ethoxy-5-butylphenyl
vinyl



1.3.732
3-n-propoxy-5-butylphenyl
vinyl



1.3.733
3-n-butoxy-5-butylphenyl
vinyl



1.3.734
3-isobutoxy-5-butylphenyl
vinyl



1.3.735
3-difluoromethoxy-5-butylphenyl
vinyl



1.3.736
3-trifluoromethoxy-5-butylphenyl
vinyl



1.3.737
3-nitro-5-butylphenyl
vinyl



1.3.738
3-acetoxy-5-butylphenyl
vinyl



1.3.739
3-methylsulfanyl-5-butylphenyl
vinyl



1.3.740
3,5-diisobutylphenyl
vinyl



1.3.741
3-tert-butyl-5-isobutylphenyl
vinyl



1.3.742
3-cyclopropyl-5-isobutylphenyl
vinyl



1.3.743
3-cyano-5-isobutylphenyl
vinyl



1.3.744
3-trifluoromethyl-5-isobutylphenyl
vinyl



1.3.745
3-(hydroxycarbonyl)-5-isobutylphenyl
vinyl



1.3.746
3-(methoxycarbonyl)-5-isobutylphenyl
vinyl



1.3.747
3-methoxy-5-isobutylphenyl
vinyl



1.3.748
3-ethoxy-5-isobutylphenyl
vinyl



1.3.749
3-n-propoxy-5-isobutylphenyl
vinyl



1.3.750
3-n-butoxy-5-isobutylphenyl
vinyl



1.3.751
3-isobutoxy-5-isobutylphenyl
vinyl



1.3.752
3-difluoromethoxy-5-isobutylphenyl
vinyl



1.3.753
3-trifluoromethoxy-5-isobutylphenyl
vinyl



1.3.754
3-nitro-5-isobutylphenyl
vinyl



1.3.755
3-acetoxy-5-isobutylphenyl
vinyl



1.3.756
3-methylsulfanyl-5-isobutylphenyl
vinyl



1.3.757
3,5-di(tert-butyl)phenyl
vinyl



1.3.758
3-cyclopropyl-5-tert-butylphenyl
vinyl



1.3.759
3-cyano-5-tert-butylphenyl
vinyl



1.3.760
3-trifluoromethyl-5-tert-butylphenyl
vinyl



1.3.761
3-(methoxycarbonyl)-5-tert-butylphenyl
vinyl



1.3.762
3-methoxy-5-tert-butylphenyl
vinyl



1.3.763
3-ethoxy-5-tert-butylphenyl
vinyl



1.3.764
3-n-propoxy-5-tert-butylphenyl
vinyl



1.3.765
3-n-butoxy-5-tert-butylphenyl
vinyl



1.3.766
3-isobutoxy-5-tert-butylphenyl
vinyl



1.3.767
3-tert-butoxy-5-tert-butylphenyl
vinyl



1.3.768
3-difluoromethoxy-5-tert-butylphenyl
vinyl



1.3.769
3-trifluoromethoxy-5-tert-butylphenyl
vinyl



1.3.770
3-nitro-5-tert-butylphenyl
vinyl



1.3.771
3-acetoxy-5-tert-butylphenyl
vinyl



1.3.772
3-methylsulfanyl-5-tert-butylphenyl
vinyl



1.3.773
3-tert-butyl-5-cyclopropylphenyl
vinyl



1.3.774
3,5-dicyclopropyl-phenyl
vinyl



1.3.775
3-cyano-5-cyclopropylphenyl
vinyl



1.3.776
3-trifluoromethyl-5-cyclopropylphenyl
vinyl



1.3.777 
3-(methoxycarbonyI)-5-cyclopropylphenyl
vinyl



1.3.778
3-methoxy-5-cyclopropylphenyl
vinyl



1.3.779
3-ethoxy-5-cyclopropylphenyl
vinyl



1.3.780
3-n-propoxy-5-cyclopropylphenyl
vinyl



1.3.781
3-n-butoxy-5-cyclopropylphenyl
vinyl



1.3.782
3-isobutoxy-5-cyclopropylphenyl
vinyl



1.3.783
3-difluoromethoxy-5-cyclopropylphenyl
vinyl



1.3.784
3-trifluoromethoxy-5-cyclopropylphenyl
vinyl



1.3.785
3-nitro-5-cyclopropylphenyl
vinyl



1.3.786
3-acetoxy-5-cyclopropylphenyl
vinyl



1.3.787
3-methylsulfanyl-5-cyclopropylphenyl
vinyl



1.3.788
3,5-dicyanophenyl
vinyl



1.3.789
3-trifluoromethyl-5-cyanophenyl
vinyl



1.3.790
3-(methoxycarbonyI)-5-cyanophenyl
vinyl



1.3.791
3-methoxy-5-cyanophenyl
vinyl



1.3.792
3-ethoxy-5-cyanophenyl
vinyl



1.3.793
3-n-propoxy-5-cyanophenyl
vinyl



1.3.794
3-n-butoxy-5-cyanophenyl
vinyl



1.3.795
3-isobutoxy-5-cyanophenyl
vinyl



1.3.796
3-difluoromethoxy-5-cyanophenyl
vinyl



1.3.797
3-trifluoromethoxy-5-cyanophenyl
vinyl



1.3.798
3-nitro-5-cyanophenyl
vinyl



1.3.799
3-acetoxy-5-cyanophenyl
vinyl



1.3.800
3-methylsulfanyl-5-cyanophenyl
vinyl



1.3.801
3,5-di(trifluoromethyl)-phenyl
vinyl



1.3.802
3-(methoxycarbonyl)-5-trifluoromethyl-
vinyl




phenyl




1.3.803
3-methoxy-5-trifluoromethylphenyl
vinyl



1.3.804
3-ethoxy-5-trifluoromethylphenyl
vinyl



1.3.805
3-n-propoxy-5-trifluoromethylphenyl
vinyl



1.3.806
3-n-butoxy-5-trifluoromethylphenyl
vinyl



1.3.807
3-isobutoxy-5-trifluoromethylphenyl
vinyl



1.3.808
3-difluoromethoxy-5-trifluoromethylphenyl
vinyl



1.3.809
3-trifluoromethoxy-5-trifluoromethylphenyl
vinyl



1.3.810
3-nitro-5-trifluoromethylphenyl
vinyl



1.3.811
3-acetoxy-5-trifluoromethylphenyl
vinyl



1.3.812
3-methylsulfanyl-5-trifluoromethylphenyl
vinyl



1.3.813
3,5-di(methoxycarbonyl)phenyl
vinyl



1.3.814
3-methoxy-5-(methoxycarbonyl)phenyl
vinyl



1.3.815
3-ethoxy-5-(methoxycarbonyl)phenyl
vinyl



1.3.816
3-n-propoxy-5-(methoxycarbonyl)phenyl
vinyl



1.3.817
3-n-butoxy-5-(methoxycarbonyl)phenyl
vinyl



1.3.818
3-isobutoxy-5-(methoxycarbonyl)phenyl
vinyl



1.3.819
3-difluoromethoxy-5-(methoxycarbonyl)-
vinyl




phenyl




1.3.820
3-trifluoromethoxy-5-(methoxycarbonyl)-
vinyl




phenyl




1.3.821
3-nitro-5-(methoxycarbonyl)phenyl
vinyl



1.3.822
3-acetoxy-5-(methoxycarbonyl)phenyl
vinyl



1.3.823
3-methylsulfanyl-5-(methoxycarbonyl)-
vinyl




phenyl




1.3.824
3,5-dimethoxyphenyl
vinyl



1.3.825
3-ethoxy-5-methoxyphenyl
vinyl



1.3.826
3-n-propoxy-5-methoxyphenyl
vinyl



1.3.827
3-n-butoxy-5-methoxyphenyl
vinyl



1.3.828
3-isobutoxy-5-methoxyphenyl
vinyl



1.3.829
3-difluoromethoxy-5-methoxyphenyl
vinyl



1.3.830
3-trifluoromethoxy-5-methoxyphenyl
vinyl



1.3.831
3-nitro-5-methoxyphenyl
vinyl



1.3.832
3-acetoxy-5-methoxyphenyl
vinyl



1.3.833
3-methylsulfanyl-5-methoxyphenyl
vinyl



1.3.834
3,5-diethoxyphenyl
vinyl



1.3.835
3-n-propoxy-5-ethoxyphenyl
vinyl



1.3.836
3-n-butoxy-5-ethoxyphenyl
vinyl



1.3.837
3-isobutoxy-5-ethoxyphenyl
vinyl



1.3.838
3-difluoromethoxy-5-ethoxyphenyl
vinyl



1.3.839
3-trifluoromethoxy-5-ethoxyphenyl
vinyl



1.3.840
3-nitro-5-ethoxyphenyl
vinyl



1.3.841
3-acetoxy-5-ethoxyphenyl
vinyl



1.3.842
3-methylsulfanyl-5-ethoxyphenyl
vinyl



1.3.843
3,5-di(isopropoxy)phenyl
vinyl



1.3.844
3-n-butoxy-5-isopropoxyphenyl
vinyl



1.3.845
3-isobutoxy-5-isopropoxyphenyl
vinyl



1.3.846
3-difluoromethoxy-5-isopropoxyphenyl
vinyl



1.3.847
3-trifluoromethoxy-5-isopropoxyphenyl
vinyl



1.3.848
3-nitro-5-isopropoxyphenyl
vinyl



1.3.849
3-acetoxy-5-isopropoxyphenyl
vinyl



1.3.850
3-methylsulfanyl-5-isopropoxyphenyl
vinyl



1.3.851
3,5-di(trifluoromethoxy)phenyl
vinyl



1.3.852
3-nitro-5-trifluoromethoxyphenyl
vinyl



1.3.853
3-acetoxy-5-tert-butoxyphenyl
vinyl



1.3.854
3-methylsulfanyl-5-trifluoromethoxy-
vinyl




phenyl




1.3.855
3,5-bis(difluoromethoxy)phenyl
vinyl



1.3.856
3,5-bis(difluoromethoxy)phenyl
1-methylvinyl



1.3.857
3,5-bis(difluoromethoxy)phenyl
allyl



1.3.858
3,5-bis(difluoromethoxy)phenyl
1-chlorovinyl



1.3.859
3-trifluoromethoxy-5-difluoromethoxy-
vinyl




phenyl




1.3.860
3-nitro-5-difluoromethoxyphenyl
vinyl



1.3.861
3-acetoxy-5-difluoromethoxyphenyl
vinyl



1.3.862
3-methylsulfanyl-5-difluoromethoxy-
vinyl




phenyl




1.3.863
3,5-bis(acetoxy)phenyl
vinyl



1.3.864
3-methylsulfanyl-5-acetoxyphenyl
vinyl



1.3.865
3-acetoxy-5-nitrophenyl
vinyl



1.3.866
3-methylsulfanyl-5-nitrophenyl
vinyl



1.3.867
3,5-di(methylsulfanyl)phenyl
vinyl



1.3.868
3,4-difluorophenyl
vinyl



1.3.869
3,4-difluorophenyl
1-methylvinyl



1.3.870
3,4-difluorophenyl
allyl



1.3.871
3,4-difluorophenyl
1-chlorovinyl



1.3.872
3,4-difluorophenyl
ethynyl



1.3.873
3-chloro-4-fluorophenyl
vinyl



1.3.874
3-chloro-4-fluorophenyl
1-methylvinyl



1.3.875
3-chloro-4-fluorophenyl
allyl



1.3.876
3-chloro-4-fluorophenyl
1-chlorovinyl



1.3.877
3-chloro-4-fluorophenyl
ethynyl



1.3.878
3-bromo-4-fluorophenyl
vinyl



1.3.879
3-methyl-4-fluorophenyl
vinyl



1.3.880
3-methyl-4-fluorophenyl
1-methylvinyl



1.3.881
3-cyclopropyl-4-fluorophenyl
vinyl



1.3.882
3-cyano-4-fluorophenyl
vinyl



1.3.883
3-methoxy-4-fluorophenyl
vinyl



1.3.884
3-ethoxy-4-fluorophenyl
vinyl



1.3.885
3-trifluoromethoxy-4-fluorophenyl
vinyl



1.3.886
3-nitro-4-fluorophenyl
vinyl



1.3.887
3-fluoro-4-chlorophenyl
vinyl



1.3.888
3,4-dichlorophenyl
vinyl



1.3.889
3-bromo-4-chlorophenyl
vinyl



1.3.890
3-methyl-4-chlorophenyl
vinyl



1.3.891
3-ethyl-4-chlorophenyl
vinyl



1.3.892
3-cyclopropyl-4-chlorophenyl
vinyl



1.3.893
3-cyano-4-chlorophenyl
vinyl



1.3.894
3-trifluoromethyl-4-chlorophenyl
vinyl



1.3.895
3-methoxy-4-chlorophenyl
vinyl



1.3.896
3-ethoxy-4-chlorophenyl
vinyl



1.3.897
3-trifluoromethoxy-4-chlorophenyl
vinyl



1.3.898
3-nitro-4-chlorophenyl
vinyl



1.3.899
3-fluoro-4-bromophenyl
vinyl



1.3.900
3-chloro-4-bromophenyl
vinyl



1.3.901
3,4-dibromophenyl
vinyl



1.3.902
3-methyl-4-bromophenyl
vinyl



1.3.903
3-ethyl-4-bromophenyl
vinyl



1.3.904
3-cyclopropyl-4-bromophenyl
vinyl



1.3.905
3-cyano-4-bromophenyl
vinyl



1.3.906
3-trifluoromethyl-4-bromophenyl
vinyl



1.3.907
3-methoxy-4-phenyl
vinyl



1.3.908
3-ethoxy-4-bromophenyl
vinyl



1.3.909
3-trifluoromethoxy-4-bromophenyl
vinyl



1.3.910
3-nitro-4-bromophenyl
vinyl



1.3.911
3-fluoro-4-iodophenyl
vinyl



1.3.912
3-chloro-4-iodophenyl
vinyl



1.3.913
3-bromo-4-iodophenyl
vinyl



1.3.914
3-methyl-4-iodophenyl
vinyl



1.3.915
3-cyclopropyl-4-iodophenyl
vinyl



1.3.916
3-cyano-4-iodophenyl
vinyl



1.3.917
3-trifluoromethyl-4-iodophenyl
vinyl



1.3.918
3-methoxy-4-iodophenyl
vinyl



1.3.919
3-ethoxy-4-iodophenyl
vinyl



1.3.920
3-trifluoromethoxy-4-iodophenyl
vinyl



1.3.921
3-nitro-4-iodophenyl
vinyl



1.3.922
3-fluoro-4-methylphenyl
vinyl



1.3.923
3-chloro-4-methylphenyl
vinyl



1.3.924
3-bromo-4-methylphenyl
vinyl



1.3.925
3,4-dimethylphenyl
vinyl



1.3.926
3,4-dimethylphenyl
1-methylvinyl



1.3.927
3,4-dimethylphenyl
allyl



1.3.928
3,4-dimethylphenyl
1-chlorovinyl



1.3.929
3,4-dimethylphenyl
ethynyl



1.3.930
3-ethyl-4-methylphenyl
vinyl



1.3.931
3-cyclopropyl-4-methylphenyl
vinyl



1.3.932
3-cyano-4-methylphenyl
vinyl



1.3.933
3-trifluoromethyl-4-methylphenyl
vinyl



1.3.934
3-methoxy-4-methylphenyl
vinyl



1.3.935
3-ethoxy-4-methylphenyl
vinyl



1.3.936
3-trifluoromethoxy-4-methylphenyl
vinyl



1.3.937
3-nitro-4-methylphenyl
vinyl



1.3.938
3-fluoro-4-ethylphenyl
vinyl



1.3.939
3-chloro-4-ethylphenyl
vinyl



1.3.940
3-bromo-4-ethylphenyl
vinyl



1.3.941
3-methyl-4-ethylphenyl
vinyl



1.3.942
3,4-diethylphenyl
vinyl



1.3.943
3-cyclopropyl-4-ethylphenyl
vinyl



1.3.944
3-cyano-4-ethylphenyl
vinyl



1.3.945
3-trifluoromethyl-4-ethylphenyl
vinyl



1.3.946
3-methoxy-4-ethylphenyl
vinyl



1.3.947
3-ethoxy-4-ethylphenyl
vinyl



1.3.948
3-trifluoromethoxy-4-ethylphenyl
vinyl



1.3.949
3-nitro-4-ethylphenyl
vinyl



1.3.950
3-fluoro-4-propylphenyl
vinyl



1.3.951
3-chloro-4-propylphenyl
vinyl



1.3.952
3-bromo-4-propylphenyl
vinyl



1.3.953
3-methyl-4-propylphenyl
vinyl



1.3.954
3-methyl-4-propylphenyl
vinyl



1.3.955
3-cyclopropyl-4-propylphenyl
vinyl



1.3.956
3-cyano-4-propylphenyl
vinyl



1.3.957
3-trifluoromethyl-4-propylphenyl
vinyl



1.3.958
3-methoxy-4-propylphenyl
vinyl



1.3.959
3-ethoxy-4-propylphenyl
vinyl



1.3.960
3-trifluoromethoxy-4-propylphenyl
vinyl



1.3.961
3-nitro-4-propylphenyl
vinyl



1.3.962
3-fluoro-4-isopropylphenyl
vinyl



1.3.963
3-chloro-4-isopropylphenyl
vinyl



1.3.964
3-bromo-4- isopropylphenyl
vinyl



1.3.965
3-methyl-4-isopropylphenyl
vinyl



1.3.966
3-cyclopropyl-4-isopropylphenyl
vinyl



1.3.967
3-cyano-4-isopropylphenyl
vinyl



1.3.968
3-trifluoromethyl-4-isopropylphenyl
vinyl



1.3.969
3-methoxy-4-isopropylphenyl
vinyl



1.3.970
3-ethoxy-4-isopropylphenyl
vinyl



1.3.971
3-trifluoromethoxy-4-isopropylphenyl
vinyl



1.3.972
3-nitro-4-isopropylphenyl
vinyl



1.3.973
3-fluoro-4-tert-butylphenyl
vinyl



1.3.974
3-chloro-4-tert-butylphenyl
vinyl



1.3.975
3-bromo-4-tert-butylphenyl
vinyl



1.3.976
3-methyl-4-tert-butylphenyl
vinyl



1.3.977
3-cyclopropyl-4-tert-butylphenyl
vinyl



1.3.978
3-cyano-4-tert-butylphenyl
vinyl



1.3.979
3-trifluoromethyl-4-tert-butylphenyl
vinyl



1.3.980
3-trifluoromethyl-4-tert-butylphenyl
1-methylvinyl



1.3.981
3-trifluoromethyl-4-tert-butylphenyl
allyl



1.3.982
3-trifluoromethyl-4-tert-butylphenyl
1-chlorovinyl



1.3.983
3-trifluoromethyl-4-tert-butylphenyl
ethynyl



1.3.984
3-methoxy-4-tert-butylphenyl
vinyl



1.3.985
3-ethoxy-4-tert-butylphenyl
vinyl



1.3.986
3-trifluoromethoxy-4-tert-butylphenyl
vinyl



1.3.987
3-nitro-4-tert-butylphenyl
vinyl



1.3.988
3-fluoro-4-cyclopropylphenyl
vinyl



1.3.989
3-chloro-4-cyclopropylphenyl
vinyl



1.3.990
3-bromo-4-cyclopropylphenyl
vinyl



1.3.991
3-methyl-4-cyclopropylphenyl
vinyl



1.3.992
3-cyclopropyl-4-cyclopropylphenyl
vinyl



1.3.993
3-cyano-4-cyclopropylphenyl
vinyl



1.3.994
3-trifluoromethyl-4-cyclopropylphenyl
vinyl



1.3.995
3-methoxy-4-cyclopropylphenyl
vinyl



1.3.996
3-ethoxy-4-cyclopropylphenyl
vinyl



1.3.997
3-trifluoromethoxy-4-cyclopropylphenyl
vinyl



1.3.998
3-fluoro-4-methoxycarbonylphenyl
vinyl



1.3.999
3-chloro-4-methoxycarbonylphenyl
vinyl



1.3.1000
3-bromo-4-methoxycarbonylphenyl
vinyl



1.3.1001
3-methyl-4-methoxycarbonylphenyl
vinyl



1.3.1002
3-cyclopropyl-4-methoxycarbonylphenyl
vinyl



1.3.1003
3-cyano-4-methoxycarbonylphenyl
vinyl



1.3.1004
3-trifluoromethyl-4-methoxycarbonyl-
vinyl




phenyl




1.3.1005
3-methoxy-4-methoxycarbonylphenyl
vinyl



1.3.1006
3-ethoxy-4-methoxycarbonylphenyl
vinyl



1.3.1007
3-trifluoromethoxy-4-methoxycarbonyl-
vinyl




phenyl




1.3.1008
3-nitro-4-methoxycarbonylphenyl
vinyl



1.3.1009
3-fluoro-4-cyanophenyl
vinyl



1.3.1010
3-chloro-4-cyanophenyl
vinyl



1.3.1011
3-bromo-4-cyanophenyl
vinyl



1.3.1012
3-methyl-4-cyanophenyl
vinyl



1.3.1013
3-cyclopropyl-4-cyanophenyl
vinyl



1.3.1014
3,4-dicyanophenyl
vinyl



1.3.1015
3-trifluoromethyl-4-cyanophenyl
vinyl



1.3.1016
3-trifluoromethyl-4-cyanophenyl
1-methylvinyl



1.3.1017
3-trifluoromethyl-4-cyanophenyl
allyl



1.3.1018
3-trifluoromethyl-4-cyanophenyl
1-chlorovinyl



1.3.1019
3-trifluoromethyl-4-cyanophenyl
ethynyl



1.3.1020
3-methoxy-4-cyanophenyl
vinyl



1.3.1021
3-ethoxy-4-cyanophenyl
vinyl



1.3.1022
3-trifluoromethoxy-4-cyanophenyl
vinyl



1.3.1023
3-nitro-4-cyanophenyl
vinyl



1.3.1024
3-fluoro-4-methoxyphenyl
vinyl



1.3.1025
3-chloro-4-methoxyphenyl
vinyl



1.3.1026
3-bromo-4-methoxyphenyl
vinyl



1.3.1027
3-methyl-4-methoxyphenyl
vinyl



1.3.1028
3-cyclopropyl-4-methoxyphenyl
vinyl



1.3.1029
3-cyano-4-methoxyphenyl
vinyl



1.3.1030
3-trifluoromethyl-4-methoxyphenyl
vinyl



1.3.1031
3,4-dimethoxyphenyl
vinyl



1.3.1032
3-ethoxy-4-methoxyphenyl
vinyl



1.3.1033
3-trifluoromethoxy-4-methoxyphenyl
vinyl



1.3.1034
3-nitro-4-methoxyphenyl
vinyl



1.3.1035
3-fluoro-4-ethoxyphenyl
vinyl



1.3.1036
3-chloro-4-ethoxyphenyl
vinyl



1.3.1037
3-chloro-4-ethoxyphenyl
1-methylvinyl



1.3.1038
3-chloro-4-ethoxyphenyl
allyl



1.3.1039
3-chloro-4-ethoxyphenyl
1-chlorovinyl



1.3.1040
3-chloro-4-ethoxyphenyl
ethynyl



1.3.1041
3-bromo-4-ethoxyphenyl
vinyl



1.3.1042
3-methyl-4-ethoxyphenyl
vinyl



1.3.1043
3-cyclopropyl-4-ethoxyphenyl
vinyl



1.3.1044
3-cyano-4-ethoxyphenyl
vinyl



1.3.1045
3-trifluoromethyl-4-ethoxyphenyl
vinyl



1.3.1046
3-methoxy-4-ethoxyphenyl
vinyl



1.3.1047
2,4-diethoxyphenyl
vinyl



1.3.1048
3-trifluoromethoxy-4-ethoxyphenyl
vinyl



1.3.1049
3-nitro-4-ethoxyphenyl
vinyl



1.3.1050
3-fluoro-4-propoxyphenyl
vinyl



1.3.1051
3-chloro-4-propoxyphenyl
vinyl



1.3.1052
3-bromo-4-propoxyphenyl
vinyl



1.3.1053
3-methyl-4-propoxyphenyl
vinyl



1.3.1054
3-cyclopropyl-4-propoxyphenyl
vinyl



1.3.1055
3-cyano-4-propoxyphenyl
vinyl



1.3.1056
3-trifluoromethyl-4-propoxyphenyl
vinyl



1.3.1057
3-methoxy-4-propoxyphenyl
vinyl



1.3.1058
3-ethoxy-4-propoxyphenyl
vinyl



1.3.1059
3-trifluoromethoxy-4-propoxyphenyl
vinyl



1.3.1060
3-nitro-4-propoxyphenyl
vinyl



1.3.1061
3-fluoro-4-isopropoxyphenyl
vinyl



1.3.1062
3-chloro-4-isopropoxyphenyl
vinyl



1.3.1063
3-bromo-4-isopropoxyphenyl
vinyl



1.3.1064
3-methyl-4-isopropoxyphenyl
vinyl



1.3.1065
3-cyclopropyl-4-isopropoxyphenyl
vinyl



1.3.1066
3-cyano-4-isopropoxyphenyl
vinyl



1.3.1067
3-trifluoromethyl-4-isopropoxyphenyl
vinyl



1.3.1068
3-methoxy-4-isopropoxyphenyl
vinyl



1.3.1069
3-ethoxy-4-isopropoxyphenyl
vinyl



1.3.1070
3-trifluoromethoxy-4-isopropoxyphenyl
vinyl



1.3.1071
3-nitro-4- isopropoxyphenyl
vinyl



1.3.1072
3-fluoro-4-trifluoromethoxyphenyl
vinyl



1.3.1073
3-chloro-4-trifluoromethoxyphenyl
vinyl



1.3.1074
3-bromo-4-trifluoromethoxyphenyl
vinyl



1.3.1075
3-methyl-4-trifluoromethoxyphenyl
vinyl



1.3.1076 
3-cyclopropyl-4-trifluoromethoxyphenyl
vinyl



1.3.1077
3-cyano-4-trifluoromethoxyphenyl
vinyl



1.3.1078
3-trifluoromethyl-4-trifluoromethoxy-
vinyl




phenyl




1.3.1079
3-methoxy-4-trifluoromethoxyphenyl
vinyl



1.3.1080
3-ethoxy-4-trifluoromethoxyphenyl
vinyl



1.3.1081
3,4-bis(trifluoromethoxy)phenyl
vinyl



1.3.1082
3-nitro-4-trifluoromethoxyphenyl
vinyl



1.3.1083
3-fluoro-4-difluoromethoxyphenyl
vinyl



1.3.1084
3-chloro-4-difluoromethoxyphenyl
vinyl



1.3.1085
3-bromo-4-difluoromethoxyphenyl
vinyl



1.3.1086
3-methyl-4-difluoromethoxyphenyl
vinyl



1.3.1087
3-cyclopropyl-4-difluoromethoxyphenyl
vinyl



1.3.1088
3-cyano-4-difluoromethoxyphenyl
vinyl



1.3.1089
3-trifluoromethyl-4-difluoromethoxyphenyl
vinyl



1.3.1090
3-methoxy-4-difluoromethoxyphenyl
vinyl



1.3.1091
3-ethoxy-4-difluoromethoxyphenyl
vinyl



1.3.1092
3-trifluoromethoxy-4-difluoromethoxy-
vinyl




phenyl




1.3.1093
3-nitro-4-difluoromethoxyphenyl
vinyl



1.3.1094
3-fluoro-4-nitrophenyl
vinyl



1.3.1095
3-chloro-4-nitrophenyl
vinyl



1.3.1096
3-bromo-4-nitrophenyl
vinyl



1.3.1097
3-methyl-4-nitrophenyl
vinyl



1.3.1098
3-cyclopropyl-4-nitrophenyl
vinyl



1.3.1099
3-cyano-4-nitrophenyl
vinyl



1.3.1100
3-trifluoromethyl-4-nitrophenyl
vinyl



1.3.1101
3-methoxy-4-nitrophenyl
vinyl



1.3.1102
3-ethoxy-4-nitrophenyl
vinyl



1.3.1103
3-trifluoromethoxy-4-nitrophenyl
vinyl



1.3.1104
3-fluoro-4-methylsulfanylphenyl
vinyl



1.3.1105
3-chloro-4-methylsulfanylphenyl
vinyl



1.3.1106
3-bromo-4-methylsulfanylphenyl
vinyl



1.3.1107
3-methyl-4-methylsulfanylphenyl
vinyl



1.3.1108
3-cyclopropyl-4-methylsulfanylphenyl
vinyl



1.3.1109
3-cyano-4-methylsulfanylphenyl
vinyl



1.3.1110
3-trifluoromethyl-4-methylsulfanylphenyl
vinyl



1.3.1111
3-methoxy-4-methylsulfanylphenyl
vinyl



1.3.1112
3-ethoxy-4-methylsulfanylphenyl
vinyl



1.3.1113
3-trifluoromethoxy-4-methylsulfanylphenyl
vinyl



1.3.1114
3-nitro-4-methylsulfanylphenyl
vinyl



1.3.1115
3,6-difluorophenyl
vinyl



1.3.1116
3,6-difluorophenyl
1-methylvinyl



1.3.1117
3,6-difluorophenyl
allyl



1.3.1118
3,6-difluorophenyl
1-chlorovinyl



1.3.1119
3,6-difluorophenyl
ethynyl



1.3.1120
3-chloro-6-fluorophenyl
vinyl



1.3.1121
3-bromo-6-fluorophenyl
vinyl



1.3.1122
3-methyl-6-fluorophenyl
vinyl



1.3.1123
3-ethyl-6-fluorophenyl
vinyl



1.3.1124
3-cyclopropyl-6-fluorophenyl
vinyl



1.3.1125
3-cyano-6-fluorophenyl
vinyl



1.3.1126
3-methoxy-6-fluorophenyl
vinyl



1.3.1127
3-ethoxy-6-fluorophenyl
vinyl



1.3.1128
3-trifluoromethoxy-6-fluorophenyl
vinyl



1.3.1129
3-nitro-6-fluorophenyl
vinyl



1.3.1130
3-fluoro-6-chlorophenyl
vinyl



1.3.1131
3-fluoro-6-chlorophenyl
1-methylvinyl



1.3.1132
3-fluoro-6-chlorophenyl
allyl



1.3.1133
3-fluoro-6-chlorophenyl
1-chlorovinyl



1.3.1134
3-fluoro-6-chlorophenyl
ethynyl



1.3.1135
3,6-dichlorophenyl
vinyl



1.3.1136
3,6-dichlorophenyl
1-methylvinyl



1.3.1137
3,6-dichlorophenyl
allyl



1.3.1138
3,6-dichlorophenyl
1-chlorovinyl



1.3.1139
3,6-dichlorophenyl
ethynyl



1.3.1140
3-bromo-6-chlorophenyl
vinyl



1.3.1141
3-methyl-6-chlorophenyl
vinyl



1.3.1142
3-cyclopropyl-6-chlorophenyl
vinyl



1.3.1143
3-cyano-6-chlorophenyl
vinyl



1.3.1144
3-trifluoromethyl-6-chlorophenyl
vinyl



1.3.1145
3-methoxy-6-chlorophenyl
vinyl



1.3.1146
3-ethoxy-6-chlorophenyl
vinyl



1.3.1147
3-trifluoromethoxy-6-chlorophenyl
vinyl



1.3.1148
3-nitro-6-chlorophenyl
vinyl



1.3.1149
3-fluoro-6-bromophenyl
vinyl



1.3.1150
3-chloro-6-bromophenyl
vinyl



1.3.1151
3,6-dibromophenyl
vinyl



1.3.1152
3-methyl-6-bromophenyl
vinyl



1.3.1153
3-cyclopropyl-6-bromophenyl
vinyl



1.3.1154
3-cyano-6-bromophenyl
vinyl



1.3.1155
3-trifluoromethyl-6-bromophenyl
vinyl



1.3.1156
3-methoxy-6-phenyl
vinyl



1.3.1157
3-ethoxy-6-bromophenyl
vinyl



1.3.1158
3-trifluoromethoxy-6-bromophenyl
vinyl



1.3.1159
3-nitro-6-bromophenyl
vinyl



1.3.1160
3-fluoro-6-iodophenyl
vinyl



1.3.1161
3-chloro-6-iodophenyl
vinyl



1.3.1162
3-bromo-6-iodophenyl
vinyl



1.3.1163
3-methyl-6-iodophenyl
vinyl



1.3.1164
3-cyclopropyl-6-iodophenyl
vinyl



1.3.1165
3-cyano-6-iodophenyl
vinyl



1.3.1166
3-trifluoromethyl-6-iodophenyl
vinyl



1.3.1167
3-methoxy-6-iodophenyl
vinyl



1.3.1168
3-ethoxy-6-iodophenyl
vinyl



1.3.1169
3-trifluoromethoxy-6-iodophenyl
vinyl



1.3.1170
3-nitro-6-iodophenyl
vinyl



1.3.1171
3-fluoro-6-methylphenyl
vinyl



1.3.1172
3-chloro-6-methylphenyl
vinyl



1.3.1173
3-bromo-6-methylphenyl
vinyl



1.3.1174
3,6-dimethylphenyl
vinyl



1.3.1175
3-ethyl-6-methylphenyl
vinyl



1.3.1176
3-cyclopropyl-6-methylphenyl
vinyl



1.3.1177
3-cyano-6-methylphenyl
vinyl



1.3.1178
3-trifluoromethyl-6-methylphenyl
vinyl



1.3.1179
3-methoxy-6-methylphenyl
vinyl



1.3.1180
3-ethoxy-6-methylphenyl
vinyl



1.3.1181
3-trifluoromethoxy-6-methylphenyl
vinyl



1.3.1182
3-nitro-6-methylphenyl
vinyl



1.3.1183
3-fluoro-6-ethylphenyl
vinyl



1.3.1184
3-chloro-6-ethylphenyl
vinyl



1.3.1185
3-bromo-6-ethylphenyl
vinyl



1.3.1186
3-methyl-6-ethylphenyl
vinyl



1.3.1187
3,6-diethylphenyl
vinyl



1.3.1188
3-cyclopropyl-6-ethylphenyl
vinyl



1.3.1189
3-cyano-6-ethylphenyl
vinyl



1.3.1190
3-trifluoromethyl-6-ethylphenyl
vinyl



1.3.1191
3-methoxy-6-ethylphenyl
vinyl



1.3.1192
3-ethoxy-6-ethylphenyl
vinyl



1.3.1193
3-trifluoromethoxy-6-ethylphenyl
vinyl



1.3.1194
3-nitro-6-ethylphenyl
vinyl



1.3.1195
3-fluoro-6-propylphenyl
vinyl



1.3.1196
3-chloro-6-propylphenyl
vinyl



1.3.1197
3-bromo-6-propylphenyl
vinyl



1.3.1198
3-methyl-6-propylphenyl
vinyl



1.3.1199
3-methyl-6-propylphenyl
vinyl



1.3.1200
3-cyclopropyl-6-propylphenyl
vinyl



1.3.1201
3-cyano-6-propylphenyl
vinyl



1.3.1202
3-trifluoromethyl-6-propylphenyl
vinyl



1.3.1203
3-methoxy-6-propylphenyl
vinyl



1.3.1204
3-ethoxy-6-propylphenyl
vinyl



1.3.1205
3-trifluoromethoxy-6-propylphenyl
vinyl



1.3.1206
3-nitro-6-propylphenyl
vinyl



1.3.1207
3-fluoro-6-isopropylphenyl
vinyl



1.3.1208
3-chloro-6-isopropylphenyl
vinyl



1.3.1209
3-bromo-6-isopropylphenyl
vinyl



1.3.1210
3-methyl-6-isopropylphenyl
vinyl



1.3.1211
3-cyclopropyl-6-isopropylphenyl
vinyl



1.3.1212
3-cyano-6-isopropylphenyl
vinyl



1.3.1213
3-trifluoromethyl-6-isopropylphenyl
vinyl



1.3.1214
3-methoxy-6-isopropylphenyl
vinyl



1.3.1215
3-ethoxy-6-isopropylphenyl
vinyl



1.3.1216
3-trifluoromethoxy-6-isopropylphenyl
vinyl



1.3.1217
3-nitro-6-isopropylphenyl
vinyl



1.3.1218
3-fluoro-6-tert-butylphenyl
vinyl



1.3.1219
3-chloro-6-tert-butylphenyl
vinyl



1.3.1220
3-bromo-6-tert-butylphenyl
vinyl



1.3.1221
3-methyl-6-tert-butylphenyl
vinyl



1.3.1222
3-cyclopropyl-6-tert-butylphenyl
vinyl



1.3.1223
3-cyano-6-tert-butylphenyl
vinyl



1.3.1224
3-trifluoromethyl-6-tert-butylphenyl
vinyl



1.3.1225
3-methoxy-6-tert-butylphenyl
vinyl



1.3.1226
3-ethoxy-6-tert-butylphenyl
vinyl



1.3.1227
3-trifluoromethoxy-6-tert-butylphenyl
vinyl



1.3.1228
3-nitro-6-tert-butylphenyl
vinyl



1.3.1229
3-fluoro-6-cyclopropylphenyl
vinyl



1.3.1230
3-chloro-6-cyclopropylphenyl
vinyl



1.3.1231
3-bromo-6-cyclopropylphenyl
vinyl



1.3.1232
3-methyl-6-cyclopropylphenyl
vinyl



1.3.1233
3-cyclopropyl-6-cyclopropylphenyl
vinyl



1.3.1234
3-cyano-6-cyclopropylphenyl
vinyl



1.3.1235
3-trifluoromethyl-6-cyclopropylphenyl
vinyl



1.3.1236
3-methoxy-6-cyclopropylphenyl
vinyl



1.3.1237
3-ethoxy-6-cyclopropylphenyl
vinyl



1.3.1238
3-trifluoromethoxy-6-cyclopropylphenyl
vinyl



1.3.1239
3-fluoro-6-methoxycarbonylphenyl
vinyl



1.3.1240
3-chloro-6-methoxycarbonylphenyl
vinyl



1.3.1241
3-bromo-6-methoxycarbonylphenyl
vinyl



1.3.1242
3-methyl-6-methoxycarbonylphenyl
vinyl



1.3.1243 
3-cyclopropyl-6-methoxycarbonylphenyl
vinyl



1.3.1244
3-cyano-6-methoxycarbonylphenyl
vinyl



1.3.1245
3-trifluoromethyl-6-methoxycarbonyl-
vinyl




phenyl




1.3.1246
3-methoxy-6-methoxycarbonylphenyl
vinyl



1.3.1247
3-ethoxy-6-methoxycarbonylphenyl
vinyl



1.3.1248
3-trifluoromethoxy-6-methoxycarbonyl-
vinyl




phenyl




1.3.1249
3-nitro-6-methoxycarbonylphenyl
vinyl



1.3.1250
3-fluoro-6-cyanophenyl
vinyl



1.3.1251
3-chloro-6-cyanophenyl
vinyl



1.3.1252
3-bromo-6-cyanophenyl
vinyl



1.3.1253
3-methyl-6-cyanophenyl
vinyl



1.3.1254
3-cyclopropyl-6-cyanophenyl
vinyl



1.3.1255
3-cyano-6-cyanophenyl
vinyl



1.3.1256
3-trifluoromethyl-6-cyanophenyl
vinyl



1.3.1257
3-methoxy-6-cyanophenyl
vinyl



1.3.1258
3-ethoxy-6-cyanophenyl
vinyl



1.3.1259
3-trifluoromethoxy-6-cyanophenyl
vinyl



1.3.1260
3-nitro-6-cyanophenyl
vinyl



1.3.1261
3-fluoro-6-methoxyphenyl
vinyl



1.3.1262
3-chloro-6-methoxyphenyl
vinyl



1.3.1263
3-bromo-6-methoxyphenyl
vinyl



1.3.1264
3-methyl-6-methoxyphenyl
vinyl



1.3.1265
3-cyclopropyl-6-methoxyphenyl
vinyl



1.3.1266
3-cyano-6-methoxyphenyl
vinyl



1.3.1267
3-trifluoromethyl-6-methoxyphenyl
vinyl



1.3.1268
3,6-dimethoxyphenyl
vinyl



1.3.1269
3-ethoxy-6-methoxyphenyl
vinyl



1.3.1270
3-trifluoromethoxy-6-methoxyphenyl
vinyl



1.3.1271
3-nitro-6-methoxyphenyl
vinyl



1.3.1272
3-fluoro-6-ethoxyphenyl
vinyl



1.3.1273
3-chloro-6-ethoxyphenyl
vinyl



1.3.1274
3-bromo-6-ethoxyphenyl
vinyl



1.3.1275
3-methyl-6-ethoxyphenyl
vinyl



1.3.1276
3-cyclopropyl-6-ethoxyphenyl
vinyl



1.3.1277
3-cyano-6-ethoxyphenyl
vinyl



1.3.1278
3-trifluoromethyl-6-ethoxyphenyl
vinyl



1.3.1279
3-methoxy-6-ethoxyphenyl
vinyl



1.3.1280
2,6-diethoxyphenyl
vinyl



1.3.1281
3-trifluoromethoxy-6-ethoxyphenyl
vinyl



1.3.1282
3-nitro-6-ethoxyphenyl
vinyl



1.3.1283
3-fluoro-6-isopropoxyphenyl
vinyl



1.3.1284
3-chloro-6-isopropoxyphenyl
vinyl



1.3.1285
3-bromo-6-isopropoxyphenyl
vinyl



1.3.1286
3-methyl-6-isopropoxyphenyl
vinyl



1.3.1287
3-cyclopropyl-6-isopropoxyphenyl
vinyl



1.3.1288
3-cyano-6-isopropoxyphenyl
vinyl



1.3.1289
3-trifluoromethyl-6-isopropoxyphenyl
vinyl



1.3.1290
3-methoxy-6-isopropoxyphenyl
vinyl



1.3.1291
3-ethoxy-6-isopropoxyphenyl
vinyl



1.3.1292 
3-trifluoromethoxy-6-isopropoxyphenyl
vinyl



1.3.1293
3-nitro-6-isopropoxyphenyl
vinyl



1.3.1294
3-fluoro-6-trifluoromethoxyphenyl
vinyl



1.3.1295
3-chloro-6-trifluoromethoxyphenyl
vinyl



1.3.1296
3-bromo-6-trifluoromethoxyphenyl
vinyl



1.3.1297
3-methyl-6-trifluoromethoxyphenyl
vinyl



1.3.1298 
3-cyclopropyl-6-trifluoromethoxyphenyl
vinyl



1.3.1299
3-cyano-6-trifluoromethoxyphenyl
vinyl



1.3.1300
3-trifluoromethyl-6-trifluoromethoxy-
vinyl




phenyl




1.3.1301
3-methoxy-6-trifluoromethoxyphenyl
vinyl



1.3.1302
3-ethoxy-6-trifluoromethoxyphenyl
vinyl



1.3.1303
3,6-bis(trifluoromethoxy)phenyl
vinyl



1.3.1304
3-nitro-6-trifluoromethoxyphenyl
vinyl



1.3.1305
3-fluoro-6-difluoromethoxyphenyl
vinyl



1.3.1306
3-chloro-6-difluoromethoxyphenyl
vinyl



1.3.1307
3-bromo-6-difluoromethoxyphenyl
vinyl



1.3.1308
3-methyl-6-difluoromethoxyphenyl
vinyl



1.3.1309 
3-cyclopropyl-6-difluoromethoxyphenyl
vinyl



1.3.1310
3-cyano-6-difluoromethoxyphenyl
vinyl



1.3.1311
3-trifluoromethyl-6-difluoromethoxyphenyl
vinyl



1.3.1312
3-methoxy-6-difluoromethoxyphenyl
vinyl



1.3.1313
3-ethoxy-6-difluoromethoxyphenyl
vinyl



1.3.1314
3-trifluoromethoxy-6-difluoromethoxy-
vinyl




phenyl




1.3.1315
3-nitro-6-difluoromethoxyphenyl
vinyl



1.3.1316
3-fluoro-6-nitrophenyl
vinyl



1.3.1317
3-chloro-6-nitrophenyl
vinyl



1.3.1318
3-bromo-6-nitrophenyl
vinyl



1.3.1319
3-methyl-6-nitrophenyl
vinyl



1.3.1320
3-cyclopropyl-6-nitrophenyl
vinyl



1.3.1321
3-cyano-6-nitrophenyl
vinyl



1.3.1322
3-trifluoromethyl-6-nitrophenyl
vinyl



1.3.1323
3-methoxy-6-nitrophenyl
vinyl



1.3.1324
3-ethoxy-6-nitrophenyl
vinyl



1.3.1325
3-trifluoromethoxy-6-nitrophenyl
vinyl



1.3.1326
3-fluoro-6-methylsulfanylphenyl
vinyl



1.3.1327
3-chloro-6-methylsulfanylphenyl
vinyl



1.3.1328
3-bromo-6-methylsulfanylphenyl
vinyl



1.3.1329
3-methyl-6-methylsulfanylphenyl
vinyl



1.3.1330
3-cyclopropyl-6-methylsulfanylphenyl
vinyl



1.3.1331
3-cyano-6-methylsulfanylphenyl
vinyl



1.3.1332
3-trifluoromethyl-6-methylsulfanylphenyl
vinyl



1.3.1333
3-methoxy-6-methylsulfanylphenyl
vinyl



1.3.1334
3-ethoxy-6-methylsulfanylphenyl
vinyl



1.3.1335
3-trifluoromethoxy-6-methylsulfanylphenyl
vinyl



1.3.1336
3-nitro-6-methylsulfanylphenyl
vinyl



1.3.1337
2,3,4-trifluorophenyl
vinyl



1.3.1338
2,3,4-trichlorophenyl
vinyl



1.3.1339
2,3,4-trimethylphenyl
vinyl



1.3.1340
2-fluoro-2-chloro-5-trifluoromethylphenyl
vinyl



1.3.1341
2,3,5-trifluorophenyl
vinyl



1.3.1342
2,3,5-trichlorophenyl
vinyl



1.3.1343
2,3,5-trimethylphenyl
vinyl



1.3.1344
2,3-dichloro-5-methoxyphenyl
vinyl



1.3.1345
2,3,6-trifluorophenyl
vinyl



1.3.1346
2,3,6-trichlorophenyl
vinyl



1.3.1347
2,3,6-trimethylphenyl
vinyl



1.3.1348
3,4,5-trifluorophenyl
vinyl



1.3.1349
3,4,5-trichlorophenyl
vinyl



1.3.1350
3,4,5-trimethylphenyl
vinyl



1.3.1351
3,5-dimethyl-4-fluorophenyl
vinyl



1.3.1352
3,5-dichloro-4-methoxyphenyl
vinyl



1.3.1353
3,5-difluoro-4-chlorophenyl
vinyl



1.3.1354
3,5-dichloro-4-hydroxyphenyl
vinyl



1.3.1355
3,5-trifluoromethyl-4-chlorophenyl
vinyl



1.3.1356
3,4,6-trifluorophenyl
vinyl



1.3.1357
3,4,6-trichlorophenyl
vinyl



1.3.1358
3,4,6-trimethylphenyl
vinyl



1.3.1359
pentafluorophenyl
vinyl
















TABLE 1.4







Inventive compounds of the general formula (I) in which W* is COOH, R1


and R2 are each hydrogen, and aryl is the radical.








 








 













Physical


No.
Aryl
Alkyl
data





1.4.1
3-fluorophenyl
methyl



1.4.2
3-fluorophenyl
ethyl



1.4.3
3-fluorophenyl
propyl



1.4.4
3-fluorophenyl
butyl



1.4.5
3-chlorophenyl
methyl



1.4.6
3-chlorophenyl
ethyl



1.4.7
3-chlorophenyl
propyl



1.4.8
3-chlorophenyl
butyl



1.4.9
3-bromophenyl
methyl



1.4.10
3-bromophenyl
ethyl



1.4.11
3-iodophenyl
methyl



1.4.12
3-iodophenyl
ethyl



1.4.13
3-methylphenyl
methyl



1.4.14
3-methylphenyl
ethyl



1.4.15
3-ethylphenyl
methyl



1.4.16
3-propylphenyl
methyl



1.4.17
3-isopropylphenyl
methyl



1.4.18
3-n-butylphenyl
methyl



1.4.19
3-i-butylphenyl
methyl



1.4.20
3-tert-butylphenyl
methyl



1.4.21
3-cyclopropylphenyl
methyl



1.4.22
3-cyclobutylphenyl
methyl



1.4.23
3-cyclopentylphenyl
methyl



1.4.24
3-vinylphenyl
methyl



1.4.25
3-ethynylphenyl
methyl



1.4.26
3-cyanophenyl
methyl



1.4.27
3-trifluoromethylphenyl
methyl



1.4.28
3-difluoromethylphenyl
methyl



1.4.29
3-(hydroxycarbonyl)phenyl
methyl



1.4.30
3-(methoxycarbonyl)phenyl
methyl



1.4.31
3-(ethoxycarbonyl)phenyl
methyl



1.4.32
3-hydroxymethylphenyl
methyl



1.4.33
3-carbamoylphenyl
methyl



1.4.34
3-hydroxyphenyl
methyl



1.4.35
3-methoxyphenyl
methyl



1.4.36
3-ethoxyphenyl
methyl



1.4.37
3-propyloxyphenyl
methyl



1.4.38
3-isopropyloxyphenyl
methyl



1.4.39
3-n-butyloxyphenyl
methyl



1.4.40
3-i-butyloxyphenyl
methyl



1.4.41
3-t-butyloxyphenyl
methyl



1.4.42
3-difluoromethoxyphenyl
methyl



1.4.43
3-trifluoromethoxyphenyl
methyl



1.4.44
3-(2,2,2-trifluoroethoxy)phenyl
methyl



1.4.45
3-(2-chloroethoxy)phenyl
methyl



1.4.46
3-(2-hydroxyethoxy)phenyl
methyl



1.4.47
3-(2-methoxyethoxy)phenyl
methyl



1.4.48
3-[(tert-butoxycarbonyl)oxy]phenyl
methyl



1.4.49
3-nitrophenyl
methyl



1.4.50
3-acetoxyphenyl
methyl



1.4.51
{3-[(tert-butoxycarbonyl)amino]phenyl}
methyl



1.4.52
3-methylsulfanylphenyl
methyl



1.4.53
3-(pentafluoro-lambda6-sulfanyl)phenyl
methyl



1.4.54
2,3-difluorophenyl
methyl



1.4.55
2,3-difluorophenyl
ethyl



1.4.56
2,3-difluorophenyl
propyl



1.4.57
2,3-difluorophenyl
butyl



1.4.58
2-chloro-3-fluorophenyl
methyl



1.4.59
2-bromo-3-fluorophenyl
methyl



1.4.60
2-methyl-3-fluorophenyl
methyl



1.4.61
2-cyclopropyl-3-fluorophenyl
methyl



1.4.62
2-cyano-3-fluorophenyl
methyl



1.4.63
2-methoxy-3-fluorophenyl
methyl



1.4.64
2-ethoxy-3-fluorophenyl
methyl



1.4.65
2-trifluoromethoxy-3-fluorophenyl
methyl



1.4.66
2-nitro-3-fluorophenyl
methyl



1.4.67
2-fluoro-3-chlorophenyl
methyl



1.4.68
2,3-dichlorophenyl
methyl



1.4.69
2,3-dichlorophenyl
ethyl



1.4.70
2,3-dichlorophenyl
propyl



1.4.71
2,3-dichlorophenyl
butyl



1.4.72
2-bromo-3-chlorophenyl
methyl



1.4.73
2-methyl-3-chlorophenyl
methyl



1.4.74
2-cyclopropyl-3-chlorophenyl
methyl



1.4.75
2-cyano-3-chlorophenyl
methyl



1.4.76
2-trifluoromethyl-2-chlorophenyl
methyl



1.4.77
2-methoxy-3-chlorophenyl
methyl



1.4.78
2-ethoxy-3-chlorophenyl
methyl



1.4.79
2-trifluoromethoxy-3-chlorophenyl
methyl



1.4.80
2-nitro-3-chlorophenyl
methyl



1.4.81
2-fluoro-3-bromophenyl
methyl



1.4.82
2-chloro-3-bromophenyl
methyl



1.4.83
2,3-dibromophenyl
methyl



1.4.84
2-methyl-3-bromophenyl
methyl



1.4.85
2-ethyl-3-bromophenyl
methyl



1.4.86
2-cyclopropyl-3-bromophenyl
methyl



1.4.87
2-cyano-3-bromophenyl
methyl



1.4.88
2-trifluoromethyl-3-bromophenyl
methyl



1.4.89
2-methoxy-3-phenyl
methyl



1.4.90
2-ethoxy-3-bromophenyl
methyl



1.4.91
2-trifluoromethoxy-3-bromophenyl
methyl



1.4.92
2-nitro-3-bromophenyl
methyl



1.4.93
2-fluoro-3-iodophenyl
methyl



1.4.94
2-chloro-3-iodophenyl
methyl



1.4.95
2-bromo-3-iodophenyl
methyl



1.4.96
2-methyl-3-iodophenyl
methyl



1.4.97
2-cyclopropyl-3-iodophenyl
methyl



1.4.98
2-cyano-3-iodophenyl
methyl



1.4.99
2-trifluoromethyl-3-iodophenyl
methyl



1.4.100
2-methoxy-3-iodophenyl
methyl



1.4.101
2-ethoxy-3-iodophenyl
methyl



1.4.102
2-trifluoromethoxy-3-iodophenyl
methyl



1.4.103
2-fluoro-3-methylphenyl
methyl



1.4.104
2-fluoro-3-methylphenyl
ethyl



1.4.105
2-fluoro-3-methylphenyl
propyl



1.4.106
2-fluoro-3-methylphenyl
butyl



1.4.107
2-chloro-3-methylphenyl
methyl



1.4.108
2-chloro-3-methylphenyl
ethyl



1.4.109
2-chloro-3-methylphenyl
propyl



1.4.110
2-chloro-3-methylphenyl
butyl



1.4.111
2-bromo-3-methylphenyl
methyl



1.4.112
2,3-dimethylphenyl
methyl



1.4.113
2,3-dimethylphenyl
ethyl



1.4.114
2,3-dimethylphenyl
propyl



1.4.115
2,3-dimethylphenyl
butyl



1.4.116
2-cyclopropyl-3-methylphenyl
methyl



1.4.117
2-cyano-3-methylphenyl
methyl



1.4.118
2-trifluoromethyl-3-methylphenyl
methyl



1.4.119
2-methoxy-3-methylphenyl
methyl



1.4.120
2-ethoxy-3-methylphenyl
methyl



1.4.121
2-trifluoromethoxy-3-methylphenyl
methyl



1.4.122
2-nitro-3-methylphenyl
methyl



1.4.123
2-fluoro-3-ethylphenyl
methyl



1.4.124
2-chloro-3-ethylphenyl
methyl



1.4.125
2-bromo-3-ethylphenyl
methyl



1.4.126
2-methyl-3-ethylphenyl
methyl



1.4.127
2,3-diethylphenyl
methyl



1.4.128
2-cyclopropyl-3-ethylphenyl
methyl



1.4.129
2-cyano-3-ethylphenyl
methyl



1.4.130
2-trifluoromethyl-3-ethylphenyl
methyl



1.4.131
2-methoxy-3-ethylphenyl
methyl



1.4.132
2-ethoxy-3-ethylphenyl
methyl



1.4.133
2-trifluoromethoxy-3-ethylphenyl
methyl



1.4.134
2-nitro-3-ethylphenyl
methyl



1.4.135
2-fluoro-3-propylphenyl
methyl



1.4.136
2-chloro-3-propylphenyl
methyl



1.4.137
2-bromo-3-propylphenyl
methyl



1.4.138
2-methyl-3-propylphenyl
methyl



1.4.139
2-cyclopropyl-3-propylphenyl
methyl



1.4.140
2-cyano-3-propylphenyl
methyl



1.4.141
2-trifluoromethyl-3-propylphenyl
methyl



1.4.142
2-methoxy-3-propylphenyl
methyl



1.4.143
2-ethoxy-3-propylphenyl
methyl



1.4.144
2-trifluoromethoxy-3-propylphenyl
methyl



1.4.145
2-nitro-3-propylphenyl
methyl



1.4.146
2-fluoro-3-isopropylphenyl
methyl



1.4.147
2-chloro-3-isopropylphenyl
methyl



1.4.148
2-bromo-3-isopropylphenyl
methyl



1.4.149
2-methyl-3-isopropylphenyl
methyl



1.4.150
2-cyclopropyl-3-isopropylphenyl
methyl



1.4.151
2-cyano-3-isopropylphenyl
methyl



1.4.152
2-trifluoromethyl-3-isopropylphenyl
methyl



1.4.153
2-methoxy-3-isopropylphenyl
methyl



1.4.154
2-ethoxy-3-isopropylphenyl
methyl



1.4.155
2-trifluoromethoxy-3-isopropylphenyl
methyl



1.4.156
2-nitro-3-isopropylphenyl
methyl



1.4.157
2-fluoro-3-tert-butylphenyl
methyl



1.4.158
2-chloro-3-tert-butylphenyl
methyl



1.4.159
2-bromo-3-tert-butylphenyl
methyl



1.4.160
2-methyl-3-tert-butylphenyl
methyl



1.4.161
2-cyano-3-tert-butylphenyl
methyl



1.4.162
2-trifluoromethyl-3-tert-butylphenyl
methyl



1.4.163
2-methoxy-3-tert-butylphenyl
methyl



1.4.164
2-ethoxy-3-tert-butylphenyl
methyl



1.4.165
2-nitro-3-tert-butylphenyl
methyl



1.4.166
2-fluoro-3-cyclopropylphenyl
methyl



1.4.167
2-chloro-3-cyclopropylphenyl
methyl



1.4.168
2-bromo-3-cyclopropylphenyl
methyl



1.4.169
2-methyl-3-cyclopropylphenyl
methyl



1.4.170
2-cyano-3-cyclopropylphenyl
methyl



1.4.171
2-trifluoromethyl-3-cyclopropylphenyl
methyl



1.4.172
2-methoxy-3-cyclopropylphenyl
methyl



1.4.173
2-trifluoromethoxy-3-cyclopropylphenyl
methyl



1.4.174
2-fluoro-3-methoxycarbonylphenyl
methyl



1.4.175
2-chloro-3-methoxycarbonylphenyl
methyl



1.4.176
2-bromo-3-methoxycarbonylphenyl
methyl



1.4.177
2-methyl-3-methoxycarbonylphenyl
methyl



1.4.178
2-cyclopropyl-3-methoxycarbonylphenyl
methyl



1.4.179
2-cyano-3-methoxycarbonylphenyl
methyl



1.4.180
2-trifluoromethyl-3-
methyl




methoxycarbonylphenyl




1.4.181
2-methoxy-3-methoxycarbonylphenyl
methyl



1.4.182
2-ethoxy-3-methoxycarbonylphenyl
methyl



1.4.183
2-trifluoromethoxy-3-
methyl




methoxycarbonylphenyl




1.4.184
2-nitro-3-methoxycarbonylphenyl
methyl



1.4.185
2-fluoro-3-cyanophenyl
methyl



1.4.186
2-chloro-3-cyanophenyl
methyl



1.4.187
2-bromo-3-cyanophenyl
methyl



1.4.188
2-methyl-3-cyanophenyl
methyl



1.4.189
2-ethyl-3-cyanophenyl
methyl



1.4.190
2-ethyl-3-cyanophenyl
ethyl



1.4.191
2-ethyl-3-cyanophenyl
propyl



1.4.192
2-ethyl-3-cyanophenyl
butyl



1.4.193
2-cyclopropyl-3-cyanophenyl
methyl



1.4.194
2-cyano-3-cyanophenyl
methyl



1.4.195
2-trifluoromethyl-3-cyanophenyl
methyl



1.4.196
2-methoxy-3-cyanophenyl
methyl



1.4.197
2-ethoxy-3-cyanophenyl
methyl



1.4.198
2-trifluoromethoxy-3-cyanophenyl
methyl



1.4.199
2-fluoro-3-methoxyphenyl
methyl



1.4.200
2-chloro-3-methoxyphenyl
methyl



1.4.201
2-bromo-3-methoxyphenyl
methyl



1.4.202
2-methyl-3-methoxyphenyl
methyl



1.4.203
2-cyclopropyl-3-methoxyphenyl
methyl



1.4.204
2-cyano-3-methoxyphenyl
methyl



1.4.205
2-trifluoromethyl-3-methoxyphenyl
methyl



1.4.206
2,3-dimethoxyphenyl
methyl



1.4.207
2-ethoxy-3-methoxyphenyl
methyl



1.4.208
2-trifluoromethoxy-3-methoxyphenyl
methyl



1.4.209
2-nitro-3-methoxyphenyl
methyl



1.4.210
2-fluoro-3-ethoxyphenyl
methyl



1.4.211
2-chloro-3-ethoxyphenyl
methyl



1.4.212
2-bromo-3-ethoxyphenyl
methyl



1.4.213
2-methyl-3-ethoxyphenyl
methyl



1.4.214
2-ethyl-3-ethoxyphenyl
methyl



1.4.215
2-cyclopropyl-3-ethoxyphenyl
methyl



1.4.216
2-cyano-3-ethoxyphenyl
methyl



1.4.217
2-trifluoromethyl-3-ethoxyphenyl
methyl



1.4.218
2-methoxy-3-ethoxyphenyl
methyl



1.4.219
2,3-diethoxyphenyl
methyl



1.4.220
2-trifluoromethoxy-3-ethoxyphenyl
methyl



1.4.221
2-nitro-3-ethoxyphenyl
methyl



1.4.222
2-fluoro-3-isopropoxyphenyl
methyl



1.4.223
2-chloro-3-isopropoxyphenyl
methyl



1.4.224
2-bromo-3-isopropoxyphenyl
methyl



1.4.225
2-methyl-3-isopropoxyphenyl
methyl



1.4.226
2-ethyl-3-isopropoxyphenyl
methyl



1.4.227
2-cyclopropyl-3-isopropoxyphenyl
methyl



1.4.228
2-cyano-3-isopropoxyphenyl
methyl



1.4.229
2-trifluoromethyl-3-isopropoxyphenyl
methyl



1.4.230
2-methoxy-3-isopropoxyphenyl
methyl



1.4.231
2-ethoxy-3-isopropoxyphenyl
methyl



1.4.232
2-trifluoromethoxy-3-isopropoxyphenyl
methyl



1.4.233
2-nitro-3-isopropoxyphenyl
methyl



1.4.234
2-fluoro-3-trifluoromethoxyphenyl
methyl



1.4.235
2-chloro-3-trifluoromethoxyphenyl
methyl



1.4.236
2-bromo-3-trifluoromethoxyphenyl
methyl



1.4.237
2-methyl-3-trifluoromethoxyphenyl
methyl



1.4.238
2-cyclopropyl-3-trifluoromethoxyphenyl
methyl



1.4.239
2-cyano-3-trifluoromethoxyphenyl
methyl



1.4.240
2-trifluoromethyl-3-trifluoromethoxy-
methyl




phenyl




1.4.241
2-methoxy-3-trifluoromethoxyphenyl
methyl



1.4.242
2-ethoxy-3-trifluoromethoxyphenyl
methyl



1.4.243
2,3-bis(trifluoromethoxy)phenyl
methyl



1.4.244
2-nitro-3-trifluoromethoxyphenyl
methyl



1.4.245
2-fluoro-3-difluoromethoxyphenyl
methyl



1.4.246
2-chloro-3-difluoromethoxyphenyl
methyl



1.4.247
2-bromo-3-difluoromethoxyphenyl
methyl



1.4.248
2-methyl-3-difluoromethoxyphenyl
methyl



1.4.249
2-cyclopropyl-3-difluoromethoxyphenyl
methyl



1.4.250
2-cyano-3-difluoromethoxyphenyl
methyl



1.4.251
2-trifluoromethyl-3-difluoromethoxy-
methyl




phenyl




1.4.252
2-methoxy-3-difluoromethoxyphenyl
methyl



1.4.253
2-ethoxy-3-difluoromethoxyphenyl
methyl



1.4.254
2-trifluoromethoxy-3-difluoromethoxy-
methyl




phenyl




1.4.255
2-nitro-3-difluoromethoxyphenyl
methyl



1.4.256
2-fluoro-3-nitrophenyl
methyl



1.4.257
2-chloro-3-nitrophenyl
methyl



1.4.258
2-bromo-3-nitrophenyl
methyl



1.4.259
2-methyl-3-nitrophenyl
methyl



1.4.260
2-cyclopropyl-3-nitrophenyl
methyl



1.4.261
2-cyano-3-nitrophenyl
methyl



1.4.262
2-trifluoromethyl-3-nitrophenyl
methyl



1.4.263
2-methoxy-3-nitrophenyl
methyl



1.4.264
2-ethoxy-3-nitrophenyl
methyl



1.4.265
2-trifluoromethoxy-3-nitrophenyl
methyl



1.4.266
2-fluoro-3-methylsulfanylphenyl
methyl



1.4.267
2-chloro-3-methylsulfanylphenyl
methyl



1.4.268
2-bromo-3-methylsulfanylphenyl
methyl



1.4.269
2-methyl-3-methylsulfanylphenyl
methyl



1.4.270
2-ethyl-3-methylsulfanylphenyl
methyl



1.4.271
2-cyclopropyl-3-methylsulfanylphenyl
methyl



1.4.272
2-trifluoromethyl-3-methylsulfanylphenyl
methyl



1.4.273
2-methoxy-3-methylsulfanylphenyl
methyl



1.4.274
3,5-difluorophenyl
methyl



1.4.275
3,5-difluorophenyl
ethyl



1.4.276
3,5-difluorophenyl
propyl



1.4.277
3,5-difluorophenyl
butyl



1.4.278
3-chloro-5-fluorophenyl
methyl



1.4.279
3-chloro-5-fluorophenyl
ethyl



1.4.280
3-chloro-5-fluorophenyl
propyl



1.4.281
3-chloro-5-fluorophenyl
butyl



1.4.282
3-bromo-5-fluorophenyl
methyl



1.4.283
3-bromo-5-fluorophenyl
ethyl



1.4.284
3-bromo-5-fluorophenyl
propyl



1.4.285
3-bromo-5-fluorophenyl
butyl



1.4.286
3-iodo-5-fluorophenyl
methyl



1.4.287
3-methyl-5-fluorophenyl
methyl



1.4.288
3-methyl-5-fluorophenyl
ethyl



1.4.289
3-methyl-5-fluorophenyl
propyl



1.4.290
3-methyl-5-fluorophenyl
butyl



1.4.291
3-propyl-5-fluorophenyl
methyl



1.4.292
3-i-propyl-5-fluorophenyl
methyl



1.4.293
3-n-butyl-5-fluorophenyl
methyl



1.4.294
3-isobutyl-5-fluorophenyl
methyl



1.4.295
3-tert-butyl-5-fluorophenyl
methyl



1.4.296
3-cyclopropyl-5-fluorophenyl
methyl



1.4.297
3-cyano-5-fluorophenyl
methyl



1.4.298
3-trifluoromethyl-5-fluorophenyl
methyl



1.4.299
3-trifluoromethyl-5-fluorophenyl
ethyl



1.4.300
3-trifluoromethyl-5-fluorophenyl
propyl



1.4.301
3-trifluoromethyl-5-fluorophenyl
butyl



1.4.302
3-(methoxycarbonyl)-5-fluorophenyl
methyl



1.4.303
3-methoxy-5-fluorophenyl
methyl



1.4.304
3-ethoxy-5-fluorophenyl
methyl



1.4.305
3-n-propoxy-5-fluorophenyl
methyl



1.4.306
3-isopropoxy-5-fluorophenyl
methyl



1.4.307
3-difluoromethoxy-5-fluorophenyl
methyl



1.4.308
3-trifluoromethoxy-5-fluorophenyl
methyl



1.4.309
3-nitro-5-fluorophenyl
methyl



1.4.310
3-acetoxy-5-fluorophenyl
methyl



1.4.311
3-methylsulfanyl-5-fluorophenyl
methyl



1.4.312
3,5-dichlorophenyl
methyl



1.4.313
3,5-dichlorophenyl
ethyl



1.4.314
3,5-dichlorophenyl
propyl



1.4.315
3,5-dichlorophenyl
butyl



1.4.316
3-bromo-5-chlorophenyl
methyl



1.4.317
3-iodo-5-chlorophenyl
methyl



1.4.318
3-methyl-5-chlorophenyl
methyl



1.4.319
3-ethyl-5-chlorophenyl
methyl



1.4.320
3-propyl-5-chlorophenyl
methyl



1.4.321
3-isopropyl-5-chlorophenyl
methyl



1.4.322
3-n-butyl-5-chlorophenyl
methyl



1.4.323
3-isobutyl-5-chlorophenyl
methyl



1.4.324
3-tert-butyl-5-chlorophenyl
methyl



1.4.325
3-cyclopropyl-5-chlorophenyl
methyl



1.4.326
3-cyano-5-chlorophenyl
methyl



1.4.327
3-trifluoromethyl-5-chlorophenyl
methyl



1.4.328
3-(methoxycarbonyl)-5-chlorophenyl
methyl



1.4.329
3-methoxy-5-chlorophenyl
methyl



1.4.330
3-ethoxy-5-chlorophenyl
methyl



1.4.331
3-n-propoxy-5-chlorophenyl
methyl



1.4.332
3-isopropoxy-5-chlorophenyl
methyl



1.4.333
3-n-butoxy-5-chlorophenyl
methyl



1.4.334
3-isobutoxy-5-chlorophenyl
methyl



1.4.335
3-tert-butoxy-5-chlorophenyl
methyl



1.4.336
3-difluoromethoxy-5-chlorophenyl
methyl



1.4.337
3-trifluoromethoxy-5-chlorophenyl
methyl



1.4.338
3-nitro-5-chlorophenyl
methyl



1.4.339
3-acetoxy-5-chlorophenyl
methyl



1.4.340
3-methylsulfanyl-5-chlorophenyl
methyl



1.4.341
3,5-dibromophenyl
methyl



1.4.342
3,5-dibromophenyl
ethyl



1.4.343
3-iodo-5-bromophenyl
methyl



1.4.344
3-methyl-5-bromophenyl
methyl



1.4.345
3-methyl-5-bromophenyl
ethyl



1.4.346
3-methyl-5-bromophenyl
propyl



1.4.347
3-methyl-5-bromophenyl
butyl



1.4.348
3-ethyl-5-bromophenyl
methyl



1.4.349
3-propyl-5-bromophenyl
methyl



1.4.350
3-isopropyl-5-bromophenyl
methyl



1.4.351
3-n-butyl-5-bromophenyl
methyl



1.4.352
3-isobutyl-5-bromophenyl
methyl



1.4.353
3-tert-butyl-5-bromophenyl
methyl



1.4.354
3-cyclopropyl-5-bromophenyl
methyl



1.4.355
3-cyano-5-bromophenyl
methyl



1.4.356
3-trifluoromethyl-5-bromophenyl
methyl



1.4.357
3-(methoxycarbonyl)-5-bromophenyl
methyl



1.4.358
3-methoxy-5-bromophenyl
methyl



1.4.359
3-ethoxy-5-bromophenyl
methyl



1.4.360
3-n-propoxy-5-bromophenyl
methyl



1.4.361
3-isopropoxy-5-bromophenyl
methyl



1.4.362
3-n-butoxy-5-bromophenyl
methyl



1.4.363
3-isobutoxy-5-bromophenyl
methyl



1.4.364
3-tert-butoxy-5-bromophenyl
methyl



1.4.365
3-difluoromethoxy-5-bromophenyl
methyl



1.4.366
3-trifluoromethoxy-5-bromophenyl
methyl



1.4.367
3-nitro-5-bromophenyl
methyl



1.4.368
3-acetoxy-5-bromophenyl
methyl



1.4.369
3-methylsulfanyl-5-bromophenyl
methyl



1.4.370
3,5-diiodophenyl
methyl



1.4.371
3-methyl-5-iodophenyl
methyl



1.4.372
3-ethyl-5-iodophenyl
methyl



1.4.373
3-propyl-5-iodophenyl
methyl



1.4.374
3-isopropyl-5-iodophenyl
methyl



1.4.375
3-n-butyl-5-iodophenyl
methyl



1.4.376
3-isobutyl-5-iodophenyl
methyl



1.4.377
3-tert-butyl-5-iodophenyl
methyl



1.4.378
3-cyclopropyl-5-iodophenyl
methyl



1.4.379
3-cyano-5-iodophenyl
methyl



1.4.380
3-trifluoromethyl-5-iodophenyl
methyl



1.4.381
3-(methoxycarbonyl)-5-iodophenyl
methyl



1.4.382
3-methoxy-5-iodophenyl
methyl



1.4.383
3-ethoxy-5-iodophenyl
methyl



1.4.384
3-n-propoxy-5-iodophenyl
methyl



1.4.385
3-isopropoxy-5-iodophenyl
methyl



1.4.386
3-isobutoxy-5-iodophenyl
methyl



1.4.387
3-difluoromethoxy-5-iodophenyl
methyl



1.4.388
3-trifluoromethoxy-5-iodophenyl
methyl



1.4.389
3-nitro-5-iodophenyl
methyl



1.4.390
3-acetoxy-5-iodophenyl
methyl



1.4.391
3-methylsulfanyl-5-iodophenyl
methyl



1.4.392
3,5-dimethylphenyl
methyl



1.4.393
3-ethyl-5-methylphenyl
methyl



1.4.394
3-propyl-5-methylphenyl
methyl



1.4.395
3-isopropyl-5-methylphenyl
methyl



1.4.396
3-n-butyl-5-methylphenyl
methyl



1.4.397
3-isobutyl-5-methylphenyl
methyl



1.4.398
3-tert-butyl-5-methylphenyl
methyl



1.4.399
3-cyclopropyl-5-methylphenyl
methyl



1.4.400
3-cyano-5-methylphenyl
methyl



1.4.401
3-trifluoromethyl-5-methylphenyl
methyl



1.4.402
3-(methoxycarbonyl)-5-methylphenyl
methyl



1.4.403
3-methoxy-5-methylphenyl
methyl



1.4.404
3-ethoxy-5-methylphenyl
methyl



1.4.405
3-n-propoxy-5-methylphenyl
methyl



1.4.406
3-n-butoxy-5-methylphenyl
methyl



1.4.407
3-isobutoxy-5-methylphenyl
methyl



1.4.408
3-difluoromethoxy-5-methylphenyl
methyl



1.4.409
3-trifluoromethoxy-5-methylphenyl
methyl



1.4.410
3-nitro-5-methylphenyl
methyl



1.4.411
3-acetoxy-5-methylphenyl
methyl



1.4.412
3-methylsulfanyl-5-methylphenyl
methyl



1.4.413
3,5-diethylphenyl
methyl



1.4.414
3-propyl-5-ethylphenyl
methyl



1.4.415
3-isopropyl-5-ethylphenyl
methyl



1.4.416
3-n-butyl-5-ethylphenyl
methyl



1.4.417
3-isobutyl-5-ethylphenyl
methyl



1.4.418
3-tert-butyl-5-ethylphenyl
methyl



1.4.419
3-cyclopropyl-5-ethylphenyl
methyl



1.4.420
3-cyano-5-ethylphenyl
methyl



1.4.421
3-trifluoromethyl-5-ethylphenyl
methyl



1.4.422
3-(methoxycarbonyl)-5-ethylphenyl
methyl



1.4.423
3-methoxy-5-ethylphenyl
methyl



1.4.424
3-ethoxy-5-ethylphenyl
methyl



1.4.425
3-n-propoxy-5-ethylphenyl
methyl



1.4.426
3-n-butoxy-5-ethylphenyl
methyl



1.4.427
3-isobutoxy-5-ethylphenyl
methyl



1.4.428
3-difluoromethoxy-5-ethylphenyl
methyl



1.4.429
3-trifluoromethoxy-5-ethylphenyl
methyl



1.4.430
3-nitro-5-ethylphenyl
methyl



1.4.431
3-acetoxy-5-ethylphenyl
methyl



1.4.432
3-methylsulfanyl-5-ethylphenyl
methyl



1.4.433
3,5-dipropylphenyl
methyl



1.4.434
3-isopropyl-5-propylphenyl
methyl



1.4.435
3-n-butyl-5-propylphenyl
methyl



1.4.436
3-isobutyl-5-propylphenyl
methyl



1.4.437
3-tert-butyl-5-propylphenyl
methyl



1.4.438
3-cyclopropyl-5-propylphenyl
methyl



1.4.439
3-cyano-5-propylphenyl
methyl



1.4.440
3-trifluoromethyl-5-propylphenyl
methyl



1.4.441
3-(methoxycarbonyl)-5-propylphenyl
methyl



1.4.442
3-methoxy-5-propylphenyl
methyl



1.4.443
3-ethoxy-5-propylphenyl
methyl



1.4.444
3-n-propoxy-5-propylphenyl
methyl



1.4.445
3-n-butoxy-5-propylphenyl
methyl



1.4.446
3-isobutoxy-5-propylphenyl
methyl



1.4.447
3-difluoromethoxy-5-propylphenyl
methyl



1.4.448
3-trifluoromethoxy-5-ethylphenyl
methyl



1.4.449
3-nitro-5-propylphenyl
methyl



1.4.450
3-acetoxy-5-propylphenyl
methyl



1.4.451
3-methylsulfanyl-5-propylphenyl
methyl



1.4.452
3,5-diisopropylphenyl
methyl



1.4.453
3-n-butyl-5-isopropylphenyl
methyl



1.4.454
3-tert-butyl-5-isopropylphenyl
methyl



1.4.455
3-cyclopropyl-5-isopropylphenyl
methyl



1.4.456
3-cyano-5-isopropylphenyl
methyl



1.4.457
3-trifluoromethyl-5-isopropylphenyl
methyl



1.4.458
3-(methoxycarbonyl)-5-isopropylphenyl
methyl



1.4.459
3-methoxy-5-isopropylphenyl
methyl



1.4.460
3-ethoxy-5-isopropylphenyl
methyl



1.4.461
3-n-propoxy-5-isopropylphenyl
methyl



1.4.462
3-n-butoxy-5-isopropylphenyl
methyl



1.4.463
3-isobutoxy-5-isopropylphenyl
methyl



1.4.464
3-difluoromethoxy-5-isopropylphenyl
methyl



1.4.465
3-trifluoromethoxy-5-isopropylphenyl
methyl



1.4.466
3-nitro-5-isopropylphenyl
methyl



1.4.467
3-acetoxy-5-isopropylphenyl
methyl



1.4.468
3-methylsulfanyl-5-isopropylphenyl
methyl



1.4.469
3,5-di isobutylphenyl
methyl



1.4.470
3-tert-butyl-5-isobutylphenyl
methyl



1.4.471
3-cyclopropyl-5-isobutylphenyl
methyl



1.4.472
3-cyano-5-isobutylphenyl
methyl



1.4.473
3-trifluoromethyl-5-isobutylphenyl
methyl



1.4.474
3-(methoxycarbonyl)-5-isobutylphenyl
methyl



1.4.475
3-methoxy-5-isobutylphenyl
methyl



1.4.476
3-ethoxy-5-isobutylphenyl
methyl



1.4.477
3-n-propoxy-5-isobutylphenyl
methyl



1.4.478
3-n-butoxy-5-isobutylphenyl
methyl



1.4.479
3-isobutoxy-5-isobutylphenyl
methyl



1.4.480
3-difluoromethoxy-5-isobutylphenyl
methyl



1.4.481
3-trifluoromethoxy-5-isobutylphenyl
methyl



1.4.482
3-nitro-5-isobutylphenyl
methyl



1.4.483
3-acetoxy-5-isobutylphenyl
methyl



1.4.484
3-methylsulfanyl-5-isobutylphenyl
methyl



1.4.485
3,5-di(tert-butyl)phenyl
methyl



1.4.486
3-cyclopropyl-5-tert-butylphenyl
methyl



1.4.487
3-cyano-5-tert-butylphenyl
methyl



1.4.488
3-trifluoromethyl-5-tert-butylphenyl
methyl



1.4.489
3-methoxy-5-tert-butylphenyl
methyl



1.4.490
3-ethoxy-5-tert-butylphenyl
methyl



1.4.491
3-n-propoxy-5-tert-butylphenyl
methyl



1.4.492
3-n-butoxy-5-tert-butylphenyl
methyl



1.4.493
3-isobutoxy-5-tert-butylphenyl
methyl



1.4.494
3-difluoromethoxy-5-tert-butylphenyl
methyl



1.4.495
3-trifluoromethoxy-5-tert-butylphenyl
methyl



1.4.496
3-nitro-5-tert-butylphenyl
methyl



1.4.497
3-acetoxy-5-tert-butylphenyl
methyl



1.4.498
3-methylsulfanyl-5-tert-butylphenyl
methyl



1.4.499
3-tert-butyl-5-cyclopropylphenyl
methyl



1.4.500
3,5-dicyclopropyl-phenyl
methyl



1.4.501
3-cyano-5-cyclopropylphenyl
methyl



1.4.502
3-trifluoromethyl-5-cyclopropylphenyl
methyl



1.4.503
3-(methoxycarbonyl)-5-cyclopropylphenyl
methyl



1.4.504
3-methoxy-5-cyclopropylphenyl
methyl



1.4.505
3-ethoxy-5-cyclopropylphenyl
methyl



1.4.506
3-n-propoxy-5-cyclopropylphenyl
methyl



1.4.507
3-n-butoxy-5-cyclopropylphenyl
methyl



1.4.508
3-isobutoxy-5-cyclopropylphenyl
methyl



1.4.509
3-difluoromethoxy-5-cyclopropylphenyl
methyl



1.4.510
3-trifluoromethoxy-5-cyclopropylphenyl
methyl



1.4.511
3-nitro-5-cyclopropylphenyl
methyl



1.4.512
3-acetoxy-5-cyclopropylphenyl
methyl



1.4.513
3-methylsulfanyl-5-cyclopropylphenyl
methyl



1.4.514
3,5-dicyanophenyl
methyl



1.4.515
3-trifluoromethyl-5-cyanophenyl
methyl



1.4.516
3-(methoxycarbonyl)-5-cyanophenyl
methyl



1.4.517
3-methoxy-5-cyanophenyl
methyl



1.4.518
3-ethoxy-5-cyanophenyl
methyl



1.4.519
3-n-propoxy-5-cyanophenyl
methyl



1.4.520
3-n-butoxy-5-cyanophenyl
methyl



1.4.521
3-isobutoxy-5-cyanophenyl
methyl



1.4.522
3-difluoromethoxy-5-cyanophenyl
methyl



1.4.523
3-trifluoromethoxy-5-cyanophenyl
methyl



1.4.524
3-nitro-5-cyanophenyl
methyl



1.4.525
3-acetoxy-5-cyanophenyl
methyl



1.4.526
3-methylsulfanyl-5-cyanophenyl
methyl



1.4.527
3,5-di(trifluoromethyl)-phenyl
methyl



1.4.528
3-(methoxycarbonyl)-5-trifluoromethyl-
methyl




phenyl




1.4.529
3-methoxy-5-trifluoromethylphenyl
methyl



1.4.530
3-ethoxy-5-trifluoromethylphenyl
methyl



1.4.531
3-n-propoxy-5-trifluoromethylphenyl
methyl



1.4.532
3-n-butoxy-5-trifluoromethylphenyl
methyl



1.4.533
3-isobutoxy-5-trifluoromethylphenyl
methyl



1.4.534
3-difluoromethoxy-5-trifluoromethyl-
methyl




phenyl




1.4.535
3-trifluoromethoxy-5-trifluoromethyl-
methyl




phenyl




1.4.536
3-nitro-5-trifluoromethylphenyl
methyl



1.4.537
3-acetoxy-5-trifluoromethylphenyl
methyl



1.4.538
3-methylsulfanyl-5-trifluoromethylphenyl
methyl



1.4.539
3-methoxy-5-(methoxycarbonyl)phenyl
methyl



1.4.540
3-ethoxy-5-(methoxycarbonyl)phenyl
methyl



1.4.541
3-n-propoxy-5-(methoxycarbonyl)phenyl
methyl



1.4.542
3-n-butoxy-5-(methoxycarbonyl)phenyl
methyl



1.4.543
3-isobutoxy-5-(methoxycarbonyl)phenyl
methyl



1.4.544
3-difluoromethoxy-5-(methoxycarbonyl)-
methyl




phenyl




1.4.545
3-trifluoromethoxy-5-(methoxycarbonyl)-
methyl




phenyl




1.4.546
3-nitro-5-(methoxycarbonyl)phenyl
methyl



1.4.547
3-acetoxy-5-(methoxycarbonyl)phenyl
methyl



1.4.548
3-methylsulfanyl-5-(methoxycarbonyl)-
methyl




phenyl




1.4.549
3,5-dimethoxyphenyl
methyl



1.4.550
3-ethoxy-5-methoxyphenyl
methyl



1.4.551
3-n-propoxy-5-methoxyphenyl
methyl



1.4.552
3-n-butoxy-5-methoxyphenyl
methyl



1.4.553
3-isobutoxy-5-methoxyphenyl
methyl



1.4.554
3-tert-butoxy-5-methoxyphenyl
methyl



1.4.555
3-difluoromethoxy-5-methoxyphenyl
methyl



1.4.556
3-trifluoromethoxy-5-methoxyphenyl
methyl



1.4.557
3-nitro-5-methoxyphenyl
methyl



1.4.558
3-acetoxy-5-methoxyphenyl
methyl



1.4.559
3-methylsulfanyl-5-methoxyphenyl
methyl



1.4.560
3,5-diethoxyphenyl
methyl



1.4.561
3-n-propoxy-5-ethoxyphenyl
methyl



1.4.562
3-n-butoxy-5-ethoxyphenyl
methyl



1.4.563
3-isobutoxy-5-ethoxyphenyl
methyl



1.4.564
3-difluoromethoxy-5-ethoxyphenyl
methyl



1.4.565
3-trifluoromethoxy-5-ethoxyphenyl
methyl



1.4.566
3-nitro-5-ethoxyphenyl
methyl



1.4.567
3-acetoxy-5-ethoxyphenyl
methyl



1.4.568
3-methylsulfanyl-5-ethoxyphenyl
methyl



1.4.569
3,5-di(isopropoxy)phenyl
methyl



1.4.570
3-n-butoxy-5-isopropoxyphenyl
methyl



1.4.571
3-isobutoxy-5-isopropoxyphenyl
methyl



1.4.572
3-difluoromethoxy-5-isopropoxyphenyl
methyl



1.4.573
3-trifluoromethoxy-5-isopropoxyphenyl
methyl



1.4.574
3-nitro-5-isopropoxyphenyl
methyl



1.4.575
3-acetoxy-5-isopropoxyphenyl
methyl



1.4.576
3-methylsulfanyl-5-isopropoxyphenyl
methyl



1.4.577
3,5-di(trifluoromethoxy)phenyl
methyl



1.4.578
3-nitro-5-trifluoromethoxyphenyl
methyl



1.4.579
3-methylsulfanyl-5-trifluoromethoxy-
methyl




phenyl




1.4.580
3,5-bis(difluoromethoxy)phenyl
methyl



1.4.581
3,5-bis(difluoromethoxy)phenyl
ethyl



1.4.582
3,5-bis(difluoromethoxy)phenyl
propyl



1.4.583
3,5-bis(difluoromethoxy)phenyl
butyl



1.4.584
3-trifluoromethoxy-5-difluoromethoxy-
methyl




phenyl




1.4.585
3-nitro-5-difluoromethoxyphenyl
methyl



1.4.586
3-acetoxy-5-difluoromethoxyphenyl
methyl



1.4.587
3-methylsulfanyl-5-difluoromethoxy-
methyl




phenyl




1.4.588
3-acetoxy-5-nitrophenyl
methyl



1.4.589
3-methylsulfanyl-5-nitrophenyl
methyl



1.4.590
3,4-difluorophenyl
methyl



1.4.591
3,4-difluorophenyl
ethyl



1.4.592
3,4-difluorophenyl
propyl



1.4.593
3,4-difluorophenyl
butyl



1.4.594
3-chloro-4-fluorophenyl
methyl



1.4.595
3-chloro-4-fluorophenyl
ethyl



1.4.596
3-chloro-4-fluorophenyl
propyl



1.4.597
3-chloro-4-fluorophenyl
butyl



1.4.598
3-bromo-4-fluorophenyl
methyl



1.4.599
3-methyl-4-fluorophenyl
methyl



1.4.600
3-methyl-4-fluorophenyl
ethyl



1.4.601
3-cyclopropyl-4-fluorophenyl
methyl



1.4.602
3-cyano-4-fluorophenyl
methyl



1.4.603
3-methoxy-4-fluorophenyl
methyl



1.4.604
3-ethoxy-4-fluorophenyl
methyl



1.4.605
3-trifluoromethoxy-4-fluorophenyl
methyl



1.4.606
3-nitro-4-fluorophenyl
methyl



1.4.607
3-fluoro-4-chlorophenyl
methyl



1.4.608
3,4-dichlorophenyl
methyl



1.4.609
3-bromo-4-chlorophenyl
methyl



1.4.610
3-methyl-4-chlorophenyl
methyl



1.4.611
3-cyclopropyl-4-chlorophenyl
methyl



1.4.612
3-cyano-4-chlorophenyl
methyl



1.4.613
3-trifluoromethyl-4-chlorophenyl
methyl



1.4.614
3-methoxy-4-chlorophenyl
methyl



1.4.615
3-ethoxy-4-chlorophenyl
methyl



1.4.616
3-trifluoromethoxy-4-chlorophenyl
methyl



1.4.617
3-nitro-4-chlorophenyl
methyl



1.4.618
3-fluoro-4-bromophenyl
methyl



1.4.619
3-chloro-4-bromophenyl
methyl



1.4.620
3,4-dibromophenyl
methyl



1.4.621
3-methyl-4-bromophenyl
methyl



1.4.622
3-cyclopropyl-4-bromophenyl
methyl



1.4.623
3-cyano-4-bromophenyl
methyl



1.4.624
3-trifluoromethyl-4-bromophenyl
methyl



1.4.625
3-methoxy-4-phenyl
methyl



1.4.626
3-ethoxy-4-bromophenyl
methyl



1.4.627
3-trifluoromethoxy-4-bromophenyl
methyl



1.4.628
3-nitro-4-bromophenyl
methyl



1.4.629
3-fluoro-4-iodophenyl
methyl



1.4.630
3-chloro-4-iodophenyl
methyl



1.4.631
3-bromo-4-iodophenyl
methyl



1.4.632
3-methyl-4-iodophenyl
methyl



1.4.633
3-cyclopropyl-4-iodophenyl
methyl



1.4.634
3-cyano-4-iodophenyl
methyl



1.4.635
3-trifluoromethyl-4-iodophenyl
methyl



1.4.636
3-methoxy-4-iodophenyl
methyl



1.4.637
3-ethoxy-4-iodophenyl
methyl



1.4.638
3-trifluoromethoxy-4-iodophenyl
methyl



1.4.639
3-nitro-4-iodophenyl
methyl



1.4.640
3-fluoro-4-methylphenyl
methyl



1.4.641
3-chloro-4-methylphenyl
methyl



1.4.642
3-bromo-4-methylphenyl
methyl



1.4.643
3,4-dimethylphenyl
methyl



1.4.644
3,4-dimethylphenyl
ethyl



1.4.645
3,4-dimethylphenyl
propyl



1.4.646
3,4-dimethylphenyl
butyl



1.4.647
3-cyclopropyl-4-methylphenyl
methyl



1.4.648
3-cyano-4-methylphenyl
methyl



1.4.649
3-trifluoromethyl-4-methylphenyl
methyl



1.4.650
3-methoxy-4-methylphenyl
methyl



1.4.651
3-ethoxy-4-methylphenyl
methyl



1.4.652
3-trifluoromethoxy-4-methylphenyl
methyl



1.4.653
3-nitro-4-methylphenyl
methyl



1.4.654
3-fluoro-4-ethylphenyl
methyl



1.4.655
3-chloro-4-ethylphenyl
methyl



1.4.656
3-bromo-4-ethylphenyl
methyl



1.4.657
3-methyl-4-ethylphenyl
methyl



1.4.658
3,4-diethylphenyl
methyl



1.4.659
3-cyclopropyl-4-ethylphenyl
methyl



1.4.660
3-cyano-4-ethylphenyl
methyl



1.4.661
3-trifluoromethyl-4-ethylphenyl
methyl



1.4.662
3-methoxy-4-ethylphenyl
methyl



1.4.663
3-ethoxy-4-ethylphenyl
methyl



1.4.664
3-trifluoromethoxy-4-ethylphenyl
methyl



1.4.665
3-nitro-4-ethylphenyl
methyl



1.4.666
3-fluoro-4-propylphenyl
methyl



1.4.667
3-chloro-4-propylphenyl
methyl



1.4.668
3-bromo-4-propylphenyl
methyl



1.4.669
3-methyl-4-propylphenyl
methyl



1.4.670
3-cyclopropyl-4-propylphenyl
methyl



1.4.671
3-cyano-4-propylphenyl
methyl



1.4.672
3-trifluoromethyl-4-propylphenyl
methyl



1.4.673
3-methoxy-4-propylphenyl
methyl



1.4.674
3-ethoxy-4-propylphenyl
methyl



1.4.675
3-trifluoromethoxy-4-propylphenyl
methyl



1.4.676
3-nitro-4-propylphenyl
methyl



1.4.677
3-fluoro-4-isopropylphenyl
methyl



1.4.678
3-chloro-4-isopropylphenyl
methyl



1.4.679
3-bromo-4-isopropylphenyl
methyl



1.4.680
3-methyl-4-isopropylphenyl
methyl



1.4.681
3-cyclopropyl-4-isopropylphenyl
methyl



1.4.682
3-cyano-4-isopropylphenyl
methyl



1.4.683
3-trifluoromethyl-4-isopropylphenyl
methyl



1.4.684
3-methoxy-4-isopropylphenyl
methyl



1.4.685
3-ethoxy-4-isopropylphenyl
methyl



1.4.686
3-trifluoromethoxy-4-isopropylphenyl
methyl



1.4.687
3-nitro-4-isopropylphenyl
methyl



1.4.688
3-fluoro-4-tert-butylphenyl
methyl



1.4.689
3-chloro-4-tert-butylphenyl
methyl



1.4.690
3-bromo-4-tert-butylphenyl
methyl



1.4.691
3-methyl-4-tert-butylphenyl
methyl



1.4.692
3-cyclopropyl-4-tert-butylphenyl
methyl



1.4.693
3-cyano-4-tert-butylphenyl
methyl



1.4.694
3-trifluoromethyl-4-tert-butylphenyl
methyl



1.4.695
3-trifluoromethyl-4-tert-butylphenyl
ethyl



1.4.696
3-trifluoromethyl-4-tert-butylphenyl
propyl



1.4.697
3-trifluoromethyl-4-tert-butylphenyl
butyl



1.4.698
3-methoxy-4-tert-butylphenyl
methyl



1.4.699
3-ethoxy-4-tert-butylphenyl
methyl



1.4.700
3-trifluoromethoxy-4-tert-butylphenyl
methyl



1.4.701
3-nitro-4-tert-butylphenyl
methyl



1.4.702
3-fluoro-4-cyclopropylphenyl
methyl



1.4.703
3-chloro-4-cyclopropylphenyl
methyl



1.4.704
3-bromo-4-cyclopropylphenyl
methyl



1.4.705
3-methyl-4-cyclopropylphenyl
methyl



1.4.706
3-trifluoromethyl-4-cyclopropylphenyl
methyl



1.4.707
3-methoxy-4-cyclopropylphenyl
methyl



1.4.708
3-ethoxy-4-cyclopropylphenyl
methyl



1.4.709
3-trifluoromethoxy-4-cyclopropylphenyl
methyl



1.4.710
3-fluoro-4-methoxycarbonylphenyl
methyl



1.4.711
3-chloro-4-methoxycarbonylphenyl
methyl



1.4.712
3-bromo-4-methoxycarbonylphenyl
methyl



1.4.713
3-methyl-4-methoxycarbonylphenyl
methyl



1.4.714
3-cyclopropyl-4-methoxycarbonylphenyl
methyl



1.4.715
3-cyano-4-methoxycarbonylphenyl
methyl



1.4.716
3-trifluoromethyl-4-methoxycarbonyl-
methyl




phenyl




1.4.717
3-methoxy-4-methoxycarbonylphenyl
methyl



1.4.718
3-ethoxy-4-methoxycarbonylphenyl
methyl



1.4.719
3-trifluoromethoxy-4-methoxycarbonyl-
methyl




phenyl




1.4.720
3-nitro-4-methoxycarbonylphenyl
methyl



1.4.721
3-fluoro-4-cyanophenyl
methyl



1.4.722
3-chloro-4-cyanophenyl
methyl



1.4.723
3-bromo-4-cyanophenyl
methyl



1.4.724
3-methyl-4-cyanophenyl
methyl



1.4.725
3-cyclopropyl-4-cyanophenyl
methyl



1.4.726
3,4-dicyanophenyl
methyl



1.4.727
3-trifluoromethyl-4-cyanophenyl
methyl



1.4.728
3-trifluoromethyl-4-cyanophenyl
ethyl



1.4.729
3-trifluoromethyl-4-cyanophenyl
propyl



1.4.730
3-trifluoromethyl-4-cyanophenyl
butyl



1.4.731
3-methoxy-4-cyanophenyl
methyl



1.4.732
3-ethoxy-4-cyanophenyl
methyl



1.4.733
3-trifluoromethoxy-4-cyanophenyl
methyl



1.4.734
3-nitro-4-cyanophenyl
methyl



1.4.735
3-fluoro-4-methoxyphenyl
methyl



1.4.736
3-chloro-4-methoxyphenyl
methyl



1.4.737
3-bromo-4-methoxyphenyl
methyl



1.4.738
3-methyl-4-methoxyphenyl
methyl



1.4.739
3-cyclopropyl-4-methoxyphenyl
methyl



1.4.740
3-cyano-4-methoxyphenyl
methyl



1.4.741
3-trifluoromethyl-4-methoxyphenyl
methyl



1.4.742
3,4-dimethoxyphenyl
methyl



1.4.743
3-ethoxy-4-methoxyphenyl
methyl



1.4.744
3-trifluoromethoxy-4-methoxyphenyl
methyl



1.4.745
3-nitro-4-methoxyphenyl
methyl



1.4.746
3-fluoro-4-ethoxyphenyl
methyl



1.4.747
3-chloro-4-ethoxyphenyl
methyl



1.4.748
3-chloro-4-ethoxyphenyl
ethyl



1.4.749
3-chloro-4-ethoxyphenyl
propyl



1.4.750
3-chloro-4-ethoxyphenyl
butyl



1.4.751
3-bromo-4-ethoxyphenyl
methyl



1.4.752
3-methyl-4-ethoxyphenyl
methyl



1.4.753
3-cyclopropyl-4-ethoxyphenyl
methyl



1.4.754
3-cyano-4-ethoxyphenyl
methyl



1.4.755
3-trifluoromethyl-4-ethoxyphenyl
methyl



1.4.756
3-methoxy-4-ethoxyphenyl
methyl



1.4.757
2,4-diethoxyphenyl
methyl



1.4.758
3-trifluoromethoxy-4-ethoxyphenyl
methyl



1.4.759
3-nitro-4-ethoxyphenyl
methyl



1.4.760
3-fluoro-4-isopropoxyphenyl
methyl



1.4.761
3-chloro-4-isopropoxyphenyl
methyl



1.4.762
3-bromo-4-isopropoxyphenyl
methyl



1.4.763
3-methyl-4-isopropoxyphenyl
methyl



1.4.764
3-cyclopropyl-4-isopropoxyphenyl
methyl



1.4.765
3-cyano-4-isopropoxyphenyl
methyl



1.4.766
3-trifluoromethyl-4-isopropoxyphenyl
methyl



1.4.767
3-methoxy-4-isopropoxyphenyl
methyl



1.4.768
3-ethoxy-4-isopropoxyphenyl
methyl



1.4.769
3-trifluoromethoxy-4-isopropoxyphenyl
methyl



1.4.770
3-nitro-4-isopropoxyphenyl
methyl



1.4.771
3-fluoro-4-trifluoromethoxyphenyl
methyl



1.4.772
3-chloro-4-trifluoromethoxyphenyl
methyl



1.4.773
3-bromo-4-trifluoromethoxyphenyl
methyl



1.4.774
3-methyl-4-trifluoromethoxyphenyl
methyl



1.4.775
3-cyclopropyl-4-trifluoromethoxyphenyl
methyl



1.4.776
3-cyano-4-trifluoromethoxyphenyl
methyl



1.4.777
3-trifluoromethyl-4-trifluoromethoxy-
methyl




phenyl




1.4.778
3-methoxy-4-trifluoromethoxyphenyl
methyl



1.4.779
3-ethoxy-4-trifluoromethoxyphenyl
methyl



1.4.780
3,4-bis(trifluoromethoxy)phenyl
methyl



1.4.781
3-nitro-4-trifluoromethoxyphenyl
methyl



1.4.782
3-fluoro-4-difluoromethoxyphenyl
methyl



1.4.783
3-chloro-4-difluoromethoxyphenyl
methyl



1.4.784
3-bromo-4-difluoromethoxyphenyl
methyl



1.4.785
3-methyl-4-difluoromethoxyphenyl
methyl



1.4.786
3-cyclopropyl-4-difluoromethoxyphenyl
methyl



1.4.787
3-cyano-4-difluoromethoxyphenyl
methyl



1.4.788
3-trifluoromethyl-4-difluoromethoxy-
methyl




phenyl




1.4.789
3-methoxy-4-difluoromethoxyphenyl
methyl



1.4.790
3-ethoxy-4-difluoromethoxyphenyl
methyl



1.4.791
3-nitro-4-difluoromethoxyphenyl
methyl



1.4.792
3-fluoro-4-nitrophenyl
methyl



1.4.793
3-chloro-4-nitrophenyl
methyl



1.4.794
3-bromo-4-nitrophenyl
methyl



1.4.795
3-methyl-4-nitrophenyl
methyl



1.4.796
3-cyclopropyl-4-nitrophenyl
methyl



1.4.797
3-cyano-4-nitrophenyl
methyl



1.4.798
3-trifluoromethyl-4-nitrophenyl
methyl



1.4.799
3-methoxy-4-nitrophenyl
methyl



1.4.800
3-ethoxy-4-nitrophenyl
methyl



1.4.801
3-trifluoromethoxy-4-nitrophenyl
methyl



1.4.802
3-fluoro-4-methylsulfanylphenyl
methyl



1.4.803
3-chloro-4-methylsulfanylphenyl
methyl



1.4.804
3-bromo-4-methylsulfanylphenyl
methyl



1.4.805
3-methyl-4-methylsulfanylphenyl
methyl



1.4.806
3-cyclopropyl-4-methylsulfanylphenyl
methyl



1.4.807
3-cyano-4-methylsulfanylphenyl
methyl



1.4.808
3-nitro-4-methylsulfanylphenyl
methyl



1.4.809
3,6-difluorophenyl
methyl



1.4.810
3,6-difluorophenyl
ethyl



1.4.811
3,6-difluorophenyl
propyl



1.4.812
3,6-difluorophenyl
butyl



1.4.813
3-chloro-6-fluorophenyl
methyl



1.4.814
3-bromo-6-fluorophenyl
methyl



1.4.815
3-methyl-6-fluorophenyl
methyl



1.4.816
3-cyclopropyl-6-fluorophenyl
methyl



1.4.817
3-cyano-6-fluorophenyl
methyl



1.4.818
3-methoxy-6-fluorophenyl
methyl



1.4.819
3-ethoxy-6-fluorophenyl
methyl



1.4.820
3-trifluoromethoxy-6-fluorophenyl
methyl



1.4.821
3-nitro-6-fluorophenyl
methyl



1.4.822
3-fluoro-6-chlorophenyl
methyl



1.4.823
3-fluoro-6-chlorophenyl
ethyl



1.4.824
3-fluoro-6-chlorophenyl
propyl



1.4.825
3-fluoro-6-chlorophenyl
butyl



1.4.826
3,6-dichlorophenyl
methyl



1.4.827
3,6-dichlorophenyl
ethyl



1.4.828
3,6-dichlorophenyl
propyl



1.4.829
3,6-dichlorophenyl
butyl



1.4.830
3-bromo-6-chlorophenyl
methyl



1.4.831
3-methyl-6-chlorophenyl
methyl



1.4.832
3-ethyl-6-chlorophenyl
methyl



1.4.833
3-cyclopropyl-6-chlorophenyl
methyl



1.4.834
3-cyano-6-chlorophenyl
methyl



1.4.835
3-trifluoromethyl-6-chlorophenyl
methyl



1.4.836
3-methoxy-6-chlorophenyl
methyl



1.4.837
3-ethoxy-6-chlorophenyl
methyl



1.4.838
3-trifluoromethoxy-6-chlorophenyl
methyl



1.4.839
3-nitro-6-chlorophenyl
methyl



1.4.840
3-fluoro-6-bromophenyl
methyl



1.4.841
3-chloro-6-bromophenyl
methyl



1.4.842
3,6-dibromophenyl
methyl



1.4.843
3-methyl-6-bromophenyl
methyl



1.4.844
3-cyclopropyl-6-bromophenyl
methyl



1.4.845
3-cyano-6-bromophenyl
methyl



1.4.846
3-trifluoromethyl-6-bromophenyl
methyl



1.4.847
3-methoxy-6-phenyl
methyl



1.4.848
3-ethoxy-6-bromophenyl
methyl



1.4.849
3-trifluoromethoxy-6-bromophenyl
methyl



1.4.850
3-nitro-6-bromophenyl
methyl



1.4.851
3-fluoro-6-iodophenyl
methyl



1.4.852
3-chloro-6-iodophenyl
methyl



1.4.853
3-bromo-6-iodophenyl
methyl



1.4.854
3-methyl-6-iodophenyl
methyl



1.4.855
3-cyclopropyl-6-iodophenyl
methyl



1.4.856
3-cyano-6-iodophenyl
methyl



1.4.857
3-trifluoromethyl-6-iodophenyl
methyl



1.4.858
3-methoxy-6-iodophenyl
methyl



1.4.859
3-ethoxy-6-iodophenyl
methyl



1.4.860
3-trifluoromethoxy-6-iodophenyl
methyl



1.4.861
3-nitro-6-iodophenyl
methyl



1.4.862
3-fluoro-6-methylphenyl
methyl



1.4.863
3-chloro-6-methylphenyl
methyl



1.4.864
3-bromo-6-methylphenyl
methyl



1.4.865
3,6-dimethylphenyl
methyl



1.4.866
3-cyclopropyl-6-methylphenyl
methyl



1.4.867
3-cyano-6-methylphenyl
methyl



1.4.868
3-trifluoromethyl-6-methylphenyl
methyl



1.4.869
3-methoxy-6-methylphenyl
methyl



1.4.870
3-ethoxy-6-methylphenyl
methyl



1.4.871
3-trifluoromethoxy-6-methylphenyl
methyl



1.4.872
3-nitro-6-methylphenyl
methyl



1.4.873
3-fluoro-6-ethylphenyl
methyl



1.4.874
3-chloro-6-ethylphenyl
methyl



1.4.875
3-bromo-6-ethylphenyl
methyl



1.4.876
3-methyl-6-ethylphenyl
methyl



1.4.877
3,6-diethylphenyl
methyl



1.4.878
3-cyclopropyl-6-ethylphenyl
methyl



1.4.879
3-cyano-6-ethylphenyl
methyl



1.4.880
3-trifluoromethyl-6-ethylphenyl
methyl



1.4.881
3-methoxy-6-ethylphenyl
methyl



1.4.882
3-ethoxy-6-ethylphenyl
methyl



1.4.883
3-trifluoromethoxy-6-ethylphenyl
methyl



1.4.884
3-nitro-6-ethylphenyl
methyl



1.4.885
3-fluoro-6-propylphenyl
methyl



1.4.886
3-chloro-6-propylphenyl
methyl



1.4.887
3-bromo-6-propylphenyl
methyl



1.4.888
3-methyl-6-propylphenyl
methyl



1.4.889
3-cyclopropyl-6-propylphenyl
methyl



1.4.890
3-cyano-6-propylphenyl
methyl



1.4.891
3-trifluoromethyl-6-propylphenyl
methyl



1.4.892
3-methoxy-6-propylphenyl
methyl



1.4.893
3-ethoxy-6-propylphenyl
methyl



1.4.894
3-trifluoromethoxy-6-propylphenyl
methyl



1.4.895
3-nitro-6-propylphenyl
methyl



1.4.896
3-fluoro-6-isopropylphenyl
methyl



1.4.897
3-chloro-6-isopropylphenyl
methyl



1.4.898
3-bromo-6-isopropylphenyl
methyl



1.4.899
3-methyl-6-isopropylphenyl
methyl



1.4.900
3-cyclopropyl-6-isopropylphenyl
methyl



1.4.901
3-cyano-6-isopropylphenyl
methyl



1.4.902
3-trifluoromethyl-6-isopropylphenyl
methyl



1.4.903
3-ethoxy-6-isopropylphenyl
methyl



1.4.904
3-trifluoromethoxy-6-isopropylphenyl
methyl



1.4.905
3-nitro-6-isopropylphenyl
methyl



1.4.906
3-fluoro-6-tert-butylphenyl
methyl



1.4.907
3-chloro-6-tert-butylphenyl
methyl



1.4.908
3-bromo-6-tert-butylphenyl
methyl



1.4.909
3-methyl-6-tert-butylphenyl
methyl



1.4.910
3-cyclopropyl-6-tert-butylphenyl
methyl



1.4.911
3-cyano-6-tert-butylphenyl
methyl



1.4.912
3-trifluoromethyl-6-tert-butylphenyl
methyl



1.4.913
3-methoxy-6-tert-butylphenyl
methyl



1.4.914
3-ethoxy-6-tert-butylphenyl
methyl



1.4.915
3-trifluoromethoxy-6-tert-butylphenyl
methyl



1.4.916
3-nitro-6-tert-butylphenyl
methyl



1.4.917
3-fluoro-6-cyclopropylphenyl
methyl



1.4.918
3-chloro-6-cyclopropylphenyl
methyl



1.4.919
3-bromo-6-cyclopropylphenyl
methyl



1.4.920
3-methyl-6-cyclopropylphenyl
methyl



1.4.921
3-cyano-6-cyclopropylphenyl
methyl



1.4.922
3-trifluoromethyl-6-cyclopropylphenyl
methyl



1.4.923
3-methoxy-6-cyclopropylphenyl
methyl



1.4.924
3-ethoxy-6-cyclopropylphenyl
methyl



1.4.925
3-trifluoromethoxy-6-cyclopropylphenyl
methyl



1.4.926
3-fluoro-6-methoxycarbonylphenyl
methyl



1.4.927
3-chloro-6-methoxycarbonylphenyl
methyl



1.4.928
3-bromo-6-methoxycarbonylphenyl
methyl



1.4.929
3-methyl-6-methoxycarbonylphenyl
methyl



1.4.930
3-cyclopropyl-6-methoxycarbonylphenyl
methyl



1.4.931
3-cyano-6-methoxycarbonylphenyl
methyl



1.4.932
3-trifluoromethyl-6-methoxycarbonyl-
methyl




phenyl




1.4.933
3-methoxy-6-methoxycarbonylphenyl
methyl



1.4.934
3-ethoxy-6-methoxycarbonylphenyl
methyl



1.4.935
3-trifluoromethoxy-6-methoxycarbonyl-
methyl




phenyl




1.4.936
3-nitro-6-methoxycarbonylphenyl
methyl



1.4.937
3-fluoro-6-cyanophenyl
methyl



1.4.938
3-chloro-6-cyanophenyl
methyl



1.4.939
3-bromo-6-cyanophenyl
methyl



1.4.940
3-methyl-6-cyanophenyl
methyl



1.4.941
3-cyclopropyl-6-cyanophenyl
methyl



1.4.942
3-cyano-6-cyanophenyl
methyl



1.4.943
3-trifluoromethyl-6-cyanophenyl
methyl



1.4.944
3-methoxy-6-cyanophenyl
methyl



1.4.945
3-ethoxy-6-cyanophenyl
methyl



1.4.946
3-trifluoromethoxy-6-cyanophenyl
methyl



1.4.947
3-nitro-6-cyanophenyl
methyl



1.4.948
3-fluoro-6-methoxyphenyl
methyl



1.4.949
3-chloro-6-methoxyphenyl
methyl



1.4.950
3-bromo-6-methoxyphenyl
methyl



1.4.951
3-methyl-6-methoxyphenyl
methyl



1.4.952
3-cyclopropyl-6-methoxyphenyl
methyl



1.4.953
3-cyano-6-methoxyphenyl
methyl



1.4.954
3-trifluoromethyl-6-methoxyphenyl
methyl



1.4.955
3,6-dimethoxyphenyl
methyl



1.4.956
3-ethoxy-6-methoxyphenyl
methyl



1.4.957
3-trifluoromethoxy-6-methoxyphenyl
methyl



1.4.958
3-nitro-6-methoxyphenyl
methyl



1.4.959
3-fluoro-6-ethoxyphenyl
methyl



1.4.960
3-chloro-6-ethoxyphenyl
methyl



1.4.961
3-bromo-6-ethoxyphenyl
methyl



1.4.962
3-methyl-6-ethoxyphenyl
methyl



1.4.963
3-cyclopropyl-6-ethoxyphenyl
methyl



1.4.964
3-cyano-6-ethoxyphenyl
methyl



1.4.965
3-trifluoromethyl-6-ethoxyphenyl
methyl



1.4.966
3-methoxy-6-ethoxyphenyl
methyl



1.4.967
2,6-diethoxyphenyl
methyl



1.4.968
3-trifluoromethoxy-6-ethoxyphenyl
methyl



1.4.969
3-nitro-6-ethoxyphenyl
methyl



1.4.970
3-fluoro-6-isopropoxyphenyl
methyl



1.4.971
3-chloro-6-isopropoxyphenyl
methyl



1.4.972
3-bromo-6-isopropoxyphenyl
methyl



1.4.973
3-methyl-6-isopropoxyphenyl
methyl



1.4.974
3-cyclopropyl-6-isopropoxyphenyl
methyl



1.4.975
3-cyano-6-isopropoxyphenyl
methyl



1.4.976
3-trifluoromethyl-6-isopropoxyphenyl
methyl



1.4.977
3-methoxy-6-isopropoxyphenyl
methyl



1.4.978
3-ethoxy-6-isopropoxyphenyl
methyl



1.4.979
3-trifluoromethoxy-6-isopropoxyphenyl
methyl



1.4.980
3-nitro-6-isopropoxyphenyl
methyl



1.4.981
3-fluoro-6-trifluoromethoxyphenyl
methyl



1.4.982
3-chloro-6-trifluoromethoxyphenyl
methyl



1.4.983
3-bromo-6-trifluoromethoxyphenyl
methyl



1.4.984
3-methyl-6-trifluoromethoxyphenyl
methyl



1.4.985
3-cyclopropyl-6-trifluoromethoxyphenyl
methyl



1.4.986
3-cyano-6-trifluoromethoxyphenyl
methyl



1.4.987
3-trifluoromethyl-6-trifluoromethoxy-
methyl




phenyl




1.4.988
3-methoxy-6-trifluoromethoxyphenyl
methyl



1.4.989
3-ethoxy-6-trifluoromethoxyphenyl
methyl



1.4.990
3,6-bis(trifluoromethoxy)phenyl
methyl



1.4.991
3-nitro-6-trifluoromethoxyphenyl
methyl



1.4.992
3-fluoro-6-difluoromethoxyphenyl
methyl



1.4.993
3-chloro-6-difluoromethoxyphenyl
methyl



1.4.994
3-bromo-6-difluoromethoxyphenyl
methyl



1.4.995
3-methyl-6-difluoromethoxyphenyl
methyl



1.4.996
3-cyclopropyl-6-difluoromethoxyphenyl
methyl



1.4.997
3-cyano-6-difluoromethoxyphenyl
methyl



1.4.998
3-trifluoromethyl-6-difluoromethoxy-
methyl




phenyl




1.4.999
3-methoxy-6-difluoromethoxyphenyl
methyl



1.4.1000
3-ethoxy-6-difluoromethoxyphenyl
methyl



1.4.1001
3-trifluoromethoxy-6-difluoromethoxy-
methyl




phenyl




1.4.1002
3-nitro-6-difluoromethoxyphenyl
methyl



1.4.1003
3-fluoro-6-nitrophenyl
methyl



1.4.1004
3-chloro-6-nitrophenyl
methyl



1.4.1005
3-bromo-6-nitrophenyl
methyl



1.4.1006
3-methyl-6-nitrophenyl
methyl



1.4.1007
3-cyclopropyl-6-nitrophenyl
methyl



1.4.1008
3-trifluoromethyl-6-nitrophenyl
methyl



1.4.1009
3-methoxy-6-nitrophenyl
methyl



1.4.1010
3-ethoxy-6-nitrophenyl
methyl



1.4.1011
3-trifluoromethoxy-6-nitrophenyl
methyl



1.4.1012
3-fluoro-6-methylsulfanylphenyl
methyl



1.4.1013
3-chloro-6-methylsulfanylphenyl
methyl



1.4.1014
3-bromo-6-methylsulfanylphenyl
methyl



1.4.1015
3-methyl-6-methylsulfanylphenyl
methyl



1.4.1016
3-cyclopropyl-6-methylsulfanylphenyl
methyl



1.4.1017
3-cyano-6-methylsulfanylphenyl
methyl



1.4.1018
3-trifluoromethyl-6-methylsulfanylphenyl
methyl



1.4.1019
2,3,4-trifluorophenyl
methyl



1.4.1020
2,3,4-trichlorophenyl
methyl



1.4.1021
2,3,4-trimethylphenyl
methyl



1.4.1022
2-fluoro-2-chloro-5-trifluoromethylphenyl
methyl



1.4.1023
2,3,5-trifluorophenyl
methyl



1.4.1024
2,3,5-trichlorophenyl
methyl



1.4.1025
2,3,5-trimethylphenyl
methyl



1.4.1026
2,3-dichloro-5-methoxyphenyl
methyl



1.4.1027
2,3,6-trifluorophenyl
methyl



1.4.1028
2,3,6-trichlorophenyl
methyl



1.4.1029
2,3,6-trimethylphenyl
methyl



1.4.1030
3,4,5-trifluorophenyl
methyl



1.4.1031
3,4,5-trichlorophenyl
methyl



1.4.1032
3,4,5-trimethylphenyl
methyl



1.4.1033
3,5-dimethyl-4-fluorophenyl
methyl



1.4.1034
3,5-dichloro-4-methoxyphenyl
methyl



1.4.1035
3,5-difluoro-4-chlorophenyl
methyl



1.4.1036
3,5-dichloro-4-hydroxyphenyl
methyl



1.4.1037
3,5-trifluoromethyl-4-chlorophenyl
methyl



1.4.1038
3,4,6-trifluorophenyl
methyl



1.4.1039
3,4,6-trichlorophenyl
methyl



1.4.1040
3,4,6-trimethylphenyl
methyl



1.4.1041
pentafluorophenyl
methyl
















TABLE 1.5







Inventive compounds of the general formula (I) in which W* is COOH, R1


and R2 are each hydrogen, and aryl is the radical.








 








 










No.
Aryl
R3
Physical data





1.5.1
3-fluorophenyl
hydroxymethyl



1.5.2
3-fluorophenyl
1-hydroxyethyl



1.5.3
3-fluorophenyl
1-hydroxypropyl



1.5.4
3-fluorophenyl
(1-hydroxy-2-





methylpropyl)



1.5.5
3-fluorophenyl
methoxymethyl



1.5.6
3-fluorophenyl
2-methoxyethyl



1.5.7
3-chlorophenyl
hydroxymethyl



1.5.8
3-chlorophenyl
1-hydroxyethyl



1.5.9
3-chlorophenyl
1-hydroxypropyl



1.5.10
3-chlorophenyl
(1-hydroxy-2-





methylpropyl)



1.5.11
3-chlorophenyl
methoxymethyl



1.5.12
3-chlorophenyl
2-methoxyethyl



1.5.13
3-bromophenyl
hydroxymethyl



1.5.14
3-bromophenyl
1-hydroxyethyl



1.5.15
3-iodophenyl
hydroxymethyl



1.5.16
3-iodophenyl
1-hydroxyethyl



1.5.17
3-methylphenyl
hydroxymethyl



1.5.18
3-methylphenyl
1-hydroxyethyl



1.5.19
3-ethylphenyl
hydroxymethyl



1.5.20
3-propylphenyl
hydroxymethyl



1.5.21
3-isopropylphenyl
hydroxymethyl



1.5.22
3-n-butylphenyl
hydroxymethyl



1.5.23
3-i-butylphenyl
hydroxymethyl



1.5.24
3-tert-butylphenyl
hydroxymethyl



1.5.25
3-cyclopropylphenyl
hydroxymethyl



1.5.26
3-cyclobutylphenyl
hydroxymethyl



1.5.27
3-cyclopentylphenyl
hydroxymethyl



1.5.28
3-vinylphenyl
hydroxymethyl



1.5.29
3-ethynylphenyl
hydroxymethyl



1.5.30
3-cyanophenyl
hydroxymethyl



1.5.31
3-trifluoromethylphenyl
hydroxymethyl



1.5.32
3-difluoromethylphenyl
hydroxymethyl



1.5.33
3-(hydroxycarbonyl)phenyl
hydroxymethyl



1.5.34
3-(methoxycarbonyl)phenyl
hydroxymethyl



1.5.35
3-(ethoxycarbonyl)phenyl
hydroxymethyl



1.5.36
3-hydroxymethylphenyl
hydroxymethyl



1.5.37
3-carbamoylphenyl
hydroxymethyl



1.5.38
3-hydroxyphenyl
hydroxymethyl



1.5.39
3-methoxyphenyl
hydroxymethyl



1.5.40
3-ethoxyphenyl
hydroxymethyl



1.5.41
3-propyloxyphenyl
hydroxymethyl



1.5.42
3-isopropyloxyphenyl
hydroxymethyl



1.5.43
3-n-butyloxyphenyl
hydroxymethyl



1.5.44
3-i-butyloxyphenyl
hydroxymethyl



1.5.45
3-t-butyloxyphenyl
hydroxymethyl



1.5.46
3-difluoromethoxyphenyl
hydroxymethyl



1.5.47
3-trifluoromethoxyphenyl
hydroxymethyl



1.5.48
3-(2,2,2-trifluoroethoxy)phenyl
hydroxymethyl



1.5.49
3-(2-chloroethoxy)phenyl
hydroxymethyl



1.5.50
3-(2-hydroxyethoxy)phenyl
hydroxymethyl



1.5.51
3-(2-methoxyethoxy)phenyl
hydroxymethyl



1.5.52
3-[(tert-butoxycarbonyl)oxy]phenyl
hydroxymethyl



1.5.53
3-nitrophenyl
hydroxymethyl



1.5.54
3-acetoxyphenyl
hydroxymethyl



1.5.55
(3-[(tert-butoxycarbonyl)amino]phenyl)
hydroxymethyl



1.5.56
3-methylsulfanylphenyl
hydroxymethyl



1.5.57
3-ethylsulfanylphenyl
hydroxymethyl



1.5.58
3-(pentafluoro-lambda6-sulfanyl)phenyl
hydroxymethyl



1.5.59
2,3-difluorophenyl
hydroxymethyl



1.5.60
2,3-difluorophenyl
1-hydroxyethyl



1.5.61
2,3-difluorophenyl
1-hydroxypropyl



1.5.62
2,3-difluorophenyl
(1-hydroxy-2-





methylpropyl)



1.5.63
2,3-difluorophenyl
methoxymethyl



1.5.64
2,3-difluorophenyl
2-methoxyethyl



1.5.65
2-chloro-3-fluorophenyl
hydroxymethyl



1.5.66
2-bromo-3-fluorophenyl
hydroxymethyl



1.5.67
2-methyl-3-fluorophenyl
hydroxymethyl



1.5.68
2-ethyl-3-fluorophenyl
hydroxymethyl



1.5.69
2-cyclopropyl-3-fluorophenyl
hydroxymethyl



1.5.70
2-vinyl-3-fluorophenyl
hydroxymethyl



1.5.71
2-ethynyl-3-fluorophenyl
hydroxymethyl



1.5.72
2-cyano-3-fluorophenyl
hydroxymethyl



1.5.73
2-methoxy-3-fluorophenyl
hydroxymethyl



1.5.74
2-ethoxy-3-fluorophenyl
hydroxymethyl



1.5.75
2-trifluoromethoxy-3-fluorophenyl
hydroxymethyl



1.5.76
2-nitro-3-fluorophenyl
hydroxymethyl



1.5.77
2-fluoro-3-chlorophenyl
hydroxymethyl



1.5.78
2,3-dichlorophenyl
hydroxymethyl



1.5.79
2,3-dichlorophenyl
1-hydroxyethyl



1.5.80
2,3-dichlorophenyl
1-hydroxypropyl



1.5.81
2,3-dichlorophenyl
(1-hydroxy-2-





methylpropyl)



1.5.82
2,3-dichlorophenyl
methoxymethyl



1.5.83
2,3-dichlorophenyl
2-methoxyethyl



1.5.84
2-bromo-3-chlorophenyl
hydroxymethyl



1.5.85
2-methyl-3-chlorophenyl
hydroxymethyl



1.5.86
2-ethyl-3-chlorophenyl
hydroxymethyl



1.5.87
2-cyclopropyl-3-chlorophenyl
hydroxymethyl



1.5.88
2-vinyl-3-chlorophenyl
hydroxymethyl



1.5.89
2-ethynyl-3-chlorophenyl
hydroxymethyl



1.5.90
2-cyano-3-chlorophenyl
hydroxymethyl



1.5.91
2-trifluoromethyl-2-chlorophenyl
hydroxymethyl



1.5.92
2-methoxy-3-chlorophenyl
hydroxymethyl



1.5.93
2-ethoxy-3-chlorophenyl
hydroxymethyl



1.5.94
2-trifluoromethoxy-3-chlorophenyl
hydroxymethyl



1.5.95
2-nitro-3-chlorophenyl
hydroxymethyl



1.5.96
2-fluoro-3-bromophenyl
hydroxymethyl



1.5.97
2-chloro-3-bromophenyl
hydroxymethyl



1.5.98
2,3-dibromophenyl
hydroxymethyl



1.5.99
2-methyl-3-bromophenyl
hydroxymethyl



1.5.100
2-ethyl-3-bromophenyl
hydroxymethyl



1.5.101
2-cyclopropyl-3-bromophenyl
hydroxymethyl



1.5.102
2-vinyl-3-bromophenyl
hydroxymethyl



1.5.103
2-ethynyl-3-bromophenyl
hydroxymethyl



1.5.104
2-cyano-3-bromophenyl
hydroxymethyl



1.5.105
2-trifluoromethyl-3-bromophenyl
hydroxymethyl



1.5.106
2-methoxy-3-phenyl
hydroxymethyl



1.5.107
2-ethoxy-3-bromophenyl
hydroxymethyl



1.5.108
2-trifluoromethoxy-3-bromophenyl
hydroxymethyl



1.5.109
2-nitro-3-bromophenyl
hydroxymethyl



1.5.110
2-fluoro-3-iodophenyl
hydroxymethyl



1.5.111
2-chloro-3-iodophenyl
hydroxymethyl



1.5.112
2-bromo-3-iodophenyl
hydroxymethyl



1.5.113
2-methyl-3-iodophenyl
hydroxymethyl



1.5.114
2-ethyl-3-iodophenyl
hydroxymethyl



1.5.115
2-cyclopropyl-3-iodophenyl
hydroxymethyl



1.5.116
2-vinyl-3-iodophenyl
hydroxymethyl



1.5.117
2-ethynyl-3-iodophenyl
hydroxymethyl



1.5.118
2-cyano-3-iodophenyl
hydroxymethyl



1.5.119
2-trifluoromethyl-3-iodophenyl
hydroxymethyl



1.5.120
2-methoxy-3-iodophenyl
hydroxymethyl



1.5.121
2-ethoxy-3-iodophenyl
hydroxymethyl



1.5.122
2-trifluoromethoxy-3-iodophenyl
hydroxymethyl



1.5.123
2-nitro-3-iodophenyl
hydroxymethyl



1.5.124
2-fluoro-3-methylphenyl
hydroxymethyl



1.5.125
2-fluoro-3-methylphenyl
1-hydroxyethyl



1.5.126
2-fluoro-3-methylphenyl
1-hydroxypropyl



1.5.127
2-fluoro-3-methylphenyl
(1-hydroxy-2-





methylpropyl)



1.5.128
2-fluoro-3-methylphenyl
methoxymethyl



1.5.129
2-fluoro-3-methylphenyl
2-methoxyethyl



1.5.130
2-chloro-3-methylphenyl
hydroxymethyl



1.5.131
2-chloro-3-methylphenyl
1-hydroxyethyl



1.5.132
2-chloro-3-methylphenyl
1-hydroxypropyl



1.5.133
2-chloro-3-methylphenyl
(1-hydroxy-2-





methylpropyl)



1.5.134
2-chloro-3-methylphenyl
methoxymethyl



1.5.135
2-chloro-3-methylphenyl
2-methoxyethyl



1.5.136
2-bromo-3-methylphenyl
hydroxymethyl



1.5.137
2,3-dimethylphenyl
hydroxymethyl



1.5.138
2,3-dimethylphenyl
1-hydroxyethyl



1.5.139
2,3-dimethylphenyl
1-hydroxypropyl



1.5.140
2,3-dimethylphenyl
(1-hydroxy-2-





methylpropyl)



1.5.141
2,3-dimethylphenyl
methoxymethyl



1.5.142
2,3-dimethylphenyl
2-methoxyethyl



1.5.143
2-ethyl-3-methylphenyl
hydroxymethyl



1.5.144
2-cyclopropyl-3-methylphenyl
hydroxymethyl



1.5.145
2-vinyl-3-methylphenyl
hydroxymethyl



1.5.146
2-ethynyl-3-methylphenyl
hydroxymethyl



1.5.147
2-cyano-3-methylphenyl
hydroxymethyl



1.5.148
2-trifluoromethyl-3-methylphenyl
hydroxymethyl



1.5.149
2-methoxy-3-methylphenyl
hydroxymethyl



1.5.150
2-ethoxy-3-methylphenyl
hydroxymethyl



1.5.151
2-trifluoromethoxy-3-methylphenyl
hydroxymethyl



1.5.152
2-nitro-3-methylphenyl
hydroxymethyl



1.5.153
2-fluoro-3-ethylphenyl
hydroxymethyl



1.5.154
2-chloro-3-ethylphenyl
hydroxymethyl



1.5.155
2-bromo-3-ethylphenyl
hydroxymethyl



1.5.156
2-methyl-3-ethylphenyl
hydroxymethyl



1.5.157
2,3-diethylphenyl
hydroxymethyl



1.5.158
2-cyclopropyl-3-ethylphenyl
hydroxymethyl



1.5.159
2-vinyl-3-ethylphenyl
hydroxymethyl



1.5.160
2-ethynyl-3-ethylphenyl
hydroxymethyl



1.5.161
2-cyano-3-ethylphenyl
hydroxymethyl



1.5.162
2-trifluoromethyl-3-ethylphenyl
hydroxymethyl



1.5.163
2-methoxy-3-ethylphenyl
hydroxymethyl



1.5.164
2-ethoxy-3-ethylphenyl
hydroxymethyl



1.5.165
2-trifluoromethoxy-3-ethylphenyl
hydroxymethyl



1.5.166
2-nitro-3-ethylphenyl
hydroxymethyl



1.5.167
2-fluoro-3-propylphenyl
hydroxymethyl



1.5.168
2-chloro-3-propylphenyl
hydroxymethyl



1.5.169
2-bromo-3-propylphenyl
hydroxymethyl



1.5.170
2-methyl-3-propylphenyl
hydroxymethyl



1.5.171
2-methyl-3-propylphenyl
hydroxymethyl



1.5.172
2-cyclopropyl-3-propylphenyl
hydroxymethyl



1.5.173
2-vinyl-3-propylphenyl
hydroxymethyl



1.5.174
2-ethynyl-3propylphenyl
hydroxymethyl



1.5.175
2-cyano-3-propylphenyl
hydroxymethyl



1.5.176
2-trifluoromethyl-3-propylphenyl
hydroxymethyl



1.5.177
2-methoxy-3-propylphenyl
hydroxymethyl



1.5.178
2-ethoxy-3-propylphenyl
hydroxymethyl



1.5.179
2-trifluoromethoxy-3-propylphenyl
hydroxymethyl



1.5.180
2-nitro-3-propylphenyl
hydroxymethyl



1.5.181
2-fluoro-3-isopropylphenyl
hydroxymethyl



1.5.182
2-chloro-3-isopropylphenyl
hydroxymethyl



1.5.183
2-bromo-3-isopropylphenyl
hydroxymethyl



1.5.184
2-methyl-3-isopropylphenyl
hydroxymethyl



1.5.185
2-ethyl-3-isopropylphenyl
hydroxymethyl



1.5.186
2-cyclopropyl-3-isopropylphenyl
hydroxymethyl



1.5.187
2-vinyl-3-isopropylphenyl
hydroxymethyl



1.5.188
2-ethynyl-3-isopropylphenyl
hydroxymethyl



1.5.189
2-cyano-3-isopropylphenyl
hydroxymethyl



1.5.190
2-trifluoromethyl-3-isopropylphenyl
hydroxymethyl



1.5.191
2-methoxy-3-isopropylphenyl
hydroxymethyl



1.5.192
2-ethoxy-3-isopropylphenyl
hydroxymethyl



1.5.193
2-trifluoromethoxy-3-isopropylphenyl
hydroxymethyl



1.5.194
2-nitro-3-isopropylphenyl
hydroxymethyl



1.5.195
2-fluoro-3-tert-butylphenyl
hydroxymethyl



1.5.196
2-chloro-3-tert-butylphenyl
hydroxymethyl



1.5.197
2-bromo-3-tert-butylphenyl
hydroxymethyl



1.5.198
2-methyl-3-tert-butylphenyl
hydroxymethyl



1.5.199
2-ethyl-3-tert-butylphenyl
hydroxymethyl



1.5.200
2-cyclopropyl-3-tert-butylphenyl
hydroxymethyl



1.5.201
2-vinyl-3-tert-butylphenyl
hydroxymethyl



1.5.202
2-ethynyl-3-tert-butylphenyl
hydroxymethyl



1.5.203
2-cyano-3-tert-butylphenyl
hydroxymethyl



1.5.204
2-trifluoromethyl-3-tert-butylphenyl
hydroxymethyl



1.5.205
2-methoxy-3-tert-butylphenyl
hydroxymethyl



1.5.206
2-ethoxy-3-tert-butylphenyl
hydroxymethyl



1.5.207
2-trifluoromethoxy-3-tert-butylphenyl
hydroxymethyl



1.5.208
2-nitro-3-tert-butylphenyl
hydroxymethyl



1.5.209
2-fluoro-3-hydroxymethylphenyl
hydroxymethyl



1.5.210
2-chloro-3-hydroxymethylphenyl
hydroxymethyl



1.5.211
2-bromo-3-hydroxymethylphenyl
hydroxymethyl



1.5.212
2-methyl-3-hydroxymethylphenyl
hydroxymethyl



1.5.213
2-ethyl-3-hydroxymethylphenyl
hydroxymethyl



1.5.214
2-cyclopropyl-3-hydroxymethylphenyl
hydroxymethyl



1.5.215
2-vinyl-3-hydroxymethylphenyl
hydroxymethyl



1.5.216
2-ethynyl-3-hydroxymethylphenyl
hydroxymethyl



1.5.217
2-cyano-3-hydroxymethylphenyl
hydroxymethyl



1.5.218
2-trifluoromethyl-3-hydroxymethylphenyl
hydroxymethyl



1.5.219
2-methoxy-3-hydroxymethylphenyl
hydroxymethyl



1.5.220
2-ethoxy-3-hydroxymethylphenyl
hydroxymethyl



1.5.221
2-trifluoromethoxy-3-
hydroxymethyl




hydroxymethylphenyl




1.5.222
2-nitro-3-hydroxymethylphenyl
hydroxymethyl



1.5.223
2-fluoro-3-cyclopropylphenyl
hydroxymethyl



1.5.224
2-chloro-3-cyclopropylphenyl
hydroxymethyl



1.5.225
2-bromo-3-cyclopropylphenyl
hydroxymethyl



1.5.226
2-methyl-3-cyclopropylphenyl
hydroxymethyl



1.5.227
2-ethyl-3-cyclopropylphenyl
hydroxymethyl



1.5.228
2-cyclopropyl-3-cyclopropylphenyl
hydroxymethyl



1.5.229
2-vinyl-3-cyclopropylphenyl
hydroxymethyl



1.5.230
2-ethynyl-3-cyclopropylphenyl
hydroxymethyl



1.5.231
2-cyano-3-cyclopropylphenyl
hydroxymethyl



1.5.232
2-trifluoromethyl-3-cyclopropylphenyl
hydroxymethyl



1.5.233
2-methoxy-3-cyclopropylphenyl
hydroxymethyl



1.5.234
2-ethoxy-3-cyclopropylphenyl
hydroxymethyl



1.5.235
2-trifluoromethoxy-3-cyclopropylphenyl
hydroxymethyl



1.5.236
2-fluoro-3-methoxycarbonylphenyl
hydroxymethyl



1.5.237
2-chloro-3-methoxycarbonylphenyl
hydroxymethyl



1.5.238
2-bromo-3-methoxycarbonylphenyl
hydroxymethyl



1.5.239
2-methyl-3-methoxycarbonylphenyl
hydroxymethyl



1.5.240
2-ethyl-3-methoxycarbonylphenyl
hydroxymethyl



1.5.241
2-cyclopropyl-3-methoxycarbonylphenyl
hydroxymethyl



1.5.242
2-vinyl-3-methoxycarbonylphenyl
hydroxymethyl



1.5.243
2-ethynyl-3-methoxycarbonylphenyl
hydroxymethyl



1.5.244
2-cyano-3-methoxycarbonylphenyl
hydroxymethyl



1.5.245
2-trifluoromethyl-3-
hydroxymethyl




methoxycarbonylphenyl




1.5.246
2-methoxy-3-methoxycarbonylphenyl
hydroxymethyl



1.5.247
2-ethoxy-3-methoxycarbonylphenyl
hydroxymethyl



1.5.248
2-trifluoromethoxy-3-
hydroxymethyl




methoxycarbonylphenyl




1.5.249
2-nitro-3-methoxycarbonylphenyl
hydroxymethyl



1.5.250
2-fluoro-3-vinylphenyl
hydroxymethyl



1.5.251
2-chloro-3-vinylphenyl
hydroxymethyl



1.5.252
2-bromo-3-vinylphenyl
hydroxymethyl



1.5.253
2-methyl-3-vinylphenyl
hydroxymethyl



1.5.254
2-ethyl-3-vinylphenyl
hydroxymethyl



1.5.255
2-cyclopropyl-3-vinylphenyl
hydroxymethyl



1.5.256
2-vinyl-3-vinylphenyl
hydroxymethyl



1.5.257
2-ethynyl-3-vinylphenyl
hydroxymethyl



1.5.258
2-cyano-3-vinylphenyl
hydroxymethyl



1.5.259
2-trifluoromethyl-3-vinylphenyl
hydroxymethyl



1.5.260
2-methoxy-3-vinylphenyl
hydroxymethyl



1.5.261
2-ethoxy-3-vinylphenyl
hydroxymethyl



1.5.262
2-trifluoromethoxy-3-vinylphenyl
hydroxymethyl



1.5.263
2-nitro-3-vinylphenyl
hydroxymethyl



1.5.264
2-fluoro-3-ethynylphenyl
hydroxymethyl



1.5.265
2-chloro-3-ethynylphenyl
hydroxymethyl



1.5.266
2-bromo-3-ethynylphenyl
hydroxymethyl



1.5.267
2-methyl-3-ethynylphenyl
hydroxymethyl



1.5.268
2-ethyl-3-ethynylphenyl
hydroxymethyl



1.5.269
2-cyclopropyl-3-ethynylphenyl
hydroxymethyl



1.5.270
2-vinyl-3-ethynylphenyl
hydroxymethyl



1.5.271
2-cyano-3-ethynylphenyl
hydroxymethyl



1.5.272
2-trifluoromethyl-3-ethynylphenyl
hydroxymethyl



1.5.273
2-methoxy-3-ethynylphenyl
hydroxymethyl



1.5.274
2-ethoxy-3-ethynylphenyl
hydroxymethyl



1.5.275
2-trifluoromethoxy-3-ethynylphenyl
hydroxymethyl



1.5.276
2-nitro-3-ethynylphenyl
hydroxymethyl



1.5.277
2-fluoro-3-ethynylphenyl
hydroxymethyl



1.5.278
2-fluoro-3-cyanophenyl
hydroxymethyl



1.5.279
2-chloro-3-cyanophenyl
hydroxymethyl



1.5.280
2-bromo-3-cyanophenyl
hydroxymethyl



1.5.281
2-methyl-3-cyanophenyl
hydroxymethyl



1.5.282
2-ethyl-3-cyanophenyl
hydroxymethyl



1.5.283
2-ethyl-3-cyanophenyl
1-hydroxyethyl



1.5.284
2-ethyl-3-cyanophenyl
1-hydroxypropyl



1.5.285
2-ethyl-3-cyanophenyl
(1-hydroxy-2-





methylpropyl)



1.5.286
2-ethyl-3-cyanophenyl
methoxymethyl



1.5.287
2-ethyl-3-cyanophenyl
2-methoxyethyl



1.5.288
2-cyclopropyl-3-cyanophenyl
hydroxymethyl



1.5.289
2-vinyl-3-cyanophenyl
hydroxymethyl



1.5.290
2-ethynyl-3-cyanophenyl
hydroxymethyl



1.5.291
2-cyano-3-cyanophenyl
hydroxymethyl



1.5.292
2-trifluoromethyl-3-cyanophenyl
hydroxymethyl



1.5.293
2-methoxy-3-cyanophenyl
hydroxymethyl



1.5.294
2-ethoxy-3-cyanophenyl
hydroxymethyl



1.5.295
2-trifluoromethoxy-3-cyanophenyl
hydroxymethyl



1.5.296
2-nitro-3-cyanophenyl
hydroxymethyl



1.5.297
2-fluoro-3-hydroxyphenyl
hydroxymethyl



1.5.298
2-chloro-3-hydroxyphenyl
hydroxymethyl



1.5.299
2-bromo-3-hydroxyphenyl
hydroxymethyl



1.5.300
2-methyl-3-hydroxyphenyl
hydroxymethyl



1.5.301
2-ethyl-3-hydroxyphenyl
hydroxymethyl



1.5.302
2-cyclopropyl-3-hydroxyphenyl
hydroxymethyl



1.5.303
2-vinyl-3-hydroxyphenyl
hydroxymethyl



1.5.304
2-ethynyl-3-hydroxyphenyl
hydroxymethyl



1.5.305
2-cyano-3-hydroxyphenyl
hydroxymethyl



1.5.306
2-trifluoromethyl-3-hydroxyphenyl
hydroxymethyl



1.5.307
2-methoxy-3-hydroxyphenyl
hydroxymethyl



1.5.308
2-ethoxy-3-hydroxyphenyl
hydroxymethyl



1.5.309
2-trifluoromethoxy-3-hydroxyphenyl
hydroxymethyl



1.5.310
2-nitro-3-hydroxyphenyl
hydroxymethyl



1.5.311
2-fluoro-3-methoxyphenyl
hydroxymethyl



1.5.312
2-chloro-3-methoxyphenyl
hydroxymethyl



1.5.313
2-bromo-3-methoxyphenyl
hydroxymethyl



1.5.314
2-methyl-3-methoxyphenyl
hydroxymethyl



1.5.315
2-ethyl-3-methoxyphenyl
hydroxymethyl



1.5.316
2-cyclopropyl-3-methoxyphenyl
hydroxymethyl



1.5.317
2-vinyl-3-methoxyphenyl
hydroxymethyl



1.5.318
2-ethynyl-3-methoxyphenyl
hydroxymethyl



1.5.319
2-cyano-3-methoxyphenyl
hydroxymethyl



1.5.320
2-trifluoromethyl-3-methoxyphenyl
hydroxymethyl



1.5.321
2,3-dimethoxyphenyl
hydroxymethyl



1.5.322
2-ethoxy-3-methoxyphenyl
hydroxymethyl



1.5.323
2-trifluoromethoxy-3-methoxyphenyl
hydroxymethyl



1.5.324
2-nitro-3-methoxyphenyl
hydroxymethyl



1.5.325
2-fluoro-3-ethoxyphenyl
hydroxymethyl



1.5.326
2-chloro-3-ethoxyphenyl
hydroxymethyl



1.5.327
2-bromo-3-ethoxyphenyl
hydroxymethyl



1.5.328
2-methyl-3-ethoxyphenyl
hydroxymethyl



1.5.329
2-ethyl-3-ethoxyphenyl
hydroxymethyl



1.5.330
2-cyclopropyl-3-ethoxyphenyl
hydroxymethyl



1.5.331
2-vinyl-3-ethoxyphenyl
hydroxymethyl



1.5.332
2-ethynyl-3-ethoxyphenyl
hydroxymethyl



1.5.333
2-cyano-3-ethoxyphenyl
hydroxymethyl



1.5.334
2-trifluoromethyl-3-ethoxyphenyl
hydroxymethyl



1.5.335
2-methoxy-3-ethoxyphenyl
hydroxymethyl



1.5.336
2,3-diethoxy--phenyl
hydroxymethyl



1.5.337
2-trifluoromethoxy-3-ethoxyphenyl
hydroxymethyl



1.5.338
2-nitro-3-ethoxyphenyl
hydroxymethyl



1.5.339
2-fluoro-3-propoxyphenyl
hydroxymethyl



1.5.340
2-chloro-3-propoxyphenyl
hydroxymethyl



1.5.341
2-bromo-3-propoxyphenyl
hydroxymethyl



1.5.342
2-methyl-3-propoxyphenyl
hydroxymethyl



1.5.343
2-ethyl-3-propoxyphenyl
hydroxymethyl



1.5.344
2-cyclopropyl-3-propoxyphenyl
hydroxymethyl



1.5.345
2-vinyl-3-propoxyphenyl
hydroxymethyl



1.5.346
2-ethynyl-3-propoxyphenyl
hydroxymethyl



1.5.347
2-cyano-3-propoxyphenyl
hydroxymethyl



1.5.348
2-trifluoromethyl-3-propoxyphenyl
hydroxymethyl



1.5.349
2-methoxy-3-propoxyphenyl
hydroxymethyl



1.5.350
2-ethoxy-3-propoxyphenyl
hydroxymethyl



1.5.351
2-trifluoromethoxy-3-propoxyphenyl
hydroxymethyl



1.5.352
2-nitro-3-propoxyphenyl
hydroxymethyl



1.5.353
2-fluoro-3-isopropoxyphenyl
hydroxymethyl



1.5.354
2-chloro-3-isopropoxyphenyl
hydroxymethyl



1.5.355
2-bromo-3-isopropoxyphenyl
hydroxymethyl



1.5.356
2-methyl-3-isopropoxyphenyl
hydroxymethyl



1.5.357
2-ethyl-3-isopropoxyphenyl
hydroxymethyl



1.5.358
2-cyclopropyl-3-isopropoxyphenyl
hydroxymethyl



1.5.359
2-vinyl-3-isopropoxyphenyl
hydroxymethyl



1.5.360
2-ethynyl-3-isopropoxyphenyl
hydroxymethyl



1.5.361
2-cyano-3-isopropoxyphenyl
hydroxymethyl



1.5.362
2-trifluoromethyl-3-isopropoxyphenyl
hydroxymethyl



1.5.363
2-methoxy-3-isopropoxyphenyl
hydroxymethyl



1.5.364
2-ethoxy-3-isopropoxyphenyl
hydroxymethyl



1.5.365
2-trifluoromethoxy-3-isopropoxyphenyl
hydroxymethyl



1.5.366
2-nitro-3-isopropoxyphenyl
hydroxymethyl



1.5.367
2-fluoro-3-tert-butoxyphenyl
hydroxymethyl



1.5.368
2-chloro-3-tert-butoxyphenyl
hydroxymethyl



1.5.369
2-bromo-3-tert-butoxyphenyl
hydroxymethyl



1.5.370
2-methyl-3-tert-butoxyphenyl
hydroxymethyl



1.5.371
2-ethyl-3-tert-butoxyphenyl
hydroxymethyl



1.5.372
2-cyclopropyl-3-tert-butoxyphenyl
hydroxymethyl



1.5.373
2-vinyl-3-tert-butoxyphenyl
hydroxymethyl



1.5.374
2-ethynyl-3-tert-butoxyphenyl
hydroxymethyl



1.5.375
2-cyano-3-tert-butoxyphenyl
hydroxymethyl



1.5.376
2-trifluoromethyl-3-tert-butoxyphenyl
hydroxymethyl



1.5.377
2-methoxy-3-tert-butoxyphenyl
hydroxymethyl



1.5.378
2-ethoxy-3-tert-butoxyphenyl
hydroxymethyl



1.5.379
2-trifluoromethoxy-3-tert-butoxyphenyl
hydroxymethyl



1.5.380
2-nitro-3-tert-butoxyphenyl
hydroxymethyl



1.5.381
2-fluoro-3-trifluoromethoxyphenyl
hydroxymethyl



1.5.382
2-chloro-3-trifluoromethoxyphenyl
hydroxymethyl



1.5.383
2-bromo-3-trifluoromethoxyphenyl
hydroxymethyl



1.5.384
2-methyl-3-trifluoromethoxyphenyl
hydroxymethyl



1.5.385
2-ethyl-3-trifluoromethoxyphenyl
hydroxymethyl



1.5.386
2-cyclopropyl-3-trifluoromethoxyphenyl
hydroxymethyl



1.5.387
2-vinyl-3-trifluoromethoxyphenyl
hydroxymethyl



1.5.388
2-ethynyl-3-trifluoromethoxyphenyl
hydroxymethyl



1.5.389
2-cyano-3-trifluoromethoxyphenyl
hydroxymethyl



1.5.390
2-trifluoromethyl-3-trifluoromethoxy-
hydroxymethyl




phenyl




1.5.391
2-methoxy-3-trifluoromethoxyphenyl
hydroxymethyl



1.5.392
2-ethoxy-3-trifluoromethoxyphenyl
hydroxymethyl



1.5.393
2,3-bis(trifluoromethoxy)phenyl
hydroxymethyl



1.5.394
2-nitro-3-trifluoromethoxyphenyl
hydroxymethyl



1.5.395
2-fluoro-3-(2,2,2-trifluoroethoxy)phenyl
hydroxymethyl



1.5.396
2-chloro-3-(2,2,2-trifluoroethoxy)phenyl
hydroxymethyl



1.5.397
2-bromo-3-(2,2,2-trifluoroethoxy)phenyl
hydroxymethyl



1.5.398
2-methyl-3-(2,2,2-trifluoroethoxy)phenyl
hydroxymethyl



1.5.399
2-ethyl-3-(2,2,2-trifluoroethoxy)phenyl
hydroxymethyl



1.5.400
2-cyclopropyl-3-(2,2,2-trifluoro-
hydroxymethyl




ethoxy)phenyl




1.5.401
2-vinyl-3-(2,2,2-trifluoroethoxy)phenyl
hydroxymethyl



1.5.402
2-ethynyl-3-(2,2,2-trifluoroethoxyphenyl
hydroxymethyl



1.5.403
2-cyano-3-(2,2,2-trifluoroethoxy)phenyl
hydroxymethyl



1.5.404
2-trifluoromethyl-3-(2,2,2-trifluoro-
hydroxymethyl




ethoxy)phenyl




1.5.405
2-methoxy-3-(2,2,2-trifluoroethoxy)-
hydroxymethyl




phenyl




1.5.406
2-ethoxy-3-(2,2,2-trifluoroethoxy)phenyl
hydroxymethyl



1.5.407
2-trifluoromethoxy-3-(2,2,2-trifluoro-
hydroxymethyl




ethoxy)phenyl




1.5.408
2-nitro-3-(2,2,2-trifluoroethoxy)phenyl
hydroxymethyl



1.5.409
2-fluoro-3-difluoromethoxyphenyl
hydroxymethyl



1.5.410
2-chloro-3-difluoromethoxyphenyl
hydroxymethyl



1.5.411
2-bromo-3-difluoromethoxyphenyl
hydroxymethyl



1.5.412
2-methyl-3-difluoromethoxyphenyl
hydroxymethyl



1.5.413
2-ethyl-3-difluoromethoxyphenyl
hydroxymethyl



1.5.414
2-cyclopropyl-3-difluoromethoxyphenyl
hydroxymethyl



1.5.415
2-vinyl-3-difluoromethoxyphenyl
hydroxymethyl



1.5.416
2-ethynyl-3-difluoromethoxyphenyl
hydroxymethyl



1.5.417
2-cyano-3-difluoromethoxyphenyl
hydroxymethyl



1.5.418
2-trifluoromethyl-3-difluoromethoxy-
hydroxymethyl




phenyl




1.5.419
2-methoxy-3-difluoromethoxyphenyl
hydroxymethyl



1.5.420
2-ethoxy-3-difluoromethoxyphenyl
hydroxymethyl



1.5.421
2-trifluoromethoxy-3-difluoromethoxy-
hydroxymethyl




phenyl




1.5.422
2-nitro-3-difluoromethoxyphenyl
hydroxymethyl



1.5.423
2-fluoro-3-(2-methoxyethoxy)phenyl
hydroxymethyl



1.5.424
2-chloro-3-(2-methoxyethoxy)phenyl
hydroxymethyl



1.5.425
2-bromo-3-(2-methoxyethoxy)phenyl
hydroxymethyl



1.5.426
2-methyl-3-(2-methoxyethoxy)phenyl
hydroxymethyl



1.5.427
2-ethyl-3-(2-methoxyethoxy)phenyl
hydroxymethyl



1.5.428
2-cyclopropyl-3-(2-methoxyethoxy)-
hydroxymethyl




phenyl




1.5.429
2-vinyl-3-(2-methoxyethoxy)phenyl
hydroxymethyl



1.5.430
2-ethynyl-3-(2-methoxyethoxy)phenyl
hydroxymethyl



1.5.431
2-cyano-3-(2-methoxyethoxy)phenyl
hydroxymethyl



1.5.432
2-trifluoromethyl-3-(2-methoxyethoxy)-
hydroxymethyl




phenyl




1.5.433
2-methoxy-3-(2-methoxyethoxy)phenyl
hydroxymethyl



1.5.434
2-ethoxy-3-(2-methoxyethoxy)phenyl
hydroxymethyl



1.5.435
2-trifluoromethoxy-(2-methoxyethoxy)-
hydroxymethyl




phenyl




1.5.436
2-nitro-3-(2-methoxyethoxy)phenyl
hydroxymethyl



1.5.437
2-fluoro-3-(tert-butoxycarbonyloxy)-
hydroxymethyl




phenyl




1.5.438
2-chloro-3-(tert-butoxycarbonyloxy)-
hydroxymethyl




phenyl




1.5.439
2-bromo-3-(tert-butoxycarbonyl-
hydroxymethyl




oxy)phenyl




1.5.440
2-methyl-3-(tert-butoxycarbonyl-
hydroxymethyl




oxy)phenyl




1.5.441
2-ethyl-3-(tert-butoxycarbonyloxy)-
hydroxymethyl




phenyl




1.5.442
2-cyclopropyl-3-(tert-butoxycarbonyl-
hydroxymethyl




oxy)phenyl




1.5.443
2-vinyl-3-(tert-butoxycarbonyloxy)-
hydroxymethyl




phenyl




1.5.444
2-ethynyl-3-(tert-butoxycarbonyl-
hydroxymethyl




oxy)phenyl




1.5.445
2-cyano-3-(tert-butoxycarbonyloxy)-
hydroxymethyl




phenyl




1.5.446
2-trifluoromethyl-3-(tert-butoxycarbonyl-
hydroxymethyl




oxy)phenyl




1.5.447
2-methoxy-3-(tert-butoxycarbonyloxy)-
hydroxymethyl




phenyl




1.5.448
2-ethoxy-3-(tert-butoxycarbonyloxy)-
hydroxymethyl




phenyl




1.5.449
2-trifluoromethoxy-3-(tert-
hydroxymethyl




butoxycarbonyl-oxy)phenyl




1.5.450
2-nitro-3-(tert-butoxycarbonyloxy)-
hydroxymethyl




phenyl




1.5.451
2-fluoro-3-nitrophenyl
hydroxymethyl



1.5.452
2-chloro-3-nitrophenyl
hydroxymethyl



1.5.453
2-bromo-3-nitrophenyl
hydroxymethyl



1.5.454
2-methyl-3-nitrophenyl
hydroxymethyl



1.5.455
2-ethyl-3-nitrophenyl
hydroxymethyl



1.5.456
2-cyclopropyl-3-nitrophenyl
hydroxymethyl



1.5.457
2-vinyl-3-nitrophenyl
hydroxymethyl



1.5.458
2-ethynyl-3-nitrophenyl
hydroxymethyl



1.5.459
2-cyano-3-nitrophenyl
hydroxymethyl



1.5.460
2-trifluoromethyl-3-nitrophenyl
hydroxymethyl



1.5.461
2-methoxy-3-nitrophenyl
hydroxymethyl



1.5.462
2-ethoxy-3-nitrophenyl
hydroxymethyl



1.5.463
2-trifluoromethoxy-3-nitrophenyl
hydroxymethyl



1.5.464
2-fluoro-3-methylsulfanylphenyl
hydroxymethyl



1.5.465
2-chloro-3-methylsulfanylphenyl
hydroxymethyl



1.5.466
2-bromo-3-methylsulfanylphenyl
hydroxymethyl



1.5.467
2-methyl-3-methylsulfanylphenyl
hydroxymethyl



1.5.468
2-ethyl-3-methylsulfanylphenyl
hydroxymethyl



1.5.469
2-cyclopropyl-3-methylsulfanylphenyl
hydroxymethyl



1.5.470
2-vinyl-3-methylsulfanylphenyl
hydroxymethyl



1.5.471
2-ethynyl-3-methylsulfanylphenyl
hydroxymethyl



1.5.472
2-cyano-3-methylsulfanylphenyl
hydroxymethyl



1.5.473
2-trifluoromethyl-3-methylsulfanylphenyl
hydroxymethyl



1.5.474
2-methoxy-3-methylsulfanylphenyl
hydroxymethyl



1.5.475
2-ethoxy-3-methylsulfanylphenyl
hydroxymethyl



1.5.476
2-trifluoromethoxy-3-
hydroxymethyl




methylsulfanylphenyl




1.5.477
2-nitro-3-methylsulfanylphenyl
hydroxymethyl



1.5.478
3,5-difluorophenyl
hydroxymethyl
[CDCl3] 2.0 (s br, 1H);





3.61 (d, 1H); 3.69





(d, 1H), 3.95 (d, 1H),





4.08 (d, 1H), 6.91





(t, 1H); 7.18 (d, 2H).


1.5.479
3,5-difluorophenyl
1-hydroxyethyl
[CDCl3] D1 1.25





(d, 3H); 1.36 (d, 1H);





3.60 (d, 1H); 3.70





(d, 1H); 4.29 (m, 1H);





6.91 (t, 1H); 7.20





(d, 2H). D2 1.29 (d, 3H);





1.42 (d, 1H); 3.60





(d, 1H); 3.69 (d, 1H);





4.22 (m, 1H); 6.91





(t, 1H); 7.20 (d, 2H).


1.5.480
3,5-difluorophenyl
1-hydroxypropyl



1.5.481
3,5-difluorophenyl
(1-hydroxy-2-





methylpropyl)



1.5.482
3,5-difluorophenyl
methoxymethyl
[CDCl3] 3.47 (s, 3H);





3.50 (d, 1H); 3.72





(d, 1H); 3.84 (s, 2H);





6.90 (m, 1H); 7.19





(m, 2H).


1.5.483
2-ethyl-3-cyanophenyl
2-methoxyethyl



1.5.484
3-chloro-5-fluorophenyl
hydroxymethyl



1.5.485
3-chloro-5-fluorophenyl
1-hydroxyethyl



1.5.486
3-chloro-5-fluorophenyl
1-hydroxypropyl



1.5.487
3-chloro-5-fluorophenyl
(1-hydroxy-2-





methylpropyl)



1.5.488
3-chloro-5-fluorophenyl
methoxymethyl



1.5.489
3-chloro-5-fluorophenyl
2-methoxyethyl



1.5.490
3-bromo-5-fluorophenyl
hydroxymethyl



1.5.491
3-bromo-5-fluorophenyl
1-hydroxyethyl



1.5.492
3-bromo-5-fluorophenyl
1-hydroxypropyl



1.5.493
3-bromo-5-fluorophenyl
(1-hydroxy-2-





methylpropyl)



1.5.494
3-bromo-5-fluorophenyl
methoxymethyl



1.5.495
3-bromo-5-fluorophenyl
2-methoxyethyl



1.5.496
3-iodo-5-fluorophenyl
hydroxymethyl



1.5.497
3-methyl-5-fluorophenyl
hydroxymethyl



1.5.498
3-methyl-5-fluorophenyl
1-hydroxyethyl



1.5.499
3-methyl-5-fluorophenyl
1-hydroxypropyl



1.5.500
3-methyl-5-fluorophenyl
(1-hydroxy-2-





methylpropyl)



1.5.501
3-methyl-5-fluorophenyl
methoxymethyl



1.5.502
3-methyl-5-fluorophenyl
2-methoxyethyl



1.5.503
3-ethyl-5-fluorophenyl
hydroxymethyl



1.5.504
3-propyl-5-fluorophenyl
hydroxymethyl



1.5.505
3-i-propyl-5-fluorophenyl
hydroxymethyl



1.5.506
3-n-butyl-5-fluorophenyl
hydroxymethyl



1.5.507
3-isobutyl-5-fluorophenyl
hydroxymethyl



1.5.508
3-tert-butyl-5-fluorophenyl
hydroxymethyl



1.5.509
3-cyclopropyl-5-fluorophenyl
hydroxymethyl



1.5.510
3-vinyl-5-fluorophenyl
hydroxymethyl



1.5.511
3-ethynyl-5-fluorophenyl
hydroxymethyl



1.5.512
3-cyano-5-fluorophenyl
hydroxymethyl



1.5.513
3-trifluoromethyl-5-fluorophenyl
hydroxymethyl



1.5.514
3-trifluoromethyl-5-fluorophenyl
1-hydroxyethyl



1.5.515
3-trifluoromethyl-5-fluorophenyl
1-hydroxypropyl



1.5.516
3-trifluoromethyl-5-fluorophenyl
(1-hydroxy-2-





methylpropyl)



1.5.517
3-trifluoromethyl-5-fluorophenyl
methoxymethyl



1.5.518
3-trifluoromethyl-5-fluorophenyl
2-methoxyethyl



1.5.519
3-(methoxycarbonyl)-5-fluorophenyl
hydroxymethyl



1.5.520
3-hydroxymethyl-5-fluorophenyl
hydroxymethyl



1.5.521
3-carbamoyl-5-fluorophenyl
hydroxymethyl



1.5.522
3-hydroxy-5-fluorophenyl
hydroxymethyl



1.5.523
3-methoxy-5-fluorophenyl
hydroxymethyl



1.5.524
3-ethoxy-5-fluorophenyl
hydroxymethyl



1.5.525
3-n-propoxy-5-fluorophenyl
hydroxymethyl



1.5.526
3-isopropoxy-5-fluorophenyl
hydroxymethyl



1.5.527
3-n-butoxy-5-fluorophenyl
hydroxymethyl



1.5.528
3-isobutoxy-5-fluorophenyl
hydroxymethyl



1.5.529
3-tert-butoxy-5-fluorophenyl
hydroxymethyl



1.5.530
3-difluoromethoxy-5-fluorophenyl
hydroxymethyl



1.5.531
3-trifluoromethoxy-5-fluorophenyl
hydroxymethyl



1.5.532
3-(2,2,2-trifluoroethoxy)-5-fluorophenyl
hydroxymethyl



1.5.533
3-(2-chloroethoxy)-5-fluorophenyl
hydroxymethyl



1.5.534
3-(2-hydroxyethoxy)-5-fluorophenyl
hydroxymethyl



1.5.535
3-[(tert-butoxycarbonyl)oxy]-5-
hydroxymethyl




fluorophenyl




1.5.536
3-nitro-5-fluorophenyl
hydroxymethyl



1.5.537
3-acetoxy-5-fluorophenyl
hydroxymethyl



1.5.538
{3-[(tert-butoxycarbonyl)amino]-5-
hydroxymethyl




fluorophenyl}




1.5.539
3-methylsulfanyl-5-fluorophenyl
hydroxymethyl



1.5.540
3,5-dichlorophenyl
hydroxymethyl
[CDCl3] 3.68 (q, 2H);





3.96 (d, 1H); 4.08 (d,





1H); 7.45 (s, 1H); 7.56





(s, 2H).


1.5.541
3,5-dichlorophenyl
1-hydroxyethyl



1.5.542
3,5-dichlorophenyl
1-hydroxypropyl



1.5.543
3,5-dichlorophenyl
(1-hydroxy-2-





methylpropyl)



1.5.544
3,5-dichlorophenyl
methoxymethyl
[CDCl3] 3.48 (s, 3H);





3.50 (d, 1H); 3.72 (d,





1H); 3.85 (q, 2H); 7.42





(m, 1H); 7.55 (m, 2H).


1.5.545
3,5-dichlorophenyl
2-methoxyethyl
[CDCl3]


1.5.546
3-bromo-5-chlorophenyl
hydroxymethyl



1.5.547
3-iodo-5-chlorophenyl
hydroxymethyl



1.5.548
3-methyl-5-chlorophenyl
hydroxymethyl



1.5.549
3-propyl-5-chlorophenyl
hydroxymethyl



1.5.550
3-isopropyl-5-chlorophenyl
hydroxymethyl



1.5.551
3-n-butyl-5-chlorophenyl
hydroxymethyl



1.5.552
3-isobutyl-5-chlorophenyl
hydroxymethyl



1.5.553
3-tert-butyl-5-chlorophenyl
hydroxymethyl



1.5.554
3-cyclopropyl-5-chlorophenyl
hydroxymethyl



1.5.555
3-cyano-5-chlorophenyl
hydroxymethyl



1.5.556
3-trifluoromethyl-5-chlorophenyl
hydroxymethyl



1.5.557
3-(methoxycarbonyl)-5-chlorophenyl
hydroxymethyl



1.5.558
3-methoxy-5-chlorophenyl
hydroxymethyl



1.5.559
3-ethoxy-5-chlorophenyl
hydroxymethyl



1.5.560
3-n-propoxy-5-chlorophenyl
hydroxymethyl



1.5.561
3-isopropoxy-5-chlorophenyl
hydroxymethyl



1.5.562
3-n-butoxy-5-chlorophenyl
hydroxymethyl



1.5.563
3-isobutoxy-5-chlorophenyl
hydroxymethyl



1.5.564
3-difluoromethoxy-5-chlorophenyl
hydroxymethyl



1.5.565
3-trifluoromethoxy-5-chlorophenyl
hydroxymethyl



1.5.566
3-nitro-5-chlorophenyl
hydroxymethyl



1.5.567
3-acetoxy-5-chlorophenyl
hydroxymethyl



1.5.568
3,5-dibromophenyl
hydroxymethyl



1.5.569
3,5-dibromophenyl
1-hydroxyethyl



1.5.570
3-iodo-5-bromophenyl
hydroxymethyl



1.5.571
3-methyl-5-bromophenyl
hydroxymethyl



1.5.572
3-methyl-5-bromophenyl
1-hydroxyethyl



1.5.573
3-methyl-5-bromophenyl
1-hydroxypropyl



1.5.574
3-methyl-5-bromophenyl
(1-hydroxy-2-





methylpropyl)



1.5.575
3-methyl-5-bromophenyl
methoxymethyl



1.5.576
3-methyl-5-bromophenyl
2-methoxyethyl



1.5.577
3-ethyl-5-bromophenyl
hydroxymethyl



1.5.578
3-propyl-5-bromophenyl
hydroxymethyl



1.5.579
3-isopropyl-5-bromophenyl
hydroxymethyl



1.5.580
3-n-butyl-5-bromophenyl
hydroxymethyl



1.5.581
3-isobutyl-5-bromophenyl
hydroxymethyl



1.5.582
3-tert-butyl-5-bromophenyl
hydroxymethyl



1.5.583
3-cyclopropyl-5-bromophenyl
hydroxymethyl



1.5.584
3-cyano-5-bromophenyl
hydroxymethyl



1.5.585
3-trifluoromethyl-5-bromophenyl
hydroxymethyl



1.5.586
3-(methoxycarbonyl)-5-bromophenyl
hydroxymethyl



1.5.587
3-methoxy-5-bromophenyl
hydroxymethyl



1.5.588
3-ethoxy-5-bromophenyl
hydroxymethyl



1.5.589
3-n-propoxy-5-bromophenyl
hydroxymethyl



1.5.590
3-isopropoxy-5-bromophenyl
hydroxymethyl



1.5.591
3-n-butoxy-5-bromophenyl
hydroxymethyl



1.5.592
3-isobutoxy-5-bromophenyl
hydroxymethyl



1.5.593
3-difluoromethoxy-5-bromophenyl
hydroxymethyl



1.5.594
3-trifluoromethoxy-5-bromophenyl
hydroxymethyl



1.5.595
3-nitro-5-bromophenyl
hydroxymethyl



1.5.596
3-acetoxy-5-bromophenyl
hydroxymethyl



1.5.597
3-methylsulfanyl-5-bromophenyl
hydroxymethyl



1.5.598
3,5-diiodophenyl
hydroxymethyl



1.5.599
3-methyl-5-iodophenyl
hydroxymethyl



1.5.600
3-ethyl-5-iodophenyl
hydroxymethyl



1.5.601
3-propyl-5-iodophenyl
hydroxymethyl



1.5.602
3-isopropyl-5-iodophenyl
hydroxymethyl



1.5.603
3-n-butyl-5-iodophenyl
hydroxymethyl



1.5.604
3-isobutyl-5-iodophenyl
hydroxymethyl



1.5.605
3-tert-butyl-5-iodophenyl
hydroxymethyl



1.5.606
3-cyclopropyl-5-iodophenyl
hydroxymethyl



1.5.607
3-cyano-5-iodophenyl
hydroxymethyl



1.5.608
3-trifluoromethyl-5-iodophenyl
hydroxymethyl



1.5.609
3-(methoxycarbonyl)-5-iodophenyl
hydroxymethyl



1.5.610
3-methoxy-5-iodophenyl
hydroxymethyl



1.5.611
3-ethoxy-5-iodophenyl
hydroxymethyl



1.5.612
3-n-propoxy-5-iodophenyl
hydroxymethyl



1.5.613
3-isopropoxy-5-iodophenyl
hydroxymethyl



1.5.614
3-n-butoxy-5-iodophenyl
hydroxymethyl



1.5.615
3-isobutoxy-5-iodophenyl
hydroxymethyl



1.5.616
3-difluoromethoxy-5-iodophenyl
hydroxymethyl



1.5.617
3-trifluoromethoxy-5-iodophenyl
hydroxymethyl



1.5.618
3-nitro-5-iodophenyl
hydroxymethyl



1.5.619
3-acetoxy-5-iodophenyl
hydroxymethyl



1.5.620
3-methylsulfanyl-5-iodophenyl
hydroxymethyl



1.5.621
3,5-dimethylphenyl
hydroxymethyl



1.5.622
3-ethyl-5-methylphenyl
hydroxymethyl



1.5.623
3-propyl-5-methylphenyl
hydroxymethyl



1.5.624
3-isopropyl-5-methylphenyl
hydroxymethyl



1.5.625
3-n-butyl-5-methylphenyl
hydroxymethyl



1.5.626
3-isobutyl-5-methylphenyl
hydroxymethyl



1.5.627
3-tert-butyl-5-methylphenyl
hydroxymethyl



1.5.628
3-cyclopropyl-5-methylphenyl
hydroxymethyl



1.5.629
3-cyano-5-methylphenyl
hydroxymethyl



1.5.630
3-trifluoromethyl-5-methylphenyl
hydroxymethyl



1.5.631
3-(methoxycarbonyl)-5-methylphenyl
hydroxymethyl



1.5.632
3-methoxy-5-methylphenyl
hydroxymethyl



1.5.633
3-ethoxy-5-methylphenyl
hydroxymethyl



1.5.634
3-n-propoxy-5-methylphenyl
hydroxymethyl



1.5.635
3-n-butoxy-5-methylphenyl
hydroxymethyl



1.5.636
3-isobutoxy-5-methylphenyl
hydroxymethyl



1.5.637
3-difluoromethoxy-5-methylphenyl
hydroxymethyl



1.5.638
3-trifluoromethoxy-5-methylphenyl
hydroxymethyl



1.5.639
3-nitro-5-methylphenyl
hydroxymethyl



1.5.640
3-acetoxy-5-methylphenyl
hydroxymethyl



1.5.641
3-methylsulfanyl-5-methylphenyl
hydroxymethyl



1.5.642
3,5-diethylphenyl
hydroxymethyl



1.5.643
3-propyl-5-ethylphenyl
hydroxymethyl



1.5.644
3-isopropyl-5-ethylphenyl
hydroxymethyl



1.5.645
3-n-butyl-5-ethylphenyl
hydroxymethyl



1.5.646
3-isobutyl-5-ethylphenyl
hydroxymethyl



1.5.647
3-tert-butyl-5-ethylphenyl
hydroxymethyl



1.5.648
3-cyclopropyl-5-ethylphenyl
hydroxymethyl



1.5.649
3-cyano-5-ethylphenyl
hydroxymethyl



1.5.650
3-trifluoromethyl-5-ethylphenyl
hydroxymethyl



1.5.651
3-(methoxycarbonyl)-5-ethylphenyl
hydroxymethyl



1.5.652
3-methoxy-5-ethylphenyl
hydroxymethyl



1.5.653
3-ethoxy-5-ethylphenyl
hydroxymethyl



1.5.654
3-n-propoxy-5-ethylphenyl
hydroxymethyl



1.5.655
3-n-butoxy-5-ethylphenyl
hydroxymethyl



1.5.656
3-isobutoxy-5-ethylphenyl
hydroxymethyl



1.5.657
3-difluoromethoxy-5-ethylphenyl
hydroxymethyl



1.5.658
3-trifluoromethoxy-5-ethylphenyl
hydroxymethyl



1.5.659
3-nitro-5-ethylphenyl
hydroxymethyl



1.5.660
3-acetoxy-5-ethylphenyl
hydroxymethyl



1.5.661
3-methylsulfanyl-5-ethylphenyl
hydroxymethyl



1.5.662
3,5-dipropylphenyl
hydroxymethyl



1.5.663
3-isopropyl-5-propylphenyl
hydroxymethyl



1.5.664
3-n-butyl-5-propylphenyl
hydroxymethyl



1.5.665
3-isobutyl-5-propylphenyl
hydroxymethyl



1.5.666
3-tert-butyl-5-propylphenyl
hydroxymethyl



1.5.667
3-cyclopropyl-5-propylphenyl
hydroxymethyl



1.5.668
3-cyano-5-propylphenyl
hydroxymethyl



1.5.669
3-trifluoromethyl-5-propylphenyl
hydroxymethyl



1.5.670
3-(methoxycarbonyl)-5-propylphenyl
hydroxymethyl



1.5.671
3-methoxy-5-propylphenyl
hydroxymethyl



1.5.672
3-ethoxy-5-propylphenyl
hydroxymethyl



1.5.673
3-n-propoxy-5-propylphenyl
hydroxymethyl



1.5.674
3-n-butoxy-5-propylphenyl
hydroxymethyl



1.5.675
3-isobutoxy-5-propylphenyl
hydroxymethyl



1.5.676
3-difluoromethoxy-5-propylphenyl
hydroxymethyl



1.5.677
3-trifluoromethoxy-5-ethylphenyl
hydroxymethyl



1.5.678
3-nitro-5-propylphenyl
hydroxymethyl



1.5.679
3-acetoxy-5-propylphenyl
hydroxymethyl



1.5.680
3-methylsulfanyl-5-propylphenyl
hydroxymethyl



1.5.681
3,5-diisopropylphenyl
hydroxymethyl



1.5.682
3-n-butyl-5-isopropylphenyl
hydroxymethyl



1.5.683
3-isobutyl-5-isopropylphenyl
hydroxymethyl



1.5.684
3-tert-butyl-5-isopropylphenyl
hydroxymethyl



1.5.685
3-cyclopropyl-5-isopropylphenyl
hydroxymethyl



1.5.686
3-cyano-5-isopropylphenyl
hydroxymethyl



1.5.687
3-trifluoromethyl-5-isopropylphenyl
hydroxymethyl



1.5.688
3-(methoxycarbonyl)-5-isopropylphenyl
hydroxymethyl



1.5.689
3-methoxy-5-isopropylphenyl
hydroxymethyl



1.5.690
3-ethoxy-5-isopropylphenyl
hydroxymethyl



1.5.691
3-n-propoxy-5-isopropylphenyl
hydroxymethyl



1.5.692
3-n-butoxy-5-isopropylphenyl
hydroxymethyl



1.5.693
3-isobutoxy-5-isopropylphenyl
hydroxymethyl



1.5.694
3-difluoromethoxy-5-isopropylphenyl
hydroxymethyl



1.5.695
3-trifluoromethoxy-5-isopropylphenyl
hydroxymethyl



1.5.696
3-nitro-5-isopropylphenyl
hydroxymethyl



1.5.697
3-acetoxy-5-isopropylphenyl
hydroxymethyl



1.5.698
3-methylsulfanyl-5-isopropylphenyl
hydroxymethyl



1.5.699
3,5-dibutylphenyl
hydroxymethyl



1.5.700
3-isobutyl-5-butylphenyl
hydroxymethyl



1.5.701
3-tert-butyl-5-butylphenyl
hydroxymethyl



1.5.702
3-cyclopropyl-5-butylphenyl
hydroxymethyl



1.5.703
3-cyano-5-butylphenyl
hydroxymethyl



1.5.704
3-trifluoromethyl-5-butylphenyl
hydroxymethyl



1.5.705
3-(methoxycarbonyl)-5-butylphenyl
hydroxymethyl



1.5.706
3-methoxy-5-butylphenyl
hydroxymethyl



1.5.707
3-ethoxy-5-butylphenyl
hydroxymethyl



1.5.708
3-n-propoxy-5-butylphenyl
hydroxymethyl



1.5.709
3-n-butoxy-5-butylphenyl
hydroxymethyl



1.5.710
3-isobutoxy-5-butylphenyl
hydroxymethyl



1.5.711
3-difluoromethoxy-5-butylphenyl
hydroxymethyl



1.5.712
3-trifluoromethoxy-5-butylphenyl
hydroxymethyl



1.5.713
3-nitro-5-butylphenyl
hydroxymethyl



1.5.714
3-acetoxy-5-butylphenyl
hydroxymethyl



1.5.715
3-methylsulfanyl-5-butylphenyl
hydroxymethyl



1.5.716
3,5-diisobutylphenyl
hydroxymethyl



1.5.717
3-tert-butyl-5-isobutylphenyl
hydroxymethyl



1.5.718
3-cyclopropyl-5-isobutylphenyl
hydroxymethyl



1.5.719
3-cyano-5-isobutylphenyl
hydroxymethyl



1.5.720
3-trifluoromethyl-5-isobutylphenyl
hydroxymethyl



1.5.721
3-(methoxycarbonyl)-5-isobutylphenyl
hydroxymethyl



1.5.722
3-methoxy-5-isobutylphenyl
hydroxymethyl



1.5.723
3-ethoxy-5-isobutylphenyl
hydroxymethyl



1.5.724
3-n-propoxy-5-isobutylphenyl
hydroxymethyl



1.5.725
3-n-butoxy-5-isobutylphenyl
hydroxymethyl



1.5.726
3-isobutoxy-5-isobutylphenyl
hydroxymethyl



1.5.727
3-difluoromethoxy-5-isobutylphenyl
hydroxymethyl



1.5.728
3-trifluoromethoxy-5-isobutylphenyl
hydroxymethyl



1.5.729
3-nitro-5-isobutylphenyl
hydroxymethyl



1.5.730
3-acetoxy-5-isobutylphenyl
hydroxymethyl



1.5.731
3-methylsulfanyl-5-isobutylphenyl
hydroxymethyl



1.5.732
3,5-di(tert-butyl)phenyl
hydroxymethyl



1.5.733
3-cyclopropyl-5-tert-butylphenyl
hydroxymethyl



1.5.734
3-cyano-5-tert-butylphenyl
hydroxymethyl



1.5.735
3-trifluoromethyl-5-tert-butylphenyl
hydroxymethyl



1.5.736
3-(methoxycarbonyl)-5-tert-butylphenyl
hydroxymethyl



1.5.737
3-methoxy-5-tert-butylphenyl
hydroxymethyl



1.5.738
3-ethoxy-5-tert-butylphenyl
hydroxymethyl



1.5.739
3-n-propoxy-5-tert-butylphenyl
hydroxymethyl



1.5.740
3-n-butoxy-5-tert-butylphenyl
hydroxymethyl



1.5.741
3-isobutoxy-5-tert-butylphenyl
hydroxymethyl



1.5.742
3-difluoromethoxy-5-tert-butylphenyl
hydroxymethyl



1.5.743
3-trifluoromethoxy-5-tert-butylphenyl
hydroxymethyl



1.5.744
3-nitro-5-tert-butylphenyl
hydroxymethyl



1.5.745
3-acetoxy-5-tert-butylphenyl
hydroxymethyl



1.5.746
3-methylsulfanyl-5-tert-butylphenyl
hydroxymethyl



1.5.747
3-tert-butyl-5-cyclopropylphenyl
hydroxymethyl



1.5.748
3,5-dicyclopropyl-phenyl
hydroxymethyl



1.5.749
3-cyano-5-cyclopropylphenyl
hydroxymethyl



1.5.750
3-trifluoromethyl-5-cyclopropylphenyl
hydroxymethyl



1.5.751
3-(hydroxycarbonyl)-5-cyclopropylphenyl
hydroxymethyl



1.5.752
3-(methoxycarbonyl)-5-
hydroxymethyl




cyclopropylphenyl




1.5.753
3-methoxy-5-cyclopropylphenyl
hydroxymethyl



1.5.754
3-ethoxy-5-cyclopropylphenyl
hydroxymethyl



1.5.755
3-n-propoxy-5-cyclopropylphenyl
hydroxymethyl



1.5.756
3-n-butoxy-5-cyclopropylphenyl
hydroxymethyl



1.5.757
3-isobutoxy-5-cyclopropylphenyl
hydroxymethyl



1.5.758
3-difluoromethoxy-5-cyclopropylphenyl
hydroxymethyl



1.5.759
3-trifluoromethoxy-5-cyclopropylphenyl
hydroxymethyl



1.5.760
3-nitro-5-cyclopropylphenyl
hydroxymethyl



1.5.761
3-acetoxy-5-cyclopropylphenyl
hydroxymethyl



1.5.762
3-methylsulfanyl-5-cyclopropylphenyl
hydroxymethyl



1.5.763
3,5-dicyanophenyl
hydroxymethyl



1.5.764
3-trifluoromethyl-5-cyanophenyl
hydroxymethyl



1.5.765
3-(methoxycarbonyl)-5-cyanophenyl
hydroxymethyl



1.5.766
3-methoxy-5-cyanophenyl
hydroxymethyl



1.5.767
3-ethoxy-5-cyanophenyl
hydroxymethyl



1.5.768
3-n-propoxy-5-cyanophenyl
hydroxymethyl



1.5.769
3-n-butoxy-5-cyanophenyl
hydroxymethyl



1.5.770
3-isobutoxy-5-cyanophenyl
hydroxymethyl



1.5.771
3-difluoromethoxy-5-cyanophenyl
hydroxymethyl



1.5.772
3-trifluoromethoxy-5-cyanophenyl
hydroxymethyl



1.5.773
3-nitro-5-cyanophenyl
hydroxymethyl



1.5.774
3-acetoxy-5-cyanophenyl
hydroxymethyl



1.5.775
3-methylsulfanyl-5-cyanophenyl
hydroxymethyl



1.5.776
3,5-di(trifluoromethyl)-phenyl
hydroxymethyl



1.5.777
3-(methoxycarbonyl)-5-trifluoromethyl-
hydroxymethyl




phenyl




1.5.778
3-methoxy-5-trifluoromethylphenyl
hydroxymethyl



1.5.779
3-ethoxy-5-trifluoromethylphenyl
hydroxymethyl



1.5.780
3-n-propoxy-5-trifluoromethylphenyl
hydroxymethyl



1.5.781
3-isobutoxy-5-trifluoromethylphenyl
hydroxymethyl



1.5.782
3-difluoromethoxy-5-
hydroxymethyl




trifluoromethylphenyl




1.5.783
3-trifluoromethoxy-5-
hydroxymethyl




trifluoromethylphenyl




1.5.784
3-nitro-5-trifluoromethylphenyl
hydroxymethyl



1.5.785
3-acetoxy-5-trifluoromethylphenyl
hydroxymethyl



1.5.786
3-methylsulfanyl-5-trifluoromethylphenyl
hydroxymethyl



1.5.787
3,5-di(methoxycarbonyl)phenyl
hydroxymethyl



1.5.788
3-methoxy-5-(methoxycarbonyl)phenyl
hydroxymethyl



1.5.789
3-ethoxy-5-(methoxycarbonyl)phenyl
hydroxymethyl



1.5.790
3-n-propoxy-5-(methoxycarbonyl)-
hydroxymethyl




phenyl




1.5.791
3-n-butoxy-5-(methoxycarbonyl)phenyl
hydroxymethyl



1.5.792
3-isobutoxy-5-(methoxycarbonyl)phenyl
hydroxymethyl



1.5.793
3-difluoromethoxy-5-(methoxycarbonyl)-
hydroxymethyl




phenyl




1.5.794
3-trifluoromethoxy-5-(methoxycarbonyl)-
hydroxymethyl




phenyl




1.5.795
3-nitro-5-(methoxycarbonyl)phenyl
hydroxymethyl



1.5.796
3-acetoxy-5-(methoxycarbonyl)phenyl
hydroxymethyl



1.5.797
3-methylsulfanyl-5-(methoxycarbonyl)-
hydroxymethyl




phenyl




1.5.798
3,5-dimethoxyphenyl
hydroxymethyl



1.5.799
3-ethoxy-5-methoxyphenyl
hydroxymethyl



1.5.800
3-n-propoxy-5-methoxyphenyl
hydroxymethyl



1.5.801
3-isobutoxy-5-methoxyphenyl
hydroxymethyl



1.5.802
3-difluoromethoxy-5-methoxyphenyl
hydroxymethyl



1.5.803
3-trifluoromethoxy-5-methoxyphenyl
hydroxymethyl



1.5.804
3-nitro-5-methoxyphenyl
hydroxymethyl



1.5.805
3-acetoxy-5-methoxyphenyl
hydroxymethyl



1.5.806
3-methylsulfanyl-5-methoxyphenyl
hydroxymethyl



1.5.807
3,5-diethoxyphenyl
hydroxymethyl



1.5.808
3-n-propoxy-5-ethoxyphenyl
hydroxymethyl



1.5.809
3-n-butoxy-5-ethoxyphenyl
hydroxymethyl



1.5.810
3-isobutoxy-5-ethoxyphenyl
hydroxymethyl



1.5.811
3-difluoromethoxy-5-ethoxyphenyl
hydroxymethyl



1.5.812
3-trifluoromethoxy-5-ethoxyphenyl
hydroxymethyl



1.5.813
3-nitro-5-ethoxyphenyl
hydroxymethyl



1.5.814
3-acetoxy-5-ethoxyphenyl
hydroxymethyl



1.5.815
3-methylsulfanyl-5-ethoxyphenyl
hydroxymethyl



1.5.816
3,5-dipropoxyphenyl
hydroxymethyl



1.5.817
3-n-butoxy-5-propoxyphenyl
hydroxymethyl



1.5.818
3-isobutoxy-5-propoxyphenyl
hydroxymethyl



1.5.819
3-difluoromethoxy-5-propoxyphenyl
hydroxymethyl



1.5.820
3-trifluoromethoxy-5-propoxyphenyl
hydroxymethyl



1.5.821
3-nitro-5-propoxyphenyl
hydroxymethyl



1.5.822
3-acetoxy-5-propoxyphenyl
hydroxymethyl



1.5.823
3-methylsulfanyl-5-propoxyphenyl
hydroxymethyl



1.5.824
3,5-di(isopropoxy)phenyl
hydroxymethyl



1.5.825
3-n-butoxy-5-isopropoxyphenyl
hydroxymethyl



1.5.826
3-isobutoxy-5-isopropoxyphenyl
hydroxymethyl



1.5.827
3-difluoromethoxy-5-isopropoxyphenyl
hydroxymethyl



1.5.828
3-trifluoromethoxy-5-isopropoxyphenyl
hydroxymethyl



1.5.829
3-nitro-5-isopropoxyphenyl
hydroxymethyl



1.5.830
3-acetoxy-5-isopropoxyphenyl
hydroxymethyl



1.5.831
3-methylsulfanyl-5-isopropoxyphenyl
hydroxymethyl



1.5.832
3,5-di(trifluoromethoxy)phenyl
hydroxymethyl



1.5.833
3-nitro-5-trifluoromethoxyphenyl
hydroxymethyl



1.5.834
3-methylsulfanyl-5-trifluoromethoxy-
hydroxymethyl




phenyl




1.5.835
3,5-bis(difluoromethoxy)phenyl
hydroxymethyl



1.5.836
3,5-bis(difluoromethoxy)phenyl
1-hydroxyethyl



1.5.837
3,5-bis(difluoromethoxy)phenyl
1-hydroxypropyl



1.5.838
3,5-bis(difluoromethoxy)phenyl
(1-hydroxy-2-





methylpropyl)



1.5.839
3-trifluoromethoxy-5-difluoromethoxy-
hydroxymethyl




phenyl




1.5.840
3-nitro-5-difluoromethoxyphenyl
hydroxymethyl



1.5.841
3-acetoxy-5-difluoromethoxyphenyl
hydroxymethyl



1.5.842
3-methylsulfanyl-5-difluoromethoxy-
hydroxymethyl




phenyl




1.5.843
3,5-bis(acetoxy)phenyl
hydroxymethyl



1.5.844
3-methylsulfanyl-5-acetoxyphenyl
hydroxymethyl



1.5.845
3,5-dinitrophenyl
hydroxymethyl



1.5.846
3-acetoxy-5-nitrophenyl
hydroxymethyl



1.5.847
3-methylsulfanyl-5-nitrophenyl
hydroxymethyl



1.5.848
3,5-di(methylsulfanyl)phenyl
hydroxymethyl



1.5.849
3,4-difluorophenyl
hydroxymethyl



1.5.850
3,4-difluorophenyl
1-hydroxyethyl



1.5.851
3,4-difluorophenyl
1-hydroxypropyl



1.5.852
3,4-difluorophenyl
(1-hydroxy-2-





methylpropyl)



1.5.853
3,4-difluorophenyl
methoxymethyl



1.5.854
3,4-difluorophenyl
2-methoxyethyl



1.5.855
3-chloro-4-fluorophenyl
hydroxymethyl



1.5.856
3-chloro-4-fluorophenyl
1-hydroxyethyl



1.5.857
3-chloro-4-fluorophenyl
1-hydroxypropyl



1.5.858
3-chloro-4-fluorophenyl
(1-hydroxy-2-





methylpropyl)



1.5.859
3-chloro-4-fluorophenyl
methoxymethyl



1.5.860
3-chloro-4-fluorophenyl
2-methoxyethyl



1.5.861
3-bromo-4-fluorophenyl
hydroxymethyl



1.5.862
3-methyl-4-fluorophenyl
hydroxymethyl



1.5.863
3-methyl-4-fluorophenyl
1-hydroxyethyl



1.5.864
3-ethyl-4-fluorophenyl
hydroxymethyl



1.5.865
3-cyclopropyl-4-fluorophenyl
hydroxymethyl



1.5.866
3-cyano-4-fluorophenyl
hydroxymethyl



1.5.867
3-methoxy-4-fluorophenyl
hydroxymethyl



1.5.868
3-ethoxy-4-fluorophenyl
hydroxymethyl



1.5.869
3-trifluoromethoxy-4-fluorophenyl
hydroxymethyl



1.5.870
3-nitro-4-fluorophenyl
hydroxymethyl



1.5.871
3-fluoro-4-chlorophenyl
hydroxymethyl



1.5.872
3,4-dichlorophenyl
hydroxymethyl



1.5.873
3-bromo-4-chlorophenyl
hydroxymethyl



1.5.874
3-methyl-4-chlorophenyl
hydroxymethyl



1.5.875
3-cyclopropyl-4-chlorophenyl
hydroxymethyl



1.5.876
3-cyano-4-chlorophenyl
hydroxymethyl



1.5.877
3-trifluoromethyl-4-chlorophenyl
hydroxymethyl



1.5.878
3-methoxy-4-chlorophenyl
hydroxymethyl



1.5.879
3-ethoxy-4-chlorophenyl
hydroxymethyl



1.5.880
3-trifluoromethoxy-4-chlorophenyl
hydroxymethyl



1.5.881
3-nitro-4-chlorophenyl
hydroxymethyl



1.5.882
3-fluoro-4-bromophenyl
hydroxymethyl



1.5.883
3-chloro-4-bromophenyl
hydroxymethyl



1.5.884
3,4-dibromophenyl
hydroxymethyl



1.5.885
3-methyl-4-bromophenyl
hydroxymethyl



1.5.886
3-cyclopropyl-4-bromophenyl
hydroxymethyl



1.5.887
3-cyano-4-bromophenyl
hydroxymethyl



1.5.888
3-trifluoromethyl-4-bromophenyl
hydroxymethyl



1.5.889
3-methoxy-4-phenyl
hydroxymethyl



1.5.890
3-ethoxy-4-bromophenyl
hydroxymethyl



1.5.891
3-trifluoromethoxy-4-bromophenyl
hydroxymethyl



1.5.892
3-nitro-4-bromophenyl
hydroxymethyl



1.5.893
3-fluoro-4-iodophenyl
hydroxymethyl



1.5.894
3-chloro-4-iodophenyl
hydroxymethyl



1.5.895
3-bromo-4-iodophenyl
hydroxymethyl



1.5.896
3-methyl-4-iodophenyl
hydroxymethyl



1.5.897
3-cyclopropyl-4-iodophenyl
hydroxymethyl



1.5.898
3-cyano-4-iodophenyl
hydroxymethyl



1.5.899
3-trifluoromethyl-4-iodophenyl
hydroxymethyl



1.5.900
3-methoxy-4-iodophenyl
hydroxymethyl



1.5.901
3-ethoxy-4-iodophenyl
hydroxymethyl



1.5.902
3-trifluoromethoxy-4-iodophenyl
hydroxymethyl



1.5.903
3-nitro-4-iodophenyl
hydroxymethyl



1.5.904
3-fluoro-4-methylphenyl
hydroxymethyl



1.5.905
3-chloro-4-methylphenyl
hydroxymethyl



1.5.906
3-bromo-4-methylphenyl
hydroxymethyl



1.5.907
3,4-dimethylphenyl
hydroxymethyl



1.5.908
3,4-dimethylphenyl
1-hydroxyethyl



1.5.909
3,4-dimethylphenyl
1-hydroxypropyl



1.5.910
3,4-dimethylphenyl
(1-hydroxy-2-





methylpropyl)



1.5.911
3,4-dimethylphenyl
methoxymethyl



1.5.912
3,4-dimethylphenyl
2-methoxyethyl



1.5.913
3-ethyl-4-methylphenyl
hydroxymethyl



1.5.914
3-cyclopropyl-4-methylphenyl
hydroxymethyl



1.5.915
3-cyano-4-methylphenyl
hydroxymethyl



1.5.916
3-trifluoromethyl-4-methylphenyl
hydroxymethyl



1.5.917
3-methoxy-4-methylphenyl
hydroxymethyl



1.5.918
3-ethoxy-4-methylphenyl
hydroxymethyl



1.5.919
3-trifluoromethoxy-4-methylphenyl
hydroxymethyl



1.5.920
3-nitro-4-methylphenyl
hydroxymethyl



1.5.921
3-fluoro-4-ethylphenyl
hydroxymethyl



1.5.922
3-chloro-4-ethylphenyl
hydroxymethyl



1.5.923
3-bromo-4-ethylphenyl
hydroxymethyl



1.5.924
3-methyl-4-ethylphenyl
hydroxymethyl



1.5.925
3,4-diethylphenyl
hydroxymethyl



1.5.926
3-cyclopropyl-4-ethylphenyl
hydroxymethyl



1.5.927
3-cyano-4-ethylphenyl
hydroxymethyl



1.5.928
3-trifluoromethyl-4-ethylphenyl
hydroxymethyl



1.5.929
3-methoxy-4-ethylphenyl
hydroxymethyl



1.5.930
3-ethoxy-4-ethylphenyl
hydroxymethyl



1.5.931
3-trifluoromethoxy-4-ethylphenyl
hydroxymethyl



1.5.932
3-nitro-4-ethylphenyl
hydroxymethyl



1.5.933
3-fluoro-4-propylphenyl
hydroxymethyl



1.5.934
3-chloro-4-propylphenyl
hydroxymethyl



1.5.935
3-bromo-4-propylphenyl
hydroxymethyl



1.5.936
3-methyl-4-propylphenyl
hydroxymethyl



1.5.937
3-cyclopropyl-4-propylphenyl
hydroxymethyl



1.5.938
3-cyano-4-propylphenyl
hydroxymethyl



1.5.939
3-trifluoromethyl-4-propylphenyl
hydroxymethyl



1.5.940
3-methoxy-4-propylphenyl
hydroxymethyl



1.5.941
3-ethoxy-4-propylphenyl
hydroxymethyl



1.5.942
3-trifluoromethoxy-4-propylphenyl
hydroxymethyl



1.5.943
3-nitro-4-propylphenyl
hydroxymethyl



1.5.944
3-fluoro-4-isopropylphenyl
hydroxymethyl



1.5.945
3-chloro-4-isopropylphenyl
hydroxymethyl



1.5.946
3-bromo-4-isopropylphenyl
hydroxymethyl



1.5.947
3-methyl-4-isopropylphenyl
hydroxymethyl



1.5.948
3-cyclopropyl-4-isopropylphenyl
hydroxymethyl



1.5.949
3-cyano-4-isopropylphenyl
hydroxymethyl



1.5.950
3-trifluoromethyl-4-isopropylphenyl
hydroxymethyl



1.5.951
3-methoxy-4-isopropylphenyl
hydroxymethyl



1.5.952
3-ethoxy-4-isopropylphenyl
hydroxymethyl



1.5.953
3-trifluoromethoxy-4-isopropylphenyl
hydroxymethyl



1.5.954
3-nitro-4-isopropylphenyl
hydroxymethyl



1.5.955
3-fluoro-4-tert-butylphenyl
hydroxymethyl



1.5.956
3-chloro-4-tert-butylphenyl
hydroxymethyl



1.5.957
3-bromo-4-tert-butylphenyl
hydroxymethyl



1.5.958
3-methyl-4-tert-butylphenyl
hydroxymethyl



1.5.959
3-cyclopropyl-4-tert-butylphenyl
hydroxymethyl



1.5.960
3-cyano-4-tert-butylphenyl
hydroxymethyl



1.5.961
3-trifluoromethyl-4-tert-butylphenyl
hydroxymethyl



1.5.962
3-trifluoromethyl-4-tert-butylphenyl
1-hydroxyethyl



1.5.963
3-trifluoromethyl-4-tert-butylphenyl
1-hydroxypropyl



1.5.964
3-trifluoromethyl-4-tert-butylphenyl
(1-hydroxy-2-





methylpropyl)



1.5.965
3-trifluoromethyl-4-tert-butylphenyl
methoxymethyl



1.5.966
3-trifluoromethyl-4-tert-butylphenyl
2-methoxyethyl



1.5.967
3-methoxy-4-tert-butylphenyl
hydroxymethyl



1.5.968
3-ethoxy-4-tert-butylphenyl
hydroxymethyl



1.5.969
3-trifluoromethoxy-4-tert-butylphenyl
hydroxymethyl



1.5.970
3-nitro-4-tert-butylphenyl
hydroxymethyl



1.5.971
3-fluoro-4-cyclopropylphenyl
hydroxymethyl



1.5.972
3-chloro-4-cyclopropylphenyl
hydroxymethyl



1.5.973
3-bromo-4-cyclopropylphenyl
hydroxymethyl



1.5.974
3-methyl-4-cyclopropylphenyl
hydroxymethyl



1.5.975
3-cyclopropyl-4-cyclopropylphenyl
hydroxymethyl



1.5.976
3-cyano-4-cyclopropylphenyl
hydroxymethyl



1.5.977
3-trifluoromethyl-4-cyclopropylphenyl
hydroxymethyl



1.5.978
3-methoxy-4-cyclopropylphenyl
hydroxymethyl



1.5.979
3-ethoxy-4-cyclopropylphenyl
hydroxymethyl



1.5.980
3-trifluoromethoxy-4-cyclopropylphenyl
hydroxymethyl



1.5.981
3-fluoro-4-methoxycarbonylphenyl
hydroxymethyl



1.5.982
3-chloro-4-methoxycarbonylphenyl
hydroxymethyl



1.5.983
3-bromo-4-methoxycarbonylphenyl
hydroxymethyl



1.5.984
3-methyl-4-methoxycarbonylphenyl
hydroxymethyl



1.5.985
3-cyclopropyl-4-methoxycarbonylphenyl
hydroxymethyl



1.5.986
3-cyano-4-methoxycarbonylphenyl
hydroxymethyl



1.5.987
3-trifluoromethyl-4-methoxycarbonyl-
hydroxymethyl




phenyl




1.5.988
3-methoxy-4-methoxycarbonylphenyl
hydroxymethyl



1.5.989
3-ethoxy-4-methoxycarbonylphenyl
hydroxymethyl



1.5.990
3-trifluoromethoxy-4-methoxycarbonyl-
hydroxymethyl




phenyl




1.5.991
3-nitro-4-methoxycarbonylphenyl
hydroxymethyl



1.5.992
3-fluoro-4-cyanophenyl
hydroxymethyl



1.5.993
3-chloro-4-cyanophenyl
hydroxymethyl



1.5.994
3-bromo-4-cyanophenyl
hydroxymethyl



1.5.995
3-methyl-4-cyanophenyl
hydroxymethyl



1.5.996
3-cyclopropyl-4-cyanophenyl
hydroxymethyl



1.5.997
3,4-dicyanophenyl
hydroxymethyl



1.5.998
3-trifluoromethyl-4-cyanophenyl
hydroxymethyl



1.5.999
3-trifluoromethyl-4-cyanophenyl
1-hydroxyethyl



1.5.1000
3-trifluoromethyl-4-cyanophenyl
1-hydroxypropyl



1.5.1001
3-trifluoromethyl-4-cyanophenyl
(1-hydroxy-2-





methylpropyl)



1.5.1002
3-trifluoromethyl-4-cyanophenyl
methoxymethyl



1.5.1003
3-trifluoromethyl-4-cyanophenyl
2-methoxyethyl



1.5.1004
3-methoxy-4-cyanophenyl
hydroxymethyl



1.5.1005
3-ethoxy-4-cyanophenyl
hydroxymethyl



1.5.1006
3-trifluoromethoxy-4-cyanophenyl
hydroxymethyl



1.5.1007
3-nitro-4-cyanophenyl
hydroxymethyl



1.5.1008
3-fluoro-4-methoxyphenyl
hydroxymethyl



1.5.1009
3-chloro-4-methoxyphenyl
hydroxymethyl



1.5.1010
3-bromo-4-methoxyphenyl
hydroxymethyl



1.5.1011
3-methyl-4-methoxyphenyl
hydroxymethyl



1.5.1012
3-cyclopropyl-4-methoxyphenyl
hydroxymethyl



1.5.1013
3-cyano-4-methoxyphenyl
hydroxymethyl



1.5.1014
3-trifluoromethyl-4-methoxyphenyl
hydroxymethyl



1.5.1015
3,4-dimethoxyphenyl
hydroxymethyl



1.5.1016
3-ethoxy-4-methoxyphenyl
hydroxymethyl



1.5.1017
3-trifluoromethoxy-4-methoxyphenyl
hydroxymethyl



1.5.1018
3-nitro-4-methoxyphenyl
hydroxymethyl



1.5.1019
3-fluoro-4-ethoxyphenyl
hydroxymethyl



1.5.1020
3-chloro-4-ethoxyphenyl
hydroxymethyl



1.5.1021
3-chloro-4-ethoxyphenyl
1-hydroxyethyl



1.5.1022
3-chloro-4-ethoxyphenyl
1-hydroxypropyl



1.5.1023
3-chloro-4-ethoxyphenyl
(1-hydroxy-2-





methylpropyl)



1.5.1024
3-chloro-4-ethoxyphenyl
methoxymethyl



1.5.1025
3-chloro-4-ethoxyphenyl
2-methoxyethyl



1.5.1026
3-bromo-4-ethoxyphenyl
hydroxymethyl



1.5.1027
3-methyl-4-ethoxyphenyl
hydroxymethyl



1.5.1028
3-ethyl-4-ethoxyphenyl
hydroxymethyl



1.5.1029
3-cyclopropyl-4-ethoxyphenyl
hydroxymethyl



1.5.1030
3-cyano-4-ethoxyphenyl
hydroxymethyl



1.5.1031
3-trifluoromethyl-4-ethoxyphenyl
hydroxymethyl



1.5.1032
3-methoxy-4-ethoxyphenyl
hydroxymethyl



1.5.1033
2,4-diethoxyphenyl
hydroxymethyl



1.5.1034
3-trifluoromethoxy-4-ethoxyphenyl
hydroxymethyl



1.5.1035
3-nitro-4-ethoxyphenyl
hydroxymethyl



1.5.1036
3-fluoro-4-isopropoxyphenyl
hydroxymethyl



1.5.1037
3-chloro-4-isopropoxyphenyl
hydroxymethyl



1.5.1038
3-bromo-4-isopropoxyphenyl
hydroxymethyl



1.5.1039
3-methyl-4-isopropoxyphenyl
hydroxymethyl



1.5.1040
3-cyclopropyl-4-isopropoxyphenyl
hydroxymethyl



1.5.1041
3-cyano-4-isopropoxyphenyl
hydroxymethyl



1.5.1042
3-trifluoromethyl-4-isopropoxyphenyl
hydroxymethyl



1.5.1043
3-methoxy-4-isopropoxyphenyl
hydroxymethyl



1.5.1044
3-ethoxy-4-isopropoxyphenyl
hydroxymethyl



1.5.1045
3-trifluoromethoxy-4-isopropoxyphenyl
hydroxymethyl



1.5.1046
3-nitro-4-isopropoxyphenyl
hydroxymethyl



1.5.1047
3-fluoro-4-trifluoromethoxyphenyl
hydroxymethyl



1.5.1048
3-chloro-4-trifluoromethoxyphenyl
hydroxymethyl



1.5.1049
3-bromo-4-trifluoromethoxyphenyl
hydroxymethyl



1.5.1050
3-methyl-4-trifluoromethoxyphenyl
hydroxymethyl



1.5.1051
3-cyclopropyl-4-trifluoromethoxyphenyl
hydroxymethyl



1.5.1052
3-cyano-4-trifluoromethoxyphenyl
hydroxymethyl



1.5.1053
3-trifluoromethyl-4-trifluoromethoxy-
hydroxymethyl




phenyl




1.5.1054
3-methoxy-4-trifluoromethoxyphenyl
hydroxymethyl



1.5.1055
3-ethoxy-4-trifluoromethoxyphenyl
hydroxymethyl



1.5.1056
3,4-bis(trifluoromethoxy)phenyl
hydroxymethyl



1.5.1057
3-nitro-4-trifluoromethoxyphenyl
hydroxymethyl



1.5.1058
3-fluoro-4-difluoromethoxyphenyl
hydroxymethyl



1.5.1059
3-chloro-4-difluoromethoxyphenyl
hydroxymethyl



1.5.1060
3-bromo-4-difluoromethoxyphenyl
hydroxymethyl



1.5.1061
3-methyl-4-difluoromethoxyphenyl
hydroxymethyl



1.5.1062
3-cyclopropyl-4-difluoromethoxyphenyl
hydroxymethyl



1.5.1063
3-cyano-4-difluoromethoxyphenyl
hydroxymethyl



1.5.1064
3-trifluoromethyl-4-difluoromethoxy-
hydroxymethyl




phenyl




1.5.1065
3-methoxy-4-difluoromethoxyphenyl
hydroxymethyl



1.5.1066
3-ethoxy-4-difluoromethoxyphenyl
hydroxymethyl



1.5.1067
3-trifluoromethoxy-4-difluoromethoxy-
hydroxymethyl




phenyl




1.5.1068
3-nitro-4-difluoromethoxyphenyl
hydroxymethyl



1.5.1069
3-fluoro-4-nitrophenyl
hydroxymethyl



1.5.1070
3-chloro-4-nitrophenyl
hydroxymethyl



1.5.1071
3-bromo-4-nitrophenyl
hydroxymethyl



1.5.1072
3-methyl-4-nitrophenyl
hydroxymethyl



1.5.1073
3-cyclopropyl-4-nitrophenyl
hydroxymethyl



1.5.1074
3-cyano-4-nitrophenyl
hydroxymethyl



1.5.1075
3-trifluoromethyl-4-nitrophenyl
hydroxymethyl



1.5.1076
3-methoxy-4-nitrophenyl
hydroxymethyl



1.5.1077
3-ethoxy-4-nitrophenyl
hydroxymethyl



1.5.1078
3-trifluoromethoxy-4-nitrophenyl
hydroxymethyl



1.5.1079
3-fluoro-4-methylsulfanylphenyl
hydroxymethyl



1.5.1080
3-chloro-4-methylsulfanylphenyl
hydroxymethyl



1.5.1081
3-bromo-4-methylsulfanylphenyl
hydroxymethyl



1.5.1082
3-methyl-4-methylsulfanylphenyl
hydroxymethyl



1.5.1083
3-cyclopropyl-4-methylsulfanylphenyl
hydroxymethyl



1.5.1084
3-cyano-4-methylsulfanylphenyl
hydroxymethyl



1.5.1085
3-trifluoromethyl-4-methylsulfanylphenyl
hydroxymethyl



1.5.1086
3-methoxy-4-methylsulfanylphenyl
hydroxymethyl



1.5.1087
3-ethoxy-4-methylsulfanylphenyl
hydroxymethyl



1.5.1088
3-trifluoromethoxy-4-
hydroxymethyl




methylsulfanylphenyl




1.5.1089
3-nitro-4-methylsulfanylphenyl
hydroxymethyl



1.5.1090
3,6-difluorophenyl
hydroxymethyl



1.5.1091
3,6-difluorophenyl
1-hydroxyethyl



1.5.1092
3,6-difluorophenyl
1-hydroxypropyl



1.5.1093
3,6-difluorophenyl
(1-hydroxy-2-





methylpropyl)



1.5.1094
3,6-difluorophenyl
methoxymethyl



1.5.1095
3,6-difluorophenyl
2-methoxyethyl



1.5.1096
3-chloro-6-fluorophenyl
hydroxymethyl



1.5.1097
3-bromo-6-fluorophenyl
hydroxymethyl



1.5.1098
3-methyl-6-fluorophenyl
hydroxymethyl



1.5.1099
3-ethyl-6-fluorophenyl
hydroxymethyl



1.5.1100
3-cyclopropyl-6-fluorophenyl
hydroxymethyl



1.5.1101
3-cyano-6-fluorophenyl
hydroxymethyl



1.5.1102
3-methoxy-6-fluorophenyl
hydroxymethyl



1.5.1103
3-ethoxy-6-fluorophenyl
hydroxymethyl



1.5.1104
3-trifluoromethoxy-6-fluorophenyl
hydroxymethyl



1.5.1105
3-nitro-6-fluorophenyl
hydroxymethyl



1.5.1106
3-fluoro-6-chlorophenyl
hydroxymethyl



1.5.1107
3-fluoro-6-chlorophenyl
1-hydroxyethyl



1.5.1108
3-fluoro-6-chlorophenyl
1-hydroxypropyl



1.5.1109
3-fluoro-6-chlorophenyl
(1-hydroxy-2-





methylpropyl)



1.5.1110
3-fluoro-6-chlorophenyl
methoxymethyl



1.5.1111
3-fluoro-6-chlorophenyl
2-methoxyethyl



1.5.1112
3,6-dichlorophenyl
hydroxymethyl



1.5.1113
3,6-dichlorophenyl
1-hydroxyethyl



1.5.1114
3,6-dichlorophenyl
1-hydroxypropyl



1.5.1115
3,6-dichlorophenyl
(1-hydroxy-2-





methylpropyl)



1.5.1116
3,6-dichlorophenyl
methoxymethyl



1.5.1117
3,6-dichlorophenyl
2-methoxyethyl



1.5.1118
3-bromo-6-chlorophenyl
hydroxymethyl



1.5.1119
3-methyl-6-chlorophenyl
hydroxymethyl



1.5.1120
3-cyclopropyl-6-chlorophenyl
hydroxymethyl



1.5.1121
3-cyano-6-chlorophenyl
hydroxymethyl



1.5.1122
3-trifluoromethyl-6-chlorophenyl
hydroxymethyl



1.5.1123
3-methoxy-6-chlorophenyl
hydroxymethyl



1.5.1124
3-ethoxy-6-chlorophenyl
hydroxymethyl



1.5.1125
3-trifluoromethoxy-6-chlorophenyl
hydroxymethyl



1.5.1126
3-nitro-6-chlorophenyl
hydroxymethyl



1.5.1127
3-fluoro-6-bromophenyl
hydroxymethyl



1.5.1128
3-chloro-6-bromophenyl
hydroxymethyl



1.5.1129
3,6-dibromophenyl
hydroxymethyl



1.5.1130
3-methyl-6-bromophenyl
hydroxymethyl



1.5.1131
3-cyclopropyl-6-bromophenyl
hydroxymethyl



1.5.1132
3-cyano-6-bromophenyl
hydroxymethyl



1.5.1133
3-trifluoromethyl-6-bromophenyl
hydroxymethyl



1.5.1134
3-methoxy-6-phenyl
hydroxymethyl



1.5.1135
3-ethoxy-6-bromophenyl
hydroxymethyl



1.5.1136
3-trifluoromethoxy-6-bromophenyl
hydroxymethyl



1.5.1137
3-nitro-6-bromophenyl
hydroxymethyl



1.5.1138
3-fluoro-6-iodophenyl
hydroxymethyl



1.5.1139
3-chloro-6-iodophenyl
hydroxymethyl



1.5.1140
3-bromo-6-iodophenyl
hydroxymethyl



1.5.1141
3-methyl-6-iodophenyl
hydroxymethyl



1.5.1142
3-cyclopropyl-6-iodophenyl
hydroxymethyl



1.5.1143
3-cyano-6-iodophenyl
hydroxymethyl



1.5.1144
3-trifluoromethyl-6-iodophenyl
hydroxymethyl



1.5.1145
3-methoxy-6-iodophenyl
hydroxymethyl



1.5.1146
3-ethoxy-6-iodophenyl
hydroxymethyl



1.5.1147
3-trifluoromethoxy-6-iodophenyl
hydroxymethyl



1.5.1148
3-nitro-6-iodophenyl
hydroxymethyl



1.5.1149
3-fluoro-6-methylphenyl
hydroxymethyl



1.5.1150
3-chloro-6-methylphenyl
hydroxymethyl



1.5.1151
3-bromo-6-methylphenyl
hydroxymethyl



1.5.1152
3,6-dimethylphenyl
hydroxymethyl



1.5.1153
3-ethyl-6-methylphenyl
hydroxymethyl



1.5.1154
3-cyclopropyl-6-methylphenyl
hydroxymethyl



1.5.1155
3-cyano-6-methylphenyl
hydroxymethyl



1.5.1156
3-trifluoromethyl-6-methylphenyl
hydroxymethyl



1.5.1157
3-methoxy-6-methylphenyl
hydroxymethyl



1.5.1158
3-ethoxy-6-methylphenyl
hydroxymethyl



1.5.1159
3-trifluoromethoxy-6-methylphenyl
hydroxymethyl



1.5.1160
3-nitro-6-methylphenyl
hydroxymethyl



1.5.1161
3-fluoro-6-ethylphenyl
hydroxymethyl



1.5.1162
3-chloro-6-ethylphenyl
hydroxymethyl



1.5.1163
3-bromo-6-ethylphenyl
hydroxymethyl



1.5.1164
3-methyl-6-ethylphenyl
hydroxymethyl



1.5.1165
3,6-diethylphenyl
hydroxymethyl



1.5.1166
3-cyclopropyl-6-ethylphenyl
hydroxymethyl



1.5.1167
3-cyano-6-ethylphenyl
hydroxymethyl



1.5.1168
3-trifluoromethyl-6-ethylphenyl
hydroxymethyl



1.5.1169
3-methoxy-6-ethylphenyl
hydroxymethyl



1.5.1170
3-ethoxy-6-ethylphenyl
hydroxymethyl



1.5.1171
3-trifluoromethoxy-6-ethylphenyl
hydroxymethyl



1.5.1172
3-nitro-6-ethylphenyl
hydroxymethyl



1.5.1173
3-fluoro-6-propylphenyl
hydroxymethyl



1.5.1174
3-chloro-6-propylphenyl
hydroxymethyl



1.5.1175
3-bromo-6-propylphenyl
hydroxymethyl



1.5.1176
3-methyl-6-propylphenyl
hydroxymethyl



1.5.1177
3-methyl-6-propylphenyl
hydroxymethyl



1.5.1178
3-cyclopropyl-6-propylphenyl
hydroxymethyl



1.5.1179
3-cyano-6-propylphenyl
hydroxymethyl



1.5.1180
3-trifluoromethyl-6-propylphenyl
hydroxymethyl



1.5.1181
3-methoxy-6-propylphenyl
hydroxymethyl



1.5.1182
3-ethoxy-6-propylphenyl
hydroxymethyl



1.5.1183
3-trifluoromethoxy-6-propylphenyl
hydroxymethyl



1.5.1184
3-nitro-6-propylphenyl
hydroxymethyl



1.5.1185
3-fluoro-6-isopropylphenyl
hydroxymethyl



1.5.1186
3-chloro-6-isopropylphenyl
hydroxymethyl



1.5.1187
3-bromo-6-isopropylphenyl
hydroxymethyl



1.5.1188
3-methyl-6-isopropylphenyl
hydroxymethyl



1.5.1189
3-cyclopropyl-6-isopropylphenyl
hydroxymethyl



1.5.1190
3-cyano-6-isopropylphenyl
hydroxymethyl



1.5.1191
3-trifluoromethyl-6-isopropylphenyl
hydroxymethyl



1.5.1192
3-ethoxy-6-isopropylphenyl
hydroxymethyl



1.5.1193
3-trifluoromethoxy-6-isopropylphenyl
hydroxymethyl



1.5.1194
3-nitro-6-isopropylphenyl
hydroxymethyl



1.5.1195
3-fluoro-6-tert-butylphenyl
hydroxymethyl



1.5.1196
3-chloro-6-tert-butylphenyl
hydroxymethyl



1.5.1197
3-bromo-6-tert-butylphenyl
hydroxymethyl



1.5.1198
3-methyl-6-tert-butylphenyl
hydroxymethyl



1.5.1199
3-cyclopropyl-6-tert-butylphenyl
hydroxymethyl



1.5.1200
3-cyano-6-tert-butylphenyl
hydroxymethyl



1.5.1201
3-trifluoromethyl-6-tert-butylphenyl
hydroxymethyl



1.5.1202
3-methoxy-6-tert-butylphenyl
hydroxymethyl



1.5.1203
3-ethoxy-6-tert-butylphenyl
hydroxymethyl



1.5.1204
3-trifluoromethoxy-6-tert-butylphenyl
hydroxymethyl



1.5.1205
3-nitro-6-tert-butylphenyl
hydroxymethyl



1.5.1206
3-fluoro-6-cyclopropylphenyl
hydroxymethyl



1.5.1207
3-chloro-6-cyclopropylphenyl
hydroxymethyl



1.5.1208
3-bromo-6-cyclopropylphenyl
hydroxymethyl



1.5.1209
3-methyl-6-cyclopropylphenyl
hydroxymethyl



1.5.1210
3-cyclopropyl-6-cyclopropyl phenyl
hydroxymethyl



1.5.1211
3-cyano-6-cyclopropylphenyl
hydroxymethyl



1.5.1212
3-trifluoromethyl-6-cyclopropylphenyl
hydroxymethyl



1.5.1213
3-methoxy-6-cyclopropylphenyl
hydroxymethyl



1.5.1214
3-ethoxy-6-cyclopropylphenyl
hydroxymethyl



1.5.1215
3-trifluoromethoxy-6-cyclopropylphenyl
hydroxymethyl



1.5.1216
3-fluoro-6-methoxycarbonylphenyl
hydroxymethyl



1.5.1217
3-chloro-6-methoxycarbonylphenyl
hydroxymethyl



1.5.1218
3-bromo-6-methoxycarbonylphenyl
hydroxymethyl



1.5.1219
3-methyl-6-methoxycarbonylphenyl
hydroxymethyl



1.5.1220
3-cyclopropyl-6-methoxycarbonylphenyl
hydroxymethyl



1.5.1221
3-cyano-6-methoxycarbonylphenyl
hydroxymethyl



1.5.1222
3-trifluoromethyl-6-methoxycarbonyl-
hydroxymethyl




phenyl




1.5.1223
3-methoxy-6-methoxycarbonylphenyl
hydroxymethyl



1.5.1224
3-ethoxy-6-methoxycarbonylphenyl
hydroxymethyl



1.5.1225
3-trifluoromethoxy-6-methoxycarbonyl-
hydroxymethyl




phenyl




1.5.1226
3-nitro-6-methoxycarbonylphenyl
hydroxymethyl



1.5.1227
3-fluoro-6-cyanophenyl
hydroxymethyl



1.5.1228
3-chloro-6-cyanophenyl
hydroxymethyl



1.5.1229
3-bromo-6-cyanophenyl
hydroxymethyl



1.5.1230
3-methyl-6-cyanophenyl
hydroxymethyl



1.5.1231
3-cyclopropyl-6-cyanophenyl
hydroxymethyl



1.5.1232
3-cyano-6-cyanophenyl
hydroxymethyl



1.5.1233
3-trifluoromethyl-6-cyanophenyl
hydroxymethyl



1.5.1234
3-methoxy-6-cyanophenyl
hydroxymethyl



1.5.1235
3-ethoxy-6-cyanophenyl
hydroxymethyl



1.5.1236
3-trifluoromethoxy-6-cyanophenyl
hydroxymethyl



1.5.1237
3-nitro-6-cyanophenyl
hydroxymethyl



1.5.1238
3-fluoro-6-methoxyphenyl
hydroxymethyl



1.5.1239
3-chloro-6-methoxyphenyl
hydroxymethyl



1.5.1240
3-bromo-6-methoxyphenyl
hydroxymethyl



1.5.1241
3-methyl-6-methoxyphenyl
hydroxymethyl



1.5.1242
3-cyclopropyl-6-methoxyphenyl
hydroxymethyl



1.5.1243
3-cyano-6-methoxyphenyl
hydroxymethyl



1.5.1244
3-trifluoromethyl-6-methoxyphenyl
hydroxymethyl



1.5.1245
3,6-dimethoxyphenyl
hydroxymethyl



1.5.1246
3-ethoxy-6-methoxyphenyl
hydroxymethyl



1.5.1247
3-trifluoromethoxy-6-methoxyphenyl
hydroxymethyl



1.5.1248
3-nitro-6-methoxyphenyl
hydroxymethyl



1.5.1249
3-fluoro-6-ethoxyphenyl
hydroxymethyl



1.5.1250
3-chloro-6-ethoxyphenyl
hydroxymethyl



1.5.1251
3-bromo-6-ethoxyphenyl
hydroxymethyl



1.5.1252
3-methyl-6-ethoxyphenyl
hydroxymethyl



1.5.1253
3-cyclopropyl-6-ethoxyphenyl
hydroxymethyl



1.5.1254
3-cyano-6-ethoxyphenyl
hydroxymethyl



1.5.1255
3-trifluoromethyl-6-ethoxyphenyl
hydroxymethyl



1.5.1256
3-methoxy-6-ethoxyphenyl
hydroxymethyl



1.5.1257
2,6-diethoxyphenyl
hydroxymethyl



1.5.1258
3-trifluoromethoxy-6-ethoxyphenyl
hydroxymethyl



1.5.1259
3-nitro-6-ethoxyphenyl
hydroxymethyl



1.5.1260
3-fluoro-6-isopropoxyphenyl
hydroxymethyl



1.5.1261
3-chloro-6-isopropoxyphenyl
hydroxymethyl



1.5.1262
3-bromo-6-isopropoxyphenyl
hydroxymethyl



1.5.1263
3-methyl-6-isopropoxyphenyl
hydroxymethyl



1.5.1264
3-cyclopropyl-6-isopropoxyphenyl
hydroxymethyl



1.5.1265
3-cyano-6-isopropoxyphenyl
hydroxymethyl



1.5.1266
3-trifluoromethyl-6-isopropoxyphenyl
hydroxymethyl



1.5.1267
3-methoxy-6-isopropoxyphenyl
hydroxymethyl



1.5.1268
3-ethoxy-6-isopropoxyphenyl
hydroxymethyl



1.5.1269
3-trifluoromethoxy-6-isopropoxyphenyl
hydroxymethyl



1.5.1270
3-nitro-6-isopropoxyphenyl
hydroxymethyl



1.5.1271
3-fluoro-6-trifluoromethoxyphenyl
hydroxymethyl



1.5.1272
3-chloro-6-trifluoromethoxyphenyl
hydroxymethyl



1.5.1273
3-bromo-6-trifluoromethoxyphenyl
hydroxymethyl



1.5.1274
3-methyl-6-trifluoromethoxyphenyl
hydroxymethyl



1.5.1275
3-cyclopropyl-6-trifluoromethoxyphenyl
hydroxymethyl



1.5.1276
3-cyano-6-trifluoromethoxyphenyl
hydroxymethyl



1.5.1277
3-trifluoromethyl-6-trifluoromethoxy-
hydroxymethyl




phenyl




1.5.1278
3-methoxy-6-trifluoromethoxyphenyl
hydroxymethyl



1.5.1279
3-ethoxy-6-trifluoromethoxyphenyl
hydroxymethyl



1.5.1280
3,6-bis(trifluoromethoxy)phenyl
hydroxymethyl



1.5.1281
3-nitro-6-trifluoromethoxyphenyl
hydroxymethyl



1.5.1282
3-fluoro-6-difluoromethoxyphenyl
hydroxymethyl



1.5.1283
3-chloro-6-difluoromethoxyphenyl
hydroxymethyl



1.5.1284
3-bromo-6-difluoromethoxyphenyl
hydroxymethyl



1.5.1285
3-methyl-6-difluoromethoxyphenyl
hydroxymethyl



1.5.1286
3-cyclopropyl-6-difluoromethoxyphenyl
hydroxymethyl



1.5.1287
3-cyano-6-difluoromethoxyphenyl
hydroxymethyl



1.5.1288
3-trifluoromethyl-6-difluoromethoxy-
hydroxymethyl




phenyl




1.5.1289
3-methoxy-6-difluoromethoxyphenyl
hydroxymethyl



1.5.1290
3-ethoxy-6-difluoromethoxyphenyl
hydroxymethyl



1.5.1291
3-trifluoromethoxy-6-difluoromethoxy-
hydroxymethyl




phenyl




1.5.1292
3-nitro-6-difluoromethoxyphenyl
hydroxymethyl



1.5.1293
3-fluoro-6-nitrophenyl
hydroxymethyl



1.5.1294
3-chloro-6-nitrophenyl
hydroxymethyl



1.5.1295
3-bromo-6-nitrophenyl
hydroxymethyl



1.5.1296
3-methyl-6-nitrophenyl
hydroxymethyl



1.5.1297
3-cyclopropyl-6-nitrophenyl
hydroxymethyl



1.5.1298
3-cyano-6-nitrophenyl
hydroxymethyl



1.5.1299
3-trifluoromethyl-6-nitrophenyl
hydroxymethyl



1.5.1300
3-methoxy-6-nitrophenyl
hydroxymethyl



1.5.1301
3-ethoxy-6-nitrophenyl
hydroxymethyl



1.5.1302
3-trifluoromethoxy-6-nitrophenyl
hydroxymethyl



1.5.1303
3-fluoro-6-methylsulfanylphenyl
hydroxymethyl



1.5.1304
3-chloro-6-methylsulfanylphenyl
hydroxymethyl



1.5.1305
3-bromo-6-methylsulfanylphenyl
hydroxymethyl



1.5.1306
3-methyl-6-methylsulfanylphenyl
hydroxymethyl



1.5.1307
3-cyclopropyl-6-methylsulfanylphenyl
hydroxymethyl



1.5.1308
3-cyano-6-methylsulfanylphenyl
hydroxymethyl



1.5.1309
3-trifluoromethyl-6-methylsulfanylphenyl
hydroxymethyl



1.5.1310
3-methoxy-6-methylsulfanylphenyl
hydroxymethyl



1.5.1311
3-ethoxy-6-methylsulfanylphenyl
hydroxymethyl



1.5.1312
3-trifluoromethoxy-6-
hydroxymethyl




methylsulfanylphenyl




1.5.1313
3-nitro-6-methylsulfanylphenyl
hydroxymethyl



1.5.1314
2,3,4-trifluorophenyl
hydroxymethyl



1.5.1315
2,3,4-trichlorophenyl
hydroxymethyl



1.5.1316
2,3,4-trimethylphenyl
hydroxymethyl



1.5.1317
2-fluoro-2-chloro-5-trifluoromethylphenyl
hydroxymethyl



1.5.1318
2,3,5-trifluorophenyl
hydroxymethyl



1.5.1319
2,3,5-trichlorophenyl
hydroxymethyl



1.5.1320
2,3,5-trimethylphenyl
hydroxymethyl



1.5.1321
2,3-dichloro-5-methoxyphenyl
hydroxymethyl



1.5.1322
2,3,6-trifluorophenyl
hydroxymethyl



1.5.1323
2,3,6-trichlorophenyl
hydroxymethyl



1.5.1324
2,3,6-trimethylphenyl
hydroxymethyl



1.5.1325
3,4,5-trifluorophenyl
hydroxymethyl



1.5.1326
3,4,5-trichlorophenyl
hydroxymethyl



1.5.1327
3,4,5-trimethylphenyl
hydroxymethyl



1.5.1328
3,5-dimethyl-4-fluorophenyl
hydroxymethyl



1.5.1329
3,5-dichloro-4-methoxyphenyl
hydroxymethyl



1.5.1330
3,5-difluoro-4-chlorophenyl
hydroxymethyl



1.5.1331
3,5-dichloro-4-hydroxyphenyl
hydroxymethyl



1.5.1332
3,5-trifluoromethyl-4-chlorophenyl
hydroxymethyl



1.5.1333
3,4,6-trifluorophenyl
hydroxymethyl



1.5.1334
3,4,6-trichlorophenyl
hydroxymethyl



1.5.1335
3,4,6-trimethylphenyl
hydroxymethyl



1.5.1336
pentafluorophenyl
hydroxymethyl
















TABLE 2.1







Inventive compounds of the general formula (I) in which W* is COOY, R1 is hydrogen, and aryl is the radical.








 








 












No.
Aryl
R2
R3
Y
Physical data





2.1.1
3-fluorophenyl
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.71 (s,







3H); 3.6 (d, 1H); 3.85 (d, 1H);







4.25 (m, 2H); 7.10 (m, 1H); 7.40







(m, 2H).


2.1.2
3-fluorophenyl
H
ethyl
ethyl
[CDCl3] 1.00 (t, 3H); 1.31 (t, 3H);







2.05 (m, 2H); 3.20 (d, 1H); 3.80







(d, 1H); 4.25 (m, 2H); 7.11 (m,







1H); 7.40 (m, 3H).


2.1.3
3-fluorophenyl
H
propyl
ethyl



2.1.4
3-fluorophenyl
H
cyclo-
ethyl






propyl




2.1.5
3-chlorophenyl
H
methyl
ethyl
[CDCl3] 1.30 (t, 3H); 1.70 (s,







3H); 3.17 (d, 1H); 3.85 (d, 1H);







4.25 (m, 2H); 7.35 (m, 2H); 7.55







(dd, 1H); 7.65 (s, 1H).


2.1.6
3-chlorophenyl
H
ethyl
ethyl



2.1.7
3-chlorophenyl
H
propyl
ethyl



2.1.8
3-chlorophenyl
H
cyclo-
ethyl






propyl




2.1.9
3-bromophenyl
H
methyl
methyl



2.1.10
3-bromophenyl
H
ethyl
ethyl



2.1.11
3-iodophenyl
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.69 (s,







3H); 3.16 (d, 1H); 3.83 (d, 1H);







4.25 (m, 2H); 7.12 (t, 1H); 7.62







(dd, 1H); 7.73 (dd, H); 7.98 d,







1H).


2.1.12
3-iodophenyl
H
ethyl
ethyl



2.1.13
3-methylphenyl
H
methyl
ethyl
[CDCl3] 1.30 (t, 3H); 1.70 (s,







3H); 2.36 (s, 3H); 3.20 (d, 1H);







3.88 (d, 1H); 4.25 (m, 2H); 7.25







(mc; 2H); 7.42 (d, 1H); 7.50 (bs,







1H).


2.1.14
3-methylphenyl
H
ethyl
ethyl



2.1.15
3-ethylphenyl
H
methyl
ethyl
[CDCl3] 1.22 (t, 3H); 1.31 (t, 3H);







1.70 (s, 3H); 2.65 (q, 2H); 3.20







(d, 1H); 3.90 (d, 1H); 4.25 (m,







2H); 7.25 (m, 1H); 7.31 (t, 1H);







7.42 (d, 1H); 7.58 (bs, 1H).


2.1.16
3-propylphenyl
H
methyl
ethyl



2.1.17
3-isopropyl-
H
methyl
ethyl
[CDCl3] 1.22 (d, 6H); 1.31 (t,



phenyl



3H); 2.91 (m, 1H); 3.21 (d, 1H);







3.91 (d, 1H); 4.25 (m, 2H); 7.28







(m, 1H); 7.32 t, 1H); 7.41 (d,







1H); 7.58 (bs, 1H).


2.1.18
3-n-butylphenyl
H
methyl
ethyl



2.1.19
3-i-butylphenyl
H
methyl
ethyl



2.1.20
3-tert-
H
methyl
ethyl




butylphenyl






2.1.21
3-cyclopropyl-
H
methyl
ethyl




phenyl






2.1.22
3-cyclobutyl-
H
methyl
ethyl




phenyl






2.1.23
3-cyclopentyl-
H
methyl
ethyl




phenyl






2.1.24
3-vinylphenyl
H
methyl
ethyl



2.1.25
3-ethynylphenyl
H
methyl
ethyl



2.1.26
3-cyanophenyl
H
methyl
ethyl
[CDCl3] 1.30 (t, 3H); 1.71 (s,







3H); 3.18 (d, 1H); 3.90 (d, 1H);







4.25 (m, 2H); 7.52 (m, 1H); 7.68







(m, 1H); 7.91 (m, 2H).


2.1.27
3-trifluoro-
H
methyl
ethyl
[CDCl3] 1.32 (t, 3H); 1.71 (s,



methylphenyl



3H); 3.21 (d, 1H); 3.91 (m, 2H);







7.53 (t, 1H); 7.68 (d, 1H); 7.88







(m, 2H).


2.1.28
3-difluoro-
H
methyl
ethyl




methylphenyl






2.1.29
3-(hydroxy-
H
methyl
ethyl




carbonyl)phenyl






2.1.30
3-(methoxy-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.72 (s,



carbonyl)phenyl



3H); 3.26 (d, 1H); 3.91 (d, 1H);







3.96 (s, 3H); 4.25 (m, 2H); 7.50







(m, 1H); 7.96 (d, 1H); 8.10 (d,







1H); 8.21 (s, 1H).


2.1.31
3-(ethoxy-
H
methyl
ethyl




carbonyl)phenyl






2.1.32
3-hydroxy-
H
methyl
ethyl




methylphenyl






2.1.33
3-acetylphenyl
H
methyl
ethyl
[CDCl3] 1.32 (t, 3H); 1.72 (s,







3H); 2.63 (s, 3H); 3.24 (d, 1H);







3.93 (d, 1H); 4.25 (q, 2H); 7.52







/t, 1H); 7.90 (d, 1H); 8.0 (d, 1H);







8.20 (s, 1H).


2.1.34
3-carbamoyl-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.70 (s,



phenyl



3H); 3.21 (d, 1H); 3.86 (d, 1h),







4.25 (dq; 2H); 6.52 (bs, 1H);







7.28-7.42 (m, 3H); 7.70 (s, 1H).


2.1.35
3-hydroxyphenyl
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.70 (s,







3H); 3.21 (d, 1H); 3.85 (d, 1H);







4.26 (m, 2H); 5.70 (bs, 1H); 6.92







(dd, 1H); 7.15 (d, 1H); 7.28 (m,







2H).


2.1.36
3-methoxy-
H
methyl
ethyl
[DMSO] 1.21 (t, 3H); 1.59 (s,



phenyl



3H); 3.25-3.45 (m, 2H); 3.80 (s,







3H); 4.15 (q, 2H); 7.05 (m, 1H);







7.22 (m, 2H); 7.48 (m, 1H).


2.1.37
3-ethoxyphenyl
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.42 (t, 3H);







1.70 (s, 3H); 3.20 (d, 1H); 3.88







(d, 3H); 4.08 (q, 2H); 4.25 (m,







2H); 6.95 (dd, 1H); 7.15 (dd,







1H); 7.31 (mc, 2H).


2.1.38
3-propyloxy-
H
methyl
ethyl




phenyl






2.1.39
3-isopropyloxy-
H
methyl
ethyl
[CDCl3] 1.31 (m, 9H); 1.70 (s,



phenyl



3H); 3.19 (d, 1H); 3.87 (d, 1H);







4.25 (m, 2H); 4.58 (m, 1H); 6.92







(dd, 1H); 7.15 (d, 1H); 7.29 (mc,







2H).


2.1.40
3-n-
H
methyl
ethyl




butyloxyphenyl






2.1.41
3-i-
H
methyl
ethyl




butyloxyphenyl






2.1.42
3-t-
H
methyl
ethyl




butyloxyphenyl






2.1.43
3-difluoro-
H
methyl
ethyl
[CDCl3] 1.30 (t, 3H); 1.71 (s,



methoxyphenyl



3H); 3.2 (d, 1H); 3.89 (d, 1H);







4.25 (m, 2H); 6.51 (t, 3H); 7.19







(d, 1H); 7.43 (m, 3H).


2.1.44
3-trifluoro-
H
methyl
ethyl
[CDCl3] 1.31 /t, 3H); 1.71 (s,



methoxyphenyl



3H); 3.20 (d, 1H); 3.91 (d, 1H);







4.25 (m, 2H); 2.25 (d, 1H); 7.42







(t, 1H); 7.55 (mc, 2H).


2.1.45
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







phenyl






2.1.46
3-(2-chloro-
H
methyl
ethyl




ethoxy)phenyl






2.1.47
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)phenyl






2.1.48
3-(2-methoxy-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.70 (s,



ethoxy)phenyl



3H), 3.16 (d, 1H); 3.45 (s, 3H);







3.75 (dd, 2H); 3.85 (d, 1H); 4.13







(dd, 2H); 4.25 (m, 2H); 7.00 (dd,







1H); 7.20 (d, 1H); 7.30 (mc, 2H).


2.1.49
3-[(tert-butoxy-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.58 (s,



carbonyl)oxy]-



9H); 1.70 (s, 3H); 3.17 (d, 1H);



phenyl



3.82 (d, 1H); 4.25 (q, 2H); 7.22







(dd, 1H); 7.40 (t, 1H); 7.50 (mc,







2H).


2.1.50
3-nitrophenyl
H
methyl
ethyl
[CDCl3] 1.32 (t, 3H); 1.72 (s,







3H); 3.25 (d, 1H); 3.95 (d, 1H);







4.30 (m, 2H); 7.60 (t, 1H); 8.07







(dd, 1H); 8.26 (dd, 1H); 8.41 (d,







1H).


2.1.51
3-acetoxyphenyl
H
methyl
ethyl
[CDCl3] 1.30 (t, 3H); 1.71 (s,







3H); 2.30 (s, 3H); 3.18 (d, 1H);







3.85 (d, 1H); 4.25 (m, 2H); 7.15







(dd, 1H); 7.40 (mc, 2H); 7.51







(dd, 1H).


2.1.52
{3-[(tert-
H
methyl
ethyl




butoxycarbonyl)







amino]phenyl}






2.1.53
3-methyl-
H
methyl
ethyl




sulfanylphenyl






2.1.54
3-ethyl-
H
methyl
ethyl




sulfanylphenyl






2.1.55
3-(pentafluoro-
H
methyl
ethyl




lambda6-







sulfanyl)phenyl






2.1.56
2,3-difluoro-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.72 (s,



phenyl



3H); 3.33 (d, 1H); 3.95 (d, 1H);







4.36 (q, 2H); 7.12 (m, 1H); 7.23







(m, 1H); 7.53 (m, 1H).


2.1.57
2,3-difluoro-
H
ethyl
ethyl




phenyl






2.1.58
2,3-difluoro-
H
propyl
ethyl




phenyl






2.1.59
2,3-difluoro-
H
cyclo-
ethyl




phenyl

propyl




2.1.60
2-chloro-3-
H
methyl
ethyl




fluorophenyl






2.1.61
2-bromo-3-
H
methyl
ethyl




fluorophenyl






2.1.62
2-methyl-3-
H
methyl
ethyl




fluorophenyl






2.1.63
2-ethyl-3-
H
methyl
ethyl




fluorophenyl






2.1.64
2-cyclopropyl-3-
H
methyl
ethyl




fluorophenyl






2.1.65
2-vinyl-3-
H
methyl
ethyl




fluorophenyl






2.1.66
2-ethynyl-3-
H
methyl
ethyl




fluorophenyl






2.1.67
2-cyano-3-
H
methyl
ethyl




fluorophenyl






2.1.68
2-methoxy-3-
H
methyl
ethyl




fluorophenyl






2.1.69
2-ethoxy-3-
H
methyl
ethyl




fluorophenyl






2.1.70
2-trifluoro-
H
methyl
ethyl




methoxy-3-







fluorophenyl






2.1.71
2-nitro-3-
H
methyl
ethyl




fluorophenyl






2.1.72
2-fluoro-3-
H
methyl
ethyl




chlorophenyl






2.1.73
2,3-dichloro-
H
methyl
ethyl
[CDCl3] 1.32 (t, 3H), 1.73 (s,



phenyl



3H), 3.39 (d, 1H), 3.92 (d, 1H),







4.28 (m, 2H), 7.25 (m, 1H), 7.51







(m, 2H)


2.1.74
2,3-dichloro-
H
ethyl
ethyl




phenyl






2.1.75
2,3-dichloro-
H
propyl
ethyl




phenyl






2.1.76
2,3-dichloro-
H
cyclo-
ethyl




phenyl

propyl




2.1.77
2-bromo-3-
H
methyl
ethyl




chlorophenyl






2.1.78
2-methyl-3-
H
methyl
ethyl




chlorophenyl






2.1.79
2-ethyl-3-
H
methyl
ethyl




chlorophenyl






2.1.80
2-cyclopropyl-3-
H
methyl
ethyl




chlorophenyl






2.1.81
2-vinyl-3-
H
methyl
ethyl




chlorophenyl






2.1.82
2-ethynyl-3-
H
methyl
ethyl




chlorophenyl






2.1.83
2-cyano-3-
H
methyl
ethyl




chlorophenyl






2.1.84
2-trifluoro-
H
methyl
ethyl




methyl-2-







chlorophenyl






2.1.85
2-methoxy-3-
H
methyl
ethyl




chlorophenyl






2.1.86
2-ethoxy-3-
H
methyl
ethyl




chlorophenyl






2.1.87
2-trifluoro-
H
methyl
ethyl




methoxy-3-







chlorophenyl






2.1.88
2-nitro-3-
H
methyl
ethyl




chlorophenyl






2.1.89
2-fluoro-3-
H
methyl
ethyl




bromophenyl






2.1.90
2-chloro-3-
H
methyl
ethyl




bromophenyl






2.1.91
2,3-dibromo-
H
methyl
ethyl




phenyl






2.1.92
2-methyl-3-
H
methyl
ethyl




bromophenyl






2.1.93
2-ethyl-3-
H
methyl
ethyl




bromophenyl






2.1.94
2-cyclopropyl-3-
H
methyl
ethyl




bromophenyl






2.1.95
2-vinyl-3-
H
methyl
ethyl




bromophenyl






2.1.96
2-ethynyl-3-
H
methyl
ethyl




bromophenyl






2.1.97
2-cyano-3-
H
methyl
ethyl




bromophenyl






2.1.98
2-trifluoro-
H
methyl
ethyl




methyl-3-







bromophenyl






2.1.99
2-methoxy-3-
H
methyl
ethyl




phenyl






2.1.100
2-ethoxy-3-
H
methyl
ethyl




bromophenyl






2.1.101
2-trifluoro-
H
methyl
ethyl




methoxy-3-







bromophenyl






2.1.102
2-nitro-3-
H
methyl
ethyl




bromophenyl






2.1.103
2-fluoro-3-
H
methyl
ethyl




iodophenyl






2.1.104
2-chloro-3-
H
methyl
ethyl




iodophenyl






2.1.105
2-bromo-3-
H
methyl
ethyl




iodophenyl






2.1.106
2-methyl-3-
H
methyl
ethyl




iodophenyl






2.1.107
2-ethyl-3-
H
methyl
ethyl




iodophenyl






2.1.108
2-cyclopropyl-3-
H
methyl
ethyl




iodophenyl






2.1.109
2-vinyl-3-
H
methyl
ethyl




iodophenyl






2.1.110
2-ethynyl-3-
H
methyl
ethyl




iodophenyl






2.1.111
2-cyano-3-
H
methyl
ethyl




iodophenyl






2.1.112
2-trifluoro-
H
methyl
ethyl




methyl-3-







iodophenyl






2.1.113
2-methoxy-3-
H
methyl
ethyl




iodophenyl






2.1.114
2-ethoxy-3-
H
methyl
ethyl




iodophenyl






2.1.115
2-trifluoro-
H
methyl
ethyl




methoxy-3-







iodophenyl






2.1.116
2-nitro-3-
H
methyl
ethyl




iodophenyl






2.1.117
2-fluoro-3-
H
methyl
ethyl




methylphenyl






2.1.118
2-fluoro-3-
H
ethyl
ethyl




methylphenyl






2.1.119
2-fluoro-3-
H
propyl
ethyl




methylphenyl






2.1.120
2-fluoro-3-
H
cyclo-
ethyl




methylphenyl

propyl




2.1.121
2-chloro-3-
H
methyl
ethyl




methylphenyl






2.1.122
2-chloro-3-
H
ethyl
ethyl




methylphenyl






2.1.123
2-chloro-3-
H
propyl
ethyl




methylphenyl






2.1.124
2-chloro-3-
H
cyclo-
ethyl




methylphenyl

propyl




2.1.125
2-bromo-3-
H
methyl
ethyl




methylphenyl






2.1.126
2,3-dimethyl-
H
methyl
ethyl




phenyl






2.1.127
2,3-dimethyl-
H
ethyl
ethyl




phenyl






2.1.128
2,3-dimethyl-
H
propyl
ethyl




phenyl






2.1.129
2,3-dimethyl-
H
cyclo-
ethyl




phenyl

propyl




2.1.130
2-ethyl-3-
H
methyl
ethyl




methylphenyl






2.1.131
2-cyclopropyl-3-
H
methyl
ethyl




methylphenyl






2.1.132
2-vinyl-3-
H
methyl
ethyl




methylphenyl






2.1.133
2-ethynyl-3-
H
methyl
ethyl




methylphenyl






2.1.134
2-cyano-3-
H
methyl
ethyl




methylphenyl






2.1.135
2-trifluoro-
H
methyl
ethyl




methyl-3-







methylphenyl






2.1.136
2-methoxy-3-
H
methyl
ethyl




methylphenyl






2.1.137
2-ethoxy-3-
H
methyl
ethyl




methylphenyl






2.1.138
2-trifluoro-
H
methyl
ethyl




methoxy-3-







methylphenyl






2.1.139
2-nitro-3-
H
methyl
ethyl




methylphenyl






2.1.140
2-fluoro-3-
H
methyl
ethyl




ethylphenyl






2.1.141
2-chloro-3-
H
methyl
ethyl




ethylphenyl






2.1.142
2-bromo-3-
H
methyl
ethyl




ethylphenyl






2.1.143
2-methyl-3-
H
methyl
ethyl




ethylphenyl






2.1.144
2,3-diethyl-
H
methyl
ethyl




phenyl






2.1.145
2-cyclopropyl-3-
H
methyl
ethyl




ethylphenyl






2.1.146
2-vinyl-3-
H
methyl
ethyl




ethylphenyl






2.1.147
2-ethynyl-3-
H
methyl
ethyl




ethylphenyl






2.1.148
2-cyano-3-
H
methyl
ethyl




ethylphenyl






2.1.149
2-trifluoro-
H
methyl
ethyl




methyl-3-







ethylphenyl






2.1.150
2-methoxy-3-
H
methyl
ethyl




ethylphenyl






2.1.151
2-ethoxy-3-
H
methyl
ethyl




ethylphenyl






2.1.152
2-trifluoro-
H
methyl
ethyl




methoxy-3-







ethylphenyl






2.1.153
2-nitro-3-
H
methyl
ethyl




ethylphenyl






2.1.154
2-fluoro-3-
H
methyl
ethyl




propylphenyl






2.1.155
2-chloro-3-
H
methyl
ethyl




propylphenyl






2.1.156
2-bromo-3-
H
methyl
ethyl




propylphenyl






2.1.157
2-methyl-3-
H
methyl
ethyl




propylphenyl






2.1.158
2-methyl-3-
H
methyl
ethyl




propylphenyl






2.1.159
2-cyclopropyl-3-
H
methyl
ethyl




propylphenyl






2.1.160
2-vinyl-3-
H
methyl
ethyl




propylphenyl






2.1.161
2-ethynyl-
H
methyl
ethyl




3propylphenyl






2.1.162
2-cyano-3-
H
methyl
ethyl




propylphenyl






2.1.163
2-trifluoro-
H
methyl
ethyl




methyl-3-







propylphenyl






2.1.164
2-methoxy-3-
H
methyl
ethyl




propylphenyl






2.1.165
2-ethoxy-3-
H
methyl
ethyl




propylphenyl






2.1.166
2-trifluoro-
H
methyl
ethyl




methoxy-3-







propylphenyl






2.1.167
2-nitro-3-
H
methyl
ethyl




propylphenyl






2.1.168
2-fluoro-3-
H
methyl
ethyl




isopropylphenyl






2.1.169
2-chloro-3-
H
methyl
ethyl




isopropylphenyl






2.1.170
2-bomo-3-
H
methyl
ethyl




isopropylphenyl






2.1.171
2-methyl-3-
H
methyl
ethyl




isopropylphenyl






2.1.172
2-ethyl-3-
H
methyl
ethyl




isopropylphenyl






2.1.173
2-cyclopropyl-3-
H
methyl
ethyl




isopropylphenyl






2.1.174
2-vinyl-3-
H
methyl
ethyl




isopropylphenyl






2.1.175
2-ethynyl-3-
H
methyl
ethyl




isopropylphenyl






2.1.176
2-cyano-3-
H
methyl
ethyl




isopropylphenyl






2.1.177
2-trifluoro-
H
methyl
ethyl




methyl-3-







isopropylphenyl






2.1.178
2-methoxy-3-
H
methyl
ethyl




isopropylphenyl






2.1.179
2-thoxy-3-
H
methyl
ethyl




isopropylphenyl






2.1.180
2-trifluoro-
H
methyl
ethyl




methoxy-3-







isopropylphenyl






2.1.181
2-nitro-3-
H
methyl
ethyl




isopropylphenyl






2.1.182
2-fluoro-3-tert-
H
methyl
ethyl




butylphenyl






2.1.183
2-chloro-3-tert-
H
methyl
ethyl




butylphenyl






2.1.184
2-bromo-3-tert-
H
methyl
ethyl




butylphenyl






2.1.185
2-methyl-3-tert-
H
methyl
ethyl




butylphenyl






2.1.186
2-ethyl-3-tert-
H
methyl
ethyl




butylphenyl






2.1.187
2-cyclopropyl-3-
H
methyl
ethyl




tert-butylphenyl






2.1.188
2-vinyl-3-tert-
H
methyl
ethyl




butylphenyl






2.1.189
2-ethynyl-3-tert-
H
methyl
ethyl




butylphenyl






2.1.190
2-cyano-3-tert-
H
methyl
ethyl




butylphenyl






2.1.191
2-trifluoro-
H
methyl
ethyl




methyl-3-tert-







butylphenyl






2.1.192
2-methoxy-3-
H
methyl
ethyl




tert-butylphenyl






2.1.193
2-ethoxy-3-tert-
H
methyl
ethyl




butylphenyl






2.1.194
2-trifluoro-
H
methyl
ethyl




methoxy-3-tert-







butylphenyl






2.1.195
2-nitro-3-tert-
H
methyl
ethyl




butylphenyl






2.1.196
2-fluoro-3-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.197
2-chloro-3-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.198
2-bromo-3-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.199
2-methyl-3-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.200
2-ethyl-3-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.201
2-cyclopropyl-3-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.202
2-vinyl-3-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.203
2-ethynyl-3-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.204
2-cyano-3-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.205
2-trifluoro-
H
methyl
ethyl




methyl-3-







hydroxymethyl-







phenyl






2.1.206
2-methoxy-3-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.207
2-ethoxy-3-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.208
2-trifluoro-
H
methyl
ethyl




methoxy-3-







hydroxymethyl-







phenyl






2.1.209
2-nitro-3-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.210
2-fluoro-3-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.211
2-chloro-3-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.212
2-bromo-3-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.213
2-methyl-3-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.214
2-ethyl-3-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.215
2-cyclopropyl-3-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.216
2-vinyl-3-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.217
2-ethynyl-3-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.218
2-cyano-3-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.219
2-trifluoro-
H
methyl
ethyl




methyl-3-







cyclopropyl-







phenyl






2.1.220
2-methoxy-3-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.221
2-ethoxy-3-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.222
2-trifluoro-
H
methyl
ethyl




methoxy-3-







cyclopropyl-







phenyl






2.1.223
2-fluoro-3-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.224
2-chloro-3-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.225
2-bromo-3-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.226
2-methyl-3-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.227
2-ethyl-3-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.228
2-cyclopropyl-3-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.229
2-vinyl-3-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.230
2-ethynyl-3-
H
methyl
ethyl




methoxycarbonyl-







phenyl






2.1.231
2-cyano-3-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.232
2-trifluoro-
H
methyl
ethyl




methyl-3-







methoxy-







carbonylphenyl






2.1.233
2-methoxy-3-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.234
2-ethoxy-3-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.235
2-trifluoro-
H
methyl
ethyl




methoxy-3-







methoxy-







carbonylphenyl






2.1.236
2-nitro-3-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.237
2-fluoro-3-
H
methyl
ethyl




vinylphenyl






2.1.238
2-chloro-3-
H
methyl
ethyl




vinylphenyl






2.1.239
2-bromo-3-
H
methyl
ethyl




vinylphenyl






2.1.240
2-methyl-3-
H
methyl
ethyl




vinylphenyl






2.1.241
2-ethyl-3-
H
methyl
ethyl




vinylphenyl






2.1.242
2-cyclopropyl-3-
H
methyl
ethyl




vinylphenyl






2.1.243
2-vinyl-3-
H
methyl
ethyl




vinylphenyl






2.1.244
2-ethynyl-3-
H
methyl
ethyl




vinylphenyl






2.1.245
2-cyano-3-
H
methyl
ethyl




vinylphenyl






2.1.246
2-trifluoromethyl-
H
methyl
ethyl




3-vinylphenyl






2.1.247
2-methoxy-3-
H
methyl
ethyl




vinylphenyl






2.1.248
2-ethoxy-3-
H
methyl
ethyl




vinylphenyl






2.1.249
2-trifluoromethoxy-
H
methyl
ethyl




3-vinylphenyl






2.1.250
2-nitro-3-
H
methyl
ethyl




vinylphenyl






2.1.251
2-fluoro-3-
H
methyl
ethyl




ethynylphenyl






2.1.252
2-chloro-3-
H
methyl
ethyl




ethynylphenyl






2.1.253
2-bromo-3-
H
methyl
ethyl




ethynylphenyl






2.1.254
2-methyl-3-
H
methyl
ethyl




ethynylphenyl






2.1.255
2-ethyl-3-
H
methyl
ethyl




ethynylphenyl






2.1.256
2-cyclopropyl-3-
H
methyl
ethyl




ethynylphenyl






2.1.257
2-vinyl-3-
H
methyl
ethyl




ethynylphenyl






2.1.258
2-cyano-3-
H
methyl
ethyl




ethynylphenyl






2.1.259
2-trifluoromethyl-
H
methyl
ethyl




3-ethynylphenyl






2.1.260
2-methoxy-3-
H
methyl
ethyl




ethynylphenyl






2.1.261
2-ethoxy-3-
H
methyl
ethyl




ethynylphenyl






2.1.262
2-trifluoromethoxy-
H
methyl
ethyl




3-ethynylphenyl






2.1.263
2-nitro-3-
H
methyl
ethyl




ethynylphenyl






2.1.264
2-fluoro-3-
H
methyl
ethyl




ethynylphenyl






2.1.265
2-fluoro-3-
H
methyl
ethyl




cyanophenyl






2.1.266
2-chloro-3-
H
methyl
ethyl




cyanophenyl






2.1.267
2-bromo-3-
H
methyl
ethyl




cyanophenyl






2.1.268
2-methyl-3-
H
methyl
ethyl




cyanophenyl






2.1.269
2-ethyl-3-
H
methyl
ethyl




cyanophenyl






2.1.270
2-ethyl-3-
H
ethyl
ethyl




cyanophenyl






2.1.271
2-ethyl-3-
H
propyl
ethyl




cyanophenyl






2.1.272
2-ethyl-3-
H
cyclo-
ethyl




cyanophenyl

propyl




2.1.273
2-cyclopropyl-3-
H
methyl
ethyl




cyanophenyl






2.1.274
2-vinyl-3-
H
methyl
ethyl




cyanophenyl






2.1.275
2-ethynyl-3-
H
methyl
ethyl




cyanophenyl






2.1.276
2-cyano-3-
H
methyl
ethyl




cyanophenyl






2.1.277
2-trifluoromethyl-
H
methyl
ethyl




3-cyanophenyl






2.1.278
2-methoxy-3-
H
methyl
ethyl




cyanophenyl






2.1.279
2-ethoxy-3-
H
methyl
ethyl




cyanophenyl






2.1.280
2-trifluoro-
H
methyl
ethyl




methoxy-3-







cyanophenyl






2.1.281
2-nitro-3-
H
methyl
ethyl




cyanophenyl






2.1.282
2-fluoro-3-
H
methyl
ethyl




hydroxyphenyl






2.1.283
2-chloro-3-
H
methyl
ethyl




hydroxyphenyl






2.1.284
2-bromo-3-
H
methyl
ethyl




hydroxyphenyl






2.1.285
2-methyl-3-
H
methyl
ethyl




hydroxyphenyl






2.1.286
2-ethyl-3-
H
methyl
ethyl




hydroxyphenyl






2.1.287
2-cyclopropyl-3-
H
methyl
ethyl




hydroxyphenyl






2.1.288
2-vinyl-3-
H
methyl
ethyl




hydroxyphenyl






2.1.289
2-ethynyl-3-
H
methyl
ethyl




hydroxyphenyl






2.1.290
2-cyano-3-
H
methyl
ethyl




hydroxyphenyl






2.1.291
2-trifluoro-
H
methyl
ethyl




methyl-3-







hydroxyphenyl






2.1.292
2-methoxy-3-
H
methyl
ethyl




hydroxyphenyl






2.1.293
2-ethoxy-3-
H
methyl
ethyl




hydroxyphenyl






2.1.294
2-trifluoro-
H
methyl
ethyl




methoxy-3-







hydroxyphenyl






2.1.295
2-nitro-3-
H
methyl
ethyl




hydroxyphenyl






2.1.296
2-fluoro-3-
H
methyl
ethyl




methoxyphenyl






2.1.297
2-chloro-3-
H
methyl
ethyl




methoxyphenyl






2.1.298
2-bromo-3-
H
methyl
ethyl




methoxyphenyl






2.1.299
2-methyl-3-
H
methyl
ethyl




methoxyphenyl






2.1.300
2-ethyl-3-
H
methyl
ethyl




methoxyphenyl






2.1.301
2-cyclopropyl-3-
H
methyl
ethyl




methoxyphenyl






2.1.302
2-vinyl-3-
H
methyl
ethyl




methoxyphenyl






2.1.303
2-ethynyl-3-
H
methyl
ethyl




methoxyphenyl






2.1.304
2-cyano-3-
H
methyl
ethyl




methoxyphenyl






2.1.305
2-trifluoro-
H
methyl
ethyl




methyl-3-







methoxyphenyl






2.1.306
2,3-dimethoxy--
H
methyl
ethyl




phenyl






2.1.307
2-ethoxy-3-
H
methyl
ethyl




methoxyphenyl






2.1.308
2-trifluoro-
H
methyl
ethyl




methoxy-3-







methoxyphenyl






2.1.309
2-nitro-3-
H
methyl
ethyl




methoxyphenyl






2.1.310
2-fluoro-3-
H
methyl
ethyl




ethoxyphenyl






2.1.311
2-chloro-3-
H
methyl
ethyl




ethoxyphenyl






2.1.312
2-bromo-3-
H
methyl
ethyl




ethoxyphenyl






2.1.313
2-methyl-3-
H
methyl
ethyl




ethoxyphenyl






2.1.314
2-ethyl-3-
H
methyl
ethyl




ethoxyphenyl






2.1.315
2-cyclopropyl-3-
H
methyl
ethyl




ethoxyphenyl






2.1.316
2-vinyl-3-
H
methyl
ethyl




ethoxyphenyl






2.1.317
2-ethynyl-3-
H
methyl
ethyl




ethoxyphenyl






2.1.318
2-cyano-3-
H
methyl
ethyl




ethoxyphenyl






2.1.319
2-trifluoro-
H
methyl
ethyl




methyl-3-







ethoxyphenyl






2.1.320
2-methoxy-3-
H
methyl
ethyl




ethoxyphenyl






2.1.321
2,3-diethoxy--
H
methyl
ethyl




phenyl






2.1.322
2-trifluoro-
H
methyl
ethyl




methoxy-3-







ethoxyphenyl






2.1.323
2-nitro-3-
H
methyl
ethyl




ethoxyphenyl






2.1.324
2-fluoro-3-
H
methyl
ethyl




propoxyphenyl






2.1.325
2-chloro-3-
H
methyl
ethyl




propoxyphenyl






2.1.326
2-bromo-3-
H
methyl
ethyl




propoxyphenyl






2.1.327
2-methyl-3-
H
methyl
ethyl




propoxyphenyl






2.1.328
2-ethyl-3-
H
methyl
ethyl




propoxyphenyl






2.1.329
2-cyclopropyl-3-
H
methyl
ethyl




propoxyphenyl






2.1.330
2-vinyl-3-
H
methyl
ethyl




propoxyphenyl






2.1.331
2-ethynyl-3-
H
methyl
ethyl




propoxyphenyl






2.1.332
2-cyano-3-
H
methyl
ethyl




propoxyphenyl






2.1.333
2-trifluoro-
H
methyl
ethyl




methyl-3-







propoxyphenyl






2.1.334
2-methoxy-3-
H
methyl
ethyl




propoxyphenyl






2.1.335
2-ethoxy-3-
H
methyl
ethyl




propoxyphenyl






2.1.336
2-trifluoro-
H
methyl
ethyl




methoxy-3-







propoxyphenyl






2.1.337
2-nitro-3-
H
methyl
ethyl




propoxyphenyl






2.1.338
2-fluoro-3-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.339
2-chloro-3-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.340
2-bromo-3-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.341
2-methyl-3-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.342
2-ethyl-3-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.343
2-cyclopropyl-3-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.344
2-vinyl-3-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.345
2-ethynyl-3-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.346
2-cyano-3-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.347
2-trifluoro-
H
methyl
ethyl




methyl-3-







isopropoxy-







phenyl






2.1.348
2-methoxy-3-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.349
2-ethoxy-3-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.350
2-trifluoro-
H
methyl
ethyl




methoxy-3-







isopropoxy-







phenyl






2.1.351
2-nitro-3-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.352
2-fluoro-3-tert-
H
methyl
ethyl




butoxyphenyl






2.1.353
2-chloro-3-tert-
H
methyl
ethyl




butoxyphenyl






2.1.354
2-bromo-3-tert-
H
methyl
ethyl




butoxyphenyl






2.1.355
2-methyl-3-tert-
H
methyl
ethyl




butoxyphenyl






2.1.356
2-ethyl-3-tert-
H
methyl
ethyl




butoxyphenyl






2.1.357
2-cyclopropyl-3-
H
methyl
ethyl




tert-butoxy-







phenyl






2.1.358
2-vinyl-3-tert-
H
methyl
ethyl




butoxyphenyl






2.1.359
2-ethynyl-3-tert-
H
methyl
ethyl




butoxyphenyl






2.1.360
2-cyano-3-tert-
H
methyl
ethyl




butoxyphenyl






2.1.361
2-trifluoro-
H
methyl
ethyl




methyl-3-tert-







butoxyphenyl






2.1.362
2-methoxy-3-
H
methyl
ethyl




tert-butoxy-







phenyl






2.1.363
2-ethoxy-3-tert-
H
methyl
ethyl




butoxyphenyl






2.1.364
2-trifluoro-
H
methyl
ethyl




methoxy-3-tert-







butoxyphenyl






2.1.365
2-nitro-3-tert-
H
methyl
ethyl




butoxyphenyl






2.1.366
2-fluoro-3-
H
methyl
ethyl




trifluoromethoxy-







phenyl






2.1.367
2-chloro-3-
H
methyl
ethyl




trifluoromethoxy-







phenyl






2.1.368
2-bromo-3-
H
methyl
ethyl




trifluoromethoxy-







phenyl






2.1.369
2-methyl-3-
H
methyl
ethyl




trifluoromethoxy-







phenyl






2.1.370
2-ethyl-3-
H
methyl
ethyl




trifluoromethoxy-







phenyl






2.1.371
2-cyclopropyl-3-
H
methyl
ethyl




trifluoromethoxy-







phenyl






2.1.372
2-vinyl-3-
H
methyl
ethyl




trifluoromethoxy-







phenyl






2.1.373
2-ethynyl-3-
H
methyl
ethyl




trifluoromethoxy-







phenyl






2.1.374
2-cyano-3-
H
methyl
ethyl




trifluoromethoxy-







phenyl






2.1.375
2-trifluoro-
H
methyl
ethyl




methyl-3-







trifluoro-







methoxyphenyl






2.1.376
2-methoxy-3-
H
methyl
ethyl




trifluoro-







methoxyphenyl






2.1.377
2-ethoxy-3-
H
methyl
ethyl




trifluoro-







methoxyphenyl






2.1.378
2,3-bis(trifluoro-
H
methyl
ethyl




methoxy)phenyl






2.1.379
2-nitro-3-
H
methyl
ethyl




trifluoromethoxy-







phenyl






2.1.380
2-fluoro-3-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxy)phenyl






2.1.381
2-chloro-3-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxy)phenyl






2.1.382
2-bromo-3-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxy)phenyl






2.1.383
2-methyl-3-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxy)phenyl






2.1.384
2-ethyl-3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







phenyl






2.1.385
2-cyclopropyl-3-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxy)phenyl






2.1.386
2-vinyl-3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







phenyl






2.1.387
2-ethynyl-3-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxyphenyl






2.1.388
2-cyano-3-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxy)phenyl






2.1.389
2-trifluoro-
H
methyl
ethyl




methyl-3-(2,2,2-







trifluoroethoxy)-







phenyl






2.1.390
2-methoxy-3-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxy)phenyl






2.1.391
2-ethoxy-3-
H
methyl
ethyl




(2,2,2-







trifluoroethoxy)-







phenyl






2.1.392
2-trifluoro-
H
methyl
ethyl




methoxy-3-







(2,2,2-trifluoro-







ethoxy)phenyl






2.1.393
2-nitro-3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







phenyl






2.1.394
2-fluoro-3-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.395
2-chloro-3-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.396
2-bromo-3-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.397
2-methyl-3-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.398
2-ethyl-3-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.399
2-cyclopropyl-3-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.400
2-vinyl-3-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.401
2-ethynyl-3-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.402
2-cyano-3-
H
methyl
ethyl




difluoro-







methoxyphenyl






2.1.403
2-trifluoromethyl-
H
methyl
ethyl




3-difluoro-







methoxyphenyl






2.1.404
2-methoxy-3-
H
methyl
ethyl




difluoro-







methoxyphenyl






2.1.405
2-ethoxy-3-
H
methyl
ethyl




difluoromethoxy







phenyl






2.1.406
2-trifluoro-
H
methyl
ethyl




methoxy-3-







difluoromethoxy-







phenyl






2.1.407
2-nitro-3-
H
methyl
ethyl




difluoromethoxy







phenyl






2.1.408
2-fluoro-3-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.409
2-chloro-3-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.410
2-bromo-3-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.411
2-methyl-3-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.412
2-ethyl-3-(2-
H
methyl
ethyl




methoxyethoxy)







phenyl






2.1.413
2-cyclopropyl-3-
H
methyl
ethyl




(2-methoxy-







ethoxy)phenyl






2.1.414
2-vinyl-3-(2-
H
methyl
ethyl




methoxyethoxy)







phenyl






2.1.415
2-ethynyl-3-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.416
2-cyano-3-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.417
2-trifluoro-
H
methyl
ethyl




methyl-3-(2-







methoxyethoxy)-







phenyl






2.1.418
2-methoxy-3-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.419
2-ethoxy-3-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.420
2-trifluoro-
H
methyl
ethyl




methoxy-(2-







methoxyethoxy)-







phenyl






2.1.421
2-nitro-3-(2-
H
methyl
ethyl




methoxyethoxy)







phenyl






2.1.422
2-fluoro-3-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.423
2-chloro-3-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.424
2-bromo-3-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.425
2-methyl-3-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.426
2-ethyl-3-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.427
2-cyclopropyl-3-
H
methyl
ethyl




(tert-butoxy-







carbonyloxy)-







phenyl






2.1.428
2-vinyl-3-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.429
2-ethynyl-3-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.430
2-cyano-3-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.431
2-trifluoro-
H
methyl
ethyl




methyl-3-(tert-







butoxycarbonyl-







oxy)phenyl






2.1.432
2-methoxy-3-
H
methyl
ethyl




(tert-butoxy-







carbonyloxy)-







phenyl






2.1.433
2-ethoxy-3-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.434
2-trifluoro-
H
methyl
ethyl




methoxy-3-(tert-







butoxycarbonyl-







oxy)phenyl






2.1.435
2-nitro-3-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.436
2-fluoro-3-
H
methyl
ethyl




nitrophenyl






2.1.437
2-chloro-3-
H
methyl
ethyl




nitrophenyl






2.1.438
2-bromo-3-
H
methyl
ethyl




nitrophenyl






2.1.439
2-methyl-3-
H
methyl
ethyl




nitrophenyl






2.1.440
2-ethyl-3-
H
methyl
ethyl




nitrophenyl






2.1.441
2-cyclopropyl-3-
H
methyl
ethyl




nitrophenyl






2.1.442
2-vinyl-3-
H
methyl
ethyl




nitrophenyl






2.1.443
2-ethynyl-3-
H
methyl
ethyl




nitrophenyl






2.1.444
2-cyano-3-
H
methyl
ethyl




nitrophenyl






2.1.445
2-trifluoro-
H
methyl
ethyl




methyl-3-







nitrophenyl






2.1.446
2-methoxy-3-
H
methyl
ethyl




nitrophenyl






2.1.447
2-ethoxy-3-
H
methyl
ethyl




nitrophenyl






2.1.448
2-trifluoro-
H
methyl
ethyl




methoxy-3-







nitrophenyl






2.1.449
2-fluoro-3-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.450
2-chloro-3-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.451
2-bromo-3-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.452
2-methyl-3-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.453
2-ethyl-3-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.454
2-cyclopropyl-3-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.455
2-vinyl-3-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.456
2-ethynyl-3-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.457
2-cyano-3-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.458
2-trifluoro-
H
methyl
ethyl




methyl-3-







methylsulfanyl-







phenyl






2.1.459
2-methoxy-3-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.460
2-ethoxy-3-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.461
2-trifluoro-
H
methyl
ethyl




methoxy-3-







methylsulfanyl-







phenyl






2.1.462
2-nitro-3-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.463
3,5-difluoro-
H
methyl
methyl




phenyl






2.1.464
(S)-3,5-
H
methyl
methyl




difluorophenyl






2.1.465
(R)-3,5-difluoro-
H
methyl
methyl




phenyl






2.1.466
3,5-difluoro-
H
methyl
ethyl
[CDCl3] 1.30 (t, 3H); 1.71 (s,



phenyl



3H); 3.15 (d, 1H); 3.85 (d, 1H);







4.25 (m, 2H); 6.85 (m, 1H); 7.18







(m, 2H).


2.1.467
rel-(4R,5R)-3,5-
Me
Me
methyl
[CDCl3] 1.22 (d, 3H); 1.65 (s,



difluorophenyl



3H); 3.76 (s, 3H); 3.92 (q, 1H);







6.89 (m, 1H); 7.21 (m, 2H).


2.1.468
rel-(4R,5R)-3,5-
ethyl
Me
ethyl
[CDCl3] 0.92 (t, 3H); 1.28 (t, 3H);



difluorophenyl



1.69 (s, 3H); 1.74 (m, 2H); 3.80







(dd, 1H); 4.21 (m, 2H), 6.86 (m,







1H); 7.20 (m, 2H).


2.1.469
rel-(4R,5R)-3,5-
trifluoro
Me
ethyl
[CDCl3] 1.32 (t, 3H); 1.86 (“t”,



difluorophenyl
methyl


3H); 4.30 (m, 2H); 4.72 (q, 1H);







6.91 (m, 1H); 7.25 (m, 2H).


2.1.470
3,5-difluorophenyl
Cl
Me
methyl



2.1.471
3,5-difluorophenyl
H
Et
ethyl
[CDCl3] 1.00 (t, 3H); 1.32 (t, 3H);







2.06 (q, 2H); 3.18 (d, 1H); 3.88







(d, 1H); 4.27 (M, 2H); 6.85 (m,







1H), 7.18 (m, 2H).


2.1.472
3,5-difluorophenyl
H
isopropyl
ethyl
[CDCl3] 0.95-1.00 (m, 6H); 1.32







(t, 3H); 2.45 (m, 1H); 3.19 (d, 1H);







3.74 (d, 1H); 4.22-4.33 (m, 2H);







6.85 (m, 1H); 7.19 (m, 2H).


2.1.473
3,5-difluorophenyl
H
cyclo-
ethyl






propyl




2.1.474
3-chloro-5-
H
methyl
ethyl
[CDCl3] 1.3 (t, 3H); 1.72 (s, 3H);



fluorophenyl



3.14 (d, 1H); 3.82 (d, 1H); 4.28







(mc, 2H); 7.15 (mc, 1H); 7.30







(mc, 1H); 7.410 (s, 1H).


2.1.475
3-chloro-5-
H
ethyl
ethyl
[CDCl3] 1.00 (t, 3H); 1.35 (t, 3H);



fluorophenyl



2.08 (q, 2H); 3.19 (d, 1H); 3.75







(d, 1H); 4.29 (m, 2H); 7.15 (m,







1H); 7.30 (m, 1H); 7.41 (s, 1H).


2.1.476
3-chloro-5-
H
isopropyl
ethyl




fluorophenyl






2.1.477
3-chloro-5-
H
cyclo-
ethyl




fluorophenyl

propyl




2.1.478
3-bromo-5-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.72 (s,



fluorophenyl



3H); 3.15 (d, 1H); 3.85 (d, 1H);







4.28 (m, 2H); 7.31 (mc; 2H);







7.55 (m, 1H).


2.1.479
3-bromo-5-
H
ethyl
ethyl




fluorophenyl






2.1.480
3-bromo-5-
H
isopropyl
ethyl




fluorophenyl






2.1.481
3-bromo-5-
H
cyclo-
ethyl




fluorophenyl

propyl




2.1.482
3-iodo-5-
H
methyl
ethyl




fluorophenyl






2.1.483
3-methyl-5-
H
methyl
ethyl
[CDCl3] 1.32 (t, 3H); 1.70 (s,



fluorophenyl



3H); 2.38 (s, 3H); 3.18 (d, 1H);







3.83 (d, 1H); 4.25 (m, 2H); 6.92







(d, 1H); 7.15 (dd, 1H); 7.24 (d,







1H).


2.1.484
3-methyl-5-
H
ethyl
ethyl




fluorophenyl






2.1.485
3-methyl-5-
H
isopropyl
ethyl




fluorophenyl






2.1.486
3-methyl-5-
H
cyclo-
ethyl




fluorophenyl

propyl




2.1.487
3-ethyl-5-
H
methyl
ethyl
[CDCl3] 1.25 (t, 3H); 1.35 (t, 3H);



fluorophenyl



1.72 (s, 3H); 2.68 (q, 2H); 3.18







(d, 1H); 3.82 (d, 1H); 4.25 (m,







2H); 6.95 (d, 1H); 7.18 (dd, 1H);







7.25 (d, 1H).


2.1.488
3-propyl-5-
H
methyl
ethyl




fluorophenyl






2.1.489
3-i-propyl-5-
H
methyl
ethyl




fluorophenyl






2.1.490
3-n-butyl-5-
H
methyl
ethyl




fluorophenyl






2.1.491
3-isobutyl-5-
H
methyl
ethyl




fluorophenyl






2.1.492
3-tert-butyl-5-
H
methyl
ethyl




fluorophenyl






2.1.493
3-cyclopropyl-5-
H
methyl
ethyl
[CDCl3] 0.7 (m, 2H); 1.1 (m, 2H);



fluorophenyl



1.32 (t, 3H); 1.70 (s, 3H); 1.90







(m, 1H); 3.15 (d, 1H); 3.82 (d,







1H); 4.25 (m, 2H); 6.78 (dd, 1H);







7.11 (dd, 1H); 7.20 (s, 1H).


2.1.494
3-vinyl-5-
H
methyl
ethyl




fluorophenyl






2.1.495
3-ethynyl-5-
H
methyl
ethyl




fluorophenyl






2.1.496
3-cyano-5-
H
methyl
ethyl




fluorophenyl






2.1.497
3-trifluoro-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.72 (s,



methyl-5-



3H); 3.18 (d, 1H); 3.89 (d, 1H);



fluorophenyl



4.25 (m, 2H); 7.35 (d, 1H); 7.58







(d, 1H); 7.65 (bs, 1H).


2.1.498
3-trifluoro-
H
ethyl
ethyl




methyl-5-







fluorophenyl






2.1.499
3-trifluoro-
H
isopropyl
ethyl




methyl-5-







fluorophenyl






2.1.500
3-trifluoro-
H
cyclo-
ethyl




methyl-5-

propyl





fluorophenyl






2.1.501
3-(methoxy-
H
methyl
ethyl




carbonyl)-5-







fluorophenyl






2.1.502
3-hydroxy-
H
methyl
ethyl




methyl-5-







fluorophenyl






2.1.503
3-carbamoyl-5-
H
methyl
ethyl




fluorophenyl






2.1.504
3-hydroxy-5-
H
methyl
ethyl




fluorophenyl






2.1.505
3-methoxy-5-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.71 (s,



fluorophenyl



3H); 3.16 (d, 1H); 3.80 (s, 3H);







3.85 (d, 1H); 4.25 (m, 2H); 6.65







(dd, 1H); 6.91 (dd, 1H); 7.02 (s,







1H).


2.1.506
3-ethoxy-5-
H
methyl
ethyl




fluorophenyl






2.1.507
3-n-propoxy-5-
H
methyl
ethyl




fluorophenyl






2.1.508
3-isopropoxy-5-
H
methyl
ethyl




fluorophenyl






2.1.509
3-n-butoxy-5-
H
methyl
ethyl




fluorophenyl






2.1.510
3-isobutoxy-5-
H
methyl
ethyl




fluorophenyl






2.1.511
3-tert-butoxy-5-
H
methyl
ethyl




fluorophenyl






2.1.512
3-difluoro-
H
methyl
ethyl




methoxy-5-







fluorophenyl






2.1.513
3-trifluoro-
H
methyl
ethyl




methoxy-5-







fluorophenyl






2.1.514
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-fluorophenyl






2.1.515
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







fluorophenyl






2.1.516
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







fluorophenyl






2.1.517
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







fluorophenyl






2.1.518
3-nitro-5-
H
methyl
ethyl




fluorophenyl






2.1.519
3-acetoxy-5-
H
methyl
ethyl




fluorophenyl






2.1.520
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-fluorophenyl}






2.1.521
3-methyl-
H
methyl
ethyl
[CDCl3] 1.32 (t, 3H); 1.70 (s,



sulfanyl-5-



3H); 2.5 (s, 3H); 3.15 (d, 1H);



fluorophenyl



3.82 (d, 1H); 6.95 (dd, 1H); 7.10







(dd, 1H); 7.25 (d, 1H).


2.1.522
3,5-dichloro-
H
methyl
ethyl
[CDCl3] 1.31 (3, 3H); 1.70 (s,



phenyl



3H); 3.15 (d, 1H); 3.82 (d, 1H);







4.25 (m, 2H); 7.40 (s, 1H); 7.52







(s, 2H).


2.1.523
3,5-dichloro-
H
methyl
methyl
[CDCl3] 1.72 (s, 3H); 3.15 (d,



phenyl



1H); 3.81 (s, 3H); 3.87 (d, 1H);







7.40 (m, 1H); 7.5 (m, 2H).


2.1.524
3,5-dichloro-
H
methyl
isopropyl
[CDCl3] 1.30 (d, 6H); 1.70 (s,



phenyl



3H); 3.12 (d, 1H); 3.82 (d, 1H);







5.10 (m, 1H); 7.40 (s, 1H); 7.52







(s, 2H).


2.1.525
(S)-3,5-
H
methyl
methyl
[CDCl3] 1.72 (s, 3H); 3.16



dichlorophenyl



(d,1H), 3.82 (s, 3H), 3.84 (d, 1H);







7.40 (s, 1H); 7.53 (s, 2H).


2.1.526
(R)-3,5-
H
methyl
methyl
[CDCl3] 1.72 (s, 3H); 3.15 (d, 1H);



dichlorophenyl



3.82 (s, 3H); 3.84 (d, 1H); 7.41







(s, 1H); 7.54 (s, 2H).


2.1.527
3,5-
H
ethyl
ethyl
[CDCl3] 1.00 (t, 3H); 1.38 (t, 3H);



dichlorophenyl



2.07 (q, 2H); 2.18 (q, 2H); 3.16







(d, 1H); 3.76 (d, 1H); 7.37 (s,







1H); 7.55 (s, 2H).


2.1.528
3,5-dichloro-
H
propyl
ethyl




phenyl






2.1.529
3,5-dichloro-
H
iPr
ethyl
[CDCl3] 0.92 (dd; mc, 6H); 1.32



phenyl



(t, 3H); 2.45 (MC, 1H); 3.18 (d,







1H); 3.74 (d, 1H); 4.25 (mc, 2H);







7.41 (s, 1H); 7.55 (s, 2H).


2.1.530
3,5-dichloro-
H
cyclo-
ethyl
[CDCl3] 0.45-0.75 (m, 4H); 1.32



phenyl

propyl

(t, 3H); 1.42 (m, 1H); 3.23 (d,







1H); 3.78 (d, 1H); 4.29 (mc, 2H);







7.38 (s, 1H); 7.51 (s, 2H).


2.1.531
3-bromo-5-
H
methyl
methyl
[CDCl3] 1.72 (s, 3H); 3.15 (d,



chlorophenyl



1H); 3.81 (s, 3H); 3.85 (d, 1H);







7.55 (m, 2H); 7.70 (m, 1H).


2.1.532
3-bromo-5-
H
methyl
ethyl
[CDCl3] 1.32 (t, 3H); 1.70 (s,



chlorophenyl



3H); 3.13 (d, 1H); 3.82 (d, 1H);







4.28 (m, 2H); 7.58 (m, 2H); 7.69







(m, 1H).


2.1.533
rel-(4R,5R)-3,5-
methyl
methyl
methyl
[CDCl3] 1.20 (d, 3H); 1.61 (s,



dichlorophenyl



3H); 3.78 (s, 3H); 3.82 (q, 1H);







7.41 (s, 1H); 7.58 (s, 2H).


2.1.534
Rel-(4R,5S)-3,5-
methyl
methyl
methyl
[CDCl3] 1.15 (d, 1H); 1.62 (s,



dichlorophenyl



3H); 3.48 (q, 1H); 3.83 (s, 3H);







7.40 (s, 1H); 7.55 (s, 2H).


2.1.535
3-methyl-5-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.70 (s,



chlorophenyl



3H); 2.35 (s, 3H); 3.15 (d, 1H);







3.85 (d, 1H); 4.25 (m, 2H); 7.21







(s, 1H); 7.37 (s, 1H); 7.42 (s, 1H).


2.1.536
3-propyl-5-
H
methyl
ethyl




chlorophenyl






2.1.537
3-isopropyl-5-
H
methyl
ethyl




chlorophenyl






2.1.538
3-n-butyl-5-
H
methyl
ethyl




chlorophenyl






2.1.539
3-isobutyl-5-
H
methyl
ethyl




chlorophenyl






2.1.540
3-tert-butyl-5-
H
methyl
ethyl




chlorophenyl






2.1.541
3-cyclopropyl-5-
H
methyl
ethyl




chlorophenyl






2.1.542
3-vinyl-5-
H
methyl
ethyl




chlorophenyl






2.1.543
3-ethynyl-5-
H
methyl
ethyl




chlorophenyl






2.1.544
3-cyano-5-
H
methyl
ethyl




chlorophenyl






2.1.545
3-trifluoro-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.72 (s,



methyl-5-



3H); 3.20 (d, 1H); 3.90 (d, 1H);



chlorophenyl



4.25 (m, 2H); 7.65 (s, 1H); 7.76







(s, 1H); 7.84 (s, 1H).


2.1.546
3-trifluoro-
H
methyl
isopropyl
[CDCl3] 1.30 (d, 6H); 1.71 (s,



methyl-5-



3H); 3.15 (d, 1H); 3.85 (d, 1H);



chlorophenyl



5.10 (m, 1H); 7.65 (s, 1H); 7.77







(s, 1H); 7.85 (s, 1H).


2.1.547
3-(hydroxy-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 3.18 (d,



carbonyl)-5-



1H); 3.85 (d, 1H); 4.25 (q, 2H);



chlorophenyl



6.15 (bs, 1H); 6.92 (d, 1H); 7.10







(s, 1H); 7.20 (s, 1H).


2.1.548
3-(methoxy-
H
methyl
ethyl




carbonyl)-5-







chlorophenyl






2.1.549
3-hydroxy-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.71 (s,



methyl-5-



3H); 3.17 (d, 1H); 3.85 (d, 1H);



chlorophenyl



4.25 (m, 2H); 4.70 (s, 2H); 7.41







(s, 1H); 7.60 (mc, 2H).


2.1.550
3-carbamoyl-5-
H
methyl
ethyl




chlorophenyl






2.1.551
3-hydroxy-5-
H
methyl
ethyl




chlorophenyl






2.1.552
3-methoxy-5-
H
methyl
ethyl
[CDCl3] 1.32 (t, 3H); 1.71 (s,



chlorophenyl



3H); 3.16 (d, 1H); 3.82 (s, 3H);







3.86 (d, 1H); 4.25 (mc, 2H); 6.95







(m, 1H); 7.16 (m, 2H).


2.1.553
3-ethoxy-5-
H
methyl
ethyl




chlorophenyl






2.1.554
3-n-propoxy-5-
H
methyl
ethyl




chlorophenyl






2.1.555
3-isopropoxy-5-
H
methyl
ethyl




chlorophenyl






2.1.556
3-n-butoxy-5-
H
methyl
ethyl




chlorophenyl






2.1.557
3-isobutoxy-5-
H
methyl
ethyl




chlorophenyl






2.1.558
3-tert-butoxy-5-
H
methyl
ethyl




chlorophenyl






2.1.559
3-difluoro-
H
methyl
ethyl




methoxy-5-







chlorophenyl






2.1.560
3-trifluoro-
H
methyl
ethyl




methoxy-5-







chlorophenyl






2.1.561
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-chlorophenyl






2.1.562
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







chlorophenyl






2.1.563
3-(2-
H
methyl
ethyl




hydroxyethoxy)-







5-chlorophenyl






2.1.564
3-[(tert-butoxy-
H
methyl
ethyl
[CDCl3] 1.30 (t, 3H); 1.55 (s,



carbonyl)oxy]-5-



9H); 1.70 (s, 3H); 3.15 (d, 1H);



chlorophenyl



3.82 (d, 1H); 4.25 (m, 2H); 7.25







(s, 1H); 7.38 (d, 1H); 7.51 (s,







1H).


2.1.565
3-nitro-5-
H
methyl
ethyl




chlorophenyl






2.1.566
3-acetoxy-5-
H
methyl
ethyl




chlorophenyl






2.1.567
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-chlorophenyl}






2.1.568
3-methyl-
H
methyl
ethyl




sulfanyl-5-







chlorophenyl






2.1.569
3,5-dibromo-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.71 (s, H);



phenyl



3.15 (d, 1H); 3.82 (d, 1H); 4.28







(m, 2H); 7.70 (s, 1H); 7.75 (s,







2H).


2.1.570
3,5-dibromo-
H
ethyl
ethyl
[CDCl3] 1.00 (t, 3H); 1.31 (t, 3H);



phenyl



2.05 (q, 2H); 3.15 (d, 1H); 3.75







(d, 1H); 4.30 (m, 2H); 7.70 (s,







1H); 7.78 (s, 2H).


2.1.571
3,5-dibromo-
H
isopropyl
ethyl




phenyl






2.1.572
3,5-dibromo-
H
cyclo-
ethyl




phenyl

propyl




2.1.573
3-iodo-5-
H
methyl
ethyl




bromophenyl






2.1.574
3-methyl-5-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.70 (s,



bromophenyl



3H); 2.35 (s, 3H); 3.15 (d, 1H);







3.85 (d, 1H); 4.26 (m, 2H); 7.38







(s, 1H); 7.43 (s, 1H); 7.58 (s,







1H).


2.1.575
3-methyl-5-
H
ethyl
ethyl




bromophenyl






2.1.576
3-methyl-5-
H
isopropyl
ethyl




bromophenyl






2.1.577
3-methyl-5-
H
cyclo-
ethyl




bromophenyl

propyl




2.1.578
3-ethyl-5-
H
methyl
ethyl




bromophenyl






2.1.579
3-propyl-5-
H
methyl
ethyl




bromophenyl






2.1.580
3-isopropyl-5-
H
methyl
ethyl




bromophenyl






2.1.581
3-n-butyl-5-
H
methyl
ethyl




bromophenyl






2.1.582
3-isobutyl-5-
H
methyl
ethyl




bromophenyl






2.1.583
3-tert-butyl-5-
H
methyl
ethyl




bromophenyl






2.1.584
3-cyclopropyl-5-
H
methyl
ethyl




bromophenyl






2.1.585
3-vinyl-5-
H
methyl
ethyl




bromophenyl






2.1.586
3-ethynyl-5-
H
methyl
ethyl




bromophenyl






2.1.587
3-cyano-5-
H
methyl
ethyl




bromophenyl






2.1.588
3-trifluoro-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.75 (s,



methyl-5-



3H); 3.2 (d, 1H); 3.89 (d, 1H);



bromophenyl



7.81 (d, 2H); 8.0 (m, 1H).


2.1.589
3-(hydroxy-
H
methyl
ethyl




carbonyl)-5-







bromophenyl






2.1.590
3-(methoxy-
H
methyl
ethyl




carbonyl)-5-







bromophenyl






2.1.591
3-hydroxy-
H
methyl
ethyl




methyl-5-







bromophenyl






2.1.592
3-carbamoyl-5-
H
methyl
ethyl




bromophenyl






2.1.593
3-hydroxy-5-
H
methyl
ethyl




bromophenyl






2.1.594
3-methoxy-5-
H
methyl
ethyl




bromophenyl






2.1.595
3-ethoxy-5-
H
methyl
ethyl




bromophenyl






2.1.596
3-n-propoxy-5-
H
methyl
ethyl




bromophenyl






2.1.597
3-isopropoxy-5-
H
methyl
ethyl




bromophenyl






2.1.598
3-n-butoxy-5-
H
methyl
ethyl




bromophenyl






2.1.599
3-isobutoxy-5-
H
methyl
ethyl




bromophenyl






2.1.600
3-tert-butoxy-5-
H
methyl
ethyl




bromophenyl






2.1.601
3-difluoro-
H
methyl
ethyl




methoxy-5-







bromophenyl






2.1.602
3-trifluoro-
H
methyl
ethyl




methoxy-5-







bromophenyl






2.1.603
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-bromophenyl






2.1.604
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







bromophenyl






2.1.605
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







bromophenyl






2.1.606
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







bromophenyl






2.1.607
3-nitro-5-
H
methyl
ethyl




bromophenyl






2.1.608
3-acetoxy-5-
H
methyl
ethyl




bromophenyl






2.1.609
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-bromophenyl}






2.1.610
3-methyl-
H
methyl
ethyl




sulfanyl-5-







bromophenyl






2.1.611
3,5-diiodophenyl
H
methyl
ethyl
[CDCl3] 1.32 (st, 3H); 1.70 (s,







3H); 3.12 (d, 1H); 3.81 (d, 1H);







7.93 (s, 2H); 8.09 (s, 1H).


2.1.612
3-methyl-5-
H
methyl
ethyl




iodophenyl






2.1.613
3-ethyl-5-
H
methyl
ethyl




iodophenyl






2.1.614
3-propyl-5-
H
methyl
ethyl




iodophenyl






2.1.615
3-isopropyl-5-
H
methyl
ethyl




iodophenyl






2.1.616
3-n-butyl-5-
H
methyl
ethyl




iodophenyl






2.1.617
3-isobutyl-5-
H
methyl
ethyl




iodophenyl






2.1.618
3-tert-butyl-5-
H
methyl
ethyl




iodophenyl






2.1.619
3-cyclopropyl-5-
H
methyl
ethyl




iodophenyl






2.1.620
3-vinyl-5-
H
methyl
ethyl




iodophenyl






2.1.621
3-ethynyl-5-
H
methyl
ethyl




iodophenyl






2.1.622
3-cyano-5-
H
methyl
ethyl




iodophenyl






2.1.623
3-trifluoro-
H
methyl
ethyl




methyl-5-







iodophenyl






2.1.624
3-(hydroxy-
H
methyl
ethyl




carbonyl)-5-







iodophenyl






2.1.625
3-(methoxycarbonyl)-
H
methyl
ethyl




5-iodophenyl






2.1.626
3-hydroxy-
H
methyl
ethyl




methyl-5-







iodophenyl






2.1.627
3-carbamoyl-5-
H
methyl
ethyl




iodophenyl






2.1.628
3-hydroxy-5-
H
methyl
ethyl




iodophenyl






2.1.629
3-methoxy-5-
H
methyl
ethyl




iodophenyl






2.1.630
3-ethoxy-5-
H
methyl
ethyl




iodophenyl






2.1.631
3-n-propoxy-5-
H
methyl
ethyl




iodophenyl






2.1.632
3-isopropoxy-5-
H
methyl
ethyl




iodophenyl






2.1.633
3-n-butoxy-5-
H
methyl
ethyl




iodophenyl






2.1.634
3-isobutoxy-5-
H
methyl
ethyl




iodophenyl






2.1.635
3-tert-butoxy-5-
H
methyl
ethyl




iodophenyl






2.1.636
3-difluoro-
H
methyl
ethyl




methoxy-5-







iodophenyl






2.1.637
3-trifluoro-
H
methyl
ethyl




methoxy-5-







iodophenyl






2.1.638
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-iodophenyl






2.1.639
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







iodophenyl






2.1.640
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







iodophenyl






2.1.641
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







iodophenyl






2.1.642
3-nitro-5-
H
methyl
ethyl




iodophenyl






2.1.643
3-acetoxy-5-
H
methyl
ethyl




iodophenyl






2.1.644
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-iodophenyl}






2.1.645
3-methyl-
H
methyl
ethyl




sulfanyl-5-







iodophenyl






2.1.646
3,5-dimethyl-
H
methyl
ethyl
[CDCl3] 1.30 (t, 3H); 1.69 (s,



phenyl



3H); 2.31 (s, 6H); 3.19 (d, 1H);







3.85 (d, 1H); 4.25 (mc, 2H); 7.05







(s, 1H); 7.25 (s, 2H).


2.1.647
3-ethyl-5-
H
methyl
ethyl




methylphenyl






2.1.648
3-propyl-5-
H
methyl
ethyl




methylphenyl






2.1.649
3-isopropyl-5-
H
methyl
ethyl




methylphenyl






2.1.650
3-n-butyl-5-
H
methyl
ethyl




methylphenyl






2.1.651
3-isobutyl-5-
H
methyl
ethyl




methylphenyl






2.1.652
3-tert-butyl-5-
H
methyl
ethyl




methylphenyl






2.1.653
3-cyclopropyl-5-
H
methyl
ethyl




methylphenyl






2.1.654
3-vinyl-5-
H
methyl
ethyl




methylphenyl






2.1.655
3-ethynyl-5-
H
methyl
ethyl




methylphenyl






2.1.656
3-cyano-5-
H
methyl
ethyl




methylphenyl






2.1.657
3-trifluoro-
H
methyl
ethyl




methyl-5-







methylphenyl






2.1.658
3-(hydroxy-
H
methyl
ethyl




carbonyl)-5-







methylphenyl






2.1.659
3-(methoxy-
H
methyl
ethyl




carbonyl)-5-







methylphenyl






2.1.660
3-hydroxy-
H
methyl
ethyl




methyl-5-







methylphenyl






2.1.661
3-carbamoyl-5-
H
methyl
ethyl




methylphenyl






2.1.662
3-hydroxy-5-
H
methyl
ethyl




methylphenyl






2.1.663
3-methoxy-5-
H
methyl
ethyl




methylphenyl






2.1.664
3-ethoxy-5-
H
methyl
ethyl




methylphenyl






2.1.665
3-n-propoxy-5-
H
methyl
ethyl




methylphenyl






2.1.666
3-n-butoxy-5-
H
methyl
ethyl




methylphenyl






2.1.667
3-isobutoxy-5-
H
methyl
ethyl




methylphenyl






2.1.668
3-tert-butoxy-5-
H
methyl
ethyl




methylphenyl






2.1.669
3-difluoro-
H
methyl
ethyl




methoxy-5-







methylphenyl






2.1.670
3-trifluoro-
H
methyl
ethyl
[CDCl3] 1.30 (t, 3H); 1.72 (s,



methoxy-5-



3H); 2.40 (s, 3H); 3.18 (d, 1H);



methylphenyl



3.86 (d, 1H); 4.25 (m, 2H); 7.08







(s, 1H); 7.31 (s, 1H); 7.41 (s,







1H).


2.1.671
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-methylphenyl






2.1.672
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







methylphenyl






2.1.673
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







methylphenyl






2.1.674
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







methylphenyl






2.1.675
3-nitro-5-
H
methyl
ethyl




methylphenyl






2.1.676
3-acetoxy-5-
H
methyl
ethyl




methylphenyl






2.1.677
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-methyl-







phenyl}






2.1.678
3-methyl-
H
methyl
ethyl




sulfanyl-5-







methylphenyl






2.1.679
3,5-diethyl-
H
methyl
ethyl




phenyl






2.1.680
3-propyl-5-
H
methyl
ethyl




ethylphenyl






2.1.681
3-isopropyl-5-
H
methyl
ethyl




ethylphenyl






2.1.682
3-n-butyl-5-
H
methyl
ethyl




ethylphenyl






2.1.683
3-isobutyl-5-
H
methyl
ethyl




ethylphenyl






2.1.684
3-tert-butyl-5-
H
methyl
ethyl




ethylphenyl






2.1.685
3-cyclopropyl-5-
H
methyl
ethyl




ethylphenyl






2.1.686
3-vinyl-5-
H
methyl
ethyl




ethylphenyl






2.1.687
3-ethynyl-5-
H
methyl
ethyl




ethylphenyl






2.1.688
3-cyano-5-
H
methyl
ethyl




ethylphenyl






2.1.689
3-trifluoro-
H
methyl
ethyl




methyl-5-







ethylphenyl






2.1.690
3-(hydroxy-
H
methyl
ethyl




carbonyl)-5-







ethylphenyl






2.1.691
3-(methoxy-
H
methyl
ethyl




carbonyl)-5-







ethylphenyl






2.1.692
3-hydroxy-
H
methyl
ethyl




methyl-5-







ethylphenyl






2.1.693
3-carbamoyl-5-
H
methyl
ethyl




ethylphenyl






2.1.694
3-hydroxy-5-
H
methyl
ethyl




ethylphenyl






2.1.695
3-methoxy-5-
H
methyl
ethyl




ethylphenyl






2.1.696
3-ethoxy-5-
H
methyl
ethyl




ethylphenyl






2.1.697
3-n-propoxy-5-
H
methyl
ethyl




ethylphenyl






2.1.698
3-n-butoxy-5-
H
methyl
ethyl




ethylphenyl






2.1.699
3-isobutoxy-5-
H
methyl
ethyl




ethylphenyl






2.1.700
3-tert-butoxy-5-
H
methyl
ethyl




ethylphenyl






2.1.701
3-difluoro-
H
methyl
ethyl




methoxy-5-







ethylphenyl






2.1.702
3-trifluoro-
H
methyl
ethyl




methoxy-5-







ethylphenyl






2.1.703
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-ethylphenyl






2.1.704
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







ethylphenyl






2.1.705
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







ethylphenyl






2.1.706
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







ethylphenyl






2.1.707
3-nitro-5-
H
methyl
ethyl




ethylphenyl






2.1.708
3-acetoxy-5-
H
methyl
ethyl




ethylphenyl






2.1.709
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-ethylphenyl}






2.1.710
3-methyl-
H
methyl
ethyl




sulfanyl-5-







ethylphenyl






2.1.711
3,5-dipropyl-
H
methyl
ethyl




phenyl






2.1.712
3-isopropyl-5-
H
methyl
ethyl




propylphenyl






2.1.713
3-n-butyl-5-
H
methyl
ethyl




propylphenyl






2.1.714
3-isobutyl-5-
H
methyl
ethyl




propylphenyl






2.1.715
3-tert-butyl-5-
H
methyl
ethyl




propylphenyl






2.1.716
3-cyclopropyl-5-
H
methyl
ethyl




propylphenyl






2.1.717
3-vinyl-5-
H
methyl
ethyl




propylphenyl






2.1.718
3-ethynyl-5-
H
methyl
ethyl




propylphenyl






2.1.719
3-cyano-5-
H
methyl
ethyl




propylphenyl






2.1.720
3-trifluoro-
H
methyl
ethyl




methyl-5-







propylphenyl






2.1.721
3-(hydroxy-
H
methyl
ethyl




carbonyl)-5-







propylphenyl






2.1.722
3-(methoxy-
H
methyl
ethyl




carbonyl)-5-







propylphenyl






2.1.723
3-hydroxy-
H
methyl
ethyl




methyl-5-







propylphenyl






2.1.724
3-carbamoyl-5-
H
methyl
ethyl




propylphenyl






2.1.725
3-hydroxy-5-
H
methyl
ethyl




propylphenyl






2.1.726
3-methoxy-5-
H
methyl
ethyl




propylphenyl






2.1.727
3-ethoxy-5-
H
methyl
ethyl




propylphenyl






2.1.728
3-n-propoxy-5-
H
methyl
ethyl




propylphenyl






2.1.729
3-n-butoxy-5-
H
methyl
ethyl




propylphenyl






2.1.730
3-isobutoxy-5-
H
methyl
ethyl




propylphenyl






2.1.731
3-tert-butoxy-5-
H
methyl
ethyl




propylphenyl






2.1.732
3-difluoro-
H
methyl
ethyl




methoxy-5-







propylphenyl






2.1.733
3-trifluoro-
H
methyl
ethyl




methoxy-5-







ethylphenyl






2.1.734
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-propylphenyl






2.1.735
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







propylphenyl






2.1.736
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







propylphenyl






2.1.737
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







propylphenyl






2.1.738
3-nitro-5-
H
methyl
ethyl




propylphenyl






2.1.739
3-acetoxy-5-
H
methyl
ethyl




propylphenyl






2.1.740
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-propylphenyl}






2.1.741
3-methyl-
H
methyl
ethyl




sulfanyl-5-







propylphenyl






2.1.742
3,5-diisopropyl-
H
methyl
ethyl




phenyl






2.1.743
3-n-butyl-5-
H
methyl
ethyl




isopropylphenyl






2.1.744
3-isobutyl-5-
H
methyl
ethyl




isopropylphenyl






2.1.745
3-tert-butyl-5-
H
methyl
ethyl




isopropylphenyl






2.1.746
3-cyclopropyl-5-
H
methyl
ethyl




isopropylphenyl






2.1.747
3-vinyl-5-
H
methyl
ethyl




isopropylphenyl






2.1.748
3-ethynyl-5-
H
methyl
ethyl




isopropylphenyl






2.1.749
3-cyano-5-
H
methyl
ethyl




isopropylphenyl






2.1.750
3-trifluoro-
H
methyl
ethyl




methyl-5-







isopropylphenyl






2.1.751
3-(hydroxy-
H
methyl
ethyl




carbonyl)-5-







isopropylphenyl






2.1.752
3-(methoxy-
H
methyl
ethyl




carbonyl)-5-







isopropylphenyl






2.1.753
3-hydroxy-
H
methyl
ethyl




methyl-5-







isopropylphenyl






2.1.754
3-carbamoyl-5-
H
methyl
ethyl




isopropylphenyl






2.1.755
3-hydroxy-5-
H
methyl
ethyl




isopropylphenyl






2.1.756
3-methoxy-5-
H
methyl
ethyl




isopropylphenyl






2.1.757
3-ethoxy-5-
H
methyl
ethyl




isopropylphenyl






2.1.758
3-n-propoxy-5-
H
methyl
ethyl




isopropylphenyl






2.1.759
3-n-butoxy-5-
H
methyl
ethyl




isopropylphenyl






2.1.760
3-isobutoxy-5-
H
methyl
ethyl




isopropylphenyl






2.1.761
3-tert-butoxy-5-
H
methyl
ethyl




isopropylphenyl






2.1.762
3-difluoro-
H
methyl
ethyl




methoxy-5-







isopropylphenyl






2.1.763
3-trifluoro-
H
methyl
ethyl




methoxy-5-







isopropylphenyl






2.1.764
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-isopropyl-







phenyl






2.1.765
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







isopropylphenyl






2.1.766
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







propylphenyl






2.1.767
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







isopropylphenyl






2.1.768
3-nitro-5-
H
methyl
ethyl




isopropylphenyl






2.1.769
3-acetoxy-5-
H
methyl
ethyl




isopropylphenyl






2.1.770
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-isopropyl-







phenyl}






2.1.771
3-methyl-
H
methyl
ethyl




sulfanyl-5-







isopropyl-phenyl






2.1.772
3,5-dibutyl-
H
methyl
ethyl




phenyl






2.1.773
3-isobutyl-5-
H
methyl
ethyl




butylphenyl






2.1.774
3-tert-butyl-5-
H
methyl
ethyl




butylphenyl






2.1.775
3-cyclopropyl-5-
H
methyl
ethyl




butylphenyl






2.1.776
3-vinyl-5-
H
methyl
ethyl




butylphenyl






2.1.777
3-ethynyl-5-
H
methyl
ethyl




butylphenyl






2.1.778
3-cyano-5-
H
methyl
ethyl




butylphenyl






2.1.779
3-trifluoro-
H
methyl
ethyl




methyl-5-







butylphenyl






2.1.780
3-(hydroxy-
H
methyl
ethyl




carbonyl)-5-







butylphenyl






2.1.781
3-(methoxy-
H
methyl
ethyl




carbonyl)-5-







butylphenyl






2.1.782
3-hydroxy-
H
methyl
ethyl




methyl-5-







butylphenyl






2.1.783
3-carbamoyl-5-
H
methyl
ethyl




butylphenyl






2.1.784
3-hydroxy-5-
H
methyl
ethyl




butylphenyl






2.1.785
3-methoxy-5-
H
methyl
ethyl




butylphenyl






2.1.786
3-ethoxy-5-
H
methyl
ethyl




butylphenyl






2.1.787
3-n-propoxy-5-
H
methyl
ethyl




butylphenyl






2.1.788
3-n-butoxy-5-
H
methyl
ethyl




butylphenyl






2.1.789
3-isobutoxy-5-
H
methyl
ethyl




butylphenyl






2.1.790
3-tert-butoxy-5-
H
methyl
ethyl




butylphenyl






2.1.791
3-difluoro-
H
methyl
ethyl




methoxy-5-







butylphenyl






2.1.792
3-trifluoro-
H
methyl
ethyl




methoxy-5-







butylphenyl






2.1.793
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-butylphenyl






2.1.794
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







butylphenyl






2.1.795
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







butylphenyl






2.1.796
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







butylphenyl






2.1.797
3-nitro-5-
H
methyl
ethyl




butylphenyl






2.1.798
3-acetoxy-5-
H
methyl
ethyl




butylphenyl






2.1.799
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-butylphenyl}






2.1.800
3-methyl-
H
methyl
ethyl




sulfanyl-5-







butylphenyl






2.1.801
3,5-diisobutyl-
H
methyl
ethyl




phenyl






2.1.802
3-tert-butyl-5-
H
methyl
ethyl




isobutylphenyl






2.1.803
3-cyclopropyl-5-
H
methyl
ethyl




isobutylphenyl






2.1.804
3-vinyl-5-
H
methyl
ethyl




isobutylphenyl






2.1.805
3-ethynyl-5-
H
methyl
ethyl




isobutylphenyl






2.1.806
3-cyano-5-
H
methyl
ethyl




isobutylphenyl






2.1.807
3-trifluoro-
H
methyl
ethyl




methyl-5-







isobutylphenyl






2.1.808
3-(hydroxy-
H
methyl
ethyl




carbonyl)-5-







isobutylphenyl






2.1.809
3-(methoxy-
H
methyl
ethyl




carbonyl)-5-







isobutylphenyl






2.1.810
3-hydroxy-
H
methyl
ethyl




methyl-5-







isobutylphenyl






2.1.811
3-carbamoyl-5-
H
methyl
ethyl




isobutylphenyl






2.1.812
3-hydroxy-5-
H
methyl
ethyl




isobutylphenyl






2.1.813
3-methoxy-5-
H
methyl
ethyl




isobutylphenyl






2.1.814
3-ethoxy-5-
H
methyl
ethyl




isobutylphenyl






2.1.815
3-n-propoxy-5-
H
methyl
ethyl




isobutylphenyl






2.1.816
3-n-butoxy-5-
H
methyl
ethyl




isobutylphenyl






2.1.817
3-isobutoxy-5-
H
methyl
ethyl




isobutylphenyl






2.1.818
3-tert-butoxy-5-
H
methyl
ethyl




isobutylphenyl






2.1.819
3-difluoro-
H
methyl
ethyl




methoxy-5-







isobutylphenyl






2.1.820
3-trifluoro-
H
methyl
ethyl




methoxy-5-







isobutylphenyl






2.1.821
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-isobutylphenyl






2.1.822
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







isobutylphenyl






2.1.823
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







isobutylphenyl






2.1.824
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







isobutylphenyl






2.1.825
3-nitro-5-
H
methyl
ethyl




isobutylphenyl






2.1.826
3-acetoxy-5-
H
methyl
ethyl




isobutylphenyl






2.1.827
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-isobutyl-







phenyl}






2.1.828
3-methyl-
H
methyl
ethyl




sulfanyl-5-







isobutylphenyl






2.1.829
3,5-di-tert-
H
methyl
ethyl




butylphenyl






2.1.830
3-cyclopropyl-5-
H
methyl
ethyl




tert-butylphenyl






2.1.831
3-vinyl-5-tert-
H
methyl
ethyl




butylphenyl






2.1.832
3-ethynyl-5-tert-
H
methyl
ethyl




butylphenyl






2.1.833
3-cyano-5-tert-
H
methyl
ethyl




butylphenyl






2.1.834
3-trifluoro-
H
methyl
ethyl




methyl-5-tert-







butylphenyl






2.1.835
3-(hydroxy-
H
methyl
ethyl




carbonyl)-5-tert-







butylphenyl






2.1.836
3-(methoxy-
H
methyl
ethyl




carbonyl)-5-tert-







butylphenyl






2.1.837
3-hydroxy-
H
methyl
ethyl




methyl-5-tert-







butylphenyl






2.1.838
3-carbamoyl-5-
H
methyl
ethyl




tert-butylphenyl






2.1.839
3-hydroxy-5-tert-
H
methyl
ethyl




butylphenyl






2.1.840
3-methoxy-5-
H
methyl
ethyl




tert-butylphenyl






2.1.841
3-ethoxy-5-tert-
H
methyl
ethyl




butylphenyl






2.1.842
3-n-propoxy-5-
H
methyl
ethyl




tert-butylphenyl






2.1.843
3-n-butoxy-5-
H
methyl
ethyl




tert-butylphenyl






2.1.844
3-isobutoxy-5-
H
methyl
ethyl




tert-butylphenyl






2.1.845
3-tert-butoxy-5-
H
methyl
ethyl




tert-butylphenyl






2.1.846
3-difluoro-
H
methyl
ethyl




methoxy-5-tert-







butylphenyl






2.1.847
3-trifluoro-
H
methyl
ethyl




methoxy-5-tert-







butylphenyl






2.1.848
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-tert-butyl-







phenyl






2.1.849
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-tert-







butylphenyl






2.1.850
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-tert-







butylphenyl






2.1.851
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







tert-butylphenyl






2.1.852
3-nitro-5-tert-
H
methyl
ethyl




butylphenyl






2.1.853
3-acetoxy-5-tert-
H
methyl
ethyl




butylphenyl






2.1.854
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-tert-butyl-







phenyl}






2.1.855
3-methyl-
H
methyl
ethyl




sulfanyl-5-tert-







butylphenyl






2.1.856
3-tert-butyl-5-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.857
3,5-dicyclo-
H
methyl
ethyl




propylphenyl






2.1.858
3-vinyl-5-cyclo-
H
methyl
ethyl




propylphenyl






2.1.859
3-ethynyl-5-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.860
3-cyano-5-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.861
3-trifluoro-
H
methyl
ethyl




methyl-5-







cyclopropyl-







phenyl






2.1.862
3-(hydroxy-
H
methyl
ethyl




carbonyl)-5-







cyclopropyl-







phenyl






2.1.863
3-(methoxy-
H
methyl
ethyl




carbonyl)-5-







cyclopropyl-







phenyl






2.1.864
3-hydroxy-
H
methyl
ethyl




methyl-5-







cyclopropyl-







phenyl






2.1.865
3-carbamoyl-5-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.866
3-hydroxy-5-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.867
3-methoxy-5-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.868
3-ethoxy-5-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.869
3-n-propoxy-5-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.870
3-n-butoxy-5-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.871
3-isobutoxy-5-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.872
3-tert-butoxy-5-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.873
3-difluoro-
H
methyl
ethyl




methoxy-5-







cyclopropyl-







phenyl






2.1.874
3-trifluoro-
H
methyl
ethyl




methoxy-5-







cyclopropyl-







phenyl






2.1.875
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-cyclopropyl-







phenyl






2.1.876
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







cyclopropyl-







phenyl






2.1.877
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







cyclopropyl-







phenyl






2.1.878
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







cyclopropyl-







phenyl






2.1.879
3-nitro-5-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.880
3-acetoxy-5-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.881
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-cyclopropyl-







phenyl}






2.1.882
3-methyl-
H
methyl
ethyl




sulfanyl-5-







cyclopropyl-







phenyl






2.1.883
3,5-divinyl-
H
methyl
ethyl




phenyl






2.1.884
3-ethynyl-5-
H
methyl
ethyl




vinylphenyl






2.1.885
3-cyano-5-
H
methyl
ethyl




vinylphenyl






2.1.886
3-trifluoro-
H
methyl
ethyl




methyl-5-







vinylphenyl






2.1.887
3-(hydroxy-
H
methyl
ethyl




carbonyl)-5-







vinylphenyl






2.1.888
3-(methoxy-
H
methyl
ethyl




carbonyl)-5-







vinylphenyl






2.1.889
3-hydroxy-
H
methyl
ethyl




methyl-5-







vinylphenyl






2.1.890
3-carbamoyl-5-
H
methyl
ethyl




vinylphenyl






2.1.891
3-hydroxy-5-
H
methyl
ethyl




vinylphenyl






2.1.892
3-methoxy-5-
H
methyl
ethyl




vinylphenyl






2.1.893
3-ethoxy-5-
H
methyl
ethyl




vinylphenyl






2.1.894
3-n-propoxy-5-
H
methyl
ethyl




vinylphenyl






2.1.895
3-n-butoxy-5-
H
methyl
ethyl




vinylphenyl






2.1.896
3-isobutoxy-5-
H
methyl
ethyl




vinylphenyl






2.1.897
3-tert-butoxy-5-
H
methyl
ethyl




vinylphenyl






2.1.898
3-difluoro-
H
methyl
ethyl




methoxy-5-







vinylphenyl






2.1.899
3-trifluoro-
H
methyl
ethyl




methoxy-5-







vinylphenyl






2.1.900
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-vinylphenyl






2.1.901
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







vinylphenyl






2.1.902
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







vinylphenyl






2.1.903
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







vinylphenyl






2.1.904
3-nitro-5-
H
methyl
ethyl




vinylphenyl






2.1.905
3-acetoxy-5-
H
methyl
ethyl




vinylphenyl






2.1.906
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-vinylphenyl}






2.1.907
3-methyl-
H
methyl
ethyl




sulfanyl-5-







vinylphenyl






2.1.908
3,5-diethynyl-
H
methyl
ethyl




phenyl






2.1.909
3-cyano-5-
H
methyl
ethyl




ethynylphenyl






2.1.910
3-trifluoro-
H
methyl
ethyl




methyl-5-







ethynylphenyl






2.1.911
3-(hydroxy-
H
methyl
ethyl




carbonyl)-5-







ethynylphenyl






2.1.912
3-(methoxy-
H
methyl
ethyl




carbonyl)-5-







ethynylphenyl






2.1.913
3-hydroxy-
H
methyl
ethyl




methyl-5-







ethynylphenyl






2.1.914
3-carbamoyl-5-
H
methyl
ethyl




ethynylphenyl






2.1.915
3-hydroxy-5-
H
methyl
ethyl




ethynylphenyl






2.1.916
3-methoxy-5-
H
methyl
ethyl




ethynylphenyl






2.1.917
3-ethoxy-5-
H
methyl
ethyl




ethynylphenyl






2.1.918
3-n-propoxy-5-
H
methyl
ethyl




ethynylphenyl






2.1.919
3-n-butoxy-5-
H
methyl
ethyl




ethynylphenyl






2.1.920
3-isobutoxy-5-
H
methyl
ethyl




ethynylphenyl






2.1.921
3-tert-butoxy-5-
H
methyl
ethyl




ethynylphenyl






2.1.922
3-difluoro-
H
methyl
ethyl




methoxy-5-







ethynylphenyl






2.1.923
3-trifluoro-
H
methyl
ethyl




methoxy-5-







ethynylphenyl






2.1.924
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-ethynylphenyl






2.1.925
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







ethynylphenyl






2.1.926
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







ethynylphenyl






2.1.927
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







ethynylphenyl






2.1.928
3-nitro-5-
H
methyl
ethyl




ethynylphenyl






2.1.929
3-acetoxy-5-
H
methyl
ethyl




ethynylphenyl






2.1.930
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-ethynyl-







phenyl}






2.1.931
3-methyl-
H
methyl
ethyl




sulfanyl-5-







ethynylphenyl






2.1.932
3,5-dicyano-
H
methyl
ethyl




phenyl






2.1.933
3-trifluoro-
H
methyl
ethyl




methyl-5-







cyanophenyl






2.1.934
3-(hydroxy-
H
methyl
ethyl




carbonyl)-5-







cyanophenyl






2.1.935
3-(methoxy-
H
methyl
ethyl




carbonyl)-5-







cyanophenyl






2.1.936
3-hydroxy-
H
methyl
ethyl




methyl-5-







cyanophenyl






2.1.937
3-carbamoyl-5-
H
methyl
ethyl




cyanophenyl






2.1.938
3-hydroxy-5-
H
methyl
ethyl




cyanophenyl






2.1.939
3-methoxy-5-
H
methyl
ethyl




cyanophenyl






2.1.940
3-ethoxy-5-
H
methyl
ethyl




cyanophenyl






2.1.941
3-n-propoxy-5-
H
methyl
ethyl




cyanophenyl






2.1.942
3-n-butoxy-5-
H
methyl
ethyl




cyanophenyl






2.1.943
3-isobutoxy-5-
H
methyl
ethyl




cyanophenyl






2.1.944
3-tert-butoxy-5-
H
methyl
ethyl




cyanophenyl






2.1.945
3-difluoro-
H
methyl
ethyl




methoxy-5-







cyanophenyl






2.1.946
3-trifluoro-
H
methyl
ethyl




methoxy-5-







cyanophenyl






2.1.947
3-(2,2,2-tri-
H
methyl
ethyl




fluoroethoxy)-5-







cyanophenyl






2.1.948
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







cyanophenyl






2.1.949
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







cyanophenyl






2.1.950
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







cyanophenyl






2.1.951
3-nitro-5-
H
methyl
ethyl




cyanophenyl






2.1.952
3-acetoxy-5-
H
methyl
ethyl




cyanophenyl






2.1.953
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-cyanophenyl}






2.1.954
3-methyl-
H
methyl
ethyl




sulfanyl-5-







cyanophenyl






2.1.955
3,5-di(trifluoro-
H
methyl
ethyl
[CDCl3] 1.30 (t, 3H); 1.75 (s,



methyl)-phenyl



3H); 3.25 (d, 1H); 3.95 (d, 1H),







4.39 (m, 2H); 7.91 (bs, 1H); 8.10







(bs, 2H).


2.1.956
3-(hydroxy-
H
methyl
ethyl




carbonyl)-5-







trifluoromethyl-







phenyl






2.1.957
3-(methoxy-
H
methyl
ethyl




carbonyl)-5-







trifluoromethyl-







phenyl






2.1.958
3-hydroxy-
H
methyl
ethyl




methyl-5-







trifluoromethyl-







phenyl






2.1.959
3-carbamoyl-5-
H
methyl
ethyl




trifluoromethyl-







phenyl






2.1.960
3-hydroxy-5-
H
methyl
ethyl




trifluoromethyl-







phenyl






2.1.961
3-methoxy-5-
H
methyl
ethyl




trifluoromethyl-







phenyl






2.1.962
3-ethoxy-5-
H
methyl
ethyl




trifluoromethyl-







phenyl






2.1.963
3-n-propoxy-5-
H
methyl
ethyl




trifluoromethyl-







phenyl






2.1.964
3-n-butoxy-5-
H
methyl
ethyl




trifluoromethyl-







phenyl






2.1.965
3-isobutoxy-5-
H
methyl
ethyl




trifluoromethyl-







phenyl






2.1.966
3-tert-butoxy-5-
H
methyl
ethyl




trifluoromethyl-







phenyl






2.1.967
3-difluoro-
H
methyl
ethyl




methoxy-5-







trifluoromethyl-







phenyl






2.1.968
3-trifluoro-
H
methyl
ethyl




methoxy-5-







trifluoromethyl-







phenyl






2.1.969
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-trifluoro-







methylphenyl






2.1.970
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







trifluoromethyl-







phenyl






2.1.971
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







trifluoromethyl-







phenyl






2.1.972
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







trifluoromethyl-







phenyl






2.1.973
3-nitro-5-
H
methyl
ethyl




trifluoromethyl-







phenyl






2.1.974
3-acetoxy-5-
H
methyl
ethyl




trifluoromethyl-







phenyl






2.1.975
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-trifluoro-







methylphenyl}






2.1.976
3-methyl-
H
methyl
ethyl




sulfanyl-5-







trifluoromethyl-







phenyl






2.1.977
3,5-bis(hydroxy-
H
methyl
ethyl




carbonyl)phenyl






2.1.978
3-(methoxy-
H
methyl
ethyl




carbonyl)-5-







(hydroxy-







carbonyl)phenyl






2.1.979
3-hydroxy-
H
methyl
ethyl




methyl-5-







(hydroxy-







carbonyl)phenyl






2.1.980
3-carbamoyl-5-
H
methyl
ethyl




(hydroxy-







carbonyl)phenyl






2.1.981
3-hydroxy-5-
H
methyl
ethyl




(hydroxy-







carbonyl)phenyl






2.1.982
3-methoxy-5-
H
methyl
ethyl




(hydroxy-







carbonyl)phenyl






2.1.983
3-ethoxy-5-
H
methyl
ethyl




(hydroxy-







carbonyl)phenyl






2.1.984
3-n-propoxy-5-
H
methyl
ethyl




(hydroxy-







carbonyl)phenyl






2.1.985
3-n-butoxy-5-
H
methyl
ethyl




(hydroxy-







carbonyl)phenyl






2.1.986
3-isobutoxy-5-
H
methyl
ethyl




(hydroxy-







carbonyl)phenyl






2.1.987
3-tert-butoxy-5-
H
methyl
ethyl




(hydroxy-







carbonyl)phenyl






2.1.988
3-difluoro-
H
methyl
ethyl




methoxy-5-







(hydroxy-







carbonyl)phenyl






2.1.989
3-trifluoro-
H
methyl
ethyl




methoxy-5-







(hydroxy-







carbonyl)phenyl






2.1.990
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-(hydroxy-







carbonyl)phenyl






2.1.991
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







(hydroxy-







carbonyl)phenyl






2.1.992
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







(hydroxy-







carbonyl)phenyl






2.1.993
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







(hydroxy-







carbonyl)phenyl






2.1.994
3-nitro-5-
H
methyl
ethyl




(hydroxy-







carbonyl)phenyl






2.1.995
3-acetoxy-5-
H
methyl
ethyl




(hydroxy-







carbonyl)phenyl






2.1.996
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-(hydroxy-







carbonyl)phenyl}






2.1.997
3-methyl-
H
methyl
ethyl




sulfanyl-5-







(hydroxy-







carbonyl)phenyl






2.1.998
3,5-di(methoxy-
H
methyl
ethyl




carbonyl)phenyl






2.1.999
3-hydroxy-
H
methyl
ethyl




methyl-5-







(methoxy-







carbonyl)phenyl






2.1.1000
3-carbamoyl-5-
H
methyl
ethyl




(methoxy-







carbonyl)phenyl






2.1.1001
3-hydroxy-5-
H
methyl
ethyl




(methoxy-







carbonyl)phenyl






2.1.1002
3-methoxy-5-
H
methyl
ethyl




(methoxy-







carbonyl)phenyl






2.1.1003
3-ethoxy-5-
H
methyl
ethyl




(methoxy-







carbonyl)phenyl






2.1.1004
3-n-propoxy-5-
H
methyl
ethyl




(methoxy-







carbonyl)phenyl






2.1.1005
3-n-butoxy-5-
H
methyl
ethyl




(methoxy-







carbonyl)phenyl






2.1.1006
3-isobutoxy-5-
H
methyl
ethyl




(methoxy-







carbonyl)phenyl






2.1.1007
3-tert-butoxy-5-
H
methyl
ethyl




(methoxy-







carbonyl)phenyl






2.1.1008
3-difluoro-
H
methyl
ethyl




methoxy-5-







(methoxy-







carbonyl)phenyl






2.1.1009
3-trifluoro-
H
methyl
ethyl




methoxy-5-







(methoxy-







carbonyl)phenyl






2.1.1010
3-(2,2,2-
H
methyl
ethyl




trifluoro-ethoxy)-







5-(methoxy-







carbonyl)phenyl






2.1.1011
3-(2-chloro-
H
methyl
ethyl




ethoxy)-







(methoxy-







carbonyl)phenyl






2.1.1012
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-







(methoxy-







carbonyl)phenyl






2.1.1013
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







(methoxy-







carbonyl)phenyl






2.1.1014
3-nitro-5-
H
methyl
ethyl




(methoxy-







carbonyl)phenyl






2.1.1015
3-acetoxy-5-
H
methyl
ethyl




(methoxy-







carbonyl)phenyl






2.1.1016
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-(methoxy-







carbonyl)phenyl)






2.1.1017
3-methyl-
H
methyl
ethyl




sulfanyl-5-







(methoxy-







carbonyl)phenyl






2.1.1018
3,5-di(hydroxy-
H
methyl
ethyl




methyl)phenyl






2.1.1019
3-carbamoyl-5-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1020
3-hydroxy-5-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1021
3-methoxy-5-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1022
3-ethoxy-5-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1023
3-n-propoxy-5-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1024
3-n-butoxy-5-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1025
3-isobutoxy-5-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1026
3-tert-butoxy-5-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1027
3-difluoro-
H
methyl
ethyl




methoxy-5-







hydroxymethyl-







phenyl






2.1.1028
3-trifluoro-
H
methyl
ethyl




methoxy-5-







hydroxymethyl-







phenyl






2.1.1029
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-hydroxy-







methylphenyl






2.1.1030
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







hydroxymethyl-







phenyl






2.1.1031
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







hydroxymethyl-







phenyl






2.1.1032
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







hydroxymethyl-







phenyl






2.1.1033
3-nitro-5-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1034
3-acetoxy-5-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1035
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-hydroxy-







methylphenyl)






2.1.1036
3-methyl-
H
methyl
ethyl




sulfanyl-5-







hydroxymethyl-







phenyl






2.1.1037
3,5-
H
methyl
ethyl




dicarbamoyl-5-







carbamoyl-







phenyl






2.1.1038
3-hydroxy-5-
H
methyl
ethyl




carbamoyl-







phenyl






2.1.1039
3-methoxy-5-
H
methyl
ethyl




carbamoyl-







phenyl






2.1.1040
3-ethoxy-5-
H
methyl
ethyl




carbamoyl-







phenyl






2.1.1041
3-n-propoxy-5-
H
methyl
ethyl




carbamoyl-







phenyl






2.1.1042
3-n-butoxy-5-
H
methyl
ethyl




carbamoyl-







phenyl






2.1.1043
3-isobutoxy-5-
H
methyl
ethyl




carbamoyl-







phenyl






2.1.1044
3-tert-butoxy-5-
H
methyl
ethyl




carbamoyl-







phenyl






2.1.1045
3-difluoro-
H
methyl
ethyl




methoxy-5-







carbamoyl-







phenyl






2.1.1046
3-trifluoro-
H
methyl
ethyl




methoxy-5-







carbamoyl-







phenyl






2.1.1047
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-carbamoyl-







phenyl






2.1.1048
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







carbamoyl-







phenyl






2.1.1049
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







carbamoyl-







phenyl






2.1.1050
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







carbamoyl-







phenyl






2.1.1051
3-nitro-5-
H
methyl
ethyl




carbamoyl-







phenyl






2.1.1052
3-acetoxy-5-
H
methyl
ethyl




carbamoyl-







phenyl






2.1.1053
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)-







amino]-5-







carbamoyl-







phenyl}






2.1.1054
3-methyl-
H
methyl
ethyl




sulfanyl-5-







carbamoyl-







phenyl






2.1.1055
3,5-dihydroxy-
H
methyl
ethyl




phenyl






2.1.1056
3-methoxy-5-
H
methyl
ethyl




hydroxyphenyl






2.1.1057
3-ethoxy-5-
H
methyl
ethyl




hydroxyphenyl






2.1.1058
3-n-propoxy-5-
H
methyl
ethyl




hydroxyphenyl






2.1.1059
3-n-butoxy-5-
H
methyl
ethyl




hydroxyphenyl






2.1.1060
3-isobutoxy-5-
H
methyl
ethyl




hydroxyphenyl






2.1.1061
3-tert-butoxy-5-
H
methyl
ethyl




hydroxyphenyl






2.1.1062
3-difluoro-
H
methyl
ethyl




methoxy-5-







hydroxyphenyl






2.1.1063
3-trifluoro-
H
methyl
ethyl




methoxy-5-







hydroxyphenyl






2.1.1064
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-hydroxyphenyl






2.1.1065
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







hydroxyphenyl






2.1.1066
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







hydroxyphenyl






2.1.1067
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







hydroxyphenyl






2.1.1068
3-nitro-5-
H
methyl
ethyl




hydroxyphenyl






2.1.1069
3-acetoxy-5-
H
methyl
ethyl




hydroxyphenyl






2.1.1070
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-hydroxy-







phenyl}






2.1.1071
3-methyl-
H
methyl
ethyl




sulfanyl-5-







hydroxyphenyl






2.1.1072
3,5-dimethoxy-
H
methyl
ethyl
[CDCl3] 1.30 (t, 3H); 1.71 (s,



phenyl



3H); 3.15 (d, 1H); 3.80 (s, 6H);







3.85 (d, 1H); 4.25 (m, 2H); 6.51







(d, 1H); 6.80 (d, 1H).


2.1.1073
3-ethoxy-5-
H
methyl
ethyl




methoxyphenyl






2.1.1074
3-n-propoxy-5-
H
methyl
ethyl




methoxyphenyl






2.1.1075
3-n-butoxy-5-
H
methyl
ethyl




methoxyphenyl






2.1.1076
3-isobutoxy-5-
H
methyl
ethyl




methoxyphenyl






2.1.1077
3-tert-butoxy-5-
H
methyl
ethyl




methoxyphenyl






2.1.1078
3-difluoro-
H
methyl
ethyl




methoxy-5-







methoxyphenyl






2.1.1079
3-trifluoro-
H
methyl
ethyl




methoxy-5-







methoxyphenyl






2.1.1080
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-methoxy-







phenyl






2.1.1081
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







methoxyphenyl






2.1.1082
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







methoxyphenyl






2.1.1083
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







methoxyphenyl






2.1.1084
3-nitro-5-
H
methyl
ethyl




methoxyphenyl






2.1.1085
3-acetoxy-5-
H
methyl
ethyl




methoxyphenyl






2.1.1086
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-methoxy-







phenyl}






2.1.1087
3-methyl-
H
methyl
ethyl




sulfanyl-5-







methoxyphenyl






2.1.1088
3,5-diethoxy-
H
methyl
ethyl




phenyl






2.1.1089
3-n-propoxy-5-
H
methyl
ethyl




ethoxyphenyl






2.1.1090
3-n-butoxy-5-
H
methyl
ethyl




ethoxyphenyl






2.1.1091
3-isobutoxy-5-
H
methyl
ethyl




ethoxyphenyl






2.1.1092
3-tert-butoxy-5-
H
methyl
ethyl




ethoxyphenyl






2.1.1093
3-difluoro-
H
methyl
ethyl




methoxy-5-







ethoxyphenyl






2.1.1094
3-trifluoro-
H
methyl
ethyl




methoxy-5-







ethoxyphenyl






2.1.1095
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-ethoxyphenyl






2.1.1096
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







ethoxyphenyl






2.1.1097
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







ethoxyphenyl






2.1.1098
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







ethoxyphenyl






2.1.1099
3-nitro-5-
H
methyl
ethyl




ethoxyphenyl






2.1.1100
3-acetoxy-5-
H
methyl
ethyl




ethoxyphenyl






2.1.1101
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-ethoxy-







phenyl}






2.1.1102
3-methyl-
H
methyl
ethyl




sulfanyl-5-







ethoxyphenyl






2.1.1103
3,5-dipropoxy-
H
methyl
ethyl




phenyl






2.1.1104
3-n-butoxy-5-
H
methyl
ethyl




propoxyphenyl






2.1.1105
3-isobutoxy-5-
H
methyl
ethyl




propoxyphenyl






2.1.1106
3-tert-butoxy-5-
H
methyl
ethyl




propoxyphenyl






2.1.1107
3-difluoro-
H
methyl
ethyl




methoxy-5-







propoxyphenyl






2.1.1108
3-trifluoro-
H
methyl
ethyl




methoxy-5-







propoxyphenyl






2.1.1109
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-propoxyphenyl






2.1.1110
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







propoxyphenyl






2.1.1111
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







propoxyphenyl






2.1.1112
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







propoxyphenyl






2.1.1113
3-nitro-5-
H
methyl
ethyl




propoxyphenyl






2.1.1114
3-acetoxy-5-
H
methyl
ethyl




propoxyphenyl






2.1.1115
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-propoxy-







phenyl}






2.1.1116
3-methyl-
H
methyl
ethyl




sulfanyl-5-







propoxyphenyl






2.1.1117
3,5-
H
methyl
ethyl




di(isopropoxy)-







phenyl






2.1.1118
3-n-butoxy-5-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.1119
3-isobutoxy-5-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.1120
3-tert-butoxy-5-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.1121
3-difluoro-
H
methyl
ethyl




methoxy-5-







isopropoxy-







phenyl






2.1.1122
3-trifluoro-
H
methyl
ethyl




methoxy-5-







isopropoxy-







phenyl






2.1.1123
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-isopropoxy-







phenyl






2.1.1124
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







isopropoxy-







phenyl






2.1.1125
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







isopropoxy-







phenyl






2.1.1126
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







isopropoxy-







phenyl






2.1.1127
3-nitro-5-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.1128
3-acetoxy-5-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.1129
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-isopropoxy-







phenyl}






2.1.1130
3-methyl-
H
methyl
ethyl




sulfanyl-5-







isopropoxy-







phenyl






2.1.1131
3,5-di(tert-
H
methyl
ethyl




butoxy)phenyl






2.1.1132
3-difluoro-
H
methyl
ethyl




methoxy-5-tert-







butoxyphenyl






2.1.1133
3-trifluoro-
H
methyl
ethyl




methoxy-5-tert-







butoxyphenyl






2.1.1134
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-tert-butoxy-







phenyl






2.1.1135
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-tert-







butoxylphenyl






2.1.1136
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-tert-







butoxyphenyl






2.1.1137
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







tert-butoxy-







phenyl






2.1.1138
3-nitro-5-tert-
H
methyl
ethyl




butoxyphenyl






2.1.1139
3-acetoxy-5-tert-
H
methyl
ethyl




butoxyphenyl






2.1.1140
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-tert-butoxy-







phenyl}






2.1.1141
3-methyl-
H
methyl
ethyl




sulfanyl-5-tert-







butoxyphenyl






2.1.1142
3,5-di(trifluoro-
H
methyl
ethyl




methoxy)phenyl






2.1.1143
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-trifluoro-







methoxyphenyl






2.1.1144
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







trifluoromethoxy-







phenyl






2.1.1145
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







trifluoro-







methoxyphenyl






2.1.1146
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







trifluoro-







methoxyphenyl






2.1.1147
3-nitro-5-
H
methyl
ethyl




trifluoro-







methoxyphenyl






2.1.1148
3-acetoxy-5-tert-
H
methyl
ethyl




butoxyphenyl






2.1.1149
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-trifluoro-







methoxyphenyl}






2.1.1150
3-methyl-
H
methyl
ethyl




sulfanyl-5-







trifluoro-







methoxyphenyl






2.1.1151
3,5-bis(difluoro-
H
methyl
ethyl




methoxy)phenyl






2.1.1152
3-trifluoro-
H
methyl
ethyl




methoxy-5-







difluoromethoxy-







phenyl






2.1.1153
3-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







5-difluoro-







methoxyphenyl






2.1.1154
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-







difluoromethoxy-







phenyl






2.1.1155
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-







difluoromethoxy-







phenyl






2.1.1156
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







difluoromethoxy-







phenyl






2.1.1157
3-nitro-5-
H
methyl
ethyl




difluoro-







methoxyphenyl






2.1.1158
3-acetoxy-5-
H
methyl
ethyl




difluoro-







methoxyphenyl






2.1.1159
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-difluoro-







methoxyphenyl}






2.1.1160
3-methyl-
H
methyl
ethyl




sulfanyl-5-







difluoromethoxy-







phenyl






2.1.1161
3,5-bis(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







phenyl






2.1.1162
3-(2-chloro-
H
methyl
ethyl




ethoxy)-5-(2,2,2-







trifluoro-







ethoxy)phenyl






2.1.1163
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-(2,2,2-







trifluoro-







ethoxy)phenyl






2.1.1164
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







(2,2,2-trifluoro-







ethoxy)phenyl






2.1.1165
3-nitro-5--(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







phenyl






2.1.1166
3-acetoxy-5-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxy)phenyl






2.1.1167
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-(2,2,2-







trifluoroethoxy)-







phenyl}






2.1.1168
3-methyl-
H
methyl
ethyl




sulfanyl-5-







(2,2,2-trifluoro-







ethoxy)phenyl






2.1.1169
3,5-bis(2-
H
methyl
ethyl




chloroethoxy)-







phenyl






2.1.1170
3-(2-hydroxy-
H
methyl
ethyl




ethoxy)-5-(2-







chloroethoxy)-







phenyl






2.1.1171
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







(2-chloro-







ethoxy)phenyl






2.1.1172
3-nitro-5-(2-
H
methyl
ethyl




chloroethoxy)-







phenyl






2.1.1173
3-acetoxy-5-(2-
H
methyl
ethyl




chloroethoxy)-







phenyl






2.1.1174
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-(2-chloro-







ethoxy)phenyl}






2.1.1175
3-methyl-
H
methyl
ethyl




sulfanyl-5-(2-







chloroethoxy)-







phenyl






2.1.1176
3,5-bis(2-
H
methyl
ethyl




hydroxy-







ethoxy)phenyl






2.1.1177
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)oxy]-5-







(2-hydroxy-







ethoxy)phenyl






2.1.1178
3-nitro-5-(2-
H
methyl
ethyl




hydroxy-







ethoxy)phenyl






2.1.1179
3-acetoxy-5-(2-
H
methyl
ethyl




hydroxyethoxy)-







phenyl






2.1.1180
3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-(2-hydroxy-







ethoxy)-phenyl






2.1.1181
3-methyl-
H
methyl
ethyl




sulfanyl-5-(2-







hydroxyethoxy)-







phenyl






2.1.1182
3,5-bis[(tert-
H
methyl
ethyl




butoxy-







carbonyl)oxy]-







phenyl






2.1.1183
3-nitro-5-[(tert-
H
methyl
ethyl




butoxy-







carbonyl)oxy]-







phenyl






2.1.1184
3-acetoxy-5-
H
methyl
ethyl




[(tert-butoxy-







carbonyl)oxy]-







phenyl






2.1.1185
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5[(tert-butoxy-







carbonyl)oxy]-







phenyl)






2.1.1186
3,5-
H
methyl
ethyl




bis(acetoxy)-







phenyl






2.1.1187
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-acetoxy-







phenyl}






2.1.1188
3-methyl-
H
methyl
ethyl




sulfanyl-5-







acetoxyphenyl






2.1.1189
3,5-dinitrophenyl
H
methyl
ethyl



2.1.1190
3-acetoxy-5-
H
methyl
ethyl




nitrophenyl






2.1.1191
{3-[(tert-butoxy-
H
methyl
ethyl




carbonyl)amino]-







5-nitrophenyl}






2.1.1192
3-methyl-
H
methyl
ethyl




sulfanyl-5-







nitrophenyl






2.1.1193
3,5-bis[(tert-
H
methyl
ethyl




butoxycarbonyl)-







amino]phenyl






2.1.1194
3-methyl-
H
methyl
ethyl




sulfanyl-5-[(tert-







butoxy-







carbonyl)amino]







phenyl






2.1.1195
3,5-di(methyl-
H
methyl
ethyl




sulfanyl)phenyl






2.1.1196
3,4-difluoro-
H
methyl
ethyl
[CDCl3] 1.35 (t, 3H); 1.72 (s,



phenyl



3H); 3.15 (d, 1H); 3.86 (d, 1H);







4.25 (m, 2H); 7.20 (m, 1H); 7.35







(m, 1H); 7.52 (m, 1H).


2.1.1197
3,4-difluoro-
H
ethyl
ethyl
[CDCl3] 1.0 (t, 3H); 1.32 (t, 3H);



phenyl



2.08 (q, 2H); 3.18 (d, 1H); 3.80







(d, 1H); 4.25 (m, 2H); 7.22 (m,







1H); 7.38 (m, 1H); 7.52 (m, 1H).


2.1.1198
3,4-difluoro-
H
isopropyl
ethyl




phenyl






2.1.1199
3,4-difluoro-
H
cyclo-
ethyl




phenyl

propyl




2.1.1200
3-chloro-4-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.71 (s,



fluorophenyl



3H); 3.15 (d, 1H); 3.82 (d, 1H);







4.25 (m, 2H); 7.18 (t, 1H); 7.55







(m, 1H); 7.70 (m, 1H).


2.1.1201
3-chloro-4-
H
ethyl
ethyl




fluorophenyl






2.1.1202
3-chloro-4-
H
isopropyl
ethyl




fluorophenyl






2.1.1203
3-chloro-4-
H
cyclo-
ethyl




fluorophenyl

propyl




2.1.1204
3-bromo-4-
H
methyl
ethyl




fluorophenyl






2.1.1205
3-methyl-4-
H
methyl
ethyl




fluorophenyl






2.1.1206
3-ethyl-4-
H
methyl
ethyl




fluorophenyl






2.1.1207
3-cyclopropyl-4-
H
methyl
ethyl




fluorophenyl






2.1.1208
3-vinyl-4-
H
methyl
ethyl




fluorophenyl






2.1.1209
3-ethynyl-4-
H
methyl
ethyl




fluorophenyl






2.1.1210
3-cyano-4-
H
methyl
ethyl




fluorophenyl






2.1.1211
3-methoxy-4-
H
methyl
ethyl




fluorophenyl






2.1.1212
3-ethoxy-4-
H
methyl
ethyl




fluorophenyl






2.1.1213
3-trifluoro-
H
methyl
ethyl




methoxy-4-







fluorophenyl






2.1.1214
3-nitro-4-
H
methyl
ethyl




fluorophenyl






2.1.1215
3-fluoro-4-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.71 (s,



chlorophenyl



3H); 3.15 (d, 1H); 3.85 (d, 1H);







4.25 (m, 2H); 7.40-7.50 (m, 3H).


2.1.1216
3,4-dichloro-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.72 (s,



phenyl



3H); 3.15 (d, 1H); 3.84 (d, 1H);







4.25 (mc, 2H); 7.5 (mc, 2H);







7.71 (s, 1H)


2.1.1217
3-bromo-4-
H
methyl
ethyl




chlorophenyl






2.1.1218
3-methyl-4-
H
methyl
ethyl




chlorophenyl






2.1.1219
3-ethyl-4-
H
methyl
ethyl




chlorophenyl






2.1.1220
3-cyclopropyl-4-
H
methyl
ethyl




chlorophenyl






2.1.1221
3-vinyl-4-
H
methyl
ethyl




chlorophenyl






2.1.1222
3-ethynyl-4-
H
methyl
ethyl




chlorophenyl






2.1.1223
3-cyano-4-
H
methyl
ethyl




chlorophenyl






2.1.1224
3-trifluoro-
H
methyl
ethyl




methyl-4-







chlorophenyl






2.1.1225
3-methoxy-4-
H
methyl
ethyl




chlorophenyl






2.1.1226
3-ethoxy-4-
H
methyl
ethyl




chlorophenyl






2.1.1227
3-trifluoro-
H
methyl
ethyl




methoxy-4-







chlorophenyl






2.1.1228
3-nitro-4-
H
methyl
ethyl




chlorophenyl






2.1.1229
3-fluoro-4-
H
methyl
ethyl




bromophenyl






2.1.1230
3-chloro-4-
H
methyl
ethyl




bromophenyl






2.1.1231
3,4-dibromo-
H
methyl
ethyl




phenyl






2.1.1232
3-methyl-4-
H
methyl
ethyl




bromophenyl






2.1.1233
3-ethyl-4-
H
methyl
ethyl




bromophenyl






2.1.1234
3-cyclopropyl-4-
H
methyl
ethyl




bromophenyl






2.1.1235
3-vinyl-4-
H
methyl
ethyl




bromophenyl






2.1.1236
3-ethynyl-4-
H
methyl
ethyl




bromophenyl






2.1.1237
3-cyano-4-
H
methyl
ethyl




bromophenyl






2.1.1238
3-trifluoro-
H
methyl
ethyl




methyl-4-







bromophenyl






2.1.1239
3-methoxy-4-
H
methyl
ethyl




phenyl






2.1.1240
3-ethoxy-4-
H
methyl
ethyl




bromophenyl






2.1.1241
3-trifluoro-
H
methyl
ethyl




methoxy-4-







bromophenyl






2.1.1242
3-nitro-4-
H
methyl
ethyl




bromophenyl






2.1.1243
3-fluoro-4-
H
methyl
ethyl




iodophenyl






2.1.1244
3-chloro-4-
H
methyl
ethyl




iodophenyl






2.1.1245
3-bromo-4-
H
methyl
ethyl




iodophenyl






2.1.1246
3-methyl-4-
H
methyl
ethyl




iodophenyl






2.1.1247
3-ethyl-4-
H
methyl
ethyl




iodophenyl






2.1.1248
3-cyclopropyl-4-
H
methyl
ethyl




iodophenyl






2.1.1249
3-vinyl-4-
H
methyl
ethyl




iodophenyl






2.1.1250
3-ethynyl-4-
H
methyl
ethyl




iodophenyl






2.1.1251
3-cyano-4-
H
methyl
ethyl




iodophenyl






2.1.1252
3-trifluoro-
H
methyl
ethyl




methyl-4-







iodophenyl






2.1.1253
3-methoxy-4-
H
methyl
ethyl




iodophenyl






2.1.1254
3-ethoxy-4-
H
methyl
ethyl




iodophenyl






2.1.1255
3-trifluoro-
H
methyl
ethyl




methoxy-4-







iodophenyl






2.1.1256
3-nitro-4-
H
methyl
ethyl




iodophenyl






2.1.1257
3-fluoro-4-
H
methyl
ethyl




methylphenyl






2.1.1258
3-chloro-4-
H
methyl
ethyl
[CDCl3] 1.32 t, 3H); 1.70 (s, 3H);



methylphenyl



2.41 (s, 3H); 3.15 (d, 1H); 3.85







(d, 1H); 4.25 (m, 2H); 7.24 (m,







1H); 7.45 (m, 1H); 7.61 (s, 1H).


2.1.1259
3-bromo-4-
H
methyl
ethyl




methylphenyl






2.1.1260
3,4-dimethyl-
H
methyl
ethyl




phenyl






2.1.1261
3,4-dimethyl-
H
ethyl
ethyl




phenyl






2.1.1262
3,4-dimethyl-
H
isopropyl
ethyl




phenyl






2.1.1263
3,4-dimethyl-
H
cyclo
ethyl




phenyl

propyl




2.1.1264
3-ethyl-4-
H
methyl
ethyl




methylphenyl






2.1.1265
3-cyclopropyl-4-
H
methyl
ethyl




methylphenyl






2.1.1266
3-vinyl-4-
H
methyl
ethyl




methylphenyl






2.1.1267
3-ethynyl-4-
H
methyl
ethyl




methylphenyl






2.1.1268
3-cyano-4-
H
methyl
ethyl




methylphenyl






2.1.1269
3-trifluoro-
H
methyl
ethyl




methyl-4-







methylphenyl






2.1.1270
3-methoxy-4-
H
methyl
ethyl




methylphenyl






2.1.1271
3-ethoxy-4-
H
methyl
ethyl




methylphenyl






2.1.1272
3-trifluoro-
H
methyl
ethyl




methoxy-4-







methylphenyl






2.1.1273
3-nitro-4-
H
methyl
ethyl




methylphenyl






2.1.1274
3-fluoro-4-
H
methyl
ethyl




ethylphenyl






2.1.1275
3-chloro-4-
H
methyl
ethyl




ethylphenyl






2.1.1276
3-bromo-4-
H
methyl
ethyl




ethylphenyl






2.1.1277
3-methyl-4-
H
methyl
ethyl




ethylphenyl






2.1.1278
3,4-diethyl-
H
methyl
ethyl




phenyl






2.1.1279
3-cyclopropyl-4-
H
methyl
ethyl




ethylphenyl






2.1.1280
3-vinyl-4-
H
methyl
ethyl




ethylphenyl






2.1.1281
3-ethynyl-4-
H
methyl
ethyl




ethylphenyl






2.1.1282
3-cyano-4-
H
methyl
ethyl




ethylphenyl






2.1.1283
3-trifluoro-
H
methyl
ethyl




methyl-4-







ethylphenyl






2.1.1284
3-methoxy-4-
H
methyl
ethyl




ethylphenyl






2.1.1285
3-ethoxy-4-
H
methyl
ethyl




ethylphenyl






2.1.1286
3-trifluoro-
H
methyl
ethyl




methoxy-4-







ethylphenyl






2.1.1287
3-nitro-4-
H
methyl
ethyl




ethylphenyl






2.1.1288
3-fluoro-4-
H
methyl
ethyl




propylphenyl






2.1.1289
3-chloro-4-
H
methyl
ethyl




propylphenyl






2.1.1290
3-bromo-4-
H
methyl
ethyl




propylphenyl






2.1.1291
3-methyl-4-
H
methyl
ethyl




propylphenyl






2.1.1292
3-methyl-4-
H
methyl
ethyl




propylphenyl






2.1.1293
3-cyclopropyl-4-
H
methyl
ethyl




propylphenyl






2.1.1294
3-vinyl-4-
H
methyl
ethyl




propylphenyl






2.1.1295
3-ethynyl-4-
H
methyl
ethyl




propylphenyl






2.1.1296
3-cyano-4-
H
methyl
ethyl




propylphenyl






2.1.1297
3-trifluoro-
H
methyl
ethyl




methyl-4-







propylphenyl






2.1.1298
3-methoxy-4-
H
methyl
ethyl




propylphenyl






2.1.1299
3-ethoxy-4-
H
methyl
ethyl




propylphenyl






2.1.1300
3-trifluoro-
H
methyl
ethyl




methoxy-4-







propylphenyl






2.1.1301
3-nitro-4-
H
methyl
ethyl




propylphenyl






2.1.1302
3-fluoro-4-
H
methyl
ethyl




isopropylphenyl






2.1.1303
3-chloro-4-
H
methyl
ethyl




isopropylphenyl






2.1.1304
3-bromo-4-
H
methyl
ethyl




isopropylphenyl






2.1.1305
3-methyl-4-
H
methyl
ethyl




isopropylphenyl






2.1.1306
3-ethyl-4-
H
methyl
ethyl




isopropylphenyl






2.1.1307
3-cyclopropyl-4-
H
methyl
ethyl




isopropylphenyl






2.1.1308
3-vinyl-4-
H
methyl
ethyl




isopropylphenyl






2.1.1309
3-ethynyl-4-
H
methyl
ethyl




isopropylphenyl






2.1.1310
3-cyano-4-
H
methyl
ethyl




isopropylphenyl






2.1.1311
3-trifluoro-
H
methyl
ethyl




methyl-4-







isopropyl-phenyl






2.1.1312
3-methoxy-4-
H
methyl
ethyl




isopropylphenyl






2.1.1313
3-thoxy-4-
H
methyl
ethyl




isopropylphenyl






2.1.1314
3-trifluoro-
H
methyl
ethyl




methoxy-4-







isopropyl-phenyl






2.1.1315
3-nitro-4-
H
methyl
ethyl




isopropylphenyl






2.1.1316
3-fluoro-4-tert-
H
methyl
ethyl




butylphenyl






2.1.1317
3-chloro-4-tert-
H
methyl
ethyl




butylphenyl






2.1.1318
3-bromo-4-tert-
H
methyl
ethyl




butylphenyl






2.1.1319
3-methyl-4-tert-
H
methyl
ethyl




butylphenyl






2.1.1320
3-ethyl-4-tert-
H
methyl
ethyl




butylphenyl






2.1.1321
3-cyclopropyl-4-
H
methyl
ethyl




tert-butylphenyl






2.1.1322
3-vinyl-4-tert-
H
methyl
ethyl




butylphenyl






2.1.1323
3-ethynyl-4-tert-
H
methyl
ethyl




butylphenyl






2.1.1324
3-cyano-4-tert-
H
methyl
ethyl




butylphenyl






2.1.1325
3-trifluoro-
H
methyl
ethyl




methyl-4-tert-







butylphenyl






2.1.1326
3-methoxy-4-
H
methyl
ethyl




tert-butylphenyl






2.1.1327
3-ethoxy-4-tert-
H
methyl
ethyl




butylphenyl






2.1.1328
3-trifluoro-
H
methyl
ethyl




methoxy-4-tert-







butylphenyl






2.1.1329
3-nitro-4-tert-
H
methyl
ethyl




butylphenyl






2.1.1330
3-fluoro-4-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1331
3-chloro-4-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1332
3-bromo-4-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1333
3-methyl-4-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1334
3-ethyl-4-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1335
3-cyclopropyl-4-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1336
3-vinyl-4-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1337
3-ethynyl-4-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1338
3-cyano-4-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1339
3-trifluoro-
H
methyl
ethyl




methyl-4-







hydroxymethyl-







phenyl






2.1.1340
3-methoxy-4-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1341
3-ethoxy-4-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1342
3-trifluoro-
H
methyl
ethyl




methoxy-4-







hydroxymethyl-







phenyl






2.1.1343
3-nitro-4-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1344
3-fluoro-4-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.1345
3-chloro-4-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.1346
3-bromo-4-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.1347
3-methyl-4-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.1348
3-ethyl-4-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.1349
3-cyclopropyl-4-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.1350
3-vinyl-4-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.1351
3-ethynyl-4-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.1352
3-cyano-4-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.1353
3-trifluoro-
H
methyl
ethyl




methyl-4-







cyclopropyl-







phenyl






2.1.1354
3-methoxy-4-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.1355
3-ethoxy-4-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.1356
3-trifluoro-
H
methyl
ethyl




methoxy-4-







cyclopropyl-







phenyl






2.1.1357
3-fluoro-4-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1358
3-chloro-4-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1359
3-bromo-4-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1360
3-methyl-4-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1361
3-ethyl-4-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1362
3-cyclopropyl-4-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1363
3-vinyl-4-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1364
3-ethynyl-4-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1365
3-cyano-4-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1366
3-trifluoro-
H
methyl
ethyl




methyl-4-







methoxy-







carbonylphenyl






2.1.1367
3-methoxy-4-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1368
3-ethoxy-4-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1369
3-trifluoro-
H
methyl
ethyl




methoxy-4-







methoxy-







carbonylphenyl






2.1.1370
3-nitro-4-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1371
3-fluoro-4-
H
methyl
ethyl




vinylphenyl






2.1.1372
3-chloro-4-
H
methyl
ethyl




vinylphenyl






2.1.1373
3-bromo-4-
H
methyl
ethyl




vinylphenyl






2.1.1374
3-methyl-4-
H
methyl
ethyl




vinylphenyl






2.1.1375
3-ethyl-4-
H
methyl
ethyl




vinylphenyl






2.1.1376
3-cyclopropyl-4-
H
methyl
ethyl




vinylphenyl






2.1.1377
3-vinyl-4-
H
methyl
ethyl




vinylphenyl






2.1.1378
3-ethynyl-4-
H
methyl
ethyl




vinylphenyl






2.1.1379
3-cyano-4-
H
methyl
ethyl




vinylphenyl






2.1.1380
3-trifluoro-
H
methyl
ethyl




methyl-4-







vinylphenyl






2.1.1381
3-methoxy-4-
H
methyl
ethyl




vinylphenyl






2.1.1382
3-ethoxy-4-
H
methyl
ethyl




vinylphenyl






2.1.1383
3-trifluoro-
H
methyl
ethyl




methoxy-4-







vinylphenyl






2.1.1384
3-nitro-4-
H
methyl
ethyl




vinylphenyl






2.1.1385
3-fluoro-4-
H
methyl
ethyl




ethynylphenyl






2.1.1386
3-chloro-4-
H
methyl
ethyl




ethynylphenyl






2.1.1387
3-bromo-4-
H
methyl
ethyl




ethynylphenyl






2.1.1388
3-methyl-4-
H
methyl
ethyl




ethynylphenyl






2.1.1389
3-ethyl-4-
H
methyl
ethyl




ethynylphenyl






2.1.1390
3-cyclopropyl-4-
H
methyl
ethyl




ethynylphenyl






2.1.1391
3-vinyl-4-
H
methyl
ethyl




ethynylphenyl






2.1.1392
3-cyano-4-
H
methyl
ethyl




ethynylphenyl






2.1.1393
3-trifluoro-
H
methyl
ethyl




methyl-4-







ethynylphenyl






2.1.1394
3-methoxy-4-
H
methyl
ethyl




ethynylphenyl






2.1.1395
3-ethoxy-4-
H
methyl
ethyl




ethynylphenyl






2.1.1396
3-trifluoro-
H
methyl
ethyl




methoxy-4-







ethynylphenyl






2.1.1397
3-nitro-4-
H
methyl
ethyl




ethynylphenyl






2.1.1398
3-fluoro-4-
H
methyl
ethyl




ethynylphenyl






2.1.1399
3-fluoro-4-
H
methyl
ethyl




cyanophenyl






2.1.1400
3-chloro-4-
H
methyl
ethyl




cyanophenyl






2.1.1401
3-bromo-4-
H
methyl
ethyl




cyanophenyl






2.1.1402
3-methyl-4-
H
methyl
ethyl




cyanophenyl






2.1.1403
3-ethyl-4-
H
methyl
ethyl




cyanophenyl






2.1.1404
3-cyclopropyl-4-
H
methyl
ethyl




cyanophenyl






2.1.1405
3-vinyl-4-
H
methyl
ethyl




cyanophenyl






2.1.1406
3-ethynyl-4-
H
methyl
ethyl




cyanophenyl






2.1.1407
3-cyano-4-
H
methyl
ethyl




cyanophenyl






2.1.1408
3-trifluoro-
H
methyl
ethyl




methyl-4-







cyanophenyl






2.1.1409
3-trifluoro-
H
ethyl
ethyl




methyl-4-







cyanophenyl






2.1.1410
3-trifluoro-
H
isopropyl
ethyl




methyl-4-







cyanophenyl






2.1.1411
3-trifluoro-
H
cyclo-
ethyl




methyl-4-

propyl





cyanophenyl






2.1.1412
3-methoxy-4-
H
methyl
ethyl




cyanophenyl






2.1.1413
3-ethoxy-4-
H
methyl
ethyl




cyanophenyl






2.1.1414
3-trifluoro-
H
methyl
ethyl




methoxy-4-







cyanophenyl






2.1.1415
3-nitro-4-
H
methyl
ethyl




cyanophenyl






2.1.1416
3-fluoro-4-
H
methyl
ethyl




hydroxyphenyl






2.1.1417
3-chloro-4-
H
methyl
ethyl




hydroxyphenyl






2.1.1418
3-bromo-4-
H
methyl
ethyl




hydroxyphenyl






2.1.1419
3-methyl-4-
H
methyl
ethyl




hydroxyphenyl






2.1.1420
3-ethyl-4-
H
methyl
ethyl




hydroxyphenyl






2.1.1421
3-cyclopropyl-4-
H
methyl
ethyl




hydroxyphenyl






2.1.1422
3-vinyl-4-
H
methyl
ethyl




hydroxyphenyl






2.1.1423
3-ethynyl-4-
H
methyl
ethyl




hydroxyphenyl






2.1.1424
3-cyano-4-
H
methyl
ethyl




hydroxyphenyl






2.1.1425
3-trifluoro-
H
methyl
ethyl




methyl-4-







hydroxyphenyl






2.1.1426
3-methoxy-4-
H
methyl
ethyl




hydroxyphenyl






2.1.1427
3-ethoxy-4-
H
methyl
ethyl




hydroxyphenyl






2.1.1428
3-trifluoro-
H
methyl
ethyl




methoxy-4-







hydroxyphenyl






2.1.1429
3-nitro-4-
H
methyl
ethyl




hydroxyphenyl






2.1.1430
3-fluoro-4-
H
methyl
ethyl




methoxyphenyl






2.1.1431
3-chloro-4-
H
methyl
ethyl




methoxyphenyl






2.1.1432
3-bromo-4-
H
methyl
ethyl




methoxyphenyl






2.1.1433
3-methyl-4-
H
methyl
ethyl




methoxyphenyl






2.1.1434
3-ethyl-4-
H
methyl
ethyl




methoxyphenyl






2.1.1435
3-cyclopropyl-4-
H
methyl
ethyl




methoxyphenyl






2.1.1436
3-vinyl-4-
H
methyl
ethyl




methoxyphenyl






2.1.1437
3-ethynyl-4-
H
methyl
ethyl




methoxyphenyl






2.1.1438
3-cyano-4-
H
methyl
ethyl




methoxyphenyl






2.1.1439
3-trifluoro-
H
methyl
ethyl




methyl-4-







methoxyphenyl






2.1.1440
3,4-dimethoxy--
H
methyl
ethyl




phenyl






2.1.1441
3-ethoxy-4-
H
methyl
ethyl




methoxyphenyl






2.1.1442
3-trifluoro-
H
methyl
ethyl




methoxy-4-







methoxyphenyl






2.1.1443
3-nitro-4-
H
methyl
ethyl




methoxyphenyl






2.1.1444
3-fluoro-4-
H
methyl
ethyl




ethoxyphenyl






2.1.1445
3-chloro-4-
H
methyl
ethyl




ethoxyphenyl






2.1.1446
3-bromo-4-
H
methyl
ethyl




ethoxyphenyl






2.1.1447
3-methyl-4-
H
methyl
ethyl




ethoxyphenyl






2.1.1448
3-ethyl-4-
H
methyl
ethyl




ethoxyphenyl






2.1.1449
3-cyclopropyl-4-
H
methyl
ethyl




ethoxyphenyl






2.1.1450
3-vinyl-4-
H
methyl
ethyl




ethoxyphenyl






2.1.1451
3-ethynyl-4-
H
methyl
ethyl




ethoxyphenyl






2.1.1452
3-cyano-4-
H
methyl
ethyl




ethoxyphenyl






2.1.1453
3-trifluoro-
H
methyl
ethyl




methyl-4-







ethoxyphenyl






2.1.1454
3-methoxy-4-
H
methyl
ethyl




ethoxyphenyl






2.1.1455
2,4-diethoxy--
H
methyl
ethyl




phenyl






2.1.1456
3-trifluoro-
H
methyl
ethyl




methoxy-4-







ethoxyphenyl






2.1.1457
3-nitro-4-
H
methyl
ethyl




ethoxyphenyl






2.1.1458
3-fluoro-4-
H
methyl
ethyl




propoxyphenyl






2.1.1459
3-chloro-4-
H
methyl
ethyl




propoxyphenyl






2.1.1460
3-bromo-4-
H
methyl
ethyl




propoxyphenyl






2.1.1461
3-methyl-4-
H
methyl
ethyl




propoxyphenyl






2.1.1462
3-ethyl-4-
H
methyl
ethyl




propoxyphenyl






2.1.1463
3-cyclopropyl-4-
H
methyl
ethyl




propoxyphenyl






2.1.1464
3-vinyl-4-
H
methyl
ethyl




propoxyphenyl






2.1.1465
3-ethynyl-4-
H
methyl
ethyl




propoxyphenyl






2.1.1466
3-cyano-4-
H
methyl
ethyl




propoxyphenyl






2.1.1467
3-trifluoro-
H
methyl
ethyl




methyl-4-







propoxyphenyl






2.1.1468
3-methoxy-4-
H
methyl
ethyl




propoxyphenyl






2.1.1469
3-ethoxy-4-
H
methyl
ethyl




propoxyphenyl






2.1.1470
3-trifluoro-
H
methyl
ethyl




methoxy-4-







propoxyphenyl






2.1.1471
3-nitro-4-
H
methyl
ethyl




propoxyphenyl






2.1.1472
3-fluoro-4-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.1473
3-chloro-4-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.1474
3-bromo-4-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.1475
3-methyl-4-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.1476
3-ethyl-4-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.1477
3-cyclopropyl-4-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.1478
3-vinyl-4-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.1479
3-ethynyl-4-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.1480
3-cyano-4-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.1481
3-trifluoro-
H
methyl
ethyl




methyl-4-







isopropoxy-







phenyl






2.1.1482
3-methoxy-4-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.1483
3-ethoxy-4-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.1484
3-trifluoro-
H
methyl
ethyl




methoxy-4-







isopropoxy-







phenyl






2.1.1485
3-nitro-4-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.1486
3-fluoro-4-tert-
H
methyl
ethyl




butoxyphenyl






2.1.1487
3-chloro-4-tert-
H
methyl
ethyl




butoxyphenyl






2.1.1488
3-bromo-4-tert-
H
methyl
ethyl




butoxyphenyl






2.1.1489
3-methyl-4-tert-
H
methyl
ethyl




butoxyphenyl






2.1.1490
3-ethyl-4-tert-
H
methyl
ethyl




butoxyphenyl






2.1.1491
3-cyclopropyl-4-
H
methyl
ethyl




tert-butoxy-







phenyl






2.1.1492
3-vinyl-4-tert-
H
methyl
ethyl




butoxyphenyl






2.1.1493
3-ethynyl-4-tert-
H
methyl
ethyl




butoxyphenyl






2.1.1494
3-cyano-4-tert-
H
methyl
ethyl




butoxyphenyl






2.1.1495
3-trifluoro-
H
methyl
ethyl




methyl-4-tert-







butoxyphenyl






2.1.1496
3-methoxy-4-
H
methyl
ethyl




tert-butoxy-







phenyl






2.1.1497
3-ethoxy-4-tert-
H
methyl
ethyl




butoxyphenyl






2.1.1498
3-trifluoro-
H
methyl
ethyl




methoxy-4-tert-







butoxyphenyl






2.1.1499
3-nitro-4-tert-
H
methyl
ethyl




butoxyphenyl






2.1.1500
3-fluoro-4-
H
methyl
ethyl




trifluoro-







methoxyphenyl






2.1.1501
3-chloro-4-
H
methyl
ethyl




trifluoro-







methoxyphenyl






2.1.1502
3-bromo-4-
H
methyl
ethyl




trifluoro-







methoxyphenyl






2.1.1503
3-methyl-4-
H
methyl
ethyl




trifluoro-







methoxyphenyl






2.1.1504
3-ethyl-4-
H
methyl
ethyl




trifluoro-







methoxyphenyl






2.1.1505
3-cyclopropyl-4-
H
methyl
ethyl




trifluoro-







methoxyphenyl






2.1.1506
3-vinyl-4-
H
methyl
ethyl




trifluoro-







methoxyphenyl






2.1.1507
3-ethynyl-4-
H
methyl
ethyl




trifluoro-







methoxyphenyl






2.1.1508
3-cyano-4-
H
methyl
ethyl




trifluoro-







methoxyphenyl






2.1.1509
3-trifluoro-
H
methyl
ethyl




methyl-4-







trifluoro-







methoxyphenyl






2.1.1510
3-methoxy-4-
H
methyl
ethyl




trifluoro-







methoxyphenyl






2.1.1511
3-ethoxy-4-
H
methyl
ethyl




trifluoro-







methoxyphenyl






2.1.1512
3,4-bis(trifluoro-
H
methyl
ethyl




methoxy)phenyl






2.1.1513
3-nitro-4-
H
methyl
ethyl




trifluoro-







methoxyphenyl






2.1.1514
3-fluoro-4-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxy)phenyl






2.1.1515
3-chloro-4-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxy)phenyl






2.1.1516
3-bromo-4-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxy)phenyl






2.1.1517
3-methyl-4-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxy)phenyl






2.1.1518
3-ethyl-4-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







phenyl






2.1.1519
3-cyclopropyl-4-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxy)phenyl






2.1.1520
3-vinyl-4-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







phenyl






2.1.1521
3-ethynyl-4-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxyphenyl






2.1.1522
3-cyano-4-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxy)phenyl






2.1.1523
3-trifluoro-
H
methyl
ethyl




methyl-4-(2,2,2 -







trifluoroethoxy)-







phenyl






2.1.1524
3-methoxy-4-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxy)phenyl






2.1.1525
3-ethoxy-4-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxy)phenyl






2.1.1526
3-trifluoro-
H
methyl
ethyl




methoxy-4-







(2,2,2-trifluoro-







ethoxy)phenyl






2.1.1527
3-nitro-4-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







phenyl






2.1.1528
3-fluoro-4-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.1529
3-chloro-4-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.1530
3-bromo-4-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.1531
3-methyl-4-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.1532
3-ethyl-4-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.1533
3-cyclopropyl-4-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.1534
3-vinyl-4-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.1535
3-ethynyl-4-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.1536
3-cyano-4-
H
methyl
ethyl




difluoromethoxy







phenyl






2.1.1537
3-trifluoro-
H
methyl
ethyl




methyl-4-







difluoromethoxy







phenyl






2.1.1538
3-methoxy-4-
H
methyl
ethyl




difluoromethoxy







phenyl






2.1.1539
3-ethoxy-4-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.1540
3-trifluoro-
H
methyl
ethyl




methoxy-4-







difluoromethoxy-







phenyl






2.1.1541
3-nitro-4-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.1542
3-fluoro-4-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.1543
3-chloro-4-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.1544
3-bromo-4-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.1545
3-methyl-4-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.1546
3-ethyl-4-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.1547
3-cyclopropyl-4-
H
methyl
ethyl




(2-methoxy-







ethoxy)phenyl






2.1.1548
3-vinyl-4-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.1549
3-ethynyl-4-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.1550
3-cyano-4-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.1551
3-trifluoro-
H
methyl
ethyl




methyl-4-(2-







methoxyethoxy)-







phenyl






2.1.1552
3-methoxy-4-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.1553
3-ethoxy-4-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.1554
3-trifluoro-
H
methyl
ethyl




methoxy-(2-







methoxyethoxy)-







phenyl






2.1.1555
3-nitro-4-(2-
H
methyl
ethyl




methoxy-







ethoxy)phenyl






2.1.1556
3-fluoro-4-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.1557
3-chloro-4-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.1558
3-bromo-4-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.1559
3-methyl-4-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.1560
3-ethyl-4-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.1561
3-cyclopropyl-4-
H
methyl
ethyl




(tert-butoxy-







carbonyloxy)-







phenyl






2.1.1562
3-vinyl-4-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.1563
3-ethynyl-4-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.1564
3-cyano-4-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.1565
3-trifluoro-
H
methyl
ethyl




methyl-4-(tert-







butoxycarbonyl-







oxy)phenyl






2.1.1566
3-methoxy-4-
H
methyl
ethyl




(tert-butoxy-







carbonyloxy)-







phenyl






2.1.1567
3-ethoxy-4-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.1568
3-trifluoro-
H
methyl
ethyl




methoxy-4-(tert-







butoxycarbonyl-







oxy)phenyl






2.1.1569
2-nitro-4-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.1570
3-fluoro-4-
H
methyl
ethyl




nitrophenyl






2.1.1571
3-chloro-4-
H
methyl
ethyl




nitrophenyl






2.1.1572
3-bromo-4-
H
methyl
ethyl




nitrophenyl






2.1.1573
3-methyl-4-
H
methyl
ethyl




nitrophenyl






2.1.1574
3-ethyl-4-
H
methyl
ethyl




nitrophenyl






2.1.1575
3-cyclopropyl-4-
H
methyl
ethyl




nitrophenyl






2.1.1576
3-vinyl-4-
H
methyl
ethyl




nitrophenyl






2.1.1577
3-ethynyl-4-
H
methyl
ethyl




nitrophenyl






2.1.1578
3-cyano-4-
H
methyl
ethyl




nitrophenyl






2.1.1579
3-trifluoro-
H
methyl
ethyl




methyl-4-







nitrophenyl






2.1.1580
3-methoxy-4-
H
methyl
ethyl




nitrophenyl






2.1.1581
3-ethoxy-4-
H
methyl
ethyl




nitrophenyl






2.1.1582
3-trifluoro-
H
methyl
ethyl




methoxy-4-







nitrophenyl






2.1.1583
3-fluoro-4-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.1584
3-chloro-4-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.1585
3-bromo-4-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.1586
3-methyl-4-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.1587
3-ethyl-4-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.1588
3-cyclopropyl-4-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.1589
3-vinyl-4-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.1590
3-ethynyl-4-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.1591
3-cyano-4-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.1592
3-trifluoro-
H
methyl
ethyl




methyl-4-







methylsulfanyl-







phenyl






2.1.1593
3-methoxy-4-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.1594
3-ethoxy-4-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.1595
3-trifluoro-
H
methyl
ethyl




methoxy-4-







methylsulfanyl-







phenyl






2.1.1596
3-nitro-4-methyl-
H
methyl
ethyl




sulfanylphenyl






2.1.1597
3,6-difluoro-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.70 (s,



phenyl



3H); 3.29 (dd, 1H); 3.92 (dd,







1H); 4.25 (q, 2H); 7.10 (m, 2H);







7.59 (m, 1H).


2.1.1598
3,6-difluoro-
H
ethyl
ethyl




phenyl






2.1.1599
3,6-difluoro-
H
isopropyl
ethyl




phenyl






2.1.1600
3,6-difluoro-
H
cyclo-
ethyl




phenyl

propyl




2.1.1601
3-chloro-6-
H
methyl
ethyl




fluorophenyl






2.1.1602
3-bromo-6-
H
methyl
ethyl
[CDCl3] 1.30 (t, 3H); 1.71 (s,



fluorophenyl



3H); 3.29 (d, 1H); 3.91 (d, 1H);







4.25 (m, 2H); 7.00 (d, 1H); 7.50







(m, 1H); 8.01 (m, 1H).


2.1.1603
3-methyl-6-
H
methyl
ethyl




fluorophenyl






2.1.1604
3-ethyl-6-
H
methyl
ethyl




fluorophenyl






2.1.1605
3-cyclopropyl-6-
H
methyl
ethyl




fluorophenyl






2.1.1606
3-vinyl-6-
H
methyl
ethyl




fluorophenyl






2.1.1607
3-ethynyl-6-
H
methyl
ethyl




fluorophenyl






2.1.1608
3-cyano-6-
H
methyl
ethyl




fluorophenyl






2.1.1609
3-methoxy-6-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.71 (s,



fluorophenyl



3H); 3.31 (dd, 1H); 3.80 (s, 3H);







3.90 (dd, 1H); 4.25 (m, 2H); 6.91







(m, 1H); 7.2 (t, 1H); 7.35 (m,







1H).


2.1.1610
3-ethoxy-6-
H
methyl
ethyl




fluorophenyl






2.1.1611
3-trifluoro-
H
methyl
ethyl




methoxy-6-







fluorophenyl






2.1.1612
3-nitro-6-
H
methyl
ethyl




fluorophenyl






2.1.1613
3-fluoro-6-
H
methyl
ethyl
[CDCl3] 1.35 (t, 3H); 1.75, (s,



chlorophenyl



3H); 3.40 (d, 1H); 3.98 (d, 1H);







4.28 (q, 2H); 7.08 (m, 1H); 7.40







(m; 2H).


2.1.1614
3-fluoro-6-
H
ethyl
ethyl




chlorophenyl






2.1.1615
3-fluoro-6-
H
propyl
ethyl




chlorophenyl






2.1.1616
3-fluoro-6-
H
cyclo-
ethyl




chlorophenyl

propyl




2.1.1617
3,6-dichloro-
H
methyl
ethyl
[CDCl3] 1.33 (t, 3H); 1.72 (s,



phenyl



3H); 3.38 (d, 1H); 3.98 (d, 1H);







4.39 (m, 2H); 7.32 (m, 2H); 7.68







(m, 1H).


2.1.1618
3-bromo-6-
H
methyl
ethyl




chlorophenyl






2.1.1619
3-methyl-6-
H
methyl
ethyl




chlorophenyl






2.1.1620
3-ethyl-6-
H
methyl
ethyl




chlorophenyl






2.1.1621
3-cyclopropyl-6-
H
methyl
ethyl




chlorophenyl






2.1.1622
3-vinyl-6-
H
methyl
ethyl




chlorophenyl






2.1.1623
3-ethynyl-6-
H
methyl
ethyl




chlorophenyl






2.1.1624
3-cyano-6-
H
methyl
ethyl




chlorophenyl






2.1.1625
3-trifluoro-
H
methyl
ethyl




methyl-6-







chlorophenyl






2.1.1626
3-hydroxy-6-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.72 (s,



chlorophenyl



3H); 3.45 (d, 1H); 3.95 (d, 1H);







4.28 (q, 2H); 6.85 (dd, 1H); 7.20







(dd, 1H); 7.28 (m, 1H).


2.1.1627
3-methoxy-6-
H
methyl
ethyl




chlorophenyl






2.1.1628
3-ethoxy-6-
H
methyl
ethyl




chlorophenyl






2.1.1629
3-trifluoro-
H
methyl
ethyl




methoxy-6-







chlorophenyl






2.1.1630
3-nitro-6-
H
methyl
ethyl




chlorophenyl






2.1.1631
3-fluoro-6-
H
methyl
ethyl




bromophenyl






2.1.1632
3-chloro-6-
H
methyl
ethyl




bromophenyl






2.1.1633
3,6-dibromo-
H
methyl
ethyl




phenyl






2.1.1634
3-methyl-6-
H
methyl
ethyl




bromophenyl






2.1.1635
3-ethyl-6-
H
methyl
ethyl




bromophenyl






2.1.1636
3-cyclopropyl-6-
H
methyl
ethyl




bromophenyl






2.1.1637
3-vinyl-6-
H
methyl
ethyl




bromophenyl






2.1.1638
3-ethynyl-6-
H
methyl
ethyl




bromophenyl






2.1.1639
3-cyano-6-
H
methyl
ethyl




bromophenyl






2.1.1640
3-trifluoro-
H
methyl
ethyl




methyl-6-







bromophenyl






2.1.1641
3-methoxy-6-
H
methyl
ethyl




phenyl






2.1.1642
3-ethoxy-6-
H
methyl
ethyl




bromophenyl






2.1.1643
3-trifluoro-
H
methyl
ethyl




methoxy-6-







bromophenyl






2.1.1644
3-nitro-6-
H
methyl
ethyl




bromophenyl






2.1.1645
3-fluoro-6-
H
methyl
ethyl




iodophenyl






2.1.1646
3-chloro-6-
H
methyl
ethyl




iodophenyl






2.1.1647
3-bromo-6-
H
methyl
ethyl




iodophenyl






2.1.1648
3-methyl-6-
H
methyl
ethyl




iodophenyl






2.1.1649
3-ethyl-6-
H
methyl
ethyl




iodophenyl






2.1.1650
3-cyclopropyl-6-
H
methyl
ethyl




iodophenyl






2.1.1651
3-vinyl-6-
H
methyl
ethyl




iodophenyl






2.1.1652
3-ethynyl-6-
H
methyl
ethyl




iodophenyl






2.1.1653
3-cyano-6-
H
methyl
ethyl




iodophenyl






2.1.1654
3-trifluoro-
H
methyl
ethyl




methyl-6-







iodophenyl






2.1.1655
3-methoxy-6-
H
methyl
ethyl




iodophenyl






2.1.1656
3-ethoxy-6-
H
methyl
ethyl




iodophenyl






2.1.1657
3-trifluoro-
H
methyl
ethyl




methoxy-6-







iodophenyl






2.1.1658
3-nitro-6-
H
methyl
ethyl




iodophenyl






2.1.1659
3-fluoro-6-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.72 (s,



methylphenyl



3H); 2.50 (s, 3H); 3.22 (d, 1H);







3.87 (d, 1H); 4.28 (m, 2H); 7.00







(m, 2H); 7.21 (m, 1H).


2.1.1660
3-chloro-6-
H
methyl
ethyl




methylphenyl






2.1.1661
3-bromo-6-
H
methyl
ethyl




methylphenyl






2.1.1662
3,6-
H
methyl
ethyl




dimethylphenyl






2.1.1663
3-ethyl-6-
H
methyl
ethyl




methylphenyl






2.1.1664
3-cyclopropyl-6-
H
methyl
ethyl




methylphenyl






2.1.1665
3-vinyl-6-
H
methyl
ethyl




methylphenyl






2.1.1666
3-ethynyl-6-
H
methyl
ethyl




methylphenyl






2.1.1667
3-cyano-6-
H
methyl
ethyl




methylphenyl






2.1.1668
3-trifluoro-
H
methyl
ethyl




methyl-6-







methylphenyl






2.1.1669
3-methoxy-6-
H
methyl
ethyl




methylphenyl






2.1.1670
3-ethoxy-6-
H
methyl
ethyl




methylphenyl






2.1.1671
3-trifluoro-
H
methyl
ethyl




methoxy-6-







methylphenyl






2.1.1672
3-nitro-6-
H
methyl
ethyl




methylphenyl






2.1.1673
3-fluoro-6-
H
methyl
ethyl




ethylphenyl






2.1.1674
3-chloro-6-
H
methyl
ethyl




ethylphenyl






2.1.1675
3-bromo-6-
H
methyl
ethyl




ethylphenyl






2.1.1676
3-methyl-6-
H
methyl
ethyl




ethylphenyl






2.1.1677
3,6-diethyl-
H
methyl
ethyl




phenyl






2.1.1678
3-cyclopropyl-6-
H
methyl
ethyl




ethylphenyl






2.1.1679
3-vinyl-6-
H
methyl
ethyl




ethylphenyl






2.1.1680
3-ethynyl-6-
H
methyl
ethyl




ethylphenyl






2.1.1681
3-cyano-6-
H
methyl
ethyl




ethylphenyl






2.1.1682
3-trifluoro-
H
methyl
ethyl




methyl-6-







ethylphenyl






2.1.1683
3-methoxy-6-
H
methyl
ethyl




ethylphenyl






2.1.1684
3-ethoxy-6-
H
methyl
ethyl




ethylphenyl






2.1.1685
3-trifluoro-
H
methyl
ethyl




methoxy-6-







ethylphenyl






2.1.1686
3-nitro-6-
H
methyl
ethyl




ethylphenyl






2.1.1687
3-fluoro-6-
H
methyl
ethyl




propylphenyl






2.1.1688
3-chloro-6-
H
methyl
ethyl




propylphenyl






2.1.1689
3-bromo-6-
H
methyl
ethyl




propylphenyl






2.1.1690
3-methyl-6-
H
methyl
ethyl




propylphenyl






2.1.1691
3-methyl-6-
H
methyl
ethyl




propylphenyl






2.1.1692
3-cyclopropyl-6-
H
methyl
ethyl




propylphenyl






2.1.1693
3-vinyl-6-
H
methyl
ethyl




propylphenyl






2.1.1694
3-ethynyl-6-
H
methyl
ethyl




propylphenyl






2.1.1695
3-cyano-6-
H
methyl
ethyl




propylphenyl






2.1.1696
3-trifluoro-
H
methyl
ethyl




methyl-6-







propylphenyl






2.1.1697
3-methoxy-6-
H
methyl
ethyl




propylphenyl






2.1.1698
3-ethoxy-6-
H
methyl
ethyl




propylphenyl






2.1.1699
3-trifluoro-
H
methyl
ethyl




methoxy-6-







propylphenyl






2.1.1700
3-nitro-6-
H
methyl
ethyl




propylphenyl






2.1.1701
3-fluoro-6-
H
methyl
ethyl




isopropylphenyl






2.1.1702
3-chloro-6-
H
methyl
ethyl




isopropylphenyl






2.1.1703
3-bromo-6-
H
methyl
ethyl




isopropylphenyl






2.1.1704
3-methyl-6-
H
methyl
ethyl




isopropylphenyl






2.1.1705
3-ethyl-6-
H
methyl
ethyl




isopropylphenyl






2.1.1706
3-cyclopropyl-6-
H
methyl
ethyl




isopropylphenyl






2.1.1707
3-vinyl-6-
H
methyl
ethyl




isopropylphenyl






2.1.1708
3-ethynyl-6-
H
methyl
ethyl




isopropylphenyl






2.1.1709
3-cyano-6-
H
methyl
ethyl




isopropylphenyl






2.1.1710
3-trifluoro-
H
methyl
ethyl




methyl-6-







isopropylphenyl






2.1.1711
3-methoxy-6-
H
methyl
ethyl




isopropylphenyl






2.1.1712
3-ethoxy-6-
H
methyl
ethyl




isopropylphenyl






2.1.1713
3-trifluoro-
H
methyl
ethyl




methoxy-6-







isopropylphenyl






2.1.1714
3-nitro-6-
H
methyl
ethyl




isopropylphenyl






2.1.1715
3-fluoro-6-tert-
H
methyl
ethyl




butylphenyl






2.1.1716
3-chloro-6-tert-
H
methyl
ethyl




butylphenyl






2.1.1717
3-bromo-6-tert-
H
methyl
ethyl




butylphenyl






2.1.1718
3-methyl-6-tert-
H
methyl
ethyl




butylphenyl






2.1.1719
3-ethyl-6-tert-
H
methyl
ethyl




butylphenyl






2.1.1720
3-cyclopropyl-6-
H
methyl
ethyl




tert-butylphenyl






2.1.1721
3-vinyl-6-tert-
H
methyl
ethyl




butylphenyl






2.1.1722
3-ethynyl-6-tert-
H
methyl
ethyl




butylphenyl






2.1.1723
3-cyano-6-tert-
H
methyl
ethyl




butylphenyl






2.1.1724
3-trifluoro-
H
methyl
ethyl




methyl-6-tert-







butylphenyl






2.1.1725
3-methoxy-6-
H
methyl
ethyl




tert-butylphenyl






2.1.1726
3-ethoxy-6-tert-
H
methyl
ethyl




butylphenyl






2.1.1727
3-trifluoro-
H
methyl
ethyl




methoxy-6-tert-







butylphenyl






2.1.1728
3-nitro-6-tert-
H
methyl
ethyl




butylphenyl






2.1.1729
3-fluoro-6-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1730
3-chloro-6-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1731
3-bromo-6-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1732
3-methyl-6-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1733
3-ethyl-6-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1734
3-cyclopropyl-6-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1735
3-vinyl-6-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1736
3-ethynyl-6-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1737
3-cyano-6-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1738
3-trifluoro-
H
methyl
ethyl




methyl-6-







hydroxymethyl-







phenyl






2.1.1739
3-methoxy-6-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1740
3-ethoxy-6-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1741
3-trifluoro-
H
methyl
ethyl




methoxy-6-







hydroxymethyl-







phenyl






2.1.1742
3-nitro-6-
H
methyl
ethyl




hydroxymethyl-







phenyl






2.1.1743
3-fluoro-6-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.1744
3-chloro-6-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.1745
3-bromo-6-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.1746
3-methyl-6-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.1747
3-ethyl-6-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.1748
3-cyclopropyl-6-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.1749
3-vinyl-6-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.1750
3-ethynyl-6-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.1751
3-cyano-6-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.1752
3-trifluoro-
H
methyl
ethyl




methyl-6-







cyclopropyl-







phenyl






2.1.1753
3-methoxy-6-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.1754
3-ethoxy-6-
H
methyl
ethyl




cyclopropyl-







phenyl






2.1.1755
3-trifluoro-
H
methyl
ethyl




methoxy-6-







cyclopropyl-







phenyl






2.1.1756
3-fluoro-6-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1757
3-chloro-6-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1758
3-bromo-6-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1759
3-methyl-6-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1760
3-ethyl-6-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1761
3-cyclopropyl-6-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1762
3-vinyl-6-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1763
3-ethynyl-6-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1764
3-cyano-6-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1765
3-trifluoro-
H
methyl
ethyl




methyl-6-







methoxy-







carbonylphenyl






2.1.1766
3-methoxy-6-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1767
3-ethoxy-6-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1768
3-trifluoro-
H
methyl
ethyl




methoxy-6-







methoxy-







carbonylphenyl






2.1.1769
3-nitro-6-
H
methyl
ethyl




methoxy-







carbonylphenyl






2.1.1770
3-fluoro-6-
H
methyl
ethyl




vinylphenyl






2.1.1771
3-chloro-6-
H
methyl
ethyl




vinylphenyl






2.1.1772
3-bromo-6-
H
methyl
ethyl




vinylphenyl






2.1.1773
3-methyl-6-
H
methyl
ethyl




vinylphenyl






2.1.1774
3-ethyl-6-
H
methyl
ethyl




vinylphenyl






2.1.1775
3-cyclopropyl-6-
H
methyl
ethyl




vinylphenyl






2.1.1776
3,6-divinyl-
H
methyl
ethyl




phenyl






2.1.1777
3-ethynyl-6-
H
methyl
ethyl




vinylphenyl






2.1.1778
3-cyano-6-
H
methyl
ethyl




vinylphenyl






2.1.1779
3-trifluoro-
H
methyl
ethyl




methyl-6-







vinylphenyl






2.1.1780
3-methoxy-6-
H
methyl
ethyl




vinylphenyl






2.1.1781
3-ethoxy-6-
H
methyl
ethyl




vinylphenyl






2.1.1782
3-trifluoro-
H
methyl
ethyl




methoxy-6-







vinylphenyl






2.1.1783
3-nitro-6-
H
methyl
ethyl




vinylphenyl






2.1.1784
3-fluoro-6-
H
methyl
ethyl




ethynylphenyl






2.1.1785
3-chloro-6-
H
methyl
ethyl




ethynylphenyl






2.1.1786
3-bromo-6-
H
methyl
ethyl




ethynylphenyl






2.1.1787
3-methyl-6-
H
methyl
ethyl




ethynylphenyl






2.1.1788
3-ethyl-6-
H
methyl
ethyl




ethynylphenyl






2.1.1789
3-cyclopropyl-6-
H
methyl
ethyl




ethynylphenyl






2.1.1790
3-vinyl-6-
H
methyl
ethyl




ethynylphenyl






2.1.1791
3-cyano-6-
H
methyl
ethyl




ethynylphenyl






2.1.1792
3-trifluoro-
H
methyl
ethyl




methyl-6-







ethynylphenyl






2.1.1793
3-methoxy-6-
H
methyl
ethyl




ethynylphenyl






2.1.1794
3-ethoxy-6-
H
methyl
ethyl




ethynylphenyl






2.1.1795
3-trifluoro-
H
methyl
ethyl




methoxy-6-







ethynylphenyl






2.1.1796
3-nitro-6-
H
methyl
ethyl




ethynylphenyl






2.1.1797
3-fluoro-6-
H
methyl
ethyl




ethynylphenyl






2.1.1798
3-fluoro-6-
H
methyl
ethyl




cyanophenyl






2.1.1799
3-chloro-6-
H
methyl
ethyl




cyanophenyl






2.1.1800
3-bromo-6-
H
methyl
ethyl




cyanophenyl






2.1.1801
3-methyl-6-
H
methyl
ethyl




cyanophenyl






2.1.1802
3-ethyl-6-
H
methyl
ethyl




cyanophenyl






2.1.1803
3-cyclopropyl-6-
H
methyl
ethyl




cyanophenyl






2.1.1804
3-vinyl-6-
H
methyl
ethyl




cyanophenyl






2.1.1805
3-ethynyl-6-
H
methyl
ethyl




cyanophenyl






2.1.1806
3-cyano-6-
H
methyl
ethyl




cyanophenyl






2.1.1807
3-trifluoro-
H
methyl
ethyl




methyl-6-







cyanophenyl






2.1.1808
3-methoxy-6-
H
methyl
ethyl




cyanophenyl






2.1.1809
3-ethoxy-6-
H
methyl
ethyl




cyanophenyl






2.1.1810
3-trifluoro-
H
methyl
ethyl




methoxy-6-







cyanophenyl






2.1.1811
3-nitro-6-
H
methyl
ethyl




cyanophenyl






2.1.1812
3-fluoro-6-
H
methyl
ethyl




hydroxyphenyl






2.1.1813
3-chloro-6-
H
methyl
ethyl




hydroxyphenyl






2.1.1814
3-bromo-6-
H
methyl
ethyl




hydroxyphenyl






2.1.1815
3-methyl-6-
H
methyl
ethyl




hydroxyphenyl






2.1.1816
3-ethyl-6-
H
methyl
ethyl




hydroxyphenyl






2.1.1817
3-cyclopropyl-6-
H
methyl
ethyl




hydroxyphenyl






2.1.1818
3-vinyl-6-
H
methyl
ethyl




hydroxyphenyl






2.1.1819
3-ethynyl-6-
H
methyl
ethyl




hydroxyphenyl






2.1.1820
3-cyano-6-
H
methyl
ethyl




hydroxyphenyl






2.1.1821
3-trifluoro-
H
methyl
ethyl




methyl-6-







hydroxyphenyl






2.1.1822
3-methoxy-6-
H
methyl
ethyl




hydroxyphenyl






2.1.1823
3-ethoxy-6-
H
methyl
ethyl




hydroxyphenyl






2.1.1824
3-trifluoro-
H
methyl
ethyl




methoxy-6-







hydroxyphenyl






2.1.1825
3-nitro-6-
H
methyl
ethyl




hydroxyphenyl






2.1.1826
3-fluoro-6-
H
methyl
ethyl




methoxyphenyl






2.1.1827
3-chloro-6-
H
methyl
ethyl




methoxyphenyl






2.1.1828
3-bromo-6-
H
methyl
ethyl




methoxyphenyl






2.1.1829
3-methyl-6-
H
methyl
ethyl




methoxyphenyl






2.1.1830
3-ethyl-6-
H
methyl
ethyl




methoxyphenyl






2.1.1831
3-cyclopropyl-6-
H
methyl
ethyl




methoxyphenyl






2.1.1832
3-vinyl-6-
H
methyl
ethyl




methoxyphenyl






2.1.1833
3-ethynyl-6-
H
methyl
ethyl




methoxyphenyl






2.1.1834
3-cyano-6-
H
methyl
ethyl




methoxyphenyl






2.1.1835
3-trifluoro-
H
methyl
ethyl




methyl-6-







methoxyphenyl






2.1.1836
3,6-dimethoxy--
H
methyl
ethyl




phenyl






2.1.1837
3-ethoxy-6-
H
methyl
ethyl




methoxyphenyl






2.1.1838
3-trifluoro-
H
methyl
ethyl




methoxy-6-







methoxyphenyl






2.1.1839
3-nitro-6-
H
methyl
ethyl




methoxyphenyl






2.1.1840
3-fluoro-6-
H
methyl
ethyl




ethoxyphenyl






2.1.1841
3-chloro-6-
H
methyl
ethyl




ethoxyphenyl






2.1.1842
3-bromo-6-
H
methyl
ethyl




ethoxyphenyl






2.1.1843
3-methyl-6-
H
methyl
ethyl




ethoxyphenyl






2.1.1844
3-ethyl-6-
H
methyl
ethyl




ethoxyphenyl






2.1.1845
3-cyclopropyl-6-
H
methyl
ethyl




ethoxyphenyl






2.1.1846
3-vinyl-6-
H
methyl
ethyl




ethoxyphenyl






2.1.1847
3-ethynyl-6-
H
methyl
ethyl




ethoxyphenyl






2.1.1848
3-cyano-6-
H
methyl
ethyl




ethoxyphenyl






2.1.1849
3-trifluoro-
H
methyl
ethyl




methyl-6-







ethoxyphenyl






2.1.1850
3-methoxy-6-
H
methyl
ethyl




ethoxyphenyl






2.1.1851
2,6-
H
methyl
ethyl




diethoxyphenyl






2.1.1852
3-trifluoro-
H
methyl
ethyl




methoxy-6-







ethoxyphenyl






2.1.1853
3-nitro-6-
H
methyl
ethyl




ethoxyphenyl






2.1.1854
3-fluoro-6-
H
methyl
ethyl




propoxyphenyl






2.1.1855
3-chloro-6-
H
methyl
ethyl




propoxyphenyl






2.1.1856
3-bromo-6-
H
methyl
ethyl




propoxyphenyl






2.1.1857
3-methyl-6-
H
methyl
ethyl




propoxyphenyl






2.1.1858
3-ethyl-6-
H
methyl
ethyl




propoxyphenyl






2.1.1859
3-cyclopropyl-6-
H
methyl
ethyl




propoxyphenyl






2.1.1860
3-vinyl-6-
H
methyl
ethyl




propoxyphenyl






2.1.1861
3-ethynyl-6-
H
methyl
ethyl




propoxyphenyl






2.1.1862
3-cyano-6-
H
methyl
ethyl




propoxyphenyl






2.1.1863
3-trifluoro-
H
methyl
ethyl




methyl-6-







propoxyphenyl






2.1.1864
3-methoxy-6-
H
methyl
ethyl




propoxy-phenyl






2.1.1865
3-ethoxy-6-
H
methyl
ethyl




propoxyphenyl






2.1.1866
3-trifluoro-
H
methyl
ethyl




methoxy-6-







propoxyphenyl






2.1.1867
3-nitro-6-
H
methyl
ethyl




propoxyphenyl






2.1.1868
3-fluoro-6-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.1869
3-chloro-6-iso-
H
methyl
ethyl




propoxyphenyl






2.1.1870
3-bromo-6-iso-
H
methyl
ethyl




propoxyphenyl






2.1.1871
3-methyl-6-iso-
H
methyl
ethyl




propoxyphenyl






2.1.1872
3-ethyl-6-iso-
H
methyl
ethyl




propoxyphenyl






2.1.1873
3-cyclopropyl-6-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.1874
3-vinyl-6-iso-
H
methyl
ethyl




propoxyphenyl






2.1.1875
3-ethynyl-6-iso-
H
methyl
ethyl




propoxyphenyl






2.1.1876
3-cyano-6-iso-
H
methyl
ethyl




propoxyphenyl






2.1.1877
3-trifluoro-
H
methyl
ethyl




methyl-6-iso-







propoxyphenyl






2.1.1878
3-methoxy-6-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.1879
3-ethoxy-6-
H
methyl
ethyl




isopropoxy-







phenyl






2.1.1880
3-trifluoro-
H
methyl
ethyl




methoxy-6-iso-







propoxyphenyl






2.1.1881
3-nitro-6-iso-
H
methyl
ethyl




propoxyphenyl






2.1.1882
3-fluoro-6-tert-
H
methyl
ethyl




butoxyphenyl






2.1.1883
3-chloro-6-tert-
H
methyl
ethyl




butoxyphenyl






2.1.1884
3-bromo-6-tert-
H
methyl
ethyl




butoxyphenyl






2.1.1885
3-methyl-6-tert-
H
methyl
ethyl




butoxyphenyl






2.1.1886
3-ethyl-6-tert-
H
methyl
ethyl




butoxyphenyl






2.1.1887
3-cyclopropyl-6-
H
methyl
ethyl




tert-butoxy-







phenyl






2.1.1888
3-vinyl-6-tert-
H
methyl
ethyl




butoxyphenyl






2.1.1889
3-ethynyl-6-tert-
H
methyl
ethyl




butoxyphenyl






2.1.1890
3-cyano-6-tert-
H
methyl
ethyl




butoxyphenyl






2.1.1891
3-trifluoro-
H
methyl
ethyl




methyl-6-tert-







butoxyphenyl






2.1.1892
3-methoxy-6-
H
methyl
ethyl




tert-butoxy-







phenyl






2.1.1893
3-ethoxy-6-tert-
H
methyl
ethyl




butoxyphenyl






2.1.1894
3-trifluoro-
H
methyl
ethyl




methoxy-6-tert-







butoxyphenyl






2.1.1895
3-nitro-6-tert-
H
methyl
ethyl




butoxyphenyl






2.1.1896
3-fluoro-6-tri-
H
methyl
ethyl




fluoromethoxy-







phenyl






2.1.1897
3-chloro-6-tri-
H
methyl
ethyl




fluoromethoxy-







phenyl






2.1.1898
3-bromo-6-tri-
H
methyl
ethyl




fluoromethoxy-







phenyl






2.1.1899
3-methyl-6-tri-
H
methyl
ethyl




fluoromethoxy-







phenyl






2.1.1900
3-ethyl-6-tri-
H
methyl
ethyl




fluoromethoxy-







phenyl






2.1.1901
3-cyclopropyl-6-
H
methyl
ethyl




trifluorometh-







oxyphenyl






2.1.1902
3-vinyl-6-tri-
H
methyl
ethyl




fluoromethoxy-







phenyl






2.1.1903
3-ethynyl-6-tri-
H
methyl
ethyl




fluoromethoxy-







phenyl






2.1.1904
3-cyano-6-tri-
H
methyl
ethyl




fluoromethoxy-







phenyl






2.1.1905
3-trifluoro-
H
methyl
ethyl




methyl-6-tri-







fluoromethoxy-







phenyl






2.1.1906
3-methoxy-6-
H
methyl
ethyl




trifluoro-







methoxyphenyl






2.1.1907
3-ethoxy-6-
H
methyl
ethyl




trifluoro-







methoxyphenyl






2.1.1908
3,6-bis(trifluoro-
H
methyl
ethyl




methoxy)phenyl






2.1.1909
3-nitro-6-tri-
H
methyl
ethyl




fluoromethoxy-







phenyl






2.1.1910
3-fluoro-6-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxy)phenyl






2.1.1911
3-chloro-6-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxy)phenyl






2.1.1912
3-bromo-6-
H
methyl
ethyl




(2,2,2-







trifluoroethoxy)-







phenyl






2.1.1913
3-methyl-6-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxy)phenyl






2.1.1914
3-ethyl-6-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







phenyl






2.1.1915
3-cyclopropyl-6-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxy)phenyl






2.1.1916
3-vinyl-6-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







phenyl






2.1.1917
3-ethynyl-6-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxyphenyl






2.1.1918
3-cyano-6-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxy)phenyl






2.1.1919
3-trifluoro-
H
methyl
ethyl




methyl-6-(2,2,2-







trifluoroethoxy)-







phenyl






2.1.1920
3-methoxy-6-
H
methyl
ethyl




(2,2,2-trifluoro-







ethoxy)phenyl






2.1.1921
3-ethoxy-6-
H
methyl
ethyl




(2,2,2-







trifluoroethoxy)-







phenyl






2.1.1922
3-trifluoro-
H
methyl
ethyl




methoxy-6-







(2,2,2-trifluoro-







ethoxy)phenyl






2.1.1923
3-nitro-6-(2,2,2-
H
methyl
ethyl




trifluoroethoxy)-







phenyl






2.1.1924
3-fluoro-6-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.1925
3-chloro-6-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.1926
3-bromo-6-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.1927
3-methyl-6-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.1928
3-ethyl-6-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.1929
3-cyclopropyl-6-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.1930
3-vinyl-6-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.1931
3-ethynyl-6-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.1932
3-cyano-6-
H
methyl
ethyl




difluoromethoxy







phenyl






2.1.1933
3-trifluoro-
H
methyl
ethyl




methyl-6-di-







fluoromethoxy-







phenyl






2.1.1934
3-methoxy-6-
H
methyl
ethyl




difluoromethoxy







phenyl






2.1.1935
3-ethoxy-6-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.1936
3-trifluoro-
H
methyl
ethyl




methoxy-6-di-







fluoromethoxy-







phenyl






2.1.1937
3-nitro-6-
H
methyl
ethyl




difluoromethoxy-







phenyl






2.1.1938
3-fluoro-6-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.1939
3-chloro-6-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.1940
3-bromo-6-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.1941
3-methyl-6-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.1942
3-ethyl-6-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.1943
3-cyclopropyl-6-
H
methyl
ethyl




(2-methoxy-







ethoxy)phenyl






2.1.1944
3-vinyl-6-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.1945
3-ethynyl-6-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.1946
3-cyano-6-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.1947
3-trifluoro-
H
methyl
ethyl




methyl-6-(2-







methoxyethoxy)-







phenyl






2.1.1948
3-methoxy-6-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.1949
3-ethoxy-6-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.1950
3-trifluoro-
H
methyl
ethyl




methoxy-(2-







methoxyethoxy)-







phenyl






2.1.1951
3-nitro-6-(2-
H
methyl
ethyl




methoxyethoxy)-







phenyl






2.1.1952
3-fluoro-6-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.1953
3-chloro-6-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.1954
3-bromo-6-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.1955
3-methyl-6-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.1956
3-ethyl-6-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.1957
3-cyclopropyl-6-
H
methyl
ethyl




(tert-butoxy-







carbonyloxy)-







phenyl






2.1.1958
3-vinyl-6-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.1959
3-ethynyl-6-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.1960
3-cyano-6-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.1961
3-trifluoro-
H
methyl
ethyl




methyl-6-(tert-







butoxycarbonyl-







oxy)phenyl






2.1.1962
3-methoxy-6-
H
methyl
ethyl




(tert-butoxy-







carbonyloxy)-







phenyl






2.1.1963
3-ethoxy-6-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.1964
3-trifluoro-
H
methyl
ethyl




methoxy-6-(tert-







butoxycarbonyl-







oxy)phenyl






2.1.1965
2-nitro-6-(tert-
H
methyl
ethyl




butoxycarbonyl-







oxy)phenyl






2.1.1966
3-fluoro-6-
H
methyl
ethyl




nitrophenyl






2.1.1967
3-chloro-6-
H
methyl
ethyl




nitrophenyl






2.1.1968
3-bromo-6-
H
methyl
ethyl




nitrophenyl






2.1.1969
3-methyl-6-
H
methyl
ethyl




nitrophenyl






2.1.1970
3-ethyl-6-
H
methyl
ethyl




nitrophenyl






2.1.1971
3-cyclopropyl-6-
H
methyl
ethyl




nitrophenyl






2.1.1972
3-vinyl-6-
H
methyl
ethyl




nitrophenyl






2.1.1973
3-ethynyl-6-
H
methyl
ethyl




nitrophenyl






2.1.1974
3-cyano-6-
H
methyl
ethyl




nitrophenyl






2.1.1975
3-trifluoro-
H
methyl
ethyl




methyl-6-







nitrophenyl






2.1.1976
3-methoxy-6-
H
methyl
ethyl




nitrophenyl






2.1.1977
3-ethoxy-6-
H
methyl
ethyl




nitrophenyl






2.1.1978
3-trifluoro-
H
methyl
ethyl




methoxy-6-







nitrophenyl






2.1.1979
3-fluoro-6-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.1980
3-chloro-6-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.1981
3-bromo-6-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.1982
3-methyl-6-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.1983
3-ethyl-6-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.1984
3-cyclopropyl-6-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.1985
3-vinyl-6-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.1986
3-ethynyl-6-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.1987
3-cyano-6-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.1988
3-trifluoro-
H
methyl
ethyl




methyl-6-







methylsulfanyl-







phenyl






2.1.1989
3-methoxy-6-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.1990
3-ethoxy-6-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.1991
3-trifluoro-
H
methyl
ethyl




methoxy-6-







methylsulfanyl-







phenyl






2.1.1992
3-nitro-6-
H
methyl
ethyl




methylsulfanyl-







phenyl






2.1.1993
2,3,4-trifluoro-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.71 (s,



phenyl



3H); 3.25 (dd, 1H); 3.92 (dd,







1H); 4.25 (q, 2H); 7.00 (m, 1H);







7.61 (m, 1H).


2.1.1994
2,3,4-trichloro-
H
methyl
ethyl




phenyl






2.1.1995
2,3,4-trimethyl-
H
methyl
ethyl




phenyl






2.1.1996
2-fluoro-2-
H
methyl
ethyl




chloro-5-tri-







fluoromethyl-







phenyl






2.1.1997
2,3,5-
H
methyl
ethyl
[CDCl3] 1.30 (t, 3H); 1.72 (s,



trifluorophenyl



3H); 3.28 (dd, 1H); 3.92 (dd,







1H); 4.25 (q, 2H); 6.97 (m, 1H);







7.39 (m, 1H).


2.1.1998
2,3,5-trichloro-
H
methyl
ethyl




phenyl






2.1.1999
2,3,5-trimethyl-
H
methyl
ethyl




phenyl






2.1.2000
2,3-dichloro-5-
H
methyl
ethyl
[CDCl3] 1.32 (t, 3H); 1.72 (s,



methoxyphenyl



3H); 3.40 (d, 1H); 3.81 (s, 3H);







3.92 (d, 1H): 4.30 (mc, 2H); 7.11







(mc, 2H).


2.1.2001
2,3,6-trifluoro-
H
methyl
ethyl




phenyl






2.1.2002
2,3,6-trichloro-
H
methyl
ethyl
[CDCl3] 1.34 (t, 3H); 1.75 (s,



phenyl



3H); 3.13 (d, 1H); 3.79 (d, 1H);







4.30 (q, 2H); 7.3 (d, 1H); 7.48







(d, 1H).


2.1.2003
2,3,6-trimethyl-
H
methyl
ethyl




phenyl






2.1.2004
3,4,5-trifluoro-
H
methyl
ethyl
[CDCl3] 1.32 (t, 3H); 1.70 (s,



phenyl



3H); 3.10 (d, 1H); 3.81 (d, 1H);







4.25 (m, 1H); 7.32 (m, 2H).


2.1.2005
3,4,5-trichloro-
H
methyl
ethyl
[CDCl3] 1.32 (t, 3H); 1.71 (s,



phenyl



3H); 3.12 (d, 1H); 3.81 (d, 1H);







4.25 (m, 2H); 7.66 (s, 2H).


2.1.2006
3,4,5-trimethyl-
H
methyl
ethyl




phenyl






2.1.2007
3,5-dimethyl-4-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.70 (s,



fluorophenyl



3H); 2.25 (s, 6H); 3.17 (d, 1H);







3.85 (d, 1H); 4.25 (m, 2H); 7.32







(d, 2H).


2.1.2008
3,5-dichloro-4-
H
methyl
ethyl
[CDCl3] 1.30 (t, 3H); 1.70 (s,



methoxyphenyl



3H); 3.14 (d, 1H); 3.82 (d, 1H);







3.91 (s, 3H); 4.28 (q, 2H); 7.60







(s, 2H).


2.1.2009
3,5-difluoro-4-
H
methyl
ethyl
[CDCl3] 1.30 (t, 3H); 1.71 (s,



chlorophenyl



3H); 3.12 (d, 1H); 3.82 (d, 1H);







4.25 (m, 2H); 7.32 (m, 2H).


2.1.2010
3,5-dichloro-4-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.71 (s,



hydroxyphenyl



3H); 3.12 (d, 1H); 3.82 (d, 1H);







4.25 (m, 2H); 7.58 (s, 2H).


2.1.2011
3,5-trifluoro-
H
methyl
ethyl




methyl-4-







chlorophenyl






2.1.2012
3,4,6-
H
methyl
ethyl




trifluorophenyl






2.1.2013
3,4,6-
H
methyl
ethyl




trichlorophenyl






2.1.2014
3,4,6-
H
methyl
ethyl




trimethylphenyl






2.1.2015
2,3,4,5-
H
methyl
ethyl
[CDCl3] 1.31 (t, 3H); 1.72 (s,



pentafluoro-



3H); 3.25 (dd, 1H); 3.90 (d, 1H);



phenyl



4.25 (m, 2H).


2.1.2016
3,5-difluoro-
Br
methyl
ethyl
One unassigned diastereomer



phenyl



[CDCl3] 1.32 (t, 3H); 1.93 (s,







3H); 4.27 (m , 2H); 5.80 (s, 1H);







6.93 (dt, 1H); 7.35 (m, 2H).


2.1.2017
3,5-difluoro-
Br
methyl
ethyl
The other unassigned



phenyl



diastereomer







[CDCl3] 1.32 (t, 3H); 1.62 (s,







3H), 4.30 (q, 2H); 5.08 (s, 1H);







6.85 (t, 1H); 7.24 (d, 2H).


2.1.2018
3,5-dichloro-
Br
methyl
ethyl
One unassigned diastereomer



phenyl



[CDCl3] 1.25 (t, 3H); 1.85 (s,







3H); 4.17 (m, 2H); 5.71 (s, 1H);







7.37 (s, 1H); 7.61 (s, 2H).


2.1.2019
3,5-dichloro-
Br
methyl
ethyl
The other unassigned



phenyl



diastereomer







[CDCl3] 1.39 (t, 3H); 1.68 (s,







3H); 4.37 (q, 2H); 5.15 (s, 1H);







7.45 (s, 1H); 7.67 (s, 2H).
















TABLE 2.2







Inventive compounds of the general formula (I) in which W* is CODY, R1


and R2 are each hydrogen, and aryl is the radical.








 








 











No.
Aryl
R3
Y
Physical data





2.2.1
3-fluorophenyl
fluoromethyl
ethyl
[CDCl3] 1.33 (t, 3H); 3.53






(d, 1H); 3.84 (d, 1H); 4.31






(q, 2H); 4.68 (d, 1H); 4.78






(d, 1H); 7.14 (t, 1H); 7.41






(m, 3H).


2.2.2
3-fluorophenyl
chloromethyl
ethyl
[CDCl3] 1.35 (t, 3H); 3.55






(d, 1H); 3.79 (d, 1H); 4.01






(dd, 2H); 4.32 (m, 2H); 7.15






(t, 1H); 7.41 (m, 3H).


2.2.3
3-fluorophenyl
bromomethyl
ethyl
[CDCl3] 1.35 (t, 3H); 3.50






(d, 1H); 3.62 (d, 1H); 3.90






(d, 1H); 4.05 (d, 1H); 4.33






(m, 2H); 7.15 (t, 1H); 7.43






(m, 3H).


2.2.4
3-fluorophenyl
difluoromethyl
ethyl



2.2.5
3-fluorophenyl
1,1-dichloroethyl
methyl
[CDCl3] 2.40 (s, 3H); 3.88






(s, 3H); 4.07 (AB, 2H); 7.16






(t, 1H); 7.39-7.46 (m, 3H).


2.2.6
3-fluorophenyl
cyano
ethyl



2.2.7
3-chlorophenyl
fluoromethyl
ethyl



2.2.8
3-chlorophenyl
chloromethyl
ethyl



2.2.9
3-chlorophenyl
bromomethyl
ethyl



2.2.10
3-chlorophenyl
difluoromethyl
ethyl



2.2.11
3-chlorophenyl
trifluoromethyl
ethyl



2.2.12
3-chlorophenyl
cyano
ethyl



2.2.13
3-bromophenyl
fluoromethyl
ethyl



2.2.14
3-bromophenyl
chloromethyl
ethyl



2.2.15
3-iodophenyl
fluoromethyl
ethyl



2.2.16
3-iodophenyl
chloromethyl
ethyl



2.2.17
3-methylphenyl
fluoromethyl
ethyl



2.2.18
3-methylphenyl
chloromethyl
ethyl



2.2.19
3-ethylphenyl
fluoromethyl
ethyl



2.2.20
3-propylphenyl
fluoromethyl
ethyl



2.2.21
3-isopropylphenyl
fluoromethyl
ethyl



2.2.22
3-n-butylphenyl
fluoromethyl
ethyl



2.2.23
3-i-butylphenyl
fluoromethyl
ethyl



2.2.24
3-tert-butylphenyl
fluoromethyl
ethyl



2.2.25
3-cyclopropylphenyl
fluoromethyl
ethyl



2.2.26
3-cyclobutylphenyl
fluoromethyl
ethyl



2.2.27
3-cyclopentylphenyl
fluoromethyl
ethyl



2.2.28
3-vinylphenyl
fluoromethyl
ethyl



2.2.29
3-ethynylphenyl
fluoromethyl
ethyl



2.2.30
3-cyanophenyl
fluoromethyl
ethyl



2.2.31
3-trifluoromethylphenyl
fluoromethyl
ethyl



2.2.32
3-difluoromethylphenyl
fluoromethyl
ethyl



2.2.33
3-(hydroxycarbonyl)-
fluoromethyl
ethyl




phenyl





2.2.34
3-(methoxycarbonyl)-
fluoromethyl
ethyl




phenyl





2.2.35
3-(ethoxycarbonyl)phenyl
fluoromethyl
ethyl



2.2.36
3-hydroxymethylphenyl
fluoromethyl
ethyl



2.2.37
3-carbamoylphenyl
fluoromethyl
ethyl



2.2.38
3-hydroxyphenyl
fluoromethyl
ethyl



2.2.39
3-methoxyphenyl
fluoromethyl
ethyl



2.2.40
3-ethoxyphenyl
fluoromethyl
ethyl



2.2.41
3-propyloxyphenyl
fluoromethyl
ethyl



2.2.42
3-isopropyloxyphenyl
fluoromethyl
ethyl



2.2.43
3-n-butyloxyphenyl
fluoromethyl
ethyl



2.2.44
3-i-butyloxyphenyl
fluoromethyl
ethyl



2.2.45
3-t-butyloxyphenyl
fluoromethyl
ethyl



2.2.46
3-difluoromethoxyphenyl
fluoromethyl
ethyl



2.2.47
3-trifluoromethoxyphenyl
fluoromethyl
ethyl



2.2.48
3-(2,2,2-trifluoroethoxy)- 
fluoromethyl
ethyl




phenyl





2.2.49
3-(2-chloroethoxy)phenyl
fluoromethyl
ethyl



2.2.50
3-(2-hydroxyethoxy)-
fluoromethyl
ethyl




phenyl





2.2.51
3-(2-methoxyethoxy)-
fluoromethyl
ethyl




phenyl





2.2.52
3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




oxy]phenyl





2.2.53
3-nitrophenyl
fluoromethyl
ethyl



2.2.54
3-acetoxyphenyl
fluoromethyl
ethyl



2.2.55
{3-[(tert-butoxycarbony1)-
fluoromethyl
ethyl




amino]phenyl}





2.2.56
3-methylsulfanylphenyl
fluoromethyl
ethyl



2.2.57
3-ethylsulfanylphenyl
fluoromethyl
ethyl



2.2.58
3-(pentafluoro-lambda6-
fluoromethyl
ethyl




sulfanyl)phenyl





2.2.59
2,3-difluorophenyl
fluoromethyl
ethyl



2.2.60
2,3-difluorophenyl
chloromethyl
ethyl



2.2.61
2,3-difluorophenyl
bromomethyl
ethyl



2.2.62
2,3-difluorophenyl
difluoromethyl
ethyl



2.2.63
2,3-difluorophenyl
trifluoromethyl
ethyl



2.2.64
2,3-difluorophenyl
cyano
ethyl



2.2.65
2-chloro-3-fluorophenyl
fluoromethyl
ethyl



2.2.66
2-bromo-3-fluorophenyl
fluoromethyl
ethyl



2.2.67
2-methyl-3-fluorophenyl
fluoromethyl
ethyl



2.2.68
2-ethyl-3-fluorophenyl
fluoromethyl
ethyl



2.2.69
2-cyclopropy1-3-
fluoromethyl
ethyl




fluorophenyl





2.2.70
2-vinyl-3-fluorophenyl
fluoromethyl
ethyl



2.2.71
2-ethynyl-3-fluorophenyl
fluoromethyl
ethyl



2.2.72
2-cyano-3-fluorophenyl
fluoromethyl
ethyl



2.2.73
2-methoxy-3-fluorophenyl
fluoromethyl
ethyl



2.2.74
2-ethoxy-3-fluorophenyl
fluoromethyl
ethyl



2.2.75
2-trifluoromethoxy-3-
fluoromethyl
ethyl




fluorophenyl





2.2.76
2-nitro-3-fluorophenyl
fluoromethyl
ethyl



2.2.77
2-fluoro-3-chlorophenyl
fluoromethyl
ethyl



2.2.78
2,3-dichlorophenyl
fluoromethyl
ethyl



2.2.79
2,3-dichlorophenyl
chloromethyl
ethyl



2.2.80
2,3-dichlorophenyl
bromomethyl
ethyl



2.2.81
2,3-dichlorophenyl
difluoromethyl
ethyl



2.2.82
2-bromo-3-chlorophenyl
fluoromethyl
ethyl



2.2.83
2-methyl-3-chlorophenyl
fluoromethyl
ethyl



2.2.84
2-ethyl-3-chlorophenyl
fluoromethyl
ethyl



2.2.85
2-cyclopropyl-3-
fluoromethyl
ethyl




chlorophenyl





2.2.86
2-vinyl-3-chlorophenyl
fluoromethyl
ethyl



2.2.87
2-ethynyl-3-chlorophenyl
fluoromethyl
ethyl



2.2.88
2-cyano-3-chlorophenyl
fluoromethyl
ethyl



2.2.89
2-trifluoromethy1-2-
fluoromethyl
ethyl




chlorophenyl





2.2.90
2-methoxy-3-chlorophenyl
fluoromethyl
ethyl



2.2.91
2-ethoxy-3-chlorophenyl
fluoromethyl
ethyl



2.2.92
2-trifluoromethoxy-3-
fluoromethyl
ethyl




chlorophenyl





2.2.93
2-nitro-3-chlorophenyl
fluoromethyl
ethyl



2.2.94
2-fluoro-3-bromophenyl
fluoromethyl
ethyl



2.2.95
2-chloro-3-bromophenyl
fluoromethyl
ethyl



2.2.96
2,3-dibromophenyl
fluoromethyl
ethyl



2.2.97
2-methyl-3-bromophenyl
fluoromethyl
ethyl



2.2.98
2-ethyl-3-bromophenyl
fluoromethyl
ethyl



2.2.99
2-cyclopropy1-3-
fluoromethyl
ethyl




bromophenyl





2.2.100
2-vinyl-3-bromophenyl
fluoromethyl
ethyl



2.2.101
2-ethynyl-3-bromophenyl
fluoromethyl
ethyl



2.2.102
2-cyano-3-bromophenyl
fluoromethyl
ethyl



2.2.103
2-trifluoromethyl-3-
fluoromethyl
ethyl




bromophenyl





2.2.104
2-methoxy-3-phenyl
fluoromethyl
ethyl



2.2.105
2-ethoxy-3-bromophenyl
fluoromethyl
ethyl



2.2.106
2-trifluoromethoxy-3-
fluoromethyl
ethyl




bromophenyl





2.2.107
2-nitro-3-bromophenyl
fluoromethyl
ethyl



2.2.108
2-fluoro-3-iodophenyl
fluoromethyl
ethyl



2.2.109
2-chloro-3-iodophenyl
fluoromethyl
ethyl



2.2.110
2-bromo-3-iodophenyl
fluoromethyl
ethyl



2.2.111
2-methyl-3-iodophenyl
fluoromethyl
ethyl



2.2.112
2-ethyl-3-iodophenyl
fluoromethyl
ethyl



2.2.113
2-cyclopropy1-3-
fluoromethyl
ethyl




iodophenyl





2.2.114
2-vinyl-3-iodophenyl
fluoromethyl
ethyl



2.2.115
2-ethynyl-3-iodophenyl
fluoromethyl
ethyl



2.2.116
2-cyano-3-iodophenyl
fluoromethyl
ethyl



2.2.117
2-trifluoromethy1-3-
fluoromethyl
ethyl




iodophenyl





2.2.118
2-methoxy-3-iodophenyl
fluoromethyl
ethyl



2.2.119
2-ethoxy-3-iodophenyl
fluoromethyl
ethyl



2.2.120
2-trifluoromethoxy-3-
fluoromethyl
ethyl




iodophenyl





2.2.121
2-nitro-3-iodophenyl
fluoromethyl
ethyl



2.2.122
2-fluoro-3-methylphenyl
fluoromethyl
ethyl



2.2.123
2-fluoro-3-methylphenyl
chloromethyl
ethyl



2.2.124
2-fluoro-3-methylphenyl
bromomethyl
ethyl



2.2.125
2-fluoro-3-methylphenyl
difluoromethyl 
ethyl



2.2.126
2-chloro-3-methylphenyl
fluoromethyl
ethyl



2.2.127
2-chloro-3-methylphenyl
chloromethyl
ethyl



2.2.128
2-chloro-3-methylphenyl
bromomethyl
ethyl



2.2.129
2-chloro-3-methylphenyl
difluoromethyl 
ethyl



2.2.130
2-bromo-3-methylphenyl
fluoromethyl
ethyl



2.2.131
2,3-dimethylphenyl
fluoromethyl
ethyl



2.2.132
2,3-dimethylphenyl
chloromethyl
ethyl



2.2.133
2,3-dimethylphenyl
bromomethyl
ethyl



2.2.134
2,3-dimethylphenyl
difluoromethyl
ethyl



2.2.135
2-ethyl-3-methylphenyl
fluoromethyl
ethyl



2.2.136
2-cyclopropy1-3-
fluoromethyl
ethyl




methylphenyl





2.2.137
2-vinyl-3-methylphenyl
fluoromethyl
ethyl



2.2.138
2-ethynyl-3-methylphenyl
fluoromethyl
ethyl



2.2.139
2-cyano-3-methylphenyl
fluoromethyl
ethyl



2.2.140
2-trifluoromethyl-3-
fluoromethyl
ethyl




methylphenyl





2.2.141
2-methoxy-3-
fluoromethyl
ethyl




methylphenyl





2.2.142
2-ethoxy-3-methylphenyl
fluoromethyl
ethyl



2.2.143
2-trifluoromethoxy-3- 
fluoromethyl
ethyl




methylphenyl





2.2.144
2-nitro-3-methylphenyl
fluoromethyl
ethyl



2.2.145
2-fluoro-3-ethylphenyl
fluoromethyl
ethyl



2.2.146
2-chloro-3-ethylphenyl
fluoromethyl
ethyl



2.2.147
2-bromo-3-ethylphenyl
fluoromethyl
ethyl



2.2.148
2-methyl-3-ethylphenyl
fluoromethyl
ethyl



2.2.149
2,3-diethylphenyl
fluoromethyl
ethyl



2.2.150
2-cyclopropyl-3-
fluoromethyl
ethyl




ethylphenyl





2.2.151
2-vinyl-3-ethylphenyl
fluoromethyl
ethyl



2.2.152
2-ethynyl-3-ethylphenyl
fluoromethyl
ethyl



2.2.153
2-cyano-3-ethylphenyl
fluoromethyl
ethyl



2.2.154
2-trifluoromethy1-3-
fluoromethyl
ethyl




ethylphenyl





2.2.155
2-methoxy-3-ethylphenyl
fluoromethyl
ethyl



2.2.156
2-ethoxy-3-ethylphenyl
fluoromethyl
ethyl



2.2.157
2-trifluoromethoxy-3-
fluoromethyl
ethyl




ethylphenyl





2.2.158
2-nitro-3-ethylphenyl
fluoromethyl
ethyl



2.2.159
2-fluoro-3-propylphenyl
fluoromethyl
ethyl



2.2.160
2-chloro-3-propylphenyl
fluoromethyl
ethyl



2.2.161
2-bromo-3-propylphenyl
fluoromethyl
ethyl



2.2.162
2-methyl-3-propylphenyl
fluoromethyl
ethyl



2.2.163
2-methyl-3-propylphenyl
fluoromethyl
ethyl



2.2.164
2-cyclopropy1-3-
fluoromethyl
ethyl




propylphenyl





2.2.165
2-vinyl-3-propylphenyl
fluoromethyl
ethyl



2.2.166
2-ethynyl-3propylphenyl
fluoromethyl
ethyl



2.2.167
2-cyano-3-propylphenyl
fluoromethyl
ethyl



2.2.168
2-trifluoromethyl-3-
fluoromethyl
ethyl




propylphenyl





2.2.169
2-methoxy-3-propylphenyl
fluoromethyl
ethyl



2.2.170
2-ethoxy-3-propylphenyl
fluoromethyl
ethyl



2.2.171
2-trifluoromethoxy-3-
fluoromethyl
ethyl




propylphenyl





2.2.172
2-nitro-3-propylphenyl
fluoromethyl
ethyl



2.2.173
2-fluoro-3-isopropylphenyl
fluoromethyl
ethyl



2.2.174
2-chloro-3-isopropyl-
fluoromethyl
ethyl




phenyl





2.2.175
2-bromo-3-isopropyl-
fluoromethyl
ethyl




phenyl





2.2.176
2-methy1-3-isopropyl-
fluoromethyl
ethyl




phenyl





2.2.177
2-ethyl-3-isopropylphenyl
fluoromethyl
ethyl



2.2.178
2-cyclopropy1-3-isopropyl-
fluoromethyl
ethyl




phenyl





2.2.179
2-vinyl-3-isopropylphenyl
fluoromethyl
ethyl



2.2.180
2-ethyny1-3-isopropyl-
fluoromethyl
ethyl




phenyl





2.2.181
2-cyano-3-isopropyl-
fluoromethyl
ethyl




phenyl





2.2.182
2-trifluoromethyl-3-
fluoromethyl
ethyl




isopropylphenyl





2.2.183
2-methoxy-3-isopropyl-
fluoromethyl
ethyl




phenyl





2.2.184
2-ethoxy-3-isopropyl-
fluoromethyl
ethyl




phenyl





2.2.185
2-trifluoromethoxy-3-
fluoromethyl
ethyl




isopropylphenyl





2.2.186
2-nitro-3-isopropylphenyl
fluoromethyl
ethyl



2.2.187
2-fluoro-3-tert-butylphenyl
fluoromethyl
ethyl



2.2.188
2-chloro-3-tert-butylphenyl
fluoromethyl
ethyl



2.2.189
2-bromo-3-tert-butyl-
fluoromethyl
ethyl




phenyl





2.2.190
2-methy1-3-tert-butyl-
fluoromethyl
ethyl




phenyl





2.2.191
2-ethyl-3-tert-butylphenyl
fluoromethyl
ethyl



2.2.192
2-cyclopropyl-3-tert-butyl-
fluoromethyl
ethyl




phenyl





2.2.193
2-vinyl-3-tert-butylphenyl
fluoromethyl
ethyl



2.2.194
2-ethyny1-3-tert-butyl-
fluoromethyl
ethyl




phenyl





2.2.195
2-cyano-3-tert-butylphenyl
fluoromethyl
ethyl



2.2.196
2-trifluoromethyl-3-tert-
fluoromethyl
ethyl




butylphenyl





2.2.197
2-methoxy-3-tert-butyl-
fluoromethyl
ethyl




phenyl





2.2.198
2-ethoxy-3-tert-butyl-
fluoromethyl
ethyl




phenyl





2.2.199
2-trifluoromethoxy-3-tert-
fluoromethyl
ethyl




butylphenyl





2.2.200
2-nitro-3-tert-butylphenyl
fluoromethyl
ethyl



2.2.201
2-fluoro-3-hydroxymethyl-
fluoromethyl
ethyl




phenyl





2.2.202
2-chloro-3-hydroxymethyl-
fluoromethyl
ethyl




phenyl





2.2.203
2-bromo-3-hydroxy-
fluoromethyl
ethyl




methylphenyl





2.2.204
2-methyl-3-hydroxy-
fluoromethyl
ethyl




methylphenyl





2.2.205
2-ethyl-3-hydroxymethyl-
fluoromethyl
ethyl




phenyl





2.2.206
2-cyclopropyl-3-hydroxy-
fluoromethyl
ethyl




methylphenyl





2.2.207
2-vinyl-3-hydroxymethyl-
fluoromethyl
ethyl




phenyl





2.2.208
2-ethynyl-3-hydroxy-
fluoromethyl
ethyl




methylphenyl





2.2.209
2-cyano-3-hydroxymethyl-
fluoromethyl
ethyl




phenyl





2.2.210
2-trifluoromethyl-3-
fluoromethyl
ethyl




hydroxymethylphenyl





2.2.211
2-methoxy-3-
fluoromethyl
ethyl




hydroxymethylphenyl





2.2.212
2-ethoxy-3-hydroxy-
fluoromethyl
ethyl




methylphenyl





2.2.213
2-trifluoromethoxy-3-
fluoromethyl
ethyl




hydroxymethylphenyl





2.2.214
2-nitro-3-hydroxymethyl-
fluoromethyl
ethyl




phenyl





2.2.215
2-fluoro-3-cyclopropyl-
fluoromethyl
ethyl




phenyl





2.2.216
2-chloro-3-cyclopropyl-
fluoromethyl
ethyl




phenyl





2.2.217
2-bromo-3-cyclopropyl-
fluoromethyl
ethyl




phenyl





2.2.218
2-methyl-3-cyclopropyl-
fluoromethyl
ethyl




phenyl





2.2.219
2-ethyl-3-cyclopropyl-
fluoromethyl
ethyl




phenyl





2.2.220
2-cyclopropy1-3-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.221
2-vinyl-3-cyclopropyl-
fluoromethyl
ethyl




phenyl





2.2.222
2-ethynyl-3-cyclopropyl-
fluoromethyl
ethyl




phenyl





2.2.223
2-cyano-3-cyclopropyl-
fluoromethyl
ethyl




phenyl





2.2.224
2-trifluoromethy1-3-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.225
2-methoxy-3-cyclopropyl-
fluoromethyl
ethyl




phenyl





2.2.226
2-ethoxy-3-cyclopropyl-
fluoromethyl
ethyl




phenyl





2.2.227
2-trifluoromethoxy-3-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.228
2-fluoro-3-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.229
2-chloro-3-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.230
2-bromo-3-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.231
2-methyl-3-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.232
2-ethy1-3-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.233
2-cyclopropyl-3-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.234
2-vinyl-3-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.235
2-ethynyl-3-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.236
2-cyano-3-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.237
2-trifluoromethyl-3-
fluoromethyl
ethyl




methoxycarbonylphenyl





2.2.238
2-methoxy-3-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.239
2-ethoxy-3-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.240
2-trifluoromethoxy-3-
fluoromethyl
ethyl




methoxycarbonylphenyl





2.2.241
2-nitro-3-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.242
2-fluoro-3-vinylphenyl
fluoromethyl
ethyl



2.2.243
2-chloro-3-vinylphenyl
fluoromethyl
ethyl



2.2.244
2-bromo-3-vinylphenyl
fluoromethyl
ethyl



2.2.245
2-methyl-3-vinylphenyl
fluoromethyl
ethyl



2.2.246
2-ethyl-3-vinylphenyl
fluoromethyl
ethyl



2.2.247
2-cyclopropy1-3-
fluoromethyl
ethyl




vinylphenyl





2.2.248
2-vinyl-3-vinylphenyl
fluoromethyl
ethyl



2.2.249
2-ethynyl-3-vinylphenyl 
fluoromethyl
ethyl



2.2.250
2-cyano-3-vinylphenyl
fluoromethyl
ethyl



2.2.251
2-trifluoromethy1-3-
fluoromethyl
ethyl




vinylphenyl





2.2.252
2-methoxy-3-vinylphenyl
fluoromethyl
ethyl



2.2.253
2-ethoxy-3-vinylphenyl
fluoromethyl
ethyl



2.2.254
2-trifluoromethoxy-3-
fluoromethyl
ethyl




vinylphenyl





2.2.255
2-nitro-3-vinylphenyl
fluoromethyl
ethyl



2.2.256
2-fluoro-3-ethynylphenyl 
fluoromethyl
ethyl



2.2.257
2-chloro-3-ethynylphenyl 
fluoromethyl
ethyl



2.2.258
2-bromo-3-ethynylphenyl
fluoromethyl
ethyl



2.2.259
2-methyl-3-ethynylphenyl
fluoromethyl
ethyl



2.2.260
2-ethyl-3-ethynylphenyl
fluoromethyl
ethyl



2.2.261
2-cyclopropyl-3-
fluoromethyl
ethyl




ethynylphenyl





2.2.262
2-vinyl-3-ethynylphenyl
fluoromethyl
ethyl



2.2.263
2-cyano-3-ethynylphenyl
fluoromethyl
ethyl



2.2.264
2-trifluoromethyl-3-
fluoromethyl
ethyl




ethynylphenyl





2.2.265
2-methoxy-3-
fluoromethyl
ethyl




ethynylphenyl





2.2.266
2-ethoxy-3-ethynylphenyl
fluoromethyl
ethyl



2.2.267
2-trifluoromethoxy-3-
fluoromethyl
ethyl




ethynylphenyl





2.2.268
2-nitro-3-ethynylphenyl
fluoromethyl
ethyl



2.2.269
2-fluoro-3-ethynylphenyl
fluoromethyl
ethyl



2.2.270
2-fluoro-3-cyanophenyl
fluoromethyl
ethyl



2.2.271
2-chloro-3-cyanophenyl
fluoromethyl
ethyl



2.2.272
2-bromo-3-cyanophenyl
fluoromethyl
ethyl



2.2.273
2-methyl-3-cyanophenyl
fluoromethyl
ethyl



2.2.274
2-ethyl-3-cyanophenyl
fluoromethyl
ethyl



2.2.275
2-ethyl-3-cyanophenyl
chloromethyl
ethyl



2.2.276
2-ethyl-3-cyanophenyl
bromomethyl
ethyl



2.2.277
2-ethyl-3-cyanophenyl
difluoromethyl 
ethyl



2.2.278
2-cyclopropyl-3-
fluoromethyl
ethyl




cyanophenyl





2.2.279
2-vinyl-3-cyanophenyl
fluoromethyl
ethyl



2.2.280
2-ethynyl-3-cyanophenyl
fluoromethyl
ethyl



2.2.281
2-cyano-3-cyanophenyl
fluoromethyl
ethyl



2.2.282
2-trifluoromethyl-3-
fluoromethyl
ethyl




cyanophenyl





2.2.283
2-methoxy-3-cyanophenyl
fluoromethyl
ethyl



2.2.284
2-ethoxy-3-cyanophenyl
fluoromethyl
ethyl



2.2.285
2-trifluoromethoxy-3-
fluoromethyl
ethyl




cyanophenyl





2.2.286
2-nitro-3-cyanophenyl
fluoromethyl
ethyl



2.2.287
2-fluoro-3-hydroxyphenyl
fluoromethyl
ethyl



2.2.288
2-chloro-3-hydroxyphenyl
fluoromethyl
ethyl



2.2.289
2-bromo-3-hydroxyphenyl
fluoromethyl
ethyl



2.2.290
2-methyl-3-hydroxyphenyl
fluoromethyl
ethyl



2.2.291
2-ethyl-3-hydroxyphenyl
fluoromethyl
ethyl



2.2.292
2-cyclopropyl-3-
fluoromethyl
ethyl




hydroxyphenyl





2.2.293
2-vinyl-3-hydroxyphenyl
fluoromethyl
ethyl



2.2.294
2-ethynyl-3-
fluoromethyl
ethyl




hydroxyphenyl





2.2.295
2-cyano-3-hydroxyphenyl
fluoromethyl
ethyl



2.2.296
2-trifluoromethyl-3-
fluoromethyl
ethyl




hydroxyphenyl





2.2.297
2-methoxy-3-
fluoromethyl
ethyl




hydroxyphenyl





2.2.298
2-ethoxy-3-hydroxyphenyl
fluoromethyl
ethyl



2.2.299
2-trifluoromethoxy-3-
fluoromethyl
ethyl




hydroxyphenyl





2.2.300
2-nitro-3-hydroxyphenyl
fluoromethyl
ethyl



2.2.301
2-fluoro-3-methoxyphenyl
fluoromethyl
ethyl



2.2.302
2-chloro-3-methoxyphenyl
fluoromethyl
ethyl



2.2.303
2-bromo-3-methoxyphenyl
fluoromethyl
ethyl



2.2.304
2-methy1-3-
fluoromethyl
ethyl




methoxyphenyl





2.2.305
2-ethyl-3-methoxyphenyl
fluoromethyl
ethyl



2.2.306
2-cyclopropyl-3-
fluoromethyl
ethyl




methoxyphenyl





2.2.307
2-vinyl-3-methoxyphenyl
fluoromethyl
ethyl



2.2.308
2-ethynyl-3-
fluoromethyl
ethyl




methoxyphenyl





2.2.309
2-cyano-3-methoxyphenyl
fluoromethyl
ethyl



2.2.310
2-trifluoromethy1-3-
fluoromethyl
ethyl




methoxyphenyl





2.2.311
2,3-dimethoxy--phenyl
fluoromethyl
ethyl



2.2.312
2-ethoxy-3-
fluoromethyl
ethyl




methoxyphenyl





2.2.313
2-trifluoromethoxy-3-
fluoromethyl
ethyl




methoxyphenyl





2.2.314
2-nitro-3-methoxyphenyl
fluoromethyl
ethyl



2.2.315
2-fluoro-3-ethoxyphenyl
fluoromethyl
ethyl



2.2.316
2-chloro-3-ethoxyphenyl
fluoromethyl
ethyl



2.2.317
2-bromo-3-ethoxyphenyl
fluoromethyl
ethyl



2.2.318
2-methyl-3-ethoxyphenyl 
fluoromethyl
ethyl



2.2.319
2-ethyl-3-ethoxyphenyl
fluoromethyl
ethyl



2.2.320
2-cyclopropy1-3-
fluoromethyl
ethyl




ethoxyphenyl





2.2.321
2-vinyl-3-ethoxyphenyl
fluoromethyl
ethyl



2.2.322
2-ethynyl-3-ethoxyphenyl
fluoromethyl
ethyl



2.2.323
2-cyano-3-ethoxyphenyl
fluoromethyl
ethyl



2.2.324
2-trifluoromethy1-3-
fluoromethyl
ethyl




ethoxyphenyl





2.2.325
2-methoxy-3-
fluoromethyl
ethyl




ethoxyphenyl





2.2.326
2,3-diethoxy--phenyl
fluoromethyl
ethyl



2.2.327
2-trifluoromethoxy-3-
fluoromethyl
ethyl




ethoxyphenyl





2.2.328
2-nitro-3-ethoxyphenyl
fluoromethyl
ethyl



2.2.329
2-fluoro-3-propoxyphenyl
fluoromethyl
ethyl



2.2.330
2-chloro-3-propoxyphenyl
fluoromethyl
ethyl



2.2.331
2-bromo-3-propoxyphenyl
fluoromethyl
ethyl



2.2.332
2-methyl-3-propoxyphenyl
fluoromethyl
ethyl



2.2.333
2-ethyl-3-propoxyphenyl
fluoromethyl
ethyl



2.2.334
2-cyclopropy1-3-
fluoromethyl
ethyl




propoxyphenyl





2.2.335
2-vinyl-3-propoxyphenyl
fluoromethyl
ethyl



2.2.336
2-ethynyl-3-
fluoromethyl
ethyl




propoxyphenyl





2.2.337
2-cyano-3-propoxyphenyl
fluoromethyl
ethyl



2.2.338
2-trifluoromethyl-3-
fluoromethyl
ethyl




propoxyphenyl





2.2.339
2-methoxy-3-
fluoromethyl
ethyl




propoxyphenyl





2.2.340 
2-ethoxy-3-propoxyphenyl
fluoromethyl
ethyl



2.2.341
2-trifluoromethoxy-3-
fluoromethyl
ethyl




propoxyphenyl





2.2.342
2-nitro-3-propoxyphenyl
fluoromethyl
ethyl



2.2.343
2-fluoro-3-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.344
2-chloro-3-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.345
2-bromo-3-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.346
2-methyl-3-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.347
2-ethyl-3-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.348
2-cyclopropyl-3-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.349
2-vinyl-3-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.350
2-ethyny1-3-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.351
2-cyano-3-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.352
2-trifluoromethy1-3-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.353
2-methoxy-3-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.354
2-ethoxy-3-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.355
2-trifluoromethoxy-3-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.356
2-nitro-3-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.357
2-fluoro-3-tert-
fluoromethyl
ethyl




butoxyphenyl





2.2.358
2-chloro-3-tert-
fluoromethyl
ethyl




butoxyphenyl





2.2.359
2-bromo-3-tert-
fluoromethyl
ethyl




butoxyphenyl





2.2.360
2-methyl-3-tert-
fluoromethyl
ethyl




butoxyphenyl





2.2.361
2-ethyl-3-tert-
fluoromethyl
ethyl




butoxyphenyl





2.2.362
2-cyclopropyl-3-tert-
fluoromethyl
ethyl




butoxyphenyl





2.2.363
2-vinyl-3-tert-
fluoromethyl
ethyl




butoxyphenyl





2.2.364
2-ethyny1-3-tert-
fluoromethyl
ethyl




butoxyphenyl





2.2.365
2-cyano-3-tert-
fluoromethyl
ethyl




butoxyphenyl





2.2.366
2-trifluoromethyl-3-tert-
fluoromethyl
ethyl




butoxyphenyl





2.2.367
2-methoxy-3-tert-
fluoromethyl
ethyl




butoxyphenyl





2.2.368
2-ethoxy-3-tert-
fluoromethyl
ethyl




butoxyphenyl





2.2.369
2-trifluoromethoxy-3-tert-
fluoromethyl
ethyl




butoxyphenyl





2.2.370
2-nitro-3-tert-
fluoromethyl
ethyl




butoxyphenyl





2.2.371
2-fluoro-3-
fluoromethyl
ethyl




trifluoromethoxy-phenyl





2.2.372
2-chloro-3-
fluoromethyl
ethyl




trifluoromethoxy-phenyl





2.2.373
2-bromo-3-
fluoromethyl
ethyl




trifluoromethoxy-phenyl





2.2.374
2-methy1-3-
fluoromethyl
ethyl




trifluoromethoxy-phenyl





2.2.375
2-ethy1-3-trifluoromethoxy- 
fluoromethyl
ethyl




phenyl





2.2.376
2-cyclopropyl-3-
fluoromethyl
ethyl




trifluoromethoxy-phenyl





2.2.377
2-vinyl-3-trifluoromethoxy- 
fluoromethyl
ethyl




phenyl





2.2.378
2-ethynyl-3-
fluoromethyl
ethyl




trifluoromethoxy-phenyl





2.2.379
2-cyano-3-
fluoromethyl
ethyl




trifluoromethoxy-phenyl





2.2.380
2-trifluoromethyl-3-
fluoromethyl
ethyl




trifluoromethoxy-phenyl





2.2.381
2-methoxy-3-
fluoromethyl
ethyl




trifluoromethoxy-phenyl





2.2.382
2-ethoxy-3-
fluoromethyl
ethyl




trifluoromethoxy-phenyl





2.2.383
2,3-bis(trifluoro-
fluoromethyl
ethyl




methoxy)phenyl





2.2.384
2-nitro-3-trifluoromethoxy- 
fluoromethyl
ethyl




phenyl





2.2.385
2-fluoro-3-(2,2,2-
fluoromethyl
ethyl




trifluoroethoxy)-phenyl





2.2.386
2-chloro-3-(2,2,2-
fluoromethyl
ethyl




trifluoroethoxy)-phenyl





2.2.387
2-bromo-3-(2,2,2-
fluoromethyl
ethyl




trifluoroethoxy)-phenyl





2.2.388
2-methyl-3-(2,2,2-
fluoromethyl
ethyl




trifluoroethoxy)-phenyl





2.2.389
2-ethyl-3-(2,2,2-
fluoromethyl
ethyl




trifluoroethoxy)-phenyl





2.2.390
2-cyclopropy1-3-(2,2,2-
fluoromethyl
ethyl




trifluoro-ethoxy)phenyl





2.2.391
2-viny1-3-(2,2,2-
fluoromethyl
ethyl




trifluoroethoxy)-phenyl





2.2.392
2-ethyny1-3-(2,2,2-
fluoromethyl
ethyl




trifluoroethoxyphenyl





2.2.393
2-cyano-3-(2,2,2-
fluoromethyl
ethyl




trifluoroethoxy)-phenyl





2.2.394
2-trifluoromethyl-3-(2,2,2-
fluoromethyl
ethyl




trifluoro-ethoxy)phenyl





2.2.395
2-methoxy-3-(2,2,2-
fluoromethyl
ethyl




trifluoroethoxy)-phenyl





2.2.396
2-ethoxy-3-(2,2,2-
fluoromethyl
ethyl




trifluoroethoxy)-phenyl





2.2.397
2-trifluoromethoxy-3-
fluoromethyl
ethyl




(2,2,2-trifluoroethoxy)-






phenyl





2.2.398
2-nitro-3-(2,2,2-trifluoro- 
fluoromethyl
ethyl




ethoxy)phenyl





2.2.399
2-fluoro-3-difluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.400
2-chloro-3-difluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.401
2-bromo-3-difluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.402
2-methyl-3-difluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.403
2-ethyl-3-difluoromethoxy-
fluoromethyl
ethyl




phenyl





2.2.404
2-cyclopropy1-3-
fluoromethyl
ethyl




difluoromethoxy-phenyl





2.2.405
2-vinyl-3-difluoromethoxy-
fluoromethyl
ethyl




phenyl





2.2.406
2-ethyny1-3-difluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.407
2-cyano-3-difluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.408
2-trifluoromethy1-3-
fluoromethyl
ethyl




difluoromethoxy-phenyl





2.2.409
2-methoxy-3-difluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.410
2-ethoxy-3-difluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.411
2-trifluoromethoxy-3-
fluoromethyl
ethyl




difluoromethoxyphenyl





2.2.412
2-nitro-3-difluoromethoxy-
fluoromethyl
ethyl




phenyl





2.2.413
2-fluoro-3-(2-methoxy-
fluoromethyl
ethyl




ethoxy)phenyl





2.2.414
2-chloro-3-(2-methoxy-
fluoromethyl
ethyl




ethoxy)phenyl





2.2.415
2-bromo-3-(2-methoxy-
fluoromethyl
ethyl




ethoxy)phenyl





2.2.416
2-methyl-3-(2-methoxy-
fluoromethyl
ethyl




ethoxy)phenyl





2.2.417
2-ethyl-3-(2-
fluoromethyl
ethyl




methoxyethoxy)phenyl





2.2.418
2-cyclopropyl-3-(2-
fluoromethyl
ethyl




methoxyethoxy)-phenyl





2.2.419
2-viny1-3-(2-methoxy-
fluoromethyl
ethyl




ethoxy)phenyl





2.2.420
2-ethyny1-3-(2-methoxy-
fluoromethyl
ethyl




ethoxy)phenyl





2.2.421
2-cyano-3-(2-methoxy-
fluoromethyl
ethyl




ethoxy)phenyl





2.2.422
2-trifluoromethyl-3-(2-
fluoromethyl
ethyl




methoxyethoxy)-phenyl





2.2.423
2-methoxy-3-(2-methoxy-
fluoromethyl
ethyl




ethoxy)phenyl





2.2.424
2-ethoxy-3-(2-methoxy-
fluoromethyl
ethyl




ethoxy)phenyl





2.2.425
2-trifluoromethoxy-(2-
fluoromethyl
ethyl




methoxyethoxy)-phenyl





2.2.426
2-nitro-3-(2-methoxy-
fluoromethyl
ethyl




ethoxy)phenyl





2.2.427
2-fluoro-3-(tert-butoxy-
fluoromethyl
ethyl




carbonyloxy)phenyl





2.2.428
2-chloro-3-(tert-butoxy-
fluoromethyl
ethyl




carbonyloxy)phenyl





2.2.429
2-bromo-3-(tert-butoxy-
fluoromethyl
ethyl




carbonyloxy)phenyl





2.2.430
2-methyl-3-(tert-butoxy-
fluoromethyl
ethyl




carbonyloxy)phenyl





2.2.431
2-ethyl-3-(tert-butoxy-
fluoromethyl
ethyl




carbonyloxy)phenyl





2.2.432
2-cyclopropyl-3-(tert-
fluoromethyl
ethyl




butoxycarbonyloxy)phenyl





2.2.433
2-vinyl-3-(tert-butoxy-
fluoromethyl
ethyl




carbonyloxy)phenyl





2.2.434
2-ethynyl-3-(tert-butoxy-
fluoromethyl
ethyl




carbonyloxy)phenyl





2.2.435
2-cyano-3-(tert-butoxy-
fluoromethyl
ethyl




carbonyloxy)phenyl





2.2.436
2-trifluoromethyl-3-(tert- 
fluoromethyl
ethyl




butoxycarbonyloxy)phenyl





2.2.437
2-methoxy-3-(tert-butoxy-
fluoromethyl
ethyl




carbonyloxy)phenyl





2.2.438
2-ethoxy-3-(tert-butoxy-
fluoromethyl
ethyl




carbonyloxy)phenyl





2.2.439
2-trifluoromethoxy-3-(tert- 
fluoromethyl
ethyl




butoxycarbonyloxy)phenyl





2.2.440
2-nitro-3-(tert-butoxy-
fluoromethyl
ethyl




carbonyloxy)phenyl





2.2.441
2-fluoro-3-nitrophenyl
fluoromethyl
ethyl



2.2.442
2-chloro-3-nitrophenyl
fluoromethyl
ethyl



2.2.443
2-bromo-3-nitrophenyl
fluoromethyl
ethyl



2.2.444
2-methyl-3-nitrophenyl
fluoromethyl
ethyl



2.2.445
2-ethyl-3-nitrophenyl
fluoromethyl
ethyl



2.2.446
2-cyclopropyl-3-
fluoromethyl
ethyl




nitrophenyl





2.2.447
2-vinyl-3-nitrophenyl
fluoromethyl
ethyl



2.2.448
2-ethynyl-3-nitrophenyl
fluoromethyl
ethyl



2.2.449
2-cyano-3-nitrophenyl
fluoromethyl
ethyl



2.2.450
2-trifluoromethy1-3-
fluoromethyl
ethyl




nitrophenyl





2.2.451
2-methoxy-3-nitrophenyl
fluoromethyl
ethyl



2.2.452
2-ethoxy-3-nitrophenyl
fluoromethyl
ethyl



2.2.453
2-trifluoromethoxy-3-
fluoromethyl
ethyl




nitrophenyl





2.2.454
2-fluoro-3-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.455
2-chloro-3-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.456
2-bromo-3-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.457
2-methy1-3-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.458
2-ethyl-3-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.459
2-cyclopropy1-3-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.460
2-vinyl-3-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.461
2-ethyny1-3-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.462
2-cyano-3-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.463
2-trifluoromethyl-3-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.464
2-methoxy-3-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.465
2-ethoxy-3-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.466
2-trifluoromethoxy-3-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2467
2-nitro-3-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.468
3,5-difluorophenyl
F
methyl
[CDCl3] 3.65 (dd, 1H); 3.96






(s, 3H); 4.12 (dd, 1H); 6.96






(t, 1H); 7.22 (d, 2H).


2.2469
3,5-difluorophenyl
fluoromethyl
ethyl
[CDCl3] 1.33 (t, 3H); 3.50






(d, 1H); 3.80 (d, 1H); 4.30






(q, 2H); 4.67 (s, 1H); 4.79






(s, 1H); 6.89 (t, 1H); 7.20






(d, 2H).


2.2.470
3,5-difluorophenyl
chloromethyl
ethyl
[CDCl3] 1.34 (t, 3H); 3.50






(d, 1H); 3.80 (d, 1H); 4.00






(dd, 2H); 4.32 (m, 2H); 6.89






(t, 1H); 7.20 (d, 2H).


2.2.471
3,5-difluorophenyl
bromomethyl
ethyl
[CDCl3] 1.36 (t, 3H); 3.48






(1H) und 3.55 (d, 1H); 3.89






(d, 1H) und 4.01 (d, 1H);






4.32 (m, 2H); 6.89 (m, 1H);






7.23 (m, 2H).


2.2.472
3,5-difluorophenyl
difluoromethyl
ethyl
[CDCl3] 1.36 (t, 3H); 3.63






(d, 1H); 3.91 (d, 1H); 4.35






(q, 2H); 6.25 (tt, 1H); 6.91






(t, 1H), 7.21 (d, 2H).


2.2.473
3,5-difluorophenyl
trifluoromethyl
ethyl



2.2.474
3,5-difluorophenyl
1,1-dichloroethyl
methyl
[CDCl3] 2.40 (s, 3H); 3.88






(s, 3H); 3.98 (d, 1H); 4.10






(d, 1H); 6.91 (t, 1H); 7.21






(d, 2H).


2.2.475
3,5-difluorophenyl
CN
ethyl
[DMSO] 1.30 (t, 3H); 4.11






(d, 1H); 4.32 (q, 2H); 4.48






(d, 1H); 7.48 (m, 3H).


2.2.476
3,5-difluorophenyl
CN
isopro-
[CDCl3] 1.40 (m, 6H); 3.91





pyl
(d, 1H); 4.12 (d, 1H); 5.20






(m, 1H); 6.96 (m, 1H); 7.19






(m, 2H).


2.2.477
3-chloro-5-fluorophenyl
fluoromethyl
ethyl



2.2.478
3-chloro-5-fluorophenyl
chloromethyl
ethyl



2.2.479
3-chloro-5-fluorophenyl
bromomethyl
ethyl



2.2.480
3-chloro-5-fluorophenyl
difluoromethyl
ethyl



2.2.481
3-chloro-5-fluorophenyl
cyano
ethyl
[CDCl3] 1.45 (t, 3H); 3.91






(d, 1H); 4.15 (d, 1H); 4.42






(q, 2H); 7.25 (m, 1H); 7.32






(d, 1H); 7.40 (s, 1H).


2.2.482
3-bromo-5-fluorophenyl
fluoromethyl
ethyl



2.2.483
3-bromo-5-fluorophenyl
chloromethyl
ethyl



2.2.484
3-bromo-5-fluorophenyl
bromomethyl
ethyl



2.2.485
3-bromo-5-fluorophenyl
difluoromethyl
ethyl



2.2.486
3-iodo-5-fluorophenyl
fluoromethyl
ethyl



2.2.487
3-methyl-5-fluorophenyl
fluoromethyl
ethyl



2.2.488
3-methyl-5-fluorophenyl
chloromethyl
ethyl



2.2.489
3-methyl-5-fluorophenyl
bromomethyl
ethyl



2.2.490
3-methyl-5-fluorophenyl
difluoromethyl
ethyl



2.2.491
3-ethyl-5-fluorophenyl
fluoromethyl
ethyl



2.2.492
3-propyl-5-fluorophenyl
fluoromethyl
ethyl



2.2.493
3-i-propyl-5-fluorophenyl 
fluoromethyl
ethyl



2.2.494
3-n-butyl-5-fluorophenyl
fluoromethyl
ethyl



2.2.495
3-isobutyl-5-fluorophenyl
fluoromethyl
ethyl



2.2.496
3-tert-butyl-5-fluorophenyl
fluoromethyl
ethyl



2.2.497
3-cyclopropy1-5-
fluoromethyl
ethyl




fluorophenyl





2.2.498
3-vinyl-5-fluorophenyl
fluoromethyl
ethyl



2.2.499
3-ethynyl-5-fluorophenyl
fluoromethyl
ethyl



2.2.500
3-cyano-5-fluorophenyl
fluoromethyl
ethyl



2.2.501
3-trifluoromethy1-5-
fluoromethyl
ethyl




fluorophenyl





2.2.502
3-trifluoromethy1-5-
chloromethyl
ethyl




fluorophenyl





2.2.503
3-trifluoromethy1-5-
bromomethyl
ethyl




fluorophenyl





2.2.504
3-trifluoromethy1-5-
difluoromethyl
ethyl




fluorophenyl





2.2.505
3-(methoxycarbonyl)-5-
fluoromethyl
ethyl




fluorophenyl





2.2.506
3-hydroxymethyl-5-
fluoromethyl
ethyl




fluorophenyl





2.2.507
3-carbamoy1-5-
fluoromethyl
ethyl




fluorophenyl





2.2.508
3-hydroxy-5-fluorophenyl
fluoromethyl
ethyl



2.2.509
3-methoxy-5-fluorophenyl
fluoromethyl
ethyl



2.2.510
3-ethoxy-5-fluorophenyl
fluoromethyl
ethyl



2.2.511
3-n-propoxy-5-
fluoromethyl
ethyl




fluorophenyl





2.2.512
3-isopropoxy-5-
fluoromethyl
ethyl




fluorophenyl





2.2.513
3-n-butoxy-5-fluorophenyl
fluoromethyl
ethyl



2.2.514
3-isobutoxy-5-
fluoromethyl
ethyl




fluorophenyl





2.2.515
3-tert-butoxy-5-
fluoromethyl
ethyl




fluorophenyl





2.2.516
3-difluoromethoxy-5-
fluoromethyl
ethyl




fluorophenyl





2.2.517
3-trifluoromethoxy-5-
fluoromethyl
ethyl




fluorophenyl





2.2.518
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl
ethyl




fluorophenyl





2.2.519
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




fluorophenyl





2.2.520
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




fluorophenyl





2.2.521
3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




oxy]-5-fluorophenyl





2.2.522
3-nitro-5-fluorophenyl
fluoromethyl
ethyl



2.2.523
3-acetoxy-5-fluorophenyl
fluoromethyl
ethyl



2.2.524
{3-[(tert-butoxy-carbonyl)-
fluoromethyl
ethyl




amino]-5-fluorophenyl}





2.2.525
3-methylsulfanyl-5-
fluoromethyl
ethyl




fluorophenyl





2.2.526
3,5-dichlorophenyl
fluoromethyl
ethyl



2.2.527
3,5-dichlorophenyl
chloromethyl
ethyl
[CDCl3] 1.35 (t, 3H); 3.51






(d, 1H); 3.80 (d, 1H); 3.96






(d, 1H); 4.03 (d, 1H); 4.33






(m, 2H); 7.43 (s, 1H); 7.58






(s, 1H).


2.2.528
3,5-dichlorophenyl
bromomethyl
ethyl
[CDCl3] 1.35 (t, 3H); 3.47






(d, 1H); 3.62 (d, 1H); 3.90






(d, 1H); 4.32 (m, 2H); 7.40






(s, 1H); 7.55 (s, 2H).


2.2.529
3,5-dichlorophenyl
difluoromethyl
ethyl



2.2.530
3,5-dichlorophenyl
trifluoromethyl
methyl
[CDCl3] 3.75 (d, 1H); 3.92






(s, 3H); 4.00 (d, 1H); 7.45






(s, 1H); 7.58 (s, 2H).


2.2.531
3,5-dichlorophenyl
cyano
ethyl
[CDCl3] 1.41 (t, 3H); 3.90






(d, 1H); 4.15 (d, 1H); 4.42






(q, 2H); 7.49 (d, 1H); 7.55






(d, 2H).


2.2.532
3-bromo-5-chlorophenyl
fluoromethyl
ethyl



2.2.533
3-iodo-5-chlorophenyl
fluoromethyl
ethyl



2.2.534
3-methyl-5-chlorophenyl
fluoromethyl
ethyl



2.2.535
3-ethyl-5-chlorophenyl
fluoromethyl
ethyl



2.2.536
3-propyl-5-chlorophenyl
fluoromethyl
ethyl



2.2.537
3-isopropyl-5-
fluoromethyl
ethyl




chlorophenyl





2.2.538
3-n-butyl-5-chlorophenyl
fluoromethyl
ethyl



2.2.539
3-isobutyl-5-chlorophenyl
fluoromethyl
ethyl



2.2.540
3-tert-butyl-5-chlorophenyl
fluoromethyl
ethyl



2.2.541
3-cyclopropyl-5-
fluoromethyl
ethyl




chlorophenyl





2.2.542
3-vinyl-5-chlorophenyl
fluoromethyl
ethyl



2.2.543
3-ethynyl-5-chlorophenyl
fluoromethyl
ethyl



2.2.544
3-cyano-5-chlorophenyl
fluoromethyl
ethyl



2.2.545
3-trifluoromethyl-5-
fluoromethyl
ethyl




chlorophenyl





2.2.546
3-(hydroxycarbonyl)-5-
fluoromethyl
ethyl




chlorophenyl





2.2.547
3-(methoxycarbonyl)-5-
fluoromethyl
ethyl




chlorophenyl





2.2.548
3-hydroxymethyl-5-
fluoromethyl
ethyl




chlorophenyl





2.2.549
3-carbamoyl-5-
fluoromethyl
ethyl




chlorophenyl





2.2.550
3-hydroxy-5-chlorophenyl
fluoromethyl
ethyl



2.2.551
3-methoxy-5-chlorophenyl
fluoromethyl
ethyl



2.2.552
3-ethoxy-5-chlorophenyl
fluoromethyl
ethyl



2.2.553
3-n-propoxy-5-
fluoromethyl
ethyl




chlorophenyl





2.2.554
3-isopropoxy-5-
fluoromethyl
ethyl




chlorophenyl





2.2.555
3-n-butoxy-5-chlorophenyl
fluoromethyl
ethyl



2.2.556
3-isobutoxy-5-
fluoromethyl
ethyl




chlorophenyl





2.2.557
3-tert-butoxy-5-
fluoromethyl
ethyl




chlorophenyl





2.2.558
3-difluoromethoxy-5-
fluoromethyl
ethyl




chlorophenyl





2.2.559
3-trifluoromethoxy-5-
fluoromethyl
ethyl




chlorophenyl





2.2.560
3-(2,2,2-trifluoroethoxy)-5- 
fluoromethyl
ethyl




chlorophenyl





2.2.561
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




chlorophenyl





2.2.562
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




chlorophenyl





2.2.563
3-[(tert-butoxy-
fluoromethyl
ethyl




carbonyl)oxy]-5-






chlorophenyl





2.2.564
3-nitro-5-chlorophenyl
fluoromethyl
ethyl



2.2.565
3-acetoxy-5-chlorophenyl
fluoromethyl
ethyl



2.2.566
{3-[(tert-butoxy-cabonyl)-
fluoromethyl
ethyl




amino]-5-chlorophenyl}





2.2.567
3-methylsulfany1-5-
fluoromethyl
ethyl




chlorophenyl





2.2.568
3,5-dibromophenyl
fluoromethyl
ethyl



2.2.569
3,5-dibromophenyl
chloromethyl
ethyl



2.2.570
3-iodo-5-bromophenyl
fluoromethyl
ethyl



2.2.571
3-methyl-5-bromophenyl
fluoromethyl
ethyl



2.2.572
3-methyl-5-bromophenyl
chloromethyl
ethyl



2.2.573
3-methyl-5-bromophenyl
bromomethyl
ethyl



2.2.574
3-methyl-5-bromophenyl
difluoromethyl
ethyl



2.2.575
3-methyl-5-bromophenyl
trifluoromethyl
ethyl



2.2.576
3-methyl-5-bromophenyl
cyano
ethyl



2.2.577
3-ethyl-5-bromophenyl
fluoromethyl
ethyl



2.2.578
3-propyl-5-bromophenyl
fluoromethyl
ethyl



2.2.579
3-isopropyl-5-
fluoromethyl
ethyl




bromophenyl





2.2.580
3-n-butyl-5-bromophenyl
fluoromethyl
ethyl



2.2.581
3-isobutyl-5-bromophenyl
fluoromethyl
ethyl



2.2.582
3-tert-butyl-5-
fluoromethyl
ethyl




bromophenyl





2.2.583
3-cyclopropyl-5-
fluoromethyl
ethyl




bromophenyl





2.2.584
3-vinyl-5-bromophenyl
fluoromethyl
ethyl



2.2.585
3-ethynyl-5-bromophenyl
fluoromethyl
ethyl



2.2.586
3-cyano-5-bromophenyl
fluoromethyl
ethyl



2.2.587
3-trifluoromethyl-5-
fluoromethyl
ethyl




bromophenyl





2.2.588
3-(hydroxycarbonyl)-5-
fluoromethyl
ethyl




bromophenyl





2.2.589
3-(methoxycarbonyl)-5-
fluoromethyl
ethyl




bromophenyl





2.2.590
3-hydroxymethy1-5-
fluoromethyl
ethyl




bromophenyl





2.2.591
3-carbamoy1-5-
fluoromethyl
ethyl




bromophenyl





2.2.592
3-hydroxy-5-bromophenyl
fluoromethyl
ethyl



2.2.593
3-methoxy-5-bromophenyl
fluoromethyl
ethyl



2.2.594
3-ethoxy-5-bromophenyl
fluoromethyl
ethyl



2.2.595
3-n-propoxy-5-
fluoromethyl
ethyl




bromophenyl





2.2.596
3-isopropoxy-5-
fluoromethyl
ethyl




bromophenyl





2.2.597
3-n-butoxy-5-
fluoromethyl
ethyl




bromophenyl





2.2.598
3-isobutoxy-5-
fluoromethyl
ethyl




bromophenyl





2.2.599
3-tert-butoxy-5-
fluoromethyl
ethyl




bromophenyl





2.2.600
3-difluoromethoxy-5-
fluoromethyl
ethyl




bromophenyl





2.2.601
3-trifluoromethoxy-5-
fluoromethyl
ethyl




bromophenyl





2.2.602
3-(2,2,2-trifluoroethoxy)-5- 
fluoromethyl
ethyl




bromophenyl





2.2.603
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




bromophenyl





2.2.604
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




bromophenyl





2.2.605
3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




oxy]-5-bromophenyl





2.2.606
3-nitro-5-bromophenyl
fluoromethyl
ethyl



2.2.607
3-acetoxy-5-bromophenyl
fluoromethyl
ethyl



2.2.608
{3-[(tert-butoxy-carbonyl)-
fluoromethyl
ethyl




amino]-5-bromophenyl}





2.2.609
3-methylsulfany1-5-
fluoromethyl
ethyl




bromophenyl





2.2.610
3,5-diiodophenyl
fluoromethyl
ethyl



2.2.611
3-methyl-5-iodophenyl
fluoromethyl
ethyl



2.2.612
3-ethyl-5-iodophenyl
fluoromethyl
ethyl



2.2.613
3-propyl-5-iodophenyl
fluoromethyl
ethyl



2.2.614
3-isopropyl-5-iodophenyl
fluoromethyl
ethyl



2.2.615
3-n-butyl-5-iodophenyl
fluoromethyl
ethyl



2.2.616
3-isobutyl-5-iodophenyl
fluoromethyl
ethyl



2.2.617
3-tert-butyl-5-iodophenyl
fluoromethyl
ethyl



2.2.618
3-cyclopropyl-5-
fluoromethyl
ethyl




iodophenyl





2.2.619
3-vinyl-5-iodophenyl
fluoromethyl
ethyl



2.2.620
3-ethynyl-5-iodophenyl
fluoromethyl
ethyl



2.2.621
3-cyano-5-iodophenyl
fluoromethyl
ethyl



2.2.622
3-trifluoromethyl-5-
fluoromethyl
ethyl




iodophenyl





2.2.623
3-(hydroxycarbonyl)-5-
fluoromethyl
ethyl




iodophenyl





2.2.624
3-(methoxycarbonyl)-5-
fluoromethyl
ethyl




iodophenyl





2.2.625
3-hydroxymethyl-5-
fluoromethyl
ethyl




iodophenyl





2.2.626
3-carbamoyl-5-iodophenyl
fluoromethyl
ethyl



2.2.627
3-hydroxy-5-iodophenyl
fluoromethyl
ethyl



2.2.628
3-methoxy-5-iodophenyl
fluoromethyl
ethyl



2.2.629
3-ethoxy-5-iodophenyl
fluoromethyl
ethyl



2.2.630
3-n-propoxy-5-iodophenyl
fluoromethyl
ethyl



2.2.631
3-isopropoxy-5-
fluoromethyl
ethyl




iodophenyl





2.2.632
3-n-butoxy-5-iodophenyl
fluoromethyl
ethyl



2.2.633
3-isobutoxy-5-iodophenyl
fluoromethyl
ethyl



2.2.634
3-tert-butoxy-5-iodophenyl
fluoromethyl
ethyl



2.2.635
3-difluoromethoxy-5-
fluoromethyl
ethyl




iodophenyl





2.2.636
3-trifluoromethoxy-5-
fluoromethyl
ethyl




iodophenyl





2.2.637
3-(2,2,2-trifluoroethoxy)-5- 
fluoromethyl
ethyl




iodophenyl





2.2.638
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




iodophenyl





2.2.639
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




iodophenyl





2.2.640
3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




oxy]-5-iodophenyl





2.2.641
3-nitro-5-iodophenyl
fluoromethyl
ethyl



2.2.642
3-acetoxy-5-iodophenyl
fluoromethyl
ethyl



2.2.643
{3-[(tert-butoxy-carbonyl)-
fluoromethyl
ethyl




amino]-5-iodophenyl}





2.2.644
3-methylsulfanyl-5-
fluoromethyl
ethyl




iodophenyl





2.2.645
3,5-dimethylphenyl
fluoromethyl
ethyl



2.2.646
3-ethyl-5-methylphenyl
fluoromethyl
ethyl



2.2.647
3-propyl-5-methylphenyl
fluoromethyl
ethyl



2.2.648
3-isopropyl-5-
fluoromethyl
ethyl




methylphenyl





2.2.649
3-n-butyl-5-methylphenyl
fluoromethyl
ethyl



2.2.650
3-isobutyl-5-methylphenyl
fluoromethyl
ethyl



2.2.651
3-tert-butyl-5-
fluoromethyl
ethyl




methylphenyl





2.2.652
3-cyclopropyl-5-
fluoromethyl
ethyl




methylphenyl





2.2.653
3-vinyl-5-methylphenyl
fluoromethyl
ethyl



2.2.654
3-ethynyl-5-methylphenyl
fluoromethyl
ethyl



2.2.655
3-cyano-5-methylphenyl
fluoromethyl
ethyl



2.2.656
3-trifluoromethyl-5-
fluoromethyl
ethyl




methylphenyl





2.2.657
3-(hydroxycarbonyl)-5-
fluoromethyl
ethyl




methylphenyl





2.2.658
3-(methoxycarbonyl)-5-
fluoromethyl
ethyl




methylphenyl





2.2.659
3-hydroxymethyl-5-
fluoromethyl
ethyl




methylphenyl





2.2.660
3-carbamoyl-5-
fluoromethyl
ethyl




methylphenyl





2.2.661
3-hydroxy-5-methylphenyl
fluoromethyl
ethyl



2.2.662
3-methoxy-5-
fluoromethyl
ethyl




methylphenyl





2.2.663
3-ethoxy-5-methylphenyl
fluoromethyl
ethyl



2.2.664
3-n-propoxy-5-
fluoromethyl
ethyl




methylphenyl





2.2.665
3-n-butoxy-5-
fluoromethyl
ethyl




methylphenyl





2.2.666
3-isobutoxy-5-
fluoromethyl
ethyl




methylphenyl





2.2.667
3-tert-butoxy-5-
fluoromethyl
ethyl




methylphenyl





2.2.668
3-difluoromethoxy-5-
fluoromethyl
ethyl




methylphenyl





2.2.669
3-trifluoromethoxy-5-
fluoromethyl
ethyl




methylphenyl





2.2.670
3-(2,2,2-trifluoroethoxy)-5- 
fluoromethyl
ethyl




methylphenyl





2.2.671
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




methylphenyl





2.2.672
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




methylphenyl





2.2.673
3-[(tert-butoxy-
fluoromethyl
ethyl




carbonyl)oxy]-5-






methylphenyl





2.2.674
3-nitro-5-methylphenyl
fluoromethyl
ethyl



2.2.675
3-acetoxy-5-methylphenyl
fluoromethyl
ethyl



2.2.676
{3-[(tert-butoxy-carbonyl)-
fluoromethyl
ethyl




amino]-5-methylphenyl}





2.2.677
3-methylsulfanyl-5-
fluoromethyl
ethyl




methylphenyl





2.2.678
3,5-diethylphenyl
fluoromethyl
ethyl



2.2.679
3-propyl-5-ethylphenyl
fluoromethyl
ethyl



2.2.680
3-isopropyl-5-ethylphenyl
fluoromethyl
ethyl



2.2.681
3-n-butyl-5-ethylphenyl
fluoromethyl
ethyl



2.2.682
3-isobutyl-5-ethylphenyl
fluoromethyl
ethyl



2.2.683
3-tert-butyl-5-ethylphenyl
fluoromethyl
ethyl



2.2.684
3-cyclopropy1-5-
fluoromethyl
ethyl




ethylphenyl





2.2.685
3-vinyl-5-ethylphenyl
fluoromethyl
ethyl



2.2.686
3-ethynyl-5-ethylphenyl
fluoromethyl
ethyl



2.2.687
3-cyano-5-ethylphenyl
fluoromethyl
ethyl



2.2.688
3-trifluoromethyl-5-
fluoromethyl
ethyl




ethylphenyl





2.2.689
3-(hydroxycarbonyl)-5-
fluoromethyl
ethyl




ethylphenyl





2.2.690
3-(methoxycarbonyl)-5-
fluoromethyl
ethyl




ethylphenyl





2.2.691
3-hydroxymethyl-5-
fluoromethyl
ethyl




ethylphenyl





2.2.692
3-carbamoyl-5-
fluoromethyl
ethyl




ethylphenyl





2.2.693
3-hydroxy-5-ethylphenyl
fluoromethyl
ethyl



2.2.694
3-methoxy-5-ethylphenyl
fluoromethyl
ethyl



2.2.695
3-ethoxy-5-ethylphenyl
fluoromethyl
ethyl



2.2.696
3-n-propoxy-5-ethylphenyl
fluoromethyl
ethyl



2.2.697
3-n-butoxy-5-ethylphenyl
fluoromethyl
ethyl



2.2.698
3-isobutoxy-5-ethylphenyl
fluoromethyl
ethyl



2.2.699
3-tert-butoxy-5-
fluoromethyl
ethyl




ethylphenyl





2.2.700
3-difluoromethoxy-5-
fluoromethyl
ethyl




ethylphenyl





2.2.701
3-trifluoromethoxy-5-
fluoromethyl
ethyl




ethylphenyl





2.2.702
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl
ethyl




ethylphenyl





2.2.703
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




ethylphenyl





2.2.704
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




ethylphenyl





2.2.705
3-[(tert-butoxy-
fluoromethyl
ethyl




carbonyl)oxy]-5-






ethylphenyl





2.2.706
3-nitro-5-ethylphenyl
fluoromethyl
ethyl



2.2.707
3-acetoxy-5-ethylphenyl
fluoromethyl
ethyl



2.2.708
{3-[(tert-butoxy-carbonyl)-
fluoromethyl
ethyl




amino]-5-ethylphenyl}





2.2.709
3-methylsulfany1-5-
fluoromethyl
ethyl




ethylphenyl





2.2.710
3,5-dipropylphenyl
fluoromethyl
ethyl



2.2.711
3-isopropy1-5-
fluoromethyl
ethyl




propylphenyl





2.2.712
3-n-butyl-5-propylphenyl
fluoromethyl
ethyl



2.2.713
3-isobutyl-5-propylphenyl
fluoromethyl
ethyl



2.2.714
3-tert-butyl-5-propylphenyl
fluoromethyl
ethyl



2.2.715
3-cyclopropy1-5-
fluoromethyl
ethyl




propylphenyl





2.2.716
3-vinyl-5-propylphenyl
fluoromethyl
ethyl



2.2.717
3-ethynyl-5-propylphenyl
fluoromethyl
ethyl



2.2.718
3-cyano-5-propylphenyl
fluoromethyl
ethyl



2.2.719
3-trifluoromethyl-5-
fluoromethyl
ethyl




propylphenyl





2.2.720
3-(hydroxycarbonyl)-5-
fluoromethyl
ethyl




propylphenyl





2.2.721
3-(methoxycarbonyl)-5-
fluoromethyl
ethyl




propylphenyl





2.2.722
3-hydroxymethy1-5-
fluoromethyl
ethyl




propylphenyl





2.2.723
3-carbamoy1-5-
fluoromethyl
ethyl




propylphenyl





2.2.724
3-hydroxy-5-propylphenyl
fluoromethyl
ethyl



2.2.725
3-methoxy-5-propylphenyl
fluoromethyl
ethyl



2.2.726
3-ethoxy-5-propylphenyl
fluoromethyl
ethyl



2.2.727
3-n-propoxy-5-
fluoromethyl
ethyl




propylphenyl





2.2.728
3-n-butoxy-5-propylphenyl
fluoromethyl
ethyl



2.2.729
3-isobutoxy-5-
fluoromethyl
ethyl




propylphenyl





2.2.730
3-tert-butoxy-5-
fluoromethyl
ethyl




propylphenyl





2.2.731
3-difluoromethoxy-5-
fluoromethyl
ethyl




propylphenyl





2.2.732
3-trifluoromethoxy-5-
fluoromethyl
ethyl




ethylphenyl





2.2.733
3-(2,2,2-trifluoroethoxy)-5- 
fluoromethyl
ethyl




propylphenyl





2.2.734
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




propylphenyl





2.2.735
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




propylphenyl





2.2.736
3-[(tert-butoxy-
fluoromethyl
ethyl




carbonyl)oxy]-5-






propylphenyl





2.2.737
3-nitro-5-propylphenyl
fluoromethyl
ethyl



2.2.738
3-acetoxy-5-propylphenyl
fluoromethyl
ethyl



2.2.739
{3-[(tert-butoxy-carbonyl)-
fluoromethyl
ethyl




amino]-5-propylphenyl}





2.2.740
3-methylsulfany1-5-
fluoromethyl
ethyl




propylphenyl





2.2.741
3,5-diisopropylphenyl
fluoromethyl
ethyl



2.2.742
3-n-buty1-5-
fluoromethyl
ethyl




isopropylphenyl





2.2.743
3-isobuty1-5-
fluoromethyl
ethyl




isopropylphenyl





2.2.744
3-tert-buty1-5-
fluoromethyl
ethyl




isopropylphenyl





2.2.745
3-cyclopropyl-5-
fluoromethyl
ethyl




isopropylphenyl





2.2.746
3-vinyl-5-isopropylphenyl
fluoromethyl
ethyl



2.2.747
3-ethyny1-5-
fluoromethyl
ethyl




isopropylphenyl





2.2.748
3-cyano-5-
fluoromethyl
ethyl




isopropylphenyl





2.2.749
3-trifluoromethy1-5-
fluoromethyl
ethyl




isopropylphenyl





2.2.750
3-(hydroxycarbonyl)-5-
fluoromethyl
ethyl




isopropylphenyl





2.2.751
3-(methoxycarbonyl)-5-
fluoromethyl
ethyl




isopropylphenyl





2.2.752
3-hydroxymethy1-5-
fluoromethyl
ethyl




isopropylphenyl





2.2.753
3-carbamoyl-5-
fluoromethyl
ethyl




isopropylphenyl





2.2.754
3-hydroxy-5-
fluoromethyl
ethyl




isopropylphenyl





2.2.755
3-methoxy-5-
fluoromethyl
ethyl




isopropylphenyl





2.2.756
3-ethoxy-5-
fluoromethyl
ethyl




isoperopylphenyl





2.2.757
3-n-propoxy-5-
fluoromethyl
ethyl




isopropylphenyl





2.2.758
3-n-butoxy-5-
fluoromethyl
ethyl




isopropylphenyl





2.2.759
3-isobutoxy-5-
fluoromethyl
ethyl




isopropylphenyl





2.2.760
3-tert-butoxy-5-
fluoromethyl
ethyl




isopropylphenyl





2.2.761
3-difluoromethoxy-5-
fluoromethyl
ethyl




isopropylphenyl





2.2.762
3-trifluoromethoxy-5-
fluoromethyl
ethyl




isopropylphenyl





2.2.763
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl
ethyl




isopropylphenyl





2.2.764
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




isopropylphenyl





2.2.765
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




propylphenyl





2.2.766
3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




oxy]-5-isopropylphenyl





2.2.767
3-nitro-5-isopropylphenyl
fluoromethyl
ethyl



2.2.768
3-acetoxy-5-
fluoromethyl
ethyl




isopropylphenyl





2.2.769
{3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




amino]-5-isopropylphenyl}





2.2.770
3-methylsulfany1-5-
fluoromethyl
ethyl




isopropylphenyl





2.2.771
3,5-dibutylphenyl
fluoromethyl
ethyl



2.2.772
3-isobutyl-5-butylphenyl
fluoromethyl
ethyl



2.2.773
3-tert-butyl-5-butylphenyl
fluoromethyl
ethyl



2.2.774
3-cyclopropy1-5-
fluoromethyl
ethyl




butylphenyl





2.2.775
3-vinyl-5-butylphenyl
fluoromethyl
ethyl



2.2.776
3-ethynyl-5-butylphenyl
fluoromethyl
ethyl



2.2.777
3-cyano-5-butylphenyl
fluoromethyl
ethyl



2.2.778
3-trifluoromethyl-5-
fluoromethyl
ethyl




butylphenyl





2.2.779
3-(hydroxycarbonyl)-5-
fluoromethyl
ethyl




butylphenyl





2.2.780
3-(methoxycarbonyl)-5-
fluoromethyl
ethyl




butylphenyl





2.2.781
3-hydroxymethy1-5-
fluoromethyl
ethyl




butylphenyl





2.2.782
3-carbamoy1-5-
fluoromethyl
ethyl




butylphenyl





2.2.783
3-hydroxy-5-butylphenyl
fluoromethyl
ethyl



2.2.784
3-methoxy-5-butylphenyl
fluoromethyl
ethyl



2.2.785
3-ethoxy-5-butylphenyl
fluoromethyl
ethyl



2.2.786
3-n-propoxy-5-butylphenyl
fluoromethyl
ethyl



2.2.787
3-n-butoxy-5-butylphenyl
fluoromethyl
ethyl



2.2.788
3-isobutoxy-5-butylphenyl
fluoromethyl
ethyl



2.2.789
3-tert-butoxy-5-
fluoromethyl
ethyl




butylphenyl





2.2.790
3-difluoromethoxy-5-
fluoromethyl
ethyl




butylphenyl





2.2.791
3-trifluoromethoxy-5-
fluoromethyl
ethyl




butylphenyl





2.2.792
3-(2,2,2-trifluoroethoxy)-5- 
fluoromethyl
ethyl




butylphenyl





2.2.793
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




butylphenyl





2.2.794
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




butylphenyl





2.2.795
3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




oxy]-5-butylphenyl





2.2.796
3-nitro-5-butylphenyl
fluoromethyl
ethyl



2.2.797
3-acetoxy-5-butylphenyl
fluoromethyl
ethyl



2.2.798
{3-[(tert-butoxy-carbonyl)-
fluoromethyl
ethyl




amino]-5-butylphenyl}





2.2.799
3-methylsulfanyl-5-
fluoromethyl
ethyl




butylphenyl





2.2.800
3,5-diisobutylphenyl
fluoromethyl
ethyl



2.2.801
3-tert-butyl-5-
fluoromethyl
ethyl




isobutylphenyl





2.2.802
3-cyclopropyl-5-
fluoromethyl
ethyl




isobutylphenyl





2.2.803
3-vinyl-5-isobutylphenyl
fluoromethyl
ethyl



2.2.804
3-ethynyl-5-isobutylphenyl
fluoromethyl
ethyl



2.2.805
3-cyano-5-isobutylphenyl
fluoromethyl
ethyl



2.2.806
3-trifluoromethyl-5-
fluoromethyl
ethyl




isobutylphenyl





2.2.807
3-(hydroxycarbonyl)-5-
fluoromethyl
ethyl




isobutylphenyl





2.2.808
3-(methoxycarbonyl)-5-
fluoromethyl
ethyl




isobutylphenyl





2.2.809
3-hydroxymethyl-5-
fluoromethyl
ethyl




isobutylphenyl





2.2.810
3-carbamoyl-5-
fluoromethyl
ethyl




isobutylphenyl





2.2.811
3-hydroxy-5-
fluoromethyl
ethyl




isobutylphenyl





2.2.812
3-methoxy-5-
fluoromethyl
ethyl




isobutylphenyl





2.2.813
3-ethoxy-5-isobutylphenyl
fluoromethyl
ethyl



2.2.814
3-n-propoxy-5-
fluoromethyl
ethyl




isobutylphenyl





2.2.815
3-n-butoxy-5-
fluoromethyl
ethyl




isobutylphenyl





2.2.816
3-isobutoxy-5-
fluoromethyl
ethyl




isobutylphenyl





2.2.817
3-tert-butoxy-5-
fluoromethyl
ethyl




isobutylphenyl





2.2.818
3-difluoromethoxy-5-
fluoromethyl
ethyl




isobutylphenyl





2.2.819
3-trifluoromethoxy-5-
fluoromethyl
ethyl




isobutylphenyl





2.2.820
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl
ethyl




isobutylphenyl





2.2.821
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




isobutylphenyl





2.2.822
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




isobutylphenyl





2.2.823
3-[(tert-butoxy-
fluoromethyl
ethyl




carbonyl)oxy]-5-






isobutylphenyl





2.2.824
3-nitro-5-isobutylphenyl
fluoromethyl
ethyl



2.2.825
3-acetoxy-5-
fluoromethyl
ethyl




isobutylphenyl





2.2.826
{3-[(tert-butoxy-carbonyl)-
fluoromethyl
ethyl




amino]-5-isobutylphenyl}





2.2.827
3-methylsulfany1-5-
fluoromethyl
ethyl




isobutylphenyl





2.2.828
3,5-di(tert-butyl)phenyl
fluoromethyl
ethyl



2.2.829
3-cyclopropyl-5-tert-
fluoromethyl
ethyl




butylphenyl





2.2.830
3-vinyl-5-tert-butylphenyl
fluoromethyl
ethyl



2.2.831
3-ethynyl-5-tert-
fluoromethyl
ethyl




butylphenyl





2.2.832
3-cyano-5-tert-butylphenyl
fluoromethyl
ethyl



2.2.833
3-trifluoromethyl-5-tert-
fluoromethyl
ethyl




butylphenyl





2.2.834
3-(hydroxycarbonyl)-5-
fluoromethyl
ethyl




tert-butylphenyl





2.2.835
3-(methoxycarbonyl)-5-
fluoromethyl
ethyl




tert-butylphenyl





2.2.836
3-hydroxymethyl-5-tert-
fluoromethyl
ethyl




butylphenyl





2.2.837
3-carbamoy1-5-tert-
fluoromethyl
ethyl




butylphenyl





2.2.838
3-hydroxy-5-tert-
fluoromethyl
ethyl




butylphenyl





2.2.839
3-methoxy-5-tert-
fluoromethyl
ethyl




butylphenyl





2.2.840
3-ethoxy-5-tert-
fluoromethyl
ethyl




butylphenyl





2.2.841
3-n-propoxy-5-tert-
fluoromethyl
ethyl




butylphenyl





2.2.842
3-n-butoxy-5-tert-
fluoromethyl
ethyl




butylphenyl





2.2.843
3-isobutoxy-5-tert-
fluoromethyl
ethyl




butylphenyl





2.2.844
3-tert-butoxy-5-tert-
fluoromethyl
ethyl




butylphenyl





2.2.845
3-difluoromethoxy-5-tert-
fluoromethyl
ethyl




butylphenyl





2.2.846
3-trifluoromethoxy-5-tert-
fluoromethyl
ethyl




butylphenyl





2.2.847
3-(2,2,2-trifluoroethoxy)-5- 
fluoromethyl
ethyl




tert-butylphenyl





2.2.848
3-(2-chloroethoxy)-5-tert-
fluoromethyl
ethyl




butylphenyl





2.2.849
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




tert-butylphenyl





2.2.850
3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




oxy]-5-tert-butylphenyl





2.2.851
3-nitro-5-tert-butylphenyl
fluoromethyl
ethyl



2.2.852
3-acetoxy-5-tert-
fluoromethyl
ethyl




butylphenyl





2.2.853
{3-[(tert-butoxy-carbonyl)-
fluoromethyl
ethyl




amino]-5-tert-butylphenyl}





2.2.854
3-methylsulfanyl-5-tert-
fluoromethyl
ethyl




butylphenyl





2.2.855
3-tert-butyl-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.856
3,5-dicyclopropylphenyl
fluoromethyl
ethyl



2.2.857
3-vinyl-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.858
3-ethyny1-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.859
3-cyano-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.860
3-trifluoromethyl-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.861
3-(hydroxycarbonyl)-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.862
3-(methoxycarbonyl)-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.863
3-hydroxymethy1-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.864
3-carbamoyl-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.865
3-hydroxy-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.866
3-methoxy-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.867
3-ethoxy-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.868
3-n-propoxy-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.869
3-n-butoxy-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.870
3-isobutoxy-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.871
3-tert-butoxy-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.872
3-difluoromethoxy-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.873
3-trifluoromethoxy-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.874
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.875
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.876
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.877
3-[(tert-butoxy-
fluoromethyl
ethyl




carbonyl)oxy]-5-






cyclopropylphenyl





2.2.878
3-nitro-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.879
3-acetoxy-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.880
{3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




amino]-5-cyclopropyl-






phenyl}





2.2.881
3-methylsulfany1-5-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.882
3,5-divinylphenyl
fluoromethyl
ethyl



2.2.883
3-ethynyl-5-vinylphenyl
fluoromethyl
ethyl



2.2.884
3-cyano-5-vinylphenyl
fluoromethyl
ethyl



2.2.885
3-trifluoromethyl-5-
fluoromethyl
ethyl




vinylphenyl





2.2.886
3-(hydroxycarbonyl)-5-
fluoromethyl
ethyl




vinylphenyl





2.2.887
3-(methoxycarbonyl)-5-
fluoromethyl
ethyl




vinylphenyl





2.2.888
3-hydroxymethy1-5-
fluoromethyl
ethyl




vinylphenyl





2.2.889
3-carbamoyl-5-vinylphenyl
fluoromethyl
ethyl



2.2.890
3-hydroxy-5-vinylphenyl
fluoromethyl
ethyl



2.2.891
3-methoxy-5-vinylphenyl
fluoromethyl
ethyl



2.2.892
3-ethoxy-5-vinylphenyl
fluoromethyl
ethyl



2.2.893
3-n-propoxy-5-vinylphenyl
fluoromethyl
ethyl



2.2.894
3-n-butoxy-5-vinylphenyl
fluoromethyl
ethyl



2.2.895
3-isobutoxy-5-vinylphenyl
fluoromethyl
ethyl



2.2.896
3-tert-butoxy-5-
fluoromethyl
ethyl




vinylphenyl





2.2.897
3-difluoromethoxy-5-
fluoromethyl
ethyl




vinylphenyl





2.2.898
3-trifluoromethoxy-5-
fluoromethyl
ethyl




vinylphenyl





2.2.899
3-(2,2,2-trifluoroethoxy)-5- 
fluoromethyl
ethyl




vinylphenyl





2.2.900
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




vinylphenyl





2.2.901
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




vinylphenyl





2.2.902
3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




oxy]-5-vinylphenyl





2.2.903
3-nitro-5-vinylphenyl
fluoromethyl
ethyl



2.2.904
3-acetoxy-5-vinylphenyl
fluoromethyl
ethyl



2.2.905
{3-[(tert-butoxy-carbonyl)-
fluoromethyl
ethyl




amino]-5-vinylphenyl}





2.2.906
3-methylsulfany1-5-
fluoromethyl
ethyl




vinylphenyl





2.2.907
3,5-diethynylphenyl
fluoromethyl
ethyl



2.2.908
3-cyano-5-ethynylphenyl
fluoromethyl
ethyl



2.2.909
3-trifluoromethyl-5-
fluoromethyl
ethyl




ethynylphenyl





2.2.910
3-(hydroxycarbonyl)-5-
fluoromethyl
ethyl




ethynylphenyl





2.2.911
3-(methoxycarbonyl)-5-
fluoromethyl
ethyl




ethynylphenyl





2.2.912
3-hydroxymethyl-5-
fluoromethyl
ethyl




ethynylphenyl





2.2.913
3-carbamoyl-5-
fluoromethyl
ethyl




ethynylphenyl





2.2.914
3-hydroxy-5-
fluoromethyl
ethyl




ethynylphenyl





2.2.915
3-methoxy-5-
fluoromethyl
ethyl




ethynylphenyl





2.2.916
3-ethoxy-5-ethynylphenyl
fluoromethyl
ethyl



2.2.917
3-n-propoxy-5-
fluoromethyl
ethyl




ethynylphenyl





2.2.918
3-n-butoxy-5-
fluoromethyl
ethyl




ethynylphenyl





2.2.919
3-isobutoxy-5-
fluoromethyl
ethyl




ethynylphenyl





2.2.920
3-tert-butoxy-5-
fluoromethyl
ethyl




ethynylphenyl





2.2.921
3-difluoromethoxy-5-
fluoromethyl
ethyl




ethynylphenyl





2.2.922
3-trifluoromethoxy-5-
fluoromethyl
ethyl




ethynylphenyl





2.2.923
3-(2,2,2-trifluoroethoxy)-5- 
fluoromethyl
ethyl




ethynylphenyl





2.2.924
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




ethynylphenyl





2.2.925
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




ethynylphenyl





2.2.926
3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




oxy]-5-ethynylphenyl





2.2.927
3-nitro-5-ethynylphenyl
fluoromethyl
ethyl



2.2.928
3-acetoxy-5-ethynylphenyl
fluoromethyl
ethyl



2.2.929
{3-[(tert-butoxy-carbonyl)-
fluoromethyl
ethyl




amino]-5-ethynylphenyl}





2.2.930
3-methylsulfany1-5-
fluoromethyl
ethyl




ethynylphenyl





2.2.931
3,5-dicyanophenyl
fluoromethyl
ethyl



2.2.932
3-trifluoromethyl-5-
fluoromethyl
ethyl




cyanophenyl





2.2.933
3-(hydroxycarbonyl)-5-
fluoromethyl
ethyl




cyanophenyl





2.2.934
3-(methoxycarbonyl)-5-
fluoromethyl
ethyl




cyanophenyl





2.2.935
3-hydroxymethy1-5-
fluoromethyl
ethyl




cyanophenyl





2.2.936
3-carbamoy1-5-
fluoromethyl
ethyl




cyanophenyl





2.2.937
3-hydroxy-5-cyanophenyl
fluoromethyl
ethyl



2.2.938
3-methoxy-5-cyanophenyl
fluoromethyl
ethyl



2.2.939
3-ethoxy-5-cyanophenyl
fluoromethyl
ethyl



2.2.940
3-n-propoxy-5-
fluoromethyl
ethyl




cyanophenyl





2.2.941
3-n-butoxy-5-cyanophenyl
fluoromethyl
ethyl



2.2.942
3-isobutoxy-5-
fluoromethyl
ethyl




cyanophenyl





2.2.943
3-tert-butoxy-5-
fluoromethyl
ethyl




cyanophenyl





2.2.944
3-difluoromethoxy-5-
fluoromethyl
ethyl




cyanophenyl





2.2.945
3-trifluoromethoxy-5-
fluoromethyl
ethyl




cyanophenyl





2.2.946
3-(2,2,2-trifluoroethoxy)-5- 
fluoromethyl
ethyl




cyanophenyl





2.2.947
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




cyanophenyl





2.2.948
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




cyanophenyl





2.2.949
3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




oxy]-5-cyanophenyl





2.2.950
3-nitro-5-cyanophenyl
fluoromethyl
ethyl



2.2.951
3-acetoxy-5-cyanophenyl
fluoromethyl
ethyl



2.2.952
{3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




amino-5-cyanophenyl}





2.2.953
3-methylsulfanyl-5-
fluoromethyl
ethyl




cyanophenyl





2.2.954
3,5-di(trifluoromethyl)-
fluoromethyl
ethyl




phenyl





2.2.955
3-(hydroxycarbonyl)-5-
fluoromethyl
ethyl




trifluoromethylphenyl





2.2.956
3-(methoxycarbonyl)-5-
fluoromethyl
ethyl




trifluoromethylphenyl





2.2.957
3-hydroxymethyl-5-
fluoromethyl
ethyl




trifluoromethylphenyl





2.2.958
3-carbamoy1-5-
fluoromethyl
ethyl




trifluoromethylphenyl





2.2.959
3-hydroxy-5-
fluoromethyl
ethyl




trifluoromethylphenyl





2.2.960
3-methoxy-5-
fluoromethyl
ethyl




trifluoromethylphenyl





2.2.961
3-ethoxy-5-
fluoromethyl
ethyl




trifluoromethylphenyl





2.2.962
3-n-propoxy-5-
fluoromethyl
ethyl




trifluoromethylphenyl





2.2.963
3-n-butoxy-5-
fluoromethyl
ethyl




trifluoromethylphenyl





2.2.964
3-isobutoxy-5-
fluoromethyl
ethyl




trifluoromethylphenyl





2.2.965
3-tert-butoxy-5-
fluoromethyl
ethyl




trifluoromethylphenyl





2.2.966
3-difluoromethoxy-5-
fluoromethyl
ethyl




trifluoromethylphenyl





2.2.967
3-trifluoromethoxy-5-
fluoromethyl
ethyl




trifluoromethylphenyl





2.2.968
3-(2,2,2-trifluoro-ethoxy)- 
fluoromethyl
ethyl




5-trifluoro-methylphenyl





2.2.969
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




trifluoromethyl-phenyl





2.2.970
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




trifluoromethyl-phenyl





2.2.971
3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




oxy]-5-trifluoromethyl-






phenyl





2.2.972
3-nitro-5-trifluoromethyl-
fluoromethyl
ethyl




phenyl





2.2.973
3-acetoxy-5-trifluoro-
fluoromethyl
ethyl




methylphenyl





2.2.974
{3-[(tert-butoxy-carbonyl)-
fluoromethyl
ethyl




amino]-5-trifluoromethyl-






phenyl}





2.2.975
3-methylsulfanyl-5-
fluoromethyl
ethyl




trifluoromethylphenyl





2.2.976
3,5-bis(hydroxy-
fluoromethyl
ethyl




carbonyl)phenyl





2.2.977
3-(methoxycarbonyl)-5-
fluoromethyl
ethyl




(hydroxycarbonyl)phenyl





2.2.978
3-hydroxymethyl-5-
fluoromethyl
ethyl




(hydroxycarbonyl)phenyl





2.2.979
3-carbamoyl-5-
fluoromethyl
ethyl




(hydroxycarbonyl)phenyl





2.2.980
3-hydroxy-5-
fluoromethyl
ethyl




(hydroxycarbonyl)phenyl





2.2.981
3-methoxy-5-
fluoromethyl
ethyl




(hydroxycarbonyl)phenyl





2.2.982
3-ethoxy-5-
fluoromethyl
ethyl




(hydroxycarbonyl)phenyl





2.2.983
3-n-propoxy-5-
fluoromethyl
ethyl




(hydroxycarbonyl)phenyl





2.2.984
3-n-butoxy-5-
fluoromethyl
ethyl




(hydroxycarbonyl)phenyl





2.2.985
3-isobutoxy-5-
fluoromethyl
ethyl




(hydroxycarbonyl)phenyl





2.2.986
3-tert-butoxy-5-
fluoromethyl
ethyl




(hydroxycarbonyl)phenyl





2.2.987
3-difluoromethoxy-5-
fluoromethyl
ethyl




(hydroxycarbonyl)phenyl





2.2.988
3-trifluoromethoxy-5-
fluoromethyl
ethyl




(hydroxycarbonyl)phenyl





2.2.989
3-(2,2,2-trifluoroethoxy)-5- 
fluoromethyl
ethyl




(hydroxycarbonyl)phenyl





2.2.990
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




(hydroxycarbonyl)phenyl





2.2.991
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




(hydroxycarbonyl)phenyl





2.2.992
3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




oxy]-5-(hydroxycarbonyl)-






phenyl





2.2.993
3-nitro-5-(hydroxy-
fluoromethyl
ethyl




carbonyl)phenyl





2.2.994
3-acetoxy-5-(hydroxy-
fluoromethyl
ethyl




carbonyl)phenyl





2.2.995
{3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




amino]-5-(hydroxy-






carbonyl)phenyl}





2.2.996
3-methylsulfanyl-5-
fluoromethyl
ethyl




(hydroxycarbonyl)phenyl





2.2.997
3,5-di(methoxy-
fluoromethyl
ethyl




carbonyl)phenyl





2.2.998
3-hydroxymethyl-5-
fluoromethyl
ethyl




(methoxycarbonyl)phenyl





2.2.999
3-carbamoyl-5-(methoxy
fluoromethyl
lethyl




carbonyl)phenyl





2.2.1000
3-hydroxy-5-(methoxy-
fluoromethyl
ethyl




carbonyl)phenyl





2.2.1001
3-methoxy-5-(methoxy-
fluoromethyl
ethyl




carbonyl)phenyl





2.2.1002
3-ethoxy-5-(methoxy-
fluoromethyl
ethyl




carbonyl)phenyl





2.2.1003
3-n-propoxy-5-(methoxy-
fluoromethyl
ethyl




carbonyl)phenyl





2.2.1004
3-n-butoxy-5-(methoxy-
fluoromethyl
ethyl




carbonyl)phenyl





2.2.1005
3-isobutoxy-5-(methoxy-
fluoromethyl
ethyl




carbonyl)phenyl





2.2.1006
3-tert-butoxy-5-(methoxy-
fluoromethyl
ethyl




carbonyl)phenyl





2.2.1007
3-difluoromethoxy-5-
fluoromethyl
ethyl




(methoxycarbonyl)phenyl





2.2.1008
3-trifluoromethoxy-5-
fluoromethyl
ethyl




(methoxycarbonyl)phenyl





2.2.1009
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl
ethyl




(methoxycarbonyl)phenyl





2.2.1010
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




(methoxycarbonyl)phenyl





2.2.1011
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




(methoxycarbonyl)-phenyl





2.2.1012
3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




oxy]-5-(methoxycarbonyl)-






phenyl





2.2.1013
3-nitro-5-(methoxy-
fluoromethyl
ethyl




carbonyl)phenyl





2.2.1014
3-acetoxy-5-(methoxy-
fluoromethyl
ethyl




carbonyl)phenyl





2.2.1015
{3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




amino]-5-(methoxy-






carbonyl)phenyl}





2.2.1016
3-methylsulfany1-5-
fluoromethyl
ethyl




(methoxycarbonyl)phenyl





2.2.1017
3,5-di(hydroxymethyl)-
fluoromethyl
ethyl




phenyl





2.2.1018
3-carbamoyl-5-hydroxy-
fluoromethyl
ethyl




methylphenyl





2.2.1019
3-hydroxy-5-hydroxy -
fluoromethyl
ethyl




methylphenyl





2.2.1020
3-methoxy-5-hydroxy-
fluoromethyl
ethyl




methylphenyl





2.2.1021
3-ethoxy-5-hydroxy-
fluoromethyl
ethyl




methylphenyl





2.2.1022
3-n-propoxy-5-hydroxy-
fluoromethyl
ethyl




methylphenyl





2.2.1023
3-n-butoxy-5- hydroxy -
fluoromethyl
ethyl




methylphenyl





2.2.1024
3-isobutoxy-5-hydroxy -
fluoromethyl
ethyl




methylphenyl





2.2.1025
3-tert-butoxy-5-hydroxy-
fluoromethyl
ethyl




methylphenyl





2.2.1026
3-difluoromethoxy-5-
fluoromethyl
ethyl




hydroxymethylphenyl





2.2.1027
3-trifluoromethoxy-5-
fluoromethyl
ethyl




hydroxymethylphenyl





2.2.1028
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl
ethyl




hydroxymethylphenyl





2.2.1029
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




hydroxymethylphenyl





2.2.1030
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




hydroxymethyl-phenyl





2.2.1031
3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




oxy]-5-hydroxymethyl-






phenyl





2.2.1032
3-nitro-5- hydroxymethyl-
fluoromethyl
ethyl




phenyl





2.2.1033
3-acetoxy-5- hydroxy -
fluoromethyl
ethyl




methylphenyl





2.2.1034
{3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




amino]-5-hydroxymethyl-






phenyl}





2.2.1035
3-methylsulfany1-5-
fluoromethyl
ethyl




hydroxymethylphenyl





2.2.1036
3,5-dicarbamoy1-5-
fluoromethyl
ethyl




carbamoylphenyl





2.2.1037
3-hydroxy-5-
fluoromethyl
ethyl




carbamoylphenyl





2.2.1038
3-methoxy-5-
fluoromethyl
ethyl




carbamoylphenyl





2.2.1039
3-ethoxy-5-
fluoromethyl
ethyl




carbamoylphenyl





2.2.1040
3-n-propoxy-5-
fluoromethyl
ethyl




carbamoylphenyl





2.2.1041
3-n-butoxy-5-
fluoromethyl
ethyl




carbamoylphenyl





2.2.1042
3-isobutoxy-5-
fluoromethyl
ethyl




carbamoylphenyl





2.2.1043
3-tert-butoxy-5-
fluoromethyl
ethyl




carbamoylphenyl





2.2.1044
3-difluoromethoxy-5-
fluoromethyl
ethyl




carbamoylphenyl





2.2.1045
3-trifluoromethoxy-5-
fluoromethyl
ethyl




carbamoylphenyl





2.2.1046
3-(2,2,2-trifluoroethoxy)-5- 
fluoromethyl
ethyl




carbamoylphenyl





2.2.1047
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




carbamoylphenyl





2.2.1048
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




carbamoylphenyl





2.2.1049
3-{(tert-butoxy-
fluoromethyl
ethyl




carbonyl)oxy]-5-






carbamoylphenyl





2.2.1050
3-nitro-5-carbamoylphenyl
fluoromethyl
ethyl



2.2.1051
3-acetoxy-5-
fluoromethyl
ethyl




carbamoylphenyl





2.2.1052
{3-[(tert-butoxy-
fluoromethyl
ethyl




carbonyl)amino]-5-






carbamoylphenyl}





2.2.1053
3-methylsulfanyl-5-
fluoromethyl
ethyl




carbamoylphenyl





2.2.1054
3,5-dihydroxyphenyl
fluoromethyl
ethyl



2.2.1055
3-methoxy-5-
fluoromethyl
ethyl




hydroxyphenyl





2.2.1056
3-ethoxy-5-hydroxyphenyl
fluoromethyl
ethyl



2.2.1057
3-n-propoxy-5-
fluoromethyl
ethyl




hydroxyphenyl





2.2.1058
3-n-butoxy-5-
fluoromethyl
ethyl




hydroxyphenyl





2.2.1059
3-isobutoxy-5-
fluoromethyl
ethyl




hydroxyphenyl





2.2.1060
3-tert-butoxy-5-
fluoromethyl
ethyl




hydroxyphenyl





2.2.1061
3-difluoromethoxy-5-
fluoromethyl
ethyl




hydroxyphenyl





2.2.1062
3-trifluoromethoxy-5-
fluoromethyl
ethyl




hydroxyphenyl





2.2.1063
3-(2,2,2-trifluoroethoxy)-5- 
fluoromethyl
ethyl




hydroxyphenyl





2.2.1064
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




hydroxyphenyl





2.2.1065
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




hydroxyphenyl





2.2.1066
3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




oxy]-5-hydroxyphenyl





2.2.1067
3-nitro-5-hydroxyphenyl
fluoromethyl
ethyl



2.2.1068
3-acetoxy-5-
fluoromethyl
ethyl




hydroxyphenyl





2.2.1069
{3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




amino]-5-hydroxyphenyl}





2.2.1070
3-methylsulfany1-5-
fluoromethyl
ethyl




hydroxyphenyl





2.2.1071
3,5-dimethoxyphenyl
fluoromethyl
ethyl



2.2.1072
3-ethoxy-5-
fluoromethyl
ethyl




methoxyphenyl





2.2.1073
3-n-propoxy-5-
fluoromethyl
ethyl




methoxyphenyl





2.2.1074
3-n-butoxy-5-
fluoromethyl
ethyl




methoxyphenyl





2.2.1075
3-isobutoxy-5-
fluoromethyl
ethyl




methoxyphenyl





2.2.1076
3-tert-butoxy-5-
fluoromethyl
ethyl




methoxyphenyl





2.2.1077
3-difluoromethoxy-5-
fluoromethyl
ethyl




methoxyphenyl





2.2.1078
3-trifluoromethoxy-5-
fluoromethyl
ethyl




methoxyphenyl





2.2.1079
3-(2,2,2-trifluoroethoxy)-5- 
fluoromethyl
ethyl




methoxyphenyl





2.2.1080
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




methoxyphenyl





2.2.1081
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




methoxyphenyl





2.2.1082
3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




oxy]-5-methoxyphenyl





2.2.1083
3-nitro-5-methoxyphenyl
fluoromethyl
ethyl



2.2.1084
3-acetoxy-5-
fluoromethyl
ethyl




methoxyphenyl





2.2.1085
{3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




amino]-5-methoxyphenyl}





2.2.1086
3-methylsulfanyl-5-
fluoromethyl
ethyl




methoxyphenyl





2.2.1087
3,5-diethoxyphenyl
fluoromethyl
ethyl



2.2.1088
3-n-propoxy-5-
fluoromethyl
ethyl




ethoxyphenyl





2.2.1089
3-n-butoxy-5-
fluoromethyl
ethyl




ethoxyphenyl





2.2.1090
3-isobutoxy-5-
fluoromethyl
ethyl




ethoxyphenyl





2.2.1091
3-tert-butoxy-5-
fluoromethyl
ethyl




ethoxyphenyl





2.2.1092
3-difluoromethoxy-5-
fluoromethyl
ethyl




ethoxyphenyl





2.2.1093
3-trifluoromethoxy-5-
fluoromethyl
ethyl




ethoxyphenyl





2.2.1094
3-(2,2,2-trifluoroethoxy)-5- 
fluoromethyl
ethyl




ethoxyphenyl





2.2.1095
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




ethoxyphenyl





2.2.1096
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




ethoxyphenyl





2.2.1097
3-[(tert-butoxy-
fluoromethyl
ethyl




carbonyl)oxy]-5-






ethoxyphenyl





2.2.1098
3-nitro-5-ethoxyphenyl
fluoromethyl
ethyl



2.2.1099
3-acetoxy-5-ethoxyphenyl
fluoromethyl
ethyl



2.2.1100
{3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




amino]-5-ethoxyphenyl}





2.2.1101
3-methylsulfany1-5-
fluoromethyl
ethyl




ethoxyphenyl





2.2.1102
3,5-dipropoxyphenyl
fluoromethyl
ethyl



2.2.1103
3-n-butoxy-5-
fluoromethyl
ethyl




propoxyphenyl





2.2.1104
3-isobutoxy-5-
fluoromethyl
ethyl




propoxyphenyl





2.2.1105
3-tert-butoxy-5-
fluoromethyl
ethyl




propoxyphenyl





2.2.1106
3-difluoromethoxy-5-
fluoromethyl
ethyl




propoxyphenyl





2.2.1107
3-trifluoromethoxy-5-
fluoromethyl
ethyl




propoxyphenyl





2.2.1108 
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl
ethyl




propoxyphenyl





2.2.1109
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




propoxyphenyl





2.2.1110
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




propoxyphenyl





2.2.1111
3-[(tert-butoxy-
fluoromethyl
ethyl




carbonyl)oxy]-5-






propoxyphenyl





2.2.1112
3-nitro-5-propoxyphenyl
fluoromethyl
ethyl



2.2.1113
3-acetoxy-5-propoxy-
fluoromethyl
ethyl




phenyl





2.2.1114
{3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




amino]-5-propoxyphenyl}





2.2.1115
3-methylsulfanyl-5-
fluoromethyl
ethyl




propoxyphenyl





2.2.1116
3,5-di(isopropoxy)phenyl
fluoromethyl
ethyl



2.2.1117
3-n-butoxy-5-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1118
3-isobutoxy-5-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1119
3-tert-butoxy-5-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1120
3-difluoromethoxy-5-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1121
3-trifluoromethoxy-5-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1122
3-(2,2,2-trifluoroethoxy)-5- 
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1123
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1124
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1125
3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




oxy]-5-isopropoxyphenyl





2.2.1126
3-nitro-5-isopropoxy-
fluoromethyl
ethyl




phenyl





2.2.1127
3-acetoxy-5-isopropoxy-
fluoromethyl
ethyl




phenyl





2.2.1128
{3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




amino]-5-isopropoxy-






phenyl}





2.2.1129
3-methylsulfanyl-5-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1130
3,5-di(tert-butoxy)phenyl
fluoromethyl
ethyl



2.2.1131
3-difluoromethoxy-5-tert-
fluoromethyl
ethyl




butoxyphenyl





2.2.1132
3-trifluoromethoxy-5-tert-
fluoromethyl
ethyl




butoxyphenyl





2.2.1133
3-(2,2,2-trifluoroethoxy)-5- 
fluoromethyl
ethyl




tert-butoxyphenyl





2.2.1134
3-(2-chloroethoxy)-5-tert-
fluoromethyl
ethyl




butoxylphenyl





2.2.1135
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




tert-butoxyphenyl





2.2.1136
3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




oxy]-5-tert-butoxyphenyl





2.2.1137
3-nitro-5-tert-
fluoromethyl
ethyl




butoxyphenyl





2.2.1138
3-acetoxy-5-tert-
fluoromethyl
ethyl




butoxyphenyl





2.2.1139
{3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




amino]-5-tert-butoxy-






phenyl}





2.2.1140
3-methylsulfanyl-5-tert-
fluoromethyl
ethyl




butoxyphenyl





2.2.1141
3,5-di(trifluoro-
fluoromethyl
ethyl




methoxy)phenyl





2.2.1142
3-(2,2,2-trifluoroethoxy)-5- 
fluoromethyl
ethyl




trifluoro-methoxyphenyl





2.2.1143
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




trifluoromethoxy-phenyl





2.2.1144
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




trifluoromethoxy-phenyl





2.2.1145
3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




oxy]-5-trifluoromethoxy-






phenyl





2.2.1146
3-nitro-5-trifluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1147
3-acetoxy-5-tert-
fluoromethyl
ethyl




butoxyphenyl





2.2.1148
{3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




amino]-5-trifluoromethoxy-






phenyl}





2.2.1149
3-methylsulfaonyl-5-
fluoromethyl
ethyl




trifluoromethoxy-phenyl





2.2.1150
3,5-bis(difluoro-
fluoromethyl
ethyl




methoxy)phenyl





2.2.1151
3,5-bis(difluoro-
chloromethyl
ethyl




methoxy)phenyl





2.2.1152
3,5-bis(difluoro-
bromomethyl
ethyl




methoxy)phenyl





2.2.1153
3,5-bis(difluoro-
fluoromethyl
ethyl




methoxy)phenyl





2.2.1154
3-trifluoromethoxy-5-
fluoromethyl
ethyl




difluoromethoxy-phenyl





2.2.1155
3-(2,2,2-trifluoroethoxy)-5-
fluoromethyl
ethyl




difluoro-methoxyphenyl





2.2.1156
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




difluoromethoxy-phenyl





2.2.1157
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




difluoromethoxy-phenyl





2.2.1158
3-[(tert-butoxycar bonyl)-
fluoromethyl
ethyl




oxy]-5-difluoromethoxy-






phenyl





2.2.1159
3-nitro-5-difluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1160
3-acetoxy-5-difluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1161
{3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




amino]-5-difluoromethoxy-






phenyl}





2.2.1162
3-methylsulfanyl-5-
fluoromethyl
ethyl




difluoromethoxy-phenyl





2.2.1163
3,5-bis(2,2,2-trifluoro-
fluoromethyl
ethyl




ethoxy)phenyl





2.2.1164
3-(2-chloroethoxy)-5-
fluoromethyl
ethyl




(2,2,2-trifluoroethoxy)-






phenyl





2.2.1165
3-(2-hydroxyethoxy)-5-
fluoromethyl
ethyl




(2,2,2-trifluoro-






ethoxy)phenyl





2.2.1166
3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




oxy]-5-(2,2,2-trifluoro-






ethoxy)phenyl





2.2.1167
3-nitro-5-(2,2,2-
fluoromethyl
ethyl




trifluoroethoxy)-phenyl





2.2.1168
3-acetoxy-5-(2,2,2-
fluoromethyl
ethyl




trifluoroethoxy)-phenyl





2.2.1169
{3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




amino]-5-(2,2,2-trifluoro-






ethoxy)-phenyl}





2.2.1170
3-methylsulfanyl-5-(2,2,2-
fluoromethyl
ethyl




trifluoroethoxy)-phenyl





2.2.1171
3,5-bis(2-chloro-
fluoromethyl
ethyl




ethoxy)phenyl





2.2.1172
3-(2-hydroxyethoxy)-5-(2-
fluoromethyl
ethyl




chloroethoxy)phenyl





2.2.1173
3-{(tert-butoxycarbonyl)-
fluoromethyl
ethyl




oxy]-5-(2-chloro-






ethoxy)phenyl





2.2.1174
3-nitro-5-(2-chloroethoxy)-
fluoromethyl
ethyl




phenyl





2.2.1175
3-acetoxy-5-(2-chloro-
fluoromethyl
ethyl




ethoxy)phenyl





2.2.1176
{3-[(tert-butoxy-carbonyl)-
fluoromethyl
ethyl




amino]-5-(2-chloro-






ethoxy)phenyl}





2.2.1177
3-methylsulfanyl-5-(2-
fluoromethyl
ethyl




chloroethoxy)-phenyl





2.2.1178
3,5-bis(2-hydroxy-
fluoromethyl
ethyl




ethoxy)phenyl





2.2.1179
3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




oxy]-5-(2-hydroxyethoxy)-






phenyl





2.2.1180
3-nitro-5-(2-hydroxy-
fluoromethyl
ethyl




ethoxy)phenyl





2.2.1181
3-acetoxy-5-(2-
fluoromethyl
ethyl




hydroxyethoxy)-phenyl





2.2.1182
3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




amino]-5-(2-hydroxy-






ethoxy)phenyl





2.2.1183
3-methylsulfanyl-5-(2-
fluoromethyl
ethyl




hydroxyethoxy)-phenyl





2.2.1184
3,5-bis[(tert-butoxy-
fluoromethyl
ethyl




carbonyl)oxy]phenyl





2.2.1185
3-nitro-5-[(tert-butoxy-
fluoromethyl
ethyl




carbonyl)oxy]phenyl





2.2.1186
3-acetoxy-5-[(tert-butoxy-
fluoromethyl
ethyl




carbonyl)oxy]phenyl





2.2.1187
{3-[(tert-butoxy-carbonyl)-
fluoromethyl
ethyl




amino]-5(tert-butoxy-






carbonyl)oxy]phenyl}





2.2.1188
3,5-bis(acetoxy)phenyl
fluoromethyl
ethyl



2.2.1189
{3-[(tert-butoxycarbonyl)-
fluoromethyl
ethyl




amino]-5-acetoxyphenyl}





2.2.1190
3-methylsulfaonyl-5-
fluoromethyl
ethyl




acetoxyphenyl





2.2.1191
3,5-dinitrophenyl
fluoromethyl
ethyl



2.2.1192
3-acetoxy-5-nitrophenyl
fluoromethyl
ethyl



2.2.1193
{3-[(tert-butoxy-carbonyl)-
fluoromethyl
ethyl




amino]-5-nitrophenyl}





2.2.1194
3-methylsulfanyl-5-
fluoromethyl
ethyl




nitrophenyl





2.2.1195
3,5-bis[(tert-butoxy-
fluoromethyl
ethyl




carbonyl)amino]phenyl





2.2.1196
3-methylsulfanyl-5-[(tert-
fluoromethyl
ethyl




butoxycarbonyl)-






amino]phenyl





2.2.1197
3,5-di(methylsulfanyl)-
fluoromethyl
ethyl




phenyl





2.2.1198
3,4-difluorophenyl
fluoromethyl
ethyl



2.2.1199
3,4-difluorophenyl
chloromethyl
ethyl



2.2.1200
3,4-difluorophenyl
bromomethyl
ethyl



2.2.1201
3,4-difluorophenyl
difluoromethyl
ethyl



2.2.1202
3,4-difluorophenyl
trifluoromethyl
ethyl



2.2.1203
3,4-difluorophenyl
cyano
ethyl



2.2.1204
3-chloro-4-fluorophenyl
fluoromethyl
ethyl



2.2.1205
3-chloro-4-fluorophenyl
chloromethyl
ethyl



2.2.1206
3-chloro-4-fluorophenyl
bromomethyl
ethyl



2.2.1207
3-chloro-4-fluorophenyl
difluoromethyl
ethyl



2.2.1208
3-chloro-4-fluorophenyl
trifluoromethyl
methyl
[CDCl3] 1.52 (s, 3H); 3.74






(d, 1H); 3.94 (s, 3H); 4.03






(d, 1H); 7.22 (m, 1H); 7.58






(m, 1H); 7.72 (m, 1H).


2.2.1209
3-chloro-4-fluorophenyl
cyano
ethyl



2.2.1210
3-bromo-4-fluorophenyl
fluoromethyl
ethyl



2.2.1211
3-methyl-4-fluorophenyl
fluoromethyl
ethyl



2.2.1212
3-methyl-4-fluorophenyl
chloromethyl
ethyl



2.2.1213
3-cyclopropyl-4-
fluoromethyl
ethyl




fluorophenyl





2.2.1214
3-cyano-4-fluorophenyl
fluoromethyl
ethyl



2.2.1215
3-methoxy-4-fluorophenyl
fluoromethyl
ethyl



2.2.1216
3-ethoxy-4-fluorophenyl
fluoromethyl
ethyl



2.2.1217
3-trifluoromethoxy-4-
fluoromethyl
ethyl




fluorophenyl





2.2.1218
3-nitro-4-fluorophenyl
fluoromethyl
ethyl



2.2.1219
3-fluoro-4-chlorophenyl
fluoromethyl
ethyl



2.2.1220
3,4-dichlorophenyl
fluoromethyl
ethyl



2.2.1221
3-bromo-4-chlorophenyl
fluoromethyl
ethyl



2.2.1222
3-methyl-4-chlorophenyl
fluoromethyl
ethyl



2.2.1223
3-cyclopropyl-4-
fluoromethyl
ethyl




chlorophenyl





2.2.1224
3-cyano-4-chlorophenyl
fluoromethyl
ethyl



2.2.1225
3-trifluoromethyl-4-
fluoromethyl
ethyl




chlorophenyl





2.2.1226
3-methoxy-4-chlorophenyl
fluoromethyl
ethyl



2.2.1227
3-ethoxy-4-chlorophenyl
fluoromethyl
ethyl



2.2.1228
3-trifluoromethoxy-4-
fluoromethyl
ethyl




chlorophenyl





2.2.1229
3-nitro-4-chlorophenyl
fluoromethyl
ethyl



2.2.1230
3-fluoro-4-bromophenyl
fluoromethyl
ethyl



2.2.1231
3-chloro-4-bromophenyl
fluoromethyl
ethyl



2.2.1232
3,4-dibromophenyl
fluoromethyl
ethyl



2.2.1233
3-methyl-4-bromophenyl
fluoromethyl
ethyl



2.2.1234
3-ethyl-4-bromophenyl
fluoromethyl
ethyl



2.2.1235
3-cyclopropy1-4-
fluoromethyl
ethyl




bromophenyl





2.2.1236 
3-cyano-4-bromophenyl
fluoromethyl
ethyl



2.2.1237
3-trifluoromethy1-4-
fluoromethyl
ethyl




bromophenyl





2.2.1238
3-methoxy-4-phenyl
fluoromethyl
ethyl



2.2.1239 
3-ethoxy-4-bromophenyl
fluoromethyl
ethyl



2.2.1240
3-trifluoromethoxy-4-
fluoromethyl
ethyl




bromophenyl





2.2.1241
3-nitro-4-bromophenyl
fluoromethyl
ethyl



2.2.1242
3-fluoro-4-iodophenyl
fluoromethyl
ethyl



2.2.1243
3-chloro-4-iodophenyl
fluoromethyl
ethyl



2.2.1244
3-bromo-4-iodophenyl
fluoromethyl
ethyl



2.2.1245
3-methyl-4-iodophenyl
fluoromethyl
ethyl



2.2.1246
3-cyclopropy1-4-
fluoromethyl
ethyl




iodophenyl





2.2.1247
3-cyano-4-iodophenyl
fluoromethyl
ethyl



2.2.1248
3-trifluoromethyl-4-
fluoromethyl
ethyl




iodophenyl





2.2.1249 
3-methoxy-4-iodophenyl
fluoromethyl
ethyl



2.2.1250
3-ethoxy-4-iodophenyl
fluoromethyl
ethyl



2.2.1251
3-trifluoromethoxy-4-
fluoromethyl
ethyl




iodophenyl





2.2.1252
3-nitro-4-iodophenyl
fluoromethyl
ethyl



2.2.1253
3-fluoro-4-methylphenyl
fluoromethyl
ethyl



2.2.1254
3-chloro-4-methylphenyl
fluoromethyl
ethyl



2.2.1255
3-bromo-4-methylphenyl
fluoromethyl
ethyl



2.2.1256
3,4-dimethylphenyl
fluoromethyl
ethyl



2.2.1257
3,4-dimethylphenyl
chloromethyl
ethyl



2.2.1258
3,4-dimethylphenyl
bromomethyl
ethyl



2.2.1259
3,4-dimethylphenyl
difluoromethyl 
ethyl



2.2.1260
3,4-dimethylphenyl
trifluoromethyl
ethyl



2.2.1261
3,4-dimethylphenyl
cyano
ethyl



2.2.1262
3-ethyl-4-methylphenyl
fluoromethyl
ethyl



2.2.1263
3-cyclopropy1-4-
fluoromethyl
ethyl




methylphenyl





2.2.1264 
3-cyano-4-methylphenyl 
fluoromethyl
ethyl



2.2.1265
3-trifluoromethy1-4-
fluoromethyl
ethyl




methylphenyl





2.2.1266
3-methoxy-4-
fluoromethyl
ethyl




methylphenyl





2.2.1267 
3-ethoxy-4-methylphenyl
fluoromethyl
ethyl



2.2.1268
3-trifluoromethoxy-4-
fluoromethyl
ethyl




methylphenyl





2.2.1269
3-nitro-4-methylphenyl
fluoromethyl
ethyl



2.2.1270
3-fluoro-4-ethylphenyl
fluoromethyl
ethyl



2.2.1271
3-chloro-4-ethylphenyl
fluoromethyl
ethyl



2.2.1272
3-bromo-4-ethylphenyl
fluoromethyl
ethyl



2.2.1273
3-methyl-4-ethylphenyl
fluoromethyl
ethyl



2.2.1274
3,4-diethylphenyl
fluoromethyl
ethyl



2.2.1275
3-cyclopropyl-4-
fluoromethyl
ethyl




ethylphenyl





2.2.1276
3-cyano-4-ethylphenyl
fluoromethyl
ethyl



2.2.1277
3-trifluoromethy1-4-
fluoromethyl
ethyl




ethylphenyl





2.2.1278
3-methoxy-4-ethylphenyl
fluoromethyl
ethyl



2.2.1279
3-ethoxy-4-ethylphenyl
fluoromethyl
ethyl



2.2.1280
3-trifluoromethoxy-4-
fluoromethyl
ethyl




ethylphenyl





2.2.1281
3-nitro-4-ethylphenyl
fluoromethyl
ethyl



2.2.1282
3-fluoro-4-propylphenyl
fluoromethyl
ethyl



2.2.1283
3-chloro-4-propylphenyl
fluoromethyl
ethyl



2.2.1284
3-bromo-4-propylphenyl
fluoromethyl
ethyl



2.2.1285
3-methyl-4-propylphenyl
fluoromethyl
ethyl



2.2.1286
3-cyclopropyl-4-
fluoromethyl
ethyl




propylphenyl





2.2.1287
3-cyano-4-propylphenyl
fluoromethyl
ethyl



2.2.1288
3-trifluoromethy1-4-
fluoromethyl
ethyl




propylphenyl





2.2.1289
3-methoxy-4-propylphenyl
fluoromethyl
ethyl



2.2.1290
3-ethoxy-4-propylphenyl
fluoromethyl
ethyl



2.2.1291
3-trifluoromethoxy-4-
fluoromethyl
ethyl




propylphenyl





2.2.1292
3-nitro-4-propylphenyl
fluoromethyl
ethyl



2.2.1293
3-fluoro-4-isopropylphenyl 
fluoromethyl
ethyl



2.2.1294
3-chloro-4-
fluoromethyl
ethyl




isopropylphenyl





2.2.1295
3-bromo-4-
fluoromethyl
ethyl




isopropylphenyl





2.2.1296
3-methyl-4-
fluoromethyl
ethyl




isopropylphenyl





2.2.1297
3-cyclopropy1-4-
fluoromethyl
ethyl




isopropylphenyl





2.2.1298
3-cyano-4-
fluoromethyl
ethyl




isopropylphenyl





2.2.1299
3-trifluoromethy1-4-
fluoromethyl
ethyl




isopropylphenyl





2.2.1300
3-methoxy-4-
fluoromethyl
ethyl




isopropylphenyl





2.2.1301
3-ethoxy-4-
fluoromethyl
ethyl




isopropylphenyl





2.2.1302
3-trifluoromethoxy-4-
fluoromethyl
ethyl




isopropylphenyl





2.2.1303 
3-nitro-4-isopropylphenyl
fluoromethyl
ethyl



2.2.1304 
3-fluoro-4-tert-butylphenyl
fluoromethyl
ethyl



2.2.1305 
3-chloro-4-tert-butylphenyl
fluoromethyl
ethyl



2.2.1306
3-bromo-4-tert-
fluoromethyl
ethyl




butylphenyl





2.2.1307
3-methyl-4-tert-
fluoromethyl
ethyl




butylphenyl





2.2.1308
3-ethyl-4-tert-butylphenyl
fluoromethyl
ethyl



2.2.1309
3-cyclopropyl-4-tert-
fluoromethyl
ethyl




butylphenyl





2.2.1310
3-cyano-4-tert-butylphenyl
fluoromethyl
ethyl



2.2.1311
3-trifluoromethyl-4-tert-
fluoromethyl
ethyl




butylphenyl





2.2.1312
3-trifluoromethyl-4-tert-
chloromethyl
ethyl




butylphenyl





2.2.1313
3-trifluoromethyl-4-tert-
bromomethyl
ethyl




butylphenyl





2.2.1314
3-trifluoromethyl-4-tert-
difluoromethyl
ethyl




butylphenyl





2.2.1315
3-methoxy-4-tert-
fluoromethyl
ethyl




butylphenyl





2.2.1316
3-ethoxy-4-tert-
fluoromethyl
ethyl




butylphenyl





2.2.1317
3-trifluoromethoxy-4-tert-
fluoromethyl
ethyl




butylphenyl





2.2.1318
3-nitro-4-tert-butylphenyl
fluoromethyl
ethyl



2.2.1319
3-fluoro-4-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.1320
3-chloro-4-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.1321
3-bromo-4-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.1322
3-methyl-4-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.1323
3-cyclopropyl-4-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.1324
3-cyano-4-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.1325
3-trifluoromethyl-4-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.1326
3-methoxy-4-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.1327
3-ethoxy-4-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.1328
3-trifluoromethoxy-4-
fluroomethyl
ethyl




cyclopropylphenyl





2.2.1329
3-fluoro-4-
fluoromethyl
ethyl




methoxycarbonylphenyl





2.2.1330
3-chloro-4-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.1331
3-bromo-4-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.1332
3-methyl-4-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.1333
3-ethyl-4-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.1334
3-cyclopropyl-4-
fluoromethyl
ethyl




methoxycarbonylphenyl





2.2.1335
3-cyano-4-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.1336
3-trifluoromethyl-4-
fluoromethyl
ethyl




methoxycarbonylphenyl





2.2.1337
3-methoxy-4-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.1338
3-ethoxy-4-
fluoromethyl
ethyl




methoxycarbonylphenyl





2.2.1339
3-trifluoromethoxy-4-
fluoromethyl
ethyl




methoxycarbonylphenyl





2.2.1340
3-nitro-4-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.1341
3-fluoro-4-cyanophenyl
fluoromethyl
ethyl



2.2.1342
3-chloro-4-cyanophenyl
fluoromethyl
ethyl



2.2.1343
3-bromo-4-cyanophenyl
fluoromethyl
ethyl



2.2.1344
3-methyl-4-cyanophenyl
fluoromethyl
ethyl



2.2.1345
3-cyclopropyl-4-
fluoromethyl
ethyl




cyanophenyl





2.2.1346
3,4-dicyanophenyl
fluoromethyl
ethyl



2.2.1347
3-trifluoromethyl-4-
fluoromethyl
ethyl




cyanophenyl





2.2.1348
3-trifluoromethyl-4-
chloromethyl
ethyl




cyanophenyl





2.2.1349
3-trifluoromethyl-4-
bromomethyl
ethyl




cyanophenyl





2.2.1350
3-trifluoromethyl-4-
difluoromethyl
ethyl




cyanophenyl





2.2.1351
3-methoxy-4-cyanophenyl
fluoromethyl
ethyl



2.2.1352
3-ethoxy-4-cyanophenyl
fluoromethyl
ethyl



2.2.1353
3-trifluoromethoxy-4-
fluoromethyl
ethyl




cyanophenyl





2.2.1354
3-nitro-4-cyanophenyl
fluoromethyl
ethyl



2.2.1355
3-fluoro-4-methoxyphenyl
fluoromethyl
ethyl



2.2.1356
3-chloro-4-methoxyphenyl
fluoromethyl
ethyl



2.2.1357
3-bromo-4-methoxyphenyl
fluoromethyl
ethyl



2.2.1358
3-methyl-4-
fluoromethyl
ethyl




methoxyphenyl





2.2.1359
3-cyclopropyl-4-
fluoromethyl
ethyl




methoxyphenyl





2.2.1360
3-cyano-4-methoxyphenyl
fluoromethyl
ethyl



2.2.1361
3-trifluoromethyl-4-
fluoromethyl
ethyl




methoxyphenyl





2.2.1362
3,4-dimethoxyphenyl
fluoromethyl
ethyl



2.2.1363
3-ethoxy-4-
fluoromethyl
ethyl




methoxyphenyl





2.2.1364
3-trifluoromethoxy-4-
fluoromethyl
ethyl




methoxyphenyl





2.2.1365
3-nitro-4-methoxyphenyl
fluoromethyl
ethyl



2.2.1366
3-fluoro-4-ethoxyphenyl
fluoormethyl
ethyl



2.2.1367
3-chloro-4-ethoxyphenyl
fluoromethyl
ethyl



2.2.1368
3-chloro-4-ethoxyphenyl
chloromethyl
ethyl



2.2.1369
3-chloro-4-ethoxyphenyl
bromomethyl
ethyl



2.2.1370
3-chloro-4-ethoxyphenyl
difluoromethyl 
ethyl



2.2.1371
3-bromo-4-ethoxyphenyl
fluoromethyl
ethyl



2.2.1372
3-methyl-4-ethoxyphenyl
fluoromethyl
ethyl



2.2.1373
3-cyclopropy1-4-
fluoromethyl
ethyl




ethoxyphenyl





2.2.1374 
3-cyano-4-ethoxyphenyl
fluoromethyl
ethyl



2.2.1375
3-trifluoromethy1-4-
fluoromethyl
ethyl




ethoxyphenyl





2.2.1376
3-methoxy-4-
fluoromethyl
ethyl




ethoxyphenyl





2.2.1377
2,4-diethoxyphenyl
fluoromethyl
ethyl



2.2.1378
3-trifluoromethoxy-4- 
fluoromethyl
ethyl




ethoxyphenyl





2.2.1379
3-nitro-4-ethoxyphenyl
fluoromethyl
ethyl



2.2.1380
3-fluoro-4-propoxyphenyl
fluoromethyl
ethyl



2.2.1381
3-chloro-4-propoxyphenyl
fluoromethyl
ethyl



2.2.1382
3-bromo-4-propoxyphenyl
fluoromethyl
ethyl



2.2.1383
3-methyl-4-propoxyphenyl
fluoromethyl
ethyl



2.2.1384
3-cyclopropy1-4-
fluoromethyl
ethyl




propoxyphenyl





2.2.1385
3-cyano-4-propoxyphenyl
fluoromethyl
ethyl



2.2.1386
3-trifluoromethy1-4-
fluoromethyl
ethyl




propoxyphenyl





2.2.1387
3-methoxy-4-
fluoromethyl
ethyl




propoxyphenyl





2.2.1388 
3-ethoxy-4-propoxyphenyl
fluoromethyl
ethyl



2.2.1389
3-trifluoromethoxy-4-
fluoromethyl
ethyl




propoxyphenyl





2.2.1390
3-nitro-4-propoxyphenyl
fluoromethyl
ethyl



2.2.1391
3-fluoro-4-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1392
3-chloro-4-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1393
3-bromo-4-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1394
3-methyl-4-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1395
3-cyclopropyl-4-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1396
3-cyano-4-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1397
3-trifluoromethy1-4-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1398
3-methoxy-4-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1399
3-ethoxy-4-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1400
3-trifluoromethoxy-4-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1401
3-nitro-4-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1402
3-fluoro-4-trifluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1403
3-chloro-4-trifluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1404
3-bromo-4-trifluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1405
3-methy1-4-trifluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1406
3-cyclopropy1-4-
fluoromethyl
ethyl




trifluoromethoxy-phenyl





2.2.1407
3-cyano-4-trifluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1408
3-trifluoromethy1-4-
fluoromethyl
ethyl




trifluoromethoxy-phenyl





2.2.1409
3-methoxy-4-
fluoromethyl
ethyl




trifluoromethoxy-phenyl





2.2.1410
3-ethoxy-4-trifluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1411
3,4-bis(trifluoro-
fluoromethyl
ethyl




methoxy)phenyl





2.2.1412
3-nitro-4-trifluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1413
3-fluoro-4-
fluoromethyl
ethyl




difluoromethoxy-phenyl





2.2.1414
3-chloro-4-
fluoromethyl
ethyl




difluoromethoxy-phenyl





2.2.1415
3-bromo-4-
fluoromethyl
ethyl




difluoromethoxy-phenyl





2.2.1416
3-methyl-4-
fluoromethyl
ethyl




difluoromethoxy-phenyl





2.2.1417
3-cyclopropyl-4-
fluoromethyl
ethyl




difluoromethoxy-phenyl





2.2.1418
3-cyano-4-
fluoromethyl
ethyl




difluoromethoxy-phenyl





2.2.1419
3-trifluoromethy1-4-
fluoromethyl
ethyl




difluoromethoxy-phenyl





2.2.1420
3-methoxy-4-
fluoromethyl
ethyl




difluoromethoxy-phenyl





2.2.1421
3-ethoxy-4-
fluoromethyl
ethyl




difluoromethoxy-phenyl





2.2.1422
3-trifluoromethoxy-4-
fluoromethyl
ethyl




difluoromethoxy-phenyl





2.2.1423 
3-nitro-4-difluoromethoxy-
fluoromethyl
ethyl




phenyl





2.2.1424
3-fluoro-4-nitrophenyl
fluoromethyl
ethyl



2.2.1425
3-chloro-4-nitrophenyl
fluoromethyl
ethyl



2.2.1426
3-bromo-4-nitrophenyl
fluoromethyl
ethyl



2.2.1427
3-methyl-4-nitrophenyl
fluoromethyl
ethyl



2.2.1428
3-cyclopropy1-4-
fluoromethyl
ethyl




nitrophenyl





2.2.1429
3-cyano-4-nitrophenyl
fluoromethyl
ethyl



2.2.1430
3-trifluoromethy1-4- 
fluoromethyl
ethyl




nitrophenyl





2.2.1431
3-methoxy-4-nitrophenyl
fluoromethyl
ethyl



2.2.1432
3-ethoxy-4-nitrophenyl
fluoromethyl
ethyl



2.2.1433
3-trifluoromethoxy-4-
fluoromethyl
ethyl




nitrophenyl





2.2.1434
3-fluoro-4-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.1435
3-chloro-4-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.1436
3-bromo-4-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.1437
3-methy1-4-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.1438
3-cyclopropyl-4-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.1439
3-cyano-4-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.1440
3-trifluoromethyl-4-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.1441
3-methoxy-4-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.1442
3-ethoxy-4-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.1443
3-trifluoromethoxy-4- 
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.1444
3-nitro-4-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.1445
3,6-difluorophenyl
fluoromethyl
ethyl



2.2.1446
3,6-difluorophenyl
chloromethyl
ethyl



2.2.1447
3,6-difluorophenyl
bromomethyl
ethyl



2.2.1448
3,6-difluorophenyl
difluoromethyl
ethyl



2.2.1449
3,6-difluorophenyl
trifluoromethyl 
ethyl



2.2.1450
3,6-difluorophenyl
cyano
ethyl



2.2.1451 
3-chloro-6-fluorophenyl
fluoromethyl
ethyl



2.2.1452 
3-bromo-6-fluorophenyl
fluoromethyl
ethyl



2.2.1453
3-methyl-6-fluorophenyl
fluoromethyl
ethyl



2.2.1454
3-ethyl-6-fluorophenyl
fluoromethyl
ethyl



2.2.1455
3-cyclopropy1-6-
fluoromethyl
ethyl




fluorophenyl





2.2.1456 
3-cyano-6-fluorophenyl
fluoromethyl
ethyl



2.2.1457
3-methoxy-6-fluorophenyl
fluoromethyl
ethyl



2.2.1458 
3-ethoxy-6-fluorophenyl
fluoromethyl
ethyl



2.2.1459
3-trifluoromethoxy-6- 
fluoromethyl
ethyl




fluorophenyl





2.2.1460
3-nitro-6-fluorophenyl
fluoromethyl
ethyl



2.2.1461
3-fluoro-6-chlorophenyl
fluoromethyl
ethyl



2.2.1462
3-fluoro-6-chlorophenyl
chloromethyl
ethyl



2.2.1463
3-fluoro-6-chlorophenyl
bromomethyl
ethyl



2.2.1464
3-fluoro-6-chlorophenyl
difluoromethyl
ethyl



2.2.1465
3,6-dichlorophenyl
fluoromethyl
ethyl



2.2.1466
3,6-dichlorophenyl
chloromethyl
ethyl



2.2.1467
3,6-dichlorophenyl
bromomethyl
ethyl



2.2.1468
3,6-dichlorophenyl
difluoromethyl
ethyl



2.2.1469
3,6-dichlorophenyl
trifluoromethyl
ethyl



2.2.1470
3,6-dichlorophenyl
cyano
ethyl



2.2.1471
3-bromo-6-chlorophenyl
fluoromethyl
ethyl



2.2.1472
3-methyl-6-chlorophenyl
fluoromethyl
ethyl



2.2.1473
3-cyclopropy1-6-
fluoromethyl
ethyl




chlorophenyl





2.2.1474
3-cyano-6-chlorophenyl
fluoromethyl
ethyl



2.2.1475
3-trifluoromethy1-6-
fluoromethyl
ethyl




chlorophenyl





2.2.1476
3-methoxy-6-chlorophenyl
fluoromethyl
ethyl



2.2.1477
3-ethoxy-6-chlorophenyl
fluoromethyl
ethyl



2.2.1478
3-trifluoromethoxy-6-
fluoromethyl
ethyl




chlorophenyl





2.2.1479
3-nitro-6-chlorophenyl
fluoromethyl
ethyl



2.2.1480
3-fluoro-6-bromophenyl
fluoromethyl
ethyl



2.2.1481
3-chloro-6-bromophenyl
fluoromethyl
ethyl



2.2.1482
3,6-dibromophenyl
fluoromethyl
ethyl



2.2.1483 
3-methyl-6-bromophenyl
fluoromethyl
ethyl



2.2.1484
3-cyclopropyl-6-
fluoromethyl
ethyl




bromophenyl





2.2.1485
3-cyano-6-bromophenyl
fluoromethyl
ethyl



2.2.1486
3-trifluoromethy1-6- 
fluoromethyl
ethyl




bromophenyl





2.2.1487
3-methoxy-6-phenyl
fluoromethyl
ethyl



2.2.1488 
3-ethoxy-6-bromophenyl
fluoromethyl
ethyl



2.2.1489
3-trifluoromethoxy-6- 
fluoromethyl
ethyl




bromophenyl





2.2.1490
3-nitro-6-bromophenyl
fluoromethyl
ethyl



2.2.1491
3-fluoro-6-iodophenyl
fluoromethyl
ethyl



2.2.1492
3-chloro-6-iodophenyl
fluoromethyl
ethyl



2.2.1493
3-bromo-6-iodophenyl
fluoromethyl
ethyl



2.2.1494
3-methyl-6-iodophenyl
fluoromethyl
ethyl



2.2.1495
3-cyclopropy1-6-
fluoromethyl
ethyl




iodophenyl





2.2.1496
3-cyano-6-iodophenyl
fluoromethyl
ethyl



2.2.1497
3-trifluoromethyl-6-
fluoromethyl
ethyl




iodophenyl





2.2.1498 
3-methoxy-6-iodophenyl
fluoromethyl
ethyl



2.2.1499 
3-ethoxy-6-iodophenyl
fluoromethyl
ethyl



2.2.1500
3-trifluoromethoxy-6-
fluoromethyl
ethyl




iodophenyl





2.2.1501
3-nitro-6-iodophenyl
fluoromethyl
ethyl



2.2.1502
3-fluoro-6-methylphenyl
fluoromethyl
ethyl



2.2.1503
3-chloro-6-methylphenyl
fluoromethyl
ethyl



2.2.1504
3-bromo-6-methylphenyl
fluoromethyl
ethyl



2.2.1505
3,6-dimethylphenyl
fluoromethyl
ethyl



2.2.1506
3-ethyl-6-methylphenyl
fluoromethyl
ethyl



2.2.1507
3-cyclopropy1-6-
fluoromethyl
ethyl




methylphenyl





2.2.1508
3-cyano-6-methylphenyl
fluoromethyl
ethyl



2.2.1509
3-trifluoromethy1-6-
fluoromethyl
ethyl




methylphenyl





2.2.1510
3-methoxy-6-
fluoromethyl
ethyl




methylphenyl





2.2.1511
3-ethoxy-6-methylphenyl
fluoromethyl
ethyl



2.2.1512
3-trifluoromethoxy-6-
fluoromethyl
ethyl




methylphenyl





2.2.1513
3-nitro-6-methylphenyl
fluoromethyl
ethyl



2.2.1514
3-fluoro-6-ethylphenyl
fluoromethyl
ethyl



2.2.1515
3-chloro-6-ethylphenyl
fluoromethyl
ethyl



2.2.1516
3-bromo-6-ethylphenyl
fluoromethyl
ethyl



2.2.1517
3-methyl-6-ethylphenyl
fluoromethyl
ethyl



2.2.1518
3,6-diethylphenyl
fluoromethyl
ethyl



2.2.1519
3-cyclopropyl-6-
fluoromethyl
ethyl




ethylphenyl





2.2.1520
3-cyano-6-ethylphenyl
fluoromethyl
ethyl



2.2.1521
3-trifluoromethyl-6-
fluoromethyl
ethyl




ethylphenyl





2.2.1522
3-methoxy-6-ethylphenyl
fluoromethyl
ethyl



2.2.1523
3-ethoxy-6-ethylphenyl
fluoromethyl
ethyl



2.2.1524
3-trifluoromethoxy-6-
fluoromethyl
ethyl




ethylphenyl





2.2.1525
3-nitro-6-ethylphenyl
fluoromethyl
ethyl



2.2.1526
3-fluoro-6-propylphenyl
fluoromethyl
ethyl



2.2.1527
3-chloro-6-propylphenyl
fluoromethyl
ethyl



2.2.1528
3-bromo-6-propylphenyl
fluoromethyl
ethyl



2.2.1529
3-methyl-6-propylphenyl
fluoromethyl
ethyl



2.2.1530
3-cyclopropyl-6-
fluoromethyl
ethyl




propylphenyl





2.2.1531
3-cyano-6-propylphenyl
fluoromethyl
ethyl



2.2.1532
3-trifluoromethyl-6-
fluoromethyl
ethyl




propylphenyl





2.2.1533
3-methoxy-6-propylphenyl
fluoromethyl
ethyl



2.2.1534
3-ethoxy-6-propylphenyl
fluoromethyl
ethyl



2.2.1535
3-trifluoromethoxy-6-
fluoromethyl
ethyl




propylphenyl





2.2.1536
3-nitro-6-propylphenyl
fluoromethyl
ethyl



2.2.1537
3-fluoro-6-isopropylphenyl
fluoromethyl
ethyl



2.2.1538
3-chloro-6-
fluoromethyl
ethyl




isopropylphenyl





2.2.1539
3-bromo-6-
fluoromethyl
ethyl




isopropylphenyl





2.2.1540
3-methyl-6-
lfuoromethyl
ethyl




isopropylphenyl





2.2.1541
3-cyclopropyl-6-
fluoromethyl
ethyl




isopropylphenyl





2.2.1542
3-cyano-6-
fluoromethyl
ethyl




isopropylphenyl





2.2.1543
3-trifluoromethyl-6-
fluoromethyl
ethyl




isopropylphenyl





2.2.1544
3-methoxy-6-
fluoromethyl
ethyl




isopropylphenyl





2.2.1545
3-ethoxy-6-
fluoromethyl
ethyl




isopropylphenyl





2.2.1546
3-trifluoromethoxy-6-
fluoromethyl
ethyl




isopropylphenyl





2.2.1547
3-nitro-6-isopropylphenyl
fluroomethyl
ethyl



2.2.1548
3-fluoro-6-tert-butylphenyl
fluoromethyl
ethyl



2.2.1549
3-chloro-6-tert-butylphenyl
fluoromethyl
ethyl



2.2.1550
3-bromo-6-tert-
fluoromethyl
ethyl




butylphenyl





2.2.1551
3-methyl-6-tert-
fluoromethyl
ethyl




butylphenyl





2.2.1552
3-cyclopropyl-6-tert-
fluoromethyl
ethyl




butylphenyl





2.2.1553
3-cyano-6-tert-butylphenyl
fluoromethyl
ethyl



2.2.1554
3-trifluoromethyl-6-tert-
fluoromethyl
ethyl




butylphenyl





2.2.1555
3-methoxy-6-tert-
fluoromethyl
ethyl




butylphenyl





2.2.1556
3-ethxoy-6-tert-
fluoromethyl
ethyl




butylphenyl





2.2.1557
3-trifluoromethoxy-6-tert-
fluoromethyl
ethyl




butylphenyl





2.2.1558
3-nitro-6-tert-butylphenyl
fluoromethyl
ethyl



2.2.1559
3-fluoro-6-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.1560
3-chloro-6-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.1561
3-bromo-6-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.1562
3-methyl-6-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.1563
3-cyclopropyl-6-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.1564
3-cyano-6-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.1565
3-trifluoromethyl-6-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.1566
3-methoxy-6-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.1567
3-ethoxy-6-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.1568
3-trifluoromethoxy-6-
fluoromethyl
ethyl




cyclopropylphenyl





2.2.1569
3-fluoro-6-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.1570
3-chloro-6-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.1571
3-bromo-6-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.1572
3-methyl-6-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.1573
3-cyclopropy1-6-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.1574
3-cyano-6-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.1575
3-trifluoromethy1-6-
fluoromethyl
ethyl




methoxycarbonylphenyl





2.2.1576
3-methoxy-6-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.1577
3-ethoxy-6-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.1578
3-trifluoromethoxy-6-
fluoromethyl
ethyl




methoxycarbonyl-phenyl





2.2.1579
3-nitro-6-methoxy-
fluoromethyl
ethyl




carbonylphenyl





2.2.1580
3-fluoro-6-cyanophenyl
fluoromethyl
ethyl



2.2.1581
3-chloro-6-cyanophenyl
fluoromethyl
ethyl



2.2.1582
3-bromo-6-cyanophenyl
fluoromethyl
ethyl



2.2.1583
3-methyl-6-cyanophenyl
fluoromethyl
ethyl



2.2.1584
3-cyclopropy1-6-
fluoromethyl
ethyl




cyanophenyl





2.2.1585
3-cyano-6-cyanophenyl
fluoromethyl
ethyl



2.2.1586
3-trifluoromethyl-6-
fluoromethyl
ethyl




cyanophenyl





2.2.1587
3-methoxy-6-cyanophenyl
fluoromethyl
ethyl



2.2.1588
3-ethoxy-6-cyanophenyl
fluoromethyl
ethyl



2.2.1589
3-trifluoromethoxy-6-
fluoromethyl
ethyl




cyanophenyl





2.2.1590
3-nitro-6-cyanophenyl
fluoromethyl
ethyl



2.2.1591
3-fluoro-6-methoxyphenyl
fluoromethyl
ethyl



2.2.1592
3-chloro-6-methoxyphenyl
fluoromethyl
ethyl



2.2.1593
3-bromo-6-methoxyphenyl
fluoromethyl
ethyl



2.2.1594
3-methyl-6-
fluoromethyl
ethyl




methoxyphenyl





2.2.1595
3-cyclopropy1-6-
fluoromethyl
ethyl




methoxyphenyl





2.2.1596
3-cyano-6-methoxyphenyl
fluoromethyl
ethyl



2.2.1597
3-trifluoromethyl-6-
fluoromethyl
ethyl




methoxyphenyl





2.2.1598
3,6-dimethoxyphenyl
fluoromethyl
ethyl



2.2.1599
3-ethoxy-6-
fluoromethyl
ethyl




methoxyphenyl





2.2.1600
3-trifluoromethoxy-6-
fluoromethyl
ethyl




methoxyphenyl





2.2.1601
3-nitro-6-methoxyphenyl
fluoromethyl
ethyl



2.2.1602
3-fluoro-6-ethoxyphenyl
fluoromethyl
ethyl



2.2.1603
3-chloro-6-ethoxyphenyl
fluoromethyl
ethyl



2.2.1604
3-bromo-6-ethoxyphenyl
fluoromethyl
ethyl



2.2.1605
3-methyl-6-ethoxyphenyl
fluoromethyl
ethyl



2.2.1606
3-cyclopropy1-6-
fluoromethyl
ethyl




ethoxyphenyl





2.2.1607
3-cyano-6-ethoxyphenyl
fluoromethyl
ethyl



2.2.1608
3-trifluoromethyl-6-
fluoromethyl
ethyl




ethoxyphenyl





2.2.1609
3-methoxy-6-
fluoromethyl
ethyl




ethoxyphenyl





2.2.1610
2,6-diethoxyphenyl
fluoromethyl
ethyl



2.2.1611
3-trifluoromethoxy-6-
fluoromethyl
ethyl




ethoxyphenyl





2.2.1612
3-nitro-6-ethoxyphenyl
fluoromethyl
ethyl



2.2.1613
3-fluoro-6-propoxyphenyl
fluoromethyl
ethyl



2.2.1614
3-chloro-6-propoxyphenyl
fluoromethyl
ethyl



2.2.1615
3-bromo-6-propoxyphenyl
fluoromethyl
ethyl



2.2.1616
3-methyl-6-propoxyphenyl
fluoromethyl
ethyl



2.2.1617
3-cyclopropyl-6-
fluoromethyl
ethyl




propoxyphenyl





2.2.1618
3-cyano-6-propoxyphenyl
fluoromethyl
ethyl



2.2.1619
3-trifluoromethyl-6-
fluoromethyl
ethyl




propoxyphenyl





2.2.1620
3-methoxy-6-
fluoromethyl
ethyl




propoxyphenyl





2.2.1621
3-ethoxy-6-propoxyphenyl
fluoromethyl
ethyl



2.2.1622
3-trifluoromethoxy-6-
fluoromethyl
ethyl




propoxyphenyl





2.2.1623
3-nitro-6-propoxyphenyl
fluoromethyl
ethyl



2.2.1624
3-fluoro-6-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1625
3-chloro-6-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1626
3-bromo-6-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1627
3-methyl-6-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1628
3-cyclopropyl-6-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1629
3-cyano-6-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1630
3-trifluoromethyl-6-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1631
3-methoxy-6-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1632
3-ethoxy-6-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1633
3-trifluoromethoxy-6-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1634
3-nitro-6-
fluoromethyl
ethyl




isopropoxyphenyl





2.2.1635
3-fluoro-6-trifluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1636
3-chloro-6-trifluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1637
3-bromo-6-trifluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1638
3-methy1-6-trifluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1639
3-cyclopropyl-6-trifluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1640
3-cyano-6-trifluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1641
3-trifluoromethyl-6-
fluoromethyl
ethyl




trifluoromethoxyphenyl





2.2.1642
3-methoxy-6-trifluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1643
3-ethoxy-6-trifluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1644
3,6-bis(trifluoro-
fluoromethyl
ethyl




methoxy)phenyl





2.2.1645 
3-nitro-6-trifluoromethoxy-
fluoromethyl
ethyl




phenyl





2.2.1646
3-fluoro-6-difluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1647
3-chloro-6-difluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1648
3-bromo-6-difluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1649
3-methy1-6-difluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1650
3-cyclopropyl-6-difluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1651
3-cyano-6-difluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1652
3-trifluoromethyl-6-
fluoromethyl
ethyl




difluoromethoxyphenyl





2.2.1653
3-methoxy-6-difluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1654
3-ethoxy-6-difluoro-
fluoromethyl
ethyl




methoxyphenyl





2.2.1655
3-trifluoromethoxy-6-
fluoromethyl
ethyl




difluoromethoxyphenyl





2.2.1656
3-nitro-6-difluoromethoxy-
fluoromethyl
ethyl




phenyl





2.2.1657
3-fluoro-6-nitrophenyl
fluoromethyl
ethyl



2.2.1658
3-chloro-6-nitrophenyl
fluoromethyl
ethyl



2.2.1659
3-bromo-6-nitrophenyl
fluoromethyl
ethyl



2.2.1660
3-methyl-6-nitrophenyl
fluoromethyl
ethyl



2.2.1661
3-cyclopropy1-6-
fluoromethyl
ethyl




nitrophenyl





2.2.1662
3-cyano-6-nitrophenyl
fluoromethyl
ethyl



2.2.1663
3-trifluoromethy1-6-
fluoromethyl
ethyl




nitrophenyl





2.2.1664
3-methoxy-6-nitrophenyl
fluoromethyl
ethyl



2.2.1665
3-ethoxy-6-nitrophenyl
fluoromethyl
ethyl



2.2.1666
3-trifluoromethoxy-6-
fluoromethyl
ethyl




nitrophenyl





2.2.1667
3-fluoro-6-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.1668
3-chloro-6-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.1669
3-bromo-6-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.1670
3-methyl-6-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.1671
3-cyclopropy1-6-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.1672
3-cyano-6-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.1673
3-trifluoromethy1-6-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.1674
3-methoxy-6-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.1675
3-ethoxy-6-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.1676
3-trifluoromethoxy-6-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.1677
3-nitro-6-
fluoromethyl
ethyl




methylsulfanylphenyl





2.2.1678
2,3,4-trifluorophenyl
fluoromethyl
ethyl



2.2.1679
2,3,4-trichlorophenyl
fluoromethyl
ethyl



2.2.1680
2,3,4-trimethylphenyl
fluoromethyl
ethyl



2.2.1681
2-fluoro-2-chloro-5-
fluoromethyl
ethyl




trifluoromethylphenyl





2.2.1682
2,3,5-trifluorophenyl
fluoromethyl
ethyl



2.2.1683
2,3,5-trichlorophenyl
fluoromethyl
ethyl



2.2.1684
2,3,5-trimethylphenyl
fluoromethyl
ethyl



2.2.1685
2,3-dichloro-5-
fluoromethyl
ethyl




methoxyphenyl





2.2.1686
2,3,6-trifluorophenyl
fluoromethyl
ethyl



2.2.1687
2,3,6-trichlorophenyl
fluoromethyl
ethyl



2.2.1688
2,3,6-trimethylphenyl
fluoromethyl
ethyl



2.2.1689
3,4,5-trifluorophenyl
fluoromethyl
ethyl



2.2.1690
3,4,5-trichlorophenyl
fluoromethyl
ethyl



2.2.1691
3,4,5-trimethylphenyl
fluoromethyl
ethyl



2.2.1692
3,5-dimethy1-4-
fluoromethyl
ethyl




fluorophenyl





2.2.1693
3,5-dichloro-4-
fluoromethyl
ethyl




methoxyphenyl





2.2.1694
3,5-difluoro-4-
fluoromethyl
ethyl




chlorophenyl





2.2.1695
3,5-dichloro-4-
fluoromethyl
ethyl




hydroxyphenyl





2.2.1696
3,5-trifluoromethy1-4- 
fluoromethyl
ethyl




chlorophenyl





2.2.1697
3,4,6-trifluorophenyl
fluoromethyl
ethyl



2.2.1698
3,4,6-trichlorophenyl
fluoromethyl
ethyl



2.2.1699
3,4,6-trimethylphenyl
fluoromethyl
ethyl



2.2.1700
pentafluorophenyl
fluoromethyl
ethyl
















TABLE 2.3







Inventive compounds of the general formula (I) in which W* is COOY, R1


R2 are each hydrogen, and aryl is the radical. 








 








 











No.
Aryl
R3
Y
Physical data





2.3.1
3-fluorophenyl
vinyl
methyl
[CDCl3] 3.37 (d, 1H);






3.84 (s, 3H); 3.96






(d, 1H); 5.37 (d,1H);






5.56 (d, 1H); 6.15






(dd, 1H); 7.13 (t, 1H);






7.37-7.42 (m, 3H).


2.3.2
3-fluorophenyl
1-methylvinyl
ethyl



2.3.3
3-fluorophenyl
allyl
ethyl



2.3.4
3-fluorophenyl
1-chlorovinyl
methyl
[CDCl3] 3.57 (d, 1H);






3.88 (s, 3H); 4.25






(d, 1H); 5.55 (s, 1H);






5.94 (s, 1H); 7.15






(t, 1H); 7.39-7.43






(m, 3H).


2.3.5
3-fluorophenyl
ethynyl
ethyl



2.3.6
3-chlorophenyl
vinyl
ethyl



2.3.7
3-chlorophenyl
1-methylvinyl
ethyl



2.3.8
3-chlorophenyl
allyl
ethyl



2.3.9
3-chlorophenyl
1-chlorovinyl
ethyl



2.3.10
3-chlorophenyl
ethynyl
ethyl



2.3.11
3-bromophenyl
vinyl
ethyl



2.3.12
3-bromophenyl
1-methylvinyl
ethyl



2.3.13
3-iodophenyl
vinyl
ethyl



2.3.14
3-iodophenyl
1-methylvinyl
ethyl



2.3.15
3-methylphenyl
vinyl
ethyl



2.3.16
3-methylphenyl
1-methylvinyl
ethyl



2.3.17
3-ethylphenyl
vinyl
ethyl



2.3.18
3-propylphenyl
vinyl
ethyl



2.3.19
3-isopropylphenyl
vinyl
ethyl



2.3.20
3-n-butylphenyl
vinyl
ethyl



2.3.21
3-i-butylphenyl
vinyl
ethyl



2.3.22
3-tert-butylphenyl
vinyl
ethyl



2.3.23
3-cyclopropylphenyl
vinyl
ethyl



2.3.24
3-cyclobutylphenyl
vinyl
ethyl



2.3.25
3-cyclopentylphenyl
vinyl
ethyl



2.3.26
3-vinylphenyl
vinyl
ethyl



2.3.27
3-ethynylphenyl
vinyl
ethyl



2.3.28
3-cyanophenyl
vinyl
ethyl



2.3.29
3-trifluoromethylphenyl
vinyl
ethyl



2.3.30
3-difluoromethylphenyl
vinyl
ethyl



2.3.31
3-(hydroxycarbonyl)-phenyl
vinyl
ethyl



2.3.32
3-(methoxycarbonyl)-phenyl
vinyl
ethyl



2.3.33
3-(ethoxycarbonyl)-phenyl
vinyl
ethyl



2.3.34
3-hydroxymethylphenyl
vinyl
ethyl



2.3.35
3-carbamoylphenyl
vinyl
ethyl



2.3.36
3-hydroxyphenyl
vinyl
ethyl



2.3.37
3-methoxyphenyl
vinyl
ethyl



2.3.38
3-ethoxyphenyl
vinyl
ethyl



2.3.39
3-propyloxyphenyl
vinyl
ethyl



2.3.40
3-isopropyloxyphenyl
vinyl
ethyl



2.3.41
3-n-butyloxyphenyl
vinyl
ethyl



2.3.42
3-i-butyloxyphenyl
vinyl
ethyl



2.3.43
3-t-butyloxyphenyl
vinyl
ethyl



2.3.44
3-difluoromethoxy-phenyl
vinyl
ethyl



2.3.45
3-trifluoromethoxy-phenyl
vinyl
ethyl



2.3.46
3-(2,2,2-trifluoroethoxy)-phenyl
vinyl
ethyl



2.3.47
3-(2-chloroethoxy)-phenyl
vinyl
ethyl



2.3.48
3-(2-hydroxyethoxy)-phenyl
vinyl
ethyl



2.3.49
3-(2-methoxyethoxy)-phenyl
vinyl
ethyl



2.3.50
3-[(tert-butoxy-
vinyl
ethyl




carbonyl)oxy]phenyl





2.3.51
3-nitrophenyl
vinyl
ethyl



2.3.52
3-acetoxyphenyl
vinyl
ethyl



2.3.53
{3-[(tert-
vinyl
ethyl




butoxycarbonyl)amino]phenyl}





2.3.54
3-methylsulfanylphenyl
vinyl
ethyl



2.3.55
3-ethylsulfanylphenyl
vinyl
ethyl



2.3.56
3-(pentafluoro-lambda6-
vinyl
ethyl




sulfanyl)phenyl





2.3.57
2,3-difluorophenyl
vinyl
ethyl



2.3.58
2,3-difluorophenyl
1-methylvinyl 
ethyl



2.3.59
2,3-difluorophenyl
allyl
ethyl



2.3.60
2,3-difluorophenyl
1-chlorovinyl
ethyl



2.3.61
2,3-difluorophenyl
ethynyl
ethyl



2.3.62
2-chloro-3-fluorophenyl
vinyl
ethyl



2.3.63
2-bromo-3-fluorophenyl
vinyl
ethyl



2.3.64
2-methyl-3-fluorophenyl
vinyl
ethyl



2.3.65
2-ethyl-3-fluorophenyl
vinyl
ethyl



2.3.66
2-cyclopropyl-3-fluorophenyl
vinyl
ethyl



2.3.67
2-vinyl-3-fluorophenyl
vinyl
ethyl



2.3.68
2-ethynyl-3-fluorophenyl
vinyl
ethyl



2.3.69
2-cyano-3-fluorophenyl
vinyl
ethyl



2.3.70
2-methoxy-3-fluorophenyl
vinyl
ethyl



2.3.71
2-ethoxy-3-fluorophenyl
vinyl
ethyl



2.3.72
2-trifluoromethoxy-3-
vinyl
ethyl




fluorophenyl





2.3.73
2-nitro-3-fluorophenyl
vinyl
ethyl



2.3.74
2-fluoro-3-chlorophenyl
vinyl
ethyl



2.3.75
2,3-dichlorophenyl
vinyl
ethyl



2.3.76
2,3-dichlorophenyl
1-methylvinyl
ethyl



2.3.77
2,3-dichlorophenyl
allyl
ethyl



2.3.78
2,3-dichlorophenyl
1-chlorovinyl
ethyl



2.3.79
2,3-dichlorophenyl
ethynyl
ethyl



2.3.80
2-bromo-3-chlorophenyl
vinyl
ethyl



2.3.81
2-methyl-3-chlorophenyl
vinyl
ethyl



2.3.82
2-ethyl-3-chlorophenyl
vinyl
ethyl



2.3.83
2-cyclopropyl-3-chlorophenyl
vinyl
ethyl



2.3.84
2-vinyl-3-chlorophenyl
vinyl
ethyl



2.3.85
2-ethynyl-3-chlorophenyl
vinyl
ethyl



2.3.86
2-cyano-3-chlorophenyl
vinyl
ethyl



2.3.87
2-trifluoromethyl-2-chlorophenyl
vinyl
ethyl



2.3.88
2-methoxy-3-chlorophenyl
vinyl
ethyl



2.3.89
2-ethoxy-3-chlorophenyl
vinyl
ethyl



2.3.90
2-trifluoromethoxy-3-
vinyl
ethyl




chlorophenyl





2.3.91
2-nitro-3-chlorophenyl
vinyl
ethyl



2.3.92
2-fluoro-3-bromophenyl
vinyl
ethyl



2.3.93
2-chloro-3-bromophenyl
vinyl
ethyl



2.3.94
2,3-dibromophenyl
vinyl
ethyl



2.3.95
2-methyl-3-bromophenyl
vinyl
ethyl



2.3.96
2-ethyl-3-bromophenyl
vinyl
ethyl



2.3.97
2-cyclopropyl-3-bromophenyl
vinyl
ethyl



2.3.98
2-vinyl-3-bromophenyl
vinyl
ethyl



2.3.99
2-ethynyl-3-bromophenyl
vinyl
ethyl



2.3.100
2-cyano-3-bromophenyl
vinyl
ethyl



2.3.101
2-trifluoromethyl-3-bromophenyl 
vinyl
ethyl



2.3.102
2-methoxy-3-phenyl
vinyl
ethyl



2.3.103
2-ethoxy-3-bromophenyl
vinyl
ethyl



2.3.104
2-trifluoromethoxy-3-
vinyl
ethyl




bromophenyl





2.3.105
2-nitro-3-bromophenyl
vinyl
ethyl



2.3.106
2-fluoro-3-iodophenyl
vinyl
ethyl



2.3.107
2-chloro-3-iodophenyl
vinyl
ethyl



2.3.108
2-bromo-3-iodophenyl
vinyl
ethyl



2.3.109
2-methyl-3-iodophenyl
vinyl
ethyl



2.3.110
2-ethyl-3-iodophenyl
vinyl
ethyl



2.3.111
2-cyclopropyl-3-iodophenyl
vinyl
ethyl



2.3.112
2-vinyl-3-iodophenyl
vinyl
ethyl



2.3.113
2-ethynyl-3-iodophenyl
vinyl
ethyl



2.3.114
2-cyano-3-iodophenyl
vinyl
ethyl



2.3.115
2-trifluoromethyl-3-iodophenyl 
vinyl
ethyl



2.3.116
2-methoxy-3-iodophenyl
vinyl
ethyl



2.3.117
2-ethoxy-3-iodophenyl
vinyl
ethyl



2.3.118
2-trifluoromethoxy-3-iodophenyl 
vinyl
ethyl



2.3.119
2-nitro-3-iodophenyl
vinyl
ethyl



2.3.120
2-fluoro-3-methylphenyl
vinyl
ethyl



2.3.121
2-fluoro-3-methylphenyl
1-methylvinyl
ethyl



2.3.122
2-fluoro-3-methylphenyl
allyl
ethyl



2.3.123
2-fluoro-3-methylphenyl
1-chlorovinyl
ethyl



2.3.124
2-fluoro-3-methylphenyl
ethynyl
ethyl



2.3.125
2-chloro-3-methylphenyl
vinyl
ethyl



2.3.126
2-chloro-3-methylphenyl
1-methylvinyl
ethyl



2.3.127
2-chloro-3-methylphenyl
allyl
ethyl



2.3.128
2-chloro-3-methylphenyl
1-chlorovinyl
ethyl



2.3.129
2-chloro-3-methylphenyl
ethynyl
ethyl



2.3.130
2-bromo-3-methylphenyl
vinyl
ethyl



2.3.131
2,3-dimethylphenyl
vinyl
ethyl



2.3.132
2,3-dimethylphenyl
1-methylvinyl
ethyl



2.3.133
2,3-dimethylphenyl
allyl
ethyl



2.3.134
2,3-dimethylphenyl
1-chlorovinyl 
ethyl



2.3.135
2,3-dimethylphenyl
ethynyl
ethyl



2.3.136
2-ethyl-3-methylphenyl
vinyl
ethyl



2.3.137
2-cyclopropyl-3-methylphenyl
vinyl
ethyl



2.3.138
2-vinyl-3-methylphenyl
vinyl
ethyl



2.3.139
2-ethynyl-3-methylphenyl
vinyl
ethyl



2.3.140
2-cyano-3-methylphenyl
vinyl
ethyl



2.3.141
2-trifluoromethyl-3-methylphenyl
vinyl
ethyl



2.3.142
2-methoxy-3-
vinyl
ethyl




methylphenyl





2.3.143
2-ethoxy-3-methylphenyl
vinyl
ethyl



2.3.144
2-trifluoromethoxy-3-
vinyl
ethyl




methylphenyl





2.3.145
2-nitro-3-methylphenyl
vinyl
ethyl



2.3.146
2-fluoro-3-ethylphenyl
vinyl
ethyl



2.3.147
2-chloro-3-ethylphenyl
vinyl
ethyl



2.3.148
2-bromo-3-ethylphenyl
vinyl
ethyl



2.3.149
2-methyl-3-ethylphenyl
vinyl
ethyl



2.3.150
2,3-diethylphenyl
vinyl
ethyl



2.3.151
2-cyclopropyl-3-ethylphenyl
vinyl
ethyl



2.3.152
2-vinyl-3-ethylphenyl
vinyl
ethyl



2.3.153
2-ethynyl-3-ethylphenyl
vinyl
ethyl



2.3.154
2-cyano-3-ethylphenyl
vinyl
ethyl



2.3.155
2-trifluoromethyl-3-ethylphenyl
vinyl
ethyl



2.3.156
2-methoxy-3-ethylphenyl
vinyl
ethyl



2.3.157
2-ethoxy-3-ethylphenyl
vinyl
ethyl



2.3.158
2-trifluoromethoxy-3-ethylphenyl
vinyl
ethyl



2.3.159
2-nitro-3-ethylphenyl
vinyl
ethyl



2.3.160
2-fluoro-3-propylphenyl
vinyl
ethyl



2.3.161
2-chloro-3-propylphenyl
vinyl
ethyl



2.3.162
2-bromo-3-propylphenyl
vinyl
ethyl



2.3.163
2-methyl-3-propylphenyl
vinyl
ethyl



2.3.164
2-methyl-3-propylphenyl
vinyl
ethyl



2.3.165
2-cyclopropyl-3-propylphenyl
vinyl
ethyl



2.3.166
2-vinyl-3-propylphenyl
vinyl
ethyl



2.3.167
2-ethynyl-3-propylphenyl
vinyl
ethyl



2.3.168
2-cyano-3-propylphenyl
vinyl
ethyl



2.3.169
2-trifluoromethyl-3-propylphenyl
vinyl
ethyl



2.3.170
2-methoxy-3-propylphenyl
vinyl
ethyl



2.3.171
2-ethoxy-3-propylphenyl
vinyl
ethyl



2.3.172
2-trifluoromethoxy-3-
vinyl
ethyl




propylphenyl





2.3.173
2-nitro-3-propylphenyl
vinyl
ethyl



2.3.174
2-fluoro-3-isopropylphenyl
vinyl
ethyl



2.3.175
2-chloro-3-isopropylphenyl
vinyl
ethyl



2.3.176
2-bromo-3-isopropylphenyl
vinyl
ethyl



2.3.177
2-methyl-3-isopropylphenyl
vinyl
ethyl



2.3.178
2-ethyl-3-isopropylphenyl
vinyl
ethyl



2.3.179
2-cyclopropyl-3-isopropylphenyl
vinyl
ethyl



2.3.180
2-vinyl-3-isopropylphenyl
vinyl
ethyl



2.3.181
2-ethynyl-3-isopropylphenyl
vinyl
ethyl



2.3.182
2-cyano-3-isopropylphenyl
vinyl
ethyl



2.3.183
2-trifluoromethyl-3-
vinyl
ethyl




isopropylphenyl





2.3.184
2-methoxy-3-isopropylphenyl
vinyl
ethyl



2.3.185
2-ethoxy-3-isopropylphenyl
vinyl
ethyl



2.3.186
2-trifluoromethoxy-3-
vinyl
ethyl




isopropylphenyl





2.3.187
2-nitro-3-isopropylphenyl
vinyl
ethyl



2.3.188
2-fluoro-3-tert-butylphenyl
vinyl
ethyl



2.3.189
2-chloro-3-tert-butylphenyl
vinyl
ethyl



2.3.190
2-bromo-3-tert-butylphenyl
vinyl
ethyl



2.3.191
2-methyl-3-tert-butylphenyl
vinyl
ethyl



2.3.192
2-ethyl-3-tert-butylphenyl
vinyl
ethyl



2.3.193
2-cyclopropyl-3-tert-butylphenyl
vinyl
ethyl



2.3.194
2-vinyl-3-tert-butylphenyl
vinyl
ethyl



2.3.195
2-ethynyl-3-tert-butylphenyl
vinyl
ethyl



2.3.196
2-cyano-3-tert-butylphenyl
vinyl
ethyl



2.3.197
2-trifluoromethyl-3-tert-
vinyl
ethyl




butylphenyl





2.3.198
2-methoxy-3-tert-butylphenyl
vinyl
ethyl



2.3.199
2-ethoxy-3-tert-butylphenyl
vinyl
ethyl



2.3.200
2-trifluoromethoxy-3-tert-
vinyl
ethyl




butylphenyl





2.3.201
2-nitro-3-tert-butylphenyl
vinyl
ethyl



2.3.202
2-fluoro-3-hydroxymethylphenyl
vinyl
ethyl



2.3.203
2-chloro-3-hydroxymethylphenyl
vinyl
ethyl



2.3.204 
2-bromo-3-hydroxymethylphenyl
vinyl
ethyl



2.3.205 
2-methyl-3-hydroxymethylphenyl
vinyl
ethyl



2.3.206 
2-ethyl-3-hydroxymethylphenyl
vinyl
ethyl



2.3.207
2-cyclopropyl-3-
vinyl
ethyl




hydroxymethylphenyl





2.3.208
2-vinyl-3-hydroxymethylphenyl
vinyl
ethyl



2.3.209
2-ethynyl-3-
vinyl
ethyl




hydroxymethylphenyl





2.3.210
2-cyano-3-hydroxymethylphenyl
vinyl
ethyl



2.3.211
2-trifluoromethyl-3-
vinyl
ethyl




hydroxymethylphenyl





2.3.212
2-methoxy-3-
vinyl
ethyl




hydroxymethylphenyl





2.3.213
2-ethoxy-3-hydroxymethylphenyl
vinyl
ethyl



2.3.214
2-trifluoromethoxy-3-
vinyl
ethyl




hydroxymethylphenyl





2.3.215
2-nitro-3-hydroxymethylphenyl
vinyl
ethyl



2.3.216
2-fluoro-3-cyclopropylphenyl
vinyl
ethyl



2.3.217
2-chloro-3-cyclopropylphenyl
vinyl
ethyl



2.3.218
2-bromo-3-cyclopropylphenyl
vinyl
ethyl



2.3.219
2-methyl-3-cyclopropylphenyl
vinyl
ethyl



2.3.220
2-ethyl-3-cyclopropylphenyl
vinyl
ethyl



2.3.221
2-cyclopropyl-3-
vinyl
ethyl




cyclopropylphenyl





2.3.222
2-vinyl-3-cyclopropylphenyl
vinyl
ethyl



2.3.223
2-ethynyl-3-cyclopropylphenyl
vinyl
ethyl



2.3.224
2-cyano-3-cyclopropylphenyl
vinyl
ethyl



2.3.225
2-trifluoromethyl-3-
vinyl
ethyl




cyclopropylphenyl





2.3.226
2-methoxy-3-cyclopropylphenyl
vinyl
ethyl



2.3.227
2-ethoxy-3-cyclopropylphenyl
vinyl
ethyl



2.3.228
2-trifluoromethoxy-3-
vinyl
ethyl




cyclopropylphenyl





2.3.229
2-fluoro-3-
vinyl
ethyl




methoxycarbonylphenyl





2.3.230
2-chloro-3-
vinyl
ethyl




methoxycarbonylphenyl





2.3.231
2-bromo-3-
vinyl
ethyl




methoxycarbonylphenyl





2.3.232
2-methyl-3-
vinyl
ethyl




methoxycarbonylphenyl





2.3.233
2-ethyl-3-
vinyl
ethyl




methoxycarbonylphenyl





2.3.234
2-cyclopropyl-3-
vinyl
ethyl




methoxycarbonyl-phenyl





2.3.235
2-vinyl-3-
vinyl
ethyl




methoxycarbonylphenyl





2.3.236
2-ethynyl-3-methoxycarbonyl-
vinyl
ethyl




phenyl





2.3.237
2-cyano-3-
vinyl
ethyl




methoxycarbonylphenyl





2.3.238
2-trifluoromethyl-3-
vinyl
ethyl




methoxycarbonylphenyl





2.3.239
2-methoxy-3-methoxycarbonyl-
vinyl
ethyl




phenyl





2.3.240
2-ethoxy-3-
vinyl
ethyl




methoxycarbonylphenyl





2.3.241
2-trifluoromethoxy-3-
vinyl
ethyl




methoxycarbonylphenyl





2.3.242
2-nitro-3-
vinyl
ethyl




methoxycarbonylphenyl





2.3.243
2-fluoro-3-vinylphenyl
vinyl
ethyl



2.3.244
2-chloro-3-vinylphenyl
vinyl
ethyl



2.3.245
2-bromo-3-vinylphenyl
vinyl
ethyl



2.3.246
2-methyl-3-vinylphenyl
vinyl
ethyl



2.3.247
2-ethyl-3-vinylphenyl
vinyl
ethyl



2.3.248
2-cyclopropyl-3-vinylphenyl
vinyl
ethyl



2.3.249
2-vinyl-3-vinylphenyl
vinyl
ethyl



2.3.250
2-ethynyl-3-vinylphenyl
vinyl
ethyl



2.3.251
2-cyano-3-vinylphenyl
vinyl
ethyl



2.3.252
2-trifluoromethyl-3-vinylphenyl
vinyl
ethyl



2.3.253
2-methoxy-3-vinylphenyl
vinyl
ethyl



2.3.254
2-ethoxy-3-vinylphenyl
vinyl
ethyl



2.3.255
2-trifluoromethoxy-3-vinylphenyl
vinyl
ethyl



2.3.256
2-nitro-3-vinylphenyl
vinyl
ethyl



2.3.257
2-fluoro-3-ethynylphenyl
vinyl
ethyl



2.3.258
2-chloro-3-ethynylphenyl
vinyl
ethyl



2.3.259
2-bromo-3-ethynylphenyl
vinyl
ethyl



2.3.260
2-methyl-3-ethynylphenyl
vinyl
ethyl



2.3.261
2-ethyl-3-ethynylphenyl
vinyl
ethyl



2.3.262
2-cyclopropyl-3-ethynylphenyl
vinyl
ethyl



2.3.263
2-vinyl-3-ethynylphenyl
vinyl
ethyl



2.3.264
2-cyano-3-ethynylphenyl
vinyl
ethyl



2.3.265
2-trifluoromethyl-3-ethynylphenyl
vinyl
ethyl



2.3.266
2-methoxy-3-ethynylphenyl
vinyl
ethyl



2.3.267
2-ethoxy-3-ethynylphenyl
vinyl
ethyl



2.3.268
2-trifluoromethoxy-3-
vinyl
ethyl




ethynylphenyl





2.3.269
2-nitro-3-ethynylphenyl
vinyl
ethyl



2.3.270
2-fluoro-3-ethynylphenyl
vinyl
ethyl



2.3.271
2-fluoro-3-cyanophenyl
vinyl
ethyl



2.3.272
2-chloro-3-cyanophenyl
vinyl
ethyl



2.3.273
2-bromo-3-cyanophenyl
vinyl
ethyl



2.3.274
2-methyl-3-cyanophenyl
vinyl
ethyl



2.3.275
2-ethyl-3-cyanophenyl
vinyl
ethyl



2.3.276
2-ethyl-3-cyanophenyl
1-methylvinyl
ethyl



2.3.277
2-ethyl-3-cyanophenyl
allyl
ethyl



2.3.278
2-ethyl-3-cyanophenyl
1-chlorovinyl 
ethyl



2.3.279
2-ethyl-3-cyanophenyl
ethynyl
ethyl



2.3.280
2-cyclopropyl-3-cyanophenyl
vinyl
ethyl



2.3.281
2-vinyl-3-cyanophenyl
vinyl
ethyl



2.3.282
2-ethynyl-3-cyanophenyl
vinyl
ethyl



2.3.283
2-cyano-3-cyanophenyl
vinyl
ethyl



2.3.284
2-trifluoromethyl-3-cyanophenyl
vinyl
ethyl



2.3.285
2-methoxy-3-cyanophenyl
vinyl
ethyl



2.3.286
2-ethoxy-3-cyanophenyl
vinyl
ethyl



2.3.287
2-trifluoromethoxy-3-
vinyl
ethyl




cyanophenyl





2.3.288
2-nitro-3-cyanophenyl
vinyl
ethyl



2.3.289
2-fluoro-3-hydroxyphenyl
vinyl
ethyl



2.3.290
2-chloro-3-hydroxyphenyl
vinyl
ethyl



2.3.291
2-bromo-3-hydroxyphenyl
vinyl
ethyl



2.3.292
2-methyl-3-hydroxyphenyl
vinyl
ethyl



2.3.293
2-ethyl-3-hydroxyphenyl
vinyl
ethyl



2.3.294
2-cyclopropyl-3-hydroxyphenyl
vinyl
ethyl



2.3.295
2-vinyl-3-hydroxyphenyl
vinyl
ethyl



2.3.296
2-ethynyl-3-hydroxyphenyl
vinyl
ethyl



2.3.297
2-cyano-3-hydroxyphenyl
vinyl
ethyl



2.3.298
2-trifluoromethyl-3-
vinyl
ethyl




hydroxyphenyl





2.3.299
2-methoxy-3-hydroxyphenyl
vinyl
ethyl



2.3.300
2-ethoxy-3-hydroxyphenyl
vinyl
ethyl



2.3.301
2-trifluoromethoxy-3-
vinyl
ethyl




hydroxyphenyl





2.3.302
2-nitro-3-hydroxyphenyl
vinyl
ethyl



2.3.303
2-fluoro-3-methoxyphenyl
vinyl
ethyl



2.3.304
2-chloro-3-methoxyphenyl
vinyl
ethyl



2.3.305
2-bromo-3-methoxyphenyl
vinyl
ethyl



2.3.306
2-methyl-3-methoxyphenyl
vinyl
ethyl



2.3.307
2-ethyl-3-methoxyphenyl
vinyl
ethyl



2.3.308
2-cyclopropyl-3-methoxyphenyl
vinyl
ethyl



2.3.309
2-vinyl-3-methoxyphenyl
vinyl
ethyl



2.3.310
2-ethynyl-3-methoxyphenyl
vinyl
ethyl



2.3.311
2-cyano-3-methoxyphenyl
vinyl
ethyl



2.3.312
2-trifluoromethyl-3-
vinyl
ethyl




methoxyphenyl





2.3.313
2,3-dimethoxyphenyl
vinyl
ethyl



2.3.314
2-ethoxy-3-methoxyphenyl
vinyl
ethyl



2.3.315
2-trifluoromethoxy-3-
vinyl
ethyl




methoxyphenyl





2.3.316
2-nitro-3-methoxyphenyl
vinyl
ethyl



2.3.317
2-fluoro-3-ethoxyphenyl
vinyl
ethyl



2.3.318
2-chloro-3-ethoxyphenyl
vinyl
ethyl



2.3.319
2-bromo-3-ethoxyphenyl
vinyl
ethyl



2.3.320
2-methyl-3-ethoxyphenyl
vinyl
ethyl



2.3.321
2-ethyl-3-ethoxyphenyl
vinyl
ethyl



2.3.322
2-cyclopropyl-3-ethoxyphenyl
vinyl
ethyl



2.3.323
2-vinyl-3-ethoxyphenyl
vinyl
ethyl



2.3.324
2-ethynyl-3-ethoxyphenyl
vinyl
ethyl



2.3.325
2-cyano-3-ethoxyphenyl
vinyl
ethyl



2.3.326
2-trifluoromethyl-3-ethoxyphenyl
vinyl
ethyl



2.3.327
2-methoxy-3-ethoxyphenyl
vinyl
ethyl



2.3.328
2,3-diethoxyphenyl
vinyl
ethyl



2.3.329
2-trifluoromethoxy-3-
vinyl
ethyl




ethoxyphenyl





2.3.330
2-nitro-3-ethoxyphenyl
vinyl
ethyl



2.3.331
2-fluoro-3-propoxyphenyl
vinyl
ethyl



2.3.332
2-chloro-3-propoxyphenyl
vinyl
ethyl



2.3.333
2-bromo-3-propoxyphenyl
vinyl
ethyl



2.3.334
2-methyl-3-propoxyphenyl
vinyl
ethyl



2.3.335
2-ethyl-3-propoxyphenyl
vinyl
ethyl



2.3.336
2-cyclopropyl-3-propoxyphenyl
vinyl
ethyl



2.3.337
2-vinyl-3-propoxyphenyl
vinyl
ethyl



2.3.338
2-ethynyl-3-propoxyphenyl
vinyl
ethyl



2.3.339
2-cyano-3-propoxyphenyl
vinyl
ethyl



2.3.340
2-trifluoromethyl-3-
vinyl
ethyl




propoxyphenyl





2.3.341
2-methoxy-3-propoxyphenyl
vinyl
ethyl



2.3.342
2-ethoxy-3-propoxyphenyl
vinyl
ethyl



2.3.343
2-trifluoromethoxy-3-
vinyl
ethyl




propoxyphenyl





2.3.344
2-nitro-3-propoxyphenyl
vinyl
ethyl



2.3.345
2-fluoro-3-isopropoxyphenyl
vinyl
ethyl



2.3.346
2-chloro-3-isopropoxyphenyl
vinyl
ethyl



2.3.347
2-bromo-3-isopropoxyphenyl
vinyl
ethyl



2.3.348
2-methyl-3-isopropoxyphenyl
vinyl
ethyl



2.3.349
2-ethyl-3-isopropoxyphenyl
vinyl
ethyl



2.3.350
2-cyclopropyl-3-
vinyl
ethyl




isopropoxyphenyl





2.3.351
2-vinyl-3-isopropoxyphenyl
vinyl
ethyl



2.3.352
2-ethynyl-3-isopropoxyphenyl
vinyl
ethyl



2.3.353
2-cyano-3-isopropoxyphenyl
vinyl
ethyl



2.3.354
2-trifluoromethyl-3-
vinyl
ethyl




isopropoxyphenyl





2.3.355
2-methoxy-3-isopropoxyphenyl
vinyl
ethyl



2.3.356
2-ethoxy-3-isopropoxyphenyl
vinyl
ethyl



2.3.357
2-trifluoromethoxy-3-
vinyl
ethyl




isopropoxyphenyl





2.3.358
2-nitro-3-isopropoxyphenyl
vinyl
ethyl



2.3.359
2-fluoro-3-tert-butoxyphenyl
vinyl
ethyl



2.3.360
2-chloro-3-tert-butoxyphenyl
vinyl
ethyl



2.3.361
2-bromo-3-tert-butoxyphenyl
vinyl
ethyl



2.3.362
2-methyl-3-tert-butoxyphenyl
vinyl
ethyl



2.3.363
2-ethyl-3-tert-butoxyphenyl
vinyl
ethyl



2.3.364
2-cyclopropyl-3-tert-
vinyl
ethyl




butoxyphenyl





2.3.365
2-vinyl-3-tert-butoxyphenyl
vinyl
ethyl



2.3.366
2-ethynyl-3-tert-butoxyphenyl
vinyl
ethyl



2.3.367
2-cyano-3-tert-butoxyphenyl
vinyl
ethyl



2.3.368
2-trifluoromethyl-3-tert-
vinyl
ethyl




butoxyphenyl





2.3.369
2-methoxy-3-tert-butoxyphenyl
vinyl
ethyl



2.3.370
2-ethoxy-3-tert-butoxyphenyl
vinyl
ethyl



2.3.371
2-trifluoromethoxy-3-tert-
vinyl
ethyl




butoxyphenyl





2.3.372
2-nitro-3-tert-butoxyphenyl
vinyl
ethyl



2.3.373
2-fluoro-3-trifluoromethoxy-
vinyl
ethyl




phenyl





2.3.374
2-chloro-3-trifluoromethoxy-
vinyl
ethyl




phenyl





2.3.375
2-bromo-3-trifluoromethoxy-
vinyl
ethyl




phenyl





2.3.376
2-methyl-3-trifluoromethoxy-
vinyl
ethyl




phenyl





2.3.377
2-ethyl-3-trifluoromethoxy-
vinyl
ethyl




phenyl





2.3.378
2-cyclopropyl-3-
vinyl
ethyl




trifluoromethoxyphenyl





2.3.379
2-vinyl-3-trifluoromethoxyphenyl
vinyl
ethyl



2.3.380
2-ethynyl-3-trifluoromethoxy-
vinyl
ethyl




phenyl





2.3.381
2-cyano-3-trifluoromethoxy-
vinyl
ethyl




phenyl





2.3.382
2-trifluoromethyl-3-
vinyl
ethyl




trifluoromethoxyphenyl





2.3.383
2-methoxy-3-trifluoromethoxy-
vinyl
ethyl




phenyl





2.3.384
2-ethoxy-3-trifluoromethoxy-
vinyl
ethyl




phenyl





2.3.385
2,3-bis(trifluoromethoxy)phenyl
vinyl
ethyl



2.3.386
2-nitro-3-trifluoromethoxyphenyl
vinyl
ethyl



2.3.387
2-fluoro-3-(2,2,2-trifluoroethoxy)-
vinyl
ethyl




phenyl





2.3.388
2-chloro-3-(2,2,2-
vinyl
ethyl




trifluoroethoxy)phenyl





2.3.389
2-bromo-3-(2,2,2-
vinyl
ethyl




trifluoroethoxy)phenyl





2.3.390
2-methyl-3-(2,2,2-
vinyl
ethyl




trifluoroethoxy)phenyl





2.3.391
2-ethyl-3-(2,2,2-trifluoroethoxy)-
vinyl
ethyl




phenyl





2.3.392
2-cyclopropyl-3-(2,2,2-trifluoro-
vinyl
ethyl




ethoxy)phenyl





2.3.393
2-vinyl-3-(2,2,2-trifluoroethoxy)-
vinyl
ethyl




phenyl





2.3.394
2-ethynyl-3-(2,2,2-
vinyl
ethyl




trifluoroethoxyphenyl





2.3.395
2-cyano-3-(2,2,2-
vinyl
ethyl




trifluoroethoxy)phenyl





2.3.396
2-trifluoromethyl-3-(2,2,2-
vinyl
ethyl




trifluoro-ethoxy)phenyl





2.3.397
2-methoxy-3-(2,2,2-
vinyl
ethyl




trifluoroethoxy)phenyl





2.3.398
2-ethoxy-3-(2,2,2-
vinyl
ethyl




trifluoroethoxy)phenyl





2.3.399
2-trifluoromethoxy-3-(2,2,2-
vinyl
ethyl




trifluoro-ethoxy)phenyl





2.3.400
2-nitro-3-(2,2,2-trifluoroethoxy)-
vinyl
ethyl




phenyl





2.3.401
2-fluoro-3-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.402
2-chloro-3-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.403
2-bromo-3-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.404
2-methyl-3-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.405
2-ethyl-3-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.406
2-cyclopropyl-3-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.407
2-vinyl-3-difluoromethoxyphenyl
vinyl
ethyl



2.3.408
2-ethynyl-3-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.409
2-cyano-3-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.410
2-trifluoromethyl-3-
vinyl
ethyl




difluoromethoxyphenyl





2.3.411
2-methoxy-3-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.412
2-ethoxy-3-
vinyl
ethyl




difluoromethoxyphenyl





2.3.413
2-trifluoromethoxy-3-
vinyl
ethyl




difluoromethoxyphenyl





2.3.414
2-nitro-3-difluoromethoxyphenyl
vinyl
ethyl



2.3.415
2-fluoro-3-(2-methoxyethoxy)-
vinyl
ethyl




phenyl





2.3.416
2-chloro-3-(2-methoxyethoxy)-
vinyl
ethyl




phenyl





2.3.417
2-bromo-3-(2-methoxyethoxy)-
vinyl
ethyl




phenyl





2.3.418
2-methyl-3-(2-methoxyethoxy)-
vinyl
ethyl




phenyl





2.3.419
2-ethyl-3-(2-
vinyl
ethyl




methoxyethoxy)phenyl





2.3.420
2-cyclopropyl-3-(2-
vinyl
ethyl




methoxyethoxy)phenyl





2.3.421
2-vinyl-3-(2-
vinyl
ethyl




methoxyethoxy)phenyl





2.3.422
2-ethynyl-3-(2-methoxyethoxy)-
vinyl
ethyl




phenyl





2.3.423
2-cyano-3-(2-methoxyethoxy)-
vinyl
ethyl




phenyl





2.3.424
2-trifluoromethyl-3-(2-
vinyl
ethyl




methoxyethoxy)phenyl





2.3.425
2-methoxy-3-(2-methoxyethoxy)-
vinyl
ethyl




phenyl





2.3.426
2-ethoxy-3-(2-methoxyethoxy)-
vinyl
ethyl




phenyl





2.3.427
2-trifluoromethoxy-(2-
vinyl
ethyl




methoxyethoxy)phenyl





2.3.428
2-nitro-3-(2-
vinyl
ethyl




methoxyethoxy)phenyl





2.3.429
2-fluoro-3-(tert-
vinyl
ethyl




butoxycarbonyloxy)phenyl





2.3.430
2-chloro-3-(tert-
vinyl
ethyl




butoxycarbonyloxy)phenyl





2.3.431
2-bromo-3-(tert-butoxycarbonyl-
vinyl
ethyl




oxy)phenyl





2.3.432
2-methyl-3-(tert-butoxycarbonyl-
vinyl
ethyl




oxy)phenyl





2.3.433
2-ethyl-3-(tert-
vinyl
ethyl




butoxycarbonyloxy)phenyl





2.3.434
2-cyclopropyl-3-(tert-
vinyl
ethyl




butoxycarbonyl-oxy)phenyl





2.3.435
2-vinyl-3-(tert-
vinyl
ethyl




butoxycarbonyloxy)phenyl





2.3.436
2-ethynyl-3-(tert-butoxycarbonyl-
vinyl
ethyl




oxy)phenyl





2.3.437
2-cyano-3-(tert-
vinyl
ethyl




butoxycarbonyloxy)phenyl





2.3.438
2-trifluoromethyl-3-(tert-
vinyl
ethyl




butoxycarbonyl-oxy)phenyl





2.3.439
2-methoxy-3-(tert-
vinyl
ethyl




butoxycarbonyloxy)phenyl





2.3.440
2-ethoxy-3-(tert-
vinyl
ethyl




butoxycarbonyloxy)phenyl





2.3.441
2-trifluoromethoxy-3-(tert-
vinyl
ethyl




butoxycarbonyl-oxy)phenyl





2.3.442
2-nitro-3-(tert-
vinyl
ethyl




butoxycarbonyloxy)phenyl





2.3.443
2-fluoro-3-nitrophenyl
vinyl
ethyl



2.3.444
2-chloro-3-nitrophenyl
vinyl
ethyl



2.3.445
2-bromo-3-nitrophenyl
vinyl
ethyl



2.3.446
2-methyl-3-nitrophenyl
vinyl
ethyl



2.3.447
2-ethyl-3-nitrophenyl
vinyl
ethyl



2.3.448
2-cyclopropyl-3-nitrophenyl
vinyl
ethyl



2.3.449
2-vinyl-3-nitrophenyl
vinyl
ethyl



2.3.450
2-ethynyl-3-nitrophenyl
vinyl
ethyl



2.3.451
2-cyano-3-nitrophenyl
vinyl
ethyl



2.3.452
2-trifluoromethyl-3-nitrophenyl
vinyl
ethyl



2.3.453
2-methoxy-3-nitrophenyl
vinyl
ethyl



2.3.454
2-ethoxy-3-nitrophenyl
vinyl
ethyl



2.3.455
2-trifluoromethoxy-3-nitrophenyl
vinyl
ethyl



2.3.456
2-fluoro-3-methylsulfanylphenyl
vinyl
ethyl



2.3.457
2-chloro-3-methylsulfanylphenyl
vinyl
ethyl



2.3.458
2-bromo-3-methylsulfanylphenyl
vinyl
ethyl



2.3.459
2-methyl-3-methylsulfanylphenyl
vinyl
ethyl



2.3.460
2-ethyl-3-methylsulfanylphenyl
vinyl
ethyl



2.3.461
2-cyclopropyl-3-
vinyl
ethyl




methylsulfanylphenyl





2.3.462
2-vinyl-3-methylsulfanylphenyl
vinyl
ethyl



2.3.463
2-ethynyl-3-
vinyl
ethyl




methylsulfanylphenyl





2.3.464
2-cyano-3-methylsulfanylphenyl
vinyl
ethyl



2.3.465
2-trifluoromethyl-3-
vinyl
ethyl




methylsulfanylphenyl





2.3.466
2-methoxy-3-
vinyl
ethyl




methylsulfanylphenyl





2.3.467
3,5-difluorophenyl
vinyl
methyl
One unassigned






enantiomer






[CDCl3] 3.34 (d, 1H);






3.84 (s, 3H); 3.94






(d, 1H); 5.38 (d, 1H);






5.55 (d, 1H); 6.14






(dd, 1H); 8.88 t, 1H);






7.18 (d, 2H).


2.3.468
3,5-difluorophenyl
vinyl
methyl
The other unassigned






enantiomer






[CDCl3] 3.34 (d, 1H);






3.84 (s, 3H); 3.94






(d, 1H); 5.38 (d, 1H);






5.55 (d, 1H); 6.14






(dd, 1H); 8.88 t, 1H);






7.18 (d, 2H).


2.3.469
3,5-difluorophenyl
2,2-difluoro-
ethyl
[CDCl3] 1.33 (t, 3H);




vinyl

3.46 (d, 1H); 4.02






(d, 1H); 4.23-4.37






(m, 2H); 4.91 (dd, 1H);






6.91 (t, 1H); 7.19






(d, 2H).


2.3.470
3,5-difluorophenyl
vinyl
ethyl
[CDCl3] 1.33 (t, 3H);






3.32 (d, 1H); 3.92






(d, 1H); 4.29 (m, 2H);






5.38 (d, 1H); 5.57






(d, 1H); 6.13 (dd, 1H);






6.89 (m, 1H); 7.19






(m, 2H).


2.3.471
3,5-difluorophenyl
1-methylvinyl
methyl
[CDCl3] 1.85 (s, 3H);






3.30 (d, 1H); 3.83






(s, 3H); 4.06 (d, 1H);






5.10 (s, 1H); 5.28






(s, 1H); 6.87 (m, 1H);






7.19 (d, 2H).


2.3.472
3,5-difluorophenyl
allyl
ethyl



2.3.473
3,5-difluorophenyl
1-chlorovinyl
methyl
[CDCl3] 3.53 (d, 1H);






3.88 (s, 3H); 4.22






(d, 1H); 5.55 (s, 1H);






5.93 (s, 1H); 6.90






(m, 1H); 7.20 (d, 2H).


2.3.474
3,5-difluorophenyl
ethynyl
ethyl



2.3.475
3-chloro-5-fluorophenyl
vinyl
methyl
[CDCl3] 3.34 (d, 1H);






3.84 (s, 3H); 3.93






(d, 1H); 5.39 (d, 1H);






5.55 (d, 1H), 6.14






(dd, 1H); 7.14 (d, 1H);






7.30 (d, 1H); 7.41






(s, 1H).


2.3.476
3-chloro-5-fluorophenyl
1-methylvinyl
methyl
[CDCl3] 1.84 (s, 3H);






3.30 (d, 1H); 3.83






(s, 3H); 4.07 (d, 1H);






5.10 (s, 1H); 5.28






(s, 1H); 7.14 (d, 1H);






7.32 (d, 1H); 7.43






(s, 1H).


2.3.477
3-chloro-5-fluorophenyl
allyl
ethyl



2.3.478
3-chloro-5-fluorophenyl
1-chlorovinyl
ethyl



2.3.479
3-chloro-5-fluorophenyl
ethynyl
ethyl



2.3.480
3-bromo-5-fluorophenyl
vinyl
ethyl



2.3.481
3-bromo-5-fluorophenyl
1-methylvinyl
ethyl



2.3.482
3-bromo-5-fluorophenyl
allyl
ethyl



2.3.483
3-bromo-5-fluorophenyl
1-chlorovinyl
ethyl



2.3.484
3-bromo-5-fluorophenyl
ethynyl
ethyl



2.3.485
3-iodo-5-fluorophenyl
vinyl
ethyl



2.3.486
3-methyl-5-fluorophenyl
vinyl
methyl
[CDCl3] 2.37 (s, 3H);






3.36 (d, 1H); 3.83






(s, 3H); 3.94 (d, 1H);






5.37 (d, 1H); 5.55






(d, 1H); 6.13 (dd, 1H);






6.94 (d, 1H); 7.18






(d, 1H); 7.24 (s, 1H).


2.3.487
3-methyl-5-fluorophenyl
1-methylvinyl
ethyl



2.3.488
3-methyl-5-fluorophenyl
allyl
ethyl



2.3.489
3-methyl-5-fluorophenyl
1-chlorovinyl
ethyl



2.3.490
3-methyl-5-fluorophenyl
ethynyl
ethyl



2.3.491
3-ethyl-5-fluorophenyl
vinyl
ethyl



2.3.492
3-propyl-5-fluorophenyl
vinyl
ethyl



2.3.493
3-i-propyl-5-fluorophenyl
vinyl
ethyl



2.3.494
3-n-butyl-5-fluorophenyl
vinyl
ethyl



2.3.495
3-isobutyl-5-fluorophenyl
vinyl
ethyl



2.3.496
3-tert-butyl-5-fluorophenyl
vinyl
ethyl



2.3.497
3-cyclopropyl-5-fluorophenyl
vinyl
ethyl



2.3.498
3-vinyl-5-fluorophenyl
vinyl
ethyl



2.3.499
3-ethynyl-5-fluorophenyl
vinyl
ethyl



2.3.500
3-cyano-5-fluorophenyl
vinyl
ethyl



2.3.501
3-trifluoromethyl-5-fluorophenyl
vinyl
ethyl



2.3.502
3-trifluoromethyl-5-fluorophenyl
1-methylvinyl
ethyl



2.3.503
3-trifluoromethyl-5-fluorophenyl
allyl
ethyl



2.3.504
3-trifluoromethyl-5-fluorophenyl
1-chlorovinyl
ethyl



2.3.505
3-trifluoromethyl-5-fluorophenyl
ethynyl
ethyl



2.3.506
3-(methoxycarbonyl)-5-
vinyl
ethyl




fluorophenyl





2.3.507
3-hydroxymethyl-5-fluorophenyl
vinyl
ethyl



2.3.508
3-carbamoyl-5-fluorophenyl
vinyl
ethyl



2.3.509
3-hydroxy-5-fluorophenyl
vinyl
ethyl



2.3.510
3-methoxy-5-fluorophenyl
vinyl
ethyl



2.3.511
3-ethoxy-5-fluorophenyl
vinyl
ethyl



2.3.512
3-n-propoxy-5-fluorophenyl
vinyl
ethyl



2.3.513
3-isopropoxy-5-fluorophenyl
vinyl
ethyl



2.3.514
3-n-butoxy-5-fluorophenyl
vinyl
ethyl



2.3.515
3-isobutoxy-5-fluorophenyl
vinyl
ethyl



2.3.516
3-tert-butoxy-5-fluorophenyl
vinyl
ethyl



2.3.517
3-difluoromethoxy-5-
vinyl
ethyl




fluorophenyl





2.3.518
3-trifluoromethoxy-5-
vinyl
ethyl




fluorophenyl





2.3.519
3-(2,2,2-trifluoroethoxy)-5-
vinyl
ethyl




fluorophenyl





2.3.520
3-(2-chloroethoxy)-5-
vinyl
ethyl




fluorophenyl





2.3.521
3-(2-hydroxyethoxy)-5-
vinyl
ethyl




fluorophenyl





2.3.522
3-[(tert-butoxycarbonyl)oxy]-5-
vinyl
ethyl




fluorophenyl





2.3.523
3-nitro-5-fluorophenyl
vinyl
ethyl



2.3.524
3-acetoxy-5-fluorophenyl
vinyl
ethyl



2.3.525
{3-[(tert-butoxy-carbonyl)amino]-
vinyl
ethyl




5-fluorophenyl}





2.3.526
3-methylsulfanyl-5-fluorophenyl
vinyl
ethyl



2.3.527
3,5-dichlorophenyl
vinyl
methyl
[CDCl3] 3.34 (d, 1H);






3.84 (s, 3H); 3.93






(d, 1H), 5.39 (d, 1H);






5.55 (d, 1H); 6.14






(dd, 1H); 7.40 (s, 1H);






7.54 (s, 2H).


2.3.528
3,5-dichlorophenyl
1-methylvinyl
methyl
[CDCl3] 1.84 (s, 3H);






3.30 (d, 1H); 3.83






(s, 3H); 4.06 (d, 1H);






5.10 (s, 1H); 5.28






(s, 1H); 7.41 (s, 1H);






7.55 (s, 2H).


2.3.529
3,5-dichlorophenyl
allyl
ethyl



2.3.530
3,5-dichlorophenyl
1-chlorovinyl
ethyl



2.3.531
3,5-dichlorophenyl
ethynyl
ethyl



2.3.532
3-bromo-5-chlorophenyl
vinyl
ethyl



2.3.533
3-iodo-5-chlorophenyl
vinyl
ethyl



2.3.534
3-methyl-5-chlorophenyl
vinyl
methyl
[CDCl3] 2.36 (s, 3H),






3.35 (d, 1H); 3.83






(s, 3H); 3.94 (d, 1H);






5.37 (d, 1H); 5.55






(d, 1H); 6.13 (dd, 1H);






7.22 (s, 1H); 7.38






(s, 1H); 7.43 (s, 1H).


2.3.535
3-methyl-5-chlorophenyl
1-methylvinyl
methyl
[CDCl3] 1.85 (s, 3H);






2.36 (s, 3H); 3.32






(d, 1H); 3.82 (s, 3H);






4.07 (d, 1H); 5.08






(s, 1H); 5.28 (s, 1H);






7.21 (s, 1H); 7.38






(s, 1H); 7.45 (s, 1H).


2.3.536
3-ethyl-5-chlorophenyl
vinyl
methyl
[CDCl3] 1.24 (t, 1H);






2.65 (q, 2H); 3.37






(d, 1H); 3.83 (s, 3H);






3.95 (d, 2H); 5.37






(d, 1H); 5.55 (d, 1H);






6.14 (dd, 1H); 7.24






(s, 1H); 7.40 (s, 1H);






7.43 (s, 1H).


2.3.537
3-propyl-5-chlorophenyl
vinyl
ethyl



2.3.538
3-isopropyl-5-chlorophenyl
vinyl
ethyl



2.3.539
3-n-butyl-5-chlorophenyl
vinyl
ethyl



2.3.540
3-isobutyl-5-chlorophenyl
vinyl
ethyl



2.3.541
3-tert-butyl-5-chlorophenyl
vinyl
ethyl



2.3.542
3-cyclopropyl-5-chlorophenyl
vinyl
ethyl



2.3.543
3-vinyl-5-chlorophenyl
vinyl
ethyl



2.3.544
3-ethynyl-5-chlorophenyl
vinyl
ethyl



2.3.545
3-cyano-5-chlorophenyl
vinyl
ethyl



2.3.546
3-trifluoromethyl-5-chlorophenyl
vinyl
ethyl



2.3.547
3-(hydroxycarbonyl)-5-
vinyl
ethyl




chlorophenyl





2.3.548
3-(methoxycarbonyl)-5-
vinyl
ethyl




chlorophenyl





2.3.549
3-hydroxymethyl-5-chlorophenyl
vinyl
ethyl



2.3.550
3-carbamoyl-5-chlorophenyl
vinyl
ethyl



2.3.551
3-hydroxy-5-chlorophenyl
vinyl
ethyl



2.3.552
3-methoxy-5-chlorophenyl
vinyl
ethyl



2.3.553
3-ethoxy-5-chlorophenyl
vinyl
ethyl



2.3.554
3-n-propoxy-5-chlorophenyl
vinyl
ethyl



2.3.555
3-isopropoxy-5-chlorophenyl
vinyl
ethyl



2.3.556
3-n-butoxy-5-chlorophenyl
vinyl
ethyl



2.3.557
3-isobutoxy-5-chlorophenyl
vinyl
ethyl



2.3.558
3-tert-butoxy-5-chlorophenyl
vinyl
ethyl



2.3.559
3-difluoromethoxy-5-
vinyl
ethyl




chlorophenyl





2.3.560
3-trifluoromethoxy-5-
vinyl
ethyl




chlorophenyl





2.3.561
3-(2,2,2-trifluoroethoxy)-5-
vinyl
ethyl




chlorophenyl





2.3.562
3-(2-chloroethoxy)-5-
vinyl
ethyl




chlorophenyl





2.3.563
3-(2-hydroxyethoxy)-5-
vinyl
ethyl




chlorophenyl





2.3.564
3-[(tert-butoxycarbonyl)oxy]-5-
vinyl
ethyl




chlorophenyl





2.3.565
3-nitro-5-chlorophenyl
vinyl
ethyl



2.3.566
3-acetoxy-5-chlorophenyl
vinyl
ethyl



2.3.567
{3-[(tert-butoxy-carbonyl)amino]-
vinyl
ethyl




5-chlorophenyl}





2.3.568
3-methylsulfanyl-5-chlorophenyl
vinyl
ethyl



2.3.569
3,5-dibromophenyl
vinyl
ethyl



2.3.570
3,5-dibromophenyl
1-methylvinyl 
ethyl



2.3.571
3-iodo-5-bromophenyl
vinyl
ethyl



2.3.572
3-methyl-5-bromophenyl
vinyl
methyl
[CDCl3] 2.35 (s, 3H),






3.35 (d, 1H); 3.83






(s, 3H); 3.93 (d, 1H);






5.35 (d, 1H), 5.55






(d, 1H); 6.13 (dd, 1H);






7.38 (s, 1H), 7.42






(s, 1H); 7.58 (s, 1H).


2.3.573
3-methyl-5-bromophenyl
1-methylvinyl
methyl
[CDCl3] 1.84 (s, 3H);






2.35 (s, 3H); 3.31






(d, 1H); 3.82 (s, 3H);






4.07 (d, 1H); 5.08






(s, 1H); 5.28 (s, 1H);






7.38 (s, 1H), 7.43






(s, 1H); 7.59 (s, 1H).


2.3.574
3-methyl-5-bromophenyl
allyl
ethyl



2.3.575
3-methyl-5-bromophenyl
1-chlorovinyl
ethyl



2.3.576
3-methyl-5-bromophenyl
ethynyl
ethyl



2.3.577
3-ethyl-5-bromophenyl
vinyl
ethyl



2.3.578
3-propyl-5-bromophenyl
vinyl
ethyl



2.3.579
3-isopropyl-5-bromophenyl
vinyl
ethyl



2.3.580
3-n-butyl-5-bromophenyl
vinyl
ethyl



2.3.581
3-isobutyl-5-bromophenyl
vinyl
ethyl



2.3.582
3-tert-butyl-5-bromophenyl
vinyl
ethyl



2.3.583
3-cyclopropyl-5-bromophenyl
vinyl
ethyl



2.3.584
3-vinyl-5-bromophenyl
vinyl
ethyl



2.3.585
3-ethynyl-5-bromophenyl
vinyl
ethyl



2.3.586
3-cyano-5-bromophenyl
vinyl
ethyl



2.3.587
3-trifluoromethyl-5-bromophenyl
vinyl
ethyl



2.3.588
3-(hydroxycarbonyl)-5-
vinyl
ethyl




bromophenyl





2.3.589
3-(methoxycarbonyl)-5-
vinyl
ethyl




bromophenyl





2.3.590
3-hydroxymethyl-5-bromophenyl
vinyl
ethyl



2.3.591
3-carbamoyl-5-bromophenyl
vinyl
ethyl



2.3.592
3-hydroxy-5-bromophenyl
vinyl
ethyl



2.3.593
3-methoxy-5-bromophenyl
vinyl
ethyl



2.3.594
3-ethoxy-5-bromophenyl
vinyl
ethyl



2.3.595
3-n-propoxy-5-bromophenyl
vinyl
ethyl



2.3.596
3-isopropoxy-5-bromophenyl
vinyl
ethyl



2.3.597
3-n-butoxy-5-bromophenyl
vinyl
ethyl



2.3.598
3-isobutoxy-5-bromophenyl
vinyl
ethyl



2.3.599
3-tert-butoxy-5-bromophenyl
vinyl
ethyl



2.3.600
3-difluoromethoxy-5-
vinyl
ethyl




bromophenyl





2.3.601
3-trifluoromethoxy-5-
vinyl
ethyl




bromophenyl





2.3.602
3-(2,2,2-trifluoroethoxy)-5-
vinyl
ethyl




bromophenyl





2.3.603
3-(2-chloroethoxy)-5-
vinyl
ethyl




bromophenyl





2.3.604
3-(2-hydroxyethoxy)-5-
vinyl
ethyl




bromophenyl





2.3.605
3-[(tert-butoxycarbonyl)oxy]-5-
vinyl
ethyl




bromophenyl





2.3.606
3-nitro-5-bromophenyl
vinyl
ethyl



2.3.607
3-acetoxy-5-bromophenyl
vinyl
ethyl



2.3.608
{3-[(tert-butoxy-carbonyl)amino]-
vinyl
ethyl




5-bromophenyl}





2.3.609
3-methylsulfanyl-5-bromophenyl
vinyl
ethyl



2.3.610
3,5-diiodophenyl
vinyl
ethyl



2.3.611
3-methyl-5-iodophenyl
vinyl
ethyl



2.3.612
3-ethyl-5-iodophenyl
vinyl
ethyl



2.3.613
3-propyl-5-iodophenyl
vinyl
ethyl



2.3.614
3-isopropyl-5-iodophenyl
vinyl
ethyl



2.3.615
3-n-butyl-5-iodophenyl
vinyl
ethyl



2.3.616
3-isobutyl-5-iodophenyl
vinyl
ethyl



2.3.617
3-tert-butyl-5-iodophenyl
vinyl
ethyl



2.3.618
3-cyclopropyl-5-iodophenyl
vinyl
ethyl



2.3.619
3-vinyl-5-iodophenyl
vinyl
ethyl



2.3.620
3-ethynyl-5-iodophenyl
vinyl
ethyl



2.3.621
3-cyano-5-iodophenyl
vinyl
ethyl



2.3.622
3-trifluoromethyl-5-iodophenyl
vinyl
ethyl



2.3.623
3-(hydroxycarbonyl)-5-
vinyl
ethyl




iodophenyl





2.3.624
3-(methoxycarbonyl)-5-
vinyl
ethyl




iodophenyl





2.3.625
3-hydroxymethyl-5-iodophenyl
vinyl
ethyl



2.3.626
3-carbamoyl-5-iodophenyl
vinyl
ethyl



2.3.627
3-hydroxy-5-iodophenyl
vinyl
ethyl



2.3.628
3-methoxy-5-iodophenyl
vinyl
ethyl



2.3.629
3-ethoxy-5-iodophenyl
vinyl
ethyl



2.3.630
3-n-propoxy-5-iodophenyl
vinyl
ethyl



2.3.631
3-isopropoxy-5-iodophenyl
vinyl
ethyl



2.3.632
3-n-butoxy-5-iodophenyl
vinyl
ethyl



2.3.633
3-isobutoxy-5-iodophenyl
vinyl
ethyl



2.3.634
3-tert-butoxy-5-iodophenyl
vinyl
ethyl



2.3.635
3-difluoromethoxy-5-iodophenyl
vinyl
ethyl



2.3.636
3-trifluoromethoxy-5-iodophenyl
vinyl
ethyl



2.3.637
3-(2,2,2-trifluoroethoxy)-5-
vinyl
ethyl




iodophenyl





2.3.638
3-(2-chloroethoxy)-5-iodophenyl
vinyl
ethyl



2.3.639
3-(2-hydroxyethoxy)-5-
vinyl
ethyl




iodophenyl





2.3.640
3-[(tert-butoxycarbonyl)oxy]-5-
vinyl
ethyl




iodophenyl





2.3.641
3-nitro-5-iodophenyl
vinyl
ethyl



2.3.642
3-acetoxy-5-iodophenyl
vinyl
ethyl



2.3.643
{3-[(tert-butoxy-carbonyl)amino]-
vinyl
ethyl




5-iodophenyl}





2.3.644
3-methylsulfanyl-5-iodophenyl
vinyl
ethyl



2.3.645
3,5-dimethylphenyl
vinyl
methyl
[CDCl3] 2.33 (s, 6H);






3.38 (d, 1H); 3.83






(s, 3H); 3.96 (d, 1H);






5.35 (d, 1H); 5.55






(d, 1H); 6.15 (dd, 1H);






7.06 (s, 1H); 7.28






(s, 2H).


2.3.646
3-ethyl-5-methylphenyl
vinyl
ethyl



2.3.647
3-propyl-5-methylphenyl
vinyl
ethyl



2.3.648
3-isopropyl-5-methylphenyl
vinyl
ethyl



2.3.649
3-n-butyl-5-methylphenyl
vinyl
ethyl



2.3.650
3-isobutyl-5-methylphenyl
vinyl
ethyl



2.3.651
3-tert-butyl-5-methylphenyl
vinyl
ethyl



2.3.652
3-cyclopropyl-5-methylphenyl
vinyl
ethyl



2.3.653
3-cyano-5-methylphenyl
vinyl
ethyl



2.3.654
3-trifluoromethyl-5-methylphenyl
vinyl
ethyl



2.3.655
3-(methoxycarbonyl)-5-
vinyl
ethyl




methylphenyl





2.3.656
3-methoxy-5-methylphenyl
vinyl
ethyl



2.3.657
3-ethoxy-5-methylphenyl
vinyl
ethyl



2.3.658
3-n-propoxy-5-methylphenyl
vinyl
ethyl



2.3.659
3-n-butoxy-5-methylphenyl
vinyl
ethyl



2.3.660
3-isobutoxy-5-methylphenyl
vinyl
ethyl



2.3.661
3-difluoromethoxy-5-
vinyl
ethyl




methylphenyl





2.3.662
3-trifluoromethoxy-5-
vinyl
ethyl




methylphenyl





2.3.663
3-nitro-5-methylphenyl
vinyl
ethyl



2.3.664
3-acetoxy-5-methylphenyl
vinyl
ethyl



2.3.665
3-methylsulfanyl-5-methylphenyl
vinyl
ethyl



2.3.666
3,5-diethylphenyl
vinyl
ethyl



2.3.667
3-propyl-5-ethylphenyl
vinyl
ethyl



2.3.668
3-isopropyl-5-ethylphenyl
vinyl
ethyl



2.3.669
3-n-butyl-5-ethylphenyl
vinyl
ethyl



2.3.670
3-isobutyl-5-ethylphenyl
vinyl
ethyl



2.3.671
3-tert-butyl-5-ethylphenyl
vinyl
ethyl



2.3.672
3-cyclopropyl-5-ethylphenyl
vinyl
ethyl



2.3.673
3-cyano-5-ethylphenyl
vinyl
ethyl



2.3.674
3-trifluoromethyl-5-ethylphenyl
vinyl
ethyl



2.3.675
3-(methoxycarbonyl)-5-
vinyl
ethyl




ethylphenyl





2.3.676
3-methoxy-5-ethylphenyl
vinyl
ethyl



2.3.677
3-ethoxy-5-ethylphenyl
vinyl
ethyl



2.3.678
3-n-propoxy-5-ethylphenyl
vinyl
ethyl



2.3.679
3-n-butoxy-5-ethylphenyl
vinyl
ethyl



2.3.680
3-isobutoxy-5-ethylphenyl
vinyl
ethyl



2.3.681
3-difluoromethoxy-5-ethylphenyl
vinyl
ethyl



2.3.682
3-trifluoromethoxy-5-ethylphenyl
vinyl
ethyl



2.3.683
3-nitro-5-ethylphenyl
vinyl
ethyl



2.3.684
3-acetoxy-5-ethylphenyl
vinyl
ethyl



2.3.685
3-methylsulfanyl-5-ethylphenyl
vinyl
ethyl



2.3.686
3,5-dipropylphenyl
vinyl
ethyl



2.3.687
3-isopropyl-5-propylphenyl
vinyl
ethyl



2.3.688
3-n-butyl-5-propylphenyl
vinyl
ethyl



2.3.689
3-isobutyl-5-propylphenyl
vinyl
ethyl



2.3.690
3-tert-butyl-5-propylphenyl
vinyl
ethyl



2.3.691
3-cyclopropyl-5-propylphenyl
vinyl
ethyl



2.3.692
3-cyano-5-propylphenyl
vinyl
ethyl



2.3.693
3-trifluoromethyl-5-propylphenyl
vinyl
ethyl



2.3.694
3-(methoxycarbonyl)-5-
vinyl
ethyl




propylphenyl





2.3.695
3-methoxy-5-propylphenyl
vinyl
ethyl



2.3.696
3-ethoxy-5-propylphenyl
vinyl
ethyl



2.3.697
3-n-propoxy-5-propylphenyl
vinyl
ethyl



2.3.698
3-n-butoxy-5-propylphenyl
vinyl
ethyl



2.3.699
3-isobutoxy-5-propylphenyl
vinyl
ethyl



2.3.700
3-difluoromethoxy-5-
vinyl
ethyl




propylphenyl





2.3.701
3-trifluoromethoxy-5-ethylphenyl
vinyl
ethyl



2.3.702
3-nitro-5-propylphenyl
vinyl
ethyl



2.3.703
3-acetoxy-5-propylphenyl
vinyl
ethyl



2.3.704
3-methylsulfanyl-5-propylphenyl
vinyl
ethyl



2.3.705
3,5-diisopropylphenyl
vinyl
ethyl



2.3.706
3-n-butyl-5-isopropylphenyl
vinyl
ethyl



2.3.707
3-isobutyl-5-isopropylphenyl
vinyl
ethyl



2.3.708
3-tert-butyl-5-isopropylphenyl
vinyl
ethyl



2.3.709
3-cyclopropyl-5-isopropylphenyl
vinyl
ethyl



2.3.710
3-cyano-5-isopropylphenyl
vinyl
ethyl



2.3.711
3-trifluoromethyl-5-
vinyl
ethyl




isopropylphenyl





2.3.712
3-(methoxycarbonyl)-5-
vinyl
ethyl




isopropylphenyl





2.3.713
3-methoxy-5-isopropylphenyl
vinyl
ethyl



2.3.714
3-ethoxy-5-isopropylphenyl
vinyl
ethyl



2.3.715
3-n-propoxy-5-isopropylphenyl
vinyl
ethyl



2.3.716
3-n-butoxy-5-isopropylphenyl
vinyl
ethyl



2.3.717
3-isobutoxy-5-isopropylphenyl
vinyl
ethyl



2.3.718
3-difluoromethoxy-5-
vinyl
ethyl




isopropylphenyl





2.3.719
3-trifluoromethoxy-5-
vinyl
ethyl




isopropylphenyl





2.3.720
3-nitro-5-isopropylphenyl
vinyl
ethyl



2.3.721
3-acetoxy-5-isopropylphenyl
vinyl
ethyl



2.3.722
3-methylsulfanyl-5-
vinyl
ethyl




isopropylphenyl





2.3.723
3,5-dibutylphenyl
vinyl
ethyl



2.3.724
3-isobutyl-5-butylphenyl
vinyl
ethyl



2.3.725
3-tert-butyl-5-butylphenyl
vinyl
ethyl



2.3.726
3-cyclopropyl-5-butylphenyl
vinyl
ethyl



2.3.727
3-cyano-5-butylphenyl
vinyl
ethyl



2.3.728
3-trifluoromethyl-5-butylphenyl
vinyl
ethyl



2.3.729
3-(methoxycarbonyl)-5-
vinyl
ethyl




butylphenyl





2.3.730
3-methoxy-5-butylphenyl
vinyl
ethyl



2.3.731
3-ethoxy-5-butylphenyl
vinyl
ethyl



2.3.732
3-n-propoxy-5-butylphenyl
vinyl
ethyl



2.3.733
3-n-butoxy-5-butylphenyl
vinyl
ethyl



2.3.734
3-isobutoxy-5-butylphenyl
vinyl
ethyl



2.3.735
3-difluoromethoxy-5-butylphenyl
vinyl
ethyl



2.3.736
3-trifluoromethoxy-5-butylphenyl
vinyl
ethyl



2.3.737
3-nitro-5-butylphenyl
vinyl
ethyl



2.3.738
3-acetoxy-5-butylphenyl
vinyl
ethyl



2.3.739
3-methylsulfanyl-5-butylphenyl
vinyl
ethyl



2.3.740
3,5-diisobutylphenyl
vinyl
ethyl



2.3.741
3-tert-butyl-5-isobutylphenyl
vinyl
ethyl



2.3.742
3-cyclopropyl-5-isobutylphenyl
vinyl
ethyl



2.3.743
3-cyano-5-isobutylphenyl
vinyl
ethyl



2.3.744
3-trifluoromethyl-5-
vinyl
ethyl




isobutylphenyl





2.3.745
3-(methoxycarbonyl)-5-
vinyl
ethyl




isobutylphenyl





2.3.746
3-methoxy-5-isobutylphenyl
vinyl
ethyl



2.3.747
3-ethoxy-5-isobutylphenyl
vinyl
ethyl



2.3.748
3-n-propoxy-5-isobutylphenyl
vinyl
ethyl



2.3.749
3-n-butoxy-5-isobutylphenyl
vinyl
ethyl



2.3.750
3-isobutoxy-5-isobutylphenyl
vinyl
ethyl



2.3.751
3-difluoromethoxy-5-
vinyl
ethyl




isobutylphenyl





2.3.752
3-trifluoromethoxy-5-
vinyl
ethyl




isobutylphenyl





2.3.753
3-nitro-5-isobutylphenyl
vinyl
ethyl



2.3.754
3-acetoxy-5-isobutylphenyl
vinyl
ethyl



2.3.755
3-methylsulfanyl-5-
vinyl
ethyl




isobutylphenyl





2.3.756
3,5-di(tert-butyl)phenyl
vinyl
ethyl



2.3.757
3-cyclopropyl-5-tert-butylphenyl
vinyl
ethyl



2.3.758
3-cyano-5-tert-butylphenyl
vinyl
ethyl



2.3.759
3-trifluoromethyl-5-tert-
vinyl
ethyl




butylphenyl





2.3.760
3-(methoxycarbonyl)-5-tert-
vinyl
ethyl




butylphenyl





2.3.761
3-methoxy-5-tert-butylphenyl
vinyl
ethyl



2.3.762
3-ethoxy-5-tert-butylphenyl
vinyl
ethyl



2.3.763
3-n-propoxy-5-tert-butylphenyl
vinyl
ethyl



2.3.764
3-n-butoxy-5-tert-butylphenyl
vinyl
ethyl



2.3.765
3-isobutoxy-5-tert-butylphenyl 
vinyl
ethyl



2.3.766
3-difluoromethoxy-5-tert-
vinyl
ethyl




butylphenyl





2.3.767
3-trifluoromethoxy-5-tert-
vinyl
ethyl




butylphenyl





2.3.768
3-nitro-5-tert-butylphenyl
vinyl
ethyl



2.3.769
3-acetoxy-5-tert-butylphenyl
vinyl
ethyl



2.3.770
3-methylsulfanyl-5-tert-
vinyl
ethyl




butylphenyl





2.3.771
3-tert-butyl-5-cyclopropylphenyl
vinyl
ethyl



2.3.772
3,5-dicyclopropyl-phenyl
vinyl
ethyl



2.3.773
3-cyano-5-cyclopropylphenyl
vinyl
ethyl



2.3.774
3-trifluoromethyl-5-
vinyl
ethyl




cyclopropylphenyl





2.3.775
3-(methoxycarbonyl)-5-
vinyl
ethyl




cyclopropylphenyl





2.3.776
3-methoxy-5-cyclopropylphenyl
vinyl
ethyl



2.3.777
3-ethoxy-5-cyclopropylphenyl
vinyl
ethyl



2.3.778
3-n-propoxy-5-cyclopropylphenyl
vinyl
ethyl



2.3.779
3-n-butoxy-5-cyclopropylphenyl
vinyl
ethyl



2.3.780
3-isobutoxy-5-cyclopropylphenyl
vinyl
ethyl



2.3.781
3-difluoromethoxy-5-
vinyl
ethyl




cyclopropylphenyl





2.3.782
3-trifluoromethoxy-5-
vinyl
ethyl




cyclopropylphenyl





2.3.783
3-nitro-5-cyclopropylphenyl
vinyl
ethyl



2.3.784
3-acetoxy-5-cyclopropylphenyl
vinyl
ethyl



2.3.785
3-methylsulfanyl-5-
vinyl
ethyl




cyclopropylphenyl





2.3.786
3,5-dicyanophenyl
vinyl
ethyl



2.3.787
3-trifluoromethyl-5-cyanophenyl
vinyl
ethyl



2.3.788
3-(methoxycarbonyl)-5-
vinyl
ethyl




cyanophenyl





2.3.789
3-methoxy-5-cyanophenyl
vinyl
ethyl



2.3.790
3-ethoxy-5-cyanophenyl
vinyl
ethyl



2.3.791
3-n-propoxy-5-cyanophenyl
vinyl
ethyl



2.3.792
3-n-butoxy-5-cyanophenyl
vinyl
ethyl



2.3.793
3-isobutoxy-5-cyanophenyl
vinyl
ethyl



2.3.794
3-difluoromethoxy-5-
vinyl
ethyl




cyanophenyl





2.3.795
3-trifluoromethoxy-5-
vinyl
ethyl




cyanophenyl





2.3.796
3-nitro-5-cyanophenyl
vinyl
ethyl



2.3.797
3-acetoxy-5-cyanophenyl
vinyl
ethyl



2.3.798
3-methylsulfanyl-5-cyanophenyl
vinyl
ethyl



2.3.799
3,5-di(trifluoromethyl)-phenyl
vinyl
ethyl



2.3.800
3-(methoxycarbonyl)-5-
vinyl
ethyl




trifluoromethyl-phenyl





2.3.801
3-methoxy-5-
vinyl
ethyl




trifluoromethylphenyl





2.3.802
3-ethoxy-5-trifluoromethylphenyl
vinyl
ethyl



2.3.803
3-n-propoxy-5-
vinyl
ethyl




trifluoromethylphenyl





2.3.804
3-isobutoxy-5-
vinyl
ethyl




trifluoromethylphenyl





2.3.805
3-difluoromethoxy-5-
vinyl
ethyl




trifluoromethylphenyl





2.3.806
3-trifluoromethoxy-5-
vinyl
ethyl




trifluoromethylphenyl





2.3.807
3-nitro-5-trifluoromethylphenyl
vinyl
ethyl



2.3.808
3-acetoxy-5-
vinyl
ethyl




trifluoromethylphenyl





2.3.809
3-methylsulfanyl-5-
vinyl
ethyl




trifluoromethylphenyl





2.3.810
3,5-di(methoxycarbonyl)phenyl
vinyl
ethyl



2.3.811
3-methoxy-5-(methoxycarbonyl)-
vinyl
ethyl




phenyl





2.3.812
3-ethoxy-5-(methoxycarbonyl)-
vinyl
ethyl




phenyl





2.3.813
3-n-propoxy-5-
vinyl
ethyl




(methoxycarbonyl)-phenyl





2.3.814
3-n-butoxy-5-(methoxycarbonyl)-
vinyl
ethyl




phenyl





2.3.815
3-isobutoxy-5-
vinyl
ethyl




(methoxycarbonyl)-phenyl





2.3.816
3-difluoromethoxy-5-
vinyl
ethyl




(methoxycarbonyl)-phenyl





2.3.817
3-trifluoromethoxy-5-
vinyl
ethyl




(methoxycarbonyl)-phenyl





2.3.818
3-nitro-5-(methoxy-
vinyl
ethyl




carbonyl)phenyl





2.3.819
3-acetoxy-5-(methoxycarbonyl)-
vinyl
ethyl




phenyl





2.3.820
3-methylsulfanyl-5-
vinyl
ethyl




(methoxycarbonyl)-phenyl





2.3.821
3,5-dimethoxyphenyl
vinyl
ethyl



2.3.822
3-ethoxy-5-methoxyphenyl
vinyl
ethyl



2.3.823
3-n-propoxy-5-methoxyphenyl
vinyl
ethyl



2.3.824
3-n-butoxy-5-methoxyphenyl
vinyl
ethyl



2.3.825
3-isobutoxy-5-methoxyphenyl
vinyl
ethyl



2.3.826
3-difluoromethoxy-5-
vinyl
ethyl




methoxyphenyl





2.3.827
3-trifluoromethoxy-5-
vinyl
ethyl




methoxyphenyl





2.3.828
3-nitro-5-methoxyphenyl
vinyl
ethyl



2.3.829
3-acetoxy-5-methoxyphenyl
vinyl
ethyl



2.3.830
3-methylsulfanyl-5-
vinyl
ethyl




methoxyphenyl





2.3.831
3,5-diethoxyphenyl
vinyl
ethyl



2.3.832
3-n-propoxy-5-ethoxyphenyl
vinyl
ethyl



2.3.833
3-n-butoxy-5-ethoxyphenyl
vinyl
ethyl



2.3.834
3-isobutoxy-5-ethoxyphenyl
vinyl
ethyl



2.3.835
3-difluoromethoxy-5-
vinyl
ethyl




ethoxyphenyl





2.3.836
3-trifluoromethoxy-5-
vinyl
ethyl




ethoxyphenyl





2.3.837
3-nitro-5-ethoxyphenyl
vinyl
ethyl



2.3.838
3-acetoxy-5-ethoxyphenyl
vinyl
ethyl



2.3.839
3-methylsulfanyl-5-ethoxyphenyl
vinyl
ethyl



2.3.840
3,5-di(isopropoxy)phenyl
vinyl
ethyl



2.3.841
3-n-butoxy-5-isopropoxyphenyl
vinyl
ethyl



2.3.842
3-isobutoxy-5-isopropoxyphenyl
vinyl
ethyl



2.3.843
3-difluoromethoxy-5-
vinyl
ethyl




isopropoxyphenyl





2.3.844
3-trifluoromethoxy-5-
vinyl
ethyl




isopropoxyphenyl





2.3.845
3-nitro-5-isopropoxyphenyl
vinyl
ethyl



2.3.846
3-acetoxy-5-isopropoxyphenyl
vinyl
ethyl



2.3.847
3-methylsulfanyl-5-
vinyl
ethyl




isopropoxyphenyl





2.3.848
3,5-di(trifluoro-methoxy)phenyl
vinyl
ethyl



2.3.849
3-nitro-5-trifluoro-methoxyphenyl
vinyl
ethyl



2.3.850
3-methylsulfanyl-5-
vinyl
ethyl




trifluoromethoxy-phenyl





2.3.851
3,5-bis(difluoro-methoxy)phenyl
vinyl
ethyl



2.3.852
3,5-bis(difluoro-methoxy)phenyl
1-methylvinyl
ethyl



2.3.853
3,5-bis(difluoro-methoxy)phenyl
allyl
ethyl



2.3.854
3,5-bis(difluoro-methoxy)phenyl
1-chlorovinyl
ethyl



2.3.855
3-trifluoromethoxy-5-
vinyl
ethyl




difluoromethoxy-phenyl





2.3.856
3-nitro-5-difluoro-methoxyphenyl
vinyl
ethyl



2.3.857
3-acetoxy-5-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.858
3-methylsulfanyl-5-
vinyl
ethyl




difluoromethoxy-phenyl





2.3.859
3,5-bis(acetoxy)phenyl
vinyl
ethyl



2.3.860
3-methylsulfanyl-5-
vinyl
ethyl




acetoxyphenyl





2.3.861
3,5-dinitrophenyl
vinyl
ethyl



2.3.862
3-acetoxy-5-nitrophenyl
vinyl
ethyl



2.3.863
3-methylsulfanyl-5-nitrophenyl
vinyl
ethyl



2.3.864
3,5-di(methylsulfanyl)phenyl
vinyl
ethyl



2.3.865
3,4-difluorophenyl
vinyl
ethyl



2.3.866
3,4-difluorophenyl
1-methylvinyl
ethyl



2.3.867
3,4-difluorophenyl
allyl
ethyl



2.3.868
3,4-difluorophenyl
1-chlorovinyl
ethyl



2.3.869
3,4-difluorophenyl
ethynyl
ethyl



2.3.870
3-chloro-4-fluorophenyl
vinyl
ethyl



2.3.871
3-chloro-4-fluorophenyl
1-methylvinyl
ethyl



2.3.872
3-chloro-4-fluorophenyl
allyl
ethyl



2.3.873
3-chloro-4-fluorophenyl
1-chlorovinyl
ethyl



2.3.874
3-chloro-4-fluorophenyl
ethynyl
ethyl



2.3.875
3-bromo-4-fluorophenyl
vinyl
ethyl



2.3.876
3-methyl-4-fluorophenyl
vinyl
ethyl



2.3.877
3-methyl-4-fluorophenyl
1-methylvinyl
ethyl



2.3.878
3-ethyl-4-fluorophenyl
vinyl
ethyl



2.3.879
3-cyclopropyl-4-fluorophenyl
vinyl
ethyl



2.3.880
3-cyano-4-fluorophenyl
vinyl
ethyl



2.3.881
3-methoxy-4-fluorophenyl
vinyl
ethyl



2.3.882
3-ethoxy-4-fluorophenyl
vinyl
ethyl



2.3.883
3-trifluoromethoxy-4-
vinyl
ethyl




fluorophenyl





2.3.884
3-nitro-4-fluorophenyl
vinyl
ethyl



2.3.885
3-fluoro-4-chlorophenyl
vinyl
ethyl



2.3.886
3,4-dichlorophenyl
vinyl
ethyl



2.3.887
3-bromo-4-chlorophenyl
vinyl
ethyl



2.3.888
3-methyl-4-chlorophenyl
vinyl
ethyl



2.3.889
3-cyclopropyl-4-chlorophenyl
vinyl
ethyl



2.3.890
3-cyano-4-chlorophenyl
vinyl
ethyl



2.3.891
3-trifluoromethyl-4-chlorophenyl
vinyl
ethyl



2.3.892
3-methoxy-4-chlorophenyl
vinyl
ethyl



2.3.893
3-ethoxy-4-chlorophenyl
vinyl
ethyl



2.3.894
3-trifluoromethoxy-4-
vinyl
ethyl




chlorophenyl





2.3.895
3-nitro-4-chlorophenyl
vinyl
ethyl



2.3.896
3-fluoro-4-bromophenyl
vinyl
ethyl



2.3.897
3-chloro-4-bromophenyl
vinyl
ethyl



2.3.898
3,4-dibromophenyl
vinyl
ethyl



2.3.899
3-methyl-4-bromophenyl
vinyl
ethyl



2.3.900
3-ethyl-4-bromophenyl
vinyl
ethyl



2.3.901
3-cyclopropyl-4-bromophenyl
vinyl
ethyl



2.3.902
3-cyano-4-bromophenyl
vinyl
ethyl



2.3.903
3-trifluoromethyl-4-bromophenyl 
vinyl
ethyl



2.3.904
3-methoxy-4-phenyl
vinyl
ethyl



2.3.905
3-ethoxy-4-bromophenyl
vinyl
ethyl



2.3.906
3-trifluoromethoxy-4-
vinyl
ethyl




bromophenyl





2.3.907
3-nitro-4-bromophenyl
vinyl
ethyl



2.3.908
3-fluoro-4-iodophenyl
vinyl
ethyl



2.3.909
3-chloro-4-iodophenyl
vinyl
ethyl



2.3.910
3-bromo-4-iodophenyl
vinyl
ethyl



2.3.911
3-methyl-4-iodophenyl
vinyl
ethyl



2.3.912
3-cyclopropyl-4-iodophenyl
vinyl
ethyl



2.3.913
3-cyano-4-iodophenyl
vinyl
ethyl



2.3.914
3-trifluoromethyl-4-iodophenyl 
vinyl
ethyl



2.3.915
3-methoxy-4-iodophenyl
vinyl
ethyl



2.3.916
3-ethoxy-4-iodophenyl
vinyl
ethyl



2.3.917
3-trifluoromethoxy-4-iodophenyl 
vinyl
ethyl



2.3.918
3-nitro-4-iodophenyl
vinyl
ethyl



2.3.919
3-fluoro-4-methylphenyl
vinyl
ethyl



2.3.920
3-chloro-4-methylphenyl
vinyl
ethyl



2.3.921
3-bromo-4-methylphenyl
vinyl
ethyl



2.3.922
3,4-dimethylphenyl
vinyl
ethyl



2.3.923
3,4-dimethylphenyl
1-methylvinyl
ethyl



2.3.924
3,4-dimethylphenyl
allyl
ethyl



2.3.925
3,4-dimethylphenyl
1-chlorovinyl
ethyl



2.3.926
3,4-dimethylphenyl
ethynyl
ethyl



2.3.927
3-ethyl-4-methylphenyl
vinyl
ethyl



2.3.928
3-cyclopropyl-4-methylphenyl
vinyl
ethyl



2.3.929
3-cyano-4-methylphenyl
vinyl
ethyl



2.3.930
3-trifluoromethyl-4-methylphenyl
vinyl
ethyl



2.3.931
3-methoxy-4-methylphenyl
vinyl
ethyl



2.3.932
3-ethoxy-4-methylphenyl
vinyl
ethyl



2.3.933
3-trifluoromethoxy-4-
vinyl
ethyl




methylphenyl





2.3.934
3-nitro-4-methylphenyl
vinyl
ethyl



2.3.935
3-fluoro-4-ethylphenyl
vinyl
ethyl



2.3.936
3-chloro-4-ethylphenyl
vinyl
ethyl



2.3.937
3-bromo-4-ethylphenyl
vinyl
ethyl



2.3.938
3-methyl-4-ethylphenyl
vinyl
ethyl



2.3.939
3,4-diethylphenyl
vinyl
ethyl



2.3.940
3-cyclopropyl-4-ethylphenyl
vinyl
ethyl



2.3.941
3-cyano-4-ethylphenyl
vinyl
ethyl



2.3.942
3-trifluoromethyl-4-ethylphenyl
vinyl
ethyl



2.3.943
3-methoxy-4-ethylphenyl
vinyl
ethyl



2.3.944
3-ethoxy-4-ethylphenyl
vinyl
ethyl



2.3.945
3-trifluoromethoxy-4-ethylphenyl
vinyl
ethyl



2.3.946
3-nitro-4-ethylphenyl
vinyl
ethyl



2.3.947
3-fluoro-4-propylphenyl
vinyl
ethyl



2.3.948
3-chloro-4-propylphenyl
vinyl
ethyl



2.3.949
3-bromo-4-propylphenyl
vinyl
ethyl



2.3.950
3-methyl-4-propylphenyl
vinyl
ethyl



2.3.951
3-cyclopropyl-4-propylphenyl
vinyl
ethyl



2.3.952
3-cyano-4-propylphenyl
vinyl
ethyl



2.3.953
3-trifluoromethyl-4-propylphenyl
vinyl
ethyl



2.3.954
3-methoxy-4-propylphenyl
vinyl
ethyl



2.3.955
3-ethoxy-4-propylphenyl
vinyl
ethyl



2.3.956
3-trifluoromethoxy-4-
vinyl
ethyl




propylphenyl





2.3.957
3-nitro-4-propylphenyl
vinyl
ethyl



2.3.958
3-fluoro-4-isopropylphenyl
vinyl
ethyl



2.3.959
3-chloro-4-isopropylphenyl
vinyl
ethyl



2.3.960
3-bromo-4-isopropylphenyl
vinyl
ethyl



2.3.961
3-methyl-4-isopropylphenyl
vinyl
ethyl



2.3.962
3-cyclopropyl-4-isopropylphenyl
vinyl
ethyl



2.3.963
3-cyano-4-isopropylphenyl
vinyl
ethyl



2.3.964
3-trifluoromethyl-4-
vinyl
ethyl




isopropylphenyl





2.3.965
3-methoxy-4-isopropylphenyl
vinyl
ethyl



2.3.966
3-ethoxy-4-isopropylphenyl
vinyl
ethyl



2.3.967
3-trifluoromethoxy-4-
vinyl
ethyl




isopropylphenyl





2.3.968
3-nitro-4-isopropylphenyl
vinyl
ethyl



2.3.969
3-fluoro-4-tert-butylphenyl
vinyl
ethyl



2.3.970
3-chloro-4-tert-butylphenyl
vinyl
ethyl



2.3.971
3-bromo-4-tert-butylphenyl
vinyl
ethyl



2.3.972
3-methyl-4-tert-butylphenyl
vinyl
ethyl



2.3.973
3-cyclopropyl-4-tert-butylphenyl
vinyl
ethyl



2.3.974
3-cyano-4-tert-butylphenyl
vinyl
ethyl



2.3.975
3-trifluoromethyl-4-tert-
vinyl
ethyl




butylphenyl





2.3.976
3-trifluoromethyl-4-tert-
1-methylvinyl 
ethyl




butylphenyl





2.3.977
3-trifluoromethyl-4-tert-
allyl
ethyl




butylphenyl





2.3.978
3-trifluoromethyl-4-tert-
1-chlorovinyl 
ethyl




butylphenyl





2.3.979
3-trifluoromethyl-4-tert-
ethynyl
ethyl




butylphenyl





2.3.980
3-methoxy-4-tert-butylphenyl
vinyl
ethyl



2.3.981
3-ethoxy-4-tert-butylphenyl
vinyl
ethyl



2.3.982
3-trifluoromethoxy-4-tert-
vinyl
ethyl




butylphenyl





2.3.983
3-nitro-4-tert-butylphenyl
vinyl
ethyl



2.3.984
3-fluoro-4-cyclopropylphenyl
vinyl
ethyl



2.3.985
3-chloro-4-cyclopropylphenyl
vinyl
ethyl



2.3.986
3-bromo-4-cyclopropylphenyl
vinyl
ethyl



2.3.987
3-methyl-4-cyclopropylphenyl
vinyl
ethyl



2.3.988
3-cyclopropyl-4-
vinyl
ethyl




cyclopropylphenyl





2.3.989
3-cyano-4-cyclopropylphenyl
vinyl
ethyl



2.3.990
3-trifluoromethyl-4-
vinyl
ethyl




cyclopropylphenyl





2.3.991
3-methoxy-4-cyclopropylphenyl
vinyl
ethyl



2.3.992
3-ethoxy-4-cyclopropylphenyl
vinyl
ethyl



2.3.993
3-trifluoromethoxy-4-
vinyl
ethyl




cyclopropylphenyl





2.3.994
3-fluoro-4-methoxycarbonyl-
vinyl
ethyl




phenyl





2.3.995
3-chloro-4-methoxy-
vinyl
ethyl




carbonylphenyl





2.3.996
3-bromo-4-methoxy-
vinyl
ethyl




carbonylphenyl





2.3.997
3-methyl-4-methoxy-
vinyl
ethyl




carbonylphenyl





2.3.998
3-cyclopropyl-4-
vinyl
ethyl




methoxycarbonyl-phenyl





2.3.999
3-cyano-4-
vinyl
ethyl




methoxycarbonylphenyl





2.3.1000
3-trifluoromethyl-4-
vinyl
ethyl




methoxycarbonyl-phenyl





2.3.1001
3-methoxy-4-methoxycarbonyl-
vinyl
ethyl




phenyl





2.3.1002
3-ethoxy-4-methoxycarbonyl-
vinyl
ethyl




phenyl





2.3.1003
3-trifluoromethoxy-4-
vinyl
ethyl




methoxycarbonyl-phenyl





2.3.1004
3-nitro-4-methoxy-
vinyl
ethyl




carbonylphenyl





2.3.1005
3-fluoro-4-cyanophenyl
vinyl
ethyl



2.3.1006
3-chloro-4-cyanophenyl
vinyl
ethyl



2.3.1007
3-bromo-4-cyanophenyl
vinyl
ethyl



2.3.1008
3-methyl-4-cyanophenyl
vinyl
ethyl



2.3.1009
3-cyclopropyl-4-cyanophenyl
vinyl
ethyl



2.3.1010
3,4-dicyanophenyl
vinyl
ethyl



2.3.1011
3-trifluoromethyl-4-cyanophenyl
vinyl
ethyl



2.3.1012
3-trifluoromethyl-4-cyanophenyl
1-methylvinyl
ethyl



2.3.1013
3-trifluoromethyl-4-cyanophenyl
allyl
ethyl



2.3.1014
3-trifluoromethyl-4-cyanophenyl
1-chlorovinyl
ethyl



2.3.1015
3-trifluoromethyl-4-cyanophenyl
ethynyl
ethyl



2.3.1016
3-methoxy-4-cyanophenyl
vinyl
ethyl



2.3.1017
3-ethoxy-4-cyanophenyl
vinyl
ethyl



2.3.1018
3-trifluoromethoxy-4-
vinyl
ethyl




cyanophenyl





2.3.1019
3-nitro-4-cyanophenyl
vinyl
ethyl



2.3.1020
3-fluoro-4-methoxyphenyl
vinyl
ethyl



2.3.1021
3-chloro-4-methoxyphenyl
vinyl
ethyl



2.3.1022
3-bromo-4-methoxyphenyl
vinyl
ethyl



2.3.1023
3-methyl-4-methoxyphenyl
vinyl
ethyl



2.3.1024
3-cyclopropyl-4-methoxyphenyl
vinyl
ethyl



2.3.1025
3-cyano-4-methoxyphenyl
vinyl
ethyl



2.3.1026
3-trifluoromethyl-4-
vinyl
ethyl




methoxyphenyl





2.3.1027
3,4-dimethoxyphenyl
vinyl
ethyl



2.3.1028
3-ethoxy-4-methoxyphenyl
vinyl
ethyl



2.3.1029
3-trifluoromethoxy-4-
vinyl
ethyl




methoxyphenyl





2.3.1030
3-nitro-4-methoxyphenyl
vinyl
ethyl



2.3.1031
3-fluoro-4-ethoxyphenyl
vinyl
ethyl



2.3.1032
3-chloro-4-ethoxyphenyl
vinyl
ethyl



2.3.1033
3-chloro-4-ethoxyphenyl
1-methylvinyl
ethyl



2.3.1034
3-chloro-4-ethoxyphenyl
allyl
ethyl



2.3.1035
3-chloro-4-ethoxyphenyl
1-chlorovinyl
ethyl



2.3.1036
3-chloro-4-ethoxyphenyl
ethynyl
ethyl



2.3.1037
3-bromo-4-ethoxyphenyl
vinyl
ethyl



2.3.1038
3-methyl-4-ethoxyphenyl
vinyl
ethyl



2.3.1039
3-cyclopropyl-4-ethoxyphenyl
vinyl
ethyl



2.3.1040
3-cyano-4-ethoxyphenyl
vinyl
ethyl



2.3.1041
3-trifluoromethyl-4-ethoxyphenyl
vinyl
ethyl



2.3.1042
3-methoxy-4-ethoxyphenyl
vinyl
ethyl



2.3.1043
2,4-diethoxyphenyl
vinyl
ethyl



2.3.1044
3-trifluoromethoxy-4-
vinyl
ethyl




ethoxyphenyl





2.3.1045
3-nitro-4-ethoxyphenyl
vinyl
ethyl



2.3.1046
3-fluoro-4-isopropoxyphenyl
vinyl
ethyl



2.3.1047
3-chloro-4-isopropoxyphenyl
vinyl
ethyl



2.3.1048
3-bromo-4-isopropoxyphenyl
vinyl
ethyl



2.3.1049
3-methyl-4-isopropoxyphenyl
vinyl
ethyl



2.3.1050
3-cyclopropyl-4-
vinyl
ethyl




isopropoxyphenyl





2.3.1051
3-cyano-4-isopropoxyphenyl
vinyl
ethyl



2.3.1052
3-trifluoromethyl-4-
vinyl
ethyl




isopropoxyphenyl





2.3.1053
3-methoxy-4-isopropoxyphenyl
vinyl
ethyl



2.3.1054
3-ethoxy-4-isopropoxyphenyl
vinyl
ethyl



2.3.1055
3-trifluoromethoxy-4-
vinyl
ethyl




isopropoxyphenyl





2.3.1056
3-nitro-4-isopropoxyphenyl
vinyl
ethyl



2.3.1057
3-fluoro-4-trifluoro-
vinyl
ethyl




methoxyphenyl





2.3.1058
3-chloro-4-trifluoro-
vinyl
ethyl




methoxyphenyl





2.3.1059
3-bromo-4-trifluoro-
vinyl
ethyl




methoxyphenyl





2.3.1060
3-methyl-4-trifluoro-
vinyl
ethyl




methoxyphenyl





2.3.1061
3-cyclopropyl-4-
vinyl
ethyl




trifluoromethoxyphenyl





2.3.1062
3-cyano-4-trifluoro-
vinyl
ethyl




methoxyphenyl





2.3.1063
3-trifluoromethyl-4-
vinyl
ethyl




trifluoromethoxyphenyl





2.3.1064
3-methoxy-4-trifluoromethoxy-
vinyl
ethyl




phenyl





2.3.1065
3-ethoxy-4-trifluoro-
vinyl
ethyl




methoxyphenyl





2.3.1066
3,4-bis(trifluoromethoxy)phenyl
vinyl
ethyl



2.3.1067
3-nitro-4-trifluoromethoxyphenyl
vinyl
ethyl



2.3.1068
3-fluoro-4-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.1069
3-chloro-4-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.1070
3-bromo-4-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.1071
3-methyl-4-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.1072
3-cyclopropyl-4-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.1073
3-cyano-4-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.1074
3-trifluoromethyl-4-
vinyl
ethyl




difluoromethoxyphenyl





2.3.1075
3-methoxy-4-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.1076
3-ethoxy-4-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.1077
3-trifluoromethoxy-4-
vinyl
ethyl




difluoromethoxyphenyl





2.3.1078
3-nitro-4-difluoromethoxyphenyl
vinyl
ethyl



2.3.1079
3-fluoro-4-nitrophenyl
vinyl
ethyl



2.3.1080
3-chloro-4-nitrophenyl
vinyl
ethyl



2.3.1081
3-bromo-4-nitrophenyl
vinyl
ethyl



2.3.1082
3-methyl-4-nitrophenyl
vinyl
ethyl



2.3.1083
3-cyclopropyl-4-nitrophenyl
vinyl
ethyl



2.3.1084
3-cyano-4-nitrophenyl
vinyl
ethyl



2.3.1085
3-trifluoromethyl-4-nitrophenyl
vinyl
ethyl



2.3.1086
3-methoxy-4-nitrophenyl
vinyl
ethyl



2.3.1087
3-ethoxy-4-nitrophenyl
vinyl
ethyl



2.3.1088
3-trifluoromethoxy-4-nitrophenyl
vinyl
ethyl



2.3.1089
3-fluoro-4-methylsulfanylphenyl
vinyl
ethyl



2.3.1090
3-chloro-4-methylsulfanylphenyl
vinyl
ethyl



2.3.1091
3-bromo-4-methylsulfanylphenyl
vinyl
ethyl



2.3.1092
3-methyl-4-methylsulfanylphenyl
vinyl
ethyl



2.3.1093
3-cyclopropyl-4-
vinyl
ethyl




methylsulfanylphenyl





2.3.1094
3-cyano-4-methylsulfanylphenyl
vinyl
ethyl



2.3.1095
3-trifluoromethyl-4-
vinyl
ethyl




methylsulfanylphenyl





2.3.1096
3-methoxy-4-
vinyl
ethyl




methylsulfanylphenyl





2.3.1097
3-ethoxy-4-methylsulfanylphenyl
vinyl
ethyl



2.3.1098
3-trifluoromethoxy-4-
vinyl
ethyl




methylsulfanylphenyl





2.3.1099
3-nitro-4-methylsulfanylphenyl 
vinyl
ethyl



2.3.1100
3,6-difluorophenyl
vinyl
ethyl



2.3.1101
3,6-difluorophenyl
1-methylvinyl
ethyl



2.3.1102
3,6-difluorophenyl
allyl
ethyl



2.3.1103
3,6-difluorophenyl
1-chlorovinyl 
ethyl



2.3.1104
3,6-difluorophenyl
ethynyl
ethyl



2.3.1105
3-chloro-6-fluorophenyl
vinyl
ethyl



2.3.1106
3-bromo-6-fluorophenyl
vinyl
ethyl



2.3.1107
3-methyl-6-fluorophenyl
vinyl
ethyl



2.3.1108
3-cyclopropyl-6-fluorophenyl
vinyl
ethyl



2.3.1109
3-cyano-6-fluorophenyl
vinyl
ethyl



2.3.1110
3-methoxy-6-fluorophenyl
vinyl
ethyl



2.3.1111
3-ethoxy-6-fluorophenyl
vinyl
ethyl



2.3.1112
3-trifluoromethoxy-6-
vinyl
ethyl




fluorophenyl





2.3.1113
3-nitro-6-fluorophenyl
vinyl
ethyl



2.3.1114
3-fluoro-6-chlorophenyl
vinyl
ethyl



2.3.1115
3-fluoro-6-chlorophenyl
1-methylvinyl
ethyl



2.3.1116
3-fluoro-6-chlorophenyl
allyl
ethyl



2.3.1117
3-fluoro-6-chlorophenyl 
1-chlorovinyl
ethyl



2.3.1118
3-fluoro-6-chlorophenyl
ethynyl
ethyl



2.3.1119
3,6-dichlorophenyl
vinyl
ethyl



2.3.1120
3,6-dichlorophenyl
1-methylvinyl 
ethyl



2.3.1121
3,6-dichlorophenyl
allyl
ethyl



2.3.1122
3,6-dichlorophenyl
1-chlorovinyl 
ethyl



2.3.1123
3,6-dichlorophenyl
ethynyl
ethyl



2.3.1124
3-bromo-6-chlorophenyl
vinyl
ethyl



2.3.1125
3-methyl-6-chlorophenyl
vinyl
ethyl



2.3.1126
3-cyclopropyl-6-chlorophenyl
vinyl
ethyl



2.3.1127
3-cyano-6-chlorophenyl
vinyl
ethyl



2.3.1128
3-trifluoromethyl-6-chlorophenyl
vinyl
ethyl



2.3.1129
3-methoxy-6-chlorophenyl
vinyl
ethyl



2.3.1130
3-ethoxy-6-chlorophenyl
vinyl
ethyl



2.3.1131
3-trifluoromethoxy-6-
vinyl
ethyl




chlorophenyl





2.3.1132
3-nitro-6-chlorophenyl
vinyl
ethyl



2.3.1133
3-fluoro-6-bromophenyl
vinyl
ethyl



2.3.1134
3-chloro-6-bromophenyl
vinyl
ethyl



2.3.1135
3,6-dibromophenyl
vinyl
ethyl



2.3.1136
3-methyl-6-bromophenyl
vinyl
ethyl



2.3.1137
3-cyclopropyl-6-bromophenyl
vinyl
ethyl



2.3.1138
3-cyano-6-bromophenyl
vinyl
ethyl



2.3.1139
3-trifluoromethyl-6-bromophenyl
vinyl
ethyl



2.3.1140
3-methoxy-6-phenyl
vinyl
ethyl



2.3.1141
3-ethoxy-6-bromophenyl
vinyl
ethyl



2.3.1142
3-trifluoromethoxy-6-
vinyl
ethyl




bromophenyl





2.3.1143
3-nitro-6-bromophenyl
vinyl
ethyl



2.3.1144
3-fluoro-6-iodophenyl
vinyl
ethyl



2.3.1145
3-chloro-6-iodophenyl
vinyl
ethyl



2.3.1146
3-bromo-6-iodophenyl
vinyl
ethyl



2.3.1147
3-methyl-6-iodophenyl
vinyl
ethyl



2.3.1148
3-cyclopropyl-6-iodophenyl
vinyl
ethyl



2.3.1149
3-cyano-6-iodophenyl
vinyl
ethyl



2.3.1150
3-trifluoromethyl-6-iodophenyl
vinyl
ethyl



2.3.1151
3-methoxy-6-iodophenyl
vinyl
ethyl



2.3.1152
3-ethoxy-6-iodophenyl
vinyl
ethyl



2.3.1153
3-trifluoromethoxy-6-iodophenyl
vinyl
ethyl



2.3.1154
3-nitro-6-iodophenyl
vinyl
ethyl



2.3.1155
3-fluoro-6-methylphenyl
vinyl
ethyl



2.3.1156
3-chloro-6-methylphenyl
vinyl
ethyl



2.3.1157
3-bromo-6-methylphenyl
vinyl
ethyl



2.3.1158
3,6-dimethylphenyl
vinyl
ethyl



2.3.1159
3-ethyl-6-methylphenyl
vinyl
ethyl



2.3.1160
3-cyclopropyl-6-methylphenyl
vinyl
ethyl



2.3.1161
3-cyano-6-methylphenyl
vinyl
ethyl



2.3.1162
3-trifluoromethyl-6-methylphenyl
vinyl
ethyl



2.3.1163
3-methoxy-6-methylphenyl
vinyl
ethyl



2.3.1164
3-ethoxy-6-methylphenyl
vinyl
ethyl



2.3.1165
3-trifluoromethoxy-6-
vinyl
ethyl




methylphenyl





2.3.1166
3-nitro-6-methylphenyl
vinyl
ethyl



2.3.1167
3-fluoro-6-ethylphenyl
vinyl
ethyl



2.3.1168
3-chloro-6-ethylphenyl
vinyl
ethyl



2.3.1169
3-bromo-6-ethylphenyl
vinyl
ethyl



2.3.1170
3-methyl-6-ethylphenyl
vinyl
ethyl



2.3.1171
3,6-diethylphenyl
vinyl
ethyl



2.3.1172
3-cyclopropyl-6-ethylphenyl
vinyl
ethyl



2.3.1173
3-cyano-6-ethylphenyl
vinyl
ethyl



2.3.1174
3-trifluoromethyl-6-ethylphenyl
vinyl
ethyl



2.3.1175
3-methoxy-6-ethylphenyl
vinyl
ethyl



2.3.1176
3-ethoxy-6-ethylphenyl
vinyl
ethyl



2.3.1177
3-trifluoromethoxy-6-ethylphenyl
vinyl
ethyl



2.3.1178
3-nitro-6-ethylphenyl
vinyl
ethyl



2.3.1179
3-fluoro-6-propylphenyl
vinyl
ethyl



2.3.1180
3-chloro-6-propylphenyl
vinyl
ethyl



2.3.1181
3-bromo-6-propylphenyl
vinyl
ethyl



2.3.1182
3-methyl-6-propylphenyl
vinyl
ethyl



2.3.1183
3-cyclopropyl-6-propylphenyl
vinyl
ethyl



2.3.1184
3-cyano-6-propylphenyl
vinyl
ethyl



2.3.1185
3-trifluoromethyl-6-propylphenyl
vinyl
ethyl



2.3.1186
3-methoxy-6-propylphenyl
vinyl
ethyl



2.3.1187
3-ethoxy-6-propylphenyl
vinyl
ethyl



2.3.1188
3-trifluoromethoxy-6-
vinyl
ethyl




propylphenyl





2.3.1189
3-nitro-6-propylphenyl
vinyl
ethyl



2.3.1190
3-fluoro-6-isopropylphenyl
vinyl
ethyl



2.3.1191
3-chloro-6-isopropylphenyl
vinyl
ethyl



2.3.1192
3-bromo-6-isopropylphenyl
vinyl
ethyl



2.3.1193
3-methyl-6-isopropylphenyl
vinyl
ethyl



2.3.1194
3-cyclopropyl-6-isopropylphenyl
vinyl
ethyl



2.3.1195
3-cyano-6-isopropylphenyl
vinyl
ethyl



2.3.1196
3-trifluoromethyl-6-
vinyl
ethyl




isopropylphenyl





2.3.1197
3-methoxy-6-isopropylphenyl
vinyl
ethyl



2.3.1198
3-ethoxy-6-isopropylphenyl
vinyl
ethyl



2.3.1199
3-trifluoromethoxy-6-
vinyl
ethyl




isopropylphenyl





2.3.1200
3-nitro-6-isopropylphenyl
vinyl
ethyl



2.3.1201
3-fluoro-6-tert-butylphenyl
vinyl
ethyl



2.3.1202
3-chloro-6-tert-butylphenyl
vinyl
ethyl



2.3.1203
3-bromo-6-tert-butylphenyl
vinyl
ethyl



2.3.1204
3-methyl-6-tert-butylphenyl
vinyl
ethyl



2.3.1205
3-ethyl-6-tert-butylphenyl
vinyl
ethyl



2.3.1206
3-cyclopropyl-6-tert-butylphenyl
vinyl
ethyl



2.3.1207
3-cyano-6-tert-butylphenyl
vinyl
ethyl



2.3.1208
3-trifluoromethyl-6-tert-
vinyl
ethyl




butylphenyl





2.3.1209
3-methoxy-6-tert-butylphenyl
vinyl
ethyl



2.3.1210
3-ethoxy-6-tert-butylphenyl
vinyl
ethyl



2.3.1211
3-trifluoromethoxy-6-tert-
vinyl
ethyl




butylphenyl





2.3.1212
3-nitro-6-tert-butylphenyl
vinyl
ethyl



2.3.1213
3-fluoro-6-cyclopropylphenyl
vinyl
ethyl



2.3.1214
3-chloro-6-cyclopropylphenyl
vinyl
ethyl



2.3.1215
3-bromo-6-cyclopropylphenyl
vinyl
ethyl



2.3.1216
3-methyl-6-cyclopropylphenyl
vinyl
ethyl



2.3.1217
3-cyclopropyl-6-
vinyl
ethyl




cyclopropylphenyl





2.3.1218
3-cyano-6-cyclopropylphenyl
vinyl
ethyl



2.3.1219
3-trifluoromethyl-6-
vinyl
ethyl




cyclopropylphenyl





2.3.1220
3-methoxy-6-cyclopropylphenyl
vinyl
ethyl



2.3.1221
3-ethoxy-6-cyclopropylphenyl
vinyl
ethyl



2.3.1222
3-trifluoromethoxy-6-
vinyl
ethyl




cyclopropylphenyl





2.3.1223
3-fluoro-6-methoxycarbonyl-
vinyl
ethyl




phenyl





2.3.1224
3-chloro-6-methoxycarbonyl-
vinyl
ethyl




phenyl





2.3.1225
3-bromo-6-methoxycarbonyl-
vinyl
ethyl




phenyl





2.3.1226
3-methyl-6-methoxycarbonyl-
vinyl
ethyl




phenyl





2.3.1227
3-cyclopropyl-6-
vinyl
ethyl




methoxycarbonyl-phenyl





2.3.1228
3-cyano-6-methoxycarbonyl-
vinyl
ethyl




phenyl





2.3.1229
3-trifluoromethyl-6-
vinyl
ethyl




methoxycarbonyl-phenyl





2.3.1230
3-methoxy-6-methoxycarbonyl-
vinyl
ethyl




phenyl





2.3.1231
3-ethoxy-6-methoxycarbonyl-
vinyl
ethyl




phenyl





2.3.1232
3-trifluoromethoxy-6-
vinyl
ethyl




methoxycarbonyl-phenyl





2.3.1233
3-nitro-6-methoxycarbonyl-
vinyl
ethyl




phenyl





2.3.1234
3-fluoro-6-cyanophenyl
vinyl
ethyl



2.3.1235
3-chloro-6-cyanophenyl
vinyl
ethyl



2.3.1236
3-bromo-6-cyanophenyl
vinyl
ethyl



2.3.1237
3-methyl-6-cyanophenyl
vinyl
ethyl



2.3.1238 
3-cyclopropyl-6-cyanophenyl
vinyl
ethyl



2.3.1239
3-cyano-6-cyanophenyl
vinyl
ethyl



2.3.1240
3-trifluoromethyl-6-cyanophenyl
vinyl
ethyl



2.3.1241
3-methoxy-6-cyanophenyl
vinyl
ethyl



2.3.1242
3-ethoxy-6-cyanophenyl
vinyl
ethyl



2.3.1243
3-trifluoromethoxy-6-
vinyl
ethyl




cyanophenyl





2.3.1244
3-nitro-6-cyanophenyl
vinyl
ethyl



2.3.1245
3-fluoro-6-methoxyphenyl
vinyl
ethyl



2.3.1246
3-chloro-6-methoxyphenyl
vinyl
ethyl



2.3.1247
3-bromo-6-methoxyphenyl
vinyl
ethyl



2.3.1248
3-methyl-6-methoxyphenyl
vinyl
ethyl



2.3.1249
3-cyclopropyl-6-methoxyphenyl
vinyl
ethyl



2.3.1250
3-cyano-6-methoxyphenyl
vinyl
ethyl



2.3.1251
3-trifluoromethyl-6-
vinyl
ethyl




methoxyphenyl





2.3.1252
3,6-dimethoxyphenyl
vinyl
ethyl



2.3.1253
3-ethoxy-6-methoxyphenyl
vinyl
ethyl



2.3.1254
3-trifluoromethoxy-6-
vinyl
ethyl




methoxyphenyl





2.3.1255
3-nitro-6-methoxyphenyl
vinyl
ethyl



2.3.1256
3-fluoro-6-ethoxyphenyl
vinyl
ethyl



2.3.1257
3-chloro-6-ethoxyphenyl
vinyl
ethyl



2.3.1258
3-bromo-6-ethoxyphenyl
vinyl
ethyl



2.3.1259
3-methyl-6-ethoxyphenyl
vinyl
ethyl



2.3.1260
3-cyclopropyl-6-ethoxyphenyl
vinyl
ethyl



2.3.1261
3-cyano-6-ethoxyphenyl
vinyl
ethyl



2.3.1262
3-trifluoromethyl-6-ethoxyphenyl
vinyl
ethyl



2.3.1263
3-methoxy-6-ethoxyphenyl
vinyl
ethyl



2.3.1264
2,6-diethoxyphenyl
vinyl
ethyl



2.3.1265
3-trifluoromethoxy-6-
vinyl
ethyl




ethoxyphenyl





2.3.1266
3-nitro-6-ethoxyphenyl
vinyl
ethyl



2.3.1267
3-fluoro-6-isopropoxyphenyl
vinyl
ethyl



2.3.1268
3-chloro-6-isopropoxyphenyl
vinyl
ethyl



2.3.1269
3-bromo-6-isopropoxyphenyl
vinyl
ethyl



2.3.1270
3-methyl-6-isopropoxyphenyl
vinyl
ethyl



2.3.1271
3-cyclopropyl-6-
vinyl
ethyl




isopropoxyphenyl





2.3.1272
3-cyano-6-isopropoxyphenyl
vinyl
ethyl



2.3.1273
3-trifluoromethyl-6-
vinyl
ethyl




isopropoxyphenyl





2.3.1274
3-methoxy-6-isopropoxyphenyl
vinyl
ethyl



2.3.1275
3-ethoxy-6-isopropoxyphenyl
vinyl
ethyl



2.3.1276
3-trifluoromethoxy-6-
vinyl
ethyl




isopropoxyphenyl





2.3.1277
3-nitro-6-isopropoxyphenyl
vinyl
ethyl



2.3.1278
3-fluoro-6-trifluoromethoxy-
vinyl
ethyl




phenyl





2.3.1279
3-chloro-6-trifluoromethoxy-
vinyl
ethyl




phenyl





2.3.1280
3-bromo-6-trifluoromethoxy-
vinyl
ethyl




phenyl





2.3.1281
3-methyl-6-trifluoromethoxy-
vinyl
ethyl




phenyl





2.3.1282
3-cyclopropyl-6-
vinyl
ethyl




trifluoromethoxyphenyl





2.3.1283
3-cyano-6-trifluoromethoxy-
vinyl
ethyl




phenyl





2.3.1284
3-trifluoromethyl-6-
vinyl
ethyl




trifluoromethoxyphenyl





2.3.1285
3-methoxy-6-trifluoromethoxy-
vinyl
ethyl




phenyl





2.3.1286
3-ethoxy-6-trifluoromethoxy-
vinyl
ethyl




phenyl





2.3.1287
3,6-bis(trifluoro-methoxy)phenyl
vinyl
ethyl



2.3.1288
3-nitro-6-trifluoromethoxyphenyl
vinyl
ethyl



2.3.1289
3-fluoro-6-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.1290
3-chloro-6-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.1291
3-bromo-6-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.1292
3-methyl-6-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.1293
3-cyclopropyl-6-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.1294
3-cyano-6-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.1295
3-trifluoromethyl-6-
vinyl
ethyl




difluoromethoxyphenyl





2.3.1296
3-methoxy-6-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.1297
3-ethoxy-6-difluoromethoxy-
vinyl
ethyl




phenyl





2.3.1298
3-trifluoromethoxy-6-
vinyl
ethyl




difluoromethoxyphenyl





2.3.1299 
3-nitro-6-difluoromethoxyphenyl
vinyl
ethyl



2.3.1300
3-fluoro-6-nitrophenyl
vinyl
ethyl



2.3.1301
3-chloro-6-nitrophenyl
vinyl
ethyl



2.3.1302
3-bromo-6-nitrophenyl
vinyl
ethyl



2.3.1303
3-methyl-6-nitrophenyl
vinyl
ethyl



2.3.1304
3-cyclopropyl-6-nitrophenyl
vinyl
ethyl



2.3.1305
3-cyano-6-nitrophenyl
vinyl
ethyl



2.3.1306
3-trifluoromethyl-6-nitrophenyl
vinyl
ethyl



2.3.1307
3-methoxy-6-nitrophenyl
vinyl
ethyl



2.3.1308
3-ethoxy-6-nitrophenyl
vinyl
ethyl



2.3.1309
3-trifluoromethoxy-6-nitrophenyl
vinyl
ethyl



2.3.1310
3-fluoro-6-methylsulfanylphenyl
vinyl
ethyl



2.3.1311
3-chloro-6-methylsulfanylphenyl
vinyl
ethyl



2.3.1312
3-bromo-6-methylsulfanylphenyl
vinyl
ethyl



2.3.1313
3-methyl-6-methylsulfanylphenyl
vinyl
ethyl



2.3.1314
3-cyclopropyl-6-
vinyl
ethyl




methylsulfanylphenyl





2.3.1315
3-cyano-6-methylsulfanylphenyl
vinyl
ethyl



2.3.1316
3-trifluoromethyl-6-
vinyl
ethyl




methylsulfanylphenyl





2.3.1317
3-methoxy-6-
vinyl
ethyl




methylsulfanylphenyl





2.3.1318
3-ethoxy-6-methylsulfanylphenyl
vinyl
ethyl



2.3.1319
3-trifluoromethoxy-6-
vinyl
ethyl




methylsulfanylphenyl





2.3.1320
3-nitro-6-methylsulfanylphenyl
vinyl
ethyl



2.3.1321
2,3,4-trifluorophenyl
vinyl
ethyl



2.3.1322
2,3,4-trichlorophenyl
vinyl
ethyl



2.3.1323
2,3,4-trimethylphenyl
vinyl
ethyl



2.3.1324
2-fluoro-2-chloro-5-
vinyl
ethyl




trifluoromethylphenyl





2.3.1325
2,3,5-trifluorophenyl
vinyl
ethyl



2.3.1326
2,3,5-trichlorophenyl
vinyl
ethyl



2.3.1327
2,3,5-trimethylphenyl
vinyl
ethyl



2.3.1328
2,3-dichloro-5-methoxyphenyl
vinyl
ethyl



2.3.1329
2,3,6-trifluorophenyl
vinyl
ethyl



2.3.1330
2,3,6-trichlorophenyl
vinyl
ethyl



2.3.1331
2,3,6-trimethylphenyl
vinyl
ethyl



2.3.1332
3,4,5-trifluorophenyl
vinyl
ethyl



2.3.1333
3,4,5-trichlorophenyl
vinyl
ethyl



2.3.1334
3,4,5-trimethylphenyl
vinyl
ethyl



2.3.1335
3,5-dimethyl-4-fluorophenyl
vinyl
ethyl



2.3.1336
3,5-dichloro-4-methoxyphenyl
vinyl
ethyl



2.3.1337
3,5-difluoro-4-chlorophenyl
vinyl
ethyl



2.3.1338
3,5-dichloro-4-hydroxyphenyl
vinyl
ethyl



2.3.1339
3,5-trifluoromethyl-4-
vinyl
ethyl




chlorophenyl





2.3.1340
3,4,6-trifluorophenyl
vinyl
ethyl



2.3.1341
3,4,6-trichlorophenyl
vinyl
ethyl



2.3.1342
3,4,6-trimethylphenyl
vinyl
ethyl



2.3.1343
pentafluorophenyl
vinyl
ethyl
















TABLE 2.4







Inventive compounds of the general formula (I) in which W* is COOY, R1


and R2 are each hydrogen, and aryl is the radical.








 








 











No.
Aryl
Alkyl
Y
Physical data





2.4.1
3-fluorophenyl
methyl
methyl
[CDCl3] 2.44 (s, 3H); 3.87






(s, 3H); 3.87 (AB, 2H);






7.12-7.20 (m, 1H); 7.38-






7.43 (m, 3H).


2.4.2
3-fluorophenyl
ethyl
ethyl



2.4.3
3-fluorophenyl
propyl
ethyl



2.4.4
3-fluorophenyl
butyl
ethyl



2.4.5
3-chlorophenyl
methyl
ethyl



2.4.6
3-chlorophenyl
ethyl
ethyl



2.4.7
3-chlorophenyl
propyl
ethyl



2.4.8
3-chlorophenyl
butyl
ethyl



2.4.9
3-bromophenyl
methyl
ethyl



2.4.10
3-bromophenyl
ethyl
ethyl



2.4.11
3-iodophenyl
methyl
ethyl



2.4.12
3-iodophenyl
ethyl
ethyl



2.4.13
3-methylphenyl
methyl
ethyl



2.4.14
3-methylphenyl
ethyl
ethyl



2.4.15
3-ethylphenyl
methyl
ethyl



2.4.16
3-propylphenyl
methyl
ethyl



2.4.17
3-isopropylphenyl
methyl
ethyl



2.4.18
3-n-butylphenyl
methyl
ethyl



2.4.19
3-i-butylphenyl
methyl
ethyl



2.4.20
3-tert-butylphenyl
methyl
ethyl



2.4.21
3-cyclopropylphenyl
methyl
ethyl



2.4.22
3-cyclobutylphenyl
methyl
ethyl



2.4.23
3-cyclopentylphenyl
methyl
ethyl



2.4.24
3-vinylphenyl
methyl
ethyl



2.4.25
3-ethynylphenyl
methyl
ethyl



2.4.26
3-cyanophenyl
methyl
ethyl



2.4.27
3-trifluoromethylphenyl
methyl
ethyl



2.4.28
3-difluoromethylphenyl
methyl
ethyl



2.4.29
3-(hydroxycarbonyl)-phenyl
methyl
ethyl



2.4.30
3-(methoxycarbonyl)-phenyl
methyl
ethyl



2.4.31
3-(ethoxycarbonyl)-phenyl
methyl
ethyl



2.4.32
3-hydroxymethylphenyl
methyl
ethyl



2.4.33
3-carbamoylphenyl
methyl
ethyl



2.4.34
3-hydroxyphenyl
methyl
ethyl



2.4.35
3-methoxyphenyl
methyl
ethyl



2.4.36
3-ethoxyphenyl
methyl
ethyl



2.4.37
3-propyloxyphenyl
methyl
ethyl



2.4.38
3-isopropyloxyphenyl
methyl
ethyl



2.4.39
3-n-butyloxyphenyl
methyl
ethyl



2.4.40
3-i-butyloxyphenyl
methyl
ethyl



2.4.41
3-t-butyloxyphenyl
methyl
ethyl



2.4.42
3-difluoromethoxyphenyl
methyl
ethyl



2.4.43
3-trifluoromethoxyphenyl
methyl
ethyl



2.4.44
3-(2,2,2-trifluoroethoxy)phenyl 
methyl
ethyl



2.4.45
3-(2-chloroethoxy)phenyl
methyl
ethyl



2.4.46
3-(2-hydroxyethoxy)phenyl
methyl
ethyl



2.4.47
3-(2-methoxyethoxy)phenyl
methyl
ethyl



2.4.48
3-[(tert-butoxycarbonyl)oxy]phenyl
methyl
ethyl



2.4.49
3-nitrophenyl
methyl
ethyl



2.4.50
3-acetoxyphenyl
methyl
ethyl



2.4.51
{3-[(tert-butoxycarbonyl)amino]-
methyl
ethyl




phenyl}





2.4.52
3-methylsulfanylphenyl
methyl
ethyl



2.4.53
3-ethylsulfanylphenyl
methyl
ethyl



2.4.54
3-(pentafluoro-lambda6-sulfanyl)-
methyl
ethyl




phenyl





2.4.55
2,3-difluorophenyl
methyl
ethyl



2.4.56
2,3-difluorophenyl
ethyl
ethyl



2.4.57
2,3-difluorophenyl
propyl
ethyl



2.4.58
2,3-difluorophenyl
butyl
ethyl



2.4.59
2-chloro-3-fluorophenyl
methyl
ethyl



2.4.60
2-bromo-3-fluorophenyl
methyl
ethyl



2.4.61
2-methyl-3-fluorophenyl
methyl
ethyl



2.4.62
2-ethyl-3-fluorophenyl
methyl
ethyl



2.4.63
2-cyclopropyl-3-fluorophenyl
methyl
ethyl



2.4.64
2-vinyl-3-fluorophenyl
methyl
ethyl



2.4.65
2-ethynyl-3-fluorophenyl
methyl
ethyl



2.4.66
2-cyano-3-fluorophenyl
methyl
ethyl



2.4.67
2-methoxy-3-fluorophenyl
methyl
ethyl



2.4.68
2-ethoxy-3-fluorophenyl
methyl
ethyl



2.4.69
2-trifluoromethoxy-3-fluorophenyl 
methyl
ethyl



2.4.70
2-nitro-3-fluorophenyl
methyl
ethyl



2.4.71
2-fluoro-3-chlorophenyl
methyl
ethyl



2.4.72
2,3-dichlorophenyl
methyl
ethyl



2.4.73
2,3-dichlorophenyl
ethyl
ethyl



2.4.74
2,3-dichlorophenyl
propyl
ethyl



2.4.75
2,3-dichlorophenyl
butyl
ethyl



2.4.76
2-bromo-3-chlorophenyl
methyl
ethyl



2.4.77
2-methyl-3-chlorophenyl
methyl
ethyl



2.4.78
2-ethyl-3-chlorophenyl
methyl
ethyl



2.4.79
2-cyclopropyl-3-chlorophenyl
methyl
ethyl



2.4.80
2-vinyl-3-chlorophenyl
methyl
ethyl



2.4.81
2-ethynyl-3-chlorophenyl
methyl
ethyl



2.4.82
2-cyano-3-chlorophenyl
methyl
ethyl



2.4.83
2-trifluoromethyl-2-chlorophenyl 
methyl
ethyl



2.4.84
2-methoxy-3-chlorophenyl
methyl
ethyl



2.4.85
2-ethoxy-3-chlorophenyl
methyl
ethyl



2.4.86
2-trifluoromethoxy-3-chlorophenyl
methyl
ethyl



2.4.87
2-nitro-3-chlorophenyl
methyl
ethyl



2.4.88
2-fluoro-3-bromophenyl
methyl
ethyl



2.4.89
2-chloro-3-bromophenyl
methyl
ethyl



2.4.90
2,3-dibromophenyl
methyl
ethyl



2.4.91
2-methyl-3-bromophenyl
methyl
ethyl



2.4.92
2-ethyl-3-bromophenyl
methyl
ethyl



2.4.93
2-cyclopropyl-3-bromophenyl
methyl
ethyl



2.4.94
2-vinyl-3-bromophenyl
methyl
ethyl



2.4.95
2-ethynyl-3-bromophenyl
methyl
ethyl



2.4.96
2-cyano-3-bromophenyl
methyl
ethyl



2.4.97
2-trifluoromethyl-3-bromophenyl 
methyl
ethyl



2.4.98
2-methoxy-3-phenyl
methyl
ethyl



2.4.99
2-ethoxy-3-bromophenyl
methyl
ethyl



2.4.100
2-trifluoromethoxy-3-bromophenyl
methyl
ethyl



2.4.101
2-nitro-3-bromophenyl
methyl
ethyl



2.4.102
2-fluoro-3-iodophenyl
methyl
ethyl



2.4.103
2-chloro-3-iodophenyl
methyl
ethyl



2.4.104
2-bromo-3-iodophenyl
methyl
ethyl



2.4.105
2-methyl-3-iodophenyl
methyl
ethyl



2.4.106
2-ethyl-3-iodophenyl
methyl
ethyl



2.4.107
2-cyclopropyl-3-iodophenyl
methyl
ethyl



2.4.108
2-vinyl-3-iodophenyl
methyl
ethyl



2.4.109
2-ethynyl-3-iodophenyl
methyl
ethyl



2.4.110
2-cyano-3-iodophenyl
methyl
ethyl



2.4.111
2-trifluoromethyl-3-iodophenyl
methyl
ethyl



2.4.112
2-methoxy-3-iodophenyl
methyl
ethyl



2.4.113
2-ethoxy-3-iodophenyl
methyl
ethyl



2.4.114
2-trifluoromethoxy-3-iodophenyl
methyl
ethyl



2.4.115
2-nitro-3- iodophenyl
methyl
ethyl



2.4.116
2-fluoro-3-methylphenyl
methyl
ethyl



2.4.117
2-fluoro-3-methylphenyl
ethyl
ethyl



2.4.118
2-fluoro-3-methylphenyl
propyl
ethyl



2.4.119
2-fluoro-3-methylphenyl
butyl
ethyl



2.4.120
2-chloro-3-methylphenyl
methyl
ethyl



2.4.121
2-chloro-3-methylphenyl
ethyl
ethyl



2.4.122
2-chloro-3-methylphenyl
propyl
ethyl



2.4.123
2-chloro-3-methylphenyl
butyl
ethyl



2.4.124
2-bromo-3-methylphenyl
methyl
ethyl



2.4.125
2,3-dimethylphenyl
methyl
ethyl



2.4.126
2,3-dimethylphenyl
ethyl
ethyl



2.4.127
2,3-dimethylphenyl
propyl
ethyl



2.4.128
2,3-dimethylphenyl
butyl
ethyl



2.4.129
2-ethyl-3-methylphenyl
methyl
ethyl



2.4.130
2-cyclopropyl-3-methylphenyl
methyl
ethyl



2.4.131
2-vinyl-3-methylphenyl
methyl
ethyl



2.4.132
2-ethynyl-3-methylphenyl
methyl
ethyl



2.4.133
2-cyano-3-methylphenyl
methyl
ethyl



2.4.134
2-trifluoromethyl-3-methylphenyl
methyl
ethyl



2.4.135
2-methoxy-3-methylphenyl
methyl
ethyl



2.4.136
2-ethoxy-3-methylphenyl
methyl
ethyl



2.4.137
2-trifluoromethoxy-3-methylphenyl
methyl
ethyl



2.4.138
2-nitro-3-methylphenyl
methyl
ethyl



2.4.139
2-fluoro-3-ethylphenyl
methyl
ethyl



2.4.140
2-chloro-3-ethylphenyl
methyl
ethyl



2.4.141
2-bromo-3-ethylphenyl
methyl
ethyl



2.4.142
2-methyl-3-ethylphenyl
methyl
ethyl



2.4.143
2,3-diethylphenyl
methyl
ethyl



2.4.144
2-cyclopropyl-3-ethylphenyl
methyl
ethyl



2.4.145
2-vinyl-3-ethylphenyl
methyl
ethyl



2.4.146
2-ethynyl-3-ethylphenyl
methyl
ethyl



2.4.147
2-cyano-3-ethylphenyl
methyl
ethyl



2.4.148
2-trifluoromethyl-3-ethylphenyl
methyl
ethyl



2.4.149
2-methoxy-3-ethylphenyl
methyl
ethyl



2.4.150
2-ethoxy-3-ethylphenyl
methyl
ethyl



2.4.151
2-trifluoromethoxy-3-ethylphenyl
methyl
ethyl



2.4.152
2-nitro-3-ethylphenyl
methyl
ethyl



2.4.153
2-fluoro-3-propylphenyl
methyl
ethyl



2.4.154
2-chloro-3-propylphenyl
methyl
ethyl



2.4.155
2-bromo-3-propylphenyl
methyl
ethyl



2.4.156
2-methyl-3-propylphenyl
methyl
ethyl



2.4.157
2-methyl-3-propylphenyl
methyl
ethyl



2.4.158
2-cyclopropyl-3-propylphenyl
methyl
ethyl



2.4.159
2-vinyl-3-propylphenyl
methyl
ethyl



2.4.160
2-ethynyl-3propylphenyl
methyl
ethyl



2.4.161
2-cyano-3-propylphenyl
methyl
ethyl



2.4.162
2-trifluoromethyl-3-propylphenyl
methyl
ethyl



2.4.163
2-methoxy-3-propylphenyl
methyl
ethyl



2.4.164
2-ethoxy-3-propylphenyl
methyl
ethyl



2.4.165
2-trifluoromethoxy-3-propylphenyl
methyl
ethyl



2.4.166
2-nitro-3-propylphenyl
methyl
ethyl



2.4.167
2-fluoro-3-isopropylphenyl
methyl
ethyl



2.4.168
2-chloro-3-isopropylphenyl
methyl
ethyl



2.4.169
2-bromo-3-isopropylphenyl
methyl
ethyl



2.4.170
2-methyl-3-isopropylphenyl
methyl
ethyl



2.4.171
2-ethyl-3-isopropylphenyl
methyl
ethyl



2.4.172
2-cyclopropyl-3-isopropylphenyl
methyl
ethyl



2.4.173
2-vinyl-3-isopropylphenyl
methyl
ethyl



2.4.174
2-ethynyl-3-isopropylphenyl
methyl
ethyl



2.4.175
2-cyano-3-isopropylphenyl
methyl
ethyl



2.4.176
2-trifluoromethyl-3-isopropylphenyl
methyl
ethyl



2.4.177
2-methoxy-3-isopropylphenyl
methyl
ethyl



2.4.178
2-ethoxy-3-isopropylphenyl
methyl
ethyl



2.4.179
2-trifluoromethoxy-3-
methyl
ethyl




isopropylphenyl





2.4.180
2-nitro-3-isopropylphenyl
methyl
ethyl



2.4.181
2-fluoro-3-tert-butylphenyl
methyl
ethyl



2.4.182
2-chloro-3-tert-butylphenyl
methyl
ethyl



2.4.183
2-bromo-3-tert-butylphenyl
methyl
ethyl



2.4.184
2-methyl-3-tert-butylphenyl
methyl
ethyl



2.4.185
2-ethyl-3-tert-butylphenyl
methyl
ethyl



2.4.186
2-cyclopropyl-3-tert-butylphenyl
methyl
ethyl



2.4.187
2-vinyl-3-tert-butylphenyl
methyl
ethyl



2.4.188
2-ethynyl-3-tert-butylphenyl
methyl
ethyl



2.4.189
2-cyano-3-tert-butylphenyl
methyl
ethyl



2.4.190
2-trifluoromethyl-3-tert-butylphenyl
methyl
ethyl



2.4.191
2-methoxy-3-tert-butylphenyl
methyl
ethyl



2.4.192
2-ethoxy-3-tert-butylphenyl
methyl
ethyl



2.4.193
2-trifluoromethoxy-3-tert-
methyl
ethyl




butylphenyl





2.4.194
2-nitro-3-tert-butylphenyl
methyl
ethyl



2.4.195
2-fluoro-3-hydroxymethylphenyl
methyl
ethyl



2.4.196
2-chloro-3-hydroxymethylphenyl
methyl
ethyl



2.4.197
2-bromo-3-hydroxymethylphenyl
methyl
ethyl



2.4.198
2-methyl-3-hydroxymethylphenyl
methyl
ethyl



2.4.199
2-ethyl-3-hydroxymethylphenyl
methyl
ethyl



2.4.200
2-cyclopropyl-3-
methyl
ethyl




hydroxymethylphenyl





2.4.201
2-vinyl-3-hydroxymethylphenyl
methyl
ethyl



2.4.202
2-ethynyl-3-hydroxymethylphenyl
methyl
ethyl



2.4.203
2-cyano-3-hydroxymethylphenyl
methyl
ethyl



2.4.204
2-trifluoromethyl-3-
methyl
ethyl




hydroxymethylphenyl





2.4.205
2-methoxy-3-hydroxymethylphenyl
methyl
ethyl



2.4.206
2-ethoxy-3-hydroxymethylphenyl
methyl
ethyl



2.4.207
2-trifluoromethoxy-3-
methyl
ethyl




hydroxymethylphenyl





2.4.208
2-nitro-3-hydroxymethylphenyl
methyl
ethyl



2.4.209
2-fluoro-3-cyclopropylphenyl
methyl
ethyl



2.4.210
2-chloro-3-cyclopropylphenyl
methyl
ethyl



2.4.211
2-bromo-3-cyclopropylphenyl
methyl
ethyl



2.4.212
2-methyl-3-cyclopropylphenyl
methyl
ethyl



2.4.213
2-ethyl-3-cyclopropylphenyl
methyl
ethyl



2.4.214
2-cyclopropyl-3-cyclopropylphenyl
methyl
ethyl



2.4.215
2-vinyl-3-cyclopropylphenyl
methyl
ethyl



2.4.216
2-ethynyl-3-cyclopropylphenyl
methyl
ethyl



2.4.217
2-cyano-3-cyclopropylphenyl
methyl
ethyl



2.4.218
2-trifluoromethyl-3-
methyl
ethyl




cyclopropylphenyl





2.4.219
2-methoxy-3-cyclopropylphenyl
methyl
ethyl



2.4.220
2-ethoxy-3-cyclopropylphenyl
methyl
ethyl



2.4.221
2-trifluoromethoxy-3-
methyl
ethyl




cyclopropylphenyl





2.4.222
2-fluoro-3-methoxycarbonylphenyl
methyl
ethyl



2.4.223
2-chloro-3-methoxycarbonylphenyl
methyl
ethyl



2.4.224
2-bromo-3-methoxycarbonylphenyl
methyl
ethyl



2.4.225
2-methyl-3-methoxycarbonylphenyl
methyl
ethyl



2.4.226
2-ethyl-3-methoxycarbonylphenyl
methyl
ethyl



2.4.227
2-cyclopropyl-3-methoxycarbonyl- 
methyl
ethyl




phenyl





2.4.228
2-vinyl-3-methoxycarbonylphenyl
methyl
ethyl



2.4.229
2-ethynyl-3-methoxycarbonyl-
methyl
ethyl




phenyl





2.4.230
2-cyano-3-methoxycarbonylphenyl
methyl
ethyl



2.4.231
2-trifluoromethyl-3-
methyl
ethyl




methoxycarbonylphenyl





2.4.232
2-methoxy-3-methoxycarbonyl-
methyl
ethyl




phenyl





2.4.233
2-ethoxy-3-methoxycarbonylphenyl
methyl
ethyl



2.4.234
2-trifluoromethoxy-3-
methyl
ethyl




methoxycarbonylphenyl





2.4.235
2-nitro-3-methoxycarbonylphenyl
methyl
ethyl



2.4.236
2-fluoro-3-vinylphenyl
methyl
ethyl



2.4.237
2-chloro-3-vinylphenyl
methyl
ethyl



2.4.238
2-bromo-3-vinylphenyl
methyl
ethyl



2.4.239
2-methyl-3-vinylphenyl
methyl
ethyl



2.4.240
2-ethyl-3-vinylphenyl
methyl
ethyl



2.4.241
2-cyclopropyl-3-vinylphenyl
methyl
ethyl



2.4.242
2-vinyl-3-vinylphenyl
methyl
ethyl



2.4.243
2-ethynyl-3-vinylphenyl
methyl
ethyl



2.4.244
2-cyano-3-vinylphenyl
methyl
ethyl



2.4.245
2-trifluoromethyl-3-vinylphenyl
methyl
ethyl



2.4.246
2-methoxy-3-vinylphenyl
methyl
ethyl



2.4.247
2-ethoxy-3-vinylphenyl
methyl
ethyl



2.4.248
2-trifluoromethoxy-3-vinylphenyl
methyl
ethyl



2.4.249
2-nitro-3-vinylphenyl
methyl
ethyl



2.4.250
2-fluoro-3-ethynylphenyl
methyl
ethyl



2.4.251
2-chloro-3-ethynylphenyl
methyl
ethyl



2.4.252
2-bromo-3-ethynylphenyl
methyl
ethyl



2.4.253
2-methyl-3-ethynylphenyl
methyl
ethyl



2.4.254
2-ethyl-3-ethynylphenyl
methyl
ethyl



2.4.255
2-cyclopropyl-3-ethynylphenyl
methyl
ethyl



2.4.256
2-vinyl-3-ethynylphenyl
methyl
ethyl



2.4.257
2-cyano-3-ethynylphenyl
methyl
ethyl



2.4.258
2-trifluoromethyl-3-ethynylphenyl
methyl
ethyl



2.4.259
2-methoxy-3-ethynylphenyl
methyl
ethyl



2.4.260
2-ethoxy-3-ethynylphenyl
methyl
ethyl



2.4.261
2-trifluoromethoxy-3-ethynylphenyl
methyl
ethyl



2.4.262
2-nitro-3-ethynylphenyl
methyl
ethyl



2.4.263
2-fluoro-3-ethynylphenyl
methyl
ethyl



2.4.264
2-fluoro-3-cyanophenyl
methyl
ethyl



2.4.265
2-chloro-3-cyanophenyl
methyl
ethyl



2.4.266
2-bromo-3-cyanophenyl
methyl
ethyl



2.4.267
2-methyl-3-cyanophenyl
methyl
ethyl



2.4.268
2-ethyl-3-cyanophenyl
methyl
ethyl



2.4.269
2-ethyl-3-cyanophenyl
ethyl
ethyl



2.4.270
2-ethyl-3-cyanophenyl
propyl
ethyl



2.4.271
2-ethyl-3-cyanophenyl
butyl
ethyl



2.4.272
2-cyclopropyl-3-cyanophenyl
methyl
ethyl



2.4.273
2-vinyl-3-cyanophenyl
methyl
ethyl



2.4.274
2-ethynyl-3-cyanophenyl
methyl
ethyl



2.4.275
2-cyano-3-cyanophenyl
methyl
ethyl



2.4.276
2-trifluoromethyl-3-cyanophenyl
methyl
ethyl



2.4.277
2-methoxy-3-cyanophenyl
methyl
ethyl



2.4.278
2-ethoxy-3-cyanophenyl
methyl
ethyl



2.4.279
2-trifluoromethoxy-3-cyanophenyl
methyl
ethyl



2.4.280
2-nitro-3-cyanophenyl
methyl
ethyl



2.4.281
2-fluoro-3-hydroxyphenyl
methyl
ethyl



2.4.282
2-chloro-3-hydroxyphenyl
methyl
ethyl



2.4.283
2-bromo-3-hydroxyphenyl
methyl
ethyl



2.4.284
2-methyl-3-hydroxyphenyl
methyl
ethyl



2.4.285
2-ethyl-3-hydroxyphenyl
methyl
ethyl



2.4.286
2-cyclopropyl-3-hydroxyphenyl
methyl
ethyl



2.4.287
2-vinyl-3-hydroxyphenyl
methyl
ethyl



2.4.288
2-ethynyl-3-hydroxyphenyl
methyl
ethyl



2.4.289
2-cyano-3-hydroxyphenyl
methyl
ethyl



2.4.290
2-trifluoromethyl-3-hydroxyphenyl
methyl
ethyl



2.4.291
2-methoxy-3-hydroxyphenyl
methyl
ethyl



2.4.292
2-ethoxy-3-hydroxyphenyl
methyl
ethyl



2.4.293
2-trifluoromethoxy-3-hydroxyphenyl
methyl
ethyl



2.4.294
2-nitro-3-hydroxyphenyl
methyl
ethyl



2.4.295
2-fluoro-3-methoxyphenyl
methyl
ethyl



2.4.296
2-chloro-3-methoxyphenyl
methyl
ethyl



2.4.297
2-bromo-3-methoxyphenyl
methyl
ethyl



2.4.298
2-methyl-3-methoxyphenyl
methyl
ethyl



2.4.299
2-ethyl-3-methoxyphenyl
methyl
ethyl



2.4.300
2-cyclopropyl-3-methoxyphenyl
methyl
ethyl



2.4.301
2-vinyl-3-methoxyphenyl
methyl
ethyl



2.4.302
2-ethynyl-3-methoxyphenyl
methyl
ethyl



2.4.303
2-cyano-3-methoxyphenyl
methyl
ethyl



2.4.304
2-trifluoromethyl-3-methoxyphenyl
methyl
ethyl



2.4.305
2,3-dimethoxyphenyl
methyl
ethyl



2.4.306
2-ethoxy-3-methoxyphenyl
methyl
ethyl



2.4.307
2-trifluoromethoxy-3-
methyl
ethyl




methoxyphenyl





2.4.308
2-nitro-3-methoxyphenyl
methyl
ethyl



2.4.309
2-fluoro-3-ethoxyphenyl
methyl
ethyl



2.4.310
2-chloro-3-ethoxyphenyl
methyl
ethyl



2.4.311
2-bromo-3-ethoxyphenyl
methyl
ethyl



2.4.312
2-methyl-3-ethoxyphenyl
methyl
ethyl



2.4.313
2-ethyl-3-ethoxyphenyl
methyl
ethyl



2.4.314
2-cyclopropyl-3-ethoxyphenyl
methyl
ethyl



2.4.315
2-vinyl-3-ethoxyphenyl
methyl
ethyl



2.4.316
2-ethynyl-3-ethoxyphenyl
methyl
ethyl



2.4.317
2-cyano-3-ethoxyphenyl
methyl
ethyl



2.4.318
2-trifluoromethyl-3-ethoxyphenyl 
methyl
ethyl



2.4.319
2-methoxy-3-ethoxyphenyl
methyl
ethyl



2.4.320
2,3-diethoxy--phenyl
methyl
ethyl



2.4.321
2-trifluoromethoxy-3-ethoxyphenyl
methyl
ethyl



2.4.322
2-nitro-3-ethoxyphenyl
methyl
ethyl



2.4.323
2-fluoro-3-propoxyphenyl
methyl
ethyl



2.4.324
2-chloro-3-propoxyphenyl
methyl
ethyl



2.4.325
2-bromo-3-propoxyphenyl
methyl
ethyl



2.4.326
2-methyl-3-propoxyphenyl
methyl
ethyl



2.4.327
2-ethyl-3-propoxyphenyl
methyl
ethyl



2.4.328
2-cyclopropyl-3-propoxyphenyl
methyl
ethyl



2.4.329
2-vinyl-3-propoxyphenyl
methyl
ethyl



2.4.330
2-ethynyl-3-propoxyphenyl
methyl
ethyl



2.4.331
2-cyano-3-propoxyphenyl
methyl
ethyl



2.4.332
2-trifluoromethyl-3-propoxyphenyl
methyl
ethyl



2.4.333
2-methoxy-3-propoxyphenyl
methyl
ethyl



2.4.334
2-ethoxy-3-propoxyphenyl
methyl
ethyl



2.4.335
2-trifluoromethoxy-3-propoxyphenyl
methyl
ethyl



2.4.336
2-nitro-3-propoxyphenyl
methyl
ethyl



2.4.337
2-fluoro-3-isopropoxyphenyl
methyl
ethyl



2.4.338
2-chloro-3-isopropoxyphenyl
methyl
ethyl



2.4.339
2-bromo-3-isopropoxyphenyl
methyl
ethyl



2.4.340
2-methyl-3-isopropoxyphenyl
methyl
ethyl



2.4.341
2-ethyl-3-isopropoxyphenyl
methyl
ethyl



2.4.342
2-cyclopropyl-3-isopropoxyphenyl
methyl
ethyl



2.4.343
2-vinyl-3-isopropoxyphenyl
methyl
ethyl



2.4.344
2-ethynyl-3-isopropoxyphenyl
methyl
ethyl



2.4.345
2-cyano-3-isopropoxyphenyl
methyl
ethyl



2.4.346
2-trifluoromethyl-3-
methyl
ethyl




isopropoxyphenyl





2.4.347
2-methoxy-3-isopropoxyphenyl
methyl
ethyl



2.4.348
2-ethoxy-3-isopropoxyphenyl
methyl
ethyl



2.4.349
2-trifluoromethoxy-3-
methyl
ethyl




isopropoxyphenyl





2.4.350
2-nitro-3-isopropoxyphenyl
methyl
ethyl



2.4.351
2-fluoro-3-tert-butoxyphenyl
methyl
ethyl



2.4.352
2-chloro-3-tert-butoxyphenyl
methyl
ethyl



2.4.353
2-bromo-3-tert-butoxyphenyl
methyl
ethyl



2.4.354
2-methyl-3-tert-butoxyphenyl
methyl
ethyl



2.4.355
2-ethyl-3-tert-butoxyphenyl
methyl
ethyl



2.4.356
2-cyclopropyl-3-tert-butoxyphenyl
methyl
ethyl



2.4.357
2-vinyl-3-tert-butoxyphenyl
methyl
ethyl



2.4.358
2-ethynyl-3-tert-butoxyphenyl
methyl
ethyl



2.4.359
2-cyano-3-tert-butoxyphenyl
methyl
ethyl



2.4.360
2-trifluoromethyl-3-tert-
methyl
ethyl




butoxyphenyl





2.4.361
2-methoxy-3-tert-butoxyphenyl
methyl
ethyl



2.4.362
2-ethoxy-3-tert-butoxyphenyl
methyl
ethyl



2.4.363
2-trifluoromethoxy-3-tert-
methyl
ethyl




butoxyphenyl





2.4.364
2-nitro-3-tert-butoxyphenyl
methyl
ethyl



2.4.365
2-fluoro-3-trifluoromethoxyphenyl
methyl
ethyl



2.4.366
2-chloro-3-trifluoromethoxyphenyl
methyl
ethyl



2.4.367
2-bromo-3-trifluoromethoxyphenyl
methyl
ethyl



2.4.368
2-methyl-3-trifluoromethoxyphenyl
methyl
ethyl



2.4.369
2-ethyl-3-trifluoromethoxyphenyl
methyl
ethyl



2.4.370
2-cyclopropyl-3-trifluoromethoxy-
methyl
ethyl




phenyl





2.4.371
2-vinyl-3-trifluoromethoxyphenyl
methyl
ethyl



2.4.372
2-ethynyl-3-trifluoromethoxyphenyl
methyl
ethyl



2.4.373
2-cyano-3-trifluoromethoxyphenyl
methyl
ethyl



2.4.374
2-trifluoromethyl-3-trifluoromethoxy-
methyl
ethyl




phenyl





2.4.375
2-methoxy-3-trifluoromethoxy-
methyl
ethyl




phenyl





2.4.376
2-ethoxy-3-trifluoromethoxyphenyl
methyl
ethyl



2.4.377
2,3-bis(trifluoromethoxy)phenyl
methyl
ethyl



2.4.378
2-nitro-3-trifluoromethoxyphenyl
methyl
ethyl



2.4.379
2-fluoro-3-(2,2,2-trifluoroethoxy)-
methyl
ethyl




phenyl





2.4.380
2-chloro-3-(2,2,2-trifluoroethoxy)-
methyl
ethyl




phenyl





2.4.381
2-bromo-3-(2,2,2-trifluoroethoxy)-
methyl
ethyl




phenyl





2.4.382
2-methyl-3-(2,2,2-trifluoroethoxy)-
methyl
ethyl




phenyl





2.4.383
2-ethyl-3-(2,2,2-trifluoroethoxy)-
methyl
ethyl




phenyl





2.4.384
2-cyclopropyl-3-(2,2,2-trifluoro-
methyl
ethyl




ethoxy)phenyl





2.4.385
2-vinyl-3-(2,2,2-trifluoroethoxy)-
methyl
ethyl




phenyl





2.4.386
2-ethynyl-3-(2,2,2-
methyl
ethyl




trifluoroethoxyphenyl





2.4.387
2-cyano-3-(2,2,2-trifluoroethoxy)-
methyl
ethyl




phenyl





2.4.388
2-trifluoromethyl-3-(2,2,2-trifluoro-
methyl
ethyl




ethoxy)phenyl





2.4.389
2-methoxy-3-(2,2,2-trifluoroethoxy)-
methyl
ethyl




phenyl





2.4.390
2-ethoxy-3-(2,2,2-trifluoroethoxy)-
methyl
ethyl




phenyl





2.4.391
2-trifluoromethoxy-3-(2,2,2-trifluoro-
methyl
ethyl




ethoxy)phenyl





2.4.392
2-nitro-3-(2,2,2-trifluoroethoxy)-
methyl
ethyl




phenyl





2.4.393
2-fluoro-3-difluoromethoxyphenyl
methyl
ethyl



2.4.394
2-chloro-3-difluoromethoxyphenyl
methyl
ethyl



2.4.395
2-bromo-3-difluoromethoxyphenyl
methyl
ethyl



2.4.396
2-methyl-3-difluoromethox-phenyl
methyl
ethyl



2.4.397
2-ethyl-3-difluoromethoxyphenyl
methyl
ethyl



2.4.398
2-cyclopropyl-3-difluoromethoxy-
methyl
ethyl




phenyl





2.4.399
2-vinyl-3-difluoromethoxyphenyl
methyl
ethyl



2.4.400
2-ethynyl-3-difluoromethoxyphenyl
methyl
ethyl



2.4.401
2-cyano-3-difluoro-methoxyphenyl
methyl
ethyl



2.4.402
2-trifluoromethyl-3-difluoromethoxy-
methyl
ethyl




phenyl





2.4.403
2-methoxy-3-difluoro-
methyl
ethyl




methoxyphenyl





2.4.404
2-ethoxy-3-difluoromethoxyphenyl
methyl
ethyl



2.4.405
2-trifluoromethoxy-3-
methyl
ethyl




difluoromethoxyphenyl





2.4.406
2-nitro-3-difluoromethoxyphenyl
methyl
ethyl



2.4.407
2-fluoro-3-(2-methoxyethoxy)-
methyl
ethyl




phenyl





2.4.408
2-chloro-3-(2-methoxyethoxy)-
methyl
ethyl




phenyl





2.4.409
2-bromo-3-(2-methoxyethoxy)-
methyl
ethyl




phenyl





2.4.410
2-methyl-3-(2-methoxyethoxy)-
methyl
ethyl




phenyl





2.4.411
2-ethyl-3-(2-methoxyethoxy)phenyl
methyl
ethyl



2.4.412
2-cyclopropyl-3-(2-methoxyethoxy)-
methyl
ethyl




phenyl





2.4.413
2-vinyl-3-(2-methoxyethoxy)phenyl
methyl
ethyl



2.4.414
2-ethynyl-3-(2-methoxyethoxy)-
methyl
ethyl




phenyl





2.4.415
2-cyano-3-(2-methoxyethoxy)-
methyl
ethyl




phenyl





2.4.416
2-trifluoromethyl-3-(2-
methyl
ethyl




methoxyethoxy)phenyl





2.4.417
2-methoxy-3-(2-methoxyethoxy)-
methyl
ethyl




phenyl





2.4.418
2-ethoxy-3-(2-methoxyethoxy)-
methyl
ethyl




phenyl





2.4.419
2-trifluoromethoxy-(2-
methyl
ethyl




methoxyethoxy)phenyl





2.4.420
2-nitro-3-(2-methoxyethoxy)phenyl
methyl
ethyl



2.4.421
2-fluoro-3-(tert-butoxycarbonyloxy)-
methyl
ethyl




phenyl





2.4.422
2-chloro-3-(tert-butoxycarbonyloxy)-
methyl
ethyl




phenyl





2.4.423
2-bromo-3-(tert-butoxycarbonyl-
methyl
ethyl




oxy)phenyl





2.4.424
2-methyl-3-(tert-butoxycarbonyl-
methyl
ethyl




oxy)phenyl





2.4.425
2-ethyl-3-(tert-butoxycarbonyloxy)- 
methyl
ethyl




phenyl





2.4.426
2-cyclopropyl-3-(tert-
methyl
ethyl




butoxycarbonyl-oxy)phenyl





2.4.427
2-vinyl-3-(tert-butoxycarbonyloxy)-
methyl
ethyl




phenyl





2.4.428
2-ethynyl-3-(tert-butoxycarbonyl-
methyl
ethyl




oxy)phenyl





2.4.429
2-cyano-3-(tert-butoxycarbonyloxy)-
methyl
ethyl




phenyl





2.4.430
2-trifluoromethyl-3-(tert-
methyl
ethyl




butoxycarbonyl-oxy)phenyl





2.4.431
2-methoxy-3-(tert-
methyl
ethyl




butoxycarbonyloxy)phenyl





2.4.432
2-ethoxy-3-(tert-
methyl
ethyl




butoxycarbonyloxy)phenyl





2.4.433
2-trifluoromethoxy-3-(tert-
methyl
ethyl




butoxycarbonyl-oxy)phenyl





2.4.434
2-nitro-3-(tert-butoxycarbonyloxy)-
methyl
ethyl




phenyl





2.4.435
2-fluoro-3-nitrophenyl
methyl
ethyl



2.4.436
2-chloro-3-nitrophenyl
methyl
ethyl



2.4.437
2-bromo-3-nitrophenyl
methyl
ethyl



2.4.438
2-methyl-3-nitrophenyl
methyl
ethyl



2.4.439
2-ethyl-3-nitrophenyl
methyl
ethyl



2.4.440
2-cyclopropyl-3-nitrophenyl
methyl
ethyl



2.4.441
2-vinyl-3-nitrophenyl
methyl
ethyl



2.4.442
2-ethynyl-3-nitrophenyl
methyl
ethyl



2.4.443
2-cyano-3-nitrophenyl
methyl
ethyl



2.4.444
2-trifluoromethyl-3-nitrophenyl
methyl
ethyl



2.4.445
2-methoxy-3-nitrophenyl
methyl
ethyl



2.4.446
2-ethoxy-3-nitrophenyl
methyl
ethyl



2.4.447
2-trifluoromethoxy-3-nitrophenyl
methyl
ethyl



2.4.448
2-fluoro-3-methylsulfanylphenyl
methyl
ethyl



2.4.449
2-chloro-3-methylsulfanylphenyl
methyl
ethyl



2.4.450
2-bromo-3-methylsulfanylphenyl
methyl
ethyl



2.4.451
2-methyl-3-methylsulfanylphenyl
methyl
ethyl



2.4.452
2-ethyl-3-methylsulfanylphenyl
methyl
ethyl



2.4.453
2-cyclopropyl-3-
methyl
ethyl




methylsulfanylphenyl





2.4.454
2-vinyl-3-methylsulfanylphenyl
methyl
ethyl



2.4.455
2-ethynyl-3-methylsulfanylphenyl
methyl
ethyl



2.4.456
2-cyano-3-methylsulfanylphenyl
methyl
ethyl



2.4.457
2-trifluoromethyl-3-
methyl
ethyl




methylsulfanylphenyl





2.4.458
2-methoxy-3-methylsulfanylphenyl
methyl
ethyl



2.4.459
2-ethoxy-3-methylsulfanylphenyl
methyl
methyl



2.4.460
2-trifluoromethoxy-3-
methyl
ethyl




methylsulfanylphenyl





2.4.61
2-nitro-3-methylsulfanylphenyl
methyl
ethyl



2.4.62
3,5-difluorophenyl
methyl
methyl
[CDCl3] 2.44 (s, 3H); 3.80






(d, 1H); 3.86 (s, 3H); 3.89






(d, 1H); 6.90 (m, 1H); 7.19






(d, 2H).


2.4.463
3,5-difluorophenyl
ethyl
methyl
[CDCl3] 1.12 (t, 3H); 2.83






(q, 2H); 3.81 (d, 1H); 3.86






(s, 4H); 6.90 (m, 1H); 7.20






(d, 2H).


2.4.464
3,5-difluorophenyl
propyl
ethyl



2.4.465
3,5-difluorophenyl
butyl
ethyl



2.4.466
3-chloro-5-fluorophenyl
methyl
methyl
[CDCl3] 2.43 (s, 3H); 3.80






(d, 1H); 3.87 (s, 3H); 3.90






(d, 1H); 7.18 (d, 1H), 7.30






(d, 1H), 7.43 (s, 1H).


2.4.467
3-chloro-5-fluorophenyl
ethyl
ethyl



2.4.468
3-chloro-5-fluorophenyl
propyl
ethyl



2.4.469
3-chloro-5-fluorophenyl
butyl
ethyl



2.4.470
3-bromo-5-fluorophenyl
methyl
ethyl



2.4.471
3-bromo-5-fluorophenyl
ethyl
ethyl



2.4.472
3-bromo-5-fluorophenyl
propyl
ethyl



2.4.473
3-bromo-5-fluorophenyl
butyl
ethyl



2.4.474
3-iodo-5-fluorophenyl
methyl
ethyl



2.4.475
3-methyl-5-fluorophenyl
methyl
ethyl



2.4.476
3-methyl-5-fluorophenyl
ethyl
ethyl



2.4.477
3-methyl-5-fluorophenyl
propyl
ethyl



2.4.478
3-methyl-5-fluorophenyl
butyl
ethyl



2.4.479
3-ethyl-5-fluorophenyl
methyl
ethyl



2.4.480
3-propyl-5-fluorophenyl
methyl
ethyl



2.4.481
3-i-propyl-5-fluorophenyl
methyl
ethyl



2.4.482
3-n-butyl-5-fluorophenyl
methyl
ethyl



2.4.483
3-isobutyl-5-fluorophenyl
methyl
ethyl



2.4.484
3-tert-butyl-5-fluorophenyl
methyl
ethyl



2.4.485
3-cyclopropyl-5-fluorophenyl
methyl
ethyl



2.4.486
3-vinyl-5-fluorophenyl
methyl
ethyl



2.4.487
3-ethynyl-5-fluorophenyl
methyl
ethyl



2.4.488
3-cyano-5-fluorophenyl
methyl
ethyl



2.4.489
3-trifluoromethyl-5-fluorophenyl
methyl
ethyl



2.4.490
3-trifluoromethyl-5-fluorophenyl
ethyl
ethyl



2.4.491
3-trifluoromethyl-5-fluorophenyl
propyl
ethyl



2.4.492
3-trifluoromethyl-5-fluorophenyl
butyl
ethyl



2.4.493
3-(methoxycarbonyl)-5-fluorophenyl
methyl
ethyl



2.4.494
3-hydroxymethyl-5-fluorophenyl
methyl
ethyl



2.4.495
3-carbamoyl-5-fluorophenyl
methyl
ethyl



2.4.496
3-hydroxy-5-fluorophenyl
methyl
ethyl



2.4.497
3-methoxy-5-fluorophenyl
methyl
ethyl



2.4.498
3-ethoxy-5-fluorophenyl
methyl
ethyl



2.4.499
3-n-propoxy-5-fluorophenyl
methyl
ethyl



2.4.500
3-isopropoxy-5-fluorophenyl
methyl
ethyl



2.4.501
3-n-butoxy-5-fluorophenyl
methyl
ethyl



2.4.502
3-isobutoxy-5-fluorophenyl
methyl
ethyl



2.4.503
3-tert-butoxy-5-fluorophenyl
methyl
ethyl



2.4.504
3-difluoromethoxy-5-fluorophenyl
methyl
ethyl



2.4.505
3-trifluoromethoxy-5-fluorophenyl
methyl
ethyl



2.4.506
3-(2,2,2-trifluoroethoxy)-5-
methyl
ethyl




fluorophenyl





2.4.507
3-(2-chloroethoxy)-5-fluorophenyl
methyl
ethyl



2.4.508
3-(2-hydroxyethoxy)-5-fluorophenyl
methyl
ethyl



2.4.509
3-[(tert-butoxycarbonyl)oxy]-5-
methyl
ethyl




fluorophenyl





2.4.510
3-nitro-5-fluorophenyl
methyl
ethyl



2.4.511
3-acetoxy-5-fluorophenyl
methyl
ethyl



2.4.512
{3-[(tert-butoxy-carbonyl)amino]-5-
methyl
ethyl




fluorophenyl}





2.4.513
3-methylsulfanyl-5-fluorophenyl
methyl
ethyl



2.4.514
3,5-difluorophenyl
methyl
methyl
[CDCl3] 2.43 (s, 3H); 3.79






(d, 1H); 3.86 (s, 3H), 3.90






(d, 1H), 7.43 (s, 1H); 7.55






(s, 2H).


2.4.515
3,5-dichlorophenyl
ethyl
methyl
[CDCl3] 1.12 (t, 3H); 2.82






(q, 2H); 3.81 (d, 1H); 3.85






(s, 3H); 7.43 (s, 1H); 7.54






(s, 2H).


2.4.516
3,5-dichlorophenyl
propyl
ethyl



2.4.517
3,5-dichlorophenyl
butyl
ethyl



2.4.518
3-bromo-5-chlorophenyl
methyl
ethyl



2.4.519
3-iodo-5-chlorophenyl
methyl
ethyl



2.4.520
3-methyl-5-chlorophenyl
methyl
methyl
[CDCl3] 2.36 (s, 3H), 2.43






(s, 3H); 3.82 (d, 1H); 3.86






(s, 4H); 7.24 (s, 1H); 7.36






(s, 1H); 7.46 (s, 1H).


2.4.521
3-ethyl-5-chlorophenyl
methyl
ethyl



2.4.522
3-propyl-5-chlorophenyl
methyl
ethyl



2.4.523
3-isopropyl-5-chlorophenyl
methyl
ethyl



2.4.524
3-n-butyl-5-chlorophenyl
methyl
ethyl



2.4.525
3-isobutyl-5-chlorophenyl
methyl
ethyl



2.4.526
3-tert-butyl-5-chlorophenyl
methyl
ethyl



2.4.527
3-cyclopropyl-5-chlorophenyl
methyl
ethyl



2.4.528
3-vinyl-5-chlorophenyl
methyl
ethyl



2.4.529
3-ethynyl-5-chlorophenyl
methyl
ethyl



2.4.530
3-cyano-5-chlorophenyl
methyl
ethyl



2.4.531
3-trifluoromethyl-5-chlorophenyl
methyl
ethyl



2.4.532
3-(hydroxycarbonyl)-5-chlorophenyl
methyl
ethyl



2.4.533
3-(methoxycarbonyl)-5-
methyl
ethyl




chlorophenyl





2.4.534
3-hydroxymethyl-5-chlorophenyl
methyl
ethyl



2.4.535
3-carbamoyl-5-chlorophenyl
methyl
ethyl



2.4.536
3-hydroxy-5-chlorophenyl
methyl
ethyl



2.4.537
3-methoxy-5-chlorophenyl
methyl
ethyl



2.4.538
3-ethoxy-5-chlorophenyl
methyl
ethyl



2.4.539
3-n-propoxy-5-chlorophenyl
methyl
ethyl



2.4.540
3-isopropoxy-5-chlorophenyl
methyl
ethyl



2.4.541
3-n-butoxy-5-chlorophenyl
methyl
ethyl



2.4.542
3-isobutoxy-5-chlorophenyl
methyl
ethyl



2.4.543
3-tert-butoxy-5-chlorophenyl
methyl
ethyl



2.4.544
3-difluoromethoxy-5-chlorophenyl
methyl
ethyl



2.4.545
3-trifluoromethoxy-5-chlorophenyl
methyl
ethyl



2.4.546
3-(2,2,2-trifluoroethoxy)-5-
methyl
ethyl




chlorophenyl





2.4.547
3-(2-chloroethoxy)-5-chlorophenyl
methyl
ethyl



2.4.548
3-(2-hydroxyethoxy)-5-chlorophenyl
methyl
ethyl



2.4.549
3-[(tert-butoxycarbonyl)oxy]-5-
methyl
ethyl




chlorophenyl





2.4.550
3-nitro-5-chlorophenyl
methyl
ethyl



2.4.551
3-acetoxy-5-chlorophenyl
methyl
ethyl



2.4.552
{3-[(tert-butoxy-carbonyl)amino]-5- 
methyl
ethyl




chlorophenyl}





2.4.553
3-methylsulfanyl-5-chlorophenyl
methyl
ethyl



2.4.554
3,5-dibromophenyl
methyl
ethyl



2.4.555
3,5-dibromophenyl
ethyl
ethyl



2.4.556
3-iodo-5-bromophenyl
methyl
ethyl



2.4.557
3-methyl-5-bromophenyl
methyl
methyl
[CDCl3] 2.36 (s, 3H); 2.43






(s, 3H); 3.81 (d, 1H), 3.86






(s, 3H); 3.89 (d, 1H); 7.41






(s, 2H); 7.61 (s, 1H).


2.4.558
3-methyl-5-bromophenyl
ethyl
ethyl



2.4.559
3-methyl-5-bromophenyl
propyl
ethyl



2.4.560
3-methyl-5-bromophenyl
butyl
ethyl



2.4.561
3-ethyl-5-bromophenyl
methyl
ethyl



2.4.562
3-propyl-5-bromophenyl
methyl
ethyl



2.4.563
3-isopropyl-5-bromophenyl
methyl
ethyl



2.4.564
3-n-butyl-5-bromophenyl
methyl
ethyl



2.4.565
3-isobutyl-5-bromophenyl
methyl
ethyl



2.4.566
3-tert-butyl-5-bromophenyl
methyl
ethyl



2.4.567
3-cyclopropyl-5-bromophenyl
methyl
ethyl



2.4.568
3-cyano-5-bromophenyl
methyl
ethyl



2.4.569
3-trifluoromethyl-5-bromophenyl
methyl
ethyl



2.4.570
3-(methoxycarbonyl)-5-
methyl
ethyl




bromophenyl





2.4.571
3-methoxy-5-bromophenyl
methyl
ethyl



2.4.572
3-ethoxy-5-bromophenyl
methyl
ethyl



2.4.573
3-n-propoxy-5-bromophenyl
methyl
ethyl



2.4.574
3-isopropoxy-5-bromophenyl
methyl
ethyl



2.4.575
3-n-butoxy-5-bromophenyl
methyl
ethyl



2.4.576
3-isobutoxy-5-bromophenyl
methyl
ethyl



2.4.577
3-difluoromethoxy-5-bromophenyl
methyl
ethyl



2.4.578
3-trifluoromethoxy-5-bromophenyl
methyl
ethyl



2.4.579
3-nitro-5-bromophenyl
methyl
ethyl



2.4.580
3-acetoxy-5-bromophenyl
methyl
ethyl



2.4.581
3-methylsulfanyl-5-bromophenyl
methyl
ethyl



2.4.582
3,5-diiodophenyl
methyl
ethyl



2.4.583
3-methyl-5-iodophenyl
methyl
ethyl



2.4.584
3-ethyl-5-iodophenyl
methyl
ethyl



2.4.585
3-propyl-5-iodophenyl
methyl
ethyl



2.4.586
3-isopropyl-5-iodophenyl
methyl
ethyl



2.4.587
3-n-butyl-5-iodophenyl
methyl
ethyl



2.4.588
3-isobutyl-5-iodophenyl
methyl
ethyl



2.4.589
3-tert-butyl-5-iodophenyl
methyl
ethyl



2.4.590
3-cyclopropyl-5-iodophenyl
methyl
ethyl



2.4.591
3-cyano-5-iodophenyl
methyl
ethyl



2.4.592
3-trifluoromethyl-5-iodophenyl
methyl
ethyl



2.4.593
3-(methoxycarbonyl)-5-iodophenyl
methyl
ethyl



2.4.594
3-methoxy-5-iodophenyl
methyl
ethyl



2.4.595
3-ethoxy-5-iodophenyl
methyl
ethyl



2.4.596
3-n-propoxy-5-iodophenyl
methyl
ethyl



2.4.597
3-isopropoxy-5-iodophenyl
methyl
ethyl



2.4.598
3-n-butoxy-5-iodophenyl
methyl
ethyl



2.4.599
3-isobutoxy-5-iodophenyl
methyl
ethyl



2.4.600
3-difluoromethoxy-5-iodophenyl
methyl
ethyl



2.4.601
3-trifluoromethoxy-5-iodophenyl
methyl
ethyl



2.4.602
3-nitro-5-iodophenyl
methyl
ethyl



2.4.603
3-acetoxy-5-iodophenyl
methyl
ethyl



2.4.604
3-methylsulfanyl-5-iodophenyl
methyl
ethyl



2.4.605
3,5-dimethylphenyl
methyl
ethyl



2.4.606
3-ethyl-5-methylphenyl
methyl
ethyl



2.4.607
3-propyl-5-methylphenyl
methyl
ethyl



2.4.608
3-isopropyl-5-methylphenyl
methyl
ethyl



2.4.609
3-n-butyl-5-methylphenyl
methyl
ethyl



2.4.610
3-isobutyl-5-methylphenyl
methyl
ethyl



2.4.611
3-tert-butyl-5-methylphenyl
methyl
ethyl



2.4.612
3-cyclopropyl-5-methylphenyl
methyl
ethyl



2.4.613
3-cyano-5-methylphenyl
methyl
ethyl



2.4.614
3-trifluoromethyl-5-methylphenyl
methyl
ethyl



2.4.615
3-(methoxycarbonyl)-5-
methyl
ethyl




methylphenyl





2.4.616
3-methoxy-5-methylphenyl
methyl
ethyl



2.4.617
3-ethoxy-5-methylphenyl
methyl
ethyl



2.4.618
3-n-propoxy-5-methylphenyl
methyl
ethyl



2.4.619
3-n-butoxy-5-methylphenyl
methyl
ethyl



2.4.620
3-isobutoxy-5-methylphenyl
methyl
ethyl



2.4.621
3-difluoromethoxy-5-methylphenyl
methyl
ethyl



2.4.622
3-trifluoromethoxy-5-methylphenyl
methyl
ethyl



2.4.623
3-nitro-5-methylphenyl
methyl
ethyl



2.4.624
3-acetoxy-5-methylphenyl
methyl
ethyl



2.4.625
3-methylsulfanyl-5-methylphenyl
methyl
ethyl



2.4.626
3,5-diethylphenyl
methyl
ethyl



2.4.627
3-propyl-5-ethylphenyl
methyl
ethyl



2.4.628
3-isopropyl-5-ethylphenyl
methyl
ethyl



2.4.629
3-n-butyl-5-ethylphenyl
methyl
ethyl



2.4.630
3-isobutyl-5-ethylphenyl
methyl
ethyl



2.4.631
3-tert-butyl-5-ethylphenyl
methyl
ethyl



2.4.632
3-cyclopropyl-5-ethylphenyl
methyl
ethyl



2.4.633
3-cyano-5-ethylphenyl
methyl
ethyl



2.4.634
3-trifluoromethyl-5-ethylphenyl
methyl
ethyl



2.4.635
3-(methoxycarbonyl)-5-ethylphenyl
methyl
ethyl



2.4.636
3-methoxy-5-ethylphenyl
methyl
ethyl



2.4.637
3-ethoxy-5-ethylphenyl
methyl
ethyl



2.4.638
3-n-propoxy-5-ethylphenyl
methyl
ethyl



2.4.639
3-n-butoxy-5-ethylphenyl
methyl
ethyl



2.4.640
3-isobutoxy-5-ethylphenyl
methyl
ethyl



2.4.641
3-difluoromethoxy-5-ethylphenyl
methyl
ethyl



2.4.642
3-trifluoromethoxy-5-ethylphenyl
methyl
ethyl



2.4.643
3-nitro-5-ethylphenyl
methyl
ethyl



2.4.644
3-acetoxy-5-ethylphenyl
methyl
ethyl



2.4.645
3-methylsulfanyl-5-ethylphenyl
methyl
ethyl



2.4.646
3,5-dipropylphenyl
methyl
ethyl



2.4.647
3-isopropyl-5-propylphenyl
methyl
ethyl



2.4.648
3-n-butyl-5-propylphenyl
methyl
ethyl



2.4.649
3-isobutyl-5-propylphenyl
methyl
ethyl



2.4.650
3-tert-butyl-5-propylphenyl
methyl
ethyl



2.4.651
3-cyclopropyl-5-propylphenyl
methyl
ethyl



2.4.652
3-cyano-5-propylphenyl
methyl
ethyl



2.4.653
3-trifluoromethyl-5-propylphenyl 
methyl
ethyl



2.4.654
3-(hydroxycarbonyl)-5-propylphenyl
methyl
ethyl



2.4.655
3-(methoxycarbonyl)-5-
methyl
ethyl




propylphenyl





2.4.656
3-methoxy-5-propylphenyl
methyl
ethyl



2.4.657
3-ethoxy-5-propylphenyl
methyl
ethyl



2.4.658
3-n-propoxy-5-propylphenyl
methyl
ethyl



2.4.659
3-n-butoxy-5-propylphenyl
methyl
ethyl



2.4.660
3-isobutoxy-5-propylphenyl
methyl
ethyl



2.4.661
3-difluoromethoxy-5-propylphenyl
methyl
ethyl



2.4.662
3-trifluoromethoxy-5-ethylphenyl
methyl
ethyl



2.4.663
3-nitro-5-propylphenyl
methyl
ethyl



2.4.664
3-acetoxy-5-propylphenyl
methyl
ethyl



2.4.665
3-methylsulfanyl-5-propylphenyl
methyl
ethyl



2.4.666
3,5-diisopropylphenyl
methyl
ethyl



2.4.667
3-n-butyl-5-isopropylphenyl
methyl
ethyl



2.4.668
3-isobutyl-5-isopropylphenyl
methyl
ethyl



2.4.669
3-tert-butyl-5-isopropylphenyl
methyl
ethyl



2.4.670
3-cyclopropyl-5-isopropylphenyl
methyl
ethyl



2.4.671
3-cyano-5-isopropylphenyl
methyl
ethyl



2.4.672
3-trifluoromethyl-5-isopropylphenyl
methyl
ethyl



2.4.673
3-(methoxycarbonyl)-5-
methyl
ethyl




isopropylphenyl





2.4.674
3-methoxy-5-isopropylphenyl
methyl
ethyl



2.4.675
3-ethoxy-5-isopropylphenyl
methyl
ethyl



2.4.676
3-n-propoxy-5-isopropylphenyl
methyl
ethyl



2.4.677
3-n-butoxy-5-isopropylphenyl
methyl
ethyl



2.4.678
3-isobutoxy-5-isopropylphenyl
methyl
ethyl



2.4.679
3-difluoromethoxy-5-
methyl
ethyl




isopropylphenyl





2.4.680
3-trifluoromethoxy-5-
methyl
ethyl




isopropylphenyl





2.4.681
3-nitro-5-isopropylphenyl
methyl
ethyl



2.4.682
3-acetoxy-5-isopropylphenyl
methyl
ethyl



2.4.683
3-methylsulfanyl-5-isopropylphenyl 
methyl
ethyl



2.4.684
3,5-dibutylphenyl
methyl
ethyl



2.4.685
3-isobutyl-5-butylphenyl
methyl
ethyl



2.4.686
3-tert-butyl-5-butylphenyl
methyl
ethyl



2.4.687
3-cyclopropyl-5-butylphenyl
methyl
ethyl



2.4.688
3-cyano-5-butylphenyl
methyl
ethyl



2.4.689
3-trifluoromethyl-5-butylphenyl
methyl
ethyl



2.4.690
3-(methoxycarbonyl)-5-butylphenyl
methyl
ethyl



2.4.691
3-methoxy-5-butylphenyl
methyl
ethyl



2.4.692
3-ethoxy-5-butylphenyl
methyl
ethyl



2.4.693
3-n-propoxy-5-butylphenyl
methyl
ethyl



2.4.694
3-n-butoxy-5-butylphenyl
methyl
ethyl



2.4.695
3-isobutoxy-5-butylphenyl
methyl
ethyl



2.4.696
3-difluoromethoxy-5-butylphenyl
methyl
ethyl



2.4.697
3-trifluoromethoxy-5-butylphenyl
methyl
ethyl



2.4.698
3-nitro-5-butylphenyl
methyl
ethyl



2.4.699
3-acetoxy-5-butylphenyl
methyl
ethyl



2.4.700
3-methylsulfanyl-5-butylphenyl
methyl
ethyl



2.4.701
3,5-diisobutylphenyl
methyl
ethyl



2.4.702
3-tert-butyl-5-isobutylphenyl
methyl
ethyl



2.4.703
3-cyclopropyl-5-isobutylphenyl
methyl
ethyl



2.4.704
3-cyano-5-isobutylphenyl
methyl
ethyl



2.4.705
3-trifluoromethyl-5-isobutylphenyl
methyl
ethyl



2.4.706
3-(methoxycarbonyl)-5-
methyl
ethyl




isobutylphenyl





2.4.707
3-methoxy-5-isobutylphenyl
methyl
ethyl



2.4.708
3-ethoxy-5-isobutylphenyl
methyl
ethyl



2.4.709
3-n-propoxy-5-isobutylphenyl
methyl
ethyl



2.4.710
3-n-butoxy-5-isobutylphenyl
methyl
ethyl



2.4.711
3-isobutoxy-5-isobutylphenyl
methyl
ethyl



2.4.712
3-difluoromethoxy-5-isobutylphenyl
methyl
ethyl



2.4.713
3-trifluoromethoxy-5-isobutylphenyl
methyl
ethyl



2.4.714
3-nitro-5-isobutylphenyl
methyl
ethyl



2.4.715
3-acetoxy-5-isobutylphenyl
methyl
ethyl



2.4.716
3-methylsulfanyl-5-isobutylphenyl
methyl
ethyl



2.4.717
3,5-di(tert-butyl)phenyl
methyl
ethyl



2.4.718
3-cyclopropyl-5-tert-butylphenyl
methyl
ethyl



2.4.719
3-cyano-5-tert-butylphenyl
methyl
ethyl



2.4.720
3-trifluoromethyl-5-tert-butylphenyl
methyl
ethyl



2.4.721
3-(methoxycarbonyl)-5-tert-
methyl
ethyl




butylphenyl





2.4.722
3-methoxy-5-tert-butylphenyl
methyl
ethyl



2.4.723
3-ethoxy-5-tert-butylphenyl
methyl
ethyl



2.4.724
3-n-propoxy-5-tert-butylphenyl
methyl
ethyl



2.4.725
3-n-butoxy-5-tert-butylphenyl
methyl
ethyl



2.4.726
3-isobutoxy-5-tert-butylphenyl
methyl
ethyl



2.4.727
3-difluoromethoxy-5-tert-
methyl
ethyl




butylphenyl





2.4.728
3-trifluoromethoxy-5-tert-
methyl
ethyl




butylphenyl





2.4.729
3-nitro-5-tert-butylphenyl
methyl
ethyl



2.4.730
3-acetoxy-5-tert-butylphenyl
methyl
ethyl



2.4.731
3-methylsulfanyl-5-tert-butylphenyl
methyl
ethyl



2.4.732
3-tert-butyl-5-cyclopropylphenyl
methyl
ethyl



2.4.733
3,5-dicyclopropyl-phenyl
methyl
ethyl



2.4.734
3-cyano-5-cyclopropylphenyl
methyl
ethyl



2.4.735
3-trifluoromethyl-5-
methyl
ethyl




cyclopropylphenyl





2.4.736
3-(methoxycarbonyl)-5-
methyl
ethyl




cyclopropylphenyl





2.4.737
3-methoxy-5-cyclopropylphenyl
methyl
ethyl



2.4.738
3-ethoxy-5-cyclopropylphenyl
methyl
ethyl



2.4.739
3-n-propoxy-5-cyclopropylphenyl
methyl
ethyl



2.4.740
3-n-butoxy-5-cyclopropylphenyl
methyl
ethyl



2.4.741
3-isobutoxy-5-cyclopropylphenyl
methyl
ethyl



2.4.742
3-difluoromethoxy-5-
methyl
ethyl




cyclopropylphenyl





2.4.743
3-trifluoromethoxy-5-
methyl
ethyl




cyclopropylphenyl





2.4.744
3-nitro-5-cyclopropylphenyl
methyl
ethyl



2.4.745
3-acetoxy-5-cyclopropylphenyl
methyl
ethyl



2.4.746
3-methylsulfanyl-5-
methyl
ethyl




cyclopropylphenyl





2.4.747
3,5-dicyanophenyl
methyl
ethyl



2.4.748
3-trifluoromethyl-5-cyanophenyl
methyl
ethyl



2.4.749
3-(methoxycarbonyl)-5-
methyl
ethyl




cyanophenyl





2.4.750
3-methoxy-5-cyanophenyl
methyl
ethyl



2.4.751
3-ethoxy-5-cyanophenyl
methyl
ethyl



2.4.752
3-n-propoxy-5-cyanophenyl
methyl
ethyl



2.4.753
3-n-butoxy-5-cyanophenyl
methyl
ethyl



2.4.754
3-isobutoxy-5-cyanophenyl
methyl
ethyl



2.4.755
3-difluoromethoxy-5-cyanophenyl
methyl
ethyl



2.4.756
3-trifluoromethoxy-5-cyanophenyl
methyl
ethyl



2.4.757
3-nitro-5-cyanophenyl
methyl
ethyl



2.4.758
3-acetoxy-5-cyanophenyl
methyl
ethyl



2.4.759
3-methylsulfanyl-5-cyanophenyl
methyl
ethyl



2.4.760
3,5-di(trifluoromethyl)-phenyl
methyl
ethyl



2.4.761
3-(methoxycarbonyl)-5-
methyl
ethyl




trifluoromethyl-phenyl





2.4.762
3-methoxy-5-trifluoromethylphenyl
methyl
ethyl



2.4.763
3-ethoxy-5-trifluoromethylphenyl
methyl
ethyl



2.4.764
3-n-propoxy-5-trifluoromethylphenyl
methyl
ethyl



2.4.765
3-n-butoxy-5-trifluoromethylphenyl
methyl
ethyl



2.4.766
3-isobutoxy-5-trifluoromethylphenyl
methyl
ethyl



2.4.767
3-difluoromethoxy-5-
methyl
ethyl




trifluoromethylphenyl





2.4.768
3-trifluoromethoxy-5-
methyl
ethyl




trifluoromethylphenyl





2.4.769
3-nitro-5-trifluoromethylphenyl
methyl
ethyl



2.4.770
3-acetoxy-5-trifluoromethylphenyl
methyl
ethyl



2.4.771
3-methylsulfanyl-5-
methyl
ethyl




trifluoromethylphenyl





2.4.772
3,5-di(methoxy-carbonyl)phenyl
methyl
ethyl



2.4.773
3-methoxy-5-(methoxycarbonyl)-
methyl
ethyl




phenyl





2.4.774
3-ethoxy-5-(methoxycarbonyl)-
methyl
ethyl




phenyl





2.4.775
3-n-propoxy-5-(methoxycarbonyl)-
methyl
ethyl




phenyl





2.4.776
3-isobutoxy-5-(methoxycarbonyl)-
methyl
ethyl




phenyl





2.4.777
3-difluoromethoxy-5-
methyl
ethyl




(methoxycarbonyl)phenyl





2.4.778
3-trifluoromethoxy-5-
methyl
ethyl




(methoxycarbonyl)phenyl





2.4.779
3-nitro-5-(methoxy-carbonyl)phenyl
methyl
ethyl



2.4.780
3-acetoxy-5-(methoxycarbonyl)-
methyl
ethyl




phenyl





2.4.781
3-methylsulfanyl-5-
methyl
ethyl




(methoxycarbonyl)phenyl





2.4.782
3,5-dimethoxyphenyl
methyl
ethyl



2.4.783
3-ethoxy-5-methoxyphenyl
methyl
ethyl



2.4.784
3-n-propoxy-5-methoxyphenyl
methyl
ethyl



2.4.785
3-n-butoxy-5-methoxyphenyl
methyl
ethyl



2.4.786
3-isobutoxy-5-methoxyphenyl
methyl
ethyl



2.4.787
3-difluoromethoxy-5-methoxyphenyl
methyl
ethyl



2.4.788
3-trifluoromethoxy-5-
methyl
ethyl




methoxyphenyl





2.4.789
3-nitro-5-methoxyphenyl
methyl
ethyl



2.4.790
3-acetoxy-5-methoxyphenyl
methyl
ethyl



2.4.791
3-methylsulfanyl-5-methoxyphenyl
methyl
ethyl



2.4.792
3,5-diethoxyphenyl
methyl
ethyl



2.4.793
3-n-propoxy-5-ethoxyphenyl
methyl
ethyl



2.4.794
3-n-butoxy-5-ethoxyphenyl
methyl
ethyl



2.4.795
3-isobutoxy-5-ethoxyphenyl
methyl
ethyl



2.4.796
3-difluoromethoxy-5-ethoxyphenyl
methyl
ethyl



2.4.797
3-trifluoromethoxy-5-ethoxyphenyl
methyl
ethyl



2.4.798
3-nitro-5-ethoxyphenyl
methyl
ethyl



2.4.799
3-acetoxy-5-ethoxyphenyl
methyl
ethyl



2.4.800
3-methylsulfanyl-5-ethoxyphenyl
methyl
ethyl



2.4.801
3,5-dipropoxyphenyl
methyl
ethyl



2.4.802
3-n-butoxy-5-propoxyphenyl
methyl
ethyl



2.4.803
3-isobutoxy-5-propoxyphenyl
methyl
ethyl



2.4.804
3-difluoromethoxy-5-propoxyphenyl
methyl
ethyl



2.4.805
3-trifluoromethoxy-5-propoxyphenyl
methyl
ethyl



2.4.806
3-nitro-5-propoxyphenyl
methyl
ethyl



2.4.807
3-acetoxy-5-propoxyphenyl
methyl
ethyl



2.4.808
3-methylsulfanyl-5-propoxyphenyl 
methyl
ethyl



2.4.809
3,5-di(isopropoxy)phenyl
methyl
ethyl



2.4.810
3-n-butoxy-5-isopropoxyphenyl
methyl
ethyl



2.4.811
3-isobutoxy-5-isopropoxyphenyl
methyl
ethyl



2.4.812
3-difluoromethoxy-5-
methyl
ethyl




isopropoxyphenyl





2.4.813
3-trifluoromethoxy-5-
methyl
ethyl




isopropoxyphenyl





2.4.814
3-nitro-5-isopropoxyphenyl
methyl
ethyl



2.4.815
3-acetoxy-5-isopropoxyphenyl
methyl
ethyl



2.4.816
3-methylsulfanyl-5-
methyl
ethyl




isopropoxyphenyl





2.4.817
3,5-di(trifluoro-methoxy)phenyl
methyl
ethyl



2.4.818
3-nitro-5-trifluoro-methoxyphenyl
methyl
ethyl



2.4.819
3-acetoxy-5-tert-butoxyphenyl
methyl
ethyl



2.4.820
3-methylsulfanyl-5-trifluoromethoxy-
methyl
ethyl




phenyl





2.4.821
3,5-bis(difluoromethoxy)phenyl
methyl
ethyl



2.4.822
3,5-bis(difluoromethoxy)phenyl
ethyl
ethyl



2.4.823
3,5-bis(difluoromethoxy)phenyl
propyl
ethyl



2.4.824
3,5-bis(difluoromethoxy)phenyl
butyl
ethyl



2.4.825
3-trifluoromethoxy-5-
methyl
ethyl




difluoromethoxyphenyl





2.4.826
3-nitro-5-difluoromethoxyphenyl
methyl
ethyl



2.4.827
3-acetoxy-5-difluoro-methoxyphenyl
methyl
ethyl



2.4.828
3-methylsulfanyl-5-difluoromethoxy-
methyl
ethyl




phenyl





2.4.829
3,5-bis(acetoxy)phenyl
methyl
ethyl



2.4.830
3-methylsulfanyl-5-acetoxyphenyl
methyl
ethyl



2.4.831
3-acetoxy-5-nitrophenyl
methyl
ethyl



2.4.832
3-methylsulfanyl-5-nitrophenyl
methyl
ethyl



2.4.833
3,5-di(methylsulfanyl)phenyl
methyl
ethyl



2.4.834
3,4-difluorophenyl
methyl
ethyl



2.4.835
3,4-difluorophenyl
ethyl
ethyl



2.4.836
3,4-difluorophenyl
propyl
ethyl



2.4.837
3,4-difluorophenyl
butyl
ethyl



2.4.838
3-chloro-4-fluorophenyl
methyl
ethyl



2.4.839
3-chloro-4-fluorophenyl
ethyl
ethyl



2.4.840
3-chloro-4-fluorophenyl
propyl
ethyl



2.4.841
3-chloro-4-fluorophenyl
butyl
ethyl



2.4.842
3-bromo-4-fluorophenyl
methyl
ethyl



2.4.843
3-methyl-4-fluorophenyl
methyl
ethyl



2.4.844
3-methyl-4-fluorophenyl
ethyl
ethyl



2.4.845
3-ethyl-4-fluorophenyl
methyl
ethyl



2.4.846
3-cyclopropyl-4-fluorophenyl
methyl
ethyl



2.4.847
3-cyano-4-fluorophenyl
methyl
ethyl



2.4.848
3-methoxy-4-fluorophenyl
methyl
ethyl



2.4.849
3-ethoxy-4-fluorophenyl
methyl
ethyl



2.4.850
3-trifluoromethoxy-4-fluorophenyl
methyl
ethyl



2.4.851
3-nitro-4-fluorophenyl
methyl
ethyl



2.4.852
3-fluoro-4-chlorophenyl
methyl
ethyl



2.4.853
3,4-dichlorophenyl
methyl
ethyl



2.4.854
3-bromo-4-chlorophenyl
methyl
ethyl



2.4.855
3-methyl-4-chlorophenyl
methyl
ethyl



2.4.856
3-cyclopropyl-4-chlorophenyl
methyl
ethyl



2.4.857
3-cyano-4-chlorophenyl
methyl
ethyl



2.4.858
3-trifluoromethyl-4-chlorophenyl
methyl
ethyl



2.4.859
3-methoxy-4-chlorophenyl
methyl
ethyl



2.4.860
3-ethoxy-4-chlorophenyl
methyl
ethyl



2.4.861
3-trifluoromethoxy-4-chlorophenyl
methyl
ethyl



2.4.862
3-nitro-4-chlorophenyl
methyl
ethyl



2.4.863
3-fluoro-4-bromophenyl
methyl
ethyl



2.4.864
3-chloro-4-bromophenyl
methyl
ethyl



2.4.865
3,4-dibromophenyl
methyl
ethyl



2.4.866
3-methyl-4-bromophenyl
methyl
ethyl



2.4.867
3-cyclopropyl-4-bromophenyl
methyl
ethyl



2.4.868
3-cyano-4-bromophenyl
methyl
ethyl



2.4.869
3-trifluoromethyl-4-bromophenyl 
methyl
ethyl



2.4.870
3-methoxy-4-phenyl
methyl
ethyl



2.4.871
3-ethoxy-4-bromophenyl
methyl
ethyl



2.4.872
3-trifluoromethoxy-4-bromophenyl
methyl
ethyl



2.4.873
3-nitro-4-bromophenyl
methyl
ethyl



2.4.874
3-fluoro-4-iodophenyl
methyl
ethyl



2.4.875
3-chloro-4-iodophenyl
methyl
ethyl



2.4.876
3-bromo-4-iodophenyl
methyl
ethyl



2.4.877
3-methyl-4-iodophenyl
methyl
ethyl



2.4.878
3-cyclopropyl-4-iodophenyl
methyl
ethyl



2.4.879
3-cyano-4-iodophenyl
methyl
ethyl



2.4.880
3-trifluoromethyl-4-iodophenyl
methyl
ethyl



2.4.881
3-methoxy-4-iodophenyl
methyl
ethyl



2.4.882
3-ethoxy-4-iodophenyl
methyl
ethyl



2.4.883
3-trifluoromethoxy-4-iodophenyl
methyl
ethyl



2.4.884
3-nitro-4-iodophenyl
methyl
ethyl



2.4.885
3-fluoro-4-methylphenyl
methyl
ethyl



2.4.886
3-chloro-4-methylphenyl
methyl
ethyl



2.4.887
3-bromo-4-methylphenyl
methyl
ethyl



2.4.888
3,4-dimethylphenyl
methyl
ethyl



2.4.889
3,4-dimethylphenyl
ethyl
ethyl



2.4.890
3,4-dimethylphenyl
propyl
ethyl



2.4.891
3,4-dimethylphenyl
butyl
ethyl



2.4.892
3-cyclopropyl-4-methylphenyl
methyl
ethyl



2.4.893
3-cyano-4-methylphenyl
methyl
ethyl



2.4.894
3-trifluoromethyl-4-methylphenyl
methyl
ethyl



2.4.895
3-methoxy-4-methylphenyl
methyl
ethyl



2.4.896
3-ethoxy-4-methylphenyl
methyl
ethyl



2.4.897
3-trifluoromethoxy-4-methylphenyl
methyl
ethyl



2.4.898
3-nitro-4-methylphenyl
methyl
ethyl



2.4.899
3-fluoro-4-ethylphenyl
methyl
ethyl



2.4.900
3-chloro-4-ethylphenyl
methyl
ethyl



2.4.901
3-bromo-4-ethylphenyl
methyl
ethyl



2.4.902
3-methyl-4-ethylphenyl
methyl
ethyl



2.4.903
3,4-diethylphenyl
methyl
ethyl



2.4.904
3-cyclopropyl-4-ethylphenyl
methyl
ethyl



2.4.905
3-cyano-4-ethylphenyl
methyl
ethyl



2.4.906
3-trifluoromethyl-4-ethylphenyl
methyl
ethyl



2.4.907
3-methoxy-4-ethylphenyl
methyl
ethyl



2.4.908
3-ethoxy-4-ethylphenyl
methyl
ethyl



2.4.909
3-trifluoromethoxy-4-ethylphenyl
methyl
ethyl



2.4.910
3-nitro-4-ethylphenyl
methyl
ethyl



2.4.911
3-fluoro-4-isopropylphenyl
methyl
ethyl



2.4.912
3-chloro-4-isopropylphenyl
methyl
ethyl



2.4.913
3-bromo-4-isopropylphenyl
methyl
ethyl



2.4.914
3-methyl-4-isopropylphenyl
methyl
ethyl



2.4.915
3-cyclopropyl-4-isopropylphenyl
methyl
ethyl



2.4.916
3-cyano-4-isopropylphenyl
methyl
ethyl



2.4.917
3-trifluoromethyl-4-isopropylphenyl
methyl
ethyl



2.4.918
3-methoxy-4-isopropylphenyl
methyl
ethyl



2.4.919
3-ethoxy-4-isopropylphenyl
methyl
ethyl



2.4.920
3-trifluoromethoxy-4-
methyl
ethyl




isopropylphenyl





2.4.921
3-nitro-4-isopropylphenyl
methyl
ethyl



2.4.922
3-fluoro-4-tert-butylphenyl
methyl
ethyl



2.4.923
3-chloro-4-tert-butylphenyl
methyl
ethyl



2.4.924
3-bromo-4-tert-butylphenyl
methyl
ethyl



2.4.925
3-methyl-4-tert-butylphenyl
methyl
ethyl



2.4.926
3-ethyl-4-tert-butylphenyl
methyl
ethyl



2.4.927
3-cyclopropyl-4-tert-butylphenyl
methyl
ethyl



2.4.928
3-cyano-4-tert-butylphenyl
methyl
ethyl



2.4.929
3-trifluoromethyl-4-tert-butylphenyl
methyl
ethyl



2.4.930
3-trifluoromethyl-4-tert-butylphenyl
ethyl
ethyl



2.4.931
3-trifluoromethyl-4-tert-butylphenyl
propyl
ethyl



2.4.932
3-trifluoromethyl-4-tert-butylphenyl
butyl
ethyl



2.4.933
3-methoxy-4-tert-butylphenyl
methyl
ethyl



2.4.934
3-ethoxy-4-tert-butylphenyl
methyl
ethyl



2.4.935
3-trifluoromethoxy-4-tert-
methyl
ethyl




butylphenyl





2.4.936
3-nitro-4-tert-butylphenyl
methyl
ethyl



2.4.937
3-fluoro-4-cyclopropylphenyl
methyl
ethyl



2.4.938
3-chloro-4-cyclopropylphenyl
methyl
ethyl



2.4.939
3-bromo-4-cyclopropylphenyl
methyl
ethyl



2.4.940
3-methyl-4-cyclopropylphenyl
methyl
ethyl



2.4.941
3-cyclopropyl-4-cyclopropylphenyl
methyl
ethyl



2.4.942
3-cyano-4-cyclopropylphenyl
methyl
ethyl



2.4.943
3-trifluoromethyl-4-
methyl
ethyl




cyclopropylphenyl





2.4.944
3-methoxy-4-cyclopropylphenyl
methyl
ethyl



2.4.945
3-ethoxy-4-cyclopropylphenyl
methyl
ethyl



2.4.946
3-trifluoromethoxy-4-
methyl
ethyl




cyclopropylphenyl





2.4.947
3-fluoro-4-methoxycarbonylphenyl
methyl
ethyl



2.4.948
3-chloro-4-methoxy-carbonylphenyl
methyl
ethyl



2.4.949
3-bromo-4-methoxy-carbonylphenyl
methyl
ethyl



2.4.950
3-methyl-4-methoxy-carbonylphenyl
methyl
ethyl



2.4.951
3-cyclopropyl-4-methoxycarbonyl-
methyl
ethyl




phenyl





2.4.952
3-cyano-4-methoxycarbonylphenyl
methyl
ethyl



2.4.953
3-trifluoromethyl-4-
methyl
ethyl




methoxycarbonylphenyl





2.4.954
3-methoxy-4-methoxycarbonyl-
methyl
ethyl




phenyl





2.4.955
3-ethoxy-4-methoxycarbonylphenyl
methyl
ethyl



2.4.956
3-trifluoromethoxy-4-
methyl
ethyl




methoxycarbonylphenyl





2.4.957
3-nitro-4-methoxy-carbonylphenyl
methyl
ethyl



2.4.958
3-fluoro-4-cyanophenyl
methyl
ethyl



2.4.959
3-chloro-4-cyanophenyl
methyl
ethyl



2.4.960
3-bromo-4-cyanophenyl
methyl
ethyl



2.4.961
3-methyl-4-cyanophenyl
methyl
ethyl



2.4.962
3-cyclopropyl-4-cyanophenyl
methyl
ethyl



2.4.963
3,4-dicyanophenyl
methyl
ethyl



2.4.964
3-trifluoromethyl-4-cyanophenyl
methyl
ethyl



2.4.965
3-trifluoromethyl-4-cyanophenyl
ethyl
ethyl



2.4.966
3-trifluoromethyl-4-cyanophenyl
propyl
ethyl



2.4.967
3-trifluoromethyl-4-cyanophenyl
butyl
ethyl



2.4.968
3-methoxy-4-cyanophenyl
methyl
ethyl



2.4.969
3-ethoxy-4-cyanophenyl
methyl
ethyl



2.4.970
3-trifluoromethoxy-4-cyanophenyl
methyl
ethyl



2.4.971
3-nitro-4-cyanophenyl
methyl
ethyl



2.4.972
3-fluoro-4-methoxyphenyl
methyl
ethyl



2.4.973
3-chloro-4-methoxyphenyl
methyl
ethyl



2.4.974
3-bromo-4-methoxyphenyl
methyl
ethyl



2.4.975
3-methyl-4-methoxyphenyl
methyl
ethyl



2.4.976
3-ethyl-4-methoxyphenyl
methyl
ethyl



2.4.977
3-cyclopropyl-4-methoxyphenyl
methyl
ethyl



2.4.978
3-cyano-4-methoxyphenyl
methyl
ethyl



2.4.979
3-trifluoromethyl-4-methoxyphenyl
methyl
ethyl



2.4.980
3,4-dimethoxyphenyl
methyl
ethyl



2.4.981
3-ethoxy-4-methoxyphenyl
methyl
ethyl



2.4.982
3-trifluoromethoxy-4-
methyl
ethyl




methoxyphenyl





2.4.983
3-nitro-4-methoxyphenyl
methyl
ethyl



2.4.984
3-fluoro-4-ethoxyphenyl
methyl
ethyl



2.4.985
3-chloro-4-ethoxyphenyl
methyl
ethyl



2.4.986
3-chloro-4-ethoxyphenyl
ethyl
ethyl



2.4.987
3-chloro-4-ethoxyphenyl
propyl
ethyl



2.4.988
3-chloro-4-ethoxyphenyl
butyl
ethyl



2.4.989
3-bromo-4-ethoxyphenyl
methyl
ethyl



2.4.990
3-methyl-4-ethoxyphenyl
methyl
ethyl



2.4.991
3-cyclopropyl-4-ethoxyphenyl
methyl
ethyl



2.4.992
3-cyano-4-ethoxyphenyl
methyl
ethyl



2.4.993
3-trifluoromethyl-4-ethoxyphenyl
methyl
ethyl



2.4.994
3-methoxy-4-ethoxyphenyl
methyl
ethyl



2.4.995
2,4-diethoxyphenyl
methyl
ethyl



2.4.996
3-trifluoromethoxy-4-ethoxyphenyl
methyl
ethyl



2.4.997
3-nitro-4-ethoxyphenyl
methyl
ethyl



2.4.998
3-fluoro-4-propoxyphenyl
methyl
ethyl



2.4.999
3-chloro-4-propoxyphenyl
methyl
ethyl



2.4.1000
3-bromo-4-propoxyphenyl
methyl
ethyl



2.4.1001
3-methyl-4-propoxyphenyl
methyl
ethyl



2.4.1002
3-cyclopropyl-4-propoxyphenyl
methyl
ethyl



2.4.1003
3-cyano-4-propoxyphenyl
methyl
ethyl



2.4.1004
3-trifluoromethyl-4-propoxyphenyl
methyl
ethyl



2.4.1005
3-methoxy-4-propoxyphenyl
methyl
ethyl



2.4.1006
3-ethoxy-4-propoxyphenyl
methyl
ethyl



2.4.1007
3-trifluoromethoxy-4-propoxyphenyl
methyl
ethyl



2.4.1008
3-nitro-4-propoxyphenyl
methyl
ethyl



2.4.1009
3-fluoro-4-isopropoxyphenyl
methyl
ethyl



2.4.1010
3-chloro-4-isopropoxyphenyl
methyl
ethyl



2.4.1011
3-bromo-4-isopropoxyphenyl
methyl
ethyl



2.4.1012
3-methyl-4-isopropoxyphenyl
methyl
ethyl



2.4.1013
3-cyclopropyl-4-isopropoxyphenyl
methyl
ethyl



2.4.1014
3-cyano-4-isopropoxyphenyl
methyl
ethyl



2.4.1015
3-trifluoromethyl-4-
methyl
ethyl




isopropoxyphenyl





2.4.1016
3-methoxy-4-isopropoxyphenyl
methyl
ethyl



2.4.1017
3-ethoxy-4-isopropoxyphenyl
methyl
ethyl



2.4.1018
3-trifluoromethoxy-4-
methyl
ethyl




isopropoxyphenyl





2.4.1019
3-nitro-4-isopropoxyphenyl
methyl
ethyl



2.4.1020
3-fluoro-4-trifluoromethoxyphenyl
methyl
ethyl



2.4.1021
3-chloro-4-trifluoromethoxyphenyl
methyl
ethyl



2.4.1022
3-bromo-4-trifluoromethoxyphenyl
methyl
ethyl



2.4.1023
3-methyl-4-trifluoromethoxyphenyl
methyl
ethyl



2.4.1024
3-cyclopropyl-4-trifluoromethoxy-
methyl
ethyl




phenyl





2.4.1025
3-cyano-4-trifluoromethoxyphenyl
methyl
ethyl



2.4.1026
3-trifluoromethyl-4-trifluoromethoxy-
methyl
ethyl




phenyl





2.4.1027
3-methoxy-4-trifluoromethoxy-
methyl
ethyl




phenyl





2.4.1028
3-ethoxy-4-trifluoromethoxyphenyl
methyl
ethyl



2.4.1029
3,4-bis(trifluoromethoxy)phenyl
methyl
ethyl



2.4.1030
3-nitro-4-trifluoromethoxyphenyl
methyl
ethyl



2.4.1031
3-fluoro-4-difluoromethoxyphenyl
methyl
ethyl



2.4.1032
3-chloro-4-difluoromethoxyphenyl
methyl
ethyl



2.4.1033
3-bromo-4-difluoromethoxyphenyl
methyl
ethyl



2.4.1034
3-methyl-4-difluoromethoxy-henyl
methyl
ethyl



2.4.1035
3-cyclopropyl-4-difluoromethoxy-
methyl
ethyl




phenyl





2.4.1036
3-cyano-4-difluoromethoxyphenyl
methyl
ethyl



2.4.1037
3-trifluoromethyl-4-difluoromethoxy-
methyl
ethyl




phenyl





2.4.1038
3-methoxy-4-difluoromethoxy-
methyl
ethyl




phenyl





2.4.1039
3-ethoxy-4-difluoromethoxyphenyl
methyl
ethyl



2.4.1040
3-trifluoromethoxy-4-
methyl
ethyl




difluoromethoxyphenyl





2.4.1041
3-nitro-4-difluoromethoxyphenyl
methyl
ethyl



2.4.1042
3-fluoro-4-nitrophenyl
methyl
ethyl



2.4.1043
3-chloro-4-nitrophenyl
methyl
ethyl



2.4.1044
3-bromo-4-nitrophenyl
methyl
ethyl



2.4.1045
3-methyl-4-nitrophenyl
methyl
ethyl



2.4.1046
3-cyclopropyl-4-nitrophenyl
methyl
ethyl



2.4.1047
3-cyano-4-nitrophenyl
methyl
ethyl



2.4.1048
3-trifluoromethyl-4-nitrophenyl
methyl
ethyl



2.4.1049
3-methoxy-4-nitrophenyl
methyl
ethyl



2.4.1050
3-ethoxy-4-nitrophenyl
methyl
ethyl



2.4.1051
3-trifluoromethoxy-4-nitrophenyl
methyl
ethyl



2.4.1052
3-fluoro-4-methylsulfanylphenyl
methyl
ethyl



2.4.1053
3-chloro-4-methylsulfanylphenyl
methyl
ethyl



2.4.1054
3-bromo-4-methylsulfanylphenyl
methyl
ethyl



2.4.1055
3-methyl-4-methylsulfanylphenyl
methyl
ethyl



2.4.1056
3-cyclopropyl-4-
methyl
ethyl




methylsulfanylphenyl





2.4.1057
3-cyano-4-methylsulfanylphenyl
methyl
ethyl



2.4.1058
3-trifluoromethyl-4-
methyl
ethyl




methylsulfanylphenyl





2.4.1059 
3-methoxy-4-methylsulfanylphenyl
methyl
ethyl



2.4.1060
3-ethoxy-4-methylsulfanylphenyl
methyl
ethyl



2.4.1061
3-trifluoromethoxy-4-
methyl
ethyl




methylsulfanylphenyl





2.4.1062
3-nitro-4-methylsulfanylphenyl
methyl
ethyl



2.4.1063
3,6-difluorophenyl
methyl
ethyl



2.4.1064
3,6-difluorophenyl
ethyl
ethyl



2.4.1065
3,6-difluorophenyl
propyl
ethyl



2.4.1066
3,6-difluorophenyl
butyl
ethyl



2.4.1067
3-chloro-6-fluorophenyl
methyl
ethyl



2.4.1068
3-bromo-6-fluorophenyl
methyl
ethyl



2.4.1069
3-methyl-6-fluorophenyl
methyl
ethyl



2.4.1070
3-ethyl-6-fluorophenyl
methyl
ethyl



2.4.1071
3-cyclopropyl-6-fluorophenyl
methyl
ethyl



2.4.1072
3-cyano-6-fluorophenyl
methyl
ethyl



2.4.1073
3-methoxy-6-fluorophenyl
methyl
ethyl



2.4.1074
3-ethoxy-6-fluorophenyl
methyl
ethyl



2.4.1075
3-trifluoromethoxy-6-fluorophenyl
methyl
ethyl



2.4.1076
3-nitro-6-fluorophenyl
methyl
ethyl



2.4.1077
3-fluoro-6-chlorophenyl
methyl
ethyl



2.4.1078
3-fluoro-6-chlorophenyl
ethyl
ethyl



2.4.1079
3-fluoro-6-chlorophenyl
propyl
ethyl



2.4.1080
3-fluoro-6-chlorophenyl
butyl
ethyl



2.4.1081
3,6-dichlorophenyl
methyl
ethyl



2.4.1082
3,6-dichlorophenyl
ethyl
ethyl



2.4.1083
3,6-dichlorophenyl
propyl
ethyl



2.4.1084
3,6-dichlorophenyl
butyl
ethyl



2.4.1085
3-bromo-6-chlorophenyl
methyl
ethyl



2.4.1086
3-methyl-6-chlorophenyl
methyl
ethyl



2.4.1087
3-ethyl-6-chlorophenyl
methyl
ethyl



2.4.1088
3-cyclopropyl-6-chlorophenyl
methyl
ethyl



2.4.1089
3-cyano-6-chlorophenyl
methyl
ethyl



2.4.1090
3-trifluoromethyl-6-chlorophenyl
methyl
ethyl



2.4.1091
3-methoxy-6-chlorophenyl
methyl
ethyl



2.4.1092
3-ethoxy-6-chlorophenyl
methyl
ethyl



2.4.1093 
3-trifluoromethoxy-6-chlorophenyl
methyl
ethyl



2.4.1094
3-nitro-6-chlorophenyl
methyl
ethyl



2.4.1095
3-fluoro-6-bromophenyl
methyl
ethyl



2.4.1096
3-chloro-6-bromophenyl
methyl
ethyl



2.4.1097
3,6-dibromophenyl
methyl
ethyl



2.4.1098
3-methyl-6-bromophenyl
methyl
ethyl



2.4.1099
3-ethyl-6-bromophenyl
methyl
ethyl



2.4.1100
3-cyclopropyl-6-bromophenyl
methyl
ethyl



2.4.1101
3-cyano-6-bromophenyl
methyl
ethyl



2.4.1102
3-trifluoromethyl-6-bromophenyl
methyl
ethyl



2.4.1103
3-methoxy-6-phenyl
methyl
ethyl



2.4.1104
3-ethoxy-6-bromophenyl
methyl
ethyl



2.4.1105
3-trifluoromethoxy-6-bromophenyl
methyl
ethyl



2.4.1106
3-nitro-6-bromophenyl
methyl
ethyl



2.4.1107
3-fluoro-6-iodophenyl
methyl
ethyl



2.4.1108
3-chloro-6-iodophenyl
methyl
ethyl



2.4.1109
3-bromo-6-iodophenyl
methyl
ethyl



2.4.1110
3-methyl-6-iodophenyl
methyl
ethyl



2.4.1111
3-ethyl-6-iodophenyl
methyl
ethyl



2.4.1112
3-cyclopropyl-6-iodophenyl
methyl
ethyl



2.4.1113
3-cyano-6-iodophenyl
methyl
ethyl



2.4.1114
3-trifluoromethyl-6-iodophenyl
methyl
ethyl



2.4.1115
3-methoxy-6-iodophenyl
methyl
ethyl



2.4.1116
3-ethoxy-6-iodophenyl
methyl
ethyl



2.4.1117
3-trifluoromethoxy-6-iodophenyl
methyl
ethyl



2.4.1118
3-nitro-6-iodophenyl
methyl
ethyl



2.4.1119
3-fluoro-6-methylphenyl
methyl
ethyl



2.4.1120
3-chloro-6-methylphenyl
methyl
ethyl



2.4.1121
3-bromo-6-methylphenyl
methyl
ethyl



2.4.1122
3,6-dimethylphenyl
methyl
ethyl



2.4.1123
3-ethyl-6-methylphenyl
methyl
ethyl



2.4.1124
3-cyclopropyl-6-methylphenyl
methyl
ethyl



2.4.1125
3-cyano-6-methylphenyl
methyl
ethyl



2.4.1126
3-trifluoromethyl-6-methylphenyl
methyl
ethyl



2.4.1127
3-methoxy-6-methylphenyl
methyl
ethyl



2.4.1128
3-ethoxy-6-methylphenyl
methyl
ethyl



2.4.1129 
3-trifluoromethoxy-6-methylphenyl
methyl
ethyl



2.4.1130
3-nitro-6-methylphenyl
methyl
ethyl



2.4.1131
3-fluoro-6-ethylphenyl
methyl
ethyl



2.4.1132
3-chloro-6-ethylphenyl
methyl
ethyl



2.4.1133
3-bromo-6-ethylphenyl
methyl
ethyl



2.4.1134
3-methyl-6-ethylphenyl
methyl
ethyl



2.4.1135
3,6-diethylphenyl
methyl
ethyl



2.4.1136
3-cyclopropyl-6-ethylphenyl
methyl
ethyl



2.4.1137
3-cyano-6-ethylphenyl
methyl
ethyl



2.4.1138
3-trifluoromethyl-6-ethylphenyl
methyl
ethyl



2.4.1139
3-methoxy-6-ethylphenyl
methyl
ethyl



2.4.1140
3-ethoxy-6-ethylphenyl
methyl
ethyl



2.4.1141
3-trifluoromethoxy-6-ethylphenyl
methyl
ethyl



2.4.1142
3-nitro-6-ethylphenyl
methyl
ethyl



2.4.1143
3-fluoro-6-propylphenyl
methyl
ethyl



2.4.1144
3-chloro-6-propylphenyl
methyl
ethyl



2.4.1145
3-bromo-6-propylphenyl
methyl
ethyl



2.4.1146
3-methyl-6-propylphenyl
methyl
ethyl



2.4.1147
3-methyl-6-propylphenyl
methyl
ethyl



2.4.1148
3-cyclopropyl-6-propylphenyl
methyl
ethyl



2.4.1149
3-cyano-6-propylphenyl
methyl
ethyl



2.4.1150
3-trifluoromethyl-6-propylphenyl
methyl
ethyl



2.4.1151
3-methoxy-6-propylphenyl
methyl
ethyl



2.4.1152
3-ethoxy-6-propylphenyl
methyl
ethyl



2.4.1153
3-trifluoromethoxy-6-propylphenyl
methyl
ethyl



2.4.1154
3-nitro-6-propylphenyl
methyl
ethyl



2.4.1155
3-fluoro-6-isopropylphenyl
methyl
ethyl



2.4.1156
3-chloro-6-isopropylphenyl
methyl
ethyl



2.4.1157
3-bromo-6-isopropylphenyl
methyl
ethyl



2.4.1158
3-methyl-6-isopropylphenyl
methyl
ethyl



2.4.1159
3-cyclopropyl-6-isopropylphenyl
methyl
ethyl



2.4.1160
3-cyano-6-isopropylphenyl
methyl
ethyl



2.4.1161
3-trifluoromethyl-6-isopropylphenyl
methyl
ethyl



2.4.1162
3-methoxy-6-isopropylphenyl
methyl
ethyl



2.4.1163
3-ethoxy-6-isopropylphenyl
methyl
ethyl



2.4.1164
3-trifluoromethoxy-6-
methyl
ethyl




isopropylphenyl





2.4.1165
3-nitro-6-isopropylphenyl
methyl
ethyl



2.4.1166
3-fluoro-6-tert-butylphenyl
methyl
ethyl



2.4.1167
3-chloro-6-tert-butylphenyl
methyl
ethyl



2.4.1168
3-bromo-6-tert-butylphenyl
methyl
ethyl



2.4.1169
3-methyl-6-tert-butylphenyl
methyl
ethyl



2.4.1170
3-cyclopropyl-6-tert-butylphenyl
methyl
ethyl



2.4.1171
3-cyano-6-tert-butylphenyl
methyl
ethyl



2.4.1172
3-trifluoromethyl-6-tert-butylphenyl
methyl
ethyl



2.4.1173
3-methoxy-6-tert-butylphenyl
methyl
ethyl



2.4.1174
3-ethoxy-6-tert-butylphenyl
methyl
ethyl



2.4.1175
3-trifluoromethoxy-6-tert-
methyl
ethyl




butylphenyl





2.4.1176
3-nitro-6-tert-butylphenyl
methyl
ethyl



2.4.1177
3-fluoro-6-cyclopropylphenyl
methyl
ethyl



2.4.1178
3-chloro-6-cyclopropylphenyl
methyl
ethyl



2.4.1179
3-bromo-6-cyclopropylphenyl
methyl
ethyl



2.4.1180
3-methyl-6-cyclopropylphenyl
methyl
ethyl



2.4.1181
3-cyclopropyl-6-cyclopropylphenyl
methyl
ethyl



2.4.1182
3-cyano-6-cyclopropylphenyl
methyl
ethyl



2.4.1183
3-trifluoromethyl-6-cyclopropylphenyl
methyl
ethyl



2.4.1184
3-methoxy-6-cyclopropylphenyl
methyl
ethyl



2.4.1185
3-ethoxy-6-cyclopropylphenyl
methyl
ethyl



2.4.1186
3-trifluoromethoxy-6-
methyl
ethyl




cyclopropylphenyl





2.4.1187
3-fluoro-6-methoxycarbonylphenyl
methyl
ethyl



2.4.1188
3-chloro-6-methoxycarbonylphenyl
methyl
ethyl



2.4.1189
3-bromo-6-methoxycarbonylphenyl
methyl
ethyl



2.4.1190
3-methyl-6-methoxycarbonylphenyl
methyl
ethyl



2.4.1191
3-cyclopropyl-6-methoxycarbonylphenyl
methyl
ethyl



2.4.1192
3-cyano-6-methoxycarbonylphenyl
methyl
ethyl



2.4.1193
3-trifluoromethyl-6-methoxycarbonylphenyl
methyl
ethyl



2.4.1194
3-methoxy-6-methoxycarbonylphenyl
methyl
ethyl



2.4.1195
3-ethoxy-6-methoxycarbonylphenyl
methyl
ethyl



2.4.1196
3-trifluoromethoxy-6-
methyl
ethyl




methoxycarbonyl-phenyl





2.4.1197
3-nitro-6-methoxycarbonylphenyl
methyl
ethyl



2.4.1198
3-fluoro-6-cyanophenyl
methyl
ethyl



2.4.1199
3-chloro-6-cyanophenyl
methyl
ethyl



2.4.1200
3-bromo-6-cyanophenyl
methyl
ethyl



2.4.1201
3-methyl-6-cyanophenyl
methyl
ethyl



2.4.1202
3-cyclopropyl-6-cyanophenyl
methyl
ethyl



2.4.1203
3-cyano-6-cyanophenyl
methyl
ethyl



2.4.1204
3-trifluoromethyl-6-cyanophenyl
methyl
ethyl



2.4.1205
3-methoxy-6-cyanophenyl
methyl
ethyl



2.4.1206
3-ethoxy-6-cyanophenyl
methyl
ethyl



2.4.1207
3-trifluoromethoxy-6-cyanophenyl
methyl
ethyl



2.4.1208
3-nitro-6-cyanophenyl
methyl
ethyl



2.4.1209
3-fluoro-6-methoxyphenyl
methyl
ethyl



2.4.1210
3-chloro-6-methoxyphenyl
methyl
ethyl



2.4.1211
3-bromo-6-methoxyphenyl
methyl
ethyl



2.4.1212
3-methyl-6-methoxyphenyl
methyl
ethyl



2.4.1213
3-cyclopropyl-6-methoxyphenyl
methyl
ethyl



2.4.1214
3-cyano-6-methoxyphenyl
methyl
ethyl



2.4.1215 
3-trifluoromethyl-6-methoxyphenyl
methyl
ethyl



2.4.1216
3,6-dimethoxyphenyl
methyl
ethyl



2.4.1217
3-ethoxy-6-methoxyphenyl
methyl
ethyl



2.4.1218
3-trifluoromethoxy-6-
methyl
ethyl




methoxyphenyl





2.4.1219
3-nitro-6-methoxyphenyl
methyl
ethyl



2.4.1220
3-fluoro-6-ethoxyphenyl
methyl
ethyl



2.4.1221
3-chloro-6-ethoxyphenyl
methyl
ethyl



2.4.1222
3-bromo-6-ethoxyphenyl
methyl
ethyl



2.4.1223
3-methyl-6-ethoxyphenyl
methyl
ethyl



2.4.1224
3-cyclopropyl-6-ethoxyphenyl
methyl
ethyl



2.4.1225
3-cyano-6-ethoxyphenyl
methyl
ethyl



2.4.1226
3-trifluoromethyl-6-ethoxyphenyl
methyl
ethyl



2.4.1227
3-methoxy-6-ethoxyphenyl
methyl
ethyl



2.4.1228
2,6-diethoxyphenyl
methyl
ethyl



2.4.1229
3-trifluoromethoxy-6-ethoxyphenyl
methyl
ethyl



2.4.1230
3-nitro-6-ethoxyphenyl
methyl
ethyl



2.4.1231
3-fluoro-6-propoxyphenyl
methyl
ethyl



2.4.1232
3-chloro-6-propoxyphenyl
methyl
ethyl



2.4.1233
3-bromo-6-propoxyphenyl
methyl
ethyl



2.4.1234
3-methyl-6-propoxyphenyl
methyl
ethyl



2.4.1235
3-cyclopropyl-6-propoxyphenyl
methyl
ethyl



2.4.1236
3-cyano-6-propoxyphenyl
methyl
ethyl



2.4.1237
3-trifluoromethyl-6-propoxyphenyl
methyl
ethyl



2.4.1238
3-methoxy-6-propoxyphenyl
methyl
ethyl



2.4.1239
3-ethoxy-6-propoxyphenyl
methyl
ethyl



2.4.1240
3-trifluoromethoxy-6-propoxyphenyl
methyl
ethyl



2.4.1241
3-nitro-6-propoxyphenyl
methyl
ethyl



2.4.1242
3-fluoro-6-isopropoxyphenyl
methyl
ethyl



2.4.1243
3-chloro-6-isopropoxyphenyl
methyl
ethyl



2.4.1244
3-bromo-6-isopropoxyphenyl
methyl
ethyl



2.4.1245
3-methyl-6-isopropoxyphenyl
methyl
ethyl



2.4.1246
3-cyclopropyl-6-isopropoxyphenyl
methyl
ethyl



2.4.1247
3-cyano-6-isopropoxyphenyl
methyl
ethyl



2.4.1248
3-trifluoromethyl-6-
methyl
ethyl




isopropoxyphenyl





2.4.1249
3-methoxy-6-isopropoxyphenyl
methyl
ethyl



2.4.1250
3-ethoxy-6-isopropoxyphenyl
methyl
ethyl



2.4.1251
3-trifluoromethoxy-6-
methyl
ethyl




isopropoxyphenyl





2.4.1252
3-nitro-6-isopropoxyphenyl
methyl
ethyl



2.4.1253
3-fluoro-6-trifluoromethoxyphenyl
methyl
ethyl



2.4.1254
3-chloro-6-trifluoromethoxyphenyl
methyl
ethyl



2.4.1255
3-bromo-6-trifluoromethoxyphenyl
methyl
ethyl



2.4.1256
3-methyl-6-trifluoromethoxyphenyl
methyl
ethyl



2.4.1257
3-cyclopropyl-6-trifluoromethoxy-
methyl
ethyl




phenyl





2.4.1258
3-cyano-6-trifluoromethoxyphenyl
methyl
ethyl



2.4.1259
3-trifluoromethyl-6-trifluoromethoxy- 
methyl
ethyl




phenyl





2.4.1260
3-methoxy-6-trifluoromethoxy-
methyl
ethyl




phenyl





2.4.1261
3-ethoxy-6-trifluoromethoxyphenyl
methyl
ethyl



2.4.1262
3,6-bis(trifluoro-methoxy)phenyl
methyl
ethyl



2.4.1263
3-nitro-6-trifluoromethoxyphenyl
methyl
ethyl



2.4.1264
3-fluoro-6-difluoromethoxyphenyl
methyl
ethyl



2.4.1265
3-chloro-6-difluoromethoxyphenyl
methyl
ethyl



2.4.1266
3-bromo-6-difluoromethoxyphenyl
methyl
ethyl



2.4.1267
3-methyl-6-difluoromethoxyphenyl
methyl
ethyl



2.4.1268
3-cyclopropyl-6-difluoromethoxy-
methyl
ethyl




phenyl





2.4.1269
3-cyano-6-difluoromethoxyphenyl
methyl
ethyl



2.4.1270
3-trifluoromethyl-6-
methyl
ethyl




difluoromethoxyphenyl





2.4.1271
3-methoxy-6-difluoromethoxy-
methyl
ethyl




phenyl





2.4.1272
3-ethoxy-6-difluoromethoxyphenyl
methyl
ethyl



2.4.1273
3-trifluoromethoxy-6-
methyl
ethyl




difluoromethoxyphenyl





2.4.1274
3-nitro-6-difluoromethoxyphenyl
methyl
ethyl



2.4.1275
3-fluoro-6-nitrophenyl
methyl
ethyl



2.4.1276
3-chloro-6-nitrophenyl
methyl
ethyl



2.4.1277
3-bromo-6-nitrophenyl
methyl
ethyl



2.4.1278
3-methyl-6-nitrophenyl
methyl
ethyl



2.4.1279
3-cyclopropyl-6-nitrophenyl
methyl
ethyl



2.4.1280
3-cyano-6-nitrophenyl
methyl
ethyl



2.4.1281
3-trifluoromethyl-6-nitrophenyl
methyl
ethyl



2.4.1282
3-methoxy-6-nitrophenyl
methyl
ethyl



2.4.1283
3-ethoxy-6-nitrophenyl
methyl
ethyl



2.4.1284
3-trifluoromethoxy-6-nitrophenyl
methyl
ethyl



2.4.1285
3-fluoro-6-methylsulfanylphenyl
methyl
ethyl



2.4.1286
3-chloro-6-methylsulfanylphenyl
methyl
ethyl



2.4.1287
3-bromo-6-methylsulfanylphenyl
methyl
ethyl



2.4.1288
3-methyl-6-methylsulfanylphenyl
methyl
ethyl



2.4.1289
3-cyclopropyl-6-
methyl
ethyl




methylsulfanylphenyl





2.4.1290
3-cyano-6-methylsulfanylphenyl
methyl
ethyl



2.4.1291
3-trifluoromethyl-6-
methyl
ethyl




methylsulfanylphenyl





2.4.1292
3-methoxy-6-methylsulfanylphenyl
methyl
ethyl



2.4.1293
3-ethoxy-6-methylsulfanylphenyl
methyl
ethyl



2.4.1294
3-trifluoromethoxy-6-
methyl
ethyl




methylsulfanylphenyl





2.4.1295
3-nitro-6-methylsulfanylphenyl
methyl
ethyl



2.4.1296
2,3,4-trifluorophenyl
methyl
ethyl



2.4.1297
2,3,4-trichlorophenyl
methyl
ethyl



2.4.1298
2,3,4-trimethylphenyl
methyl
ethyl



2.4.1299
2-fluoro-2-chloro-5-trifluoromethyl-
methyl
ethyl




phenyl





2.4.1300
2,3,5-trifluorophenyl
methyl
ethyl



2.4.1301
2,3,5-trichlorophenyl
methyl
ethyl



2.4.1302
2,3,5-trimethylphenyl
methyl
ethyl



2.4.1303
2,3-dichloro-5-methoxyphenyl
methyl
ethyl



2.4.1304
2,3,6-trifluorophenyl
methyl
ethyl



2.4.1305
2,3,6-trichlorophenyl
methyl
ethyl



2.4.1306
2,3,6-trimethylphenyl
methyl
ethyl



2.4.1307
3,4,5-trifluorophenyl
methyl
ethyl



2.4.1308
3,4,5-trichlorophenyl
methyl
ethyl



2.4.1309
3,4,5-trimethylphenyl
methyl
ethyl



2.4.1310
3,5-dimethyl-4-fluorophenyl
methyl
ethyl



2.4.1311
3,5-dichloro-4-methoxyphenyl
methyl
ethyl



2.4.1312
3,5-difluoro-4-chlorophenyl
methyl
ethyl



2.4.1313
3,5-dichloro-4-hydroxyphenyl
methyl
ethyl



2.4.1314
3,5-trifluoromethyl-4-chlorophenyl
methyl
ethyl



2.4.1315
3,4,6-trifluorophenyl
methyl
ethyl



2.4.1316
3,4,6-trichlorophenyl
methyl
ethyl



2.4.1317
3,4,6-trimethylphenyl
methyl
ethyl



2.4.1318
pentafluorophenyl
methyl
ethyl
















TABLE 2.5







Inventive compounds of the general formula (I) in which W* is COOY, 


R1 and R2 are each hydrogen, and aryl is the radical.








 











No.
Aryl
R3
Y
Physical data





2.5.1
3-fluorophenyl
hydroxymethyl
ethyl



2.5.2
3-fluorophenyl
1-hydroxyethyl
methyl
[CDCl3] D1 1.20






(d, 3H); 2.39 (d br, 1H);






3.60 (d, 1H); 3.71






(d, 1H); 3.83 (s, 3H);






4.30-4.37 (m, 1H); 7.13






(t, 1H); 7.34-7.45






(m, 2H). D2 1.28






(d, 3H); 2.1 7(d br, 1H);






3.56 (d, 1H); 3.76






(d, 1H); 3.84 (s, 3H);






4.20-4.28 (m, 1H); 7.13






(t, 1H); 7.34-7.45






(m, 3H).


2.5.3
3-fluorophenyl
1-hydroxypropyl
ethyl



2.5.4
3-fluorophenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.5
3-fluorophenyl
methoxymethyl
ethyl



2.5.6
3-fluorophenyl
2-methoxyethyl
ethyl



2.5.7
3-chlorophenyl
hydroxymethyl
ethyl



2.5.8
3-chlorophenyl
1-hydroxyethyl
ethyl



2.5.9
3-chlorophenyl
1-hydroxypropyl
ethyl



2.5.10
3-chlorophenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.11
3-chlorophenyl
methoxymethyl
ethyl



2.5.12
3-chlorophenyl
2-methoxyethyl
ethyl



2.5.13
3-bromophenyl
hydroxymethyl
ethyl



2.5.14
3-bromophenyl
1-hydroxyethyl
ethyl



2.5.15
3-iodophenyl
hydroxymethyl
ethyl



2.5.16
3-iodophenyl
1-hydroxyethyl
ethyl



2.5.17
3-methylphenyl
hydroxymethyl
ethyl



2.5.18
3-methylphenyl
1-hydroxyethyl
ethyl



2.5.19
3-ethylphenyl
hydroxymethyl
ethyl



2.5.20
3-propylphenyl
hydroxymethyl
ethyl



2.5.21
3-isopropylphenyl
hydroxymethyl
ethyl



2.5.22
3-n-butylphenyl
hydroxymethyl
ethyl



2.5.23
3-i-butylphenyl
hydroxymethyl
ethyl



2.5.24
3-tert-butylphenyl
hydroxymethyl
ethyl



2.5.25
3-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.26
3-cyclobutylphenyl
hydroxymethyl
ethyl



2.5.27
3-cyclopentylphenyl
hydroxymethyl
ethyl



2.5.28
3-vinylphenyl
hydroxymethyl
ethyl



2.5.29
3-ethynylphenyl
hydroxymethyl
ethyl



2.5.30
3-cyanophenyl
hydroxymethyl
ethyl



2.5.31
3-trifluoromethylphenyl
hydroxymethyl
ethyl



2.5.32
3-difluoromethylphenyl
hydroxymethyl
ethyl



2.5.33
3-(hydroxycarbonyl)phenyl
hydroxymethyl
ethyl



2.5.34
3-(methoxycarbonyl)phenyl
hydroxymethyl
ethyl



2.5.35
3-(ethoxycarbonyl)phenyl
hydroxymethyl
ethyl



2.5.36
3-hydroxymethylphenyl
hydroxymethyl
ethyl



2.5.37
3-carbamoylphenyl
hydroxymethyl
ethyl



2.5.38
3-hydroxyphenyl
hydroxymethyl
ethyl



2.5.39
3-methoxyphenyl
hydroxymethyl
ethyl



2.5.40
3-ethoxyphenyl
hydroxymethyl
ethyl



2.5.41
3-propyloxyphenyl
hydroxymethyl
ethyl



2.5.42
3-isopropyloxyphenyl
hydroxymethyl
ethyl



2.5.43
3-n-butyloxyphenyl
hydroxymethyl
ethyl



2.5.44
3-i-butyloxyphenyl
hydroxymethyl
ethyl



2.5.45
3-t-butyloxyphenyl
hydroxymethyl
ethyl



2.5.46
3-difluoromethoxyphenyl
hydroxymethyl
ethyl



2.5.47
3-trifluoromethoxyphenyl
hydroxymethyl
ethyl



2.5.48
3-(2,2,2-trifluoroethoxy)phenyl
hydroxymethyl
ethyl



2.5.49
3-(2-chloroethoxy)phenyl
hydroxymethyl
ethyl



2.5.50
3-(2-hydroxyethoxy)phenyl
hydroxymethyl
ethyl



2.5.51
3-(2-methoxyethoxy)phenyl
hydroxymethyl
ethyl



2.5.52
3-[(tert-butoxycarbonyl)oxy]-phenyl
hydroxymethyl
ethyl



2.5.53
3-nitrophenyl
hydroxymethyl
ethyl



2.5.54
3-acetoxyphenyl
hydroxymethyl
ethyl



2.5.55
{3-[(tert-butoxycarbonyl)amino]-
hydroxymethyl
ethyl




phenyl}





2.5.56
3-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.57
3-ethylsulfanylphenyl
hydroxymethyl
ethyl



2.5.58
3-(pentafluoro-lambda6-sulfanyl)phenyl
hydroxymethyl
ethyl



2.5.59
2,3-difluorophenyl
hydroxymethyl
ethyl



2.5.60
2,3-difluorophenyl
1-hydroxyethyl
ethyl



2.5.61
2,3-difluorophenyl
1-hydroxypropyl
ethyl



2.5.62
2,3-difluorophenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.63
2,3-difluorophenyl
methoxymethyl
ethyl



2.5.64
2,3-difluorophenyl
2-methoxyethyl
ethyl



2.5.65
2-chloro-3-fluorophenyl
hydroxymethyl
ethyl



2.5.66
2-bromo-3-fluorophenyl
hydroxymethyl
ethyl



2.5.67
2-methyl-3-fluorophenyl
hydroxymethyl
ethyl



2.5.68
2-ethyl-3-fluorophenyl
hydroxymethyl
ethyl



2.5.69
2-cyclopropyl-3-fluorophenyl
hydroxymethyl
ethyl



2.5.70
2-vinyl-3-fluorophenyl
hydroxymethyl
ethyl



2.5.71
2-ethynyl-3-fluorophenyl
hydroxymethyl
ethyl



2.5.72
2-cyano-3-fluorophenyl
hydroxymethyl
ethyl



2.5.73
2-methoxy-3-fluorophenyl
hydroxymethyl
ethyl



2.5.74
2-ethoxy-3-fluorophenyl
hydroxymethyl
ethyl



2.5.75
2-trifluoromethoxy-3-fluorophenyl
hydroxymethyl
ethyl



2.5.76
2-nitro-3-fluorophenyl
hydroxymethyl
ethyl



2.5.77
2-fluoro-3-chlorophenyl
hydroxymethyl
ethyl



2.5.78
2,3-dichlorophenyl
hydroxymethyl
ethyl



2.5.79
2,3-dichlorophenyl
1-hydroxyethyl
ethyl



2.5.80
2,3-dichlorophenyl
1-hydroxypropyl
ethyl



2.5.81
2,3-dichlorophenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.82
2,3-dichlorophenyl
methoxymethyl
ethyl



2.5.83
2,3-dichlorophenyl
2-methoxyethyl
ethyl



2.5.84
2-bromo-3-chlorophenyl
hydroxymethyl
ethyl



2.5.85
2-methyl-3-chlorophenyl
hydroxymethyl
ethyl



2.5.86
2-ethyl-3-chlorophenyl
hydroxymethyl
ethyl



2.5.87
2-cyclopropyl-3-chlorophenyl
hydroxymethyl
ethyl



2.5.88
2-vinyl-3-chlorophenyl
hydroxymethyl
ethyl



2.5.89
2-ethynyl-3-chlorophenyl
hydroxymethyl
ethyl



2.5.90
2-cyano-3-chlorophenyl
hydroxymethyl
ethyl



2.5.91
2-trifluoromethyl-2-chlorophenyl
hydroxymethyl
ethyl



2.5.92
2-methoxy-3-chlorophenyl
hydroxymethyl
ethyl



2.5.93
2-ethoxy-3-chlorophenyl
hydroxymethyl
ethyl



2.5.94
2-trifluoromethoxy-3-chlorophenyl
hydroxymethyl
ethyl



2.5.95
2-nitro-3-chlorophenyl
hydroxymethyl
ethyl



2.5.96
2-fluoro-3-bromophenyl
hydroxymethyl
ethyl



2.5.97
2-chloro-3-bromophenyl
hydroxymethyl
ethyl



2.5.98
2,3-dibromophenyl
hydroxymethyl
ethyl



2.5.99
2-methyl-3-bromophenyl
hydroxymethyl
ethyl



2.5.100
2-ethyl-3-bromophenyl
hydroxymethyl
ethyl



2.5.101
2-cyclopropyl-3-bromophenyl
hydroxymethyl
ethyl



2.5.102
2-vinyl-3-bromophenyl
hydroxymethyl
ethyl



2.5.103
2-ethynyl-3-bromophenyl
hydroxymethyl
ethyl



2.5.104
2-cyano-3-bromophenyl
hydroxymethyl
ethyl



2.5.105
2-trifluoromethyl-3-bromophenyl
hydroxymethyl
ethyl



2.5.106
2-methoxy-3-phenyl
hydroxymethyl
ethyl



2.5.107
2-ethoxy-3-bromophenyl
hydroxymethyl
ethyl



2.5.108
2-trifluoromethoxy-3-bromophenyl
hydroxymethyl
ethyl



2.5.109
2-nitro-3-bromophenyl
hydroxymethyl
ethyl



2.5.110
2-fluoro-3-iodophenyl
hydroxymethyl
ethyl



2.5.111
2-chloro-3-iodophenyl
hydroxymethyl
ethyl



2.5.112
2-bromo-3-iodophenyl
hydroxymethyl
ethyl



2.5.113
2-methyl-3-iodophenyl
hydroxymethyl
ethyl



2.5.114
2-ethyl-3-iodophenyl
hydroxymethyl
ethyl



2.5.115
2-cyclopropyl-3-iodophenyl
hydroxymethyl
ethyl



2.5.116
2-vinyl-3-iodophenyl
hydroxymethyl
ethyl



2.5.117
2-ethynyl-3-iodophenyl
hydroxymethyl
ethyl



2.5.118
2-cyano-3-iodophenyl
hydroxymethyl
ethyl



2.5.119
2-trifluoromethyl-3-iodophenyl
hydroxymethyl
ethyl



2.5.120
2-methoxy-3-iodophenyl
hydroxymethyl
ethyl



2.5.121
2-ethoxy-3-iodophenyl
hydroxymethyl
ethyl



2.5.122
2-trifluoromethoxy-3-iodophenyl
hydroxymethyl
ethyl



2.5.123
2-nitro-3-iodophenyl
hydroxymethyl
ethyl



2.5.124
2-fluoro-3-methylphenyl
hydroxymethyl
ethyl



2.5.125
2-fluoro-3-methylphenyl
1-hydroxyethyl
ethyl



2.5.126
2-fluoro-3-methylphenyl
1-hydroxypropyl
ethyl



2.5.127
2-fluoro-3-methylphenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.128
2-fluoro-3-methylphenyl
methoxymethyl
ethyl



2.5.129
2-fluoro-3-methylphenyl
2-methoxyethyl
ethyl



2.5.130
2-chloro-3-methylphenyl
hydroxymethyl
ethyl



2.5.131
2-chloro-3-methylphenyl
1-hydroxyethyl
ethyl



2.5.132
2-chloro-3-methylphenyl
1-hydroxypropyl
ethyl



2.5.133
2-chloro-3-methylphenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.134
2-chloro-3-methylphenyl
methoxymethyl
ethyl



2.5.135
2-chloro-3-methylphenyl
2-methoxyethyl
ethyl



2.5.136
2-bromo-3-methylphenyl
hydroxymethyl
ethyl



2.5.137
2,3-dimethylphenyl
hydroxymethyl
ethyl



2.5.138
2,3-dimethylphenyl
1-hydroxyethyl
ethyl



2.5.139
2,3-dimethylphenyl
1-hydroxypropyl
ethyl



2.5.140
2,3-dimethylphenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.141
2,3-dimethylphenyl
methoxymethyl
ethyl



2.5.142
2,3-dimethylphenyl
2-methoxyethyl
ethyl



2.5.143
2-ethyl-3-methylphenyl
hydroxymethyl
ethyl



2.5.144
2-cyclopropyl-3-methylphenyl
hydroxymethyl
ethyl



2.5.145
2-vinyl-3-methylphenyl
hydroxymethyl
ethyl



2.5.146
2-ethynyl-3-methylphenyl
hydroxymethyl
ethyl



2.5.147
2-cyano-3-methylphenyl
hydroxymethyl
ethyl



2.5.148
2-trifluoromethyl-3-methylphenyl
hydroxymethyl
ethyl



2.5.149
2-methoxy-3-methylphenyl
hydroxymethyl
ethyl



2.5.150
2-ethoxy-3-methylphenyl
hydroxymethyl
ethyl



2.5.151
2-trifluoromethoxy-3-methylphenyl
hydroxymethyl
ethyl



2.5.152
2-nitro-3-methylphenyl
hydroxymethyl
ethyl



2.5.153
2-fluoro-3-ethylphenyl
hydroxymethyl
ethyl



2.5.154
2-chloro-3-ethylphenyl
hydroxymethyl
ethyl



2.5.155
2-bromo-3-ethylphenyl
hydroxymethyl
ethyl



2.5.156
2-methyl-3-ethylphenyl
hydroxymethyl
ethyl



2.5.157
2,3-diethylphenyl
hydroxymethyl
ethyl



2.5.158
2-cyclopropyl-3-ethylphenyl
hydroxymethyl
ethyl



2.5.159
2-vinyl-3-ethylphenyl
hydroxymethyl
ethyl



2.5.160
2-ethynyl-3-ethylphenyl
hydroxymethyl
ethyl



2.5.161
2-cyano-3-ethylphenyl
hydroxymethyl
ethyl



2.5.162
2-trifluoromethyl-3-ethylphenyl
hydroxymethyl
ethyl



2.5.163
2-methoxy-3-ethylphenyl
hydroxymethyl
ethyl



2.5.164
2-ethoxy-3-ethylphenyl
hydroxymethyl
ethyl



2.5.165
2-trifluoromethoxy-3-ethylphenyl
hydroxymethyl
ethyl



2.5.166
2-nitro-3-ethylphenyl
hydroxymethyl
ethyl



2.5.167
2-fluoro-3-propylphenyl
hydroxymethyl
ethyl



2.5.168
2-chloro-3-propylphenyl
hydroxymethyl
ethyl



2.5.169
2-bromo-3-propylphenyl
hydroxymethyl
ethyl



2.5.170
2-methyl-3-propylphenyl
hydroxymethyl
ethyl



2.5.171
2-methyl-3-propylphenyl
hydroxymethyl
ethyl



2.5.172
2-cyclopropyl-3-propylphenyl
hydroxymethyl
ethyl



2.5.173
2-vinyl-3-propylphenyl
hydroxymethyl
ethyl



2.5.174
2-ethynyl-3propylphenyl
hydroxymethyl
ethyl



2.5.175
2-cyano-3-propylphenyl
hydroxymethyl
ethyl



2.5.176
2-trifluoromethyl-3-propylphenyl
hydroxymethyl
ethyl



2.5.177
2-methoxy-3-propylphenyl
hydroxymethyl
ethyl



2.5.178
2-ethoxy-3-propylphenyl
hydroxymethyl
ethyl



2.5.179
2-trifluoromethoxy-3-propylphenyl
hydroxymethyl
ethyl



2.5.180
2-nitro-3-propylphenyl
hydroxymethyl
ethyl



2.5.181
2-fluoro-3-isopropylphenyl
hydroxymethyl
ethyl



2.5.182
2-chloro-3-isopropylphenyl
hydroxymethyl
ethyl



2.5.183
2-bromo-3-isopropylphenyl
hydroxymethyl
ethyl



2.5.184
2-methyl-3-isopropylphenyl
hydroxymethyl
ethyl



2.5.185
2-ethyl-3-isopropylphenyl
hydroxymethyl
ethyl



2.5.186
2-cyclopropyl-3-isopropylphenyl 
hydroxymethyl
ethyl



2.5.187
2-vinyl-3-isopropylphenyl
hydroxymethyl
ethyl



2.5.188
2-ethynyl-3-isopropylphenyl
hydroxymethyl
ethyl



2.5.189
2-cyano-3-isopropylphenyl
hydroxymethyl
ethyl



2.5.190
2-trifluoromethyl-3-isopropylphenyl
hydroxymethyl
ethyl



2.5.191
2-methoxy-3-isopropylphenyl
hydroxymethyl
ethyl



2.5.192
2-ethoxy-3-isopropylphenyl
hydroxymethyl
ethyl



2.5.193
2-trifluoromethoxy-3-isopropylphenyl
hydroxymethyl
ethyl



2.5.194
2-nitro-3-isopropylphenyl
hydroxymethyl
ethyl



2.5.195
2-fluoro-3-tert-butylphenyl
hydroxymethyl
ethyl



2.5.196
2-chloro-3-tert-butylphenyl
hydroxymethyl
ethyl



2.5.197
2-bromo-3-tert-butylphenyl
hydroxymethyl
ethyl



2.5.198
2-methyl-3-tert-butylphenyl
hydroxymethyl
ethyl



2.5.199
2-ethyl-3-tert-butylphenyl
hydroxymethyl
ethyl



2.5.200
2-cyclopropyl-3-tert-butylphenyl
hydroxymethyl
ethyl



2.5.201
2-vinyl-3-tert-butylphenyl
hydroxymethyl
ethyl



2.5.202
2-ethynyl-3-tert-butylphenyl
hydroxymethyl
ethyl



2.5.203
2-cyano-3-tert-butylphenyl
hydroxymethyl
ethyl



2.5.204
2-trifluoromethyl-3-tert-butylphenyl
hydroxymethyl
ethyl



2.5.205
2-methoxy-3-tert-butylphenyl
hydroxymethyl
ethyl



2.5.206
2-ethoxy-3-tert-butylphenyl
hydroxymethyl
ethyl



2.5.207
2-trifluoromethoxy-3-tert-butylphenyl
hydroxymethyl
ethyl



2.5.208
2-nitro-3-tert-butylphenyl
hydroxymethyl
ethyl



2.5.209
2-fluoro-3-hydroxymethylphenyl
hydroxymethyl
ethyl



2.5.210
2-chloro-3-hydroxymethylphenyl
hydroxymethyl
ethyl



2.5.211
2-bromo-3-hydroxymethylphenyl
hydroxymethyl
ethyl



2.5.212
2-methyl-3-hydroxymethylphenyl
hydroxymethyl
ethyl



2.5.213
2-ethyl-3-hydroxymethylphenyl
hydroxymethyl
ethyl



2.5.214
2-cyclopropyl-3-hydroxymethylphenyl
hydroxymethyl
ethyl



2.5.215
2-vinyl-3-hydroxymethylphenyl
hydroxymethyl
ethyl



2.5.216
2-ethynyl-3-hydroxymethylphenyl
hydroxymethyl
ethyl



2.5.217
2-cyano-3-hydroxymethylphenyl
hydroxymethyl
ethyl



2.5.218
2-trifluoromethyl-3-
hydroxymethyl
ethyl




hydroxymethylphenyl





2.5.219
2-methoxy-3-hydroxymethylphenyl
hydroxymethyl
ethyl



2.5.220
2-ethoxy-3-hydroxymethylphenyl
hydroxymethyl
ethyl



2.5.221
2-trifluoromethoxy-3-
hydroxymethyl
ethyl




hydroxymethylphenyl





2.5.222
2-nitro-3-hydroxymethylphenyl
hydroxymethyl
ethyl



2.5.223
2-fluoro-3-cyclopropylphenyl 
hydroxymethyl
ethyl



2.5.224
2-chloro-3-cyclopropylphenyl 
hydroxymethyl
ethyl



2.5.225
2-bromo-3-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.226
2-methyl-3-cyclopropylphenyl 
hydroxymethyl
ethyl



2.5.227
2-ethyl-3-cyclopropylphenyl 
hydroxymethyl
ethyl



2.5.228
2-cyclopropyl-3-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.229
2-vinyl-3-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.230
2-ethynyl-3-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.231
2-cyano-3-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.232
2-trifluoromethyl-3-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.233
2-methoxy-3-cyclopropylphenyl 
hydroxymethyl
ethyl



2.5.234
2-ethoxy-3-cyclopropylphenyl 
hydroxymethyl
ethyl



2.5.235
2-trifluoromethoxy-3-
hydroxymethyl
ethyl




cyclopropylphenyl





2.5.236
2-fluoro-3-methoxycarbonylphenyl
hydroxymethyl
ethyl



2.5.237
2-chloro-3-methoxycarbonylphenyl
hydroxymethyl
ethyl



2.5.238
2-bromo-3-methoxycarbonylphenyl
hydroxymethyl
ethyl



2.5.239
2-methyl-3-methoxycarbonylphenyl
hydroxymethyl
ethyl



2.5.240
2-ethyl-3-methoxycarbonylphenyl
hydroxymethyl
ethyl



2.5.241
2-cyclopropyl-3-methoxycarbonyl-
hydroxymethyl
ethyl




phenyl





2.5.242
2-vinyl-3-methoxycarbonylphenyl
hydroxymethyl
ethyl



2.5.243
2-ethynyl-3-methoxycarbonyl-phenyl
hydroxymethyl
ethyl



2.5.244
2-cyano-3-methoxycarbonylphenyl
hydroxymethyl
ethyl



2.5.245
2-trifluoromethyl-3-
hydroxymethyl
ethyl




methoxycarbonylphenyl





2.5.246
2-methoxy-3-methoxycarbonyl-phenyl
hydroxymethyl
ethyl



2.5.247
2-ethoxy-3-methoxycarbonylphenyl
hydroxymethyl
ethyl



2.5.248
2-trifluoromethoxy-3-
hydroxymethyl
ethyl




methoxycarbonylphenyl





2.5.249
2-nitro-3-methoxycarbonylphenyl
hydroxymethyl
ethyl



2.5.250
2-fluoro-3-vinylphenyl
hydroxymethyl
ethyl



2.5.251
2-chloro-3-vinylphenyl
hydroxymethyl
ethyl



2.5.252
2-bromo-3-vinylphenyl
hydroxymethyl
ethyl



2.5.253
2-methyl-3-vinylphenyl
hydroxymethyl
ethyl



2.5.254
2-ethyl-3-vinylphenyl
hydroxymethyl
ethyl



2.5.255
2-cyclopropyl-3-vinylphenyl
hydroxymethyl
ethyl



2.5.256
2-vinyl-3-vinylphenyl
hydroxymethyl
ethyl



2.5.257
2-ethynyl-3-vinylphenyl
hydroxymethyl
ethyl



2.5.258
2-cyano-3-vinylphenyl
hydroxymethyl
ethyl



2.5.259
2-trifluoromethyl-3-vinylphenyl
hydroxymethyl
ethyl



2.5.260
2-methoxy-3-vinylphenyl
hydroxymethyl
ethyl



2.5.261
2-ethoxy-3-vinylphenyl
hydroxymethyl
ethyl



2.5.262
2-trifluoromethoxy-3-vinylphenyl
hydroxymethyl
ethyl



2.5.263
2-nitro-3-vinylphenyl
hydroxymethyl
ethyl



2.5.264
2-fluoro-3-ethynylphenyl
hydroxymethyl
ethyl



2.5.265
2-chloro-3-ethynylphenyl
hydroxymethyl
ethyl



2.5.266
2-bromo-3-ethynylphenyl
hydroxymethyl
ethyl



2.5.267
2-methyl-3-ethynylphenyl
hydroxymethyl
ethyl



2.5.268
2-ethyl-3-ethynylphenyl
hydroxymethyl
ethyl



2.5.269
2-cyclopropyl-3-ethynylphenyl
hydroxymethyl
ethyl



2.5.270
2-vinyl-3-ethynylphenyl
hydroxymethyl
ethyl



2.5.271
2-cyano-3-ethynylphenyl
hydroxymethyl
ethyl



2.5.272
2-trifluoromethyl-3-ethynylphenyl
hydroxymethyl
ethyl



2.5.273
2-methoxy-3-ethynylphenyl
hydroxymethyl
ethyl



2.5.274
2-ethoxy-3-ethynylphenyl
hydroxymethyl
ethyl



2.5.275
2-trifluoromethoxy-3-ethynylphenyl 
hydroxymethyl
ethyl



2.5.276
2-nitro-3-ethynylphenyl
hydroxymethyl
ethyl



2.5.277
2-fluoro-3-ethynylphenyl
hydroxymethyl
ethyl



2.5.278
2-fluoro-3-cyanophenyl
hydroxymethyl
ethyl



2.5.279
2-chloro-3-cyanophenyl
hydroxymethyl
ethyl



2.5.280
2-bromo-3-cyanophenyl
hydroxymethyl
ethyl



2.5.281
2-methyl-3-cyanophenyl
hydroxymethyl
ethyl



2.5.282
2-ethyl-3-cyanophenyl
hydroxymethyl
ethyl



2.5.283
2-ethyl-3-cyanophenyl
1-hydroxyethyl
ethyl



2.5.284
2-ethyl-3-cyanophenyl
1-hydroxypropyl
ethyl



2.5.285
2-ethyl-3-cyanophenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.286
2-ethyl-3-cyanophenyl
methoxymethyl
ethyl



2.5.287
2-ethyl-3-cyanophenyl
2-methoxyethyl
ethyl



2.5.288
2-cyclopropyl-3-cyanophenyl
hydroxymethyl
ethyl



2.5.289
2-vinyl-3-cyanophenyl
hydroxymethyl
ethyl



2.5.290
2-ethynyl-3-cyanophenyl
hydroxymethyl
ethyl



2.5.291
2-cyano-3-cyanophenyl
hydroxymethyl
ethyl



2.5.292
2-trifluoromethyl-3-cyanophenyl
hydroxymethyl
ethyl



2.5.293
2-methoxy-3-cyanophenyl
hydroxymethyl
ethyl



2.5.294
2-ethoxy-3-cyanophenyl
hydroxymethyl
ethyl



2.5.295
2-trifluoromethoxy-3-cyanophenyl
hydroxymethyl
ethyl



2.5.296
2-nitro-3-cyanophenyl
hydroxymethyl
ethyl



2.5.297
2-fluoro-3-hydroxyphenyl
hydroxymethyl
ethyl



2.5.298
2-chloro-3-hydroxyphenyl
hydroxymethyl
ethyl



2.5.299
2-bromo-3-hydroxyphenyl
hydroxymethyl
ethyl



2.5.300
2-methyl-3-hydroxyphenyl
hydroxymethyl
ethyl



2.5.301
2-ethyl-3-hydroxyphenyl
hydroxymethyl
ethyl



2.5.302
2-cyclopropyl-3-hydroxyphenyl
hydroxymethyl
ethyl



2.5.303
2-vinyl-3-hydroxyphenyl
hydroxymethyl
ethyl



2.5.304
2-ethynyl-3-hydroxyphenyl
hydroxymethyl
ethyl



2.5.305
2-cyano-3-hydroxyphenyl
hydroxymethyl
ethyl



2.5.306
2-trifluoromethyl-3-hydroxyphenyl
hydroxymethyl
ethyl



2.5.307
2-methoxy-3-hydroxyphenyl
hydroxymethyl
ethyl



2.5.308
2-ethoxy-3-hydroxyphenyl
hydroxymethyl
ethyl



2.5.309
2-trifluoromethoxy-3-hydroxyphenyl
hydroxymethyl
ethyl



2.5.310
2-nitro-3-hydroxyphenyl
hydroxymethyl
ethyl



2.5.311
2-fluoro-3-methoxyphenyl
hydroxymethyl
ethyl



2.5.312
2-chloro-3-methoxyphenyl
hydroxymethyl
ethyl



2.5.313
2-bromo-3-methoxyphenyl
hydroxymethyl
ethyl



2.5.314
2-methyl-3-methoxyphenyl
hydroxymethyl
ethyl



2.5.315
2-ethyl-3-methoxyphenyl
hydroxymethyl
ethyl



2.5.316
2-cyclopropyl-3-methoxyphenyl
hydroxymethyl
ethyl



2.5.317
2-vinyl-3-methoxyphenyl
hydroxymethyl
ethyl



2.5.318
2-ethynyl-3-methoxyphenyl
hydroxymethyl
ethyl



2.5.319
2-cyano-3-methoxyphenyl
hydroxymethyl
ethyl



2.5.320
2-trifluoromethyl-3-methoxyphenyl
hydroxymethyl
ethyl



2.5.321
2,3-dimethoxyphenyl
hydroxymethyl
ethyl



2.5.322
2-ethoxy-3-methoxyphenyl
hydroxymethyl
ethyl



2.5.323
2-trifluoromethoxy-3-methoxyphenyl
hydroxymethyl
ethyl



2.5.324
2-nitro-3-methoxyphenyl
hydroxymethyl
ethyl



2.5.325
2-fluoro-3-ethoxyphenyl
hydroxymethyl
ethyl



2.5.326
2-chloro-3-ethoxyphenyl
hydroxymethyl
ethyl



2.5.327
2-bromo-3-ethoxyphenyl
hydroxymethyl
ethyl



2.5.328
2-methyl-3-ethoxyphenyl
hydroxymethyl
ethyl



2.5.329
2-ethyl-3-ethoxyphenyl
hydroxymethyl
ethyl



2.5.330
2-cyclopropyl-3-ethoxyphenyl
hydroxymethyl
ethyl



2.5.331
2-vinyl-3-ethoxyphenyl
hydroxymethyl
ethyl



2.5.332
2-ethynyl-3-ethoxyphenyl
hydroxymethyl
ethyl



2.5.333
2-cyano-3-ethoxyphenyl
hydroxymethyl
ethyl



2.5.334
2-trifluoromethyl-3-ethoxyphenyl
hydroxymethyl
ethyl



2.5.335
2-methoxy-3-ethoxyphenyl
hydroxymethyl
ethyl



2.5.336
2,3-diethoxy--phenyl
hydroxymethyl
ethyl



2.5.337
2-trifluoromethoxy-3-ethoxyphenyl
hydroxymethyl
ethyl



2.5.338
2-nitro-3-ethoxyphenyl
hydroxymethyl
ethyl



2.5.339
2-fluoro-3-propoxyphenyl
hydroxymethyl
ethyl



2.5.340
2-chloro-3-propoxyphenyl
hydroxymethyl
ethyl



2.5.341
2-bromo-3-propoxyphenyl
hydroxymethyl
ethyl



2.5.342
2-methyl-3-propoxyphenyl
hydroxymethyl
ethyl



2.5.343
2-ethyl-3-propoxyphenyl
hydroxymethyl
ethyl



2.5.344
2-cyclopropyl-3-propoxyphenyl
hydroxymethyl
ethyl



2.5.345
2-vinyl-3-propoxyphenyl
hydroxymethyl
ethyl



2.5.346
2-ethynyl-3-propoxyphenyl
hydroxymethyl
ethyl



2.5.347
2-cyano-3-propoxyphenyl
hydroxymethyl
ethyl



2.5.348
2-trifluoromethyl-3-propoxyphenyl
hydroxymethyl
ethyl



2.5.349
2-methoxy-3-propoxyphenyl
hydroxymethyl
ethyl



2.5.350
2-ethoxy-3-propoxyphenyl
hydroxymethyl
ethyl



2.5.351
2-trifluoromethoxy-3-propoxyphenyl
hydroxymethyl
ethyl



2.5.352
2-nitro-3-propoxyphenyl
hydroxymethyl
ethyl



2.5.353
2-fluoro-3-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.354
2-chloro-3-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.355
2-bromo-3-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.356
2-methyl-3-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.357
2-ethyl-3-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.358
2-cyclopropyl-3-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.359
2-vinyl-3-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.360
2-ethynyl-3-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.361
2-cyano-3-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.362
2-trifluoromethyl-3-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.363
2-methoxy-3-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.364
2-ethoxy-3-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.365
2-trifluoromethoxy-3-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.366
2-nitro-3-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.367
2-fluoro-3-tert-butoxyphenyl
hydroxymethyl
ethyl



2.5.368
2-chloro-3-tert-butoxyphenyl
hydroxymethyl
ethyl



2.5.369
2-bromo-3-tert-butoxyphenyl
hydroxymethyl
ethyl



2.5.370
2-methyl-3-tert-butoxyphenyl
hydroxymethyl
ethyl



2.5.371
2-ethyl-3-tert-butoxyphenyl
hydroxymethyl
ethyl



2.5.372
2-cyclopropyl-3-tert-butoxyphenyl
hydroxymethyl
ethyl



2.5.373
2-vinyl-3-tert-butoxyphenyl
hydroxymethyl
ethyl



2.5.374
2-ethynyl-3-tert-butoxyphenyl 
hydroxymethyl
ethyl



2.5.375
2-cyano-3-tert-butoxyphenyl
hydroxymethyl
ethyl



2.5.376
2-trifluoromethyl-3-tert-butoxyphenyl
hydroxymethyl
ethyl



2.5.377
2-methoxy-3-tert-butoxyphenyl
hydroxymethyl
ethyl



2.5.378
2-ethoxy-3-tert-butoxyphenyl
hydroxymethyl
ethyl



2.5.379
2-trifluoromethoxy-3-tert-butoxyphenyl
hydroxymethyl
ethyl



2.5.380
2-nitro-3-tert-butoxyphenyl
hydroxymethyl
ethyl



2.5.381
2-fluoro-3-trifluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.382
2-chloro-3-trifluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.383
2-bromo-3-trifluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.384
2-methyl-3-trifluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.385
2-ethyl-3-trifluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.386
2-cyclopropyl-3-trifluoromethoxyphenyl
hydroxymethyl
ethyl



2.5.387
2-vinyl-3-trifluoromethoxyphenyl
hydroxymethyl
ethyl



2.5.388
2-ethynyl-3-trifluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.389
2-cyano-3-trifluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.390
2-trifluoromethyl-3-
hydroxymethyl
ethyl




trifluoromethoxyphenyl





2.5.391
2-methoxy-3-trifluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.392
2-ethoxy-3-trifluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.393
2,3-bis(trifluoromethoxy)phenyl
hydroxymethyl
ethyl



2.5.394
2-nitro-3-trifluoromethoxyphenyl
hydroxymethyl
ethyl



2.5.395
2-fluoro-3-(2,2,2-trifluoroethoxy)-phenyl
hydroxymethyl
ethyl



2.5.396
2-chloro-3-(2,2,2-trifluoroethoxy)phenyl
hydroxymethyl
ethyl



2.5.397
2-bromo-3-(2,2,2-trifluoroethoxy)phenyl
hydroxymethyl
ethyl



2.5.398
2-methyl-3-(2,2,2-trifluoroethoxy)phenyl
hydroxymethyl
ethyl



2.5.399
2-ethyl-3-(2,2,2-trifluoroethoxy)-phenyl
hydroxymethyl
ethyl



2.5.400
2-cyclopropyl-3-(2,2,2-trifluoro-
hydroxymethyl
ethyl




ethoxy)phenyl





2.5.401
2-vinyl-3-(2,2,2-trifluoroethoxy)-phenyl
hydroxymethyl
ethyl



2.5.402
2-ethynyl-3-(2,2,2-trifluoroethoxyphenyl
hydroxymethyl
ethyl



2.5.403
2-cyano-3-(2,2,2-trifluoroethoxy)phenyl
hydroxymethyl
ethyl



2.5.404
2-trifluoromethyl-3-(2,2,2-trifluoro-
hydroxymethyl
ethyl




ethoxy)phenyl





2.5.405
2-methoxy-3-(2,2,2-
hydroxymethyl
ethyl




trifluoroethoxy)phenyl





2.5.406
2-ethoxy-3-(2,2,2-trifluoroethoxy)phenyl
hydroxymethyl
ethyl



2.5.407
2-trifluoromethoxy-3-(2,2,2-trifluoro-
hydroxymethyl
ethyl




ethoxy)phenyl





2.5.408
2-nitro-3-(2,2,2-trifluoroethoxy)-phenyl
hydroxymethyl
ethyl



2.5.409
2-fluoro-3-difluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.410
2-chloro-3-difluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.411
2-bromo-3-difluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.412
2-methyl-3-difluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.413
2-ethyl-3-difluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.414
2-cyclopropyl-3-difluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.415
2-vinyl-3-difluoromethoxyphenyl
hydroxymethyl
ethyl



2.5.416
2-ethynyl-3-difluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.417
2-cyano-3-difluoro-methoxyphenyl
hydroxymethyl
ethyl



2.5.418
2-trifluoromethyl-3-
hydroxymethyl
ethyl




difluoromethoxyphenyl





2.5.419
2-methoxy-3-difluoro-methoxyphenyl
hydroxymethyl
ethyl



2.5.420
2-ethoxy-3-difluoromethoxyphenyl
hydroxymethyl
ethyl



2.5.421
2-trifluoromethoxy-3-
hydroxymethyl
ethyl




difluoromethoxyphenyl





2.5.422
2-nitro-3-difluoromethoxyphenyl
hydroxymethyl
ethyl



2.5.423
2-fluoro-3-(2-methoxyethoxy)-phenyl
hydroxymethyl
ethyl



2.5.424
2-chloro-3-(2-methoxyethoxy)-phenyl
hydroxymethyl
ethyl



2.5.425
2-bromo-3-(2-methoxyethoxy)-phenyl
hydroxymethyl
ethyl



2.5.426
2-methyl-3-(2-methoxyethoxy)-phenyl
hydroxymethyl
ethyl



2.5.427
2-ethyl-3-(2-methoxyethoxy)phenyl
hydroxymethyl
ethyl



2.5.428
2-cyclopropyl-3-(2-
hydroxymethyl
ethyl




methoxyethoxy)phenyl





2.5.429
2-vinyl-3-(2-methoxyethoxy)phenyl
hydroxymethyl
ethyl



2.5.430
2-ethynyl-3-(2-methoxyethoxy)-phenyl
hydroxymethyl
ethyl



2.5.431
2-cyano-3-(2-methoxyethoxy)-phenyl
hydroxymethyl
ethyl



2.5.432
2-trifluoromethyl-3-(2-
hydroxymethyl
ethyl




methoxyethoxy)phenyl





2.5.433
2-methoxy-3-(2-methoxyethoxy)-phenyl
hydroxymethyl
ethyl



2.5.434
2-ethoxy-3-(2-methoxyethoxy)-phenyl
hydroxymethyl
ethyl



2.5.435
2-trifluoromethoxy-(2-
hydroxymethyl
ethyl




methoxyethoxy)phenyl





2.5.436
2-nitro-3-(2-methoxyethoxy)phenyl
hydroxymethyl
ethyl



2.5.437
2-fluoro-3-(tert-
hydroxymethyl
ethyl




butoxycarbonyloxy)phenyl





2.5.438
2-chloro-3-(tert-
hydroxymethyl
ethyl




butoxycarbonyloxy)phenyl





2.5.439
2-bromo-3-(tert-butoxycarbonyl-
hydroxymethyl
ethyl




oxy)phenyl





2.5.440
2-methyl-3-(tert-butoxycarbonyl-
hydroxymethyl
ethyl




oxy)phenyl





2.5.441
2-ethyl-3-(tert-
hydroxymethyl
ethyl




butoxycarbonyloxy)phenyl





2.5.442
2-cyclopropyl-3-(tert-butoxycarbonyl-
hydroxymethyl
ethyl




oxy)phenyl





2.5.443
2-vinyl-3-(tert-
hydroxymethyl
ethyl




butoxycarbonyloxy)phenyl





2.5.444
2-ethynyl-3-(tert-butoxycarbonyl-
hydroxymethyl
ethyl




oxy)phenyl





2.5.445
2-cyano-3-(tert-
hydroxymethyl
ethyl




butoxycarbonyloxy)phenyl





2.5.446
2-trifluoromethyl-3-(tert-
hydroxymethyl
ethyl




butoxycarbonyl-oxy)phenyl





2.5.447
2-methoxy-3-(tert-
hydroxymethyl
ethyl




butoxycarbonyloxy)phenyl





2.5.448
2-ethoxy-3-(tert-
hydroxymethyl
ethyl




butoxycarbonyloxy)phenyl





2.5.449
2-trifluoromethoxy-3-(tert-
hydroxymethyl
ethyl




butoxycarbonyl-oxy)phenyl





2.5.450
2-nitro-3-(tert-
hydroxymethyl
ethyl




butoxycarbonyloxy)phenyl





2.5.451
2-fluoro-3-nitrophenyl
hydroxymethyl
ethyl



2.5.452
2-chloro-3-nitrophenyl
hydroxymethyl
ethyl



2.5.453
2-bromo-3-nitrophenyl
hydroxymethyl
ethyl



2.5.454
2-methyl-3-nitrophenyl
hydroxymethyl
ethyl



2.5.455
2-ethyl-3-nitrophenyl
hydroxymethyl
ethyl



2.5.456
2-cyclopropyl-3-nitrophenyl
hydroxymethyl
ethyl



2.5.457
2-vinyl-3-nitrophenyl
hydroxymethyl
ethyl



2.5.458
2-ethynyl-3-nitrophenyl
hydroxymethyl
ethyl



2.5.459
2-cyano-3-nitrophenyl
hydroxymethyl
ethyl



2.5.460
2-trifluoromethyl-3-nitrophenyl
hydroxymethyl
ethyl



2.5.461
2-methoxy-3-nitrophenyl
hydroxymethyl
ethyl



2.5.462
2-ethoxy-3-nitrophenyl
hydroxymethyl
ethyl



2.5.463
2-trifluoromethoxy-3-nitrophenyl
hydroxymethyl
ethyl



2.5.464
2-fluoro-3-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.465
2-chloro-3-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.466
2-bromo-3-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.467
2-methyl-3-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.468
2-ethyl-3-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.469
2-cyclopropyl-3-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.470
2-vinyl-3-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.471
2-ethynyl-3-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.472
2-cyano-3-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.473
2-trifluoromethyl-3-
hydroxymethyl
ethyl




methylsulfanylphenyl





2.5.474
2-methoxy-3-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.475
2-ethoxy-3-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.476
2-trifluoromethoxy-3-
hydroxymethyl
ethyl




methylsulfanylphenyl





2.5.477
2-nitro-3-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.478
3,5-difluorophenyl
hydroxymethyl
ethyl
[CDCl3] 1.32 (t, 3H);






2.23 (m, 1H); 3.56-3.69






(m, 2H); 3.90 (m, 1H);






4.02 (m, 1H); 4.29






(m, 2H); 6.88 (m, 1H);






7.19 (m, 2H).


2.5.479
3,5-difluorophenyl
1-hydroxyethyl
methyl
[CDCl3] D1 1.06






(t, 3H); 1.30-1.49






(m, 2H); 2.27 (d, 1H);






3.52 (d, 1H); 3.73






(d, 1H); 3.83 (s, 3H);






4.05 (m, 1H); 6.88






(t, 1H); 7.20 (d, 2H).






[CDCl3] D2 1.06






(t, 3H); 1.55 (m, 2H);






1.97 (d, 1H); 3.58






(d, 1H); 3.70 (d, 1H);






3.83 (s, 3H); 3.94






(t, 1H); 6.88 (t, 1H);






7.18 (d, 2H).


2.5.480
3,5-difluorophenyl
1-hydroxypropyl
ethyl



2.5.481
3,5-difluorophenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.482
3,5-difluorophenyl
methoxymethyl
ethyl
[CDCl3] 1.33 (t, 3H);






3.44 (s, 3H); 3.47-3.51






(d, 1H); 3.72-3.83






(m, 3H); 4.29 (m, 2H):






6.88 (m, 1H); 7.20






(m, 2H).


2.5.483
2-ethyl-3-cyanophenyl
2-methoxyethyl
ethyl



2.5.484
3-chloro-5-fluorophenyl
hydroxymethyl
ethyl



2.5.485
3-chloro-5-fluorophenyl
1-hydroxyethyl
methyl
[CDCl3] D1 1.19






(d, 3H); 2.42 (s br, 1H);






3.53 (d, 1H); 3.68






(d, 1H); 3.83 (s, 3H);






4.34 (m, 1H); 7.14






(d, 1H); 7.31 (d, 1H);






7.44 (s, 1H). D2 1.29






(d, 3H); 2.18 (s br, 1H);






3.58 (d, 1H); 3.73






(d, 1H); 3.73 (s, 3H);






4.22 (m, 1H); 7.14






(d, 1H); 7.31 (d, 1H);






7.42 (s, 1H).


2.5.486
3-chloro-5-fluorophenyl
1-hydroxypropyl
ethyl



2.5.487
3-chloro-5-fluorophenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.488
3-chloro-5-fluorophenyl
methoxymethyl
ethyl



2.5.489
3-chloro-5-fluorophenyl
2-methoxyethyl
ethyl



2.5.490
3-bromo-5-fluorophenyl
hydroxymethyl
ethyl



2.5.491
3-bromo-5-fluorophenyl
1-hydroxyethyl
ethyl



2.5.492
3-bromo-5-fluorophenyl
1-hydroxypropyl
ethyl



2.5.493
3-bromo-5-fluorophenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.494
3-bromo-5-fluorophenyl
methoxymethyl
ethyl



2.5.495
3-bromo-5-fluorophenyl
2-methoxyethyl
ethyl



2.5.496
3-iodo-5-fluorophenyl
hydroxymethyl
ethyl



2.5.497
3-methyl-5-fluorophenyl
hydroxymethyl
ethyl



2.5.498
3-methyl-5-fluorophenyl
1-hydroxyethyl
methyl
[CDCl3] D1 1.20






(d, 3H); 2.37 (d, 1H);






2.38 (s, 3H); 3.54






(d, 1H), 3.69 (d, 1H);






3.83 (s, 3H); 4.33






(m, 1H); 6.96 (s, 1H);






7.23 (s, 1H); 7.25






(s, 1H). D2 1.26 (d, 3H);






2.18 (d, 1H); 2.38






(s, 3H); 3.60 (d, 1H);






3.72 (d, 1H); 3.83






(s, 3H); 4.22 (m, 1H);






6.93 (s, 1H); 7.21






(s, 1H); 7.25 (s, 1H)


2.5.499
3-methyl-5-fluorophenyl
1-hydroxypropyl
ethyl



2.5.500
3-methyl-5-fluorophenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.501
3-methyl-5-fluorophenyl
methoxymethyl
ethyl



2.5.502
3-methyl-5-fluorophenyl
2-methoxyethyl
ethyl



2.5.503
3-ethyl-5-fluorophenyl
hydroxymethyl
ethyl



2.5.504
3-propyl-5-fluorophenyl
hydroxymethyl
ethyl



2.5.505
3-i-propyl-5-fluorophenyl
hydroxymethyl
ethyl



2.5.506
3-n-butyl-5-fluorophenyl
hydroxymethyl
ethyl



2.5.507
3-isobutyl-5-fluorophenyl
hydroxymethyl
ethyl



2.5.508
3-tert-butyl-5-fluorophenyl
hydroxymethyl
ethyl



2.5.509
3-cyclopropyl-5-fluorophenyl
hydroxymethyl
ethyl



2.5.510
3-vinyl-5-fluorophenyl
hydroxymethyl
ethyl



2.5.511
3-ethynyl-5-fluorophenyl
hydroxymethyl
ethyl



2.5.512
3-cyano-5-fluorophenyl
hydroxymethyl
ethyl



2.5.513
3-trifluoromethyl-5-fluorophenyl
hydroxymethyl
ethyl



2.5.514
3-trifluoromethyl-5-fluorophenyl
1-hydroxyethyl
ethyl



2.5.515
3-trifluoromethyl-5-fluorophenyl
1-hydroxypropyl
ethyl



2.5.516
3-trifluoromethyl-5-fluorophenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.517
3-trifluoromethyl-5-fluorophenyl
methoxymethyl
ethyl



2.5.518
3-trifluoromethyl-5-fluorophenyl
2-methoxyethyl
ethyl



2.5.519
3-(methoxycarbonyl)-5-fluorophenyl
hydroxymethyl
ethyl



2.5.520
3-hydroxymethyl-5-fluorophenyl
hydroxymethyl
ethyl



2.5.521
3-carbamoyl-5-fluorophenyl
hydroxymethyl
ethyl



2.5.522
3-hydroxy-5-fluorophenyl
hydroxymethyl
ethyl



2.5.523
3-methoxy-5-fluorophenyl
hydroxymethyl
ethyl



2.5.524
3-ethoxy-5-fluorophenyl
hydroxymethyl
ethyl



2.5.525
3-n-propoxy-5-fluorophenyl
hydroxymethyl
ethyl



2.5.526
3-isopropoxy-5-fluorophenyl
hydroxymethyl
ethyl



2.5.527
3-n-butoxy-5-fluorophenyl
hydroxymethyl
ethyl



2.5.528
3-isobutoxy-5-fluorophenyl
hydroxymethyl
ethyl



2.5.529
3-tert-butoxy-5-fluorophenyl
hydroxymethyl
ethyl



2.5.530
3-difluoromethoxy-5-fluorophenyl
hydroxymethyl
ethyl



2.5.531
3-trifluoromethoxy-5-fluorophenyl
hydroxymethyl
ethyl



2.5.532
3-(2,2,2-trifluoroethoxy)-5-fluorophenyl
hydroxymethyl
ethyl



2.5.533
3-(2-chloroethoxy)-5-fluorophenyl
hydroxymethyl
ethyl



2.5.534
3-(2-hydroxyethoxy)-5-fluorophenyl
hydroxymethyl
ethyl



2.5.535
3-[(tert-butoxycarbonyl)oxy]-
hydroxymethyl
ethyl




5-fluorophenyl





2.5.536
3-nitro-5-fluorophenyl
hydroxymethyl
ethyl



2.5.537
3-acetoxy-5-fluorophenyl
hydroxymethyl
ethyl



2.5.538
{3-[(tert-butoxycarbonyl)amino]-
hydroxymethyl
ethyl




5-fluorophenyl}





2.5.539
3-methylsulfanyl-5-fluorophenyl
hydroxymethyl
ethyl



2.5.540
3,5-dichlorophenyl
hydroxymethyl
ethyl
[CDCl3] 1.31 (t, 3H);






2.05 (m, 1H, OH) 3.65






(q, 2H); 3.90 (m, 1H);






4.01 (m, 1H): 4.29 (q,






2H); 7.40 (s, 1H): 7.55






(s, 2H).


2.5.541
3,5-dichlorophenyl
1-hydroxyethyl
methyl
[CDCl3] D1 1.08






(t, 3H); 1.36-1.51






(m, 2H); 2.27 (s, 1H);






3.53 (d, 1H); 3.73






(d, 1H); 3.84 (s, 3H);






4.06 (m, 1H); 7.42






(s, 1H) 7.55 (s, 2H). D2






1.08 (t, 3H); 1.36-1.51






(m, 2H); 1.96 (s, 1H);






3.53 (d, 1H); 3.73






(d, 1H); 3.84 (s, 3H);






3.95 (m, 1H); 7.42






(s, 1H) 7.55 (s, 2H).


2.5.542
3,5-dichlorophenyl
1-hydroxypropyl
ethyl



2.5.543
3,5-dichlorophenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.544
3,5-dichlorophenyl
methoxymethyl
methyl
[CDCl3] 3.43 (s, 3H);






3.50 (d, 1H); 3.72 (d,






1H); 3.80 (mc, 2H);






3.82 (s, 3H); 7.41 (m,






1H); 7.55 (s, 2H).


2.5.545
3,5-dichlorophenyl
2-methoxyethyl
methyl
[CDCl3] 1.55 (s, 3H);






2.30 (m, 2H), 3.22 (s,






3H); 3.42 (d, 1H); 3.55






(m, 2H); 3.75 (d, 1H);






3.82 (s, 3H), 7.40 (s,






1H); 7.55 (s, 2H).


2.5.546
3-bromo-5-chlorophenyl
1-hydroxyethyl
methyl
[CDCl3] D1 1.19






(d, 3H); 2.35 (d br, 1H);






3.53 (d, 1H); 3.73






(d, 1H); 3.83 (s, 3H);






4.30-4.37 (m, 1H);






7.56-7.61 (m, 2H);






7.68-7.72 (m, 1H). D2






1.28 (d, 3H); 2.10 (d






br, 1H); 3.58 (d, 1H);






3.68 (d, 1H); 3.83






(s, 3H);


2.5.547
3-iodo-5-chlorophenyl
hydroxymethyl
ethyl



2.5.548
3-methyl-5-chlorophenyl
hydroxymethyl
ethyl



2.5.549
3-methyl-5-chlorophenyl
1-hydroxyethyl
methyl
[CDCl3] D1 1.20






(d, 3H); 2.33 (d, 1H);






2.36 (s, 3H); 3.54






(d, 1H); 3.69 (d, 1H);






3.83 (s, 3H); 4.33






(m, 1H); 7.23 (s, 1H);






7.38 (s, 1H); 7.46






(s, 1H). D2 1.29 (d, 3H)






2.14 (d, 1H); 2.36






(s, 3H); 3.59 (d, 1H);






3.74 (d, 1H); 3.83






(s, 3H); 4.23 (m, 1H);






7.23 (s, 1H); 7.37






(s, 1H); 7.44 (s, 1H).


2.5.550
3-ethyl-5-chlorophenyl
1-hydroxyethyl
methyl
One unassigned






diastereomer






[CDCl3] 1.24 (t, 3H);






1.28 (d, 3H); 2.14






(d, 1H); 2.65 (q, 2H);






3.64 (AB, 2H); 4.20-






4.28 (m,1H); 7.24






(s, 1H); 7.40 (s, 1H);






7.45 (1H).


2.5.551
3-ethyl-5-chlorophenyl
1-hydroxyethyl
methyl
One unassigned






diastereomer






[CDCl3] 1.20 (d, 3H);






1.25 (t, 3H); 2.33






(d, 1H); 2.65 (q, 2H);






3.55 (d, 1H); 3.74






(d, 1H); 3.83 (s, 3H);






4.30-4.36 (m, 1H); 7.24






(s, 1H); 7.41 (s, 1H);






7.47 (s,1H)


2.5.552
3-ethyl-5-chlorophenyl
1-hydroxyethyl
ethyl
[CDCl3] D1 1.20






(d, 3H); 1.25 (t, 3H);






2.33 (d, 1H); 2.65






(q, 2H); 3.55 (d, 1H);






3.74 (d, 1H); 3.83






(s, 3H); 4.30-4.36






(m, 1H); 7.24 (s, 1H);






7.41 (s, 1H); 7.47






(s, 1H). D2 1.24 (t, 3H);






1.28 (d, 3H); 2.14






(d, 1H); 2.65 (q, 2H);






3.64 (AB, 2H); 4.20-






4.28 (m, 1H); 7.24






(s, 1H); 7.40 s, 1H);






7.45 (1H).


2.5.553
3-n-butyl-5-chlorophenyl
hydroxymethyl
ethyl



2.5.554
3-isobutyl-5-chlorophenyl
hydroxymethyl
ethyl



2.5.555
3-tert-butyl-5-chlorophenyl
hydroxymethyl
ethyl



2.5.556
3-cyclopropyl-5-chlorophenyl
hydroxymethyl
ethyl



2.5.557
3-vinyl-5-chlorophenyl
hydroxymethyl
ethyl



2.5.558
3-ethynyl-5-chlorophenyl
hydroxymethyl
ethyl



2.5.559
3-cyano-5-chlorophenyl
hydroxymethyl
ethyl



2.5.560
3-trifluoromethyl-5-chlorophenyl
hydroxymethyl
ethyl



2.5.561
3-(hydroxycarbonyl)-5-chlorophenyl
hydroxymethyl
ethyl



2.5.562
3-(methoxycarbonyl)-5-chlorophenyl
hydroxymethyl
ethyl



2.5.563
3-hydroxymethyl-5-chlorophenyl
hydroxymethyl
ethyl



2.5.564
3-carbamoyl-5-chlorophenyl
hydroxymethyl
ethyl



2.5.565
3-hydroxy-5-chlorophenyl
hydroxymethyl
ethyl



2.5.566
3-methoxy-5-chlorophenyl
hydroxymethyl
ethyl



2.5.567
3-ethoxy-5-chlorophenyl
hydroxymethyl
ethyl



2.5.568
3-n-propoxy-5-chlorophenyl
hydroxymethyl
ethyl



2.5.569
3-isopropoxy-5-chlorophenyl
hydroxymethyl
ethyl



2.5.570
3-n-butoxy-5-chlorophenyl
hydroxymethyl
ethyl



2.5.571
3-isobutoxy-5-chlorophenyl
hydroxymethyl
ethyl



2.5.572
3-tert-butoxy-5-chlorophenyl
hydroxymethyl
ethyl



2.5.573
3-difluoromethoxy-5-chlorophenyl
hydroxymethyl
ethyl



2.5.574
3-trifluoromethoxy-5-chlorophenyl
hydroxymethyl
ethyl



2.5.575
3-(2,2,2-trifluoroethoxy)-5-chlorophenyl
hydroxymethyl
ethyl



2.5.576
3-(2-chloroethoxy)-5-chlorophenyl
hydroxymethyl
ethyl



2.5.577
3-(2-hydroxyethoxy)-5-chlorophenyl
hydroxymethyl
ethyl



2.5.578
3-[(tert-butoxycarbonyl)oxy]-5-
hydroxymethyl
ethyl




chlorophenyl





2.5.579
3-nitro-5-chlorophenyl
hydroxymethyl
ethyl



2.5.580
3-acetoxy-5-chlorophenyl
hydroxymethyl
ethyl



2.5.581
{3-[(tert-butoxycarbonyl)amino]-5-
hydroxymethyl
ethyl




chlorophenyl}





2.5.582
3-methylsulfanyl-5-chlorophenyl
hydroxymethyl
ethyl



2.5.583
3,5-dibromophenyl
hydroxymethyl
ethyl



2.5.584
3,5-dibromophenyl
1-hydroxyethyl
ethyl



2.5.585
3-iodo-5-bromophenyl
hydroxymethyl
ethyl



2.5.586
3-methyl-5-bromophenyl
hydroxymethyl
ethyl



2.5.587
3-methyl-5-bromophenyl
1-hydroxyethyl
methyl
[CDCl3] D1 1.20 (d, 3H); 1.55 (s br, 1H); 2.36 (s, 3H); 3.53 (d, 1H); 3.68 (d, 1H); 3.83 (s, 3H); 4.32 (m, 1H); 7.38 (s, 1H); 7.43 (s, 1H); 7.62 (s, 1H). D2 1.28 (d, 3H); 2.14 (d, 1H); 2.36 (s, 3H); 3.58 (d, 1H); 3.73 (d, 1H); 3.83 (s, 3H); 4.25 (m, 1H); 7.39 (s, 1H); 7.41 (s, 1H); 7.60 (s, 1H).


2.5.588
3-methyl-5-bromophenyl
1-hydroxypropyl
ethyl



2.5.589
3-methyl-5-bromophenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.590
3-methyl-5-bromophenyl
methoxymethyl
ethyl



2.5.591
3-methyl-5-bromophenyl
2-methoxyethyl
ethyl



2.5.592
3-ethyl-5-bromophenyl
hydroxymethyl
ethyl



2.5.593
3-propyl-5-bromophenyl
hydroxymethyl
ethyl



2.5.594
3-isopropyl-5-bromophenyl
hydroxymethyl
ethyl



2.5.595
3-n-butyl-5-bromophenyl
hydroxymethyl
ethyl



2.5.596
3-isobutyl-5-bromophenyl
hydroxymethyl
ethyl



2.5.597
3-tert-butyl-5-bromophenyl
hydroxymethyl
ethyl



2.5.598
3-cyclopropyl-5-bromophenyl
hydroxymethyl
ethyl



2.5.599
3-vinyl-5-bromophenyl
hydroxymethyl
ethyl



2.5.600
3-ethynyl-5-bromophenyl
hydroxymethyl
ethyl



2.5.601
3-cyano-5-bromophenyl
hydroxymethyl
ethyl



2.5.602
3-trifluoromethyl-5-bromophenyl
hydroxymethyl
ethyl



2.5.603
3-(hydroxycarbonyl)-5-bromophenyl
hydroxymethyl
ethyl



2.5.604
3-(methoxycarbonyl)-5-bromophenyl
hydroxymethyl
ethyl



2.5.605
3-hydroxymethyl-5-bromophenyl
hydroxymethyl
ethyl



2.5.606
3-carbamoyl-5-bromophenyl
hydroxymethyl
ethyl



2.5.607
3-hydroxy-5-bromophenyl
hydroxymethyl
ethyl



2.5.608
3-methoxy-5-bromophenyl
hydroxymethyl
ethyl



2.5.609
3-ethoxy-5-bromophenyl
hydroxymethyl
ethyl



2.5.610
3-n-propoxy-5-bromophenyl
hydroxymethyl
ethyl



2.5.611
3-isopropoxy-5-bromophenyl
hydroxymethyl
ethyl



2.5.612
3-n-butoxy-5-bromophenyl
hydroxymethyl
ethyl



2.5.613
3-isobutoxy-5-bromophenyl
hydroxymethyl
ethyl



2.5.614
3-tert-butoxy-5-bromophenyl
hydroxymethyl
ethyl



2.5.615
3-difluoromethoxy-5-bromophenyl
hydroxymethyl
ethyl



2.5.616
3-trifluoromethoxy-5-bromophenyl
hydroxymethyl
ethyl



2.5.617
3-(2,2,2-trifluoroethoxy)-5-bromophenyl
hydroxymethyl
ethyl



2.5.618
3-(2-chloroethoxy)-5-bromophenyl
hydroxymethyl
ethyl



2.5.619
3-(2-hydroxyethoxy)-5-bromophenyl
hydroxymethyl
ethyl



2.5.620
3-[(tert-butoxycarbonyl)oxy]-
hydroxymethyl
ethyl




5-bromophenyl





2.5.621
3-nitro-5-bromophenyl
hydroxymethyl
ethyl



2.5.622
3-acetoxy-5-bromophenyl
hydroxymethyl
ethyl



2.5.623
{3-[(tert-butoxy-carbonyl)amino]-
hydroxymethyl
ethyl




5-bromophenyl}





2.5.624
3-methylsulfanyl-5-bromophenyl
hydroxymethyl
ethyl



2.5.625
3,5-diiodophenyl
hydroxymethyl
ethyl



2.5.626
3-methyl-5-iodophenyl
hydroxymethyl
ethyl



2.5.627
3-ethyl-5-iodophenyl
hydroxymethyl
ethyl



2.5.628
3-propyl-5-iodophenyl
hydroxymethyl
ethyl



2.5.629
3-isopropyl-5-iodophenyl
hydroxymethyl
ethyl



2.5.630
3-n-butyl-5-iodophenyl
hydroxymethyl
ethyl



2.5.631
3-isobutyl-5-iodophenyl
hydroxymethyl
ethyl



2.5.632
3-tert-butyl-5-iodophenyl
hydroxymethyl
ethyl



2.5.633
3-cyclopropyl-5-iodophenyl
hydroxymethyl
ethyl



2.5.634
3-vinyl-5-iodophenyl
hydroxymethyl
ethyl



2.5.635
3-ethynyl-5-iodophenyl
hydroxymethyl
ethyl



2.5.636
3-cyano-5-iodophenyl
hydroxymethyl
ethyl



2.5.637
3-trifluoromethyl-5-iodophenyl
hydroxymethyl
ethyl



2.5.638
3-(hydroxycarbonyl)-5-iodophenyl
hydroxymethyl
ethyl



2.5.639
3-(methoxycarbonyl)-5-iodophenyl
hydroxymethyl
ethyl



2.5.640
3-hydroxymethyl-5-iodophenyl
hydroxymethyl
ethyl



2.5.641
3-carbamoyl-5-iodophenyl
hydroxymethyl
ethyl



2.5.642
3-hydroxy-5-iodophenyl
hydroxymethyl
ethyl



2.5.643
3-methoxy-5-iodophenyl
hydroxymethyl
ethyl



2.5.644
3-ethoxy-5-iodophenyl
hydroxymethyl
ethyl



2.5.645
3-n-propoxy-5-iodophenyl
hydroxymethyl
ethyl



2.5.646
3-isopropoxy-5-iodophenyl
hydroxymethyl
ethyl



2.5.647
3-n-butoxy-5-iodophenyl
hydroxymethyl
ethyl



2.5.648
3-isobutoxy-5-iodophenyl
hydroxymethyl
ethyl



2.5.649
3-tert-butoxy-5-iodophenyl
hydroxymethyl
ethyl



2.5.650
3-difluoromethoxy-5-iodophenyl
hydroxymethyl
ethyl



2.5.651
3-trifluoromethoxy-5-iodophenyl
hydroxymethyl
ethyl



2.5.652
3-(2,2,2-trifluoroethoxy)-5-iodophenyl
hydroxymethyl
ethyl



2.5.653
3-(2-chloroethoxy)-5-iodophenyl
hydroxymethyl
ethyl



2.5.654
3-(2-hydroxyethoxy)-5-iodophenyl
hydroxymethyl
ethyl



2.5.655
3-[(tert-butoxycarbonyl)oxy]-
hydroxymethyl
ethyl




5-iodophenyl





2.5.656
3-nitro-5-iodophenyl
hydroxymethyl
ethyl



2.5.657
3-acetoxy-5-iodophenyl
hydroxymethyl
ethyl



2.5.658
{3-[(tert-butoxycarbonyl)amino]-
hydroxymethyl
ethyl




5-iodophenyl}





2.5.659
3-methylsulfanyl-5-iodophenyl
hydroxymethyl
ethyl



2.5.660
3,5-dimethylphenyl
hydroxymethyl
ethyl



2.5.661
3,5-dimethylphenyl
1-hydroxyethyl
methyl
[CDCl3] D1 1.29






(d, 3H), 2.19 (d, 1H);






2.35 (s, 6H); 3.56






(d, 1H); 3.75 (d, 1H);






3.82 (s, 3H); 4.31






(m, 1H); 7.07 (s, 1H);






7.29 (s, 2H). D2 1.20






(d, 3H); 1.40 (d, 1H);






2.35 (s, 6H); 3.62






(d, 1H); 3.78 (d, 1H);






3.83 (s, 3H); 4.22






(m, 1H); 7.07 (s, 1H);






7.29 (s, 2H).


2.5.662
3-ethyl-5-methylphenyl
hydroxymethyl
ethyl



2.5.663
3-propyl-5-methylphenyl
hydroxymethyl
ethyl



2.5.664
3-isopropyl-5-methylphenyl
hydroxymethyl
ethyl



2.5.665
3-n-butyl-5-methylphenyl
hydroxymethyl
ethyl



2.5.666
3-isobutyl-5-methylphenyl
hydroxymethyl
ethyl



2.5.667
3-tert-butyl-5-methylphenyl
hydroxymethyl
ethyl



2.5.668
3-cyclopropyl-5-methylphenyl
hydroxymethyl
ethyl



2.5.669
3-cyano-5-methylphenyl
hydroxymethyl
ethyl



2.5.670
3-trifluoromethyl-5-methylphenyl
hydroxymethyl
ethyl



2.5.671
3-(methoxycarbonyl)-5-methylphenyl
hydroxymethyl
ethyl



2.5.672
3-methoxy-5-methylphenyl
hydroxymethyl
ethyl



2.5.673
3-ethoxy-5-methylphenyl
hydroxymethyl
ethyl



2.5.674
3-n-propoxy-5-methylphenyl
hydroxymethyl
ethyl



2.5.675
3-isobutoxy-5-methylphenyl
hydroxymethyl
ethyl



2.5.676
3-difluoromethoxy-5-methylphenyl
hydroxymethyl
ethyl



2.5.677
3-trifluoromethoxy-5-methylphenyl
hydroxymethyl
ethyl



2.5.678
3-nitro-5-methylphenyl
hydroxymethyl
ethyl



2.5.679
3-acetoxy-5-methylphenyl
hydroxymethyl
ethyl



2.5.680
3-methylsulfanyl-5-methylphenyl
hydroxymethyl
ethyl



2.5.681
3,5-diethylphenyl
hydroxymethyl
ethyl



2.5.682
3-propyl-5-ethylphenyl
hydroxymethyl
ethyl



2.5.683
3-isopropyl-5-ethylphenyl
hydroxymethyl
ethyl



2.5.684
3-n-butyl-5-ethylphenyl
hydroxymethyl
ethyl



2.5.685
3-isobutyl-5-ethylphenyl
hydroxymethyl
ethyl



2.5.686
3-tert-butyl-5-ethylphenyl
hydroxymethyl
ethyl



2.5.687
3-cyclopropyl-5-ethylphenyl
hydroxymethyl
ethyl



2.5.688
3-cyano-5-ethylphenyl
hydroxymethyl
ethyl



2.5.689
3-trifluoromethyl-5-ethylphenyl
hydroxymethyl
ethyl



2.5.690
3-(methoxycarbonyl)-5-ethylphenyl
hydroxymethyl
ethyl



2.5.691
3-methoxy-5-ethylphenyl
hydroxymethyl
ethyl



2.5.692
3-ethoxy-5-ethylphenyl
hydroxymethyl
ethyl



2.5.693
3-n-propoxy-5-ethylphenyl
hydroxymethyl
ethyl



2.5.694
3-isobutoxy-5-ethylphenyl
hydroxymethyl
ethyl



2.5.695
3-difluoromethoxy-5-ethylphenyl 
hydroxymethyl
ethyl



2.5.696
3-trifluoromethoxy-5-ethylphenyl
hydroxymethyl
ethyl



2.5.697
3-nitro-5-ethylphenyl
hydroxymethyl
ethyl



2.5.698
3-acetoxy-5-ethylphenyl
hydroxymethyl
ethyl



2.5.699
3-methylsulfanyl-5-ethylphenyl
hydroxymethyl
ethyl



2.5.700
3,5-dipropylphenyl
hydroxymethyl
ethyl



2.5.701
3-isopropyl-5-propylphenyl
hydroxymethyl
ethyl



2.5.702
3-n-butyl-5-propylphenyl
hydroxymethyl
ethyl



2.5.703
3-isobutyl-5-propylphenyl
hydroxymethyl
ethyl



2.5.704
3-tert-butyl-5-propylphenyl
hydroxymethyl
ethyl



2.5.705
3-cyclopropyl-5-propylphenyl
hydroxymethyl
ethyl



2.5.706
3-cyano-5-propylphenyl
hydroxymethyl
ethyl



2.5.707
3-trifluoromethyl-5-propylphenyl
hydroxymethyl
ethyl



2.5.708
3-(methoxycarbonyl)-5-propylphenyl
hydroxymethyl
ethyl



2.5.709
3-methoxy-5-propylphenyl
hydroxymethyl
ethyl



2.5.710
3-ethoxy-5-propylphenyl
hydroxymethyl
ethyl



2.5.711
3-n-propoxy-5-propylphenyl
hydroxymethyl
ethyl



2.5.712
3-isobutoxy-5-propylphenyl
hydroxymethyl
ethyl



2.5.713
3-difluoromethoxy-5-propylphenyl
hydroxymethyl
ethyl



2.5.714
3-trifluoromethoxy-5-ethylphenyl
hydroxymethyl
ethyl



2.5.715
3-nitro-5-propylphenyl
hydroxymethyl
ethyl



2.5.716
3-acetoxy-5-propylphenyl
hydroxymethyl
ethyl



2.5.717
3-methylsulfanyl-5-propylphenyl 
hydroxymethyl
ethyl



2.5.718
3,5-diisopropylphenyl
hydroxymethyl
ethyl



2.5.719
3-n-butyl-5-isopropylphenyl
hydroxymethyl
ethyl



2.5.720
3-isobutyl-5-isopropylphenyl
hydroxymethyl
ethyl



2.5.721
3-tert-butyl-5-isopropylphenyl
hydroxymethyl
ethyl



2.5.722
3-cyclopropyl-5-isopropylphenyl 
hydroxymethyl
ethyl



2.5.723
3-cyano-5-isopropylphenyl
hydroxymethyl
ethyl



2.5.724
3-trifluoromethyl-5-isopropylphenyl 
hydroxymethyl
ethyl



2.5.725
3-(methoxycarbonyl)-5-isopropylphenyl
hydroxymethyl
ethyl



2.5.726
3-methoxy-5-isopropylphenyl
hydroxymethyl
ethyl



2.5.727
3-ethoxy-5-isopropylphenyl
hydroxymethyl
ethyl



2.5.728
3-n-propoxy-5-isopropylphenyl
hydroxymethyl
ethyl



2.5.729
3-isobutoxy-5-isopropylphenyl
hydroxymethyl
ethyl



2.5.730
3-difluoromethoxy-5-isopropylphenyl
hydroxymethyl
ethyl



2.5.731
3-trifluoromethoxy-5-isopropylphenyl
hydroxymethyl
ethyl



2.5.732
3-nitro-5-isopropylphenyl
hydroxymethyl
ethyl



2.5.733
3-acetoxy-5-isopropylphenyl
hydroxymethyl
ethyl



2.5.734
3-methylsulfanyl-5-isopropylphenyl
hydroxymethyl
ethyl



2.5.735
3,5-dibutylphenyl
hydroxymethyl
ethyl



2.5.736
3-isobutyl-5-butylphenyl
hydroxymethyl
ethyl



2.5.737
3-tert-butyl-5-butylphenyl
hydroxymethyl
ethyl



2.5.738
3-cyclopropyl-5-butylphenyl
hydroxymethyl
ethyl



2.5.739
3-cyano-5-butylphenyl
hydroxymethyl
ethyl



2.5.740
3-trifluoromethyl-5-butylphenyl
hydroxymethyl
ethyl



2.5.741
3-(methoxycarbonyl)-5-butylphenyl
hydroxymethyl
ethyl



2.5.742
3-methoxy-5-butylphenyl
hydroxymethyl
ethyl



2.5.743
3-ethoxy-5-butylphenyl
hydroxymethyl
ethyl



2.5.744
3-n-propoxy-5-butylphenyl
hydroxymethyl
ethyl



2.5.745
3-isobutoxy-5-butylphenyl
hydroxymethyl
ethyl



2.5.746
3-difluoromethoxy-5-butylphenyl 
hydroxymethyl
ethyl



2.5.747
3-trifluoromethoxy-5-butylphenyl
hydroxymethyl
ethyl



2.5.748
3-nitro-5-butylphenyl
hydroxymethyl
ethyl



2.5.749
3-acetoxy-5-butylphenyl
hydroxymethyl
ethyl



2.5.750
3-methylsulfanyl-5-butylphenyl 
hydroxymethyl
ethyl



2.5.751
3,5-diisobutylphenyl
hydroxymethyl
ethyl



2.5.752
3-tert-butyl-5-isobutylphenyl 
hydroxymethyl
ethyl



2.5.753
3-cyclopropyl-5-isobutylphenyl 
hydroxymethyl
ethyl



2.5.754
3-cyano-5-isobutylphenyl
hydroxymethyl
ethyl



2.5.755
3-trifluoromethyl-5-isobutylphenyl
hydroxymethyl
ethyl



2.5.756
3-(methoxycarbonyl)-5-isobutylphenyl
hydroxymethyl
ethyl



2.5.757
3-methoxy-5-isobutylphenyl
hydroxymethyl
ethyl



2.5.758
3-ethoxy-5-isobutylphenyl
hydroxymethyl
ethyl



2.5.759
3-n-propoxy-5-isobutylphenyl
hydroxymethyl
ethyl



2.5.760
3-isobutoxy-5-isobutylphenyl
hydroxymethyl
ethyl



2.5.761
3-difluoromethoxy-5-isobutylphenyl
hydroxymethyl
ethyl



2.5.762
3-trifluoromethoxy-5-isobutylphenyl
hydroxymethyl
ethyl



2.5.763
3-nitro-5-isobutylphenyl
hydroxymethyl
ethyl



2.5.764
3-acetoxy-5-isobutylphenyl
hydroxymethyl
ethyl



2.5.765
3-methylsulfanyl-5-isobutylphenyl
hydroxymethyl
ethyl



2.5.766
3,5-(di-tert-butyl)phenyl
hydroxymethyl
ethyl



2.5.767
3-cyclopropyl-5-tert-butylphenyl
hydroxymethyl
ethyl



2.5.768
3-cyano-5-tert-butylphenyl
hydroxymethyl
ethyl



2.5.769
3-trifluoromethyl-5-tert-butylphenyl
hydroxymethyl
ethyl



2.5.770
3-(methoxycarbonyl)-5-tert-butylphenyl
hydroxymethyl
ethyl



2.5.771
3-methoxy-5-tert-butylphenyl
hydroxymethyl
ethyl



2.5.772
3-ethoxy-5-tert-butylphenyl
hydroxymethyl
ethyl



2.5.773
3-n-propoxy-5-tert-butylphenyl
hydroxymethyl
ethyl



2.5.774
3-isobutoxy-5-tert-butylphenyl 
hydroxymethyl
ethyl



2.5.775
3-difluoromethoxy-5-tert-butylphenyl
hydroxymethyl
ethyl



2.5.776
3-trifluoromethoxy-5-tert-butylphenyl
hydroxymethyl
ethyl



2.5.777
3-nitro-5-tert-butylphenyl
hydroxymethyl
ethyl



2.5.778
3-acetoxy-5-tert-butylphenyl
hydroxymethyl
ethyl



2.5.779
3-methylsulfanyl-5-tert-butylphenyl
hydroxymethyl
ethyl



2.5.780
3-tert-butyl-5-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.781
3,5-dicyclopropyl-phenyl
hydroxymethyl
ethyl



2.5.782
3-cyano-5-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.783
3-trifluoromethyl-5-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.784
3-(methoxycarbonyl)-5-
hydroxymethyl
ethyl




cyclopropylphenyl





2.5.785
3-methoxy-5-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.786
3-ethoxy-5-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.787
3-n-propoxy-5-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.788
3-isobutoxy-5-cyclopropylphenyl 
hydroxymethyl
ethyl



2.5.789
3-difluoromethoxy-5-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.790
3-trifluoromethoxy-5-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.791
3-nitro-5-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.792
3-acetoxy-5-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.793
3-methylsulfanyl-5-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.794
3,5-dicyanophenyl
hydroxymethyl
ethyl



2.5.795
3-trifluoromethyl-5-cyanophenyl
hydroxymethyl
ethyl



2.5.796
3-(methoxycarbonyl)-5-cyanophenyl
hydroxymethyl
ethyl



2.5.797
3-methoxy-5-cyanophenyl
hydroxymethyl
ethyl



2.5.798
3-ethoxy-5-cyanophenyl
hydroxymethyl
ethyl



2.5.799
3-n-propoxy-5-cyanophenyl
hydroxymethyl
ethyl



2.5.800
3-isobutoxy-5-cyanophenyl
hydroxymethyl
ethyl



2.5.801
3-difluoromethoxy-5-cyanophenyl
hydroxymethyl
ethyl



2.5.802
3-trifluoromethoxy-5-cyanophenyl
hydroxymethyl
ethyl



2.5.803
3-nitro-5-cyanophenyl
hydroxymethyl
ethyl



2.5.804
3-acetoxy-5-cyanophenyl
hydroxymethyl
ethyl



2.5.805
3-methylsulfanyl-5-cyanophenyl
hydroxymethyl
ethyl



2.5.806
3,5-di(trifluoromethyl)phenyl 
hydroxymethyl
ethyl



2.5.807
3-(methoxycarbonyl)-5-
hydroxymethyl
ethyl




trifluoromethylphenyl





2.5.808
3-methoxy-5-trifluoromethylphenyl
hydroxymethyl
ethyl



2.5.809
3-ethoxy-5-trifluoromethylphenyl
hydroxymethyl
ethyl



2.5.810
3-n-propoxy-5-trifluoromethylphenyl
hydroxymethyl
ethyl



2.5.811
3-isobutoxy-5-trifluoromethylphenyl
hydroxymethyl
ethyl



2.5.812
3-difluoromethoxy-5-
hydroxymethyl
ethyl




trifluoromethylphenyl





2.5.813
3-trifluoromethoxy-5-
hydroxymethyl
ethyl




trifluoromethylphenyl





2.5.814
3-nitro-5-trifluoromethylphenyl
hydroxymethyl
ethyl



2.5.815
3-acetoxy-5-trifluoromethylphenyl
hydroxymethyl
ethyl



2.5.816
3-methylsulfanyl-5-
hydroxymethyl
ethyl




trifluoromethylphenyl





2.5.817
3,5-di(methoxycarbonyl)phenyl
hydroxymethyl
ethyl



2.5.818
3-methoxy-5-(methoxycarbonyl)-phenyl
hydroxymethyl
ethyl



2.5.819
3-ethoxy-5-(methoxycarbonyl)-phenyl
hydroxymethyl
ethyl



2.5.820
3-n-propoxy-5-(methoxycarbonyl)-
hydroxymethyl
ethyl




phenyl





2.5.821
3-isobutoxy-5-(methoxycarbonyl)-
hydroxymethyl
ethyl




phenyl





2.5.822
3-difluoromethoxy-5-
hydroxymethyl
ethyl




(methoxycarbonyl)-phenyl





2.5.823
3-trifluoromethoxy-5-
hydroxymethyl
ethyl




(methoxycarbonyl)-phenyl





2.5.824
3-nitro-5-(methoxy-carbonyl)phenyl
hydroxymethyl
ethyl



2.5.825
3-acetoxy-5-(methoxycarbonyl)-phenyl
hydroxymethyl
ethyl



2.5.826
3-methylsulfanyl-5-
hydroxymethyl
ethyl




(methoxycarbonyl)-phenyl





2.5.827
3,5-dimethoxyphenyl
hydroxymethyl
ethyl



2.5.828
3-ethoxy-5-methoxyphenyl
hydroxymethyl
ethyl



2.5.829
3-n-propoxy-5-methoxyphenyl
hydroxymethyl
ethyl



2.5.830
3-isobutoxy-5-methoxyphenyl
hydroxymethyl
ethyl



2.5.831
3-difluoromethoxy-5-methoxyphenyl
hydroxymethyl
ethyl



2.5.832
3-trifluoromethoxy-5-methoxyphenyl
hydroxymethyl
ethyl



2.5.833
3-nitro-5-methoxyphenyl
hydroxymethyl
ethyl



2.5.834
3-acetoxy-5-methoxyphenyl
hydroxymethyl
ethyl



2.5.835
3-methylsulfanyl-5-methoxyphenyl
hydroxymethyl
ethyl



2.5.836
3,5-diethoxyphenyl
hydroxymethyl
ethyl



2.5.837
3-n-propoxy-5-ethoxyphenyl
hydroxymethyl
ethyl



2.5.838
3-isobutoxy-5-ethoxyphenyl
hydroxymethyl
ethyl



2.5.839
3-difluoromethoxy-5-ethoxyphenyl
hydroxymethyl
ethyl



2.5.840
3-trifluoromethoxy-5-ethoxyphenyl
hydroxymethyl
ethyl



2.5.841
3-nitro-5-ethoxyphenyl
hydroxymethyl
ethyl



2.5.842
3-acetoxy-5-ethoxyphenyl
hydroxymethyl
ethyl



2.5.843
3-methylsulfanyl-5-ethoxyphenyl
hydroxymethyl
ethyl



2.5.844
3,5-di(isopropoxy)phenyl
hydroxymethyl
ethyl



2.5.845
3-isobutoxy-5-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.846
3-difluoromethoxy-5-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.847
3-trifluoromethoxy-5-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.848
3-nitro-5-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.849
3-acetoxy-5-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.850
3-methylsulfanyl-5-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.851
3,5-di(trifluoro-methoxy)phenyl 
hydroxymethyl
ethyl



2.5.852
3-nitro-5-trifluoro-methoxyphenyl
hydroxymethyl
ethyl



2.5.853
3-methylsulfanyl-5-
hydroxymethyl
ethyl




trifluoromethoxyphenyl





2.5.854
3,5-bis(difluoromethoxy)phenyl
hydroxymethyl
ethyl



2.5.855
3,5-bis(difluoromethoxy)phenyl
1-hydroxyethyl
ethyl



2.5.856
3,5-bis(difluoromethoxy)phenyl 
1-hydroxypropyl
ethyl



2.5.857
3,5-bis(difluoromethoxy)phenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.858
3-trifluoromethoxy-5-
hydroxymethyl
ethyl




difluoromethoxyphenyl





2.5.859
3-nitro-5-difluoromethoxyphenyl
hydroxymethyl
ethyl



2.5.860
3-acetoxy-5-difluoromethoxy-phenyl 
hydroxymethyl
ethyl



2.5.861
3-methylsulfanyl-5-
hydroxymethyl
ethyl




difluoromethoxyphenyl





2.5.862
3,5-bis(acetoxy)phenyl
hydroxymethyl
ethyl



2.5.863
3-methylsulfanyl-5-acetoxyphenyl
hydroxymethyl
ethyl



2.5.864
3-acetoxy-5-nitrophenyl
hydroxymethyl
ethyl



2.5.865
3-methylsulfanyl-5-nitrophenyl
hydroxymethyl
ethyl



2.5.866
3,4-difluorophenyl
hydroxymethyl
ethyl



2.5.867
3,4-difluorophenyl
1-hydroxyethyl
ethyl



2.5.868
3,4-difluorophenyl
1-hydroxypropyl
ethyl



2.5.869
3,4-difluorophenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.870
3,4-difluorophenyl
methoxymethyl
ethyl



2.5.871
3,4-difluorophenyl
2-methoxyethyl
ethyl



2.5.872
3-chloro-4-fluorophenyl
hydroxymethyl
ethyl



2.5.873
3-chloro-4-fluorophenyl
1-hydroxyethyl
ethyl



2.5.874
3-chloro-4-fluorophenyl
1-hydroxypropyl
ethyl



2.5.875
3-chloro-4-fluorophenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.876
3-chloro-4-fluorophenyl
methoxymethyl
ethyl



2.5.877
3-chloro-4-fluorophenyl
2-methoxyethyl
ethyl



2.5.878
3-bromo-4-fluorophenyl
hydroxymethyl
ethyl



2.5.879
3-methyl-4-fluorophenyl
hydroxymethyl
ethyl



2.5.880
3-methyl-4-fluorophenyl
1-hydroxyethyl
ethyl



2.5.881
3-cyclopropyl-4-fluorophenyl
hydroxymethyl
ethyl



2.5.882
3-cyano-4-fluorophenyl
hydroxymethyl
ethyl



2.5.883
3-methoxy-4-fluorophenyl
hydroxymethyl
ethyl



2.5.884
3-ethoxy-4-fluorophenyl
hydroxymethyl
ethyl



2.5.885
3-trifluoromethoxy-4-fluorophenyl
hydroxymethyl
ethyl



2.5.886
3-nitro-4-fluorophenyl
hydroxymethyl
ethyl



2.5.887
3-fluoro-4-chlorophenyl
hydroxymethyl
ethyl



2.5.888
3,4-dichlorophenyl
hydroxymethyl
ethyl



2.5.889
3-bromo-4-chlorophenyl
hydroxymethyl
ethyl



2.5.890
3-methyl-4-chlorophenyl
hydroxymethyl
ethyl



2.5.891
3-cyclopropyl-4-chlorophenyl
hydroxymethyl
ethyl



2.5.892
3-cyano-4-chlorophenyl
hydroxymethyl
ethyl



2.5.893
3-trifluoromethyl-4-chlorophenyl
hydroxymethyl
ethyl



2.5.894
3-methoxy-4-chlorophenyl
hydroxymethyl
ethyl



2.5.895
3-ethoxy-4-chlorophenyl
hydroxymethyl
ethyl



2.5.896
3-trifluoromethoxy-4-chlorophenyl
hydroxymethyl
ethyl



2.5.897
3-nitro-4-chlorophenyl
hydroxymethyl
ethyl



2.5.898
3-fluoro-4-bromophenyl
hydroxymethyl
ethyl



2.5.899
3-chloro-4-bromophenyl
hydroxymethyl
ethyl



2.5.900
3,4-dibromophenyl
hydroxymethyl
ethyl



2.5.901
3-methyl-4-bromophenyl
hydroxymethyl
ethyl



2.5.902
3-cyclopropyl-4-bromophenyl
hydroxymethyl
ethyl



2.5.903
3-cyano-4-bromophenyl
hydroxymethyl
ethyl



2.5.904
3-trifluoromethyl-4-bromophenyl
hydroxymethyl
ethyl



2.5.905
3-methoxy-4-phenyl
hydroxymethyl
ethyl



2.5.906
3-ethoxy-4-bromophenyl
hydroxymethyl
ethyl



2.5.907
3-trifluoromethoxy-4-bromophenyl
hydroxymethyl
ethyl



2.5.908
3-nitro-4-bromophenyl
hydroxymethyl
ethyl



2.5.909
3-fluoro-4-iodophenyl
hydroxymethyl
ethyl



2.5.910
3-chloro-4-iodophenyl
hydroxymethyl
ethyl



2.5.911
3-bromo-4-iodophenyl
hydroxymethyl
ethyl



2.5.912
3-methyl-4-iodophenyl
hydroxymethyl
ethyl



2.5.913
3-cyclopropyl-4-iodophenyl
hydroxymethyl
ethyl



2.5.914
3-cyano-4-iodophenyl
hydroxymethyl
ethyl



2.5.915
3-trifluoromethyl-4-iodophenyl
hydroxymethyl
ethyl



2.5.916
3-methoxy-4-iodophenyl
hydroxymethyl
ethyl



2.5.917
3-ethoxy-4-iodophenyl
hydroxymethyl
ethyl



2.5.918
3-trifluoromethoxy-4-iodophenyl
hydroxymethyl
ethyl



2.5.919
3-nitro-4-iodophenyl
hydroxymethyl
ethyl



2.5.920
3-fluoro-4-methylphenyl
hydroxymethyl
ethyl



2.5.921
3-chloro-4-methylphenyl
hydroxymethyl
ethyl



2.5.922
3-bromo-4-methylphenyl
hydroxymethyl
ethyl



2.5.923
3,4-dimethylphenyl
hydroxymethyl
ethyl



2.5.924
3,4-dimethylphenyl
1-hydroxyethyl
ethyl



2.5.925
3,4-dimethylphenyl
1-hydroxypropyl
ethyl



2.5.926
3,4-dimethylphenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.927
3,4-dimethylphenyl
methoxymethyl
ethyl



2.5.928
3,4-dimethylphenyl
2-methoxyethyl
ethyl



2.5.929
3-cyclopropyl-4-methylphenyl
hydroxymethyl
ethyl



2.5.930
3-cyano-4-methylphenyl
hydroxymethyl
ethyl



2.5.931
3-trifluoromethyl-4-methylphenyl
hydroxymethyl
ethyl



2.5.932
3-methoxy-4-methylphenyl
hydroxymethyl
ethyl



2.5.933
3-ethoxy-4-methylphenyl
hydroxymethyl
ethyl



2.5.934
3-trifluoromethoxy-4-methylphenyl
hydroxymethyl
ethyl



2.5.935
3-nitro-4-methylphenyl
hydroxymethyl
ethyl



2.5.936
3-fluoro-4-ethylphenyl
hydroxymethyl
ethyl



2.5.937
3-chloro-4-ethylphenyl
hydroxymethyl
ethyl



2.5.938
3-bromo-4-ethylphenyl
hydroxymethyl
ethyl



2.5.939
3-methyl-4-ethylphenyl
hydroxymethyl
ethyl



2.5.940
3,4-diethylphenyl
hydroxymethyl
ethyl



2.5.941
3-cyclopropyl-4-ethylphenyl
hydroxymethyl
ethyl



2.5.942
3-cyano-4-ethylphenyl
hydroxymethyl
ethyl



2.5.943
3-trifluoromethyl-4-ethylphenyl 
hydroxymethyl
ethyl



2.5.944
3-methoxy-4-ethylphenyl
hydroxymethyl
ethyl



2.5.945
3-ethoxy-4-ethylphenyl
hydroxymethyl
ethyl



2.5.946
3-trifluoromethoxy-4-ethylphenyl
hydroxymethyl
ethyl



2.5.947
3-nitro-4-ethylphenyl
hydroxymethyl
ethyl



2.5.948
3-fluoro-4-propylphenyl
hydroxymethyl
ethyl



2.5.949
3-chloro-4-propylphenyl
hydroxymethyl
ethyl



2.5.950
3-bromo-4-propylphenyl
hydroxymethyl
ethyl



2.5.951
3-methyl-4-propylphenyl
hydroxymethyl
ethyl



2.5.952
3-cyclopropyl-4-propylphenyl
hydroxymethyl
ethyl



2.5.953
3-cyano-4-propylphenyl
hydroxymethyl
ethyl



2.5.954
3-trifluoromethyl-4-propylphenyl
hydroxymethyl
ethyl



2.5.955
3-methoxy-4-propylphenyl
hydroxymethyl
ethyl



2.5.956
3-ethoxy-4-propylphenyl
hydroxymethyl
ethyl



2.5.957
3-trifluoromethoxy-4-propylphenyl
hydroxymethyl
ethyl



2.5.958
3-nitro-4-propylphenyl
hydroxymethyl
ethyl



2.5.959
3-fluoro-4-isopropylphenyl
hydroxymethyl
ethyl



2.5.960
3-chloro-4-isopropylphenyl
hydroxymethyl
ethyl



2.5.961
3-bromo-4-isopropylphenyl
hydroxymethyl
ethyl



2.5.962
3-methyl-4-isopropylphenyl
hydroxymethyl
ethyl



2.5.963
3-cyclopropyl-4-isopropylphenyl 
hydroxymethyl
ethyl



2.5.964
3-cyano-4-isopropylphenyl
hydroxymethyl
ethyl



2.5.965
3-trifluoromethyl-4-isopropylphenyl
hydroxymethyl
ethyl



2.5.966
3-methoxy-4-isopropylphenyl
hydroxymethyl
ethyl



2.5.967
3-ethoxy-4-isopropylphenyl
hydroxymethyl
ethyl



2.5.968
3-trifluoromethoxy-4-isopropylphenyl
hydroxymethyl
ethyl



2.5.969
3-nitro-4-isopropylphenyl
hydroxymethyl
ethyl



2.5.970
3-fluoro-4-tert-butylphenyl
hydroxymethyl
ethyl



2.5.971
3-chloro-4-tert-butylphenyl
hydroxymethyl
ethyl



2.5.972
3-bromo-4-tert-butylphenyl
hydroxymethyl
ethyl



2.5.973
3-methyl-4-tert-butylphenyl
hydroxymethyl
ethyl



2.5.974
3-cyclopropyl-4-tert-butylphenyl
hydroxymethyl
ethyl



2.5.975
3-cyano-4-tert-butylphenyl
hydroxymethyl
ethyl



2.5.976
3-trifluoromethyl-4-tert-butylphenyl
hydroxymethyl
ethyl



2.5.977
3-trifluoromethyl-4-tert-butylphenyl
1-hydroxyethyl
ethyl



2.5.978
3-trifluoromethyl-4-tert-butylphenyl
1-hydroxypropyl
ethyl



2.5.979
3-trifluoromethyl-4-tert-butylphenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.980
3-trifluoromethyl-4-tert-butylphenyl
methoxymethyl
ethyl



2.5.981
3-trifluoromethyl-4-tert-butylphenyl
2-methoxyethyl
ethyl



2.5.982
3-methoxy-4-tert-butylphenyl
hydroxymethyl
ethyl



2.5.983
3-ethoxy-4-tert-butylphenyl
hydroxymethyl
ethyl



2.5.984
3-trifluoromethoxy-4-tert-butylphenyl
hydroxymethyl
ethyl



2.5.985
3-nitro-4-tert-butylphenyl
hydroxymethyl
ethyl



2.5.986
3-fluoro-4-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.987
3-chloro-4-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.988
3-bromo-4-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.989
3-methyl-4-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.990
3-cyano-4-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.991
3-trifluoromethyl-4-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.992
3-methoxy-4-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.993
3-ethoxy-4-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.994
3-trifluoromethoxy-4-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.995
3-fluoro-4-methoxycarbonyl-phenyl
hydroxymethyl
ethyl



2.5.996
3-chloro-4-methoxy-carbonylphenyl
hydroxymethyl
ethyl



2.5.997
3-bromo-4-methoxy-carbonylphenyl
hydroxymethyl
ethyl



2.5.998
3-methyl-4-methoxy-carbonylphenyl
hydroxymethyl
ethyl



2.5.999
3-cyclopropyl-4-methoxycarbonyl-
hydroxymethyl
ethyl




phenyl





2.5.1000
3-cyano-4-methoxycarbonylphenyl
hydroxymethyl
ethyl



2.5.1001
3-trifluoromethyl-4-methoxycarbonyl-
hydroxymethyl
ethyl




phenyl





2.5.1002
3-methoxy-4-methoxycarbonyl-phenyl
hydroxymethyl
ethyl



2.5.1003
3-ethoxy-4-methoxycarbonyl-phenyl
hydroxymethyl
ethyl



2.5.1004
3-trifluoromethoxy-4-
hydroxymethyl
ethyl




methoxycarbonyl-phenyl





2.5.1005
3-nitro-4-methoxy-carbonylphenyl
hydroxymethyl
ethyl



2.5.1006
3-fluoro-4-cyanophenyl
hydroxymethyl
ethyl



2.5.1007
3-chloro-4-cyanophenyl
hydroxymethyl
ethyl



2.5.1008
3-bromo-4-cyanophenyl
hydroxymethyl
ethyl



2.5.1009
3-methyl-4-cyanophenyl
hydroxymethyl
ethyl



2.5.1010
3-cyclopropyl-4-cyanophenyl
hydroxymethyl
ethyl



2.5.1011
3,4-dicyanophenyl
hydroxymethyl
ethyl



2.5.1012
3-trifluoromethyl-4-cyanophenyl
hydroxymethyl
ethyl



2.5.1013
3-trifluoromethyl-4-cyanophenyl
1-hydroxyethyl
ethyl



2.5.1014
3-trifluoromethyl-4-cyanophenyl
1-hydroxypropyl
ethyl



2.5.1015
3-trifluoromethyl-4-cyanophenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.1016
3-trifluoromethyl-4-cyanophenyl
methoxymethyl
ethyl



2.5.1017
3-trifluoromethyl-4-cyanophenyl
2-methoxyethyl
ethyl



2.5.1018
3-methoxy-4-cyanophenyl
hydroxymethyl
ethyl



2.5.1019
3-ethoxy-4-cyanophenyl
hydroxymethyl
ethyl



2.5.1020
3-trifluoromethoxy-4-cyanophenyl
hydroxymethyl
ethyl



2.5.1021
3-nitro-4-cyanophenyl
hydroxymethyl
ethyl



2.5.1022
3-fluoro-4-methoxyphenyl
hydroxymethyl
ethyl



2.5.1023
3-chloro-4-methoxyphenyl
hydroxymethyl
ethyl



2.5.1024
3-bromo-4-methoxyphenyl
hydroxymethyl
ethyl



2.5.1025
3-methyl-4-methoxyphenyl
hydroxymethyl
ethyl



2.5.1026
3-cyclopropyl-4-methoxyphenyl
hydroxymethyl
ethyl



2.5.1027
3-cyano-4-methoxyphenyl
hydroxymethyl
ethyl



2.5.1028
3-trifluoromethyl-4-methoxyphenyl
hydroxymethyl
ethyl



2.5.1029
3,4-dimethoxyphenyl
hydroxymethyl
ethyl



2.5.1030
3-ethoxy-4-methoxyphenyl
hydroxymethyl
ethyl



2.5.1031
3-trifluoromethoxy-4-methoxyphenyl
hydroxymethyl
ethyl



2.5.1032
3-nitro-4-methoxyphenyl
hydroxymethyl
ethyl



2.5.1033
3-fluoro-4-ethoxyphenyl
hydroxymethyl
ethyl



2.5.1034
3-chloro-4-ethoxyphenyl
hydroxymethyl
ethyl



2.5.1035
3-chloro-4-ethoxyphenyl
1-hydroxyethyl
ethyl



2.5.1036
3-chloro-4-ethoxyphenyl
1-hydroxypropyl
ethyl



2.5.1037
3-chloro-4-ethoxyphenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.1038
3-chloro-4-ethoxyphenyl
methoxymethyl
ethyl



2.5.1039
3-chloro-4-ethoxyphenyl
2-methoxyethyl
ethyl



2.5.1040
3-bromo-4-ethoxyphenyl
hydroxymethyl
ethyl



2.5.1041
3-methyl-4-ethoxyphenyl
hydroxymethyl
ethyl



2.5.1042
3-cyclopropyl-4-ethoxyphenyl
hydroxymethyl
ethyl



2.5.1043
3-cyano-4-ethoxyphenyl
hydroxymethyl
ethyl



2.5.1044 
3-trifluoromethyl-4-ethoxyphenyl
hydroxymethyl
ethyl



2.5.1045
3-methoxy-4-ethoxyphenyl
hydroxymethyl
ethyl



2.5.1046
2,4-diethoxyphenyl
hydroxymethyl
ethyl



2.5.1047
3-trifluoromethoxy-4-ethoxyphenyl
hydroxymethyl
ethyl



2.5.1048
3-nitro-4-ethoxyphenyl
hydroxymethyl
ethyl



2.5.1049
3-fluoro-4-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.1050
3-chloro-4-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.1051
3-bromo-4-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.1052
3-methyl-4-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.1053
3-cyclopropyl-4-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.1054
3-cyano-4-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.1055
3-trifluoromethyl-4-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.1056
3-methoxy-4-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.1057
3-ethoxy-4-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.1058
3-trifluoromethoxy-4-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.1059
3-nitro-4-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.1060
3-fluoro-4-trifluoro-methoxyphenyl
hydroxymethyl
ethyl



2.5.1061
3-chloro-4-trifluoro-methoxyphenyl
hydroxymethyl
ethyl



2.5.1062
3-bromo-4-trifluoro-methoxyphenyl
hydroxymethyl
ethyl



2.5.1063
3-methyl-4-trifluoro-methoxyphenyl
hydroxymethyl
ethyl



2.5.1064
3-cyclopropyl-4-trifluoromethoxyphenyl
hydroxymethyl
ethyl



2.5.1065
3-cyano-4-trifluoro-methoxyphenyl
hydroxymethyl
ethyl



2.5.1066
3-trifluoromethyl-4-
hydroxymethyl
ethyl




trifluoromethoxyphenyl





2.5.1067
3-methoxy-4-trifluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1068
3-ethoxy-4-trifluoro-methoxyphenyl
hydroxymethyl
ethyl



2.5.1069
3,4-bis(trifluoromethoxy)phenyl
hydroxymethyl
ethyl



2.5.1070
3-nitro-4-trifluoromethoxyphenyl
hydroxymethyl
ethyl



2.5.1071
3-fluoro-4-difluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1072
3-chloro-4-difluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1073
3-bromo-4-difluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1074
3-methyl-4-difluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1075
3-cyclopropyl-4-difluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1076
3-cyano-4-difluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1077
3-trifluoromethyl-4-
hydroxymethyl
ethyl




difluoromethoxyphenyl





2.5.1078
3-methoxy-4-difluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1079
3-ethoxy-4-difluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1080
3-trifluoromethoxy-4-
hydroxymethyl
ethyl




difluoromethoxyphenyl





2.5.1081
3-nitro-4-difluoromethoxyphenyl
hydroxymethyl
ethyl



2.5.1082
3-fluoro-4-nitrophenyl
hydroxymethyl
ethyl



2.5.1083
3-chloro-4-nitrophenyl
hydroxymethyl
ethyl



2.5.1084
3-bromo-4-nitrophenyl
hydroxymethyl
ethyl



2.5.1085
3-methyl-4-nitrophenyl
hydroxymethyl
ethyl



2.5.1086
3-cyclopropyl-4-nitrophenyl
hydroxymethyl
ethyl



2.5.1087
3-cyano-4-nitrophenyl
hydroxymethyl
ethyl



2.5.1088
3-trifluoromethyl-4-nitrophenyl 
hydroxymethyl
ethyl



2.5.1089
3-methoxy-4-nitrophenyl
hydroxymethyl
ethyl



2.5.1090
3-ethoxy-4-nitrophenyl
hydroxymethyl
ethyl



2.5.1091
3-trifluoromethoxy-4-nitrophenyl
hydroxymethyl
ethyl



2.5.1092
3-fluoro-4-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.1093
3-chloro-4-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.1094
3-bromo-4-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.1095
3-methyl-4-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.1096
3-cyclopropyl-4-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.1097
3-cyano-4-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.1098
3-trifluoromethyl-4-
hydroxymethyl
ethyl




methylsulfanylphenyl





2.5.1099
3-methoxy-4-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.1100
3-ethoxy-4-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.1101
3-trifluoromethoxy-4-
hydroxymethyl
ethyl




methylsulfanylphenyl





2.5.1102
3-nitro-4-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.1103
3,6-difluorophenyl
hydroxymethyl
ethyl



2.5.1104
3,6-difluorophenyl
1-hydroxyethyl
ethyl



2.5.1105
3,6-difluorophenyl
1-hydroxypropyl
ethyl



2.5.1106
3,6-difluorophenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.1107
3,6-difluorophenyl
methoxymethyl
ethyl



2.5.1108
3,6-difluorophenyl
2-methoxyethyl
ethyl



2.5.1109
3-chloro-6-fluorophenyl
hydroxymethyl
ethyl



2.5.1110
3-bromo-6-fluorophenyl
hydroxymethyl
ethyl



2.5.1111
3-methyl-6-fluorophenyl
hydroxymethyl
ethyl



2.5.1112
3-cyclopropyl-6-fluorophenyl
hydroxymethyl
ethyl



2.5.1113
3-cyano-6-fluorophenyl
hydroxymethyl
ethyl



2.5.1114
3-methoxy-6-fluorophenyl
hydroxymethyl
ethyl



2.5.1115
3-ethoxy-6-fluorophenyl
hydroxymethyl
ethyl



2.5.1116
3-trifluoromethoxy-6-fluorophenyl
hydroxymethyl
ethyl



2.5.1117
3-nitro-6-fluorophenyl
hydroxymethyl
ethyl



2.5.1118
3-fluoro-6-chlorophenyl
hydroxymethyl
ethyl



2.5.1119
3-fluoro-6-chlorophenyl
1-hydroxyethyl
ethyl



2.5.1120
3-fluoro-6-chlorophenyl
1-hydroxypropyl
ethyl



2.5.1121
3-fluoro-6-chlorophenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.1122
3-fluoro-6-chlorophenyl
methoxymethyl
ethyl



2.5.1123
3-fluoro-6-chlorophenyl
2-methoxyethyl
ethyl



2.5.1124
3,6-dichlorophenyl
hydroxymethyl
ethyl



2.5.1125
3,6-dichlorophenyl
1-hydroxyethyl
ethyl



2.5.1126
3,6-dichlorophenyl
1-hydroxypropyl
ethyl



2.5.1127
3,6-dichlorophenyl
(1-hydroxy-2-
ethyl





methylpropyl)




2.5.1128
3,6-dichlorophenyl
methoxymethyl
ethyl



2.5.1129
3,6-dichlorophenyl
2-methoxyethyl
ethyl



2.5.1130
3-bromo-6-chlorophenyl
hydroxymethyl
ethyl



2.5.1131
3-methyl-6-chlorophenyl
hydroxymethyl
ethyl



2.5.1132
3-ethyl-6-chlorophenyl
hydroxymethyl
ethyl



2.5.1133
3-cyclopropyl-6-chlorophenyl
hydroxymethyl
ethyl



2.5.1134
3-cyano-6-chlorophenyl
hydroxymethyl
ethyl



2.5.1135
3-trifluoromethyl-6-chlorophenyl
hydroxymethyl
ethyl



2.5.1136
3-methoxy-6-chlorophenyl
hydroxymethyl
ethyl



2.5.1137
3-ethoxy-6-chlorophenyl
hydroxymethyl
ethyl



2.5.1138
3-trifluoromethoxy-6-chlorophenyl
hydroxymethyl
ethyl



2.5.1139
3-nitro-6-chlorophenyl
hydroxymethyl
ethyl



2.5.1140
3-fluoro-6-bromophenyl
hydroxymethyl
ethyl



2.5.1141
3-chloro-6-bromophenyl
hydroxymethyl
ethyl



2.5.1142
3,6-dibromophenyl
hydroxymethyl
ethyl



2.5.1143
3-methyl-6-bromophenyl
hydroxymethyl
ethyl



2.5.1144
3-cyclopropyl-6-bromophenyl
hydroxymethyl
ethyl



2.5.1145
3-cyano-6-bromophenyl
hydroxymethyl
ethyl



2.5.1146
3-trifluoromethyl-6-bromophenyl
hydroxymethyl
ethyl



2.5.1147
3-methoxy-6-phenyl
hydroxymethyl
ethyl



2.5.1148
3-ethoxy-6-bromophenyl
hydroxymethyl
ethyl



2.5.1149
3-trifluoromethoxy-6-bromophenyl
hydroxymethyl
ethyl



2.5.1150
3-nitro-6-bromophenyl
hydroxymethyl
ethyl



2.5.1151
3-fluoro-6-iodophenyl
hydroxymethyl
ethyl



2.5.1152
3-chloro-6-iodophenyl
hydroxymethyl
ethyl



2.5.1153
3-bromo-6-iodophenyl
hydroxymethyl
ethyl



2.5.1154
3-methyl-6-iodophenyl
hydroxymethyl
ethyl



2.5.1155
3-cyclopropyl-6-iodophenyl
hydroxymethyl
ethyl



2.5.1156
3-cyano-6-iodophenyl
hydroxymethyl
ethyl



2.5.1157
3-trifluoromethyl-6-iodophenyl
hydroxymethyl
ethyl



2.5.1158
3-methoxy-6-iodophenyl
hydroxymethyl
ethyl



2.5.1159
3-ethoxy-6-iodophenyl
hydroxymethyl
ethyl



2.5.1160
3-trifluoromethoxy-6-iodophenyl
hydroxymethyl
ethyl



2.5.1161
3-nitro-6-iodophenyl
hydroxymethyl
ethyl



2.5.1162
3-fluoro-6-methylphenyl
hydroxymethyl
ethyl



2.5.1163
3-chloro-6-methylphenyl
hydroxymethyl
ethyl



2.5.1164
3-bromo-6-methylphenyl
hydroxymethyl
ethyl



2.5.1165
3,6-dimethylphenyl
hydroxymethyl
ethyl



2.5.1166
3-cyclopropyl-6-methylphenyl
hydroxymethyl
ethyl



2.5.1167
3-cyano-6-methylphenyl
hydroxymethyl
ethyl



2.5.1168
3-trifluoromethyl-6-methylphenyl
hydroxymethyl
ethyl



2.5.1169
3-methoxy-6-methylphenyl
hydroxymethyl
ethyl



2.5.1170
3-ethoxy-6-methylphenyl
hydroxymethyl
ethyl



2.5.1171
3-trifluoromethoxy-6-methylphenyl
hydroxymethyl
ethyl



2.5.1172
3-nitro-6-methylphenyl
hydroxymethyl
ethyl



2.5.1173
3-fluoro-6-ethylphenyl
hydroxymethyl
ethyl



2.5.1174
3-chloro-6-ethylphenyl
hydroxymethyl
ethyl



2.5.1175
3-bromo-6-ethylphenyl
hydroxymethyl
ethyl



2.5.1176
3-methyl-6-ethylphenyl
hydroxymethyl
ethyl



2.5.1177
3,6-diethylphenyl
hydroxymethyl
ethyl



2.5.1178
3-cyclopropyl-6-ethylphenyl
hydroxymethyl
ethyl



2.5.1179
3-cyano-6-ethylphenyl
hydroxymethyl
ethyl



2.5.1180
3-trifluoromethyl-6-ethylphenyl
hydroxymethyl
ethyl



2.5.1181
3-methoxy-6-ethylphenyl
hydroxymethyl
ethyl



2.5.1182
3-ethoxy-6-ethylphenyl
hydroxymethyl
ethyl



2.5.1183 
3-trifluoromethoxy-6-ethylphenyl
hydroxymethyl
ethyl



2.5.1184
3-nitro-6-ethylphenyl
hydroxymethyl
ethyl



2.5.1185
3-fluoro-6-isopropylphenyl
hydroxymethyl
ethyl



2.5.1186
3-chloro-6-isopropylphenyl
hydroxymethyl
ethyl



2.5.1187
3-bromo-6-isopropylphenyl
hydroxymethyl
ethyl



2.5.1188
3-methyl-6-isopropylphenyl
hydroxymethyl
ethyl



2.5.1189
3-ethyl-6-isopropylphenyl
hydroxymethyl
ethyl



2.5.1190
3-cyclopropyl-6-isopropylphenyl
hydroxymethyl
ethyl



2.5.1191
3-cyano-6-isopropylphenyl
hydroxymethyl
ethyl



2.5.1192
3-trifluoromethyl-6-isopropylphenyl
hydroxymethyl
ethyl



2.5.1193
3-methoxy-6-isopropylphenyl
hydroxymethyl
ethyl



2.5.1194
3-ethoxy-6-isopropylphenyl
hydroxymethyl
ethyl



2.5.1195
3-trifluoromethoxy-6-isopropylphenyl
hydroxymethyl
ethyl



2.5.1196
3-nitro-6-isopropylphenyl
hydroxymethyl
ethyl



2.5.1197
3-fluoro-6-tert-butylphenyl
hydroxymethyl
ethyl



2.5.1198
3-chloro-6-tert-butylphenyl
hydroxymethyl
ethyl



2.5.1199
3-bromo-6-tert-butylphenyl
hydroxymethyl
ethyl



2.5.1200
3-methyl-6-tert-butylphenyl 
hydroxymethyl
ethyl



2.5.1201 
3-cyclopropyl-6-tert-butylphenyl
hydroxymethyl
ethyl



2.5.1202
3-cyano-6-tert-butylphenyl
hydroxymethyl
ethyl



2.5.1203
3-trifluoromethyl-6-tert-butylphenyl
hydroxymethyl
ethyl



2.5.1204
3-methoxy-6-tert-butylphenyl
hydroxymethyl
ethyl



2.5.1205
3-ethoxy-6-tert-butylphenyl
hydroxymethyl
ethyl



2.5.1206
3-trifluoromethoxy-6-tert-butylphenyl
hydroxymethyl
ethyl



2.5.1207
3-nitro-6-tert-butylphenyl
hydroxymethyl
ethyl



2.5.1208
3-fluoro-6-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.1209
3-chloro-6-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.1210
3-bromo-6-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.1211
3-methyl-6-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.1212
3,6-dicyclopropylphenyl
hydroxymethyl
ethyl



2.5.1213
3-cyano-6-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.1214
3-trifluoromethyl-6-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.1215 
3-methoxy-6-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.1216
3-ethoxy-6-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.1217
3-trifluoromethoxy-6-cyclopropylphenyl
hydroxymethyl
ethyl



2.5.1218
3-fluoro-6-methoxycarbonyl-phenyl
hydroxymethyl
ethyl



2.5.1219
3-chloro-6-methoxycarbonyl-phenyl
hydroxymethyl
ethyl



2.5.1220
3-bromo-6-methoxycarbonyl-phenyl
hydroxymethyl
ethyl



2.5.1221
3-methyl-6-methoxycarbonyl-phenyl
hydroxymethyl
ethyl



2.5.1222
3-cyclopropyl-6-methoxycarbonyl-
hydroxymethyl
ethyl




phenyl





2.5.1223
3-cyano-6-methoxycarbonyl-phenyl
hydroxymethyl
ethyl



2.5.1224
3-trifluoromethyl-6-
hydroxymethyl
ethyl




methoxycarbonyl-phenyl





2.5.1225
3-methoxy-6-methoxycarbonyl-phenyl
hydroxymethyl
ethyl



2.5.1226
3-ethoxy-6-methoxycarbonyl-phenyl
hydroxymethyl
ethyl



2.5.1227
3-trifluoromethoxy-6-
hydroxymethyl
ethyl




methoxycarbonyl-phenyl





2.5.1228
3-nitro-6-methoxycarbonyl-phenyl
hydroxymethyl
ethyl



2.5.1229
3-fluoro-6-cyanophenyl
hydroxymethyl
ethyl



2.5.1230
3-chloro-6-cyanophenyl
hydroxymethyl
ethyl



2.5.1231
3-bromo-6-cyanophenyl
hydroxymethyl
ethyl



2.5.1232
3-methyl-6-cyanophenyl
hydroxymethyl
ethyl



2.5.1233
3-cyclopropyl-6-cyanophenyl
hydroxymethyl
ethyl



2.5.1234
3,6-dicyanophenyl
hydroxymethyl
ethyl



2.5.1235
3-trifluoromethyl-6-cyanophenyl
hydroxymethyl
ethyl



2.5.1236
3-methoxy-6-cyanophenyl
hydroxymethyl
ethyl



2.5.1237
3-ethoxy-6-cyanophenyl
hydroxymethyl
ethyl



2.5.1238
3-trifluoromethoxy-6-cyanophenyl
hydroxymethyl
ethyl



2.5.1239
3-nitro-6-cyanophenyl
hydroxymethyl
ethyl



2.5.1240
3-fluoro-6-methoxyphenyl
hydroxymethyl
ethyl



2.5.1241
3-chloro-6-methoxyphenyl
hydroxymethyl
ethyl



2.5.1242
3-bromo-6-methoxyphenyl
hydroxymethyl
ethyl



2.5.1243
3-methyl-6-methoxyphenyl
hydroxymethyl
ethyl



2.5.1244
3-cyclopropyl-6-methoxyphenyl
hydroxymethyl
ethyl



2.5.1245
3-cyano-6-methoxyphenyl
hydroxymethyl
ethyl



2.5.1246
3-trifluoromethyl-6-methoxyphenyl
hydroxymethyl
ethyl



2.5.1247
3,6-dimethoxyphenyl
hydroxymethyl
ethyl



2.5.1248
3-ethoxy-6-methoxyphenyl
hydroxymethyl
ethyl



2.5.1249
3-trifluoromethoxy-6-methoxyphenyl
hydroxymethyl
ethyl



2.5.1250
3-nitro-6-methoxyphenyl
hydroxymethyl
ethyl



2.5.1251
3-fluoro-6-ethoxyphenyl
hydroxymethyl
ethyl



2.5.1252
3-chloro-6-ethoxyphenyl
hydroxymethyl
ethyl



2.5.1253
3-bromo-6-ethoxyphenyl
hydroxymethyl
ethyl



2.5.1254
3-methyl-6-ethoxyphenyl
hydroxymethyl
ethyl



2.5.1255
3-cyclopropyl-6-ethoxyphenyl
hydroxymethyl
ethyl



2.5.1256
3-cyano-6-ethoxyphenyl
hydroxymethyl
ethyl



2.5.1257
3-trifluoromethyl-6-ethoxyphenyl
hydroxymethyl
ethyl



2.5.1258
3-methoxy-6-ethoxyphenyl
hydroxymethyl
ethyl



2.5.1259
2,6-diethoxyphenyl
hydroxymethyl
ethyl



2.5.1260
3-trifluoromethoxy-6-ethoxyphenyl
hydroxymethyl
ethyl



2.5.1261
3-nitro-6-ethoxyphenyl
hydroxymethyl
ethyl



2.5.1262
3-fluoro-6-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.1263
3-chloro-6-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.1264
3-bromo-6-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.1265
3-methyl-6-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.1266
3-cyclopropyl-6-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.1267
3-cyano-6-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.1268
3-trifluoromethyl-6-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.1269
3-methoxy-6-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.1270
3-trifluoromethoxy-6-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.1271
3-nitro-6-isopropoxyphenyl
hydroxymethyl
ethyl



2.5.1272
3-fluoro-6-trifluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1273
3-chloro-6-trifluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1274
3-bromo-6-trifluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1275
3-methyl-6-trifluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1276
3-cyclopropyl-6-trifluoromethoxyphenyl
hydroxymethyl
ethyl



2.5.1277
3-cyano-6-trifluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1278
3-trifluoromethyl-6-
hydroxymethyl
ethyl




trifluoromethoxyphenyl





2.5.1279
3-methoxy-6-trifluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1280
3-ethoxy-6-trifluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1281
3,6-bis(trifluoromethoxy)phenyl 
hydroxymethyl
ethyl



2.5.1282
3-nitro-6-trifluoromethoxyphenyl
hydroxymethyl
ethyl



2.5.1283
3-fluoro-6-difluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1284
3-chloro-6-difluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1285
3-bromo-6-difluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1286
3-methyl-6-difluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1287
3-ethyl-6-difluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1288
3-cyclopropyl-6-difluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1289
3-cyano-6-difluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1290
3-trifluoromethyl-6-
hydroxymethyl
ethyl




difluoromethoxyphenyl





2.5.1291
3-methoxy-6-difluoromethoxy-phenyl
hydroxymethyl
ethyl



2.5.1292
3-nitro-6-difluoromethoxyphenyl
hydroxymethyl
ethyl



2.5.1293
3-fluoro-6-nitrophenyl
hydroxymethyl
ethyl



2.5.1294
3-chloro-6-nitrophenyl
hydroxymethyl
ethyl



2.5.1295
3-bromo-6-nitrophenyl
hydroxymethyl
ethyl



2.5.1296
3-methyl-6-nitrophenyl
hydroxymethyl
ethyl



2.5.1297
3-cyclopropyl-6-nitrophenyl
hydroxymethyl
ethyl



2.5.1298
3-cyano-6-nitrophenyl
hydroxymethyl
ethyl



2.5.1299
3-trifluoromethyl-6-nitrophenyl 
hydroxymethyl
ethyl



2.5.1300
3-methoxy-6-nitrophenyl
hydroxymethyl
ethyl



2.5.1301
3-trifluoromethoxy-6-nitrophenyl 
hydroxymethyl
ethyl



2.5.1302
3-fluoro-6-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.1303
3-chloro-6-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.1304
3-bromo-6-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.1305
3-methyl-6-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.1306
3-cyclopropyl-6-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.1307
3-cyano-6-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.1308
3-trifluoromethyl-6-
hydroxymethyl
ethyl




methylsulfanylphenyl





2.5.1309
3-methoxy-6-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.1310
3-trifluoromethoxy-6-
hydroxymethyl
ethyl




methylsulfanylphenyl





2.5.1311
3-nitro-6-methylsulfanylphenyl
hydroxymethyl
ethyl



2.5.1312
2,3,4-trifluorophenyl
hydroxymethyl
ethyl



2.5.1313
2,3,4-trichlorophenyl
hydroxymethyl
ethyl



2.5.1314
2,3,4-trimethylphenyl
hydroxymethyl
ethyl



2.5.1315
2-fluoro-2-chloro-5-
hydroxymethyl
ethyl




trifluoromethylphenyl





2.5.1316
2,3,5-trifluorophenyl
hydroxymethyl
ethyl



2.5.1317
2,3,5-trichlorophenyl
hydroxymethyl
ethyl



2.5.1318
2,3,5-trimethylphenyl
hydroxymethyl
ethyl



2.5.1319
2,3-dichloro-5-methoxyphenyl
hydroxymethyl
ethyl



2.5.1320
2,3,6-trifluorophenyl
hydroxymethyl
ethyl



2.5.1321
2,3,6-trichlorophenyl
hydroxymethyl
ethyl



2.5.1322
2,3,6-trimethylphenyl
hydroxymethyl
ethyl



2.5.1323
3,4,5-trifluorophenyl
hydroxymethyl
ethyl



2.5.1324
3,4,5-trichlorophenyl
hydroxymethyl
ethyl



2.5.1325
3,4,5-trimethylphenyl
hydroxymethyl
ethyl



2.5.1326
3,5-dimethyl-4-fluorophenyl
hydroxymethyl
ethyl



2.5.1327
3,5-dichloro-4-methoxyphenyl
hydroxymethyl
ethyl



2.5.1328
3,5-difluoro-4-chlorophenyl
hydroxymethyl
ethyl



2.5.1329
3,5-dichloro-4-hydroxyphenyl
hydroxymethyl
ethyl



2.5.1330
3,5-trifluoromethyl-4-chlorophenyl
hydroxymethyl
ethyl



2.5.1331
3,4,6-trifluorophenyl
hydroxymethyl
ethyl



2.5.1332
3,4,6-trichlorophenyl
hydroxymethyl
ethyl



2.5.1333
3,4,6-trimethylphenyl
hydroxymethyl
ethyl



2.5.1334
pentafluorophenyl
hydroxymethyl
ethyl
















TABLE 2.6







Inventive compounds of the general formula (I) in which W* is COOY, R1 and R2 are each hydrogen, and aryl is the radical.








 











No.
Aryl
R3
Y
Physical data





2.6.1
3-fluorophenyl
methyl
(cyclohex-2-en-1-one)-3-yl



2.6.2
3-fluorophenyl
methyl
(propan-1-ol)-3-yl



2.6.3
3-fluorophenyl
methyl
(2,2-dimethylpropan-1-ol)-3-yl



2.6.4
3-fluorophenyl
methyl
(methyl 2,2-dimethyl 






propanoate)-3-yl



2.6.5
3-fluorophenyl
methyl
(methyl propanoate)-3-yl



2.6.6
3-fluorophenyl
methyl
(ethyl propanoate)-3-yl



2.6.7
3-fluorophenyl
methyl
4-ethoxy-4-oxobutan-2-yl



2.6.8
3-fluorophenyl
methyl
(ethyl (3R)-4,4,4-






trifluorobutanoate)-3-yl



2.6.9
3-fluorophenyl
methyl
(butan-1-ol)-4-yl
[CDCl3] 1.55 (bs , 1H); 1.65 (mc, 2H); 1.75 






(s, 3H); 1.80 (mc, 2H); 3.18 (d, 1H); 3.68 (t, 






2H); 3.85 (d, 1H); 4.25 (t, 2H); 7.11 (m, 1H); 






7.40 (m, 3H).


2.6.10
3-fluorophenyl
methyl
(3-methylbutan-2-one)-4-yl



2.6.11
3-fluorophenyl
methyl
(pent-3-en-2-one)-4-yl



2.6.12
3-fluorophenyl
methyl
((2S)-dimethyl butanedioate)-






2-yl



2.6.13
3-fluorophenyl
methyl
(dimethyl pentanedioate)-3-yl



2.6.14
3-fluorophenyl
ethyl
(dimethyl pentanedioate)-3-yl
[CDCl3] D1 0.98 (t, 3H); 1.24 (t, 3H); 1.35 






(d, 3H); 1.95-2.12 (m, 2H); 2.50-2.75 (m, 






2H); 3.18 (d, 1H); 3.81 (d, 1H); 3.98-4.09 






(m, 2H); 5.33-5.42 (m, 1H); 7.12 (t, 1H); 






7.33-7.43 (m 3H). D2 1.02 (t, 3H); 1.19 (t, 






3H); 1.36 (d, 3H); 1.95-2.12 (m, 2H); 






2.50-2.75 (m, 2H); 3.20 (d, 1H); 3.76 (d, 






1H); 4.09-4.17 (m, 2H); 5.33-5.42 (m, 1H); 






7.12 (t, 1H); 7.33-7.43 (m 3H).


2.6.15
3-fluorophenyl
methyl
(methyl (2R)-2-methyl 






propanoate)-3-yl



2.6.16
3-fluorophenyl
methyl
4-methoxycarbonylbenzyl



2.6.17
3-fluorophenyl
methyl
3,5-difluorobenzyl



2.6.18
3-fluorophenyl
methyl
3,4-difluorobenzyl



2.6.19
3-fluorophenyl
methyl
2,6-difluorobenzyl



2.6.20
3-fluorophenyl
methyl
(5-methylpyridin-3-yl)methyl
[CDCl3] 1.73 (s, 3H); 2.36 (s, 3H); 3.20 (d, 






1H); 3.85 (d, 1H); 5.22 (s, 2H); 7.13 (m, 1H); 






7.39 (m, 3H); 7.51 (s, 1H); 8.42 (d, 2H).


2.6.21
3-fluorophenyl
methyl
(tetrahydrofuran)-3-yl



2.6.22
3-fluorophenyl
ethyl
4-ethoxy-4-oxobutan-2-yl



2.6.23
3-chlorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.24
3-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.25
3-iodophenyl
ethyl
(ethyl butanoate)-3-yl



2.6.26
3-methylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.27
3-methylphenyl
ethyl
(ethyl butanoate)-3-yl



2.6.28
3-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.29
3-propylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.30
3-isopropylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.31
3-n-butylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.32
3-i-butylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.33
3-tert-butylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.34
3-cyclopropyl-phenyl
methyl
(ethyl butanoate)-3-yl



2.6.35
3-cyclobutyl-phenyl
methyl
(ethyl butanoate)-3-yl



2.6.36
3-cyclopentyl-phenyl
methyl
(ethyl butanoate)-3-yl



2.6.37
3-vinylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.38
3-ethynylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.39
3-cyanophenyl
methyl
(ethyl butanoate)-3-yl



2.6.40
3-trifluoromethyl-
methyl
(ethyl butanoate)-3-yl




phenyl





2.6.41
3-difluoromethyl-
methyl
(ethyl butanoate)-3-yl




phenyl





2.6.42
3-(hydroxy-
methyl
(ethyl butanoate)-3-yl




carbonyl)phenyl





2.6.43
3-(methoxy-
methyl
(ethyl butanoate)-3-yl




carbonyl)phenyl





2.6.44
3-(ethoxy-
methyl
(ethyl butanoate)-3-yl




carbonyl)phenyl





2.6.45
3-hydroxymethyl-
methyl
(ethyl butanoate)-3-yl




phenyl





2.6.46
3-acetylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.47
3-carbamoyl-phenyl
methyl
(ethyl butanoate)-3-yl



2.6.48
3-hydroxyphenyl
methyl
(ethyl butanoate)-3-yl



2.6.49
3-methoxyphenyl
methyl
(ethyl butanoate)-3-yl



2.6.50
3-ethoxyphenyl
methyl
(ethyl butanoate)-3-yl



2.6.51
3-propyloxyphenyl
methyl
(ethyl butanoate)-3-yl



2.6.52
3-isopropyloxy-phenyl
methyl
(ethyl butanoate)-3-yl



2.6.53
3-n-butyloxy-phenyl
methyl
(ethyl butanoate)-3-yl



2.6.54
3-i-butyloxyphenyl
methyl
(ethyl butanoate)-3-yl



2.6.55
3-t-butyloxyphenyl
methyl
(ethyl butanoate)-3-yl



2.6.56
3-difluoro-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.57
3-trifluoro-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.58
3-(2,2,2-trifluoro-
methyl
(ethyl butanoate)-3-yl




ethoxy)phenyl





2.6.59
3-(2-chloro-
methyl
(ethyl butanoate)-3-yl




ethoxy)phenyl





2.6.60
3-(2-hydroxy-
methyl
(ethyl butanoate)-3-yl




ethoxy)phenyl





2.6.61
3-(2-methoxy-
methyl
(ethyl butanoate)-3-yl




ethoxy)phenyl





2.6.62
3-[(tert-butoxy-
methyl
(ethyl butanoate)-3-yl




carbonyl)oxy]-phenyl





2.6.63
3-nitrophenyl
methyl
(ethyl butanoate)-3-yl



2.6.64
3-acetoxyphenyl
methyl
(ethyl butanoate)-3-yl



2.6.65
{3-[(tert-butoxy-
methyl
(ethyl butanoate)-3-yl




carbonyl)amino]-






phenyl}





2.6.66
3-methylsulfanyl-
methyl
(ethyl butanoate)-3-yl




phenyl





2.6.67
3-ethylsulfanyl-phenyl
methyl
(ethyl butanoate)-3-yl



2.6.68
3-(pentafluoro-
methyl
(ethyl butanoate)-3-yl




lambda6-sulfanyl)-






phenyl





2.6.69
2,3-difluorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.70
2-chloro-3-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.71
2-bromo-3-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.72
2-methyl-3-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.73
2-ethyl-3-fluorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.74
2-cyclopropyl-3-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.75
2-vinyl-3-fluorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.76
2-ethynyl-3-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.77
2-cyano-3-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.78
2-methoxy-3-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.79
2-ethoxy-3-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.80
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.81
2-nitro-3-fluorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.82
2-fluoro-3-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.83
2,3-dichloro-phenyl
methyl
(ethyl butanoate)-3-yl



2.6.84
2-bromo-3-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.85
2-methyl-3-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.86
2-ethyl-3-chlorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.87
2-cyclopropyl-3-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.88
2-vinyl-3-chlorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.89
2-ethynyl-3-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.90
2-cyano-3-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.91
2-trifluoromethyl-2-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.92
2-methoxy-3-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.93
2-ethoxy-3-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.94
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.95
2-nitro-3-chlorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.96
2-fluoro-3-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.97
2-chloro-3-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.98
2,3-dibromo-phenyl
methyl
(ethyl butanoate)-3-yl



2.6.99
2-methyl-3-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.100
2-ethyl-3-bromophenyl
methyl
(ethyl butanoate)-3-yl



2.6.101
2-cyclopropyl-3-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.102
2-vinyl-3-bromophenyl
methyl
(ethyl butanoate)-3-yl



2.6.103
2-ethynyl-3-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.104
2-cyano-3-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.105
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.106
2-methoxy-3-phenyl
methyl
(ethyl butanoate)-3-yl



2.6.107
2-ethoxy-3-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.108
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.109
2-nitro-3-bromophenyl
methyl
(ethyl butanoate)-3-yl



2.6.110
2-fluoro-3-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.111
2-chloro-3-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.112
2-bromo-3-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.113
2-methyl-3-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.114
2-ethyl-3-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.115
2-cyclopropyl-3-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.116
2-vinyl-3-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.117
2-ethynyl-3-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.118
2-cyano-3-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.119
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.120
2-methoxy-3-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.121
2-ethoxy-3-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.122
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.123
2-nitro-3-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.124
2-fluoro-3-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.125
2-chloro-3-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.126
2-bromo-3-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.127
2,3-dimethyl-phenyl
methyl
(ethyl butanoate)-3-yl



2.6.128
2-ethyl-3-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.129
2-cyclopropyl-3-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.130
2-vinyl-3-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.131
2-ethynyl-3-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.132
2-cyano-3-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.133
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.134
2-methoxy-3-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.135
2-ethoxy-3-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.136
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.137
2-nitro-3-methylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.138
2-fluoro-3-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.139
2-chloro-3-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.140
2-bromo-3-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.141
2-methyl-3-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.142
2,3-diethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.143
2-cyclopropyl-3-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.144
2-vinyl-3-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.145
2-ethynyl-3-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.146
2-cyano-3-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.147
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.148
2-methoxy-3-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.149
2-ethoxy-3-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.150
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.151
2-nitro-3-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.152
2-fluoro-3-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.153
2-chloro-3-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.154
2-bromo-3-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.155
2-methyl-3-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.156
2-methyl-3-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.157
2-cyclopropyl-3-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.158
2-vinyl-3-propylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.159
2-ethynyl-
methyl
(ethyl butanoate)-3-yl




3propylphenyl





2.6.160
2-cyano-3-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.161
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.162
2-methoxy-3-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.163
2-ethoxy-3-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.164
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.165
2-nitro-3-propylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.166
2-fluoro-3-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.167
2-chloro-3-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.168
2-bromo-3-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.169
2-methyl-3-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.170
2-ethyl-3-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.171
2-cyclopropyl-3-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.172
2-vinyl-3-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.173
2-ethynyl-3-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.174
2-cyano-3-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.175
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.176
2-methoxy-3-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.177
2-ethoxy-3-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.178
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.179
2-nitro-3-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.180
2-fluoro-3-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.181
2-chloro-3-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.182
2-bromo-3-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.183
2-methyl-3-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.184
2-ethyl-3-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.185
2-cyclopropyl-3-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.186
2-vinyl-3-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.187
2-ethynyl-3-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.188
2-cyano-3-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.189
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




tert-butylphenyl





2.6.190
2-methoxy-3-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.191
2-ethoxy-3-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.192
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




tert-butylphenyl





2.6.193
2-nitro-3-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.194
2-fluoro-3-hydroxy-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.195
2-chloro-3-hydroxy-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.196
2-bromo-3-hydroxy-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.197
2-methyl-3-hydroxy-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.198
2-ethyl-3-hydroxy-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.199
2-cyclopropyl-3-
methyl
(ethyl butanoate)-3-yl




hydroxymethylphenyl





2.6.200
2-vinyl-3-hydroxy-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.201
2-ethynyl-3-hydroxy-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.202
2-cyano-3-hydroxy-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.203
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




hydroxy-methylphenyl





2.6.204
2-methoxy-3-hydroxy-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.205
2-ethoxy-3-hydroxy-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.206
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




hydroxymethyl-phenyl





2.6.207
2-nitro-3-hydroxy-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.208
2-fluoro-3-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.209
2-chloro-3-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.210
2-bromo-3-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.211
2-methyl-3-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.212
2-ethyl-3-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.213
2-cyclopropyl-3-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.214
2-vinyl-3-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.215
2-ethynyl-3-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.216
2-cyano-3-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.217
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




cyclopropyl-phenyl





2.6.218
2-methoxy-3-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.219
2-ethoxy-3-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.220
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.221
2-fluoro-3-methoxy-
methyl
(ethyl butanoate)-3-yl




carbonylphenyl





2.6.222
2-chloro-3-methoxy-
methyl
(ethyl butanoate)-3-yl




carbonylphenyl





2.6.223
2-bromo-3-methoxy-
methyl
(ethyl butanoate)-3-yl




carbonylphenyl





2.6.224
2-methyl-3-methoxy-
methyl
(ethyl butanoate)-3-yl




carbonylphenyl





2.6.225
2-ethyl-3-methoxy-
methyl
(ethyl butanoate)-3-yl




carbonylphenyl





2.6.226
2-cyclopropyl-3-
methyl
(ethyl butanoate)-3-yl




methoxycarbonyl-






phenyl





2.6.227
2-vinyl-3-methoxy-
methyl
(ethyl butanoate)-3-yl




carbonylphenyl





2.6.228
2-ethynyl-3-
methyl
(ethyl butanoate)-3-yl




methoxycarbonyl-






phenyl





2.6.229
2-cyano-3-methoxy-
methyl
(ethyl butanoate)-3-yl




carbonylphenyl





2.6.230
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




methoxy-






carbonylphenyl





2.6.231
2-methoxy-3-
methyl
(ethyl butanoate)-3-yl




methoxycarbonyl-






phenyl





2.6.232
2-ethoxy-3-methoxy-
methyl
(ethyl butanoate)-3-yl




carbonylphenyl





2.6.233
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




methoxy-






carbonylphenyl





2.6.234
2-nitro-3-methoxy-
methyl
(ethyl butanoate)-3-yl




carbonylphenyl





2.6.235
2-fluoro-3-vinylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.236
2-chloro-3-vinylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.237
2-bromo-3-vinylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.238
2-methyl-3-
methyl
(ethyl butanoate)-3-yl




vinylphenyl





2.6.239
2-ethyl-3-vinylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.240
2-cyclopropyl-3-
methyl
(ethyl butanoate)-3-yl




vinylphenyl





2.6.241
2-vinyl-3-vinylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.242
2-ethynyl-3-
methyl
(ethyl butanoate)-3-yl




vinylphenyl





2.6.243
2-cyano-3-vinylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.244
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




vinylphenyl





2.6.245
2-methoxy-3-
methyl
(ethyl butanoate)-3-yl




vinylphenyl





2.6.246
2-ethoxy-3-
methyl
(ethyl butanoate)-3-yl




vinylphenyl





2.6.247
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




vinylphenyl





2.6.248
2-nitro-3-vinylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.249
2-fluoro-3-
methyl
(ethyl butanoate)-3-yl




ethynylphenyl





2.6.250
2-chloro-3-
methyl
(ethyl butanoate)-3-yl




ethynylphenyl





2.6.251
2-bromo-3-
methyl
(ethyl butanoate)-3-yl




ethynylphenyl





2.6.252
2-methyl-3-
methyl
(ethyl butanoate)-3-yl




ethynylphenyl





2.6.253
2-ethyl-3-
methyl
(ethyl butanoate)-3-yl




ethynylphenyl





2.6.254
2-cyclopropyl-3-
methyl
(ethyl butanoate)-3-yl




ethynylphenyl





2.6.255
2-vinyl-3-
methyl
(ethyl butanoate)-3-yl




ethynylphenyl





2.6.256
2-cyano-3-
methyl
(ethyl butanoate)-3-yl




ethynylphenyl





2.6.257
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




ethynylphenyl





2.6.258
2-methoxy-3-
methyl
(ethyl butanoate)-3-yl




ethynylphenyl





2.6.259
2-ethoxy-3-
methyl
(ethyl butanoate)-3-yl




ethynylphenyl





2.6.260
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




ethynylphenyl





2.6.261
2-nitro-3-
methyl
(ethyl butanoate)-3-yl




ethynylphenyl





2.6.262
2-fluoro-3-
methyl
(ethyl butanoate)-3-yl




ethynylphenyl





2.6.263
2-fluoro-3-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.264
2-chloro-3-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.265
2-bromo-3-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.266
2-methyl-3-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.267
2-ethyl-3-cyanophenyl
methyl
(ethyl butanoate)-3-yl



2.6.268
2-ethyl-3-cyanophenyl
ethyl
(ethyl butanoate)-3-yl



2.6.269
2-ethyl-3-cyanophenyl
propyl
(ethyl butanoate)-3-yl



2.6.270
2-ethyl-3-cyanophenyl
cyclopropyl
(ethyl butanoate)-3-yl



2.6.271
2-cyclopropyl-3-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.272
2-vinyl-3-cyanophenyl
methyl
(ethyl butanoate)-3-yl



2.6.273
2-ethynyl-3-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.274
2-cyano-3-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.275
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.276
2-methoxy-3-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.277
2-ethoxy-3-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.278
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.279
2-nitro-3-cyanophenyl
methyl
(ethyl butanoate)-3-yl



2.6.280
2-fluoro-3-
methyl
(ethyl butanoate)-3-yl




hydroxyphenyl





2.6.281
2-chloro-3-
methyl
(ethyl butanoate)-3-yl




hydroxyphenyl





2.6.282
2-bromo-3-
methyl
(ethyl butanoate)-3-yl




hydroxyphenyl





2.6.283
2-methyl-3-
methyl
(ethyl butanoate)-3-yl




hydroxyphenyl





2.6.284
2-ethyl-3-
methyl
(ethyl butanoate)-3-yl




hydroxyphenyl





2.6.285
2-cyclopropyl-3-
methyl
(ethyl butanoate)-3-yl




hydroxyphenyl





2.6.286
2-vinyl-3-
methyl
(ethyl butanoate)-3-yl




hydroxyphenyl





2.6.287
2-ethynyl-3-
methyl
(ethyl butanoate)-3-yl




hydroxyphenyl





2.6.288
2-cyano-3-
methyl
(ethyl butanoate)-3-yl




hydroxyphenyl





2.6.289
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




hydroxyphenyl





2.6.290
2-methoxy-3-
methyl
(ethyl butanoate)-3-yl




hydroxyphenyl





2.6.291
2-ethoxy-3-
methyl
(ethyl butanoate)-3-yl




hydroxyphenyl





2.6.292
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




hydroxyphenyl





2.6.293
2-nitro-3-
methyl
(ethyl butanoate)-3-yl




hydroxyphenyl





2.6.294
2-fluoro-3-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.295
2-chloro-3-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.296
2-bromo-3-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.297
2-methyl-3-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.298
2-ethyl-3-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.299
2-cyclopropyl-3-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.300
2-vinyl-3-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.301
2-ethynyl-3-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.302
2-cyano-3-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.303
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.304
2,3-dimethoxyphenyl
methyl
(ethyl butanoate)-3-yl



2.6.305
2-ethoxy-3-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.306
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.307
2-nitro-3-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.308
2-fluoro-3-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.309
2-chloro-3-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.310
2-bromo-3-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.311
2-methyl-3-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.312
2-ethyl-3-ethoxyphenyl
methyl
(ethyl butanoate)-3-yl



2.6.313
2-cyclopropyl-3-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.314
2-vinyl-3-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.315
2-ethynyl-3-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.316
2-cyano-3-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.317
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.318
2-methoxy-3-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.319
2,3-diethoxy--phenyl
methyl
(ethyl butanoate)-3-yl



2.6.320
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.321
2-nitro-3-ethoxyphenyl
methyl
(ethyl butanoate)-3-yl



2.6.322
2-fluoro-3-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.323
2-chloro-3-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.324
2-bromo-3-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.325
2-methyl-3-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.326
2-ethyl-3-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.327
2-cyclopropyl-3-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.328
2-vinyl-3-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.329
2-ethynyl-3-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.330
2-cyano-3-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.331
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.332
2-methoxy-3-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.333
2-ethoxy-3-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.334
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.335
2-nitro-3-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.336
2-fluoro-3-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.337
2-chloro-3-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.338
2-bromo-3-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.339
2-methyl-3-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.340
2-ethyl-3-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.341
2-cyclopropyl-3-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.342
2-vinyl-3-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.343
2-ethynyl-3-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.344
2-cyano-3-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.345
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




isopropoxy-phenyl





2.6.346
2-methoxy-3-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.347
2-ethoxy-3-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.348
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.349
2-nitro-3-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.350
2-fluoro-3-tert-
methyl
(ethyl butanoate)-3-yl




butoxyphenyl





2.6.351
2-chloro-3-tert-
methyl
(ethyl butanoate)-3-yl




butoxyphenyl





2.6.352
2-bromo-3-tert-
methyl
(ethyl butanoate)-3-yl




butoxyphenyl





2.6.353
2-methyl-3-tert-
methyl
(ethyl butanoate)-3-yl




butoxyphenyl





2.6.354
2-ethyl-3-tert-
methyl
(ethyl butanoate)-3-yl




butoxyphenyl





2.6.355
2-cyclopropyl-3-tert-
methyl
(ethyl butanoate)-3-yl




butoxyphenyl





2.6.356
2-vinyl-3-tert-
methyl
(ethyl butanoate)-3-yl




butoxyphenyl





2.6.357
2-ethynyl-3-tert-
methyl
(ethyl butanoate)-3-yl




butoxyphenyl





2.6.358
2-cyano-3-tert-
methyl
(ethyl butanoate)-3-yl




butoxyphenyl





2.6.359
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




tert-butoxy-phenyl





2.6.360
2-methoxy-3-tert-
methyl
(ethyl butanoate)-3-yl




butoxyphenyl





2.6.361
2-ethoxy-3-tert-
methyl
(ethyl butanoate)-3-yl




butoxyphenyl





2.6.362
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




tert-butoxyphenyl





2.6.363
2-nitro-3-tert-
methyl
(ethyl butanoate)-3-yl




butoxyphenyl





2.6.364
2-fluoro-3-
methyl
(ethyl butanoate)-3-yl




trifluoromethoxy-






phenyl





2.6.365
2-chloro-3-
methyl
(ethyl butanoate)-3-yl




trifluoromethoxy-






phenyl





2.6.366
2-bromo-3-
methyl
(ethyl butanoate)-3-yl




trifluoromethoxy-






phenyl





2.6.367
2-methyl-3-
methyl
(ethyl butanoate)-3-yl




trifluoromethoxy-






phenyl





2.6.368
2-ethyl-3-
methyl
(ethyl butanoate)-3-yl




trifluoromethoxy-






phenyl





2.6.369
2-cyclopropyl-3-
methyl
(ethyl butanoate)-3-yl




trifluoromethoxy-






phenyl





2.6.370
2-vinyl-3-
methyl
(ethyl butanoate)-3-yl




trifluoromethoxy-






phenyl





2.6.371
2-ethynyl-3-
methyl
(ethyl butanoate)-3-yl




trifluoromethoxy-






phenyl





2.6.372
2-cyano-3-
methyl
(ethyl butanoate)-3-yl




trifluoromethoxy-






phenyl





2.6.373
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




trifluoro-methoxy-






phenyl





2.6.374
2-methoxy-3-
methyl
(ethyl butanoate)-3-yl




trifluoromethoxy-






phenyl





2.6.375
2-ethoxy-3-
methyl
(ethyl butanoate)-3-yl




trifluoromethoxy-






phenyl





2.6.376
2,3-bis(trifluoro-
methyl
(ethyl butanoate)-3-yl




methoxy)phenyl





2.6.377
2-nitro-3-trifluoro-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.378
2-fluoro-3-(2,2,2-
methyl
(ethyl butanoate)-3-yl




trifluoroethoxy)-phenyl





2.6.379
2-chloro-3-(2,2,2-
methyl
(ethyl butanoate)-3-yl




trifluoroethoxy)-phenyl





2.6.380
2-bromo-3-(2,2,2-
methyl
(ethyl butanoate)-3-yl




trifluoroethoxy)-phenyl





2.6.381
2-methyl-3-(2,2,2-
methyl
(ethyl butanoate)-3-yl




trifluoroethoxy)-phenyl





2.6.382
2-ethyl-3-(2,2,2-
methyl
(ethyl butanoate)-3-yl




trifluoroethoxy)-phenyl





2.6.383
2-cyclopropyl-3-(2,2,2-
methyl
(ethyl butanoate)-3-yl




trifluoro-ethoxy)phenyl





2.6.384
2-vinyl-3-(2,2,2-
methyl
(ethyl butanoate)-3-yl




trifluoroethoxy)-phenyl





2.6.385
2-ethynyl-3-(2,2,2-
methyl
(ethyl butanoate)-3-yl




trifluoro-ethoxyphenyl





2.6.386
2-cyano-3-(2,2,2-
methyl
(ethyl butanoate)-3-yl




trifluoroethoxy)-phenyl





2.6.387
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




(2,2,2-trifluoro-






ethoxy)phenyl





2.6.388
2-methoxy-3-(2,2,2-
methyl
(ethyl butanoate)-3-yl




trifluoro-ethoxy)phenyl





2.6.389
2-ethoxy-3-(2,2,2-
methyl
(ethyl butanoate)-3-yl




trifluoroethoxy)-phenyl





2.6.390
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




(2,2,2-trifluoroethoxy)-






phenyl





2.6.391
2-nitro-3-(2,2,2-
methyl
(ethyl butanoate)-3-yl




trifluoroethoxy)-phenyl





2.6.392
2-fluoro-3-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.393
2-chloro-3-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.394
2-bromo-3-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.395
2-methyl-3-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.396
2-ethyl-3-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.397
2-cyclopropyl-3-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.398
2-vinyl-3-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.399
2-ethynyl-3-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.400
2-cyano-3-difluoro-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.401
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




difluoro-






methoxyphenyl





2.6.402
2-methoxy-3-difluoro-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.403
2-ethoxy-3-
methyl
(ethyl butanoate)-3-yl




difluoromethoxyphenyl





2.6.404
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.405
2-nitro-3-difluoro-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.406
2-fluoro-3-(2-
methyl
(ethyl butanoate)-3-yl




methoxyethoxy)-






phenyl





2.6.407
2-chloro-3-(2-
methyl
(ethyl butanoate)-3-yl




methoxyethoxy)-






phenyl





2.6.408
2-bromo-3-(2-
methyl
(ethyl butanoate)-3-yl




methoxyethoxy)-






phenyl





2.6.409
2-methyl-3-(2-
methyl
(ethyl butanoate)-3-yl




methoxyethoxy)-






phenyl





2.6.410
2-ethyl-3-(2-
methyl
(ethyl butanoate)-3-yl




methoxyethoxy)phenyl





2.6.411
2-cyclopropyl-3-(2-
methyl
(ethyl butanoate)-3-yl




methoxy-






ethoxy)phenyl





2.6.412
2-vinyl-3-(2-
methyl
(ethyl butanoate)-3-yl




methoxyethoxy)phenyl





2.6.413
2-ethynyl-3-(2-
methyl
(ethyl butanoate)-3-yl




methoxyethoxy)-






phenyl





2.6.414
2-cyano-3-(2-
methyl
(ethyl butanoate)-3-yl




methoxyethoxy)-






phenyl





2.6.415
2-trifluoromethyl-3-(2-
methyl
(ethyl butanoate)-3-yl




methoxy-






ethoxy)phenyl





2.6.416
2-methoxy-3-(2-
methyl
(ethyl butanoate)-3-yl




methoxyethoxy)-






phenyl





2.6.417
2-ethoxy-3-(2-
methyl
(ethyl butanoate)-3-yl




methoxyethoxy)-






phenyl





2.6.418
2-trifluoro-methoxy-
methyl
(ethyl butanoate)-3-yl




(2-methoxyethoxy)-






phenyl





2.6.419
2-nitro-3-(2-
methyl
(ethyl butanoate)-3-yl




methoxyethoxy)phenyl





2.6.420
2-fluoro-3-(tert-
methyl
(ethyl butanoate)-3-yl




butoxycarbonyloxy)-






phenyl





2.6.421
2-chloro-3-(tert-
methyl
(ethyl butanoate)-3-yl




butoxycarbonyloxy)-






phenyl





2.6.422
2-bromo-3-(tert-
methyl
(ethyl butanoate)-3-yl




butoxycarbonyl-






oxy)phenyl





2.6.423
2-methyl-3-(tert-
methyl
(ethyl butanoate)-3-yl




butoxycarbonyl-






oxy)phenyl





2.6.424
2-ethyl-3-(tert-
methyl
(ethyl butanoate)-3-yl




butoxycarbonyloxy)-






phenyl





2.6.425
2-cyclopropyl-3-(tert-
methyl
(ethyl butanoate)-3-yl




butoxy-carbonyloxy)-






phenyl





2.6.426
2-vinyl-3-(tert-
methyl
(ethyl butanoate)-3-yl




butoxycarbonyl-oxy)-






phenyl





2.6.427
2-ethynyl-3-(tert-
methyl
(ethyl butanoate)-3-yl




butoxycarbonyl-






oxy)phenyl





2.6.428
2-cyano-3-(tert-
methyl
(ethyl butanoate)-3-yl




butoxycarbonyl-oxy)-






phenyl





2.6.429
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




(tert-butoxy-






carbonyloxy)-phenyl





2.6.430
2-methoxy-3-(tert-
methyl
(ethyl butanoate)-3-yl




butoxycarbonyl-oxy)-






phenyl





2.6.431
2-ethoxy-3-(tert-
methyl
(ethyl butanoate)-3-yl




butoxycarbonyl-oxy)-






phenyl





2.6.432
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




(tert-butoxycarbonyl-






oxy)phenyl





2.6.433
2-nitro-3-(tert-
methyl
(ethyl butanoate)-3-yl




butoxycarbonyl-oxy)-






phenyl





2.6.434
2-fluoro-3-nitrophenyl
methyl
(ethyl butanoate)-3-yl



2.6.435
2-chloro-3-nitrophenyl
methyl
(ethyl butanoate)-3-yl



2.6.436
2-bromo-3-nitrophenyl
methyl
(ethyl butanoate)-3-yl



2.6.437
2-methyl-3-nitrophenyl
methyl
(ethyl butanoate)-3-yl



2.6.438
2-ethyl-3-nitrophenyl
methyl
(ethyl butanoate)-3-yl



2.6.439
2-cyclopropyl-3-
methyl
(ethyl butanoate)-3-yl




nitrophenyl





2.6.440
2-vinyl-3-nitrophenyl
methyl
(ethyl butanoate)-3-yl



2.6.441
2-ethynyl-3-
methyl
(ethyl butanoate)-3-yl




nitrophenyl





2.6.442
2-cyano-3-nitrophenyl
methyl
(ethyl butanoate)-3-yl



2.6.443
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




nitrophenyl





2.6.444
2-methoxy-3-
methyl
(ethyl butanoate)-3-yl




nitrophenyl





2.6.445
2-ethoxy-3-nitrophenyl
methyl
(ethyl butanoate)-3-yl



2.6.446
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




nitrophenyl





2.6.447
2-fluoro-3-methyl-
methyl
(ethyl butanoate)-3-yl




sulfanylphenyl





2.6.448
2-chloro-3-methyl-
methyl
(ethyl butanoate)-3-yl




sulfanylphenyl





2.6.449
2-bromo-3-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.450
2-methyl-3-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.451
2-ethyl-3-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.452
2-cyclopropyl-3-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.453
2-vinyl-3-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.454
2-ethynyl-3-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.455
2-cyano-3-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.456
2-trifluoromethyl-3-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.457
2-methoxy-3-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.458
2-ethoxy-3-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.459
2-trifluoro-methoxy-3-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.460
2-nitro-3-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.461
3,5-difluorophenyl
methyl
(cyclohex-2-en-1-one)-3-yl



2.6.462
3,5-difluorophenyl
methyl
(propan-1-ol)-3-yl
[CDCl3] 1.73 (s, 3H); 1.94 (quin, 2H); 3.15 






(d, 1H); 3.73 (t, 2H); 3.85 (d, 1H); 4.38 (t, 






2H); 6.88 (t, 1H); 7.17 (d, 2H).


2.6.463
3,5-difluorophenyl
methyl
(2,2-dimethylpropan-1-ol)-3-yl
[CDCl3] 0.89 (d, 6H), 1.74 (s, 3H), 3.16 (d, 






1H); 3.33 (s, 2H); 3.84 (d, 1H); 4.07 (s, 2H), 






6.88 (t, 1H); 7.18 (d, 2H).


2.6.464
3,5-difluorophenyl
methyl
(methyl 2,2-dimethyl 
[CDCl3] 1.24 (d, 6H); 1.71 (s, 3H); 3.14 (d, 





propanoate)-3-yl
1H); 3.65 (s, 3H); 3.81 (d, 1H); 4.22 (s, 2H); 






6.87 (t, 1H); 7.18 (d, 2H).


2.6.465
3,5-difluorophenyl
methyl
(methyl propanoate)-3-yl
[CDCl3] 1.71 (s, 3H), 2.72 (t, 2H); 3.14 (d, 






1H); 3.68 (s, 3H); 3.82 (d, 1H); 4.47 (m, 2H); 






6.86 (t, 1H); 7.18 (d, 2H).


2.6.466
3,5-difluorophenyl
methyl
(ethyl propanoate)-3-yl



2.6.467
3,5-difluorophenyl
methyl
(ethyl butanoate)-3-yl
[CDCl3] 1.17-1.26 (m, 3H); 1.36 (d, 3H); 






1.69 (d, 3H); 2.55 (m, 1H); 2.69 (m, 1H); 






3.11 (dd, 1H); 3.81 (dd, 1H); 4.03-4.15 (m, 






2H); 5.35 (m, 1H); 6.87 (t, 1H); 7.17 (m, 






2H).


2.6.468
3,5-difluorophenyl
methyl
(ethyl (3R)-4,4,4-
[CDCl3] 1.20 (t, 3H); 1.75 (s, 3H); 2.85 (t, 





trifluorobutanoate)-3-yl one 
2H); 3.19 (d, 1H); 3.85 (d, 1H); 4.09 (m, 





diastereomer
2H); 5.82 (m, 1H); 6.88 (t, 1H); 7.17 (d, 2H).


2.6.469
3,5-difluorophenyl
methyl
(ethyl (3R)-4,4,4-
[CDCl3] 1.25 (t, 3H); 1.74 (s, 3H); 2.86 (d, 





trifluorobutanoate)-3-yl the 
2H); 3.20 (d, 1H); 3.80 (d, 1H); 4.15 (q, 2H); 





other diastereomer
5.80 (m, 1H); 6.88 (t, 1H); 7.18 (d, 2H).


2.6.470
3,5-difluorophenyl
methyl
(butan-2-one)-4-yl
[CDCl3] 1.70 (s, 3H); 2.18 (s, 3H); 2.83 (q, 






2H); 3.15 (d, 1H), 3.83 (d, 1H), 4.44 (m, 2H); 






6.87 (t, 1H); 7.18 (d, 2H).


2.6.471
3,5-difluorophenyl
methyl
(3-methylbutan-2-one)-4-yl
[CDCl3] 1.16 (t, 3H), 1.70 (d, 3H), 2.19 (d, 






3H); 2.95 (quin, 1H), 3.11 (dd, 1H); 3.81 (d, 






1H); 4.21 (dd, 1H); 4.37 (dd, 1H); 6.87 (t, 






1H); 7.18 (m, 2H).


2.6.472
3,5-difluorophenyl
methyl
(pent-3-en-2-one)-4-yl



2.6.473
3,5-difluorophenyl
methyl
((2S)-dimethyl butanedioate)-
[CDCl3] 1.75 (d, 3H); 2.95 (m, 2H); 3.18 (dd, 





2-yl
1H); 3.68 (d, 3H); 3.76 (d, 3H); 3.88 (dd, 






1H); 5.55 (t, 1H); 6.87 (t, 1H); 7.18 (d, 2H).


2.6.474
3,5-difluorophenyl
methyl
(dimethyl pentanedioate)-3-yl
[CDCl3] 1.69 (s, 3H); 2.75 (t, 4H); 3.13 (d, 






1H); 3.62 (s, 3H); 3.69 (s, 3H); 3.83 (d, 1H); 






5.58 (quin, 1H); 6.87 (t, 1H); 7.18 (d, 2H).


2.6.475
3,5-difluorophenyl
methyl
(methyl (2R)-2-methyl 
[CDCl3] D1: 1.22 (t, 3H), 1.71 (s, 3H); 2.88 





propanoate)-3-yl
(m, 1H), 3.15 (d, 1H), 3.66 (s, 3H); 3.81 (d, 






1H), 4.29 (m, 1H); 4.37 (m, 1H), 6.87 (t, 






1H); 7.17 (d, 2H). D2: 1.22 (t, 3H), 1.71 (s, 






3H); 2.88 (m, 1H), 3.15 (d, 1H), 3.67 (s, 3H); 






3.83 (d, 1H), 4.29 (m, 1H); 4.37 (m, 1H), 






6.87 (t, 1H); 7.17 (d, 2H).


2.6.476
3,5-difluorophenyl
methyl
4-methoxycarbonylbenzyl
[CDCl3] 1.75 (s, 3H); 3.17 (d, 1H), 3.84 (d, 






1H); 3.92 (s, 3H); 5.28 (d, 2H); 6.88 (t, 1H); 






7.17 (d, 2H); 7.42 (d, 2H); 8.04 (d, 2H).


2.6.477
3,5-difluorophenyl
methyl
3,5-difluorobenzyl
[CDCl3] 1.76 (s, 3H); 3.19 (d, 1H); 3.84 (d, 






1H); 5.19 (d, 2H); 6.76 (t, 1H); 6.88 (m, 3H); 






7.17 (d, 2H).


2.6.478
3,5-difluorophenyl
methyl
3,4-difluorobenzyl
[CDCl3] 1.73 (s, 3H), 3.17 (d, 1H), 3.82 (d, 






1H); 5.18 (d, 2H); 6.87 (t, 1H); 7.10 (m, 1H); 






7.15 (m, 4H).


2.6.479
3,5-diluorophenyl
methyl
2,6-difluorobenzyl
[CDCl3] 1.72 (s, 3H); 3.15 (d, 1H); 3.82 (d, 






1H); 3.33 (d, 2H); 6.86 (t, 1H); 6.94 (t, 2H); 






7.16 (d, 2H); 7.35 (m, 1H).


2.6.480
3,5-diluorophenyl
methyl
(5-methylpyridin-3-yl)methyl
[CDCl3] 1.73 (s, 3H), 2.34 (s, 3H), 3.17 (d, 






1H); 3.82 (d, 1H); 5.22 (d, 2H); 6.88 (t, 1H); 






7.17 (d, 2H), 7.51 (s, 1H); 8.43 (s, 2H).


2.6.481
3,5-diluorophenyl
methyl
(tetrahydrofuran)-3yl
[CDCl3] 1.72 (s, 3H); 2.06 (m, 1H), 2.22 (m, 






1H); 3.17 (dd, 1H); 3.81-3.99 (m, 5H); 5.38 






(m, 1H); 6.89 (t, 1H); 7.17 (d, 2H).


2.6.482
3,5-diluorophenyl
ethyl
(cyclohex-2-en-1-one)-3-yl



2.6.483
3,5-diluorophenyl
ethyl
(propan-1-ol)-3-yl



2.6.484
3,5-diluorophenyl
ethyl
(2,2-dimethylpropan-1-ol)-3-yl



2.6.485
3,5-diluorophenyl
ethyl
(methyl 2,2-dimethyl 






propanoate)-3-yl



2.6.486
3,5-diluorophenyl
ethyl
(methyl propanoate)-3-yl
[CDCl3] 0.99 (t, 3H); 2.01-2.07 (m, 2H); 2.72 






(t, 2H), 3.17 (d, 1H); 3.68 (s, 3H); 3.75 (d, 






1H); 4.41-4.53 (m, 2H); 6.86 (t, 1H); 7.18 (d, 






2H).


2.6.487
3,5-diluorophenyl
ethyl
(ethyl propanoate)-3-yl



2.6.488
3,5-diluorophenyl
ethyl
(ethyl butanoate)-3-yl
[CDCl3] D1 0.98 (t, 3H); 1.27 (t, 3H); 1.36 






(d, 3H); 1.95-2.12 (m, 2H); 2.51-2.73 (m, 






2H); 3.14 (d, 1H); 3.78 (d, 1H); 4.07-4.18 






(m, 2H); 5.32-5.43 (m, 1H); 6.86 (t, 1H); 






7.13-7.22 (m, 2H). D2 1.00 (t, 3H); 1.22 (t, 






3H); 1.35 (d, 3H); 1.95-2.12 (m, 2H); 






2.51-2.73 (m, 2H); 3.17 (d, 1H); 3.72 (d, 






1H); 4.00-4.07(m, 2H); 5.32-5.43 (m, 1H); 






6.86 (t, 1H); 7.13-7.22 (m, 2H).


2.6.489
3,5-difluorophenyl
ethyl
(ethyl (3R)-4,4,4-
[CDCl3] D1 1.01 (t, 3H); 1.19 (t, 3H); 





trifluorobutanoate)-3-yl one 
2.05-2.11 (m, 2H); 2.81-2.91 (m, 2H); 3.21 





diastereomer
(d, 1H); 3.77 (d, 1H); 4.04-4.11 (m, 2H); 






5.84 (m, 1H); 6.87 (t, 1H); 7.17 (d, 2H).


2.6.490
3,5-difluorophenyl
ethyl
(ethyl (3R)-4,4,4-
[CDCl3] 1.01 (t, 3H); 1.24 (t, 3H); 2.01-2.13 





trifluorobutanoate)-3-yl the 
(m, 2H); 2.85 (d, 2H); 3.23 (d, 1H); 3.72 (d, 





other diastereomer
1H); 4.13 (q, 2H); 5.83 (m, 1H); 6.87 (t, 1H); 






7.16 (d, 2H).


2.6.491
3,5-difluorophenyl
ethyl
(butan-2-one)-4-yl



2.6.492
3,5-difluorophenyl
ethyl
(3-methylbutan-2-one)-4-yl



2.6.493
3,5-difluorophenyl
ethyl
(pent-3-en-2-one)-4-yl



2.6.494
3,5-difluorophenyl
ethyl
((2S)-dimethyl butanedioate)-
[CDCl3] D1 1.02-1.07 (m, 3H), 2.02-2.15 (m, 





2-yl
2H); 2.95 (m, 2H); 3.21 (d, 1H); 3.69 (s, 3H), 






3.75 (s, 3H), 3.79 (d, 1H), 5.58 (t, 1H); 6.87 






(t, 1H); 7.19 (d, 2H). D2 1.02-1.07 (m, 3H); 






2.02-2.15 (m, 2H); 2.95 (m, 2H); 3.22 (d, 






1H); 3.68 (s, 3H); 3.77 (s, 3H), 3.81 (d, 1H); 






5.58 (t, 1H); 6.87 (t, 1H); 7.19 (d, 2H).


2.6.495
3,5-difluorophenyl
ethyl
(dimethyl pentanedioate)-3-yl
[CDCl3] 0.99 (t, 3H); 1.97-2.06 (m, 2H); 2.75 






(m, 4H); 3.16 (d, 1H); 3.62 (s, 3H); 3.67 (s, 






3H); 3.75 (d, 1H); 5.60 (quin, 1H); 6.86 (t, 






1H); 7.19 (d, 2H).


2.6.496
3,5-difluorophenyl
ethyl
(methyl (2R)-2-methyl 






propanoate)-3-yl



2.6.497
3,5-difluorophenyl
ethyl
4-methoxycarbonylbenzyl



2.6.498
3,5-difluorophenyl
ethyl
3,5-difluorobenzyl



2.6.499
3,5-difluorophenyl
ethyl
3,4-difluorobenzyl



2.6.500
3,5-difluorophenyl
ethyl
2,6-difluorobenzyl



2.6.501
3,5-difluorophenyl
ethyl
(5-methylpyridin-3-yl)-methyl



2.6.502
3,5-difluorophenyl
ethyl
(tetrahydrofuran)-3-yl



2.6.503
(S)-3,5-difluorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.504
(R)-3,5-difluorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.505
3-chloro-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.506
3-bromo-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.507
3-iodo-5-fluorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.508
3-methyl-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.509
3-ethyl-5-fluorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.510
3-propyl-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.511
3-i-propyl-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.512
3-n-butyl-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.513
3-isobutyl-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.514
3-tert-butyl-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.515
3-cyclopropyl-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.516
3-vinyl-5-fluorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.517
3-ethynyl-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.518
3-cyano-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.519
3-trifluoromethyl-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.520
3-(methoxy-carbonyl)-
methyl
(ethyl butanoate)-3-yl




5-fluorophenyl





2.6.521
3-hydroxymethyl-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.522
3-carbamoyl-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.523
3-hydroxy-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.524
3-methoxy-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.525
3-ethoxy-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.526
3-n-propoxy-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.527
3-isopropoxy-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.528
3-n-butoxy-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.529
3-isobutoxy-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.530
3-tert-butoxy-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.531
3-difluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.532
3-trifluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.533
3-(2,2,2-trifluoro-
methyl
(ethyl butanoate)-3-yl




ethoxy)-5-fluorophenyl





2.6.534
3-(2-chloro-ethoxy)-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.535
3-(2-hydroxy-ethoxy)-
methyl
(ethyl butanoate)-3-yl




5-fluorophenyl





2.6.536
3-[(tert-butoxy-
methyl
(ethyl butanoate)-3-yl




carbonyl)oxy]-5-






fluorophenyl





2.6.537
3-nitro-5-fluorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.538
3-acetoxy-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.539
{3-[(tert-butoxy-
methyl
(ethyl butanoate)-3-yl




carbonyl)amino]-5-






fluorophenyl}





2.6.540
3-methylsulfanyl-5-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.541
3,5-dichlorophenyl
methyl
(cyclohex-2-en-1-one)-3-yl
[CDCl3] 1.79 (s, 3H); 2.08 (quin, 2H); 2.43 






(t, 2H), 2.58 (t, 2H); 3.22 (d, 1H); 3.88 (d, 






1H); 5.97 (s, 1H); 7.42 (s, 1H); 7.53 (s, 2H).


2.6.542
3,5-dichlorophenyl
methyl
(propan-1-ol)-3-yl



2.6.543
3,5-dichlorophenyl
methyl
(2,2-dimethylpropan-1-ol)-3-yl



2.6.544
3,5-dichlorophenyl
methyl
(methyl 2,2-dimethyl 






propanoate)-3-yl



2.6.545
3,5-dichlorophenyl
methyl
(methyl propanoate)-3-yl
[CDCl3] 1.71 (s, 3H); 2.72 (t, 2H); 3.15 (d, 






1H); 3.68 (s, 3H); 3.83 (d, 1H); 4.46 (t, 2H); 






7.40 (s, 1H); 7.53 (s, 2H).


2.6.546
3,5-dichlorophenyl
methyl
(ethyl propanoate)-3-yl
[CDCl3] 1.23 (t, 3H), 1.70 (s, 3H); 2.70 (t, 






2H); 3.15 (d, 1H); 3.82 (d, 1H); 4.12 (q, 2H), 






4.47 (t, 2H); 7.40 (s, 1H); 7.52 (s, 2H).


2.6.547
3,5-dichlorophenyl
methyl
(ethyl butanoate)-3-yl
[CDCl3] 1.18-1.27 (m, 3H); 1.36 (d, 3H); 






1.68 (d, 3H); 2.55 (m, 1H); 2.67 (m, 1H); 






3.12 (dd, 1H); 3.81 (dd, 1H), 4.03-4.16 (m, 






2H); 5.36 (m, 1H); 7.39 (s, 1H); 7.53 (s, 2H).


2.6.548
3,5-dichlorophenyl
methyl
(ethyl (3R)-4,4,4-
[CDCl3] (t, 3H); 1.75 (s, 3H); 2.85 (m, 2H); 





trifluorobutanoate)-3-yl (1 
3.19 (d, 1H); 3.84 (d, 1H); 4.09 (m, 2H); 5.81 





diastereomer)
(m, 1H); 7.41 (s, 1H); 7.52 (s, 2H). 6-1-1


2.6.549
3,5-dichlorophenyl
methyl
(ethyl (3R)-4,4,4-
[CDCl3] 1.25 (t, 3H); 1.74 (s, 3H); 2.86 (d, 





trifluorobutanoate)-3-yl (the 
2H); 3.20 (d, 1H); 3.80 (d, 1H); 4.16 (q, 2H); 





other diastereomer)
5.81 (m, 1H); 7.41 (s, 1H); 7.53 (s, 2H).


2.6.550
3,5-dichlorophenyl
methyl
(butan-1-ol)-4-yl
[CDCl3] 1.58 (bs, 1H); 1.65 (m, 2H); 1.72 (s, 






3H); 1.80 (mc, 2H); 3.13 (d, 1H); 3.68 (t, 






2H); 3.82 (d, 1H); 4.25 (t, 2H); 7.40 (d, 1H); 






7.52 (s, 2d).


2.6.551
3,5-dichlorophenyl
methyl
(3-methylbutan-2-one)-4-yl



2.6.552
3,5-dichlorophenyl
methyl
(pent-3-en-2-one)-4-yl (E or Z)
[CDCl3] 1.79 (s, 3H); 2.21 (s, 3H); 2.33 (s, 






3H); 3.21 (d, 1H); 3.89 (d, 1H); 6.11 (s, 1H); 






7.41 (s, 1H); 7.55 (s, 2H).


2.6.553
3,5-dichlorophenyl
methyl
(pent-3-en-2-one)-4-yl (Z or E)
[CDCl3] 1.80 (s, 3H); 2.10 (s, 6H); 3.22 (d, 






1H); 4.20 (d, 1H); 5.96 (s, 1H); 7.40 (s, 1H); 






7.58 (s, 2H).


2.6.554
3,5-dichlorophenyl
methyl
((2S)-dimethyl butanedioate)-
[CDCl3] 1.75 (d, 3H); 2.96 (m, 2H); 3.20 (dd, 





2-yl
1H); 3.68 (d, 3H); 3.77 (d, 3H); 3.90 (dd, 






1H); 5.57 (t, 1H); 7.41 (s, 1H); 7.53 (s, 2H).


2.6.555
3,5-dichlorophenyl
methyl
(dimethyl pentanedioate)-3-yl
[CDCl3] 1.68 (s, 3H); 2.75 (t, 4H); 3.11 (d, 






1H); 3.62 (s, 3H); 3.69 (s, 3H); 3.81 (d, 1H); 






5.58 (quin, 1H); 7.41 (s, 1H), 7.53 (s, 2H).


2.6.556
3,5-dichlorophenyl
methyl
(methyl (2R)-2-methyl 






propanoate)-3-yl



2.6.557
3,5-dichlorophenyl
methyl
4-methoxycarbonylbenzyl



2.6.558
3,5-dichlorophenyl
methyl
3,5-difluorobenzyl



2.6.559
3,5-dichlorophenyl
methyl
3,4-difluorobenzyl



2.6.560
3,5-dichlorophenyl
methyl
2,6-difluorobenzyl



2.6.561
3,5-dichlorophenyl
methyl
(5-methylpyridin-3-yl)methyl
[CDCl3] 1.72 (s, 3H); 2.34 (s, 3H); 3.17 (d, 






1H); 3.82 (d, 1H); 5.22 (d, 2H); 7.41 (s, 1H); 






7.51 (m, 3H); 8.43 (s, 2H).


2.6.562
3,5-dichlorophenyl
methyl
(tetrahydrofuran)-3-yl



2.6.563
3,5-dichlorophenyl
ethyl
(cyclohex-2-en-1-one)-3-yl



2.6.564
3,5-dichlorophenyl
ethyl
(propan-1-ol)-3-yl



2.6.565
3,5-dichlorophenyl
ethyl
(2,2-dimethylpropan-1-ol)-3-yl



2.6.566
3,5-dichlorophenyl
ethyl
(methyl 2,2-dimethyl 






propanoate)-3-yl



2.6.567
3,5-dichlorophenyl
ethyl
(methyl propanoate)-3-yl



2.6.568
3,5-dichlorophenyl
ethyl
(ethyl propanoate)-3-yl



2.6.569
3,5-dichlorophenyl
ethyl
(ethyl butanoate)-3-yl



2.6.570
3,5-dichlorophenyl
ethyl
(ethyl (3R)-4,4,4-






trifluorobutanoate)-3-yl



2.6.571
3,5-dichlorophenyl
ethyl
(butan-2-one)-4-yl



2.6.572
3,5-dichlorophenyl
ethyl
(3-methylbutan-2-one)-4-yl



2.6.573
3,5-dichlorophenyl
ethyl
(pent-3-en-2-one)-4-yl



2.6.574
3,5-dichlorophenyl
ethyl
((2S)-dimethyl butanedioate)-






2-yl



2.6.575
3,5-dichlorophenyl
ethyl
(dimethyl pentanedioate)-3-yl



2.6.576
3,5-dichlorophenyl
ethyl
(methyl (2R)-2-methyl 






propanoate)-3-yl



2.6.577
3,5-dichlorophenyl
ethyl
4-methoxycarbonylbenzyl



2.6.578
3,5-dichlorophenyl
ethyl
3,5-difluorobenzyl



2.6.579
3,5-dichlorophenyl
ethyl
3,4-difluorobenzyl



2.6.580
3,5-dichlorophenyl
ethyl
2,6-difluorobenzyl



2.6.581
3,5-dichlorophenyl
ethyl
(5-methylpyridin-3-yl)methyl



2.6.582
3,5-dichlorophenyl
ethyl
(tetrahydrofuran)-3-yl



2.6.583
(S)-3,5-dichlorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.584
(R)-3,5-dichlorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.585
3-bromo-5-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.586
3-iodo-5-chlorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.587
3-methyl-5-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.588
3-ethyl-5-chlorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.589
3-propyl-5-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.590
3-isopropyl-5-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.591
3-n-butyl-5-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.592
3-isobutyl-5-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.593
3-tert-butyl-5-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.594
3-cyclopropyl-5-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.595
3-cyano-5-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.596
3-trifluoromethyl-5-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.597
3-trifluoromethyl-5-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.598
3-(hydroxy-carbonyl)-
methyl
(ethyl butanoate)-3-yl




5-chlorophenyl





2.6.599
3-(methoxy-carbonyl)-
methyl
(ethyl butanoate)-3-yl




5-chlorophenyl





2.6.600
3-methoxy-5-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.601
3-ethoxy-5-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.602
3-n-propoxy-5-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.603
3-isopropoxy-5-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.604
3-n-butoxy-5-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.605
3-isobutoxy-5-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.606
3-difluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.607
3-trifluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.608
3-nitro-5-chlorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.609
3-acetoxy-5-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.610
3-methylsulfanyl-5-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.611
3,5-dibromophenyl
methyl
(ethyl butanoate)-3-yl



2.6.612
3-iodo-5-bromophenyl
methyl
(ethyl butanoate)-3-yl



2.6.613
3-methyl-5-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.614
3-ethyl-5-bromophenyl
methyl
(ethyl butanoate)-3-yl



2.6.615
3-propyl-5-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.616
3-isopropyl-5-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.617
3-n-butyl-5-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.618
3-isobutyl-5-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.619
3-tert-butyl-5-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.620
3-cyclopropyl-5-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.621
3-cyano-5-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.622
3-trifluoromethyl-5-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.623
3-(hydroxy-carbonyl)-
methyl
(ethyl butanoate)-3-yl




5-bromophenyl





2.6.624
3-(methoxy-carbonyl)-
methyl
(ethyl butanoate)-3-yl




5-bromophenyl





2.6.625
3-methoxy-5-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.626
3-ethoxy-5-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.627
3-n-propoxy-5-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.628
3-isopropoxy-5-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.629
3-n-butoxy-5-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.630
3-isobutoxy-5-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.631
3-difluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.632
3-trifluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.633
3-nitro-5-bromophenyl
methyl
(ethyl butanoate)-3-yl



2.6.634
3-acetoxy-5-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.635
3-methylsulfanyl-5-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.636
3,5-diiodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.637
3-methyl-5-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.638
3-ethyl-5-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.639
3-propyl-5-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.640
3-isopropyl-5-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.641
3-n-butyl-5-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.642
3-isobutyl-5-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.643
3-tert-butyl-5-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.644
3-cyclopropyl-5-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.645
3-cyano-5-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.646
3-trifluoromethyl-5-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.647
3-(hydroxy-carbonyl)-
methyl
(ethyl butanoate)-3-yl




5-iodophenyl





2.6.648
3-(methoxy-carbonyl)-
methyl
(ethyl butanoate)-3-yl




5-iodophenyl





2.6.649
3-methoxy-5-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.650
3-ethoxy-5-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.651
3-n-propoxy-5-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.652
3-isopropoxy-5-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.653
3-n-butoxy-5-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.654
3-isobutoxy-5-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.655
3-difluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.656
3-trifluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.657
3-nitro-5-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.658
3-acetoxy-5-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.659
3-methylsulfanyl-5-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.660
3,5-dimethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.661
3-ethyl-5-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.662
3-propyl-5-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.663
3-isopropyl-5-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.664
3-n-butyl-5-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.665
3-isobutyl-5-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.666
3-tert-butyl-5-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.667
3-cyclopropyl-5-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.668
3-cyano-5-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.669
3-trifluoromethyl-5-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.670
3-(hydroxy-carbonyl)-
methyl
(ethyl butanoate)-3-yl




5-methylphenyl





2.6.671
3-(methoxy-carbonyl)-
methyl
(ethyl butanoate)-3-yl




5-methylphenyl





2.6.672
3-methoxy-5-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.673
3-ethoxy-5-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.674
3-propoxy-5-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.675
3-butoxy-5-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.676
3-isobutoxy-5-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.677
3-difluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.678
3-trifluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.679
3-nitro-5-methylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.680
3-acetoxy-5-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.681
3-methylsulfanyl-5-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.682
3,5-diethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.683
3-propyl-5-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.684
3-isopropyl-5-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.685
3-n-butyl-5-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.686
3-isobutyl-5-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.687
3-tert-butyl-5-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.688
3-cyclopropyl-5-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.689
3-cyano-5-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.690
3-trifluoromethyl-5-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.691
3-(hydroxy-carbonyl)-
methyl
(ethyl butanoate)-3-yl




5-ethylphenyl





2.6.692
3-(methoxy-carbonyl)-
methyl
(ethyl butanoate)-3-yl




5-ethylphenyl





2.6.693
3-methoxy-5-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.694
3-ethoxy-5-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.695
3-n-propoxy-5-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.696
3-n-butoxy-5-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.697
3-isobutoxy-5-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.698
3-difluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.699
3-trifluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.700
3-nitro-5-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.701
3-acetoxy-5-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.702
3-methylsulfanyl-5-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.703
3,5-dipropylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.704
3-isopropyl-5-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.705
3-n-butyl-5-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.706
3-isobutyl-5-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.707
3-tert-butyl-5-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.708
3-cyclopropyl-5-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.709
3-cyano-5-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.710
3-trifluoromethyl-5-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.711
3-(hydroxy-carbonyl)-
methyl
(ethyl butanoate)-3-yl




5-propylphenyl





2.6.712
3-(methoxy-carbonyl)-
methyl
(ethyl butanoate)-3-yl




5-propylphenyl





2.6.713
3-methoxy-5-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.714
3-ethoxy-5-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.715
3-n-propoxy-5-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.716
3-isobutoxy-5-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.717
3-difluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.718
3-trifluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.719
3-nitro-5-propylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.720
3-acetoxy-5-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.721
3-methylsulfanyl-5-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.722
3,5-diisopropylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.723
3-n-butyl-5-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.724
3-isobutyl-5-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.725
3-tert-butyl-5-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.726
3-cyclopropyl-5-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.727
3-cyano-5-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.728
3-trifluoromethyl-5-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.729
3-(hydroxy-carbonyl)-
methyl
(ethyl butanoate)-3-yl




5-isopropylphenyl





2.6.730
3-(methoxy-carbonyl)-
methyl
(ethyl butanoate)-3-yl




5-isopropylphenyl





2.6.731
3-methoxy-5-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.732
3-ethoxy-5-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.733
3-n-propoxy-5-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.734
3-isobutoxy-5-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.735
3-difluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.736
3-trifluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.737
3-nitro-5-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.738
3-acetoxy-5-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.739
3-methylsulfanyl-5-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.740
3,5-diisobutylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.741
3-tert-butyl-5-
methyl
(ethyl butanoate)-3-yl




isobutylphenyl





2.6.742
3-cyclopropyl-5-
methyl
(ethyl butanoate)-3-yl




isobutylphenyl





2.6.743
3-cyano-5-
methyl
(ethyl butanoate)-3-yl




isobutylphenyl





2.6.744
3-trifluoromethyl-5-
methyl
(ethyl butanoate)-3-yl




isobutylphenyl





2.6.745
3-(methoxy-carbonyl)-
methyl
(ethyl butanoate)-3-yl




5-isobutylphenyl





2.6.746
3-methoxy-5-
methyl
(ethyl butanoate)-3-yl




isobutylphenyl





2.6.747
3-ethoxy-5-
methyl
(ethyl butanoate)-3-yl




isobutylphenyl





2.6.748
3-n-propoxy-5-
methyl
(ethyl butanoate)-3-yl




isobutylphenyl





2.6.749
3-isobutoxy-5-
methyl
(ethyl butanoate)-3-yl




isobutylphenyl





2.6.750
3-difluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




isobutylphenyl





2.6.751
3-trifluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




isobutylphenyl





2.6.752
3-nitro-5-
methyl
(ethyl butanoate)-3-yl




isobutylphenyl





2.6.753
3-acetoxy-5-
methyl
(ethyl butanoate)-3-yl




isobutylphenyl





2.6.754
3-methylsulfanyl-5-
methyl
(ethyl butanoate)-3-yl




isobutylphenyl





2.6.755
3,5-di-tert-butylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.756
3-cyclopropyl-5-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.757
3-cyano-5-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.758
3-trifluoromethyl-5-
methyl
(ethyl butanoate)-3-yl




tert-butylphenyl





2.6.759
3-(hydroxy-carbonyl)-
methyl
(ethyl butanoate)-3-yl




5-tert-butylphenyl





2.6.760
3-(methoxy-carbonyl)-
methyl
(ethyl butanoate)-3-yl




5-tert-butylphenyl





2.6.761
3-methoxy-5-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.762
3-ethoxy-5-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.763
3-n-propoxy-5-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.764
3-isobutoxy-5-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.765
3-difluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




tert-butylphenyl





2.6.766
3-trifluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




tert-butylphenyl





2.6.767
3-nitro-5-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.768
3-acetoxy-5-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.769
3-methylsulfanyl-5-
methyl
(ethyl butanoate)-3-yl




tert-butylphenyl





2.6.770
3-tert-butyl-5-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.771
3,5-dicyclopropyl-
methyl
(ethyl butanoate)-3-yl




phenyl





2.6.772
3-cyano-5-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.773
3-trifluoromethyl-5-
methyl
(ethyl butanoate)-3-yl




cyclopropyl-phenyl





2.6.774
3-(hydroxy-carbonyl)-
methyl
(ethyl butanoate)-3-yl




5-cyclopropylphenyl





2.6.775
3-(methoxy-carbonyl)-
methyl
(ethyl butanoate)-3-yl




5-cyclopropylphenyl





2.6.776
3-methoxy-5-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.777
3-ethoxy-5-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.778
3-n-propoxy-5-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.779
3-isobutoxy-5-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.780
3-difluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.781
3-trifluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.782
3-nitro-5-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.783
3-acetoxy-5-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.784
3-methylsulfanyl-5-
methyl
(ethyl butanoate)-3-yl




cyclopropyl-phenyl





2.6.785
3,5-dicyanophenyl
methyl
(ethyl butanoate)-3-yl



2.6.786
3-trifluoromethyl-5-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.787
3-(methoxy-carbonyl)-
methyl
(ethyl butanoate)-3-yl




5-cyanophenyl





2.6.788
3-methoxy-5-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.789
3-ethoxy-5-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.790
3-n-propoxy-5-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.791
3-n-butoxy-5-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.792
3-isobutoxy-5-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.793
3-difluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.794
3-trifluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.795
3-nitro-5-cyanophenyl
methyl
(ethyl butanoate)-3-yl



2.6.796
3-acetoxy-5-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.797
3-methylsulfanyl-5-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.798
3,5-di(trifluoro-
methyl
(ethyl butanoate)-3-yl




methyl)-phenyl





2.6.799
3-(hydroxy-carbonyl)-
methyl
(ethyl butanoate)-3-yl




5-trifluoromethyl-






phenyl





2.6.800
3-(methoxy-carbonyl)-
methyl
(ethyl butanoate)-3-yl




5-trifluoromethyl-






phenyl





2.6.801
3-methoxy-5-
methyl
(ethyl butanoate)-3-yl




trifluoromethyl-phenyl





2.6.802
3-ethoxy-5-
methyl
(ethyl butanoate)-3-yl




trifluoromethyl-phenyl





2.6.803
3-n-propoxy-5-
methyl
(ethyl butanoate)-3-yl




trifluoromethyl-phenyl





2.6.804
3-isobutoxy-5-
methyl
(ethyl butanoate)-3-yl




trifluoromethyl-phenyl





2.6.805
3-difluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




trifluoromethyl-phenyl





2.6.806
3-trifluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




trifluoromethyl-phenyl





2.6.807
3-nitro-5-
methyl
(ethyl butanoate)-3-yl




trifluoromethyl-phenyl





2.6.808
3-acetoxy-5-
methyl
(ethyl butanoate)-3-yl




trifluoromethyl-phenyl





2.6.809
3-methylsulfanyl-5-
methyl
(ethyl butanoate)-3-yl




trifluoromethyl-phenyl





2.6.810
3,5-di(methoxy-
methyl
(ethyl butanoate)-3-yl




carbonyl)phenyl





2.6.811
3-methoxy-5-
methyl
(ethyl butanoate)-3-yl




(methoxycarbonyl)-






phenyl





2.6.812
3-ethoxy-5-
methyl
(ethyl butanoate)-3-yl




(methoxycarbonyl)-






phenyl





2.6.813
3-n-propoxy-5-
methyl
(ethyl butanoate)-3-yl




(methoxycarbonyl)-






phenyl





2.6.814
3-isobutoxy-5-
methyl
(ethyl butanoate)-3-yl




(methoxycarbonyl)-






phenyl





2.6.815
3-difluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




(methoxy-






carbonyl)phenyl





2.6.816
3-trifluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




(methoxy-






carbonyl)phenyl





2.6.817
3-nitro-5-(methoxy-
methyl
(ethyl butanoate)-3-yl




carbonyl)phenyl





2.6.818
3-acetoxy-5-(methoxy-
methyl
(ethyl butanoate)-3-yl




carbonyl)phenyl





2.6.819
3-methylsulfanyl-5-
methyl
(ethyl butanoate)-3-yl




(methoxy-






carbonyl)phenyl





2.6.820
3,5-dimethoxyphenyl
methyl
(ethyl butanoate)-3-yl



2.6.821
3-ethoxy-5-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.822
3-n-propoxy-5-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.823
3-isobutoxy-5-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.824
3-difluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.825
3-trifluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.826
3-nitro-5-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.827
3-acetoxy-5-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.828
3-methylsulfanyl-5-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.829
3,5-diethoxyphenyl
methyl
(ethyl butanoate)-3-yl



2.6.830
3-n-propoxy-5-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.831
3-isobutoxy-5-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.832
3-difluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.833
3-trifluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.834
3-nitro-5-ethoxyphenyl
methyl
(ethyl butanoate)-3-yl



2.6.835
3-acetoxy-5-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.836
3-methylsulfanyl-5-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.837
3,5-di(isopropoxy)-
methyl
(ethyl butanoate)-3-yl




phenyl





2.6.838
3-n-butoxy-5-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.839
3-isobutoxy-5-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.840
3-difluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.841
3-trifluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.842
3-nitro-5-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.843
3-acetoxy-5-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.844
3-methylsulfanyl-5-
methyl
(ethyl butanoate)-3-yl




isopropoxy-phenyl





2.6.845
3,5-di(trifluoro-
methyl
(ethyl butanoate)-3-yl




methoxy)phenyl





2.6.846
3-nitro-5-trifluoro-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.847
3-methylsulfanyl-5-
methyl
(ethyl butanoate)-3-yl




trifluoro-methoxy-






phenyl





2.6.848
3,5-bis(difluoro-
methyl
(ethyl butanoate)-3-yl




methoxy)phenyl





2.6.849
3-trifluoro-methoxy-5-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.850
3-nitro-5-difluoro-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.851
3-acetoxy-5-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.852
3-methylsulfanyl-5-
methyl
(ethyl butanoate)-3-yl




difluoro-






methoxyphenyl





2.6.853
3,5-bis(acetoxy)-
methyl
(ethyl butanoate)-3-yl




phenyl





2.6.854
3-methylsulfanyl-5-
methyl
(ethyl butanoate)-3-yl




acetoxyphenyl





2.6.855
3,5-dinitrophenyl
methyl
(ethyl butanoate)-3-yl



2.6.856
3-acetoxy-5-
methyl
(ethyl butanoate)-3-yl




nitrophenyl





2.6.857
3-methylsulfanyl-5-
methyl
(ethyl butanoate)-3-yl




nitrophenyl





2.6.858
3,5-di(methyl-
methyl
(ethyl butanoate)-3-yl




sulfanyl)phenyl





2.6.859
3,4-difluorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.860
3-chloro-4-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.861
3-bromo-4-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.862
3-methyl-4-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.863
3-ethyl-4-fluorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.864
3-cyclopropyl-4-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.865
3-cyano-4-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.866
3-methoxy-4-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.867
3-ethoxy-4-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.868
3-trifluoro-methoxy-4-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.869
3-nitro-4-fluorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.870
3-fluoro-4-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.871
3,4-dichlorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.872
3-bromo-4-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.873
3-methyl-4-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.874
3-cyclopropyl-4-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.875
3-cyano-4-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.876
3-trifluoromethyl-4-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.877
3-methoxy-4-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.878
3-ethoxy-4-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.879
3-trifluoro-methoxy-4-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.880
3-nitro-4-chlorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.881
3-fluoro-4-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.882
3-chloro-4-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.883
3,4-dibromophenyl
methyl
(ethyl butanoate)-3-yl



2.6.884
3-methyl-4-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.885
3-ethyl-4-bromophenyl
methyl
(ethyl butanoate)-3-yl



2.6.886
3-cyclopropyl-4-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.887
3-cyano-4-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.888
3-trifluoromethyl-4-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.889
3-methoxy-4-phenyl
methyl
(ethyl butanoate)-3-yl



2.6.890
3-ethoxy-4-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.891
3-trifluoro-methoxy-4-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.892
3-nitro-4-bromophenyl
methyl
(ethyl butanoate)-3-yl



2.6.893
3-fluoro-4-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.894
3-chloro-4-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.895
3-bromo-4-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.896
3-methyl-4-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.897
3-cyclopropyl-4-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.898
3-cyano-4-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.899
3-trifluoromethyl-4-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.900
3-methoxy-4-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.901
3-ethoxy-4-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.902
3-trifluoro-methoxy-4-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.903
3-nitro-4-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.904
3-fluoro-4-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.905
3-chloro-4-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.906
3-bromo-4-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.907
3,4-dimethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.908
3,4-dimethylphenyl
ethyl
(ethyl butanoate)-3-yl



2.6.909
3,4-dimethylphenyl
isopropyl
(ethyl butanoate)-3-yl



2.6.910
3,4-dimethylphenyl
cyclo-
(ethyl butanoate)-3-yl





propyl




2.6.911
3-ethyl-4-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.912
3-cyclopropyl-4-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.913
3-cyano-4-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.914
3-trifluoromethyl-4-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.915
3-methoxy-4-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.916
3-ethoxy-4-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.917
3-trifluoro-methoxy-4-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.918
3-nitro-4-methylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.919
3-fluoro-4-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.920
3-chloro-4-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.921
3-bromo-4-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.922
3-methyl-4-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.923
3,4-diethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.924
3-cyclopropyl-4-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.925
3-cyano-4-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.926
3-trifluoromethyl-4-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.927
3-methoxy-4-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.928
3-ethoxy-4-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.929
3-trifluoro-methoxy-4-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.930
3-nitro-4-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.931
3-fluoro-4-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.932
3-chloro-4-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.933
3-bromo-4-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.934
3-methyl-4-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.935
3-methyl-4-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.936
3-cyclopropyl-4-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.937
3-cyano-4-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.938
3-trifluoromethyl-4-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.939
3-methoxy-4-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.940
3-ethoxy-4-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.941
3-trifluoro-methoxy-4-
methyl
(ethyl butanoate)-3-yl




propylphenyl





2.6.942
3-nitro-4-propylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.943
3-fluoro-4-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.944
3-chloro-4-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.945
3-bromo-4-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.946
3-methyl-4-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.947
3-cyclopropyl-4-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.948
3-cyano-4-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.949
3-trifluoromethyl-4-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.950
3-methoxy-4-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.951
3-thoxy-4-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.952
3-trifluoro-methoxy-4-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.953
3-nitro-4-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.954
3-fluoro-4-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.955
3-chloro-4-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.956
3-bromo-4-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.957
3-methyl-4-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.958
3-cyclopropyl-4-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.959
3-cyano-4-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.960
3-trifluoromethyl-4-
methyl
(ethyl butanoate)-3-yl




tert-butylphenyl





2.6.961
3-methoxy-4-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.962
3-ethoxy-4-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.963
3-trifluoro-methoxy-4-
methyl
(ethyl butanoate)-3-yl




tert-butylphenyl





2.6.964
3-nitro-4-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.965
3-fluoro-4-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.966
3-chloro-4-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.967
3-bromo-4-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.968
3-methyl-4-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.969
3,4-dicyclopropyl-
methyl
(ethyl butanoate)-3-yl




phenyl





2.6.970
3-cyano-4-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.971
3-trifluoromethyl-4-
methyl
(ethyl butanoate)-3-yl




cyclopropyl-phenyl





2.6.972
3-methoxy-4-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.973
3-ethoxy-4-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.974
3-trifluoro-methoxy-4-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.975
3-fluoro-4-
methyl
(ethyl butanoate)-3-yl




methoxycarbonyl-






phenyl





2.6.976
3-chloro-4-methoxy-
methyl
(ethyl butanoate)-3-yl




carbonylphenyl





2.6.977
3-bromo-4-methoxy-
methyl
(ethyl butanoate)-3-yl




carbonylphenyl





2.6.978
3-methyl-4-methoxy-
methyl
(ethyl butanoate)-3-yl




carbonylphenyl





2.6.979
3-cyclopropyl-4-
methyl
(ethyl butanoate)-3-yl




methoxycarbonyl-






phenyl





2.6.980
3-cyano-4-methoxy-
methyl
(ethyl butanoate)-3-yl




carbonylphenyl





2.6.981
3-trifluoromethyl-4-
methyl
(ethyl butanoate)-3-yl




methoxy-






carbonylphenyl





2.6.982
3-methoxy-4-
methyl
(ethyl butanoate)-3-yl




methoxycarbonyl-






phenyl





2.6.983
3-ethoxy-4-
methyl
(ethyl butanoate)-3-yl




methoxycarbonyl-






phenyl





2.6.984
3-trifluoro-
methyl
(ethyl butanoate)-3-yl




methoxycarbonyl-






phenyl





2.6.985
3-nitro-4-methoxy-
methyl
(ethyl butanoate)-3-yl




carbonylphenyl





2.6.986
3-fluoro-4-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.987
3-chloro-4-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.988
3-bromo-4-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.989
3-methyl-4-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.990
3-cyclopropyl-4-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.991
3-cyano-4-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.992
3-trifluoromethyl-4-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.993
3-methoxy-4-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.994
3-ethoxy-4-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.995
3-trifluoro-methoxy-4-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.996
3-nitro-4-cyanophenyl
methyl
(ethyl butanoate)-3-yl



2.6.997
3-fluoro-4-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.998
3-chloro-4-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.999
3-bromo-4-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1000
3-methyl-4-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1001
3-cyclopropyl-4-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1002
3-cyano-4-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1003
3-trifluoromethyl-4-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1004
3,4-dimethoxyphenyl
methyl
(ethyl butanoate)-3-yl



2.6.1005
3-ethoxy-4-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1006
3-trifluoro-methoxy-4-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1007
3-nitro-4-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1008
3-fluoro-4-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.1009
3-chloro-4-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.1010
3-bromo-4-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.1011
3-methyl-4-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.1012
3-cyclopropyl-4-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.1013
3-cyano-4-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.1014
3-trifluoromethyl-4-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.1015
3-methoxy-4-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.1016
2,4-diethoxyphenyl
methyl
(ethyl butanoate)-3-yl



2.6.1017
3-trifluoro-methoxy-4-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.1018
3-nitro-4-ethoxyphenyl
methyl
(ethyl butanoate)-3-yl



2.6.1019
3-fluoro-4-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.1020
3-chloro-4-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.1021
3-bromo-4-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.1022
3-methyl-4-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.1023
3-cyclopropyl-4-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.1024
3-cyano-4-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.1025
3-trifluoromethyl-4-
methyl
(ethyl butanoate)-3-yl




isopropoxy-phenyl





2.6.1026
3-methoxy-4-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.1027
3-ethoxy-4-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.1028
3-trifluoro-methoxy-4-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.1029
3-nitro-4-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.1030
3-fluoro-4-trifluoro-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1031
3-chloro-4-trifluoro-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1032
3-bromo-4-trifluoro-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1033
3-methyl-4-trifluoro-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1034
3-cyclopropyl-4-
methyl
(ethyl butanoate)-3-yl




trifluoromethoxy-






phenyl





2.6.1035
3-cyano-4-trifluoro-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1036
3-trifluoromethyl-4-
methyl
(ethyl butanoate)-3-yl




trifluoro-






methoxyphenyl





2.6.1037
3-methoxy-4-
methyl
(ethyl butanoate)-3-yl




trifluoromethoxy-






phenyl





2.6.1038
3-ethoxy-4-trifluoro-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1039
3, 4-bis(trifluoro-
methyl
(ethyl butanoate)-3-yl




methoxy)phenyl





2.6.1040
3-nitro-4-trifluoro-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1041
3-fluoro-4-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.1042
3-chloro-4-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.1043
3-bromo-4-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.1044
3-methyl-4-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.1045
3-cyclopropyl-4-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.1046
3-cyano-4-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.1047
3-trifluoromethyl-4-
methyl
(ethyl butanoate)-3-yl




difluoro-






methoxyphenyl





2.6.1048
3-methoxy-4-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.1049
3-ethoxy-4-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.1050
3-trifluoro-methoxy-4-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.1051
3-nitro-4-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.1052
3-fluoro-4-nitrophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1053
3-chloro-4-nitrophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1054
3-bromo-4-nitrophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1055
3-methyl-4-nitrophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1056
3-ethyl-4-nitrophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1057
3-cyclopropyl-4-
methyl
(ethyl butanoate)-3-yl




nitrophenyl





2.6.1058
3-cyano-4-nitrophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1059
3-trifluoromethyl-4-
methyl
(ethyl butanoate)-3-yl




nitrophenyl





2.6.1060
3-methoxy-4-
methyl
(ethyl butanoate)-3-yl




nitrophenyl





2.6.1061
3-ethoxy-4-nitrophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1062
3-trifluoro-methoxy-4-
methyl
(ethyl butanoate)-3-yl




nitrophenyl





2.6.1063
3-fluoro-4-
methyl
(ethyl butanoate)-3-yl




methylsulfanylphenyl





2.6.1064
3-chloro-4-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.1065
3-bromo-4-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.1066
3-methyl-4-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.1067
3-cyclopropyl-4-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.1068
3-cyano-4-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.1069
3-trifluoromethyl-4-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.1070
3-methoxy-4-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.1071
3-ethoxy-4-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.1072
3-trifluoro-methoxy-4-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.1073
3-nitro-4-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.1074
3,6-difluorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1075
3-chloro-6-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.1076
3-bromo-6-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.1077
3-methyl-6-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.1078
3-ethyl-6-fluorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1079
3-cyclopropyl-6-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.1080
3-cyano-6-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.1081
3-methoxy-6-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.1082
3-ethoxy-6-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.1083
3-trifluoro-methoxy-6-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.1084
3-nitro-6-fluorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1085
3-fluoro-6-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.1086
3,6-dichlorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1087
3-bromo-6-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.1088
3-methyl-6-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.1089
3-cyclopropyl-6-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.1090
3-cyano-6-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.1091
3-trifluoromethyl-6-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.1092
3-methoxy-6-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.1093
3-ethoxy-6-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.1094
3-trifluoro-methoxy-6-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.1095
3-nitro-6-chlorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1096
3-fluoro-6-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.1097
3-chloro-6-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.1098
3,6-dibromophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1099
3-methyl-6-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.1100
3-ethyl-6-bromophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1101
3-cyclopropyl-6-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.1102
3-cyano-6-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.1103
3-trifluoromethyl-6-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.1104
3-methoxy-6-phenyl
methyl
(ethyl butanoate)-3-yl



2.6.1105
3-ethoxy-6-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.1106
3-trifluoro-methoxy-6-
methyl
(ethyl butanoate)-3-yl




bromophenyl





2.6.1107
3-nitro-6-bromophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1108
3-fluoro-6-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1109
3-chloro-6-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1110
3-bromo-6-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1111
3-methyl-6-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1112
3-cyclopropyl-6-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.1113
3-cyano-6-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1114
3-trifluoromethyl-6-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.1115
3-methoxy-6-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.1116
3-ethoxy-6-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1117
3-trifluoro-methoxy-6-
methyl
(ethyl butanoate)-3-yl




iodophenyl





2.6.1118
3-nitro-6-iodophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1119
3-fluoro-6-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.1120
3-chloro-6-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.1121
3-bromo-6-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.1122
3,6-dimethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.1123
3-cyclopropyl-6-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.1124
3-cyano-6-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.1125
3-trifluoromethyl-6-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.1126
3-methoxy-6-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.1127
3-ethoxy-6-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.1128
3-trifluoro-methoxy-6-
methyl
(ethyl butanoate)-3-yl




methylphenyl





2.6.1129
3-nitro-6-methylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.1130
3-fluoro-6-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.1131
3-chloro-6-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.1132
3-bromo-6-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.1133
3-methyl-6-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.1134
3,6-diethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.1135
3-cyclopropyl-6-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.1136
3-cyano-6-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.1137
3-trifluoromethyl-6-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.1138
3-methoxy-6-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.1139
3-ethoxy-6-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.1140
3-trifluoro-methoxy-6-
methyl
(ethyl butanoate)-3-yl




ethylphenyl





2.6.1141
3-nitro-6-ethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.1142
3-fluoro-6-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.1143
3-chloro-6-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.1144
3-bromo-6-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.1145
3-methyl-6-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.1146
3-ethyl-6-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.1147
3-cyclopropyl-6-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.1148
3-cyano-6-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.1149
3-trifluoromethyl-6-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.1150
3-methoxy-6-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.1151
3-thoxy-6-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.1152
3-trifluoro-methoxy-6-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.1153
3-nitro-6-
methyl
(ethyl butanoate)-3-yl




isopropylphenyl





2.6.1154
3-fluoro-6-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.1155
3-chloro-6-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.1156
3-bromo-6-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.1157
3-methyl-6-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.1158
3-cyclopropyl-6-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.1159
3-cyano-6-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.1160
3-trifluoromethyl-6-
methyl
(ethyl butanoate)-3-yl




tert-butylphenyl





2.6.1161
3-methoxy-6-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.1162
3-ethoxy-6-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.1163
3-trifluoro-methoxy-6-
methyl
(ethyl butanoate)-3-yl




tert-butylphenyl





2.6.1164
3-nitro-6-tert-
methyl
(ethyl butanoate)-3-yl




butylphenyl





2.6.1165
3-fluoro-6-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.1166
3-chloro-6-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.1167
3-bromo-6-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.1168
3-methyl-6-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.1169
3-cyano-6-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.1170
3-trifluoromethyl-6-
methyl
(ethyl butanoate)-3-yl




cyclopropyl-phenyl





2.6.1171
3-methoxy-6-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.1172
3-ethoxy-6-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.1173
3-trifluoro-methoxy-6-
methyl
(ethyl butanoate)-3-yl




cyclopropylphenyl





2.6.1174
3-fluoro-6-
methyl
(ethyl butanoate)-3-yl




methoxycarbonyl-






phenyl





2.6.1175
3-chloro-6-
methyl
(ethyl butanoate)-3-yl




methoxycarbonyl-






phenyl





2.6.1176
3-bromo-6-
methyl
(ethyl butanoate)-3-yl




methoxycarbonyl-






phenyl





2.6.1177
3-methyl-6-
methyl
(ethyl butanoate)-3-yl




methoxycarbonyl-






phenyl





2.6.1178
3-cyclopropyl-6-
methyl
(ethyl butanoate)-3-yl




methoxycarbonyl-






phenyl





2.6.1179
3-cyano-6-
methyl
(ethyl butanoate)-3-yl




methoxycarbonyl-






phenyl





2.6.1180
3-trifluoromethyl-6-
methyl
(ethyl butanoate)-3-yl




methoxy-






carbonylphenyl





2.6.1181
3-methoxy-6-
methyl
(ethyl butanoate)-3-yl




methoxycarbonyl-






phenyl





2.6.1182
3-ethoxy-6-
methyl
(ethyl butanoate)-3-yl




methoxycarbonyl-






phenyl





2.6.1183
3-trifluoro-methoxy-6-
methyl
(ethyl butanoate)-3-yl




methoxycarbonyl-






phenyl





2.6.1184
3-nitro-6-
methyl
(ethyl butanoate)-3-yl




methoxycarbonyl-






phenyl





2.6.1185
3-fluoro-6-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.1186
3-chloro-6-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.1187
3-bromo-6-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.1188
3-methyl-6-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.1189
3-cyclopropyl-6-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.1190
3-cyano-6-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.1191
3-trifluoromethyl-6-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.1192
3-methoxy-6-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.1193
3-ethoxy-6-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.1194
3-trifluoro-methoxy-6-
methyl
(ethyl butanoate)-3-yl




cyanophenyl





2.6.1195
3-nitro-6-cyanophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1196
3-fluoro-6-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1197
3-chloro-6-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1198
3-bromo-6-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1199
3-methyl-6-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1200
3-cyclopropyl-6-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1201
3-cyano-6-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1202
3-trifluoromethyl-6-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1203
3,6-dimethoxyphenyl
methyl
(ethyl butanoate)-3-yl



2.6.1204
3-ethoxy-6-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1205
3-trifluoro-methoxy-6-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1206
3-nitro-6-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1207
3-fluoro-6-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.1208
3-chloro-6-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.1209
3-bromo-6-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.1210
3-methyl-6-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.1211
3-cyclopropyl-6-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.1212
3-cyano-6-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.1213
3-trifluoromethyl-6-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.1214
3-methoxy-6-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.1215
2,6-diethoxyphenyl
methyl
(ethyl butanoate)-3-yl



2.6.1216
3-trifluoro-methoxy-6-
methyl
(ethyl butanoate)-3-yl




ethoxyphenyl





2.6.1217
3-nitro-6-ethoxyphenyl
methyl
(ethyl butanoate)-3-yl



2.6.1218
3-fluoro-6-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.1219
3-chloro-6-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.1220
3-bromo-6-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.1221
3-methyl-6-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.1222
3-cyclopropyl-6-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.1223
3-cyano-6-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.1224
3-trifluoromethyl-6-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.1225
3-meihoxy-6-propoxy -
methyl
(ethyl butanoate)-3-yl




phenyl





2.6.1226
3-ethoxy-6-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.1227
3-trifluoro-methoxy-6-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.1228
3-nitro-6-
methyl
(ethyl butanoate)-3-yl




propoxyphenyl





2.6.1229
3-fluoro-6-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.1230
3-chloro-6-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.1231
3-bromo-6-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.1232
3-methyl-6-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.1233
3-cyclopropyl-6-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.1234
3-cyano-6-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.1235
3-trifluoromethyl-6-
methyl
(ethyl butanoate)-3-yl




isopropoxy-phenyl





2.6.1236
3-methoxy-6-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.1237
3-ethoxy-6-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.1238
3-trifluoro-methoxy-6-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.1239
3-nitro-6-
methyl
(ethyl butanoate)-3-yl




isopropoxyphenyl





2.6.1240
3-fluoro-6-
methyl
(ethyl butanoate)-3-yl




trifluoromethoxy-






phenyl





2.6.1241
3-chloro-6-
methyl
(ethyl butanoate)-3-yl




trifluoromethoxy-






phenyl





2.6.1242
3-bromo-6-
methyl
(ethyl butanoate)-3-yl




trifluoromethoxy-






phenyl





2.6.1243
3-methyl-6-
methyl
(ethyl butanoate)-3-yl




trifluoromethoxy-






phenyl





2.6.1244
3-cyclopropyl-6-
methyl
(ethyl butanoate)-3-yl




trifluoromethoxy-






phenyl





2.6.1245
3-cyano-6-
methyl
(ethyl butanoate)-3-yl




trifluoromethoxy-






phenyl





2.6.1246
3-trifluoromethyl-6-
methyl
(ethyl butanoate)-3-yl




trifluoro-






methoxyphenyl





2.6.1247
3-methoxy-6-
methyl
(ethyl butanoate)-3-yl




trifluoromethoxy-






phenyl





2.6.1248
3-ethoxy-6-
methyl
(ethyl butanoate)-3-yl




trifluoromethoxy-






phenyl





2.6.1249
3,6-bis(trifluoro-
methyl
(ethyl butanoate)-3-yl




methoxy)phenyl





2.6.1250
3-nitro-6-
methyl
(ethyl butanoate)-3-yl




trifluoromethoxy-






phenyl





2.6.1251
3-fluoro-6-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.1252
3-chloro-6-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.1253
3-bromo-6-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.1254
3-methyl-6-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.1255
3-cyclopropyl-6-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.1256
3-cyano-6-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.1257
3-trifluoromethyl-6-
methyl
(ethyl butanoate)-3-yl




difluoro-






methoxyphenyl





2.6.1258
3-methoxy-6-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.1259
3-ethoxy-6-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.1260
3-trifluoro-methoxy-6-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.1261
3-nitro-6-
methyl
(ethyl butanoate)-3-yl




difluoromethoxy-






phenyl





2.6.1262
3-fluoro-6-nitrophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1263
3-chloro-6-nitrophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1264
3-bromo-6-nitrophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1265
3-methyl-6-nitrophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1266
3-cyclopropyl-6-
methyl
(ethyl butanoate)-3-yl




nitrophenyl





2.6.1267
3-cyano-6-nitrophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1268
3-trifluoromethyl-6-
methyl
(ethyl butanoate)-3-yl




nitrophenyl





2.6.1269
3-methoxy-6-
methyl
(ethyl butanoate)-3-yl




nitrophenyl





2.6.1270
3-ethoxy-6-nitrophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1271
3-trifluoro-methoxy-6-
methyl
(ethyl butanoate)-3-yl




nitrophenyl





2.6.1272
3-fluoro-6-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.1273
3-chloro-6-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.1274
3-bromo-6-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.1275
3-methyl-6-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.1276
3-cyclopropyl-6-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.1277
3-cyano-6-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.1278
3-trifluoromethyl-6-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.1279
3-methoxy-6-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.1280
3-ethoxy-6-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.1281
3-trifluoro-methoxy-6-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.1282
3-nitro-6-
methyl
(ethyl butanoate)-3-yl




methylsulfanyl-phenyl





2.6.1283
2,3,4-trifluorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1284
2,3,4-trichlorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1285
2,3,4-trimethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.1286
2-fluoro-2-chloro-5-
methyl
(ethyl butanoate)-3-yl




trifluoromethyl-phenyl





2.6.1287
2,3,5-trifluorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1288
2,3,5-trichlorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1289
2,3,5-trimethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.1290
2, 3-dichloro-5-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1291
2,3,6-trifluorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1292
2,3,6-trichlorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1293
2,3,6-trimethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.1294
3,4,5-trifluorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1295
3,4,5-trichlorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1296
3,4,5-trimethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.1297
3,5-dimethyl-4-
methyl
(ethyl butanoate)-3-yl




fluorophenyl





2.6.1298
3,5-dichloro-4-
methyl
(ethyl butanoate)-3-yl




methoxyphenyl





2.6.1299
3,5-difluoro-4-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.1300
3,5-dichloro-4-
methyl
(ethyl butanoate)-3-yl




hydroxyphenyl





2.6.1301
3,5-trifluoromethyl-4-
methyl
(ethyl butanoate)-3-yl




chlorophenyl





2.6.1302
3,4,6-trifluorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1303
3,4,6-trichlorophenyl
methyl
(ethyl butanoate)-3-yl



2.6.1304
3,4,6-trimethylphenyl
methyl
(ethyl butanoate)-3-yl



2.6.1305
2,3,4,5-pentafluoro-
methyl
(ethyl butanoate)-3-yl




phenyl
















TABLE 3







Inventive compounds of the general formula (I) in which W* is CN, R1 and


R2 are each hydrogen, and aryl is the radical.








 








 










No.
Aryl
R3
Physical data





3.1
3-fluorophenyl
methyl



3.2
3-fluorophenyl
ethyl



3.3
3-fluorophenyl
CN



3.4
3-fluorophenyl
fluoromethyl



3.5
3-fluorophenyl
hydroxymethyl



3.6
3-fluorophenyl
vinyl



3.7
3-fluorophenyl
1-chlorovinyl



3.8
3-fluorophenyl
ethynyl



3.9
3-chlorophenyl
methyl



3.10
3-chlorophenyl
ethyl



3.11
3-chlorophenyl
CN



3.12
3-chlorophenyl
fluoromethyl



3.13
3-chlorophenyl
hydroxymethyl



3.14
3-chlorophenyl
fluoromethyl



3.15
3-chlorophenyl
ethynyl



3.16
3-bromophenyl
methyl



3.17
3-bromophenyl
ethyl



3.18
3-bromophenyl
vinyl



3.19
3-iodophenyl
methyl



3.20
3-methylphenyl
methyl



3.21
3-ethylphenyl
methyl



3.22
3-propylphenyl
methyl



3.23
3-isopropylphenyl
methyl



3.24
3-n-butylphenyl
methyl



3.25
3-i-butylphenyl
methyl



3.26
3-tert-butylphenyl
methyl



3.27
3-cyclopropylphenyl
methyl



3.28
3-cyclobutylphenyl
methyl



3.29
3-cyclopentylphenyl
methyl



3.30
3-vinylphenyl
methyl



3.31
3-ethynylphenyl
methyl



3.32
3-cyanophenyl
methyl



3.33
3-trifluoromethylphenyl
methyl



3.34
3-difluoromethylphenyl
methyl



3.35
3-(hydroxycarbonyl)phenyl
methyl



3.36
3-(methoxycarbonyl)phenyl
methyl



3.37
3-(ethoxycarbonyl)phenyl
methyl



3.38
3-hydroxymethylphenyl
methyl



3.39
3-carbamoylphenyl
methyl



3.40
3-hydroxyphenyl
methyl



3.41
3-methoxyphenyl
methyl



3.42
3-methoxyphenyl
ethyl



3.43
3-methoxyphenyl
CN



3.44
3-methoxyphenyl
fluoromethyl



3.45
3-methoxyphenyl
hydroxymethyl



3.46
3-methoxyphenyl
ethynyl



3.47
3-ethoxyphenyl
methyl



3.48
3-propyloxyphenyl
methyl



3.49
3-isopropyloxyphenyl
methyl



3.50
3-n-butyloxyphenyl
methyl



3.51
3-i-butyloxyphenyl
methyl



3.52
3-t-butyloxyphenyl
methyl



3.53
3-difluoromethoxyphenyl
methyl



3.54
3-trifluoromethoxyphenyl
methyl



3.55
3-trifluoromethoxyphenyl
ethyl



3.56
3-trifluoromethoxyphenyl
CN



3.57
3-trifluoromethoxyphenyl
fluoromethyl



3.58
3-trifluoromethoxy
hydroxymethyl



3.59
3-trifluoromethoxyphenyl
ethynyl



3.60
3-(2,2,2-trifluoroethoxy)phenyl
methyl



3.61
3-nitrophenyl
methyl



3.62
3-acetoxyphenyl
methyl



3.63
(3-[(tert-butoxycarbonyl)amino]phenyl}
methyl



3.64
3-methylsulfanylphenyl
methyl



3.65
3-ethylsulfanylphenyl
methyl



3.66
3-(pentafluoro-lambda6-sulfanyl)phenyl
methyl



3.67
2,3-difluorophenyl
methyl



3.68
2,3-difluorophenyl
ethyl



3.69
2,3-difluorophenyl
CN



3.70
2,3-difluorophenyl
fluoromethyl



3.71
2,3-difluorophenyl
hydroxymethyl



3.72
2,3-difluorophenyl
ethynyl



3.73
2-chloro-3-fluorophenyl
methyl



3.74
2-bromo-3-fluorophenyl
methyl



3.75
2-methyl-3-fluorophenyl
methyl



3.76
2-ethyl-3-fluorophenyl
methyl



3.77
2-cyclopropyl-3-fluorophenyl
methyl



3.78
2-cyano-3-fluorophenyl
methyl



3.79
2-methoxy-3-fluorophenyl
methyl



3.80
2-ethoxy-3-fluorophenyl
methyl



3.81
2-trifluoromethoxy-3-fluorophenyl
methyl



3.82
2-nitro-3-fluorophenyl
methyl



3.83
2-fluoro-3-chlorophenyl
methyl



3.84
2,3-dichlorophenyl
methyl



3.85
2,3-dichlorophenyl
ethyl



3.86
2,3-dichlorophenyl
CN



3.87
2,3-dichlorophenyl
fluoromethyl



3.88
2,3-dichlorophenyl
hydroxymethyl



3.89
2,3-dichlorophenyl
ethynyl



3.90
2-bromo-3-chlorophenyl
methyl



3.91
2-methyl-3-chlorophenyl
methyl



3.92
2-methyl-3-chlorophenyl
ethyl



3.93
2-methyl-3-chlorophenyl
CN



3.94
2-methyl-3-chlorophenyl
fluoromethyl



3.95
2-methyl-3-chlorophenyl
hydroxymethyl



3.96
2-methyl-3-chlorophenyl
ethynyl



3.97
2-ethyl-3-chlorophenyl
methyl



3.98
2-cyclopropyl-3-chlorophenyl
methyl



3.99
2-cyano-3-chlorophenyl
methyl



3.100
2-trifluoromethyl-2-chlorophenyl
methyl



3.101
2-methoxy-3-chlorophenyl
methyl



3.102
2-ethoxy-3-chlorophenyl
methyl



3.103
2-trifluoromethoxy-3-chlorophenyl
methyl



3.104
2-nitro-3-chlorophenyl
methyl



3.105
2-fluoro-3-bromophenyl
methyl



3.106
2-chloro-3-bromophenyl
methyl



3.107
2,3-dibromophenyl
methyl



3.108
2-methyl-3-bromophenyl
methyl



3.109
2-ethyl-3-bromophenyl
methyl



3.110
2-cyclopropyl-3-bromophenyl
methyl



3.111
2-cyano-3-bromophenyl
methyl



3.112
2-trifluoromethyl-3-bromophenyl
methyl



3.113
2-methoxy-3-phenyl
methyl



3.114
2-ethoxy-3-bromophenyl
methyl



3.115
2-trifluoromethoxy-3-bromophenyl
methyl



3.116
2-nitro-3-bromophenyl
methyl



3.117
2-fluoro-3-iodophenyl
methyl



3.118
2-chloro-3-iodophenyl
methyl



3.119
2-bromo-3-iodophenyl
methyl



3.120
2-methyl-3-iodophenyl
methyl



3.121
2-ethyl-3-iodophenyl
methyl



3.122
2-cyclopropyl-3-iodophenyl
methyl



3.123
2-cyano-3-iodophenyl
methyl



3.124
2-trifluoromethyl-3-iodophenyl
methyl



3.125
2-methoxy-3-iodophenyl
methyl



3.126
2-ethoxy-3-iodophenyl
methyl



3.127
2-trifluoromethoxy-3-iodophenyl
methyl



3.128
2-nitro-3-iodophenyl
methyl



3.129
2-fluoro-3-methylphenyl
methyl



3.130
2-fluoro-3-methylphenyl
ethyl



3.131
2-fluoro-3-methylphenyl
CN



3.132
2-fluoro-3-methylphenyl
fluoromethyl



3.133
2-fluoro-3-methylphenyl
hydroxymethyl



3.134
2-fluoro-3-methylphenyl
ethynyl



3.135
2-chloro-3-methylphenyl
methyl



3.136
2-chloro-3-methylphenyl
ethyl



3.137
2-chloro-3-methylphenyl
CN



3.138
2-chloro-3-methylphenyl
fluoromethyl



3.139
2-chloro-3-methylphenyl
hydroxymethyl



3.140
2-chloro-3-methylphenyl
ethynyl



3.141
2-bromo-3-methylphenyl
methyl



3.142
2,3-dimethylphenyl
methyl



3.143
2-ethyl-3-methylphenyl
methyl



3.144
2-cyclopropyl-3-methylphenyl
methyl



3.145
2-cyano-3-methylphenyl
methyl



3.146
2-trifluoromethyl-3-methylphenyl
methyl



3.147
2-methoxy-3-methylphenyl
methyl



3.148
2-ethoxy-3-methylphenyl
methyl



3.149
2-trifluoromethoxy-3-methylphenyl
methyl



3.150
2-nitro-3-methylphenyl
methyl



3.151
2-fluoro-3-ethylphenyl
methyl



3.152
2-chloro-3-ethylphenyl
methyl



3.153
2-bromo-3-ethylphenyl
methyl



3.154
2-methyl-3-ethylphenyl
methyl



3.155
2,3-diethylphenyl
methyl



3.156
2-cyclopropyl-3-ethylphenyl
methyl



3.157
2-cyano-3-ethylphenyl
methyl



3.158
2-trifluoromethyl-3-ethylphenyl
methyl



3.159
2-methoxy-3-ethylphenyl
methyl



3.160
2-ethoxy-3-ethylphenyl
methyl



3.161
2-trifluoromethoxy-3-ethylphenyl
methyl



3.162
2-nitro-3-ethylphenyl
methyl



3.163
2-fluoro-3-propylphenyl
methyl



3.164
2-chloro-3-propylphenyl
methyl



3.165
2-bromo-3-propylphenyl
methyl



3.166
2-methyl-3-propylphenyl
methyl



3.167
2-methyl-3-propylphenyl
methyl



3.168
2-cyclopropyl-3-propylphenyl
methyl



3.169
2-cyano-3-propylphenyl
methyl



3.170
2-trifluoromethyl-3-propylphenyl
methyl



3.171
2-methoxy-3-propylphenyl
methyl



3.172
2-ethoxy-3-propylphenyl
methyl



3.173
2-trifluoromethoxy-3-propylphenyl
methyl



3.174
2-nitro-3-propylphenyl
methyl



3.175
2-fluoro-3-isopropylphenyl
methyl



3.176
2-chloro-3-isopropylphenyl
methyl



3.177
2-bromo-3- isopropylphenyl
methyl



3.178
2-methyl-3-isopropylphenyl
methyl



3.179
2-ethyl-3-isopropylphenyl
methyl



3.180
2-cyclopropyl-3-isopropylphenyl
methyl



3.181
2-cyano-3-isopropylphenyl
methyl



3.182
2-trifluoromethyl-3-isopropylphenyl
methyl



3.183
2- methoxy-3-isopropylphenyl
methyl



3.184
2-ethoxy-3-isopropylphenyl
methyl



3.185
2-trifluoromethoxy-3-isopropylphenyl
methyl



3.186
2-nitro-3-isopropylphenyl
methyl



3.187
2-fluoro-3-tert-butylphenyl
methyl



3.188
2-fluoro-3-tert-butylphenyl
ethyl



3.189
2-fluoro-3-tert-butylphenyl
CN



3.190
2-fluoro-3-tert-butylphenyl
fluoromethyl



3.191
2-fluoro-3-tert-butylphenyl
hydroxymethyl



3.192
2-fluoro-3-tert-butylphenyl
ethynyl



3.193
2-chloro-3-tert-butylphenyl
methyl



3.194
2-bromo-3-tert-butylphenyl
methyl



3.195
2-methyl-3-tert-butylphenyl
methyl



3.196
2-ethyl-3-tert-butylphenyl
methyl



3.197
2-cyclopropyl-3-tert-butylphenyl
methyl



3.198
2-cyano-3-tert-butylphenyl
methyl



3.199
2-trifluoromethyl-3-tert-butylphenyl
methyl



3.200
2- methoxy-3-tert-butylphenyl
methyl



3.201
2-ethoxy-3-tert-butylphenyl
methyl



3.202
2-trifluoromethoxy-3-tert-butylphenyl
methyl



3.203
2-nitro-3-tert-butylphenyl
methyl



3.204
2-fluoro-3-cyclopropylphenyl
methyl



3.205
2-chloro-3-cyclopropylphenyl
methyl



3.206
2-bromo-3-cyclopropylphenyl
methyl



3.207
2-methyl-3-cyclopropylphenyl
methyl



3.208
2-ethyl-3-cyclopropylphenyl
methyl



3.209
2-cyclopropy1-3-cyclopropyl phenyl
methyl



3.210
2-cyano-3-cyclopropylphenyl
methyl



3.211
2-trifluoromethyl-3-cyclopropylphenyl 
methyl



3.212
2-methoxy-3-cyclopropylphenyl
methyl



3.213
2-ethoxy-3-cyclopropylphenyl
methyl



3.214
2-trifluoromethoxy-3-cyclopropylphenyl
methyl



3.215
2-fluoro-3-methoxycarbonylphenyl
methyl



3.216
2-chloro-3-methoxycarbonylphenyl
methyl



3.217
2-bromo-3-methoxycarbonylphenyl
methyl



3.218
2-methyl-3-methoxycarbonylphenyl
methyl



3.219
2-methyl-3-methoxycarbonylphenyl
ethyl



3.220
2-methyl-3-methoxycarbonylphenyl
CN



3.221
2-methyl-3-methoxycarbonylphenyl
vinyl



3.222
2-methyl-3-methoxycarbonylphenyl
fluoromethyl



3.223
2-methyl-3-methoxycarbonylphenyl
hydroxymethyl



3.224
2-methyl-3-methoxycarbonylphenyl
ethynyl



3.225
2-ethyl-3-methoxycarbonylphenyl
methyl



3.226
2-cyclopropyl-3-methoxycarbonyl-phenyl
methyl



3.227
2-cyano-3-methoxycarbonylphenyl
methyl



3.228
2-trifluoromethy1-3-
methyl




methoxycarbonylphenyl




3.229
2-methoxy-3-methoxycarbonylphenyl
methyl



3.230
2-ethoxy-3-methoxycarbonylphenyl
methyl



3.231
2-trifluoromethoxy-3-
methyl




methoxycarbonylphenyl




3.232
2-nitro-3-methoxycarbonylphenyl
methyl



3.233
2-fluoro-3-cyanophenyl
methyl



3.234
2-fluoro-3-cyanophenyl
ethyl



3.235
2-fluoro-3-cyanophenyl
CN



3.236
2-fluoro-3-cyanophenyl
vinyl



3.237
2-fluoro-3-cyanophenyl
fluoromethyl



3.238
2-fluoro-3-cyanophenyl
hydroxymethyl



3.239
2-fluoro-3-cyanophenyl
ethynyl



3.240
2-chloro-3-cyanophenyl
methyl



3.241
2-chloro-3-cyanophenyl
ethyl



3.242
2-chloro-3-cyanophenyl
CN



3.243
2-chloro-3-cyanophenyl
vinyl



3.244
2-chloro-3-cyanophenyl
fluoromethyl



3.245
2-chloro-3-cyanophenyl
hydroxymethyl



3.246
2-chloro-3-cyanophenyl
ethynyl



3.247
2-bromo-3-cyanophenyl
methyl



3.248
2-methyl-3-cyanophenyl
methyl



3.249
2-ethyl-3-cyanophenyl
methyl



3.250
2-cyclopropyl-3-cyanophenyl
methyl



3.251
2-cyano-3-cyanophenyl
methyl



3.252
2-trifluoromethyl-3-cyanophenyl
methyl



3.253
2-methoxy-3-cyanophenyl
methyl



3.254
2-ethoxy-3-cyanophenyl
methyl



3.255
2-trifluoromethoxy-3-cyanophenyl
methyl



3.256
2-nitro-3-cyanophenyl
methyl



3.257
2-chloro-3-methoxyphenyl
methyl



3.258
2-bromo-3-methoxyphenyl
methyl



3.259
2-methyl-3-methoxyphenyl
methyl



3.260
2-ethyl-3-methoxyphenyl
methyl



3.261
2-cyclopropyl-3-methoxyphenyl
methyl



3.262
2-cyano-3-methoxyphenyl
methyl



3.263
2-trifluoromethyl-3-methoxyphenyl
methyl



3.264
2,3-dimethoxyphenyl
methyl



3.265
2-ethoxy-3-methoxyphenyl
methyl



3.266
2-trifluoromethoxy-3-methoxyphenyl
methyl



3.267
2- nitro-3-methoxyphenyl
methyl



3.268
2-fluoro-3-ethoxyphenyl
methyl



3.269
2-chloro-3-ethoxyphenyl
methyl



3.270
2-bromo-3-ethoxyphenyl
methyl



3.271
2-methyl-3-ethoxyphenyl
methyl



3.272
2-ethyl-3-ethoxyphenyl
methyl



3.273
2-cyclopropyl-3-ethoxyphenyl
methyl



3.274
2-cyano-3-ethoxyphenyl
methyl



3.275
2-trifluoromethyl-3-ethoxyphenyl
methyl



3.276
2-methoxy-3-ethoxyphenyl
methyl



3.277
2,3-diethoxyphenyl
methyl



3.278
2-trifluoromethoxy-3-ethoxyphenyl
methyl



3.279
2-nitro-3-ethoxyphenyl
methyl



3.280
2-fluoro-3-propoxyphenyl
methyl



3.281
2-chloro-3-propoxyphenyl
methyl



3.282
2-bromo-3-propoxyphenyl
methyl



3.283
2-methyl-3-propoxyphenyl
methyl



3.284
2-ethyl-3-propoxyphenyl
methyl



3.285
2-cyclopropyl-3-propoxyphenyl
methyl



3.286
2-vinyl-3-propoxyphenyl
methyl



3.287
2-ethynyl-3-propoxyphenyl
methyl



3.288
2-cyano-3-propoxyphenyl
methyl



3.289
2-trifluoromethyl-3-propoxyphenyl
methyl



3.290
2-methoxy-3-propoxyphenyl
methyl



3.291
2-ethoxy-3-propoxyphenyl
methyl



3.292
2-trifluoromethoxy-3-propoxyphenyl
methyl



3.293
2-nitro-3-propoxyphenyl
methyl



3.294
2-fluoro-3-isopropoxyphenyl
methyl



3.295
2-chloro-3-isopropoxyphenyl
methyl



3.296
2-bromo-3-isopropoxyphenyl
methyl



3.297
2- methyl-3-isopropoxyphenyl
methyl



3.298
2-ethyl-3-isopropoxyphenyl
methyl



3.299
2-cyclopropyl-3-isopropoxyphenyl
methyl



3.300
2-vinyl-3-isopropoxyphenyl
methyl



3.301
2-ethynyl-3-isopropoxyphenyl
methyl



3.302
2-cyano-3-isopropoxyphenyl
methyl



3.303
2-trifluoromethyl-3-isopropoxyphenyl
methyl



3.304
2-methoxy-3-isopropoxyphenyl
methyl



3.305
2-ethoxy-3-isopropoxyphenyl
methyl



3.306
2-trifluoromethoxy-3-isopropoxyphenyl
methyl



3.307
2-nitro-3-isopropoxyphenyl
methyl



3.308
2-fluoro-3-trifluoromethoxyphenyl
methyl



3.309
2-chloro-3-trifluoromethoxyphenyl 
methyl



3.310
2-bromo-3-trifluoromethoxyphenyl 
methyl



3.311
2-methyl-3-trifluoromethoxyphenyl
methyl



3.312
2-ethyl-3-trifluoromethoxyphenyl
methyl



3.313
2-cyclopropyl-3-trifluoromethoxyphenyl
methyl



3.314
2-cyano-3-trifluoromethoxyphenyl
methyl



3.315
2-trifluoromethyl-3-trifluoromethoxy-
methyl




phenyl




3.316
2-methoxy-3-trifluoromethoxyphenyl
methyl



3.317
2-ethoxy-3-trifluoromethoxyphenyl
methyl



3.318
2,3-bis(trifluoromethoxy)phenyl
methyl



3.319
2-nitro-3-trifluoromethoxyphenyl
methyl



3.320
2-fluoro-3-difluoromethoxyphenyl
methyl



3.321
2-chloro-3-difluoromethoxyphenyl
methyl



3.322
2-bromo-3-difluoromethoxyphenyl
methyl



3.323
2-methyl-3-difluoromethoxyphenyl
methyl



3.324
2-ethyl-3-difluoromethoxyphenyl
methyl



3.325
2-cyclopropyl-3-difluoromethoxyphenyl
methyl



3.326
2-cyano-3-difluoromethoxyphenyl
methyl



3.327
2-trifluoromethyl-3-difluoromethoxyphenyl
methyl



3.328
2-methoxy-3-difluoromethoxyphenyl
methyl



3.329
2-ethoxy-3-difluoromethoxyphenyl
methyl



3.330
2-trifluoromethoxy-3-difluoromethoxy-
methyl




phenyl




3.331
2-nitro-3-difluoromethoxyphenyl
methyl



3.332
2-fluoro-3-nitrophenyl
methyl



3.333
2-chloro-3-nitrophenyl
methyl



3.334
2-bromo-3-nitrophenyl
methyl



3.335
2-methyl-3-nitrophenyl
methyl



3.336
2-ethyl-3-nitrophenyl
methyl



3.337
2-cyclopropyl-3-nitrophenyl
methyl



3.338
2-cyano-3-nitrophenyl
methyl



3.339
2-trifluoromethyl-3-nitrophenyl
methyl



3.340
2-methoxy-3-nitrophenyl
methyl



3.341
2-ethoxy-3-nitrophenyl
methyl



3.342
2-trifluoromethoxy-3-nitrophenyl
methyl



3.343
2-fluoro-3-methylsulfanylphenyl
methyl



3.344
2-chloro-3-methylsulfanylphenyl
methyl



3.345
2-bromo-3-methylsulfanylphenyl
methyl



3.346
2-methyl-3-methylsulfanylphenyl
methyl



3.347
2-ethyl-3-methylsulfanylphenyl
methyl



3.348
2-cyclopropyl-3-methylsulfanylphenyl
methyl



3.349
2-cyano-3-methylsulfanylphenyl
methyl



3.350
2-trifluoromethyl-3-methylsulfanylpheny
lmethyl



3.351
2-methoxy-3-methylsulfanylphenyl
methyl



3.352
2-ethoxy-3-methylsulfanylphenyl
methyl



3.353
2-trifluoromethoxy-3-methylsulfanylphenyl
methyl



3.354
2-nitro-3-methylsulfanylphenyl
methyl



3.355
3,5-difluorophenyl
methyl
[CDCl3] 1.91 (s, 3H),





3.38 (d, 1H), 3.81 (d,





1H), 6.93 (m, 1H),





7.18 (m, 2H)


3.356
3,5-difluorophenyl
ethyl



3.357
3,5-difluorophenyl
CN



3.358
3,5-difluorophenyl
vinyl



3.359
3,5-difluorophenyl
fluoromethyl



3.360
3,5-difluorophenyl
hydroxymethyl



3.361
3,5-difluorophenyl
ethynyl



3.362
3-chloro-5-fluorophenyl
methyl



3.363
3-chloro-5-fluorophenyl
ethyl



3.364
3-chloro-5-fluorophenyl
CN



3.365
3-chloro-5-fluorophenyl
vinyl



3.366
3-chloro-5-fluorophenyl
fluoromethyl



3.367
3-chloro-5-fluorophenyl
hydroxymethyl



3.368
3-chloro-5-fluorophenyl
ethynyl



3.369
3-bromo-5-fluorophenyl
methyl



3.370
3-iodo-5-fluorophenyl
methyl



3.371
3-methyl-5-fluorophenyl
methyl



3.372
3-methyl-5-fluorophenyl
ethyl



3.373
3-methyl-5-fluorophenyl
CN



3.374
3-methyl-5-fluorophenyl
vinyl



3.375
3-methyl-5-fluorophenyl
fluoromethyl



3.376
3-methyl-5-fluorophenyl
hydroxymethyl



3.377
3-methyl-5-fluorophenyl
ethynyl



3.378
3-ethyl-5-fluorophenyl
methyl



3.379
3-propyl-5-fluorophenyl
methyl



3.380
3-i-propyl-5-fluorophenyl
methyl



3.381
3-n-butyl-5-fluorophenyl
methyl



3.382
3-isobutyl-5-fluorophenyl
methyl



3.383
3-tert-butyl-5-fluorophenyl
methyl



3.384
3-tert-butyl-5-fluorophenyl
ethyl



3.385
3-tert-butyl-5-fluorophenyl
CN



3.386
3-tert-butyl-5-fluorophenyl
vinyl



3.387
3-tert-butyl-5-fluorophenyl
fluoromethyl



3.388
3-tert-butyl-5-fluorophenyl
hydroxymethyl



3.389
3-tert-butyl-5-fluorophenyl
ethynyl



3.390
3-cyclopropyl-5-fluorophenyl
methyl



3.391
3-cyano-5-fluorophenyl
methyl



3.392
3-cyano-5-fluorophenyl
ethyl



3.393
3-cyano-5-fluorophenyl
CN



3.394
3-cyano-5-fluorophenyl
vinyl



3.395
3-cyano-5-fluorophenyl
fluoromethyl



3.396
3-cyano-5-fluorophenyl
hydroxymethyl



3.397
3-cyano-5-fluorophenyl
ethynyl



3.398
3-trifluoromethyl-5-fluorophenyl
methyl



3.399
3-(methoxycarbonyI)-5-fluorophenyl
methyl



3.400
3-methoxy-5-fluorophenyl
methyl



3.401
3-methoxy-5-fluorophenyl
ethyl



3.402
3-methoxy-5-fluorophenyl
CN



3.403
3-methoxy-5-fluorophenyl
vinyl



3.404
3-methoxy-5-fluorophenyl
fluoromethyl



3.405
3-methoxy-5-fluorophenyl
hydroxymethyl



3.406
3-methoxy-5-fluorophenyl
ethynyl



3.407
3-ethoxy-5-fluorophenyl
methyl



3.408
3-n-propoxy-5-fluorophenyl
methyl



3.409
3-isopropoxy-5-fluorophenyl
methyl



3.410
3-n-butoxy-5-fluorophenyl
methyl



3.411
3-isobutoxy-5-fluorophenyl
methyl



3.412
3-difluoromethoxy-5-fluorophenyl
methyl



3.413
3-trifluoromethoxy-5-fluorophenyl
methyl



3.414
3-nitro-5-fluorophenyl
methyl



3.415
3-acetoxy-5-fluorophenyl
methyl



3.416
3-methylsulfanyl-5-fluorophenyl 
methyl



3.417
3,5-dichlorophenyl
methyl
[CDCl3] 1.91 (s, 3H);





3.38 (d, 1H); 3.80 (d,





1H); 7.45 (s, 1H); 7.52





(s, 1H).


3.418
3,5-dichlorophenyl
ethyl



3.419
3,5-dichlorophenyl
isopropyl
[DMSO] 1.06 (d, 3H);





1.10 (d, 3H); 2.25 (m,





1H); 3.85 (d, 1H); 4.10





(d, 1H); 7.74 (d, 1H);





7.79 (d, 1H).


3.420
3,5-dichlorophenyl
vinyl



3.421
3,5-dichlorophenyl
fluoromethyl



3.422
3,5-dichlorophenyl
hydroxymethyl



3.423
3,5-dichlorophenyl
ethynyl



3.424
3-bromo-5-chlorophenyl
methyl



3.425
3-iodo-5-chlorophenyl
methyl



3.426
3-methyl-5-chlorophenyl
methyl



3.427
3-methyl-5-chlorophenyl
ethyl



3.428
3-methyl-5-chlorophenyl
CN



3.429
3-methyl-5-chlorophenyl
vinyl



3.430
3-methyl-5-chlorophenyl
fluoromethyl



3.431
3-methyl-5-chlorophenyl
hydroxymethyl



3.432
3-methyl-5-chlorophenyl
ethynyl



3.433
3-ethyl-5-chlorophenyl
methyl



3.434
3-propyl-5-chlorophenyl
methyl



3.435
3-isopropyl-5-chlorophenyl
methyl



3.436
3-n-butyl-5-chlorophenyl
methyl



3.437
3-isobutyl-5-chlorophenyl
methyl



3.438
3-tert-butyl-5-chlorophenyl
methyl



3.439
3-cyclopropyl-5-chlorophenyl
methyl



3.440
3-cyano-5-chlorophenyl
methyl



3.441
3-cyano-5-chlorophenyl
ethyl



3.442
3-cyano-5-chlorophenyl
CN



3.443
3-cyano-5-chlorophenyl
vinyl



3.444
3-cyano-5-chlorophenyl
fluoromethyl



3.445
3-cyano-5-chlorophenyl
hydroxymethyl



3.446
3-cyano-5-chlorophenyl
ethynyl



3.447
3-trifluoromethyl-5-chlorophenyl
methyl



3.448
3-trifluoromethyl-5-chlorophenyl
ethyl



3.449
3-trifluoromethyl-5-chlorophenyl
CN



3.450
3-trifluoromethyl-5-chlorophenyl
vinyl



3.451
3-trifluoromethyl-5-chlorophenyl
fluoromethyl



3.452
3-trifluoromethyl-5-chlorophenyl
hydroxymethyl



3.453
3-trifluoromethyl-5-chlorophenyl
ethynyl



3.454
3-(methoxycarbony1)-5-chlorophenyl
methyl



3.455
3-methoxy-5-chlorophenyl
methyl



3.456
3-methoxy-5-chlorophenyl
ethyl



3.457
3-methoxy-5-chlorophenyl
CN



3.458
3-methoxy-5-chlorophenyl
vinyl



3.459
3-methoxy-5-chlorophenyl
fluoromethyl



3.460
3-methoxy-5-chlorophenyl
hydroxymethyl



3.461
3-methoxy-5-chlorophenyl
ethynyl



3.462
3-ethoxy-5-chlorophenyl
methyl



3.463
3-n-propoxy-5-chlorophenyl
methyl



3.464
3-isopropoxy-5-chlorophenyl
methyl



3.465
3-isobutoxy-5-chlorophenyl
methyl



3.466
3-difluoromethoxy-5-chlorophenyl
methyl



3.467
3-trifluoromethoxy-5-chlorophenyl
methyl



3.468
3-trifluoromethoxy-5-chlorophenyl
ethyl



3.469
3-trifluoromethoxy-5-chlorophenyl
CN



3.470
3-trifluoromethoxy-5-chlorophenyl
vinyl



3.471
3-trifluoromethoxy-5-chlorophenyl
fluoromethyl



3.472
3-trifluoromethoxy-5-chlorophenyl
hydroxymethyl



3.473
3-trifluoromethoxy-5-chlorophenyl
ethynyl



3.474
3-nitro-5-chlorophenyl
methyl



3.475
3-acetoxy-5-chlorophenyl
methyl



3.476
3-methylsulfanyl-5-chlorophenyl
methyl



3.477
3,5-dibromophenylphenyl
methyl



3.478
3-iodo-5-bromophenyl
methyl



3.479
3-methyl-5-bromophenyl
methyl



3.480
3-ethyl-5-bromophenyl
methyl



3.481
3-propyl-5-bromophenyl
methyl



3.482
3-isopropyl-5-bromophenyl
methyl



3.483
3-n-butyl-5-bromophenyl
methyl



3.484
3-isobutyl-5-bromophenyl
methyl



3.485
3-tert-butyl-5-bromophenyl
methyl



3.486
3-cyclopropyl-5-bromophenyl
methyl



3.487
3-cyano-5-bromophenyl
methyl



3.488
3-trifluoromethyl-5-bromophenyl
methyl



3.489
3-(methoxycarbonyl)-5-bromophenyl
methyl



3.490
3-methoxy-5-bromophenyl
methyl



3.491
3-ethoxy-5-bromophenyl
methyl



3.492
3-n-propoxy-5-bromophenyl
methyl



3.493
3-isopropoxy-5-bromophenyl
methyl



3.494
3-n-butoxy-5-bromophenyl
methyl



3.495
3-isobutoxy-5-bromophenyl
methyl



3.496
3-difluoromethoxy-5-bromophenyl
methyl



3.497
3-trifluoromethoxy-5-bromophenyl
methyl



3.498
3-nitro-5-bromophenyl
methyl



3.499
3-acetoxy-5-bromophenyl
methyl



3.500
3-methylsulf anyl-5-bromophenyl
methyl



3.501
3,5-diiodophenyl
methyl



3.502
3-methyl-5-iodophenyl
methyl



3.503
3-ethyl-5-iodophenyl
methyl



3.504
3-propyl-5-iodophenyl
methyl



3.505
3-isopropyl-5-iodophenyl
methyl



3.506
3-n-butyl-5-iodophenyl
methyl



3.507
3-isobutyl-5-iodophenyl
methyl



3.508
3-tert-butyl-5-iodophenyl
methyl



3.509
3-cyclopropyl-5-iodophenyl
methyl



3.510
3-cyano-5-iodophenyl
methyl



3.511
3-trifluoromethyl-5-iodophenyl
methyl



3.512
3-(methoxycarbonyl)-5-iodophenyl
methyl



3.513
3-methoxy-5-iodophenyl
methyl



3.514
3-ethoxy-5-iodophenyl
methyl



3.515
3-n-propoxy-5-iodophenyl
methyl



3.516
3-isopropoxy-5-iodophenyl
methyl



3.517
3- n-butoxy-5-iodophenyl
methyl



3.518
3-isobutoxy-5-iodophenyl
methyl



3.519
3-difluoromethoxy-5-iodophenyl
methyl



3.520
3-trifluoromethoxy-5-iodophenyl
methyl



3.521
3-nitro-5-iodophenyl
methyl



3.522
3-acetoxy-5-iodophenyl
methyl



3.523
3-methylsulfanyl-5-iodophenyl
methyl



3.524
3,5-dimethylphenyl
methyl



3.525
3-ethyl-5-methylphenyl
methyl



3.526
3-propyl-5-methylphenyl
methyl



3.527
3-isopropyl-5-methylphenyl
methyl



3.528
3-n-butyl-5-methylphenyl
methyl



3.529
3-isobutyl-5-methylphenyl
methyl



3.530
3-tert-butyl-5-methylphenyl
methyl



3.531
3-cyclopropyl-5-methylphenyl
methyl



3.532
3-cyano-5-methylphenyl
methyl



3.533
3-trifluoromethyl-5-methylphenyl
methyl



3.534
3-(methoxycarbonyl)-5-methylphenyl
methyl



3.535
3-methoxy-5-methylphenyl
methyl



3.536
3-ethoxy-5-methylphenyl
methyl



3.537
3-n-propoxy-5-methylphenyl
methyl



3.538
3-isobutoxy-5-methylphenyl
methyl



3.539
3-difluoromethoxy-5-methylphenyl
methyl



3.540
3-trifluoromethoxy-5-methylphenyl
methyl



3.541
3-nitro-5-methylphenyl
methyl



3.542
3-acetoxy-5-methylphenyl
methyl



3.543
3-methylsulfanyl-5-methylphenyl
methyl



3.544
3,5-diethylphenyl
methyl



3.545
3-propyl-5-ethylphenyl
methyl



3.546
3-isopropyl-5-ethylphenyl
methyl



3.547
3-n-butyl-5-ethylphenyl
methyl



3.548
3-isobutyl-5-ethylphenyl
methyl



3.549
3-cyclopropyl-5-ethylphenyl
methyl



3.550
3-cyano-5-ethylphenyl
methyl



3.551
3-trifluoromethyl-5-ethylphenyl
methyl



3.552
3-(methoxycarbonyl)-5-ethylphenyl
methyl



3.553
3-methoxy-5-ethylphenyl
methyl



3.554
3-ethoxy-5-ethylphenyl
methyl



3.555
3-n-propoxy-5-ethylphenyl
methyl



3.556
3-n-butoxy-5-ethylphenyl
methyl



3.557
3-isobutoxy-5-ethylphenyl
methyl



3.558
3-difluoromethoxy-5-ethylphenyl
methyl



3.559
3-trifluoromethoxy-5-ethylphenyl
methyl



3.560
3-nitro-5-ethylphenyl
methyl



3.561
3-acetoxy-5-ethylphenyl
methyl



3.562
3-methylsulfanyl-5-ethylphenyl
methyl



3.563
3,5-dipropylphenyl
methyl



3.564
3-isopropyl-5-propylphenyl
methyl



3.565
3-n-butyl-5-propylphenyl
methyl



3.566
3-isobutyl-5-propylphenyl
methyl



3.567
3-tert-butyl-5-propylphenyl
methyl



3.568
3-cyclopropyl-5-propylphenyl
methyl



3.569
3-cyano-5-propylphenyl
methyl



3.570
3-trifluoromethyl-5-propylphenyl
methyl



3.571
3-(methoxycarbonyl)-5-propylphenyl
methyl



3.572
3-methoxy-5-propylphenyl
methyl



3.573
3-ethoxy-5-propylphenyl
methyl



3.574
3-n-propoxy-5-propylphenyl
methyl



3.575
3-isobutoxy-5-propylphenyl
methyl



3.576
3-difluoromethoxy-5-propylphenyl 
methyl



3.577
3-trifluoromethoxy-5-ethylphenyl 
methyl



3.578
3-nitro-5-propylphenyl
methyl



3.579
3-acetoxy-5-propylphenyl
methyl



3.580
3-methylsulfanyl-5-propylphenyl
methyl



3.581
3,5-diisopropylphenyl
methyl



3.582
3-n-butyl-5-isopropylphenyl
methyl



3.583
3-isobutyl-5-isopropylphenyl
methyl



3.584
3-tert-butyl-5-isopropylphenyl
methyl



3.585
3-cyclopropyl-5-isopropylphenyl
methyl



3.586
3-cyano-5-isopropylphenyl
methyl



3.587
3-trifluoromethyl-5-isopropylphenyl
methyl



3.588
3-(methoxycarbonyl)-5-isopropylphenyl
methyl



3.589
3- methoxy-5-isopropylphenyl
methyl



3.590
3-ethoxy-5-isopropylphenyl
methyl



3.591
3-n-propoxy-5-isopropylphenyl
methyl



3.592
3-isobutoxy-5- isopropylphenyl
methyl



3.593
3-difluoromethoxy-5- isopropylphenyl
methyl



3.594
3-trifluoromethoxy-5-isopropylphenyl
methyl



3.595
3-nitro-5-isopropylphenyl
methyl



3.596
3-acetoxy-5-isopropylphenyl
methyl



3.597
3-methylsulfanyl-5-isopropylphenyl
methyl



3.598
3,5-diisobutylphenyl
methyl



3.599
3-tert-butyl-5-isobutylphenyl
methyl



3.600
3-cyclopropyl-5-isobutylphenyl
methyl



3.601
3-cyano-5-isobutylphenyl
methyl



3.602
3-trifluoromethyl-5-isobutylphenyl
methyl



3.603
3-(methoxycarbonyl)-5-isobutylphenyl
methyl



3.604
3-ethoxy-5-isobutylphenyl
methyl



3.605
3-n-propoxy-5-isobutylphenyl
methyl



3.606
3-isobutoxy-5-isobutylphenyl
methyl



3.607
3-difluoromethoxy-5-isobutylphenyl
methyl



3.608
3-trifluoromethoxy-5-isobutylphenyl
methyl



3.609
3-nitro-5- isobutylphenyl
methyl



3.610
3-acetoxy-5-isobutylphenyl
methyl



3.611
3-methylsulfanyl-5-isobutylphenyl
methyl



3.612
3,5-d i-tert-butylphenyl
methyl



3.613
3-cyclopropyl-5-tert-butylphenyl
methyl



3.614
3-cyano-5-tert-butylphenyl
methyl



3.615
3-trifluoromethyl-5-tert-butylphenyl
methyl



3.616
3-(methoxycarbonyl)-5-tert-butylphenyl
methyl



3.617
3-methoxy-5-tert-butylphenyl
methyl



3.618
3-ethoxy-5-tert-butylphenyl
methyl



3.619
3-n-propoxy-5-tert-butylphenyl
methyl



3.620
3-isobutoxy-5-tert-butylphenyl
methyl



3.621
3-difluoromethoxy-5-tert-butylphenyl
methyl



3.622
3-trifluoromethoxy-5-tert-butylphenyl
methyl



3.623
3-nitro-5-tert-butylphenyl
methyl



3.624
3-acetoxy-5-tert-butylphenyl
methyl



3.625
3-methylsulfanyl-5-tert-butylphenyl
methyl



3.626
3-tert-butyl-5-cyclopropylphenyl
methyl



3.627
3,5-dicyclopropylphenyl
methyl



3.628
3-cyano-5-cyclopropylphenyl
methyl



3.629
3-cyano-5-cyclopropylphenyl
ethyl



3.630
3-cyano-5-cyclopropylphenyl
CN



3.631
3-cyano-5-cyclopropylphenyl
vinyl



3.632
3-cyano-5-cyclopropylphenyl
fluoromethyl



3.633
3-cyano-5-cyclopropylphenyl
hydroxymethyl



3.634
3-cyano-5-cyclopropylphenyl
ethynyl



3.635
3-trifluoromethyl-5-cyclopropylphenyl
methyl



3.636
3-(methoxycarbonyl)-5-cyclopropylphenyl
methyl



3.637
3-methoxy-5-cyclopropylphenyl
methyl



3.638
3-ethoxy-5-cyclopropylphenyl
methyl



3.639
3-n-propoxy-5-cyclopropylphenyl
methyl



3.640
3-isobutoxy-5-cyclopropylphenyl
methyl



3.641
3-difluoromethoxy-5-cyclopropylphenyl
methyl



3.642
3-trifluoromethoxy-5-cyclopropylphenyl
methyl



3.643
3-nitro-5-cyclopropylphenyl
methyl



3.644
3-acetoxy-5-cyclopropylphenyl
methyl



3.645
3-methylsulfanyl-5-cyclopropylphenyl
methyl



3.646
3,5-dicyanophenyl
methyl



3.647
3-trifluoromethyl-5-cyanophenyl
methyl



3.648
3-(methoxycarbonyl)-5-cyanophenyl
methyl



3.649
3-methoxy-5-cyanophenyl
methyl



3.650
3-ethoxy-5-cyanophenyl
methyl



3.651
3-n-propoxy-5-cyanophenyl
methyl



3.652
3-isobutoxy-5-cyanophenyl
methyl



3.653
3-difluoromethoxy-5-cyanophenyl
methyl



3.654
3-trifluoromethoxy-5-cyanophenyl
methyl



3.655
3-nitro-5-cyanophenyl
methyl



3.656
3-acetoxy-5-cyanophenyl
methyl



3.657
3-methylsulfanyl-5-cyanophenyl
methyl



3.658
3,5-di(trifluoromethyl)phenyl
methyl



3.659
3,5-di(trifluoromethyl)phenyl
ethyl



3.660
3,5-di(trifluoromethyl)phenyl
CN



3.661
3,5-di(trifluoromethyl)phenyl
vinyl



3.662
3,5-di(trifluoromethyl)phenyl
fluoromethyl



3.663
3,5-di(trifluoromethyl)phenyl
hydroxymethyl



3.664
3,5-di(trifluoromethyl)phenyl
ethynyl



3.665
3-(methoxycarbonyl)-5-trifluoromethyl-
methyl




phenyl




3.666
3-methoxy-5-trifluoromethylphenyl
methyl



3.667
3-ethoxy-5-trifluoromethylphenyl
methyl



3.668
3-n-propoxy-5-trifluoromethylphenyl
methyl



3.669
3-n-butoxy-5-trifluoromethylphenyl
methyl



3.670
3-isobutoxy-5-trifluoromethylphenyl
methyl



3.671
3-difluoromethoxy-5-trifluoromethylphenyl
methyl



3.672
3-trifluoromethoxy-5-trifluoromethylphenyl
methyl



3.673
3-nitro-5-trifluoromethylphenyl
methyl



3.674
3-acetoxy-5-trifluoromethylphenyl
methyl



3.675
3-methylsulfanyl-5-trifluoromethylphenyl
methyl



3.676
3,5-di(methoxycarbonyl)phenyl
methyl



3.677
3-methoxy-5-(methoxycarbonyl)phenyl
methyl



3.678
3-ethoxy-5-(methoxycarbonyl)phenyl
methyl



3.679
3-n-propoxy-5-(methoxycarbonyl)phenyl
methyl



3.680
3-isobutoxy-5-(methoxycarbonyl)phenyl
methyl



3.681
3-difluoromethoxy-5-(methoxycarbonyl)-
methyl




phenyl




3.682
3-trifluoromethoxy-5-(methoxycarbonyl)-
methyl




phenyl




3.683
3-nitro-5-(methoxycarbonyl)phenyl
methyl



3.684
3-acetoxy-5-(methoxycarbonyl)phenyl
methyl



3.685
3-methylsulfanyl-5-(methoxycarbonyl)-
methyl




phenyl




3.686
3,5-dimethoxyphenyl
methyl



3.687
3,5-dimethoxyphenyl
ethyl



3.688
3,5-dimethoxyphenyl
CN



3.689
3,5-dimethoxyphenyl
vinyl



3.690
3,5-dimethoxyphenyl
fluoromethyl



3.691
3,5-dimethoxyphenyl
hydroxymethyl



3.692
3,5-dimethoxyphenyl
ethynyl



3.693
3-ethoxy-5-methoxyphenyl
methyl



3.694
3-n-propoxy-5-methoxyphenyl
methyl



3.695
3-isobutoxy-5-methoxyphenyl
methyl



3.696
3-difluoromethoxy-5-methoxyphenyl
methyl



3.697
3-trifluoromethoxy-5-methoxyphenyl
methyl



3.698
3-nitro-5-methoxyphenyl
methyl



3.699
3-acetoxy-5-methoxyphenyl
methyl



3.700
3-methylsulfanyl-5-methoxyphenyl
methyl



3.701
3,5-diethoxyphenyl
methyl



3.702
3-n-propoxy-5-ethoxyphenyl
methyl



3.703
3-n-butoxy-5-ethoxyphenyl
methyl



3.704
3-isobutoxy-5-ethoxyphenyl
methyl



3.705
3-difluoromethoxy-5-ethoxyphenyl
methyl



3.706
3-trifluoromethoxy-5-ethoxyphenyl
methyl



3.707
3-nitro-5-ethoxyphenyl
methyl



3.708
3-acetoxy-5-ethoxyphenyl
methyl



3.709
3-methylsulfanyl-5-ethoxyphenyl
methyl



3.710
3,5-di(isopropoxy)phenyl
methyl



3.711
3-isobutoxy-5-isopropoxyphenyl
methyl



3.712
3-difluoromethoxy-5-isopropoxyphenyl
methyl



3.713
3-trifluoromethoxy-5-isopropoxyphenyl
methyl



3.714
3-nitro-5-isopropoxyphenyl
methyl



3.715
3-acetoxy-5-isopropoxyphenyl
methyl



3.716
3-methylsulfanyl-5-isopropoxyphenyl
methyl



3.717
3,5-di(trifluoro-methoxy)phenyl
methyl



3.718
3-nitro-5-trifluoro-methoxyphenyl
methyl



3.719
3-methylsulfany1-5-trifluoromethoxy-
methyl




phenyl




3.720
3,5-bis(difluoro-methoxy)phenyl
methyl



3.721
3-nitro-5-difluoro-methoxyphenyl
methyl



3.722
3-acetoxy-5-difluoromethoxyphenyl
methyl



3.723
3-methylsulfanyl-5-acetoxyphenyl
methyl



3.724
3-acetoxy-5-nitrophenyl
methyl



3.725
3-methylsulfanyl-5-nitrophenyl
methyl



3.726
3,5-di(methylsulfanyl)phenyl
methyl



3.727
3,4-difluorophenyl
methyl



3.728
3,4-difluorophenyl
ethyl



3.729
3,4-difluorophenyl
CN



3.730
3,4-difluorophenyl
vinyl



3.731
3,4-difluorophenyl
fluoromethyl



3.732
3,4-difluorophenyl
hydroxymethyl



3.733
3,4-difluorophenyl
ethynyl



3.734
3-chloro-4-fluorophenyl
methyl



3.735
3-bromo-4-fluorophenyl
methyl



3.736
3-methyl-4-fluorophenyl
methyl



3.737
3-methyl-4-fluorophenyl
ethyl



3.738
3-methyl-4-fluorophenyl
CN



3.739
3-methyl-4-fluorophenyl
vinyl



3.740
3-methyl-4-fluorophenyl
fluoromethyl



3.741
3-methyl-4-fluorophenyl
hydroxymethyl



3.742
3-methyl-4-fluorophenyl
ethynyl



3.743
3-ethyl-4-fluorophenyl
methyl



3.744
3-cyclopropyl-4-fluorophenyl
methyl



3.745
3-cyano-4-fluorophenyl
methyl



3.746
3-methoxy-4-fluorophenyl
methyl



3.747
3-ethoxy-4-fluorophenyl
methyl



3.748
3-trifluoromethoxy-4-fluorophenyl
methyl



3.749
3-nitro-4-fluorophenyl
methyl



3.750
3-fluoro-4-chlorophenyl
methyl



3.751
3,4-dichlorophenyl
methyl
[CDCl3] 1.92 (s, 3H),





3.38 (d, 1H), 3.82 (d,





1H), 7.5 (m, 2H), 7.7





(d, 1H).


3.752
3,4-dichlorophenyl
tert-butyl
[DMSO] 1.10 (s, 9H);





4.2 (dd, 2H); 7.75 (m,





2H); 7.95 (d, 1H).


3.753
3-,4-dichlorophenyl
isopropyl
[DMSO] 1.09 (2d; 6H);





2.28 (m, 1H); 3.85 (d,





1H); 4.10 (d, 1H); 7.72





(dd, 1H); 7.78 (d, 1H);





7.93 (d, 1H).


3.754
3-cyclopropyl-4-chlorophenyl
methyl



3.755
3-cyano-4-chlorophenyl
methyl



3.756
3-trifluoromethyl-4-chlorophenyl
methyl



3.757
3-methoxy-4-chlorophenyl
methyl



3.758
3-ethoxy-4-chlorophenyl
methyl



3.759
3-trifluoromethoxy-4-chlorophenyl
methyl



3.760
3-nitro-4-chlorophenyl
methyl



3.761
3-fluoro-4-bromophenyl
methyl



3.762
3-chloro-4-bromophenyl
methyl



3.763
3,4-dibromophenyl
methyl



3.764
3-methyl-4-bromophenyl
methyl



3.765
3-cyclopropyl-4-bromophenyl
methyl



3.766
3-cyano-4-bromophenyl
methyl



3.767
3-trifluoromethyl-4-bromophenyl
methyl



3.768
3-methoxy-4-phenyl
methyl



3.769
3-ethoxy-4-bromophenyl
methyl



3.770
3-trifluoromethoxy-4-bromophenyl
methyl



3.771
3-nitro-4-bromophenyl
methyl



3.772
3-fluoro-4-iodophenyl
methyl



3.773
3-chloro-4-iodophenyl
methyl



3.774
3-bromo-4-iodophenyl
methyl



3.775
3-methyl-4-iodophenyl
methyl



3.776
3-cyclopropyl-4-iodophenyl
methyl



3.777
3-cyano-4-iodophenyl
methyl



3.778
3-trifluoromethyl-4-iodophenyl
methyl



3.779
3-methoxy-4-iodophenyl
methyl



3.780
3-ethoxy-4-iodophenyl
methyl



3.781
3-trifluoromethoxy-4-iodophenyl
methyl



3.782
3-nitro-4-iodophenyl
methyl



3.783
3-fluoro-4-methylphenyl
methyl



3.784
3-chloro-4-methylphenyl
methyl



3.785
3-chloro-4-methylphenyl
ethyl



3.786
3-chloro-4-methylphenyl
CN



3.787
3-chloro-4-methylphenyl
vinyl



3.788
3-chloro-4-methylphenyl
fluoromethyl



3.789
3-chloro-4-methylphenyl
hydroxymethyl



3.790
3-chloro-4-methylphenyl
ethynyl



3.791
3-bromo-4-methylphenyl
methyl



3.792
3,4-dimethylphenyl
methyl



3.793
3-cyclopropyl-4-methylphenyl
methyl



3.794
3-cyano-4-methylphenyl
methyl



3.795
3-trifluoromethyl-4-methylphenyl
methyl



3.796
3-methoxy-4-methylphenyl
methyl



3.797
3-ethoxy-4-methylphenyl
methyl



3.798
3-trifluoromethoxy-4-methylphenyl
methyl



3.799
3-nitro-4-methylphenyl
methyl



3.800
3-fluoro-4-ethylphenyl
methyl



3.801
3-chloro-4-ethylphenyl
methyl



3.802
3-bromo-4-ethylphenyl
methyl



3.803
3-methyl-4-ethylphenyl
methyl



3.804
3,4-diethylphenyl
methyl



3.805
3-cyclopropyl-4-ethylphenyl
methyl



3.806
3-cyano-4-ethylphenyl
methyl



3.807
3-trifluoromethyl-4-ethylphenyl
methyl



3.808
3-methoxy-4-ethylphenyl
methyl



3.809
3-ethoxy-4-ethylphenyl
methyl



3.810
3-trifluoromethoxy-4-ethylphenyl
methyl



3.811
3-nitro-4-ethylphenyl
methyl



3.812
3-fluoro-4-propylphenyl
methyl



3.813
3-chloro-4-propylphenyl
methyl



3.814
3-bromo-4-propylphenyl
methyl



3.815
3-methyl-4-propylphenyl
methyl



3.816
3-cyclopropyl-4-propylphenyl
methyl



3.817
3-cyano-4-propylphenyl
methyl



3.818
3-trifluoromethyl-4-propylphenyl
methyl



3.819
3-methoxy-4-propylphenyl
methyl



3.820
3-ethoxy-4-propylphenyl
methyl



3.821
3-trifluoromethoxy-4-propylphenyl
methyl



3.822
3-nitro-4-propylphenyl
methyl



3.823
3-fluoro-4-isopropylphenyl
methyl



3.824
3-chloro-4-isopropylphenyl
methyl



3.825
3-bromo-4- isopropylphenyl
methyl



3.826
3-methyl-4-isopropylphenyl
methyl



3.827
3-cyclopropyl-4-isopropylphenyl
methyl



3.828
3-cyano-4-isopropylphenyl
methyl



3.829
3-trifluoromethyl-4-isopropylphenyl
methyl



3.830
3- methoxy-4-isopropylphenyl
methyl



3.831
3-ethoxy-4-isopropylphenyl
methyl



3.832
3-trifluoromethoxy-4-isopropylphenyl
methyl



3.833
3-nitro-4-isopropylphenyl
methyl



3.834
3-fluoro-4-tert-butylphenyl
methyl



3.835
3-fluoro-4-tert-butylphenyl
ethyl



3.836
3-fluoro-4-tert-butylphenyl
CN



3.837
3-fluoro-4-tert-butylphenyl
vinyl



3.838
3-fluoro-4-tert-butylphenyl
fluoromethyl



3.839
3-fluoro-4-tert-butylphenyl
hydroxymethyl



3.840
3-fluoro-4-tert-butylphenyl
ethynyl



3.841
3-chloro-4-tert-butylphenyl
methyl



3.842
3-bromo-4-tert-butylphenyl
methyl



3.843
3-methyl-4-tert-butylphenyl
methyl



3.844
3-ethyl-4-tert-butylphenyl
methyl



3.845
3-cyclopropyl-4-tert-butylphenyl
methyl



3.846
3-cyano-4-tert-butylphenyl
methyl



3.847
3-trifluoromethyl-4-tert-butylphenyl
methyl



3.848
3-methoxy-4-tert-butylphenyl
methyl



3.849
3-ethoxy-4-tert-butylphenyl
methyl



3.850
3-trifluoromethoxy-4-tert-butylphenyl
methyl



3.851
3-nitro-4-tert-butylphenyl
methyl



3.852
3-fluoro-4-cyclopropylphenyl
methyl



3.853
3-chloro-4-cyclopropylphenyl
methyl



3.854
3-bromo-4-cyclopropylphenyl
methyl



3.855
3-methyl-4-cyclopropylphenyl
methyl



3.856
3-cyclopropyl-4-cyclopropylphenyl
methyl



3.857
3-cyano-4-cyclopropylphenyl
methyl



3.858
3-trifluoromethyl-4-cyclopropylphenyl
methyl



3.859
3-methoxy-4-cyclopropylphenyl
methyl



3.860
3-ethoxy-4-cyclopropylphenyl
methyl



3.861
3-trifluoromethoxy-4-cyclopropylphenyl
methyl



3.862
3-fluoro-4-methoxycarbonyl-phenyl
methyl



3.863
3-chloro-4-methoxycarbonylphenyl
methyl



3.864
3-bromo-4-methoxycarbonylphenyl
methyl



3.865
3-methyl-4-methoxycarbonylphenyl
methyl



3.866
3-cyclopropyl-4-methoxycarbonylphenyl 
methyl



3.867
3-cyano-4-methoxycarbonylphenyl
methyl



3.868
3-trifluoromethyl-4-methoxycarbonyl-
methyl




phenyl




3.869
3-methoxy-4-methoxycarbonylphenyl
methyl



3.870
3-ethoxy-4-methoxycarbonylphenyl
methyl



3.871
3-nitro-4-methoxycarbonylphenyl
methyl



3.872
3-fluoro-4-cyanophenyl
methyl



3.873
3-chloro-4-cyanophenyl
methyl



3.874
3-bromo-4-cyanophenyl
methyl



3.875
3-methyl-4-cyanophenyl
methyl



3.876
3-cyclopropyl-4-cyanophenyl
methyl



3.877
3-cyano-4-cyanophenyl
methyl



3.878
3-trifluoromethyl-4-cyanophenyl
methyl



3.879
3-methoxy-4-cyanophenyl
methyl



3.880
3-ethoxy-4-cyanophenyl
methyl



3.881
3-trifluoromethoxy-4-cyanophenyl
methyl



3.882
3-nitro-4-cyanophenyl
methyl



3.883
3-fluoro-4-methoxyphenyl
methyl



3.884
3-chloro-4-methoxyphenyl
methyl



3.885
3-bromo-4-methoxyphenyl
methyl



3.886
3-methyl-4-methoxyphenyl
methyl



3.887
3-cyclopropyl-4-methoxyphenyl
methyl



3.888
3-cyano-4-methoxyphenyl
methyl



3.889
3-trifluoromethyl-4-methoxyphenyl
methyl



3.890
3,4-dimethoxyphenyl
methyl



3.891
3-ethoxy-4-methoxyphenyl
methyl



3.892
3-trifluoromethoxy-4-methoxyphenyl
methyl



3.893
3-nitro-4-methoxyphenyl
methyl



3.894
3-fluoro-4-ethoxyphenyl
methyl



3.895
3-chloro-4-ethoxyphenyl
methyl



3.896
3-bromo-4-ethoxyphenyl
methyl



3.897
3-methyl-4-ethoxyphenyl
methyl



3.898
3-cyclopropyl-4-ethoxyphenyl
methyl



3.899
3-cyano-4-ethoxyphenyl
methyl



3.900
3-trifluoromethyl-4-ethoxyphenyl
methyl



3.901
3-methoxy-4-ethoxyphenyl
methyl



3.902
2,4-diethoxyphenyl
methyl



3.903
3-trifluoromethoxy-4-ethoxyphenyl
methyl



3.904
3-nitro-4-ethoxyphenyl
methyl



3.905
3-fluoro-4-isopropoxyphenyl
methyl



3.906
3-chloro-4-isopropoxyphenyl
methyl



3.907
3-bromo-4-isopropoxyphenyl
methyl



3.908
3-methy1-4-isopropoxyphenyl
methyl



3.909
3-cyclopropyl-4-isopropoxyphenyl
methyl



3.910
3-cyano-4-isopropoxyphenyl
methyl



3.911
3-trifluoromethyl-4-isopropoxyphenyl
methyl



3.912
3-methoxy-4-isopropoxyphenyl
methyl



3.913
3-ethoxy-4-isopropoxyphenyl
methyl



3.914
3-trifluoromethoxy-4-isopropoxyphenyl
methyl



3.915
3-nitro-4-isopropoxyphenyl
methyl



3.916
3-fluoro-4-trifluoromethoxyphenyl
methyl



3.917
3-chloro-4-trifluoromethoxyphenyl
methyl



3.918
3-bromo-4-trifluoromethoxyphenyl
methyl



3.919
3-methyl-4-trifluoromethoxyphenyl
methyl



3.920
3-ethyl-4-trifluoromethoxyphenyl
methyl



3.921
3-cyclopropyl-4-trifluoromethoxyphenyl
methyl



3.922
3-cyano-4-trifluoromethoxyphenyl
methyl



3.923
3-trifluoromethyl-4-trifluoromethoxy-
methyl




phenyl




3.924
3-methoxy-4-trifluoromethoxyphenyl
methyl



3.925
3-ethoxy-4-trifluoro-methoxyphenyl
methyl



3.926
3,4-bis(trifluoro-methoxy)phenyl
methyl



3.927
3-nitro-4-trifluoro- methoxyphenyl
methyl



3.928
3-fluoro-4-difluoromethoxyphenyl
methyl



3.929
3-chloro-4-difluoromethoxyphenyl
methyl



3.930
3-bromo-4-difluoromethoxyphenyl
methyl



3.931
3-methyl-4-difluoromethoxyphenyl
methyl



3.932
3-cyclopropyl-4-difluoromethoxyphenyl
methyl



3.933
3-cyano-4-difluoromethoxyphenyl
methyl



3.934
3-trifluoromethyl-4-difluoromethoxyphenyl
methyl



3.935
3-methoxy-4-difluoromethoxyphenyl
methyl



3.936
3-ethoxy-4-difluoromethoxyphenyl
methyl



3.937
3-nitro-4-difluoromethoxyphenyl
methyl



3.938
3-fluoro-4-nitrophenyl
methyl



3.939
3-chloro-4-nitrophenyl
methyl



3.940
3-bromo-4-nitrophenyl
methyl



3.941
3-methyl-4-nitrophenyl
methyl



3.942
3-cyclopropyl-4-nitrophenyl
methyl



3.943
3-cyano-4-nitrophenyl
methyl



3.944
3-trifluoromethyl-4-nitrophenyl
methyl



3.945
3-methoxy-4-nitrophenyl
methyl



3.946
3-ethoxy-4-nitrophenyl
methyl



3.947
3-trifluoromethoxy-4-nitrophenyl
methyl



3.948
3-fluoro-4-methylsulfanylphenyl
methyl



3.949
3-chloro-4-methylsulfanylphenyl
methyl



3.950
3-bromo-4-methylsulfanylphenyl
methyl



3.951
3-methyl-4-methylsulfanylphenyl
methyl



3.952
3-cyclopropyl-4-methylsulfanylphenyl
methyl



3.953
3-cyano-4-methylsulfanylphenyl
methyl



3.954
3-trifluoromethyl-4-methylsulfanylphenyl
methyl



3.955
3-methoxy-4-methylsulfanylphenyl
methyl



3.956
3-ethoxy-4-methylsulfanylphenyl
methyl



3.957
3-trifluoromethoxy-4-methylsulfanylphenyl
methyl



3.958
3-nitro-4-methylsulfanylphenyl
methyl



3.959
3,6-difluorophenyl
methyl



3.960
3,6-difluorophenyl
ethyl



3.961
3,6-difluorophenyl
CN



3.962
3,6-difluorophenyl
vinyl



3.963
3,6-difluorophenyl
fluoromethyl



3.964
3,6-difluorophenyl
hydroxymethyl



3.965
3,6-difluorophenyl
ethynyl



3.966
3-chloro-6-fluorophenyl
methyl



3.967
3-bromo-6-fluorophenyl
methyl



3.968
3-methyl-6-fluorophenyl
methyl



3.969
3-cyclopropyl-6-fluorophenyl
methyl



3.970
3-cyano-6-fluorophenyl
methyl



3.971
3-methoxy-6-fluorophenyl
methyl



3.972
3-ethoxy-6-fluorophenyl
methyl



3.973
3-trifluoromethoxy-6-fluorophenyl
methyl



3.974
3-nitro-6-fluorophenyl
methyl



3.975
3-fluoro-6-chlorophenyl
methyl



3.976
3,6-dichlorophenyl
methyl



3.977
3-bromo-6-chlorophenyl
methyl



3.978
3-methyl-6-chlorophenyl
methyl



3.979
3-cyclopropyl-6-chlorophenyl
methyl



3.980
3-cyano-6-chlorophenyl
methyl



3.981
3-trifluoromethyl-6-chlorophenyl
methyl



3.982
3-methoxy-6-chlorophenyl
methyl



3.983
3-ethoxy-6-chlorophenyl
methyl



3.984
3-trifluoromethoxy-6-chlorophenyl
methyl



3.985
3-nitro-6-chlorophenyl
methyl



3.986
3-fluoro-6-bromophenyl
methyl



3.987
3-chloro-6-bromophenyl
methyl



3.988
3,6-dibromophenyl
methyl



3.989
3-methyl-6-bromophenyl
methyl



3.990
3-ethyl-6-bromophenyl
methyl



3.991
3-cyclopropyl-6-bromophenyl
methyl



3.992
3-cyano-6-bromophenyl
methyl



3.993
3-trifluoromethyl-6-bromophenyl
methyl



3.994
3-methoxy-6-phenyl
methyl



3.995
3-ethoxy-6-bromophenyl
methyl



3.996
3-trifluoromethoxy-6-bromophenyl
methyl



3.997
3-nitro-6-bromophenyl
methyl



3.998
3-fluoro-6-iodophenyl
methyl



3.999
3-chloro-6-iodophenyl
methyl



3.1000
3-bromo-6-iodophenyl
methyl



3.1001
3-methyl-6-iodophenyl
methyl



3.1002
3-cyclopropyl-6-iodophenyl
methyl



3.1003
3-cyano-6-iodophenyl
methyl



3.1004
3-trifluoromethyl-6-iodophenyl
methyl



3.1005
3-methoxy-6-iodophenyl
methyl



3.1006
3-ethoxy-6-iodophenyl
methyl



3.1007
3-trifluoromethoxy-6-iodophenyl
methyl



3.1008
3-nitro-6-iodophenyl
methyl



3.1009
3-fluoro-6-methylphenyl
methyl



3.1010
3-chloro-6-methylphenyl
methyl



3.1011
3-bromo-6-methylphenyl
methyl



3.1012
3,6-dimethylphenyl
methyl



3.1013
3,6-dimethylphenyl
ethyl



3.1014
3,6-dimethylphenyl
CN



3.1015
3,6-dimethylphenyl
vinyl



3.1016
3,6-dimethylphenyl
fluoromethyl



3.1017
3,6-dimethylphenyl
hydroxymethyl



3.1018
3,6-dimethylphenyl
ethynyl



3.1019
3-cyclopropyl-6-methylphenyl
methyl



3.1020
3-cyano-6-methylphenyl
methyl



3.1021
3-trifluoromethyl-6-methylphenyl
methyl



3.1022
3-methoxy-6-methylphenyl
methyl



3.1023
3-ethoxy-6-methylphenyl
methyl



3.1024
3-trifluoromethoxy-6-methylphenyl
methyl



3.1025
3-nitro-6-methylphenyl
methyl



3.1026
3-fluoro-6-ethylphenyl
methyl



3.1027
3-chloro-6-ethylphenyl
methyl



3.1028
3-bromo-6-ethylphenyl
methyl



3.1029
3-methyl-6-ethylphenyl
methyl



3.1030
3,6-diethylphenyl
methyl



3.1031
3-cyclopropyl-6-ethylphenyl
methyl



3.1032
3-cyano-6-ethylphenyl
methyl



3.1033
3-trifluoromethyl-6-ethylphenyl
methyl



3.1034
3-methoxy-6-ethylphenyl
methyl



3.1035
3-ethoxy-6-ethylphenyl
methyl



3.1036
3-trifluoromethoxy-6-ethylphenyl
methyl



3.1037
3-nitro-6-ethylphenyl
methyl



3.1038
3-fluoro-6-isopropylphenyl
methyl



3.1039
3-chloro-6-isopropylphenyl
methyl



3.1040
3-bromo-6-isopropylphenyl
methyl



3.1041
3-methyl-6-isopropylphenyl
methyl



3.1042
3-cyclopropyl-6-isopropylphenyl
methyl



3.1043
3-cyano-6-isopropylphenyl
methyl



3.1044
3-trifluoromethyl-6-isopropylphenyl
methyl



3.1045
3-methoxy-6-isopropylphenyl
methyl



3.1046
3-ethoxy-6-isopropylphenyl
methyl



3.1047
3-trifluoromethoxy-6-isopropylphenyl
methyl



3.1048
3-nitro-6-isopropylphenyl
methyl



3.1049
3-fluoro-6-tert-butylphenyl
methyl



3.1050
3-chloro-6-tert-butylphenyl
methyl



3.1051
3-bromo-6-tert-butylphenyl
methyl



3.1052
3-methyl-6-tert-butylphenyl
methyl



3.1053
3-cyclopropyl-6-tert-butylphenyl
methyl



3.1054
3-cyano-6-tert-butylphenyl
methyl



3.1055
3-trifluoromethyl-6-tert-butylphenyl
methyl



3.1056
3-methoxy-6-tert-butylphenyl
methyl



3.1057
3-ethoxy-6-tert-butylphenyl
methyl



3.1058
3-trifluoromethoxy-6-tert-butylphenyl
methyl



3.1059
3-nitro-6-tert-butylphenyl
methyl



3.1060
3-fluoro-6-cyclopropylphenyl
methyl



3.1061
3-chloro-6-cyclopropylphenyl
methyl



3.1062
3-bromo-6-cyclopropylphenyl
methyl



3.1063
3-methyl-6-cyclopropylphenyl
methyl



3.1064
3-ethyl-6-cyclopropylphenyl
methyl



3.1065
3-cyclopropyl-6-cyclopropylphenyl
methyl



3.1066
3-cyano-6-cyclopropylphenyl
methyl



3.1067
3-trifluoromethyl-6-cyclopropylphenyl
methyl



3.1068
3-methoxy-6-cyclopropylphenyl
methyl



3.1069
3-ethoxy-6-cyclopropylphenyl
methyl



3.1070
3-trifluoromethoxy-6-cyclopropylphenyl
methyl



3.1071
3-fluoro-6-methoxycarbonylphenyl
methyl



3.1072
3-chloro-6-methoxycarbonylphenyl
methyl



3.1073
3-bromo-6-methoxycarbonylphenyl
methyl



3.1074
3-methyl-6-methoxycarbonylphenyl
methyl



3.1075
3-cyclopropyl-6-methoxycarbonylphenyl
methyl



3.1077
3-trifluoromethyl-6-methoxycarbonyl-
methyl




phenyl




3.1076
3-cyano-6-methoxycarbonylphenyl
methyl



3.1078
3-methoxy-6-methoxycarbonylphenyl
methyl



3.1079
3-ethoxy-6-methoxycarbonylphenyl
methyl



3.1080
3-trifluoromethoxy-6-methoxycarbonyl-
methyl




phenyl




3.1081
3-nitro-6-methoxycarbonylphenyl
methyl



3.1082
3-fluoro-6-cyanophenyl
methyl



3.1083
3-chloro-6-cyanophenyl
methyl



3.1084
3-bromo-6-cyanophenyl
methyl



3.1085
3-methyl-6-cyanophenyl
methyl



3.1086
3-cyclopropyl-6-cyanophenyl
methyl



3.1087
3-cyano-6-cyanophenyl
methyl



3.1088
3-trifluoromethyl-6-cyanophenyl
methyl



3.1089
3-methoxy-6-cyanophenyl
methyl



3.1090
3-ethoxy-6-cyanophenyl
methyl



3.1091
3-trifluoromethoxy-6-cyanophenyl
methyl



3.1092
3-nitro-6-cyanophenyl
methyl



3.1093
3-fluoro-6-methoxyphenyl
methyl



3.1094
3-chloro-6-methoxyphenyl
methyl



3.1095
3-bromo-6-methoxyphenyl
methyl



3.1096
3-methyl-6-methoxyphenyl
methyl



3.1097
3-cyclopropyl-6-methoxyphenyl
methyl



3.1098
3-cyano-6-methoxyphenyl
methyl



3.1099
3-trifluoromethyl-6-methoxyphenyl
methyl



3.1100
3,6-dimethoxy--phenyl
methyl



3.1101
3-ethoxy-6-methoxyphenyl
methyl



3.1102
3-trifluoromethoxy-6-methoxyphenyl
methyl



3.1103
3- nitro-6-methoxyphenyl
methyl



3.1104
3-fluoro-6-ethoxyphenyl
methyl



3.1105
3-chloro-6-ethoxyphenyl
methyl



3.1106
3-bromo-6-ethoxyphenyl
methyl



3.1107
3-methyl-6-ethoxyphenyl
methyl



3.1108
3-cyclopropyl-6-ethoxyphenyl
methyl



3.1109
3-cyano-6-ethoxyphenyl
methyl



3.1110
3-trifluoromethyl-6-ethoxyphenyl
methyl



3.1111
3-methoxy-6-ethoxyphenyl
methyl



3.1112
2,6-diethoxyphenyl
methyl



3.1113
3-trifluoromethoxy-6-ethoxyphenyl
methyl



3.1114
3-nitro-6-ethoxyphenyl
methyl



3.1115
3-fluoro-6-isopropoxyphenyl
methyl



3.1116
3-chloro-6-isopropoxyphenyl
methyl



3.1117
3-bromo-6-isopropoxyphenyl
methyl



3.1118
3-methy1-6-isopropoxyphenyl
methyl



3.1119
3-cyclopropyl-6-isopropoxyphenyl
methyl



3.1120
3-cyano-6-isopropoxyphenyl
methyl



3.1121
3-trifluoromethyl-6-isopropoxyphenyl
methyl



3.1122
3-methoxy-6-isopropoxyphenyl
methyl



3.1123
3-ethoxy-6-isopropoxyphenyl
methyl



3.1124
3-trifluoromethoxy-6-isopropoxyphenyl
methyl



3.1125
3-nitro-6-isopropoxyphenyl
methyl



3.1126
3-fluoro-6-trifluoromethoxyphenyl
methyl



3.1127
3-chloro-6-trifluoromethoxyphenyl
methyl



3.1128
3-bromo-6-trifl uoromethoxyphenyl
methyl



3.1129
3-methyl-6-trifluoromethoxyphenyl
methyl



3.1130
3-ethyl-6-trifluoromethoxyphenyl
methyl



3.1131
3-cyclopropyl-6-trifluoromethoxyphenyl
methyl



3.1132
3-cyano-6-trifluoromethoxyphenyl
methyl



3.1133
3-trifluoromethyl-6-trifluoromethoxy-
methyl




phenyl




3.1134
3-methoxy-6-trifluoromethoxyphenyl
methyl



3.1135
3-ethoxy-6-trifluoromethoxyphenyl
methyl



3.1136
3,6-bis(trifluoro-methoxy)phenyl
methyl



3.1137
3-nitro-6-trifluoromethoxyphenyl
methyl



3.1138
3-fluoro-6-difluoromethoxyphenyl
methyl



3.1139
3-chloro-6-difluoromethoxyphenyl
methyl



3.1140
3-bromo-6-difluoromethoxyphenyl
methyl



3.1141
3-methyl-6-difluoromethoxyphenyl
methyl



3.1142
3-cyclopropyl-6-difluoromethoxyphenyl
methyl



3.1143
3-cyano-6-difluoromethoxyphenyl
methyl



3.1144
3-trifluoromethyl-6-difluoromethoxyphenyl
methyl



3.1145
3-methoxy-6-difluoromethoxyphenyl
methyl



3.1146
3-ethoxy-6-difluoromethoxyphenyl
methyl



3.1147
3-nitro-6-difluoromethoxyphenyl
methyl



3.1148
3-fluoro-6-nitrophenyl
methyl



3.1149
3-chloro-6-nitrophenyl
methyl



3.1150
3-bromo-6-nitrophenyl
methyl



3.1151
3-methyl-6-nitrophenyl
methyl



3.1152
3-ethyl-6-nitrophenyl
methyl



3.1153
3-cyclopropyl-6-nitrophenyl
methyl



3.1154
3-cyano-6-nitrophenyl
methyl



3.1155
3-trifluoromethyl-6-nitrophenyl
methyl



3.1156
3-methoxy-6-nitrophenyl
methyl



3.1157
3-ethoxy-6-nitrophenyl
methyl



3.1158
3-trifluoromethoxy-6-nitrophenyl
methyl



3.1159
3-fluoro-6-methylsulfanylphenyl
methyl



3.1160
3-chloro-6-methylsulfanylphenyl
methyl



3.1161
3-bromo-6-methylsulfanylphenyl
methyl



3.1162
3-methyl-6-methylsulfanylphenyl
methyl



3.1163
3-cyclopropyl-6-methylsulfanylphenyl
methyl



3.1164
3-cyano-6-methylsulfanylphenyl
methyl



3.1165
3-trifluoromethyl-6-methylsulfanylphenyl 
methyl



3.1166
3-methoxy-6-methylsulfanylphenyl
methyl



3.1167
3-ethoxy-6-methylsulfanylphenyl
methyl



3.1168
3-trifluoromethoxy-6-methylsulfanylphenyl 
methyl



3.1169
3-nitro-6-methylsulfanylphenyl
methyl



3.1170
2,3,4-trifluorophenyl
methyl



3.1171
2,3,4-trichlorophenyl
methyl



3.1172
2,3,4-trimethylphenyl
methyl



3.1173
2-fluoro-2-chloro-5-trifluoromethylphenyl
methyl



3.1174
2,3,5-trifluorophenyl
methyl



3.1175
2,3,5-trichlorophenyl
methyl
[CDCl3] 1.92 (s, 3H);





3.40 (d, 1H); 3.95 (d,





1H); 7.58 (s, 1H); 7.85





(s, 1H)


3.1176
2,3,5-trichlorophenyl
isopropyl
[DMSO] 1.10 (2d, 6H);





2.30 (m, 1H); 3.89 (d,





1H); 4.08 (d, 1H).


3.1177
2,3,5-trichlorophenyl
tert-butyl
[CDCl3] 1.17 (s, 9H);





3.73 (dd, 2H); 7.57 (s,





1H); 7.80 (s, 1H)


3.1178
2,3,6-trifluorophenyl
methyl



3.1179
2,3,6-trichlorophenyl
methyl



3.1180
2,3,6-trimethylphenyl
methyl



3.1181
3,4,5-trifluorophenyl
methyl



3.1182
3,4,6-trifluorophenyl
methyl



3.1183
3,4,6-trichlorophenyl
methyl
[CDCl3] 1.94 (s, 3H),





3.51 (d, 1H), 3.95 (d,





1H), 7.58 (s, 1H), 7.83





(s, 1H).


3.1184
3,4,6-trichlorophenyl
ethyl



3.1185
3,4,6-trichlorophenyl
CN



3.1186
3,4,6-trichlorophenyl
vinyl



3.1187
3,4,6-trichlorophenyl
fluoromethyl



3.1188
3,4,6-trichlorophenyl
hydroxymethyl



3.1189
3,4,6-trichlorophenyl
ethynyl



3.1190
3,4,5-trimethylphenyl
methyl



3.1191
3,5-dimethyl-4-fluorophenyl
methyl



3.1192
3,5-dichloro-4-methoxyphenyl
methyl



3.1193
3,5-difluoro-4-chlorophenyl
methyl



3.1194
3,5-dichloro-4-hydroxyphenyl
methyl



3.1195
3,5-trifluoromethyl-4-chlorophenyl
methyl



3.1196
3,4,6-trifluorophenyl
methyl



3.1197
3,4,6-trichlorophenyl
methyl



3.1198
3,4,6-trimethylphenyl
methyl



3.1199
2,3,4,5-pentafluoro-phenyl
methyl
















TABLE 4







Inventive compounds of the general formula (I) in which W* is CHO, R1


and R2 are each hydrogen, and aryl is the radical.








 








 










No.
Aryl
R3
Physical data





4.1
3-fluorophenyl
methyl



4.2
3-fluorophenyl
ethyl



4.3
3-fluorophenyl
CN



4.4
3-fluorophenyl
fluoromethyl



4.5
3-fluorophenyl
methylcarbonyl



4.6
3-fluorophenyl
hydroxymethyl



4.7
3-fluorophenyl
vinyl



4.8
3-fluorophenyl
1-chlorovinyl



4.9
3-fluorophenyl
ethynyl



4.10
3-chlorophenyl
methyl



4.11
3-chlorophenyl
ethyl



4.12
3-chlorophenyl
CN



4.13
3-chlorophenyl
fluoromethyl



4.14
3-chlorophenyl
hydroxymethyl



4.15
3-chlorophenyl
methylcarbonyl



4.16
3-chlorophenyl
fluoromethyl



4.17
3-chlorophenyl
ethynyl



4.18
3-bromophenyl
methyl



4.19
3-bromophenyl
ethyl



4.20
3-bromophenyl
vinyl



4.21
3-iodophenyl
methyl



4.22
3-methylphenyl
methyl



4.23
3-ethylphenyl
methyl



4.24
3-propylphenyl
methyl



4.25
3-isopropylphenyl
methyl



4.26
3-n-butylphenyl
methyl



4.27
3-i-butylphenyl
methyl



4.28
3-tert-butylphenyl
methyl



4.29
3-cyclopropylphenyl
methyl



4.30
3-cyclobutylphenyl
methyl



4.31
3-cyclopentylphenyl
methyl



4.32
3-vinylphenyl
methyl



4.33
3-ethynylphenyl
methyl



4.34
3-cyanophenyl
methyl



4.35
3-trifluoromethylphenyl
methyl



4.36
3-difluoromethylphenyl
methyl



4.37
3-(methoxycarbonyl)phenyl
methyl



4.38
3-(ethoxycarbonyl)phenyl
methyl



4.39
3-hydroxymethylphenyl
methyl



4.40
3-methoxyphenyl
methyl



4.41
3-methoxyphenyl
ethyl



4.42
3-methoxyphenyl
CN



4.43
3-methoxyphenyl
fluoromethyl



4.44
3-methoxyphenyl
methylcarbonyl



4.45
3-methoxyphenyl
hydroxymethyl



4.46
3-methoxyphenyl
ethynyl



4.47
3-ethoxyphenyl
methyl



4.48
3-propyloxyphenyl
methyl



4.49
3-isopropyloxyphenyl
methyl



4.50
3-i-butyloxyphenyl
methyl



4.51
3-t-butyloxyphenyl
methyl



4.52
3-difluoromethoxyphenyl
methyl



4.53
3-trifluoromethoxyphenyl
methyl



4.54
3-trifluoromethoxyphenyl
ethyl



4.55
3-trifluoromethoxyphenyl
CN



4.56
3-trifluoromethoxyphenyl
fluoromethyl



4.57
3-trifluoromethoxyphenyl
methylcarbonyl



4.58
3-trifluoromethoxy
hydroxymethyl



4.59
3-trifluoromethoxyphenyl
ethynyl



4.60
3-nitrophenyl
methyl



4.61
3-acetoxyphenyl
methyl



4.62
3-methylsulfanylphenyl
methyl



4.63
3-ethylsulfanylphenyl
methyl



4.64
3-(pentafluoro-lambda6-sulfanyl)phenyl
methyl



4.65
2,3-difluorophenyl
methyl



4.66
2,3-difluorophenyl
ethyl



4.67
2,3-difluorophenyl
CN



4.68
2,3-difluorophenyl
fluoromethyl



4.69
2,3-difluorophenyl
methylcarbonyl



4.70
2,3-difluorophenyl
hydroxymethyl



4.71
2,3-difluorophenyl
ethynyl



4.72
2-chloro-3-fluorophenyl
methyl



4.73
2-bromo-3-fluorophenyl
methyl



4.74
2-methyl-3-fluorophenyl
methyl



4.75
2-ethyl-3-fluorophenyl
methyl



4.76
2-cyclopropyl-3-fluorophenyl
methyl



4.77
2-cyano-3-fluorophenyl
methyl



4.78
2-methoxy-3-fluorophenyl
methyl



4.79
2-trifluoromethoxy-3-fluorophenyl
methyl



4.80
2-nitro-3-fluorophenyl
methyl



4.81
2-fluoro-3-chlorophenyl
methyl



4.82
2,3-dichlorophenyl
methyl



4.83
2,3-dichlorophenyl
ethyl



4.84
2,3-dichlorophenyl
CN



4.85
2,3-dichlorophenyl
fluoromethyl



4.86
2,3-dichlorophenyl
methylcarbonyl



4.87
2,3-dichlorophenyl
hydroxymethyl



4.88
2,3-dichlorophenyl
ethynyl



4.89
2-bromo-3-chlorophenyl
methyl



4.90
2-methyl-3-chlorophenyl
methyl



4.91
2-methyl-3-chlorophenyl
ethyl



4.92
2-methyl-3-chlorophenyl
CN



4.93
2-methyl-3-chlorophenyl
fluoromethyl



4.94
2-methyl-3-chlorophenyl
methylcarbonyl



4.95
2-methyl-3-chlorophenyl
hydroxymethyl



4.96
2-methyl-3-chlorophenyl
ethynyl



4.97
2-ethyl-3-chlorophenyl
methyl



4.98
2-cyclopropyl-3-chlorophenyl
methyl



4.99
2-cyano-3-chlorophenyl
methyl



4.100
2-trifluoromethyl-2-chlorophenyl
methyl



4.101
2-methoxy-3-chlorophenyl
methyl



4.102
2-ethoxy-3-chlorophenyl
methyl



4.103
2-trifluoromethoxy-3-chlorophenyl
methyl



4.104
2-nitro-3-chlorophenyl
methyl



4.105
2-fluoro-3-bromophenyl
methyl



4.106
2-chloro-3-bromophenyl
methyl



4.107
2,3-dibromophenyl
methyl



4.108
2-methyl-3-bromophenyl
methyl



4.109
2-ethyl-3-bromophenyl
methyl



4.110
2-cyclopropyl-3-bromophenyl
methyl



4.111
2-cyano-3-bromophenyl
methyl



4.112
2-trifluoromethyl-3-bromophenyl
methyl



4.113
2-methoxy-3-phenyl
methyl



4.114
2-trifluoromethoxy-3-bromophenyl
methyl



4.115
2-nitro-3-bromophenyl
methyl



4.116
2-fluoro-3-iodophenyl
methyl



4.117
2-chloro-3-iodophenyl
methyl



4.118
2-bromo-3-iodophenyl
methyl



4.119
2-methyl-3-iodophenyl
methyl



4.120
2-ethyl-3-iodophenyl
methyl



4.121
2-cyclopropyl-3-iodophenyl
methyl



4.122
2-cyano-3-iodophenyl
methyl



4.123
2-trifluoromethyl-3-iodophenyl
methyl



4.124
2-methoxy-3-iodophenyl
methyl



4.125
2-trifluoromethoxy-3-iodophenyl
methyl



4.126
2-nitro-3-iodophenyl
methyl



4.127
2-fluoro-3-methylphenyl
methyl



4.128
2-fluoro-3-methylphenyl
ethyl



4.129
2-fluoro-3-methylphenyl
CN



4.130
2-fluoro-3-methylphenyl
fluoromethyl



4.131
2-fluoro-3-methylphenyl
hydroxymethyl



4.132
2-fluoro-3-methylphenyl
ethynyl



4.133
2-chloro-3-methylphenyl
methyl



4.134
2-chloro-3-methylphenyl
ethyl



4.135
2-chloro-3-methylphenyl
CN



4.136
2-chloro-3-methylphenyl
fluoromethyl



4.137
2-chloro-3-methylphenyl
methylcarbonyl



4.138
2-chloro-3-methylphenyl
hydroxymethyl



4.139
2-chloro-3-methylphenyl
ethynyl



4.140
2-bromo-3-methylphenyl
methyl



4.141
2,3-dimethylphenyl
methyl



4.142
2-ethyl-3-methylphenyl
methyl



4.143
2-cyclopropyl-3-methylphenyl
methyl



4.144
2-cyano-3-methylphenyl
methyl



4.145
2-trifluoromethyl-3-methylphenyl
methyl



4.146
2-methoxy-3-methylphenyl
methyl



4.147
2-trifluoromethoxy-3-methylphenyl
methyl



4.148
2-nitro-3-methylphenyl
methyl



4.149
2-fluoro-3-ethylphenyl
methyl



4.150
2-chloro-3-ethylphenyl
methyl



4.151
2-bromo-3-ethylphenyl
methyl



4.152
2-methyl-3-ethylphenyl
methyl



4.153
2,3-diethylphenyl
methyl



4.154
2-cyclopropyl-3-ethylphenyl
methyl



4.155
2-cyano-3-ethylphenyl
methyl



4.156
2-trifluoromethyl-3-ethylphenyl
methyl



4.157
2-methoxy-3-ethylphenyl
methyl



4.158
2-trifluoromethoxy-3-ethylphenyl
methyl



4.159
2-nitro-3-ethylphenyl
methyl



4.160
2-fluoro-3-propylphenyl
methyl



4.161
2-chloro-3-propylphenyl
methyl



4.162
2-bromo-3-propylphenyl
methyl



4.163
2-methyl-3-propylphenyl
methyl



4.164
2-methyl-3-propylphenyl
methyl



4.165
2-cyclopropyl-3-propylphenyl
methyl



4.166
2-cyano-3-propylphenyl
methyl



4.167
2-trifluoromethyl-3-propylphenyl
methyl



4.168
2-methoxy-3-propylphenyl
methyl



4.169
2-trifluoromethoxy-3-propylphenyl
methyl



4.170
2-nitro-3-propylphenyl
methyl



4.171
2-fluoro-3-isopropylphenyl
methyl



4.172
2-chloro-3-isopropylphenyl
methyl



4.173
2-bromo-3-isopropylphenyl
methyl



4.174
2-methyl-3-isopropylphenyl
methyl



4.175
2-cyclopropyl-3-isopropylphenyl
methyl



4.176
2-cyano-3-isopropylphenyl
methyl



4.177
2-trifluoromethyl-3-isopropylphenyl
methyl



4.178
2-methoxy-3-isopropylphenyl
methyl



4.179
2-trifluoromethoxy-3-isopropylphenyl
methyl



4.180
2-nitro-3-isopropylphenyl
methyl



4.181
2-fluoro-3-tert-butylphenyl
methyl



4.182
2-fluoro-3-tert-butylphenyl
ethyl



4.183
2-fluoro-3-tert-butylphenyl
CN



4.184
2-fluoro-3-tert-butylphenyl
fluoromethyl



4.185
2-fluoro-3-tert-butylphenyl
methylcarbonyl



4.186
2-fluoro-3-tert-butylphenyl
hydroxymethyl



4.187
2-fluoro-3-tert-butylphenyl
ethynyl



4.188
2-chloro-3-tert-butylphenyl
methyl



4.189
2-bromo-3-tert-butylphenyl
methyl



4.190
2-methyl-3-tert-butylphenyl
methyl



4.191
2-cyclopropyl-3-tert-butylphenyl
methyl



4.192
2-cyano-3-tert-butylphenyl
methyl



4.193
2-trifluoromethyl-3-tert-butylphenyl
methyl



4.194
2-methoxy-3-tert-butylphenyl
methyl



4.195
2-trifluoromethoxy-3-tert-butylphenyl
methyl



4.196
2-nitro-3-tert-butylphenyl
methyl



4.197
2-fluoro-3-cyclopropylphenyl
methyl



4.198
2-chloro-3-cyclopropylphenyl
methyl



4.199
2-bromo-3-cyclopropylphenyl
methyl



4.200
2-methyl-3-cyclopropylphenyl
methyl



4.201
2-cyclopropyl-3-cyclopropylphenyl
methyl



4.202
2-cyano-3-cyclopropylphenyl
methyl



4.203
2-trifluoromethyl-3-cyclopropylphenyl
methyl



4.204
2-methoxy-3-cyclopropylphenyl
methyl



4.205
2-ethoxy-3-cyclopropylphenyl
methyl



4.206
2-trifluoromethoxy-3-cyclopropylphenyl
methyl



4.207
2-fluoro-3-methoxycarbonylphenyl
methyl



4.208
2-chloro-3-methoxycarbonylphenyl
methyl



4.209
2-bromo-3-methoxycarbonylphenyl
methyl



4.210
2-methyl-3-methoxycarbonylphenyl
methyl



4.211
2-methyl-3-methoxycarbonylphenyl
ethyl



4.212
2-methyl-3-methoxycarbonylphenyl
CN



4.213
2-methyl-3-methoxycarbonylphenyl
vinyl



4.214
2-methyl-3-methoxycarbonylphenyl
fluoromethyl



4.215
2-methyl-3-methoxycarbonylphenyl
methylcarbonyl



4.216
2-methyl-3-methoxycarbonylphenyl
hydroxymethyl



4.217
2-methyl-3-methoxycarbonylphenyl
ethynyl



4.218
2-cyclopropyl-3-methoxycarbonylphenyl
methyl



4.219
2-cyano-3-methoxycarbonylphenyl
methyl



4.220
2-trifluoromethyl-3-
methyl




methoxycarbonylphenyl




4.221
2-methoxy-3-methoxycarbonylphenyl
methyl



4.222
2-ethoxy-3-methoxycarbonylphenyl
methyl



4.223
2-trifluoromethoxy-3-
methyl




methoxycarbonylphenyl




4.224
2-nitro-3-methoxycarbonylphenyl
methyl



4.225
2-fluoro-3-cyanophenyl
methyl



4.226
2-fluoro-3-cyanophenyl
ethyl



4.227
2-fluoro-3-cyanophenyl
CN



4.228
2-fluoro-3-cyanophenyl
vinyl



4.229
2-fluoro-3-cyanophenyl
fluoromethyl



4.230
2-fluoro-3-cyanophenyl
methylcarbonyl



4.231
2-fluoro-3-cyanophenyl
hydroxymethyl



4.232
2-fluoro-3-cyanophenyl
ethynyl



4.233
2-chloro-3-cyanophenyl
methyl



4.234
2-chloro-3-cyanophenyl
ethyl



4.235
2-chloro-3-cyanophenyl
CN



4.236
2-chloro-3-cyanophenyl
vinyl



4.237
2-chloro-3-cyanophenyl
fluoromethyl



4.238
2-chloro-3-cyanophenyl
methylcarbonyl



4.239
2-chloro-3-cyanophenyl
hydroxymethyl



4.240
2-chloro-3-cyanophenyl
ethynyl



4.241
2-bromo-3-cyanophenyl
methyl



4.242
2-methyl-3-cyanophenyl
methyl



4.243
2-ethyl-3-cyanophenyl
methyl



4.244
2-cyclopropyl-3-cyanophenyl
methyl



4.245
2-cyano-3-cyanophenyl
methyl



4.246
2-trifluoromethyl-3-cyanophenyl
methyl



4.247
2-methoxy-3-cyanophenyl
methyl



4.248
2-trifluoromethoxy-3-cyanophenyl
methyl



4.249
2-nitro-3-cyanophenyl
methyl



4.250
2-fluoro-3-methoxyphenyl
methyl



4.251
2-chloro-3-methoxyphenyl
methyl



4.252
2-bromo-3-methoxyphenyl
methyl



4.253
2-methyl-3-methoxyphenyl
methyl



4.254
2-cyclopropyl-3-methoxyphenyl
methyl



4.255
2-cyano-3-methoxyphenyl
methyl



4.256
2-trifluoromethyl-3-methoxyphenyl
methyl



4.257
2,3-dimethoxyphenyl
methyl



4.258
2-ethoxy-3-methoxyphenyl
methyl



4.259
2-trifluoromethoxy-3-methoxyphenyl
methyl



4.260
2-nitro-3-methoxyphenyl
methyl



4.261
2-fluoro-3-ethoxyphenyl
methyl



4.262
2-chloro-3-ethoxyphenyl
methyl



4.263
2-bromo-3-ethoxyphenyl
methyl



4.264
2-methyl-3-ethoxyphenyl
methyl



4.265
2-cyclopropyl-3-ethoxyphenyl
methyl



4.266
2-cyano-3-ethoxyphenyl
methyl



4.267
2-trifluoromethyl-3-ethoxyphenyl
methyl



4.268
2-methoxy-3-ethoxyphenyl
methyl



4.269
2,3-diethoxyphenyl
methyl



4.270
2-trifluoromethoxy-3-ethoxyphenyl
methyl



4.271
2-nitro-3-ethoxyphenyl
methyl



4.272
2-fluoro-3-isopropoxyphenyl
methyl



4.273
2-chloro-3-isopropoxyphenyl
methyl



4.274
2-bromo-3-isopropoxyphenyl
methyl



4.275
2-methyl-3-isopropoxyphenyl
methyl



4.276
2-cyclopropyl-3-isopropoxyphenyl
methyl



4.277
2-cyano-3-isopropoxyphenyl
methyl



4.278
2-trifluoromethyl-3-isopropoxyphenyl
methyl



4.279
2-methoxy-3-isopropoxyphenyl
methyl



4.280
2-trifluoromethoxy-3-isopropoxyphenyl
methyl



4.281
2-nitro-3-isopropoxyphenyl
methyl



4.282
2-fluoro-3-trifluoromethoxyphenyl
methyl



4.283
2-chloro-3-trifluoromethoxyphenyl
methyl



4.284
2-bromo-3-trifluoromethoxyphenyl
methyl



4.285
2-methyl-3-trifluoromethoxyphenyl
methyl



4.286
2-cyclopropyl-3-trifluoromethoxyphenyl
methyl



4.287
2-cyano-3-trifluoromethoxyphenyl
methyl



4.288
2-trifluoromethyl-3-trifluoromethoxy-
methyl




phenyl




4.289
2-methoxy-3-trifluoromethoxyphenyl
methyl



4.290
2,3-bis(trifluoromethoxy)phenyl
methyl



4.291
2-nitro-3-trifluoromethoxyphenyl
methyl



4.292
2-fluoro-3-difluoromethoxyphenyl
methyl



4.293
2-chloro-3-difluoromethoxyphenyl
methyl



4.294
2-bromo-3-difluoromethoxyphenyl
methyl



4.295
2-methyl-3-difluoromethoxyphenyl
methyl



4.296
2-cyclopropyl-3-difluoromethoxyphenyl
methyl



4.297
2-cyano-3-difluoromethoxyphenyl
methyl



4.298
2-trifluoromethyl-3-difluoromethoxyphenyl
methyl



4.299
2-methoxy-3-difluoromethoxyphenyl
methyl



4.300
2-ethoxy-3-difluoromethoxyphenyl
methyl



4.301
2-nitro-3-difluoromethoxyphenyl
methyl



4.302
2-fluoro-3-nitrophenyl
methyl



4.303
2-chloro-3-nitrophenyl
methyl



4.304
2-bromo-3-nitrophenyl
methyl



4.305
2-methyl-3-nitrophenyl
methyl



4.306
2-cyclopropyl-3-nitrophenyl
methyl



4.307
2-cyano-3-nitrophenyl
methyl



4.308
2-trifluoromethyl-3-nitrophenyl
methyl



4.309
2-methoxy-3-nitrophenyl
methyl



4.310
2-ethoxy-3-nitrophenyl
methyl



4.311
2-trifluoromethoxy-3-nitrophenyl
methyl



4.312
2-fluoro-3-methylsulfanylphenyl
methyl



4.313
2-chloro-3-methylsulfanylphenyl
methyl



4.314
2-bromo-3-methylsulfanylphenyl
methyl



4.315
2-methyl-3-methylsulfanylphenyl
methyl



4.316
2-ethyl-3-methylsulfanylphenyl
methyl



4.317
2-cyclopropyl-3-methylsulfanylphenyl
methyl



4.318
2-cyano-3-methylsulfanylphenyl
methyl



4.319
2-trifluoromethyl-3-methylsulfanylphenyl
methyl



4.320
2-methoxy-3-methylsulfanylphenyl
methyl



4.321
2-ethoxy-3-methylsulfanylphenyl
methyl



4.322
2-trifluoromethoxy-3-methylsulfanylphenyl
methyl



4.323
2-nitro-3-methylsulfanylphenyl
methyl



4.324
3,5-difluorophenyl
methyl
[CDCl3] 1.61 (s, 3H);





3.05 (d, 1H); 3.68 (d,





1H); 6.88 (m, 1H);





7.15 (m, 2H); 9.65 (s,





1H).


4.325
3,5-difluorophenyl
ethyl



4.326
3,5-difluorophenyl
CN



4.327
3,5-difluorophenyl
vinyl



4.328
3,5-difluorophenyl
fluoromethyl



4.329
3,5-difluorophenyl
methylcarbonyl



4.330
3,5-difluorophenyl
hydroxymethyl



4.331
3,5-difluorophenyl
ethynyl



4.332
3-chloro-5-fluorophenyl
methyl



4.333
3-chloro-5-fluorophenyl
ethyl



4.334
3-chloro-5-fluorophenyl
CN



4.335
3-chloro-5-fluorophenyl
vinyl



4.336
3-chloro-5-fluorophenyl
fluoromethyl



4.337
3-chloro-5-fluorophenyl
methylcarbonyl



4.338
3-chloro-5-fluorophenyl
hydroxymethyl



4.339
3-chloro-5-fluorophenyl
ethynyl



4.340
3-bromo-5-fluorophenyl
methyl



4.341
3-iodo-5-fluorophenyl
methyl



4.342
3-methyl-5-fluorophenyl
methyl



4.343
3-methyl-5-fluorophenyl
ethyl



4.344
3-methyl-5-fluorophenyl
CN



4.345
3-methyl-5-fluorophenyl
vinyl



4.346
3-methyl-5-fluorophenyl
fluoromethyl



4.347
3-methyl-5-fluorophenyl
methylcarbonyl



4.348
3-methyl-5-fluorophenyl
hydroxymethyl



4.349
3-methyl-5-fluorophenyl
ethynyl



4.350
3-ethyl-5-fluorophenyl
methyl



4.351
3-propyl-5-fluorophenyl
methyl



4.352
3-i-propyl-5-fluorophenyl
methyl



4.353
3-n-butyl-5-fluorophenyl
methyl



4.354
3-isobutyl-5-fluorophenyl
methyl



4.355
3-tert-butyl-5-fluorophenyl
methyl



4.356
3-tert-butyl-5-fluorophenyl
ethyl



4.357
3-tert-butyl-5-fluorophenyl
CN



4.358
3-tert-butyl-5-fluorophenyl
vinyl



4.359
3-tert-butyl-5-fluorophenyl
fluoromethyl



4.360
3-tert-butyl-5-fluorophenyl
methylcarbonyl



4.361
3-tert-butyl-5-fluorophenyl
hydroxymethyl



4.362
3-tert-butyl-5-fluorophenyl
ethynyl



4.363
3-cyclopropyl-5-fluorophenyl
methyl



4.364
3-cyano-5-fluorophenyl
methyl



4.365
3-cyano-5-fluorophenyl
ethyl



4.366
3-cyano-5-fluorophenyl
CN



4.367
3-cyano-5-fluorophenyl
vinyl



4.368
3-cyano-5-fluorophenyl
fluoromethyl



4.369
3-cyano-5-fluorophenyl
methylcarbonyl



4.370
3-cyano-5-fluorophenyl
hydroxymethyl



4.371
3-cyano-5-fluorophenyl
ethynyl



4.372
3-trifluoromethyl-5-fluorophenyl
methyl



4.373
3-(methoxycarbonyl)-5-fluorophenyl
methyl



4.374
3-methoxy-5-fluorophenyl
methyl



4.375
3-methoxy-5-fluorophenyl
ethyl



4.376
3-methoxy-5-fluorophenyl
CN



4.377
3-methoxy-5-fluorophenyl
vinyl



4.378
3-methoxy-5-fluorophenyl
fluoromethyl



4.379
3-methoxy-5-fluorophenyl
methylcarbonyl



4.380
3-methoxy-5-fluorophenyl
hydroxymethyl



4.381
3-methoxy-5-fluorophenyl
ethynyl



4.382
3-ethoxy-5-fluorophenyl
methyl



4.383
3-n-propoxy-5-fluorophenyl
methyl



4.384
3-isopropoxy-5-fluorophenyl
methyl



4.385
3-n-butoxy-5-fluorophenyl
methyl



4.386
3-isobutoxy-5-fluorophenyl
methyl



4.387
3-difluoromethoxy-5-fluorophenyl
methyl



4.388
3-trifluoromethoxy-5-fluorophenyl
methyl



4.389
3-nitro-5-fluorophenyl
methyl



4.390
3-acetoxy-5-fluorophenyl
methyl



4.391
3-methylsulfanyl-5-fluorophenyl
methyl



4.392
3,5-dichlorophenyl
methyl



4.393
3,5-dichlorophenyl
ethyl



4.394
3,5-dichlorophenyl
CN



4.395
3,5-dichlorophenyl
vinyl



4.396
3,5-dichlorophenyl
fluoromethyl



4.397
3,5-dichlorophenyl
methylcarbonyl



4.398
3,5-dichlorophenyl
hydroxymethyl



4.399
3,5-dichlorophenyl
ethynyl



4.400
3-bromo-5-chlorophenyl
methyl



4.401
3-iodo-5-chlorophenyl
methyl



4.402
3-methyl-5-chlorophenyl
methyl



4.403
3-methyl-5-chlorophenyl
ethyl



4.404
3-methyl-5-chlorophenyl
CN



4.405
3-methyl-5-chlorophenyl
vinyl



4.406
3-methyl-5-chlorophenyl
fluoromethyl



4.407
-methyl-5-chlorophenyl
methylcarbonyl



4.408
3-methyl-5-chlorophenyl
hydroxymethyl



4.409
3-methyl-5-chlorophenyl
ethynyl



4.410
3-ethyl-5-chlorophenyl
methyl



4.411
3-propyl-5-chlorophenyl
methyl



4.412
3-isopropyl-5-chlorophenyl
methyl



4.413
3-isobutyl-5-chlorophenyl
methyl



4.414
3-tert-butyl-5-chlorophenyl
methyl



4.415
3-cyclopropyl-5-chlorophenyl
methyl



4.416
3-cyano-5-chlorophenyl
methyl



4.417
3-cyano-5-chlorophenyl
ethyl



4.418
3-cyano-5-chlorophenyl
CN



4.419
3-cyano-5-chlorophenyl
vinyl



4.420
3-cyano-5-chlorophenyl
fluoromethyl



4.421
3-cyano-5-chlorophenyl
methylcarbonyl



4.422
3-cyano-5-chlorophenyl
hydroxymethyl



4.423
3-cyano-5-chlorophenyl
ethynyl



4.424
3-trifluoromethyl-5-chlorophenyl
methyl



4.425
3-trifluoromethyl-5-chlorophenyl
ethyl



4.426
3-trifluoromethyl-5-chlorophenyl
CN



4.427
3-trifluoromethyl-5-chlorophenyl
vinyl



4.428
3-trifluoromethyl-5-chlorophenyl
fluoromethyl



4.429
3-trifluoromethyl-5-chlorophenyl
methylcarbonyl



4.430
3-trifluoromethyl-5-chlorophenyl
hydroxymethyl



4.431
3-trifluoromethyl-5-chlorophenyl
ethynyl



4.432
3-(methoxycarbonyl)-5-chlorophenyl
methyl



4.433
3-methoxy-5-chlorophenyl
methyl



4.434
3-methoxy-5-chlorophenyl
ethyl



4.435
3-methoxy-5-chlorophenyl
CN



4.436
3-methoxy-5-chlorophenyl
vinyl



4.437
3-methoxy-5-chlorophenyl
fluoromethyl



4.438
3-methoxy-5-chlorophenyl
methylcarbonyl



4.439
3-methoxy-5-chlorophenyl
hydroxymethyl



4.440
3-methoxy-5-chlorophenyl
ethynyl



4.441
3-ethoxy-5-chlorophenyl
methyl



4.442
3-n-propoxy-5-chlorophenyl
methyl



4.443
3-isopropoxy-5-chlorophenyl
methyl



4.444
3-n-butoxy-5-chlorophenyl
methyl



4.445
3-isobutoxy-5-chlorophenyl
methyl



4.446
3-difluoromethoxy-5-chlorophenyl
methyl



4.447
3-trifluoromethoxy-5-chlorophenyl
methyl



4.448
3-trifluoromethoxy-5-chlorophenyl
ethyl



4.449
3-trifluoromethoxy-5-chlorophenyl
CN



4.450
3-trifluoromethoxy-5-chlorophenyl
vinyl



4.451
3-trifluoromethoxy-5-chlorophenyl
fluoromethyl



4.452
3trifluoromethoxy-5-chlorophenyl
methylcarbonyl



4.453
3-trifluoromethoxy-5-chlorophenyl
hydroxymethyl



4.454
3-trifluoromethoxy-5-chlorophenyl
ethynyl



4.455
3-nitro-5-chlorophenyl
methyl



4.456
3-acetoxy-5-chlorophenyl
methyl



4.457
3-methylsulfanyl-5-chlorophenyl
methyl



4.458
3,5-dibromophenylphenyl
methyl



4.459
3-iodo-5-bromophenyl
methyl



4.460
3-methyl-5-bromophenyl
methyl



4.461
3-ethyl-5-bromophenyl
methyl



4.462
3-propyl-5-bromophenyl
methyl



4.463
3-isopropyl-5-bromophenyl
methyl



4.464
3-isobutyl-5-bromophenyl
methyl



4.465
3-tert-butyl-5-bromophenyl
methyl



4.466
3-cyclopropyl-5-bromophenyl
methyl



4.467
3-cyano-5-bromophenyl
methyl



4.468
3-trifluoromethyl-5-bromophenyl
methyl



4.469
3-(methoxycarbonyl)-5-bromophenyl
methyl



4.470
3-methoxy-5-bromophenyl
methyl



4.471
3-ethoxy-5-bromophenyl
methyl



4.472
3-n-propoxy-5-bromophenyl
methyl



4.473
3-isopropoxy-5-bromophenyl
methyl



4.474
3-n-butoxy-5-bromophenyl
methyl



4.475
3-isobutoxy-5-bromophenyl
methyl



4.476
3-tert-butoxy-5-bromophenyl
methyl



4.477
3-difluoromethoxy-5-bromophenyl
methyl



4.478
3-trifluoromethoxy-5-bromophenyl
methyl



4.479
3-nitro-5-bromophenyl
methyl



4.480
3-acetoxy-5-bromophenyl
methyl



4.481
3-methylsulfanyl-5-bromophenyl
methyl



4.482
3,5-diiodophenyl
methyl



4.483
3-methyl-5-iodophenyl
methyl



4.484
3-ethyl-5-iodophenyl
methyl



4.485
3-propyl-5-iodophenyl
methyl



4.486
3-isopropyl-5-iodophenyl
methyl



4.487
3-n-butyl-5-iodophenyl
methyl



4.488
3-isobutyl-5-iodophenyl
methyl



4.489
3-tert-butyl-5-iodophenyl
methyl



4.490
3-cyclopropyl-5-iodophenyl
methyl



4.491
3-cyano-5-iodophenyl
methyl



4.492
3-trifluoromethyl-5-iodophenyl
methyl



4.493
3-(methoxycarbonyl)-5-iodophenyl
methyl



4.494
3-methoxy-5-iodophenyl
methyl



4.495
3-ethoxy-5-iodophenyl
methyl



4.496
3-n-propoxy-5-iodophenyl
methyl



4.497
3-isopropoxy-5-iodophenyl
methyl



4.498
3-n-butoxy-5-iodophenyl
methyl



4.499
3-isobutoxy-5-iodophenyl
methyl



4.500
3-difluoromethoxy-5-iodophenyl
methyl



4.501
3-trifluoromethoxy-5-iodophenyl
methyl



4.502
3-nitro-5-iodophenyl
methyl



4.503
3-acetoxy-5-iodophenyl
methyl



4.504
3-methylsulfanyl-5-iodophenyl
methyl



4.505
3,5-dimethylphenyl
methyl



4.506
3-ethyl-5-methylphenyl
methyl



4.507
3-propyl-5-methylphenyl
methyl



4.508
3-isopropyl-5-methylphenyl
methyl



4.509
3-n-butyl-5-methylphenyl
methyl



4.510
3-isobutyl-5-methylphenyl
methyl



4.511
3-tert-butyl-5-methylphenyl
methyl



4.512
3-cyclopropyl-5-methylphenyl
methyl



4.513
3-cyano-5-methylphenyl
methyl



4.514
3-trifluoromethyl-5-methylphenyl
methyl



4.515
3-(methoxycarbonyl)-5-methylphenyl
methyl



4.516
3-methoxy-5-methylphenyl
methyl



4.517
3-ethoxy-5-methylphenyl
methyl



4.518
3-n-propoxy-5-methylphenyl
methyl



4.519
3-n-butoxy-5-methylphenyl
methyl



4.520
3-isobutoxy-5-methylphenyl
methyl



4.521
3-difluoromethoxy-5-methylphenyl
methyl



4.522
3-trifluoromethoxy-5-methylphenyl
methyl



4.523
3-nitro-5-methylphenyl
methyl



4.524
3-acetoxy-5-methylphenyl
methyl



4.525
3-methylsulfanyl-5-methylphenyl
methyl



4.526
3,5-diethylphenyl
methyl



4.527
3-propyl-5-ethylphenyl
methyl



4.528
3-isopropyl-5-ethylphenyl
methyl



4.529
3-n-butyl-5-ethylphenyl
methyl



4.530
3-isobutyl-5-ethylphenyl
methyl



4.531
3-tert-butyl-5-ethylphenyl
methyl



4.532
3-cyclopropyl-5-ethylphenyl
methyl



4.533
3-cyano-5-ethylphenyl
methyl



4.534
3-trifluoromethyl-5-ethylphenyl
methyl



4.535
3-(methoxycarbonyl)-5-ethylphenyl
methyl



4.536
3-methoxy-5-ethylphenyl
methyl



4.537
3-ethoxy-5-ethylphenyl
methyl



4.538
3-n-propoxy-5-ethylphenyl
methyl



4.539
3-n-butoxy-5-ethylphenyl
methyl



4.540
3-isobutoxy-5-ethylphenyl
methyl



4.541
3-difluoromethoxy-5-ethylphenyl
methyl



4.542
3-trifluoromethoxy-5-ethylphenyl
methyl



4.543
3-nitro-5-ethylphenyl
methyl



4.544
3-acetoxy-5-ethylphenyl
methyl



4.545
3-methylsulfanyl-5-ethylphenyl
methyl



4.546
3,5-dipropylphenyl
methyl



4.547
3-isopropyl-5-propylphenyl
methyl



4.548
3-n-butyl-5-propylphenyl
methyl



4.549
3-isobutyl-5-propylphenyl
methyl



4.550
3-tert-butyl-5-propylphenyl
methyl



4.551
3-cyclopropyl-5-propylphenyl
methyl



4.552
3-cyano-5-propylphenyl
methyl



4.553
3-trifluoromethyl-5-propylphenyl
methyl



4.554
3-(methoxycarbonyl)-5-propylphenyl
methyl



4.555
3-methoxy-5-propylphenyl
methyl



4.556
3-ethoxy-5-propylphenyl
methyl



4.557
3-n-propoxy-5-propylphenyl
methyl



4.558
3-n-butoxy-5-propylphenyl
methyl



4.559
3-isobutoxy-5-propylphenyl
methyl



4.560
3-tert-butoxy-5-propylphenyl
methyl



4.561
3-difluoromethoxy-5-propylphenyl
methyl



4.562
3-trifluoromethoxy-5-ethylphenyl
methyl



4.563
3-nitro-5-propylphenyl
methyl



4.564
3-acetoxy-5-propylphenyl
methyl



4.565
3-methylsulfanyl-5-propylphenyl
methyl



4.566
3,5-diisopropylphenyl
methyl



4.567
3-n-butyl-5-isopropylphenyl
methyl



4.568
3-isobutyl-5-isopropylphenyl
methyl



4.569
3-tert-butyl-5-isopropylphenyl
methyl



4.570
3-cyclopropyl-5-isopropylphenyl
methyl



4.571
3-cyano-5-isopropylphenyl
methyl



4.572
3-trifluoromethyl-5-isopropylphenyl
methyl



4.573
3-(methoxycarbonyl)-5-isopropylphenyl
methyl



4.574
3-methoxy-5-isopropylphenyl
methyl



4.575
3-ethoxy-5-isopropylphenyl
methyl



4.576
3-n-propoxy-5-isopropylphenyl
methyl



4.577
3-n-butoxy-5-isopropylphenyl
methyl



4.578
3-isobutoxy-5-isopropylphenyl
methyl



4.579
3-tert-butoxy-5-isopropylphenyl
methyl



4.580
3-difluoromethoxy-5-isopropylphenyl
methyl



4.581
3-trifluoromethoxy-5-isopropylphenyl
methyl



4.582
3-nitro-5-isopropylphenyl
methyl



4.583
3-acetoxy-5-isopropylphenyl
methyl



4.584
3-methylsulfanyl-5-isopropylphenyl
methyl



4.585
3,5-diisobutylphenyl
methyl



4.586
3-tert-butyl-5-isobutylphenyl
methyl



4.587
3-cyclopropyl-5-isobutylphenyl
methyl



4.588
3-cyano-5-isobutylphenyl
methyl



4.589
3-trifluoromethyl-5-isobutylphenyl
methyl



4.590
3-(methoxycarbonyl)-5-isobutylphenyl
methyl



4.591
3-methoxy-5-isobutylphenyl
methyl



4.592
3-ethoxy-5-isobutylphenyl
methyl



4.593
3-n-propoxy-5-isobutylphenyl
methyl



4.594
3-n-butoxy-5-isobutylphenyl
methyl



4.595
3-isobutoxy-5-isobutylphenyl
methyl



4.596
3-tert-butoxy-5-isobutylphenyl
methyl



4.597
3-difluoromethoxy-5-isobutylphenyl
methyl



4.598
3-trifluoromethoxy-5-isobutylphenyl
methyl



4.599
3-nitro-5-isobutylphenyl
methyl



4.600
3-acetoxy-5-isobutylphenyl
methyl



4.601
3-methylsulfanyl-5-isobutylphenyl
methyl



4.602
3-tert-butyl-5-cyclopropylphenyl
methyl



4.603
3,5-dicyclopropylphenyl
methyl



4.604
3-cyano-5-cyclopropylphenyl
methyl



4.605
3-cyano-5-cyclopropylphenyl
ethyl



4.606
3-cyano-5-cyclopropylphenyl
CN



4.607
3-cyano-5-cyclopropylphenyl
vinyl



4.608
3-cyano-5-cyclopropylphenyl
fluoromethyl



4.609
3-cyano-5-cyclopropylphenyl
methylcarbonyl



4.610
3-cyano-5-cyclopropylphenyl
hydroxymethyl



4.611
3-cyano-5-cyclopropylphenyl
ethynyl



4.612
3-trifluoromethyl-5-cyclopropylphenyl
methyl



4.613
3-(methoxycarbonyl)-5-cyclopropylphenyl
methyl



4.614
3-methoxy-5-cyclopropylphenyl
methyl



4.615
3-ethoxy-5-cyclopropylphenyl
methyl



4.616
3-n-propoxy-5-cyclopropylphenyl
methyl



4.617
3-n-butoxy-5-cyclopropylphenyl
methyl



4.618
3-isobutoxy-5-cyclopropylphenyl
methyl



4.619
3-difluoromethoxy-5-cyclopropylphenyl
methyl



4.620
3-trifluoromethoxy-5-cyclopropylphenyl
methyl



4.621
3-nitro-5-cyclopropylphenyl
methyl



4.622
3-acetoxy-5-cyclopropylphenyl
methyl



4.623
3-methylsulfanyl-5-cyclopropylphenyl
methyl



4.624
3,5-dicyanophenyl
methyl



4.625
3-trifluoromethyl-5-cyanophenyl
methyl



4.626
3-(methoxycarbonyl)-5-cyanophenyl
methyl



4.627
3-methoxy-5-cyanophenyl
methyl



4.628
3-ethoxy-5-cyanophenyl
methyl



4.629
3-n-propoxy-5-cyanophenyl
methyl



4.630
3-n-butoxy-5-cyanophenyl
methyl



4.631
3-isobutoxy-5-cyanophenyl
methyl



4.632
3-difluoromethoxy-5-cyanophenyl
methyl



4.633
3-trifluoromethoxy-5-cyanophenyl
methyl



4.634
3-nitro-5-cyanophenyl
methyl



4.635
3-acetoxy-5-cyanophenyl
methyl



4.636
3-methylsulfanyl-5-cyanophenyl
methyl



4.637
3,5-di(trifluoromethyl)phenyl
methyl



4.638
3,5-di(trifluoromethyl)phenyl
ethyl



4.639
3,5-di(trifluoromethyl)phenyl
CN



4.640
3,5-di(trifluoromethyl)phenyl
vinyl



4.641
3,5-di(trifluoromethyl)phenyl
fluoromethyl



4.642
3,5-di(trifluoromethyl)phenyl
methylcarbonyl



4.643
3,5-di(trifluoromethyl)phenyl
hydroxymethyl



4.644
3,5-di(trifluoromethyl)phenyl
ethynyl



4. 645
3-(methoxycarbonyl)-5-trifluoromethyl-
methyl




phenyl




4.646
3-methoxy-5-trifluoromethylphenyl
methyl



4.647
3-ethoxy-5-trifluoromethylphenyl
methyl



4.648
3-n-propoxy-5-trifluoromethylphenyl
methyl



4.649
3-n-butoxy-5-trifluoromethylphenyl
methyl



4.650
3-isobutoxy-5-trifluoromethylphenyl
methyl



4.651
3-difluoromethoxy-5-trifluoromethylphenyl
methyl



4.652
3-trifluoromethoxy-5-trifluoromethylphenyl
methyl



4.653
3-nitro-5-trifluoromethylphenyl
methyl



4.654
3-acetoxy-5-trifluoromethylphenyl
methyl



4.655
3-methylsulfanyl-5-trifluoromethylphenyl
methyl



4.656
3,5-di(methoxycarbonyl)phenyl
methyl



4.657
3-methoxy-5-(methoxycarbonyl)phenyl
methyl



4.658
3-ethoxy-5-(methoxycarbonyl)phenyl
methyl



4.659
3-n-propoxy-5-(methoxycarbonyl)phenyl
methyl



4.660
3-n-butoxy-5-(methoxycarbonyl)phenyl
methyl



4.661
3-isobutoxy-5-(methoxycarbonyl)phenyl
methyl



4.662
3-difluoromethoxy-5-(methoxycarbonyl)-
methyl




phenyl




4.663
3-trifluoromethoxy-5-(methoxycarbonyl)-
methyl




phenyl




4.664
3-nitro-5-(methoxycarbonyl)phenyl
methyl



4.665
3-acetoxy-5-(methoxycarbonyl)phenyl
methyl



4.666
3-methylsulfanyl-5-(methoxycarbonyl)-
methyl




phenyl




4.667
3,5-dimethoxyphenyl
methyl



4.668
3,5-dimethoxyphenyl
ethyl



4.669
3,5-dimethoxyphenyl
CN



4.670
3,5-dimethoxyphenyl
vinyl



4.671
3,5-dimethoxyphenyl
fluoromethyl



4.672
3,5-dimethoxyphenyl
methylcarbonyl



4.673
3,5-dimethoxyphenyl
hydroxymethyl



4.674
3,5-dimethoxyphenyl
ethynyl



4.675
3-ethoxy-5-methoxyphenyl
methyl



4.676
3-n-propoxy-5-methoxyphenyl
methyl



4.677
3-n-butoxy-5-methoxyphenyl
methyl



4.678
3-isobutoxy-5-methoxyphenyl
methyl



4.679
3-difluoromethoxy-5-methoxyphenyl
methyl



4.680
3-trifluoromethoxy-5-methoxyphenyl
methyl



4.681
3-nitro-5-methoxyphenyl
methyl



4.682
3-acetoxy-5-methoxyphenyl
methyl



4.683
3-methylsulfanyl-5-methoxyphenyl
methyl



4.684
3,5-diethoxyphenyl
methyl



4.685
3-n-propoxy-5-ethoxyphenyl
methyl



4.686
3-n-butoxy-5-ethoxyphenyl
methyl



4.687
3-isobutoxy-5-ethoxyphenyl
methyl



4.688
3-tert-butoxy-5-ethoxyphenyl
methyl



4.689
3-difluoromethoxy-5-ethoxyphenyl
methyl



4.690
3-trifluoromethoxy-5-ethoxyphenyl
methyl



4.691
3-nitro-5-ethoxyphenyl
methyl



4.692
3-acetoxy-5-ethoxyphenyl
methyl



4.693
3-methylsulfanyl-5-ethoxyphenyl
methyl



4.694
3,5-di(trifluoromethoxy)phenyl
methyl



4.695
3-nitro-5-trifluoromethoxyphenyl
methyl



4.696
3-methylsulfanyl-5-trifluoromethoxy-
methyl




phenyl




4.697
3,5-bis(difluoromethoxy)phenyl
methyl



4.698
3-trifluoromethoxy-5-difluoromethoxy-
methyl




phenyl




4.699
3-nitro-5-difluoromethoxyphenyl
methyl



4.700
3-acetoxy-5-difluoromethoxyphenyl
methyl



4.701
3-methylsulfanyl-5-difluoromethoxy-
methyl




phenyl




4.702
3-methylsulfanyl-5-acetoxyphenyl
methyl



4.703
3-acetoxy-5-nitrophenyl
methyl



4.704
3-methylsulfanyl-5-nitrophenyl
methyl



4.705
3,5-di(methylsulfanyl)phenyl
methyl



4.706
3,4-difluorophenyl
methyl



4.707
3,4-difluorophenyl
ethyl



4.708
3,4-difluorophenyl
CN



4.709
3,4-difluorophenyl
vinyl



4.710
3,4-difluorophenyl
fluoromethyl



4.711
3,4-difluorophenyl
methylcarbonyl



4.712
3,4-difluorophenyl
hydroxymethyl



4.713
3,4-difluorophenyl
ethynyl



4.714
3-chloro-4-fluorophenyl
methyl



4.715
3-bromo-4-fluorophenyl
methyl



4.716
3-methyl-4-fluorophenyl
methyl



4.717
3-methyl-4-fluorophenyl
ethyl



4.718
3-methyl-4-fluorophenyl
CN



4.719
3-methyl-4-fluorophenyl
vinyl



4.720
3-methyl-4-fluorophenyl
fluoromethyl



4.721
3-methyl-4-fluorophenyl
methylcarbonyl



4.722
3-methyl-4-fluorophenyl
hydroxymethyl



4.723
3-methyl-4-fluorophenyl
ethynyl



4.724
3-ethyl-4-fluorophenyl
methyl



4.725
3-cyclopropyl-4-fluorophenyl
methyl



4.726
3-cyano-4-fluorophenyl
methyl



4.727
3-methoxy-4-fluorophenyl
methyl



4.728
3-ethoxy-4-fluorophenyl
methyl



4.729
3-trifluoromethoxy-4-fluorophenyl
methyl



4.730
3-nitro-4-fluorophenyl
methyl



4.731
3-fluoro-4-chlorophenyl
methyl



4.732
3,4-dichlorophenyl
methyl



4.733
3-bromo-4-chlorophenyl
methyl



4.734
3-methyl-4-chlorophenyl
methyl



4.735
3-cyclopropyl-4-chlorophenyl
methyl



4.736
3-cyano-4-chlorophenyl
methyl



4.737
3-trifluoromethyl-4-chlorophenyl
methyl



4.738
3-methoxy-4-chlorophenyl
methyl



4.739
3-ethoxy-4-chlorophenyl
methyl



4.740
3-trifluoromethoxy-4-chlorophenyl
methyl



4.741
3-nitro-4-chlorophenyl
methyl



4.742
3-fluoro-4-bromophenyl
methyl



4.743
3-chloro-4-bromophenyl
methyl



4.744
3,4-dibromophenyl
methyl



4.745
3-methyl-4-bromophenyl
methyl



4.746
3-cyclopropyl-4-bromophenyl
methyl



4.747
3-cyano-4-bromophenyl
methyl



4.748
3-trifluoromethyl-4-bromophenyl
methyl



4.749
3-methoxy-4-phenyl
methyl



4.750
3-ethoxy-4-bromophenyl
methyl



4.751
3-trifluoromethoxy-4-bromophenyl
methyl



4.752
3-nitro-4-bromophenyl
methyl



4.753
3-fluoro-4-iodophenyl
methyl



4.754
3-chloro-4-iodophenyl
methyl



4.755
3-bromo-4-iodophenyl
methyl



4.756
3-methyl-4-iodophenyl
methyl



4.757
3-cyclopropyl-4-iodophenyl
methyl



4.758
3-cyano-4-iodophenyl
methyl



4.759
3-trifluoromethyl-4-iodophenyl
methyl



4.760
3-methoxy-4-iodophenyl
methyl



4.761
3-ethoxy-4-iodophenyl
methyl



4.762
3-trifluoromethoxy-4-iodophenyl
methyl



4.763
3-nitro-4-iodophenyl
methyl



4.764
3-fluoro-4-methylphenyl
methyl



4.765
3-chloro-4-methylphenyl
methyl



4.766
3-chloro-4-methylphenyl
ethyl



4.767
3-chloro-4-methylphenyl
CN



4.768
3-chloro-4-methylphenyl
vinyl



4.769
3-chloro-4-methylphenyl
fluoromethyl



4.770
3-chloro-4-methylphenyl
methylcarbonyl



4.771
3-chloro-4-methylphenyl
hydroxymethyl



4.772
3-chloro-4-methylphenyl
ethynyl



4.773
3-bromo-4-methylphenyl
methyl



4.774
3,4-dimethylphenyl
methyl



4.775
3-ethyl-4-methylphenyl
methyl



4.776
3-cyclopropyl-4-methylphenyl
methyl



4.777
3-cyano-4-methylphenyl
methyl



4.778
3-trifluoromethyl-4-methylphenyl
methyl



4.779
3-methoxy-4-methylphenyl
methyl



4.780
3-ethoxy-4-methylphenyl
methyl



4.781
3-trifluoromethoxy-4-methylphenyl
methyl



4.782
3-nitro-4-methylphenyl
methyl



4.783
3-fluoro-4-ethylphenyl
methyl



4.784
3-chloro-4-ethylphenyl
methyl



4.785
3-bromo-4-ethylphenyl
methyl



4.786
3-methyl-4-ethylphenyl
methyl



4.787
3,4-diethylphenyl
methyl



4.788
3-cyclopropyl-4-ethylphenyl
methyl



4.789
3-cyano-4-ethylphenyl
methyl



4.790
3-trifluoromethyl-4-ethylphenyl
methyl



4.791
3-methoxy-4-ethylphenyl
methyl



4.792
3-ethoxy-4-ethylphenyl
methyl



4.793
3-trifluoromethoxy-4-ethylphenyl
methyl



4.794
3-nitro-4-ethylphenyl
methyl



4.795
3-fluoro-4-propylphenyl
methyl



4.796
3-chloro-4-propylphenyl
methyl



4.797
3-bromo-4-propylphenyl
methyl



4.798
3-methyl-4-propylphenyl
methyl



4.799
3-cyclopropyl-4-propylphenyl
methyl



4.800
3-cyano-4-propylphenyl
methyl



4.801
3-trifluoromethyl-4-propylphenyl
methyl



4.802
3-methoxy-4-propylphenyl
methyl



4.803
3-ethoxy-4-propylphenyl
methyl



4.804
3-trifluoromethoxy-4-propylphenyl
methyl



4.805
3-nitro-4-propylphenyl
methyl



4.806
3-fluoro-4-isopropylphenyl
methyl



4.807
3-chloro-4-isopropylphenyl
methyl



4.808
3-bromo-4-isopropylphenyl
methyl



4.809
3-methyl-4-isopropylphenyl
methyl



4.810
3-cyclopropyl-4-isopropylphenyl
methyl



4.811
3-cyano-4-isopropylphenyl
methyl



4.812
3-trifluoromethyl-4-isopropylphenyl
methyl



4.813
3-methoxy-4-isopropylphenyl
methyl



4.814
3-ethoxy-4-isopropylphenyl
methyl



4.815
3-trifluoromethoxy-4-isopropylphenyl
methyl



4.816
3-nitro-4-isopropylphenyl
methyl



4.817
3-fluoro-4-tert-butylphenyl
methyl



4.818
3-fluoro-4-tert-butylphenyl
ethyl



4.819
3-fluoro-4-tert-butylphenyl
CN



4.820
3-fluoro-4-tert-butylphenyl
vinyl



4.821
3-fluoro-4-tert-butylphenyl
fluoromethyl



4.822
3-fluoro-4-tert-butylphenyl
methylcarbonyl



4.823
3-fluoro-4-tert-butylphenyl
hydroxymethyl



4.824
3-fluoro-4-tert-butylphenyl
ethynyl



4.825
3-chloro-4-tert-butylphenyl
methyl



4.826
3-bromo-4-tert-butylphenyl
methyl



4.827
3-methyl-4-tert-butylphenyl
methyl



4.828
3-cyclopropyl-4-tert-butylphenyl
methyl



4.829
3-cyano-4-tert-butylphenyl
methyl



4.830
3-trifluoromethyl-4-tert-butylphenyl
methyl



4.831
3-methoxy-4-tert-butylphenyl
methyl



4.832
3-ethoxy-4-tert-butylphenyl
methyl



4.833
3-trifluoromethoxy-4-tert-butylphenyl
methyl



4.834
3-nitro-4-tert-butylphenyl
methyl



4.835
3-fluoro-4-cyclopropylphenyl
methyl



4.836
3-chloro-4-cyclopropylphenyl
methyl



4.837
3-bromo-4-cyclopropylphenyl
methyl



4.838
3-methyl-4-cyclopropylphenyl
methyl



4.839
3-cyclopropyl-4-cyclopropylphenyl
methyl



4.840
3-cyano-4-cyclopropylphenyl
methyl



4.841
3-trifluoromethyl-4-cyclopropylphenyl
methyl



4.842
3-methoxy-4-cyclopropylphenyl
methyl



4.843
3-ethoxy-4-cyclopropylphenyl
methyl



4.844
3-trifluoromethoxy-4-cyclopropylphenyl
methyl



4.845
3-fluoro-4-methoxycarbonylphenyl
methyl



4.846
3-chloro-4-methoxycarbonylphenyl
methyl



4.847
3-bromo-4-methoxycarbonylphenyl
methyl



4.848
3-methyl-4-methoxycarbonylphenyl
methyl



4.849
3-cyclopropyl-4-methoxycarbonylphenyl
methyl



4.850
3-cyano-4-methoxycarbonylphenyl
methyl



4.851
3-trifluoromethyl-4-methoxycarbonyl-
methyl




phenyl




4.852
3-methoxy-4-methoxycarbonylphenyl
methyl



4.853
3-ethoxy-4-methoxycarbonylphenyl
methyl



4.854
3-trifluoromethoxy-4-methoxycarbonyl-
methyl




phenyl




4.855
3-nitro-4-methoxycarbonylphenyl
methyl



4.856
3-fluoro-4-cyanophenyl
methyl



4.857
3-chloro-4-cyanophenyl
methyl



4.858
3-bromo-4-cyanophenyl
methyl



4.859
3-methyl-4-cyanophenyl
methyl



4.860
3-cyclopropyl-4-cyanophenyl
methyl



4.861
3-cyano-4-cyanophenyl
methyl



4.862
3-trifluoromethyl-4-cyanophenyl
methyl



4.863
3-methoxy-4-cyanophenyl
methyl



4.864
3-ethoxy-4-cyanophenyl
methyl



4.865
3-trifluoromethoxy-4-cyanophenyl
methyl



4.866
3-nitro-4-cyanophenyl
methyl



4.867
3-fluoro-4-methoxyphenyl
methyl



4.868
3-chloro-4-methoxyphenyl
methyl



4.869
3-bromo-4-methoxyphenyl
methyl



4.870
3-methyl-4-methoxyphenyl
methyl



4.871
3-cyclopropyl-4-methoxyphenyl
methyl



4.872
3-cyano-4-methoxyphenyl
methyl



4.873
3-trifluoromethyl-4-methoxyphenyl
methyl



4.874
3,4-dimethoxyphenyl
methyl



4.875
3-ethoxy-4-methoxyphenyl
methyl



4.876
3-trifluoromethoxy-4-methoxyphenyl
methyl



4.877
3-nitro-4-methoxyphenyl
methyl



4.878
3-fluoro-4-ethoxyphenyl
methyl



4.879
3-chloro-4-ethoxyphenyl
methyl



4.880
3-bromo-4-ethoxyphenyl
methyl



4.881
3-methyl-4-ethoxyphenyl
methyl



4.882
3-cyclopropyl-4-ethoxyphenyl
methyl



4.883
3-cyano-4-ethoxyphenyl
methyl



4.884
3-trifluoromethyl-4-ethoxyphenyl
methyl



4.885
3-methoxy-4-ethoxyphenyl
methyl



4.886
2,4-diethoxyphenyl
methyl



4.887
3-trifluoromethoxy-4-ethoxyphenyl
methyl



4.888
3-nitro-4-ethoxyphenyl
methyl



4.889
3-fluoro-4-isopropoxyphenyl
methyl



4.890
3-chloro-4-isopropoxyphenyl
methyl



4.891
3-bromo-4-isopropoxyphenyl
methyl



4.892
3-methyl-4-isopropoxyphenyl
methyl



4.893
3-cyclopropyl-4-isopropoxyphenyl
methyl



4.894
3-cyano-4-isopropoxyphenyl
methyl



4.895
3-trifluoromethyl-4-isopropoxyphenyl
methyl



4.896
3-methoxy-4-isopropoxyphenyl
methyl



4.897
3-ethoxy-4-isopropoxyphenyl
methyl



4.898
3-trifluoromethoxy-4-isopropoxyphenyl
methyl



4.899
3-nitro-4-isopropoxyphenyl
methyl



4.900
3-fluoro-4-trifluoromethoxyphenyl
methyl



4.901
3-chloro-4-trifluoromethoxyphenyl
methyl



4.902
3-bromo-4-trifluoromethoxyphenyl
methyl



4.903
3-methyl-4-trifluoromethoxyphenyl
methyl



4.904
3-cyclopropyl-4-trifluoromethoxyphenyl
methyl



4.905
3-cyano-4-trifluoromethoxyphenyl
methyl



4.906
3-trifluoromethyl-4-trifluoromethoxy-
methyl




phenyl




4.907
3-methoxy-4-trifluoromethoxyphenyl
methyl



4.908
3-ethoxy-4-trifluoromethoxyphenyl
methyl



4.909
3,4-bis(trifluoromethoxy)phenyl
methyl



4.910
3-nitro-4-trifluoromethoxyphenyl
methyl



4.911
3-fluoro-4-difluoromethoxyphenyl
methyl



4.912
3-chloro-4-difluoromethoxyphenyl
methyl



4.913
3-bromo-4-difluoromethoxyphenyl
methyl



4.914
3-methyl-4-difluoromethoxyphenyl
methyl



4.915
3-cyclopropyl-4-difluoromethoxyphenyl
methyl



4.916
3-cyano-4-difluoromethoxyphenyl
methyl



4.917
3-trifluoromethyl-4-difluoromethoxyphenyl
methyl



4.918
3-methoxy-4-difluoromethoxyphenyl
methyl



4.919
3-ethoxy-4-difluoromethoxyphenyl
methyl



4.920
3-trifluoromethoxy-4-difluoromethoxy-
methyl




phenyl




4.921
3-nitro-4-difluoromethoxyphenyl
methyl



4.922
3-fluoro-4-nitrophenyl
methyl



4.923
3-chloro-4-nitrophenyl
methyl



4.924
3-bromo-4-nitrophenyl
methyl



4.925
3-methyl-4-nitrophenyl
methyl



4.926
3-cyclopropyl-4-nitrophenyl
methyl



4.927
3-cyano-4-nitrophenyl
methyl



4.928
3-trifluoromethyl-4-nitrophenyl
methyl



4.929
3-methoxy-4-nitrophenyl
methyl



4.930
3-ethoxy-4-nitrophenyl
methyl



4.931
3-trifluoromethoxy-4-nitrophenyl
methyl



4.932
3-fluoro-4-methylsulfanylphenyl
methyl



4.933
3-chloro-4-methylsulfanylphenyl
methyl



4.934
3-bromo-4-methylsulfanylphenyl
methyl



4.935
3-methyl-4-methylsulfanylphenyl
methyl



4.936
3-cyclopropyl-4-methylsulfanylphenyl
methyl



4.937
3-cyano-4-methylsulfanylphenyl
methyl



4.938
3-trifluoromethyl-4-methylsulfanylphenyl
methyl



4.939
3-methoxy-4-methylsulfanylphenyl
methyl



4.940
3-ethoxy-4-methylsulfanylphenyl
methyl



4.941
3-trifluoromethoxy-4-methylsulfanylphenyl
methyl



4.942
3-nitro-4-methylsulfanylphenyl
methyl



4.943
3,6-difluorophenyl
methyl



4.944
3,6-difluorophenyl
ethyl



4.945
3,6-difluorophenyl
CN



4.946
3,6-difluorophenyl
vinyl



4.947
3,6-difluorophenyl
fluoromethyl



4.948
3,6-difluorophenyl
methylcarbonyl



4.949
3,6-difluorophenyl
hydroxymethyl



4.950
3,6-difluorophenyl
ethynyl



4.951
3-chloro-6-fluorophenyl
methyl



4.952
3-bromo-6-fluorophenyl
methyl



4.953
3-methyl-6-fluorophenyl
methyl



4.954
3-cyclopropyl-6-fluorophenyl
methyl



4.955
3-cyano-6-fluorophenyl
methyl



4.956
3-methoxy-6-fluorophenyl
methyl



4.957
3-ethoxy-6-fluorophenyl
methyl



4.958
3-trifluoromethoxy-6-fluorophenyl
methyl



4.959
3-nitro-6-fluorophenyl
methyl



4.960
3-fluoro-6-chlorophenyl
methyl



4.961
3,6-dichlorophenyl
methyl



4.962
3-bromo-6-chlorophenyl
methyl



4.963
3-methyl-6-chlorophenyl
methyl



4.964
3-cyclopropyl-6-chlorophenyl
methyl



4.965
3-cyano-6-chlorophenyl
methyl



4.966
3-trifluoromethyl-6-chlorophenyl
methyl



4.967
3-methoxy-6-chlorophenyl
methyl



4.968
3-ethoxy-6-chlorophenyl
methyl



4.969
3-trifluoromethoxy-6-chlorophenyl
methyl



4.970
3-nitro-6-chlorophenyl
methyl



4.971
3-fluoro-6-bromophenyl
methyl



4.972
3-chloro-6-bromophenyl
methyl



4.973
3,6-dibromophenyl
methyl



4.974
3-methyl-6-bromophenyl
methyl



4.975
3-cyclopropyl-6-bromophenyl
methyl



4.976
3-cyano-6-bromophenyl
methyl



4.977
3-trifluoromethyl-6-bromophenyl
methyl



4.978
3-methoxy-6-phenyl
methyl



4.979
3-ethoxy-6-bromophenyl
methyl



4.980
3-trifluoromethoxy-6-bromophenyl
methyl



4.981
3-nitro-6-bromophenyl
methyl



4.982
3-fluoro-6-iodophenyl
methyl



4.983
3-chloro-6-iodophenyl
methyl



4.984
3-bromo-6-iodophenyl
methyl



4.985
3-methyl-6-iodophenyl
methyl



4.986
3-ethyl-6-iodophenyl
methyl



4.987
3-cyclopropyl-6-iodophenyl
methyl



4.988
3-cyano-6-iodophenyl
methyl



4.989
3-trifluoromethyl-6-iodophenyl
methyl



4.990
3-methoxy-6-iodophenyl
methyl



4.991
3-ethoxy-6-iodophenyl
methyl



4.992
3-trifluoromethoxy-6-iodophenyl
methyl



4.993
3-nitro-6-iodophenyl
methyl



4.994
3-fluoro-6-methylphenyl
methyl



4.995
3-chloro-6-methylphenyl
methyl



4.996
3-bromo-6-methylphenyl
methyl



4.997
3,6-dimethylphenyl
methyl



4.998
3,6-dimethylphenyl
ethyl



4.999
3,6-dimethylphenyl
CN



4.1000
3,6-dimethylphenyl
vinyl



4.1001
3,6-dimethylphenyl
fluoromethyl



4.1002
3,6-dimethylphenyl
methylcarbonyl



4.1003
3,6-dimethylphenyl
hydroxymethyl



4.1004
3,6-dimethylphenyl
ethynyl



4.1005
3-cyclopropyl-6-methylphenyl
methyl



4.1006
3-cyano-6-methylphenyl
methyl



4.1007
3-trifluoromethyl-6-methylphenyl
methyl



4.1008
3-methoxy-6-methylphenyl
methyl



4.1009
3-ethoxy-6-methylphenyl
methyl



4.1010
3-trifluoromethoxy-6-methylphenyl
methyl



4.1011
3-nitro-6-methylphenyl
methyl



4.1012
3-fluoro-6-ethylphenyl
methyl



4.1013
3-chloro-6-ethylphenyl
methyl



4.1014
3-bromo-6-ethylphenyl
methyl



4.1015
3-methyl-6-ethylphenyl
methyl



4.1016
3,6-diethylphenyl
methyl



4.1017
3-cyclopropyl-6-ethylphenyl
methyl



4.1018
3-cyano-6-ethylphenyl
methyl



4.1019
3-trifluoromethyl-6-ethylphenyl
methyl



4.1020
3-methoxy-6-ethylphenyl
methyl



4.1021
3-ethoxy-6-ethylphenyl
methyl



4.1022
3-trifluoromethoxy-6-ethylphenyl
methyl



4.1023
3-nitro-6-ethylphenyl
methyl



4.1024
3-fluoro-6-isopropylphenyl
methyl



4.1025
3-chloro-6-isopropylphenyl
methyl



4.1026
3-bromo-6-isopropylphenyl
methyl



4.1027
3-methyl-6-isopropylphenyl
methyl



4.1028
3-cyclopropyl-6-isopropylphenyl
methyl



4.1029
3-cyano-6-isopropylphenyl
methyl



4.1030
3-trifluoromethyl-6-isopropylphenyl
methyl



4.1031
3-methoxy-6-isopropylphenyl
methyl



4.1032
3-ethoxy-6-isopropylphenyl
methyl



4.1033
3-trifluoromethoxy-6-isopropylphenyl
methyl



4.1034
3-nitro-6-isopropylphenyl
methyl



4.1035
3-fluoro-6-tert-butylphenyl
methyl



4.1036
3-chloro-6-tert-butylphenyl
methyl



4.1037
3-bromo-6-tert-butylphenyl
methyl



4.1038
3-methyl-6-tert-butylphenyl
methyl



4.1039
3-ethyl-6-tert-butylphenyl
methyl



4.1040
3-cyclopropyl-6-tert-butylphenyl
methyl



4.1041
3-cyano-6-tert-butylphenyl
methyl



4.1042
3-trifluoromethyl-6-tert-butylphenyl
methyl



4.1043
3-methoxy-6-tert-butylphenyl
methyl



4.1044
3-ethoxy-6-tert-butylphenyl
methyl



4.1045
3-trifluoromethoxy-6-tert-butylphenyl
methyl



4.1046
3-nitro-6-tert-butylphenyl
methyl



4.1047
3-fluoro-6-cyclopropylphenyl
methyl



4.1048
3-chloro-6-cyclopropylphenyl
methyl



4.1049
3-bromo-6-cyclopropylphenyl
methyl



4.1050
3-methyl-6-cyclopropylphenyl
methyl



4.1051
3-cyclopropyl-6-cyclopropylphenyl
methyl



4.1052
3-cyano-6-cyclopropylphenyl
methyl



4.1053
3-trifluoromethyl-6-cyclopropylphenyl
methyl



4.1054
3-methoxy-6-cyclopropylphenyl
methyl



4.1055
3-ethoxy-6-cyclopropylphenyl
methyl



4.1056
3-trifluoromethoxy-6-cyclopropylphenyl
methyl



4.1057
3-fluoro-6-methoxycarbonylphenyl
methyl



4.1058
3-chloro-6-methoxycarbonylphenyl
methyl



4.1059
3-bromo-6-methoxycarbonylphenyl
methyl



4.1060
3-methyl-6-methoxycarbonylphenyl
methyl



4.1061
3-cyclopropyl-6-methoxycarbonylphenyl
methyl



4.1062
3-cyano-6-methoxycarbonylphenyl
methyl



4.1063
3-trifluoromethyl-6-methoxycarbonyl-
methyl




phenyl




4.1064
3-methoxy-6-methoxycarbonylphenyl
methyl



4.1065
3-ethoxy-6-methoxycarbonylphenyl
methyl



4.1066
3-trifluoromethoxy-6-methoxycarbonyl-
methyl




phenyl




4.1067
3-nitro-6-methoxycarbonylphenyl
methyl



4.1068
3-fluoro-6-cyanophenyl
methyl



4.1069
3-chloro-6-cyanophenyl
methyl



4.1070
3-bromo-6-cyanophenyl
methyl



4.1071
3-methyl-6-cyanophenyl
methyl



4.1072
3-cyclopropyl-6-cyanophenyl
methyl



4.1073
3-cyano-6-cyanophenyl
methyl



4.1074
3-trifluoromethyl-6-cyanophenyl
methyl



4.1075
3-methoxy-6-cyanophenyl
methyl



4.1076
3-ethoxy-6-cyanophenyl
methyl



4.1077
3-trifluoromethoxy-6-cyanophenyl
methyl



4.1078
3-nitro-6-cyanophenyl
methyl



4.1079
3-fluoro-6-methoxyphenyl
methyl



4.1080
3-chloro-6-methoxyphenyl
methyl



4.1081
3-bromo-6-methoxyphenyl
methyl



4.1082
3-methyl-6-methoxyphenyl
methyl



4.1083
3-cyclopropyl-6-methoxyphenyl
methyl



4.1084
3-cyano-6-methoxyphenyl
methyl



4.1085
3-trifluoromethyl-6-methoxyphenyl
methyl



4.1086
3,6-dimethoxyphenyl
methyl



4.1087
3-ethoxy-6-methoxyphenyl
methyl



4.1088
3-trifluoromethoxy-6-methoxyphenyl
methyl



4.1089
3-nitro-6-methoxyphenyl
methyl



4.1090
3-fluoro-6-ethoxyphenyl
methyl



4.1091
3-chloro-6-ethoxyphenyl
methyl



4.1092
3-bromo-6-ethoxyphenyl
methyl



4.1093
3-methyl-6-ethoxyphenyl
methyl



4.1094
3-cyclopropyl-6-ethoxyphenyl
methyl



4.1095
3-cyano-6-ethoxyphenyl
methyl



4.1096
3-trifluoromethyl-6-ethoxyphenyl
methyl



4.1097
3-methoxy-6-ethoxyphenyl
methyl



4.1098
2,6-diethoxyphenyl
methyl



4.1099
3-trifluoromethoxy-6-ethoxyphenyl
methyl



4.1100
3-nitro-6-ethoxyphenyl
methyl



4.1101
3-fluoro-6-isopropoxyphenyl
methyl



4.1102
3-chloro-6-isopropoxyphenyl
methyl



4.1103
3-bromo-6-isopropoxyphenyl
methyl



4.1104
3-methyl-6-isopropoxyphenyl
methyl



4.1105
3-cyclopropyl-6-isopropoxyphenyl
methyl



4.1106
3-cyano-6-isopropoxyphenyl
methyl



4.1107
3-trifluoromethyl-6-isopropoxyphenyl
methyl



4.1108
3-methoxy-6-isopropoxyphenyl
methyl



4.1109
3-ethoxy-6-isopropoxyphenyl
methyl



4.1110
3-trifluoromethoxy-6-isopropoxyphenyl
methyl



4.1111
3-nitro-6-isopropoxyphenyl
methyl



4.1112
3-fluoro-6-trifluoromethoxyphenyl
methyl



4.1113
3-chloro-6-trifluoromethoxyphenyl
methyl



4.1114
3-bromo-6-trifluoromethoxyphenyl
methyl



4.1115
3-methyl-6-trifluoromethoxyphenyl
methyl



4.1116
3-cyclopropyl-6-trifluoromethoxyphenyl
methyl



4.1117
3-cyano-6-trifluoromethoxyphenyl
methyl



4.1118
3-trifluoromethyl-6-trifluoromethoxy-
methyl




phenyl




4.1119
3-methoxy-6-trifluoromethoxyphenyl
methyl



4.1120
3-ethoxy-6-trifluoromethoxyphenyl
methyl



4.1121
3,6-bis(trifluoromethoxy)phenyl
methyl



4.1122
3-nitro-6-trifluoromethoxyphenyl
methyl



4.1123
3-fluoro-6-difluoromethoxyphenyl
methyl



4.1124
3-chloro-6-difluoromethoxyphenyl
methyl



4.1125
3-bromo-6-difluoromethoxyphenyl
methyl



4.1126
3-methyl-6-difluoromethoxyphenyl
methyl



4.1127
3-cyclopropyl-6-difluoromethoxyphenyl
methyl



4.1128
3-cyano-6-difluoromethoxyphenyl
methyl



4.1129
3-trifluoromethyl-6-difluoromethoxyphenyl
methyl



4.1130
3-methoxy-6-difluoromethoxyphenyl
methyl



4.1131
3-ethoxy-6-difluoromethoxyphenyl
methyl



4.1132
3-trifluoromethoxy-6-difluoromethoxy-
methyl




phenyl




4.1133
3-nitro-6-difluoromethoxyphenyl
methyl



4.1134
3-fluoro-6-nitrophenyl
methyl



4.1135
3-chloro-6-nitrophenyl
methyl



4.1136
3-bromo-6-nitrophenyl
methyl



4.1137
3-methyl-6-nitrophenyl
methyl



4.1138
3-cyclopropyl-6-nitrophenyl
methyl



4.1139
3-cyano-6-nitrophenyl
methyl



4.1140
3-trifluoromethyl-6-nitrophenyl
methyl



4.1141
3-methoxy-6-nitrophenyl
methyl



4.1142
3-ethoxy-6-nitrophenyl
methyl



4.1143
3-trifluoromethoxy-6-nitrophenyl
methyl



4.1144
3-fluoro-6-methylsulfanylphenyl
methyl



4.1145
3-chloro-6-methylsulfanylphenyl
methyl



4.1146
3-bromo-6-methylsulfanylphenyl
methyl



4.1147
3-methyl-6-methylsulfanylphenyl
methyl



4.1148
3-ethyl-6-methylsulfanylphenyl
methyl



4.1149
3-cyclopropyl-6-methylsulfanylphenyl
methyl



4.1150
3-cyano-6-methylsulfanylphenyl
methyl



4.1151
3-trifluoromethyl-6-methylsulfanylphenyl
methyl



4.1152
3-methoxy-6-methylsulfanylphenyl
methyl



4.1153
3-ethoxy-6-methylsulfanylphenyl
methyl



4.1154
3-trifluoromethoxy-6-methylsulfanylphenyl
methyl



4.1155
3-nitro-6-methylsulfanylphenyl
methyl



4.1156
2,3,4-trifluorophenyl
methyl



4.1157
2,3,4-trichlorophenyl
methyl



4.1158
2,3,4-trimethylphenyl
methyl



4.1159
2-fluoro-2-chloro-5-trifluoromethylphenyl
methyl



4.1160
2,3,5-trifluorophenyl
methyl



4.1161
2,3,5-trichlorophenyl
methyl



4.1162
2,3,5-trimethylphenyl
methyl



4.1163
2,3-dichloro-5-methoxyphenyl
methyl



4.1164
2,3,6-trifluorophenyl
methyl



4.1165
2,3,6-trichlorophenyl
methyl



4.1166
2,3,6-trimethylphenyl
methyl



4.1167
3,4,5-trifluorophenyl
methyl



4.1168
3,4,6-trifluorophenyl
methyl



4.1169
3,4,6-trichlorophenyl
methyl



4.1170
3,4,6-trichlorophenyl
ethyl



4.1171
3,4,6-trichlorophenyl
CN



4.1172
3,4,6-trichlorophenyl
vinyl



4.1173
3,4,6-trichlorophenyl
fluoromethyl



4.1174
3,4,6-trichlorophenyl
methylcarbonyl



4.1175
3,4,6-trichlorophenyl
hydroxymethyl



4.1176
3,4,6-trichlorophenyl
ethynyl



4.1177
3,4,5-trimethylphenyl
methyl



4.1178
3,5-dimethyl-4-fluorophenyl
methyl



4.1179
3,5-dichloro-4-methoxyphenyl
methyl



4.1180
3,5-difluoro-4-chlorophenyl
methyl



4.1181
3,5-dichloro-4-hydroxyphenyl
methyl



4.1182
3,5-trifluoromethyl-4-chlorophenyl
methyl



4.1183
3,4,6-trifluorophenyl
methyl



4.1184
3,4,6-trichlorophenyl
methyl



4.1185
3,4,6-trimethylphenyl
methyl



4.1186
2,3,4,5-pentafluorophenyl
methyl









B. FORMULATION EXAMPLES
1. Dusting Products
A dusting product is obtained by mixing 10 parts by weight of a compound of the formula (I) and 90 parts by weight of talc as an inert substance and comminuting the mixture in a hammer mill.
2. Dispersible Powder
A readily water-dispersible wettable powder is obtained by mixing 25 parts by weight of a compound of the formula (I), 64 parts by weight of kaolin-containing quartz as an inert substance, 10 parts by weight of potassium lignosulfonate and 1 part by weight of sodium oleoylmethyltaurate as a wetting agent and dispersant, and grinding the mixture in a pinned-disk mill.
3. Dispersion Concentrate
A readily water-dispersible dispersion concentrate is obtained by mixing 20 parts by weight of a compound of the formula (I) with 6 parts by weight of alkylphenol polyglycol ether (®Triton X 207), 3 parts by weight of isotridecanol polyglycol ether (8 EO) and 71 parts by weight of paraffinic mineral oil (boiling range for example about 255 to above 277° C.) and grinding the mixture in a ball mill to a fineness of below 5 microns.
4. Emulsifiable Concentrate
An emulsifiable concentrate is obtained from 15 parts by weight of a compound of the formula (I), 75 parts by weight of cyclohexanone as a solvent and 10 parts by weight of ethoxylated nonylphenol as an emulsifier.
5. Water-Dispersible Granules
Water-dispersible granules are obtained by mixing
75 parts by weight of a compound of the formula (I),
10 parts by weight of calcium lignosulfonate,
5 parts by weight of sodium laurylsulfate,
3 parts by weight of polyvinyl alcohol and
7 parts by weight of kaolin,
grinding the mixture in a pinned-disk mill, and granulating the powder in a fluidized bed by spray application of water as a granulating liquid.
Water-dispersible granules are also obtained by homogenizing and precomminuting, in a colloid mill,
25 parts by weight of a compound of the formula (I),
5 parts by weight of sodium 2,2′-dinaphthylmethane-6,6′-disulfonate,
2 parts by weight of sodium oleoylmethyltaurinate,
1 part by weight of polyvinyl alcohol,
17 parts by weight of calcium carbonate and
50 parts by weight of water,
then grinding the mixture in a bead mill and atomizing and drying the suspension thus obtained in a spray tower by means of a one-phase nozzle.
C. BIOLOGICAL EXAMPLES
1. Pre-Emergence Herbicidal Action Against Harmful Plants
Seeds or rhizome pieces of mono- and dicotyledonous harmful plants are placed in sandy loam soil in pots having a diameter of 9 to 13 cm and covered with soil. The herbicides, formulated as emulsifiable concentrates or dusting products, are then applied in various dosages in the form of aqueous dispersions or suspensions or emulsions at an application rate of 300 to 800 I of water/ha (converted) to the surface of the covering soil. For further cultivation of the plants, the pots are then kept under optimal conditions in a greenhouse. After the test plants have been left to stand in the greenhouse for 3 to 4 weeks under optimal growth conditions, the activity of the inventive compounds is scored visually. For example, compounds No. 1.1.054, 1.1.2008, 1.1.462, 1.1.463, 1.1.494, 1.1.520, 1.1.527, 1.1.580, 1.1.603, 1.3.470, 1.2.471, 1.3.001, 1.3.473, 2.1.466, 2.1.478, 1.3.527, 2.1.522, 2.1.526, 2.1.546, 2.1.588, 2.2.472, 2.3.475, 2.3.528, 2.3.572, 2.6.462, 2.6.463, 2.6.464, 2.6.465, 2.6.467, 2.6.468, 2.6.469, 2.6.470, 2.6.471, 2.6.473, 2.6.474, 2.6.479, 2.6.480, 2.6.481, 2.6.486, 2.6.488, 2.6.489, 2.6.490, 2.6.541, 2.6.547, 2.6.553, 2.6.555 and 2.6.561 at an application rate of 320 grams per hectare each showed at least 80% efficacy against Avena fatua. Compounds No. 1.1.471, 1.1.519, 1.1.540, 1.1.580, 1.3.476, 1.3.571, 1.3.644, 2.1.523, 2.1.524, 2.1.532, 2.1.569, 2.2.530, 2.3.527, 2.3.534, 2.6.545, 2.6.548, 2.6.549, 2.6.550 and 2.6.552 at an application rate of 320 grams per hectare each showed at least 80% efficacy against Stellaria media. Compounds No. 1.1.566, 1.3.474, 2.1.531, 2.6.475 and 2.6.478 at an application rate of 320 grams per hectare each showed at least 80% efficacy against Lolium multiflorum. 
2. Post-Emergence Herbicidal Action Against Harmful Plants
Seeds of monocotyledonous and dicotyledonous harmful plants are laid out in sandy loam in cardboard pots, covered with soil and cultivated in a greenhouse under good growth conditions. Two to three weeks after sowing, the test plants are treated at the three-leaf stage. The inventive compounds, formulated as wettable powders or as emulsion concentrates, are sprayed onto the surface of the green parts of the plants at an application rate of 600 to 800 l of water/ha (converted). After the test plants have been left to stand in the greenhouse for 3 to 4 weeks under optimal growth conditions, the activity of the inventive compounds is scored visually. For example, compounds No. 1.1.2009, 1.1.462, 1.1.463, 1.1.494, 1.1.519, 1.1.520, 1.1.529, 1.1.540, 1.1.566, 1.1.580, 1.2.470, 1.2.471, 1.2.525, 1.3.001, 1.3.004, 1.3.470, 1.3.472, 1.3.474, 1.3.473, 1.3.476, 1.3.486, 1.3.527, 1.3.528, 1.3.571, 1.3.644, 2.1.466, 2.1.478, 2.1.522, 2.1.526, 2.1.527, 2.1.530, 2.1.532, 2.1.546, 2.1.570, 2.1.588, 2.2.471, 2.2.472, 2.2.527, 2.3.475, 2.3.476, 2.3.527, 2.3.528, 2.3.534, 2.3.535, 2.3.572, 2.3.645, 2.6.009, 2.6.462, 2.6.463, 2.6.464, 2.6.467, 2.6.468, 2.6.469, 2.6.470, 2.6.471, 2.6.473, 2.6.474, 2.6.475, 2.6.476, 2.6.477, 2.6.478, 2.6.479, 2.6.480, 2.6.481, 2.6.486, 2.6.488, 2.6.489, 2.6.490, 2.6.494, 2.6.495, 2.6.541, 2.6.545, 2.6.546, 2.6.547, 2.6.548, 2.6.549, 2.6.552, 2.6.553, 2.6.554, 2.6.555 and 2.6.561 at an application rate of 320 grams per hectare each showed at least 80% efficacy against Avena fatua. 
Compounds No. 1.1.2008, 1.1.1211, 1.1.527, 1.1.502, 1.1.925, 1.2.002, 1.2.528, 2.1.523, 2.1.524, 2.1.531, 2.1.670, 2.2.475, 2.6.465 and 2.6.550
at an application rate of 320 grams per hectare each showed at least 80% efficacy against Veronica persica.

## Claims

1. A 3-phenylisoxazoline derivative and/or salt thereof, of formula (I)




in which
R1 and R2 are each independently hydrogen, fluorine, chlorine, bromine, iodine, cyano, or (C1-C4)-alkyl or (C1-C4)-alkoxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine and cyano,

or
R1 and R2 together with the carbon atom to which they are bonded form a saturated or partly or fully unsaturated three-, four- or five-membered ring formed from q carbon atoms and p oxygen atoms;
R3 is fluorine, chlorine, cyano, (C1-C3)-alkylcarbonyloxy or S(O)nR5,
or (C1-C6)-alkyl, (C3-C6)-cycloalkyl, (C2-C6)-alkenyl or (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano, (C1-C4)-alkoxy and hydroxyl,
or (C1-C6)-alkylcarbonyl, (C2-C6)-alkenylcarbonyl or (C3-C6)-cycloalkylcarbonyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, and cyano;
R5 is (C1-C6)-alkyl or (C3-C6)-cycloalkyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and hydroxyl;
R6 is hydrogen or R5;
R7 is hydrogen or (C1-C6)-alkyl, (C3-C6)-cycloalkyl, (C2-C4)-alkenyl or (C2-C4)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano and (C1-C2)-alkoxy;
R8 is R7;
W* is COOH, COOY, CN or CHO;
Y is (C1-C8)-alkyl which is substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano, hydroxyl and COO—(C1-C8)-alkyl and which is interrupted by n heteroatoms from the group consisting of oxygen, sulfur and nitrogen, or
a radical from the group consisting of (cyclohex-2-en-1-one)-3-yl, (propan-1-ol)-3-yl, (2,2-dimethylpropan-1-ol)-3-yl, (methyl 2,2-dimethylpropanoate)-3-yl, (methyl propanoate)-3-yl, (ethyl propanoate)-3-yl, (ethyl butanoate)-3-yl, (ethyl (3R)-4,4,4-trifluorobutanoate)-3-yl, (butan-2-one)-4-yl, (3-methylbutan-2-one)-4-yl, (pent-3-en-2-one)-4-yl,((2S)-dimethyl butanedioate)-2-yl, (dimethyl pentanedioate)-3-yl, (methyl (2R)-2-methylpropanoate)-3-yl, 4-methoxycarbonylbenzyl, 3,5-difluorobenzyl, 3,4-difluorobenzyl, 2,6-difluorobenzyl, 5-methylpyridin-3-ylmethyl, tetrahydrofuran-3-yl and (butan-1-ol)-4-yl;
X2, X4 and X6 are each independently hydrogen, fluorine, chlorine, bromine, iodine, cyano, nitro,
or (C1-C4)-alkyl, (C3-C5)-cycloalkyl, (C2-C4)-alkenyl, (C2-C4)-alkynyl, (C1-C4)-alkoxy, (C2-C4)-alkenyloxy, (C2-C4)-alkynyloxy or (C1-C4)-alkylcarbonyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C4)-alkoxy;
X3 is fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8OSO2R5, CONR6R8, COR6, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)nR5, SO2NR6R8, OSO2NR6R8,
or (C1-C6)-alkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano,
or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy;
X5 is hydrogen, fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8SO2R5, CONR6R8, COR6, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)n R5, SO2NR6R8, OSO2NR6R8,
or (C1-C6)-alkyl, (C3-C5)-cycloalkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano,
or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy, (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy;
m is 0, 1, 2, 3, 4 or 5;
n is 0, 1 or 2;
p is 0 or 1;
q is 3, 4 or 5;

with the proviso that
a) X3 and X4 are not both substituted or unsubstituted alkoxy,
b) in the compounds in which R3 is methyl and W* is COOH, X5 is not hydrogen, and
c) the compounds methyl 3-(3-cyanophenyl)-5-(isopropoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 5-(butoxymethyl)-3-(3-cyanophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 3-(3-cyanophenyl)-5-(methoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 3-(3-cyanophenyl)-5-(2-methoxyethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, 3-(3-cyanophenyl)-5-(trifluoromethyl)-4,5-dihydro-1,2-oxazole-5-carboxylic acid, methyl 3-(3-cyanophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate, ethyl 3-(3-cyanophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 5-methyl-3-(3-nitrophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 3-(3,5-di-tert-butyl-4-hydroxyphenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate and ethyl 3-(3-chlorophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate are excluded.

2. A 3-phenylisoxazoline derivative and/or salt as claimed in claim 1, in which
R1 and R2 are each hydrogen,
R3 is (C1-C6)-alkyl, (C1-C4)-alkoxy-(C1-C4)-alkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl, halo-(C1-C6)-alkyl or halo-(C2-C6)-alkenyl;
R5 is (C1-C6)-alkyl or (C3-C6)-cycloalkyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and hydroxyl;
R6 is hydrogen or R5;
R7 is hydrogen or (C1-C6)-alkyl, (C3-C6)-cycloalkyl, (C2-C4)-alkenyl or (C2-C4)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano and (C1-C2)-alkoxy;
R8 is R7;
W* is COOH or COOP;
Y is (C1-C6)-alkyl which is substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano, hydroxyl and COO—(C1-C4)-alkyl and which is interrupted by n oxygen atoms, or
a radical from the group consisting of (cyclohex-2-en-1-one)-3-yl, (propan-1-ol)-3-yl, (2,2-dimethylpropan-1-ol)-3-yl, (methyl 2,2-dimethylpropanoate)-3-yl, (methyl propanoate)-3-yl, (ethyl propanoate)-3-yl, (ethyl butanoate)-3-yl, (ethyl (3R)-4,4,4-trifluorobutanoate)-3-yl, (butan-2-one)-4-yl, (3-methylbutan-2-one)-4-yl, (pent-3-en-2-one)-4-yl,((2S)-dimethyl butanedioate)-2-yl, (dimethyl pentanedioate)-3-yl, (methyl (2R)-2-methylpropanoate)-3-yl, 4-methoxycarbonylbenzyl, 3,5-difluorobenzyl, 3,4-difluorobenzyl, 2,6-difluorobenzyl, 5-methylpyridin-3-ylmethyl, tetrahydrofuran-3-yl and (butan-1-ol)-4-yl;
X2, X4 and X6 are each independently hydrogen, fluorine, chlorine, bromine, iodine, cyano, nitro,
or (C1-C4)-alkyl, (C3-C5)-cycloalkyl, (C2-C4)-alkenyl, (C2-C4)-alkynyl, (C1-C4)-alkoxy, (C2-C4)-alkenyloxy, (C2-C4)-alkynyloxy or (C1-C4)-alkylcarbonyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C4)-alkoxy;
X3 is fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8SO2R5, CONR6R8, COR6, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)nR5, SO2NR6R8, OSO2NR6R8,
or (C1-C6)-alkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano,
or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy;
X5 is hydrogen, fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8SO2R5, CONR6R8, COR6, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)nR5, SO2NR6R8, OSO2NR6R8,
or (C1-C6)-alkyl, (C3-C5)-cycloalkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano,
or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy, (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy;
m is 0, 1, 2, 3, 4 or 5;
n is 0, 1 or 2;

with the proviso that
a) X3 and X4 are not both substituted or unsubstituted alkoxy,
b) in the compounds in which R3 is methyl and W* is COOH, X5 is not hydrogen, and
c) the compounds methyl 3-(3-cyanophenyl)-5-(isopropoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 5-(butoxymethyl)-3-(3-cyanophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 3-(3-cyanophenyl)-5-(methoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 3-(3-cyanophenyl)-5-(2-methoxyethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, 3-(3-cyanophenyl)-5-(trifluoromethyl)-4,5-dihydro-1,2-oxazole-5-carboxylic acid, methyl 3-(3-cyanophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate, ethyl 3-(3-cyanophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 5-methyl-3-(3-nitrophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 3-(3,5-di-tert-butyl-4-hydroxyphenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate and ethyl 3-(3-chlorophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate are excluded.

3. A 3-phenylisoxazoline derivative and/or salt as claimed in claim 1, in which
R1 and R2 are each hydrogen,
R3 is (C1-C4)-alkyl, (C1-C4)-alkoxy-(C1-C4)-alkyl, vinyl, (C2-C4)-alkynyl, halo-(C1-C4)-alkyl or halo-(C2-C4)-alkenyl;
R5 is methyl or ethyl;
R6 is hydrogen or R5;
R7 is hydrogen or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine;
R8 is R7;
W* is COOH or COOP;
Y is (C1-C6)-alkyl which is substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano, hydroxyl and COO—(C1-C4)-alkyl and which is interrupted by n oxygen atoms, or
a radical from the group consisting of (cyclohex-2-en-1-one)-3-yl, (propan-1-ol)-3-yl, (2,2-dimethyl propan-1-ol)-3-yl, (methyl 2,2-dimethylpropanoate)-3-yl, (methyl propanoate)-3-yl, (ethyl propanoate)-3-yl, (ethyl butanoate)-3-yl, (ethyl (3R)-4,4,4-trifluorobutanoate)-3-yl, (butan-2-one)-4-yl, (3-methylbutan-2-one)-4-yl, (pent-3-en-2-one)-4-yl,((2S)-dimethyl butanedioate)-2-yl, (dimethyl pentanedioate)-3-yl, (methyl (2R)-2-methylpropanoate)-3-yl, 4-methoxycarbonylbenzyl, 3,5-difluorobenzyl, 3,4-difluorobenzyl, 2,6-difluorobenzyl, 5-methylpyridin-3-ylmethyl, tetrahydrofuran-3-yl and (butan-1-ol)-4-yl;
X2, X4 and X6 are each independently hydrogen, fluorine, or chlorine,
or (C1-C4)-alkyl or (C1-C4)-alkoxy each substituted by m radicals from the group consisting of fluorine, chlorine, cyano and (C1-C4)-alkoxy;
X3 is fluorine, chlorine, bromine, cyano,
or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine,
or (C1-C6)-alkoxy substituted by m radicals from the group consisting of fluorine and chlorine;
X5 is hydrogen, fluorine, chlorine, bromine, cyano,
or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine,
or (C1-C6)-alkoxy substituted by m radicals from the group consisting of fluorine and chlorine;
m is 0, 1, 2 or 3;
n is 0, 1 or 2;

with the proviso that
a) X3 and X4 are not both substituted or unsubstituted alkoxy,
b) in the compounds in which R3 is methyl and W* is COOH, X5 is not hydrogen, and
c) the compounds methyl 3-(3-cyanophenyl)-5-(isopropoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 5-(butoxymethyl)-3-(3-cyanophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 3-(3-cyanophenyl)-5-(methoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 3-(3-cyanophenyl)-5-(2-methoxyethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, 3-(3-cyanophenyl)-5-(trifluoromethyl)-4,5-dihydro-1,2-oxazole-5-carboxylic acid, methyl 3-(3-cyanophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate, ethyl 3-(3-cyanophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 5-methyl-3-(3-nitrophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 3-(3,5-di-tert-butyl-4-hydroxyphenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate and ethyl 3-(3-chlorophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate are excluded.

4. A 3-phenylisoxazoline derivative and/or salt as claimed in claim 3, in which
X5 is fluorine, chlorine, bromine, cyano,
or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine,
or (C1-C6)-alkoxy substituted by m radicals from the group consisting of fluorine and chlorine.

5. A herbicidal composition, comprising a herbicidally active content of at least one compound of the formula (I) and/or salt




in which
R1 and R2 are each independently hydrogen, fluorine, chlorine, bromine, iodine, cyano, or (C1-C4)-alkyl or (C1-C4)-alkoxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine and cyano,

or
R1 and R2 together with the carbon atom to which they are bonded form a saturated or partly or fully unsaturated three-, four- or five-membered ring formed from q carbon atoms and p oxygen atoms;
R3 is fluorine, chlorine, cyano, (C1-C3)-alkylcarbonyloxy or S(O)nR5,
or (C1-C6)-alkyl, (C3-C6)-cycloalkyl, (C2-C6)-alkenyl or (C2-C6)-alkenyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano, (C1-C4)-alkoxy and hydroxyl,
or (C1-C6)-alkylcarbonyl, (C2-C6)-alkenylcarbonyl or (C3-C6)-cycloalkylcarbonyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C6)-alkoxy;
R5 is (C1-C6)-alkyl or (C3-C6)-cycloalkyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and hydroxyl;
R6 is hydrogen or R5,
R7 is hydrogen or (C1-C6)-alkyl, (C3-C6)-cycloalkyl, (C2-C4)-alkenyl or (C2-C4)-alkenyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano and (C1-C2)-alkoxy;
R8 is R7,
W* is COOH, COOY, CN or CHO;
Y is (C1-C8)-alkyl which is substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano, hydroxyl and COO—(C1-C8)-alkyl and which is interrupted by n heteroatoms from the group consisting of oxygen, sulfur and nitrogen, or
a radical from the group consisting of (cyclohex-2-en-1-one)-3-yl, (propan-1-ol)-3-yl, (2,2-dimethylpropan-1-ol)-3-yl, (methyl 2,2-dimethylpropanoate)-3-yl, (methyl propanoate)-3-yl, (ethyl propanoate)-3-yl, (ethyl butanoate)-3-yl, (ethyl (3R)-4,4,4-trifluorobutanoate)-3-yl, (butan-2-one)-4-yl, (3-methylbutan-2-one)-4-yl, (pent-3-en-2-one)-4-yl,((2S)-dimethyl butanedioate)-2-yl, (dimethyl pentanedioate)-3-yl, (methyl (2R)-2-methylpropanoate)-3-yl, 4-methoxycarbonylbenzyl, 3,5-difluorobenzyl, 3,4-difluorobenzyl, 2,6-difluorobenzyl, 5-methylpyridin-3-ylmethyl, tetrahydrofuran-3-yl and (butan-1-ol)-4-yl;
X2, X4 and X6 are each independently hydrogen, fluorine, chlorine, bromine, iodine, cyano, nitro,
or (C1-C4)-alkyl, (C3-C5)-cycloalkyl, (C2-C4)-alkenyl, (C2-C4)-alkynyl, (C1-C4)-alkoxy, (C2-C4)-alkenyloxy, (C2-C4)-alkynyloxy or (C1-C4)-alkylcarbonyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C4)-alkoxy;
X3 is fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8SO2R5, CONR6R8, COR6, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)nR5, SO2NR6R8, OSO2NR6R8,
or (C1-C6)-alkyl, (C3-C5)-cycloalkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano,
or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy;
X5 is hydrogen, fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8SO2R5, CONR6R8, COR6, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)nR5, SO2NR6R8, OSO2NR6R8,
or (C1-C6)-alkyl, (C3-C5)-cycloalkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano,
or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy, (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy;
m is 0, 1, 2, 3, 4 or 5;
n is 0, 1 or 2;
p is 0 or 1;
q is 3, 4 or 5;

with the proviso that
a) X3 and X4 are not both substituted or unsubstituted alkoxy,
b) in the compounds in which R3 is methyl and W* is COOH, X5 is not hydrogen, and
c) the compounds methyl 3-(3-cyanophenyl)-5-(isopropoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 5-(butoxymethyl)-3-(3-cyanophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 3-(3-cyanophenyl)-5-(methoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 3-(3-cyanophenyl)-5-(2-methoxyethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, 3-(3-cyanophenyl)-5-(trifluoromethyl)-4,5-dihydro-1,2-oxazole-5-carboxylic acid, methyl 3-(3-cyanophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate, ethyl 3-(3-cyanophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 5-methyl-3-(3-nitrophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 3-(3,5-di-tert-butyl-4-hydroxyphenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate and ethyl 3-(3-chlorophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate are excluded.

6. The herbicidal composition as claimed in claim 5 in a mixture with one or more formulation auxiliaries.

7. The herbicidal composition as claimed in claim 5, comprising at least one further pesticidally active substance selected from the group consisting of insecticides, acaricides, herbicides, fungicides, safeners and growth regulators.

8. The herbicidal composition as claimed in claim 7, comprising a safener.

9. The herbicidal composition as claimed in claim 8, in which the safener is selected from the group consisting of mefenpyr-diethyl, cyprosulfamide, isoxadifen-ethyl, cloquintocet-mexyl, benoxacor and dichlormid.

10. The herbicidal composition as claimed in claim 7, comprising a further herbicide.

11. A method for controlling one or more unwanted plants comprising applying an effective amount of at least one compound of formula (Ia) to the one or more plants and/or a site of unwanted vegetation, wherein the compound of formula (Ia) is a 3-phenylisoxazoline derivative of formula (Ia)




in which
R1 and R2 are each independently hydrogen, fluorine, chlorine, bromine, iodine, cyano, or (C1-C4)-alkyl or (C1-C4)-alkoxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine and cyano,

or
R1 and R2 together with the carbon atom to which they are bonded form a saturated or partly or fully unsaturated three-, four- or five-membered ring formed from q carbon atoms and p oxygen atoms;
R3 is fluorine, chlorine, cyano, (C1-C3)-alkylcarbonyloxy or S(O)nR5,
or (C1-C6)-alkyl, (C3-C6)-cycloalkyl, (C2-C6)-alkenyl or (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano, (C1-C4)-alkoxy and hydroxyl,
or (C1-C6)-alkylcarbonyl, (C2-C6)-alkenylcarbonyl or (C3-C6)-cycloalkylcarbonyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C6)-alkoxy;
R5 is (C1-C6)-alkyl or (C3-C6)-cycloalkyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and hydroxyl;
R6 is hydrogen or R5;
R7 is hydrogen or (C1-C6)-alkyl, (C3-C6)-cycloalkyl, (C2-C4)-alkenyl or (C2-C4)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano and (C1-C2)-alkoxy;
R8 is R7;
W* is COOH, COOY, CN or CHO;
Y is (C1-C8)-alkyl which is substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano, hydroxyl and COO—(C1-C8)-alkyl and which is interrupted by n heteroatoms from the group consisting of oxygen, sulfur and nitrogen, or
a radical from the group consisting of (cyclohex-2-en-1-one)-3-yl, (propan-1-ol)-3-yl, (2,2-dimethylpropan-1-ol)-3-yl, (methyl 2,2-dimethylpropanoate)-3-yl, (methyl propanoate)-3-yl, (ethyl propanoate)-3-yl, (ethyl butanoate)-3-yl, (ethyl (3R)-4,4,4-trifluorobutanoate)-3-yl, (butan-2-one)-4-yl, (3-methylbutan-2-one)-4-yl, (pent-3-en-2-one)-4-yl,((2S)-dimethyl butanedioate)-2-yl, (dimethyl pentanedioate)-3-yl, (methyl (2R)-2-methylpropanoate)-3-yl, 4-methoxycarbonylbenzyl, 3,5-difluorobenzyl, 3,4-difluorobenzyl, 2,6-difluorobenzyl, 5-methylpyridin-3-ylmethyl, tetrahydrofuran-3-yl and (butan-1-ol)-4-yl;
X2, X4 and X6 are each independently hydrogen, fluorine, chlorine, bromine, iodine, cyano, nitro,
or (C1-C4)-alkyl, (C3-C5)-cycloalkyl, (C2-C4)-alkenyl, (C2-C4)-alkynyl, (C1-C4)-alkoxy, (C2-C4)-alkenyloxy, (C2-C4)-alkynyloxy or (C1-C4)-alkylcarbonyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine iodine, cyano and (C1-C4)-alkoxy;
X3 is fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8SO2R5, CONR6R8, CORE, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)nR5, SO2NR6R8, OSO2NR6R8,
or (C1-C6)-alkyl, (C3-C5)-cycloalkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano,
or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy;
X5 is hydrogen, fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8SO2R5, CONR6R8, CORE, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)n R5, SO2NR6R8, OSO2NR6R8,
or (C1-C6)-alkyl, (C3-C5)-cycloalkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano,
or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy, (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy;
m is 0, 1, 2, 3, 4 or 5;
n is 0, 1 or 2;
p is 0 or 1;
q is 3, 4 or 5.

12. The method as claimed in claim 11, in which
R1 and R2 are each hydrogen,
R3 is (C1-C6)-alkyl, (C1-C4)-alkoxy-(C1-C4)-alkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl, halo-(C1-C6)-alkyl or halo-(C2-C6)-alkenyl;
R5 is (C1-C6)-alkyl or (C3-C6)-cycloalkyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and hydroxyl;
R6 is hydrogen or R5;
R7 is hydrogen or (C1-C6)-alkyl, (C3-C6)-cycloalkyl, (C2-C4)-alkenyl or (C2-C4)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano and (C1-C2)-alkoxy;
R8 is R7;
W* is COOH or COOP;
Y is (C1-C6)-alkyl which is substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano, hydroxyl and COO—(C1-C4)-alkyl and which is interrupted by n oxygen atoms, or
a radical from the group consisting of (cyclohex-2-en-1-one)-3-yl, (propan-1-ol)-3-yl, (2,2-dimethylpropan-1-ol)-3-yl, (methyl 2,2-dimethylpropanoate)-3-yl, (methyl propanoate)-3-yl, (ethyl propanoate)-3-yl, (ethyl butanoate)-3-yl, (ethyl (3R)-4,4,4-trifluorobutanoate)-3-yl, (butan-2-one)-4-yl, (3-methylbutan-2-one)-4-yl, (pent-3-en-2-one)-4-yl,((2S)-dimethyl butanedioate)-2-yl, (dimethyl pentanedioate)-3-yl, (methyl (2R)-2-methylpropanoate)-3-yl, 4-methoxycarbonylbenzyl, 3,5-difluorobenzyl, 3,4-difluorobenzyl, 2,6-difluorobenzyl, 5-methylpyridin-3-ylmethyl, tetrahydrofuran-3-yl and (butan-1-ol)-4-yl;
X2, X4 and X6 are each independently hydrogen, fluorine, chlorine, bromine, iodine, cyano, nitro,
or (C1-C4)-alkyl, (C3-C5)-cycloalkyl, (C2-C4)-alkenyl, (C2-C4)-alkynyl, (C1-C4)-alkoxy, (C2-C4)-alkenyloxy, (C2-C4)-alkynyloxy or (C1-C4)-alkylcarbonyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C4)-alkoxy;
X3 is fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8SO2R5, CONR6R8, COR6, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)nR5, SO2NR6R8, OSO2NR6R8,
or (C1-C6)-alkyl, (C3-C5)-cycloalkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano,
or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy, (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy;
X5 is hydrogen, fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8SO2R5, CONR6R8, COR6, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)nR5, SO2NR6R8, OSO2NR6R8,
or (C1-C6)-alkyl, (C3-C5)-cycloalkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano,
or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy, (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy;
m is 0, 1, 2, 3, 4 or 5;
n is 0, 1 or 2.

13. The method as claimed in claim 11, in which
R1 and R2 are each hydrogen,
R3 is (C1-C4)-alkyl, (C1-C4)-alkoxy-(C1-C4)-alkyl, vinyl, (C2-C4)-alkynyl, halo-(C1-C4)-alkyl or halo-(C2-C4)-alkenyl;
R5 is methyl or ethyl,
R6 is hydrogen or R5;
R7 is hydrogen or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine;
R8 is R7;
W* is COOH or COOP;
Y is (C1-C6)-alkyl which is substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano, hydroxyl and COO—(C1-C4)-alkyl and which is interrupted by n oxygen atoms;
X2, X4 and X6 are each independently hydrogen, fluorine, or chlorine,
or (C1-C4)-alkyl or (C1-C4)-alkoxy each substituted by m radicals from the group consisting of fluorine, chlorine, cyano and C1-C4)-alkoxy;
X3 is fluorine, chlorine, bromine, cyano,
or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine,
or (C1-C6)-alkoxy substituted by m radicals from the group consisting of fluorine and chlorine;
X5 is hydrogen, fluorine, chlorine, bromine, cyano,
or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine,
or (C1-C6)-alkoxy substituted by m radicals from the group consisting of fluorine and chlorine;
m is 0, 1, 2 or 3;
n is 0, 1 or 2.

14. The method as claimed in claim 13, in which
X5 is fluorine, chlorine, bromine, cyano,
or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine,
or (C1-C6)-alkoxy substituted by m radicals from the group consisting of fluorine and chlorine.

15. A method for preparing a herbicidally active 3-phenylisoxazoline-5-carboxamide and/or 3-phenylisoxazoline-5-thioamide comprising employing a 3 phenylisoxazoline derivative of formula (Ia)




in which
R1 and R2 are each independently hydrogen, fluorine, chlorine, bromine, iodine, cyano, or (C1-C4)-alkyl or (C1-C4)-alkoxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine and cyano,

or
R1 and R2 together with the carbon atom to which they are bonded form a saturated or partly or fully unsaturated three-, four- or five-membered ring formed from q carbon atoms and p oxygen atoms;
R3 is fluorine, chlorine, cyano, (C1-C3)-alkylcarbonyloxy or S(O)nR5,
or (C1-C6)-alkyl, (C3-C6)-cycloalkyl, (C2-C6)-alkenyl or (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano, (C1-C4)-alkoxy and hydroxyl,
or (C1-C6)-alkylcarbonyl, (C2-C6)-alkenylcarbonyl or (C3-C6)-cycloalkylcarbonyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C6)-alkoxy;
R5 is (C1-C6)-alkyl or (C3-C6)-cycloalkyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and hydroxyl;
R6 is hydrogen or R5;
R7 is hydrogen or (C1-C6)-alkyl, (C3-C6)-cycloalkyl, (C2-C4)-alkenyl or (C2-C4)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano and (C1-C2)-alkoxy;
R8 is R7;
W* is COOH, COOY, CN or CHO;
Y is (C1-C8)-alkyl which is substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano, hydroxyl and COO—(C1-C8)-alkyl and which is interrupted by n heteroatoms from the group consisting of oxygen, sulfur and nitrogen, or
a radical from the group consisting of (cyclohex-2-en-1-one)-3-yl, (propan-1-ol)-3-yl, (2,2-dimethylpropan-1-ol)-3-yl, (methyl 2,2-dimethylpropanoate)-3-yl, (methyl propanoate)-3-yl, (ethyl propanoate)-3-yl, (ethyl butanoate)-3-yl, (ethyl (3R)-4,4,4-trifluorobutanoate)-3-yl, (butan-2-one)-4-yl, (3-methylbutan-2-one)-4-yl, (pent-3-en-2-one)-4-yl,((2S)-dimethyl butanedioate)-2-yl, (dimethyl pentanedioate)-3-yl, (methyl (2R)-2-methylpropanoate)-3-yl, 4-methoxycarbonylbenzyl, 3,5-difluorobenzyl, 3,4-difluorobenzyl, 2,6-difluorobenzyl, 5-methylpyridin-3-ylmethyl, tetrahydrofuran-3-yl and (butan-1-ol)-4-yl;
X2, X4 and X6 are each independently hydrogen, fluorine, chlorine, bromine, iodine, cyano, nitro,
or (C1-C4)-alkyl, (C3-C5)-cycloalkyl, (C2-C4)-alkenyl, (C2-C4)-alkynyl, (C1-C4)-alkoxy, (C2-C4)-alkenyloxy, (C2-C4)-alkynyloxy or (C1-C4)-alkylcarbonyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine iodine, cyano and (C1-C4)-alkoxy;
X3 is fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8SO2R5, CONR6R8, COR6, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)nR5, SO2NR6R8, OSO2NR6R8,
or (C1-C6)-alkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano,
or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy, (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy;
X5 is hydrogen, fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8SO2R5, CONR6R8, COR6, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)nR5, SO2NR6R8, OSO2NR6R8,
or (C1-C6)-alkyl, (C3-C5)-cycloalkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano,
or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy, (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy;
m is 0, 1, 2, 3, 4 or 5;
n is 0, 1 or 2;
p is 0 or 1;
q is 3, 4 or 5.

16. The method as claimed in claim 15, in which
R1 and R2 are each hydrogen,
R3 is (C1-C6)-alkyl, (C1-C4)-alkoxy-(C1-C4)-alkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl, halo-(C1-C4)-alkyl or halo-(C2-C4)-alkenyl;
R5 is (C1-C6)-alkyl or (C3-C6)-cycloalkyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and hydroxyl;
R6 is hydrogen or R5;
R7 is hydrogen or (C1-C6)-alkyl, (C3-C6)-cycloalkyl, (C2-C4)-alkenyl or (C2-C4)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano and (C1-C2)-alkoxy;
R8 is R7;
W* is COOH or COOP;
Y is (C1-C6)-alkyl which is substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano, hydroxyl and COO—(C1-C4)-alkyl and which is interrupted by n oxygen atoms, or
a radical from the group consisting of (cyclohex-2-en-1-one)-3-yl, (propan-1-ol)-3-yl, (2,2-dimethylpropan-1-ol)-3-yl, (methyl 2,2-dimethylpropanoate)-3-yl, (methyl propanoate)-3-yl, (ethyl propanoate)-3-yl, (ethyl butanoate)-3-yl, (ethyl (3R)-4,4,4-trifluorobutanoate)-3-yl, (butan-2-one)-4-yl, (3-methylbutan-2-one)-4-yl, (pent-3-en-2-one)-4-yl,((2S)-dimethyl butanedioate)-2-yl, (dimethyl pentanedioate)-3-yl, (methyl (2R)-2-methylpropanoate)-3-yl, 4-methoxycarbonylbenzyl, 3,5-difluorobenzyl, 3,4-difluorobenzyl, 2,6-difluorobenzyl, 5-methylpyridin-3-ylmethyl, tetrahydrofuran-3-yl and (butan-1-ol)-4-yl;
X2, X4 and X6 are each independently hydrogen, fluorine, chlorine, bromine, iodine, cyano, nitro,
or (C1-C4)-alkyl, (C3-C5)-cycloalkyl, (C2-C4)-alkenyl, (C2-C4)-alkynyl, (C1-C4)-alkoxy, (C2-C4)-alkenyloxy, (C2-C4)-alkynyloxy or (C1-C4)-alkylcarbonyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C4)-alkoxy;
X3 is fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8SO2R5, CONR6R8, COR6, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)nR5, SO2NR6R8, OSO2NR6R8,
or (C1-C6)-alkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano,
or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy;
X5 is hydrogen, fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8SO2R5, CONR6R8, COR6, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)nR5, SO2NR6R8, OSO2NR6R8,
or (C1-C6)-alkyl, (C3-C5)-cycloalkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano,
or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy, (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy;
m is 0, 1, 2, 3, 4 or 5;
n is 0, 1 or 2.

17. The method as claimed in claim 15, in which R1 and R2 are each hydrogen,
R3 is (C1-C4)-alkyl, (C1-C4)-alkoxy-(C1-C4)-alkyl, vinyl, (C2-C4)-alkynyl, halo-(C1-C4)-alkyl or halo-(C2-C4)-alkenyl;
R5 is methyl or ethyl,
R6 is hydrogen or R5;
R7 is hydrogen or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine;
R8 is R7;
W* is COOH or COOP;
Y is (C1-C6)-alkyl which is substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano, hydroxyl and COO—(C1-C4)-alkyl and which is interrupted by n oxygen atoms, or
a radical from the group consisting of (cyclohex-2-en-1-one)-3-yl, (propan-1-ol)-3-yl, (2,2-dimethylpropan-1-ol)-3-yl, (methyl 2,2-dimethylpropanoate)-3-yl, (methyl propanoate)-3-yl, (ethyl propanoate)-3-yl, (ethyl butanoate)-3-yl, (ethyl (3R)-4,4,4-trifluorobutanoate)-3-yl, (butan-2-one)-4-yl, (3-methylbutan-2-one)-4-yl, (pent-3-en-2-one)-4-yl,((2S)-dimethyl butanedioate)-2-yl, (dimethyl pentanedioate)-3-yl, (methyl (2R)-2-methylpropanoate)-3-yl, 4-methoxycarbonylbenzyl, 3,5-difluorobenzyl, 3,4-difluorobenzyl, 2,6-difluorobenzyl, 5-methylpyridin-3-ylmethyl, tetrahydrofuran-3-yl and (butan-1-ol)-4-yl;
X2, X4 and X6 are each independently hydrogen, fluorine, or chlorine,
or (C1-C4)-alkyl or (C1-C4)-alkoxy each substituted by m radicals from the group consisting of fluorine, chlorine, cyano and (C1-C4)-alkoxy;
X3 is fluorine, chlorine, bromine, cyano,
or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine,
or (C1-C6)-alkoxy substituted by m radicals from the group consisting of fluorine and chlorine;
X5 is hydrogen, fluorine, chlorine, bromine, cyano,
or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine,
or (C1-C6)-alkoxy substituted by m radicals from the group consisting of fluorine and chlorine;
m is 0, 1, 2 or 3;
n is 0, 1 or 2.

18. The method as claimed in claim 17, in which
X5 is fluorine, chlorine, bromine, cyano,
or (C1-C6)-alkyl substituted by m radicals from the group consisting of fluorine and chlorine,
or (C1-C6)-alkoxy substituted by m radicals from the group consisting of fluorine and chlorine.

19. A method for controlling one or more unwanted plants, comprising applying an effective amount of at least one compound of formula (I) as claimed in claim 1 to the one or more plants and/or a site of unwanted vegetation.

20. A method for controlling one or more unwanted plants, comprising applying an effective amount of the composition as claimed in claim 5 to the one or more unwanted plants and/or site of unwanted vegetation.

21. A method for controlling one or more unwanted plants in one or more crops of one or more useful plants, comprising applying an effective amount of the compound as claimed in claim 2 to the one or more unwanted plants and/or site of unwanted vegetation.

22. The method as claimed in claim 21, wherein the one or more useful plants are one or more transgenic useful plants.

23. The 3-phenylisoxazoline derivative as claimed in claim 1, which is compound 1.1.462, in which
R1 and R2 are each hydrogen,
R3 is methyl;
W* is COOH;
X2, X4 and X6 are each independently hydrogen; and
X3 and X5 are each independently fluorine.

24. The 3-phenylisoxazoline derivative as claimed in claim 1, which is compound 1.1.519, in which
R1 and R2 are each hydrogen,
R3 is methyl;
W* is COOH;
X2, X4 and X6 are each independently hydrogen; and
X3 and X5 are each independently chlorine.

25. The 3-phenylisoxazoline derivative as claimed in claim 1, which is compound 1.1.580, in which
R1 and R2 are each hydrogen,
R3 is methyl;
W* is COOH;
X2, X4 and X6 are each independently hydrogen;
X3 is trifluoromethyl; and
X5 is bromine.

26. The 3-phenylisoxazoline derivative as claimed in claim 1, which is compound 1.3.4, in which
R1 and R2 are each hydrogen,
R3 is 1-chlorovinyl;
W* is COOH;
X4, X5 and X6 are each independently hydrogen; and
X3 is fluorine.

27. The 3-phenylisoxazoline derivative as claimed in claim 1, which is compound 1.3.470, in which
R1 and R2 are each hydrogen,
R3 is vinyl;
W* is COOH;
X2, X4 and X6 are each independently hydrogen; and
X3 and X5 are each independently fluorine.

28. The 3-phenylisoxazoline derivative as claimed in claim 1, which is compound 2.1.33, in which
R1 and R2 are each hydrogen,
R3 is methyl;
W* is COOP;
X2, X4, X5 and X6 are each independently hydrogen;
X3 is acetyl; and
Y is ethyl.

29. The 3-phenylisoxazoline derivative as claimed in claim 1, which is compound 2.2.472, in which
R1 and R2 are each hydrogen,
R3 is difluoromethyl;
W* is COOP;
X2, X4 and X6 are each independently hydrogen;
X3 and X5 are each independently fluorine; and
Y is ethyl.

30. The 3-phenylisoxazoline derivative as claimed in claim 1, which is compound 2.2.527, in which
R1 and R2 are each hydrogen,
R3 is chloromethyl;
W* is COOP;
X2, X4 and X6 are each independently hydrogen;
X3 and X5 are each independently chlorine; and
Y is ethyl.

31. The 3-phenylisoxazoline derivative as claimed in claim 1, which is compound 2.3.475, in which
R1 and R2 are each hydrogen,
R3 is vinyl;
W* is COOP;
X2, X4 and X6 are each independently hydrogen;
X3 is chlorine;
X5 is fluorine; and
Y is methyl.

32. The 3-phenylisoxazoline derivative as claimed in claim 1, which is compound 2.6.546, in which
R1 and R2 are each hydrogen,
R3 is methyl;
W* is COOP;
X2, X4 and X6 are each independently hydrogen;
X3 and X5 are each independently chlorine; and
Y is (ethyl propanoate)-3-yl.