Contributed papers
November 21 (Tue)
16:40-18:40		
Poster Session A (Rooms C, D and E)
				
PA(C)-01 — PA(C)-84 (Room C)				PA(D)-01 — PA(D)-46 (Room D)				PA(E)-01 — PA(E)-57 (Room E)

Room C
PA(C)-01 Jukiya Sakamoto, Mariko Kitajimas, Hayato Ishikawa
	Divergent Total Synthesis of Monoterpenoid Indole Alkaloids via Strictosidine
Aglycones
PA(C)-02 Yuji Otsuka, Toshihiro Yamamoto	Synthesis of 4-Nitroarene Protected Thioglycosides and Their Reactivity on
Chemical Glycosylation
PA(C)-03 Yuki Kurihara, Minori Yagi, Takashi Noguchi, Haruka Yasufuku, Ayane Okita,
Keisuke Fukaya, Daisuke Urabe, Noritaka Chida, Toshitaka Okamura,
Takaaki Sato
Total Synthesis of Keramaphidin B
PA(C)-04 Ghayah Bahatheg, Rajesh Kuppusamy, Muhammad Yasir, David StC. Black,
Mark Willcox, Naresh Kumar
	”Short Cationic Peptoid Dimers: Novel antibacterial therapy for a Post-Antibiotic Era”
PA(C)-05 Shota Iiyama, Keisuke Fukaya, Yu Yamaguchi, Ami Watanabe,
Hiroaki Yamamoto, Shota Mochizuki, Ryosuke Saio, Takashi Noguchi,
Takeshi Oishi, Takaaki Sato, Noritaka Chida
Total Synthesis of Paclitaxel
PA(C)-06 Takahiro Kawajiri, Akihito Kijima, Nobuaki Fukui, Shuichi Yanagisawa,Kazushi Agura
Process Development of Ensitrelvir, COVID-19 AntiviralPA(C)-07 Toyonobu Usuki
Synthesis and Analysis of Elastin Crosslinker Desmosine and the Cyclic Peptide
PA(C)-08 Zazybin Alexey, Bayazit Sarah, Basharimova Anna, Yessinaminov Temirlan,
Tursynbek Saniya, Zolotareva Darya, Dauletbakov Anuar, Belyankova Yelizaveta
	Synthesis and Biological Evaluation of the New Derivatives of Kazcaine,
Tolperisone and Diphenhydramine
PA(C)-09 Hla Myo, Desy Liana, Anuchit Phanumartwiwath	Neuroprotective Potential of dietary plant Centella asiatica L. as inhibitors of
5-lipoxygenase
PA(C)-10 Kaho Oishi, Hiroto Yanuma, Toyonobu Usuki
Synthesis and Analysis of Elastin Crosslinkers Neodesmosine and Merodesmosine1

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Mina Yamane, Hiroki Umeda, Moe Toyobe, Atsushi Iwai, Genki Kudo,
Harunobu Mitsunuma, Masamitsu Okada, Mitsuharu Ueda, Yukio Ando,
Takatsugu Hirokawa, Shigehiro Kawashima, Youhei Sohma,
Kunitoshi Yamanaka, Motomu Kanai
Development of Amyloid Breakers: Catalytic Photooxygenation of Transthyretin
Amyloids in vivo
Haruki Taguchi, Mayuko Kawaguchi, Tohru Nagamitsu, Masaki Ohtawa
Concise Syntheses of (–)-Habiterpenol and (+)-2,3-Epi-Habiterpenol via MHATInitiated Redox Radical Cyclization of Alkenylsilane
Kenji Kimura, Naoya Oku, Atsumi Hasada, Ryo Katsuta, Arata Yajima,
Tomoo Nukada, Yasuhiro Igarashi, Ken Ishigami
Stereoselective Synthesis of New Ether Lipid and Determination of Its
Stereochemistry.
Hiroaki Tanaka, Seiya Miyagi, Takemasa Sakaguchi, Toyonobu Usuki
Synthesis and Cell-Based Evaluation of Umifenovir Analogues as Anti-SARSCoV-2 Agents
Ryosuke Shigeta, Ibuki Haishima, Takahiro Suzuki, Kazuki Kaneko,
Hiroaki Tanaka, Ayano Tanaka-Yanuma, Toyonobu Usuki
Synthetic Study of Jamaicamides
Saki Nagayasu, Hinata Togo, Shoji Kobayashi
Biomimetic Divergent Syntheses of Sterol Metabolites in Mushrooms
Yasukazu Sugiyama, Daiki Kaneko, Seiya Katahara, Mina Yamane,
Yukinori Komiya, Noritaka Chida, Toshitaka Okamura, Takaaki Sato
Total Syntheses of Eburnan and Aspidosperma Type Indole Alkaloids by Lactam
Strategy
Yoshiyuki Manabe, Hersa Milawati, Julinton Sianturi, Takuya Matsumoto,Kazuya Kabayama, Koichi Fukase
Development of Antibody Recruiting Strategy for Novel Cancer Immunotherapy
Yuko Tsuyuguchi, Satoru Hirabayashi, Noriko Ota, Yue Li, Yusuke Yoshikawa,
Bangzhong Lin, Megumi Fumimoto, Junichi Haruta, Keisuke Nimura,
Mitsuhiro Arisawa
Design and Synthesis of Spliceostatin A derivatives toward Castration resistant
prostate cancer
Ryo Katsuta, Ryo Shimizu, Keita Takeda, Shinnosuke Wakamori,Arata Yajima, Shigefumi Kuwahara, Tomoo Nukada, Ken Ishigami
Divergent Synthesis of Aspinolides B–I and Revision of Cremenolide Structure
Risa Maeda, Keiya Uezono, Hiroaki Matoba, Makoto Yoritate, Go Hirai
Inhibition Machinery of Sialoglycans with 3-Exomethylene Functionality
Shaheen Kasim Mulani, Subarna Jyoti Kalita, Sandeep Ramesharao Tapkir,
Maheshwara Reddy Nadiveedhi, Masahiko Seki, Kazushi Mashima
Synthesis of SGLT2 Inhibitors by Means of Metal-Mediated Coupling Reaction
with Grignard Reagent

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Tsukiho Osawa, Kohki Fujikawa, Keiko ShimamotoImportance of the Pyrophosphate Group and the C6 Position of GlcNAc of the
Glycolipid MPIase Essential for the Membrane Protein Integration in Escherichia coli.
Natsuki Mori, Toyonobu Usuki
Extraction of Essential Oils from Aromatic Plants using Deep Eutectic Solvent
Taishi Miura, Makoto Yoritate, Go Hirai
Photoredox-Catalyzed Protecting-Group-Free C-Glycosylation with Glycosyl Sulfinate
Tomonori Teranishi, Keisuke Nishikawa, Toshiki Niwa, Kengo Morita,
Subaru Hashimoto, Akihiro Hoshino, Yoshiki MorimotoEstablishment of “Ring-Size-Divergent” Synthetic Strategy of Terpeonoids Having
Five-, Six-, and Seven-Membered Ether Rings from Identical Polyepoxides
Keitaro Umeno, Hisaaki Onoue, Keiichi Konoki, Kohei Torikai, Yoko Yasuno,
Masayuki Satake, Tohru Oishi
Convergent Synthesis of the WXYZA’B’C’D’E’F’ Ring Segment of Maitotoxin
Rikako Nakamura, Takeru Yamazaki, Yui Kondo, Miho Tsukada,Yusuke Miyamoto, Nozomi Arakawa, Yuto Sumida, Taketoshi Kiya,
Satoshi Arai, Hirohisa Ohmiya
Radical Caging Strategy
Ryuto Terada, Atsuki Tsuboi, Narihito Ogawa
Total Synthesis of (–)-Pinellic Acid, (12R,13R)-Isomer, and (11R,12S,15S)-THETA
Shunki Mamada, Narihito Ogawa
Synthesis of C1-C13 Intermediate of Lactomycin A
Eigo Fukuda, Ibuki Fujiwara, Kenichiro Hamamoto, Keita Ozawa,
Shoki Maruno, Kaiki Motomura, Atsushi Nakayama, Tetsuro Shinada
Total Synthesis and Structure Determination of Bipenicilisorin
Yudai Itagaki, Shota Nagasawa, Shogo Fujiki, Yusuke Sasano, Eunsang Kwon,
Yoshiharu IwabuchiAerobic Stereoselective Synthesis of Benzoxanthenone Lignans Employing
Chromium-salen / Nitroxyl Radical Cooperative Catalysis
Shunki Mamada, Kosuke Niwa, Yoshiya Seto, Narihito Ogawa
Stereoselective Synthesis of Volicitin
Seiya Endo, Keita Ozawa, Yuki Yamamoto, Eigo Fukuda, Atsushi Nakayama,
Yoko Yasuno, Daijiro Ueda, Tsutomu Sato, Tetsuro Shinada
Synthesis of Drimane-8α,11-diol Using Terpene Cyclase from Bacillus Megaterium
Yoko Yasuno, Yuma Karita, Seiji Marubayashi, Tetsuro Shinada, Tohru Oishi
Synthetic Study of Phomopsin A
Yuto Fumimoto, Yuji Mori, Takeo Sakai
Synthetic Study of Serratinine-Type Lycopodium Alkaloids Using the Cascade
Reaction
Kenji Arimitsu, Ikumi Nakazawa, Hiroki Iwasaki, Yoshimi Hirokawa,
Naoyoshi Maezaki
D-Allulopyranosylation Reaction Using Thioglycoside Prepared Directly from Rare
Sugar D-allulose

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Keita Komine, Yuta Yamazaki, Hayato Fukuda, Jun Ishihara
Synthetic Studies on Lyconesidine A Based on Three-Component Radical Coupling
Ryuki Ota, Keisuke Yoshida, Daiki Furukawa, Yuri Imaizumi, Arisa Hidaka,
Yuri Fukami, Masaya Kako, Shinji Kitagaki
Synthetic Study Toward the Total Synthesis of Proaporphine Alkaloids
Sora Iwamoto, Reki Nakano, Keiji Sasaki, Koya Takei, Shoichiro Kobayashi,Reiji Kawakita, Ayako Tokuyama, Noritaka Chida, Toshitaka Okamura,
Takaaki Sato
Synthetic Study of Calyciphylline B
Soichiro Yasui, Shona Banjo, Yoshiyuki Nagashima, Yuto Okada,Keisuke Nakata, Kao Yoshikawa, Eiko Nakasuji, Noritaka Chida,Toshitaka Okamura, Takaaki Sato
Total Synthesis of Lobatamides
Nguyen Ngoc Thanh Luan, Okada Takuya, Toyooka Naoki
Total Synthesis of Natural Product Contained Phloroglucinol Core
Hiroto Aihara, Daisuke Kounai, Akihiko Kasamatsu, Junya Shiraiwa,
Akinobu Matsuzawa, Shogo Kamo, Kazuyuki Sugita
Enantioselective, Protecting-Group-Free Total Syntheses of Boscartins
Kazuki Hori, Shogo Kamo, Kazuyuki Sugita
Total Syntheses of (−)-Oregonensin A and Related Natural Products
Tomoya Mashiko, Yuta shingai, Shogo Kamo, Kazuyuki Sugita
Enantioselective Total Syntheses of (−)-Cochlearol B and (+)-Ganocin A
Patamawadee Silalai, Anan Athipornchai, Jiraporn Tocharus,
Nittaya Boonmuen, Arthit Chairoungdua, Rungnapha Saeeng
New Triazole-Genipin Analogues and Their Biological Activity
Motohiro Sonoda, Haruta Shinoda, Kotaro Fujino, Yusuke Mimura,
Shizuki Noda, Atsushi Okazawa
Synthesis of Aryloxyacetylthioureas for Inhibition of Orobanche minor Radicle
Elongation and its Evaluation
Ryosuke Ashizaki, Ryo Katsuta, Shinnosuke Wakamori, Tomoo Nukada,
Ken Ishigami
Synthetic Studies of Gomadalactones
Yuta Inagaki, Kouki Hashimoto, Daisuke Kaida, Shinnosuke Wakamori,Ryo Katsuta, Ken Ishigami
Synthesis, Cell Growth Inhibition and Structure-Activity Relationship of CGK733
analogs.
Kiyono Uchida, Yusuke Ogura, Hironori Okamura, Hirosato Takikawa
Synthesis of Orobanchol, Based on Acid-Mediated Cascade Cyclization
Davie Kenneth, Atsushi Shimoyama, Haruki Yamaura, Yusuke Yamanaka,
Koichi Fukase
Chemical Synthesis of Monophosphoryl Lipid As from Alcaligenes and a Conjugateof Lipid A with Tumor-Associated Carbohydrate Tn Antigen

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Atsushi Ueda, Sana Kakazu, Takuma Kato, Akihiro Iyoshi, Yui Makura,
Mitsunobu Doi, Masakazu Tanaka
Ring-Closing Metathesis of Side Chains of Helical Peptide: Effects of α-Position
Stereochemistry and Sequence
Soyoung Park
Development of New Biohybrid Materials by Merging of DNA and Amino Acids
Tomoya Suwa, Atsushi Umehara, Makoto Sasaki
Synthetic Studies on Irijimasides Using Ni-Catalyzed Ketone Coupling
Daisuke Sato, Atsushi Umehara, Makoto Sasaki
Synthetic Studies toward the Total Synthesis of Portimine
Shota Nagasawa, Kan Fujiwara, Ryusei Maeyama, Ryosuke Segawa,
Noriyasu Hirasawa, Takatsugu Hirokawa, Yoshiharu Iwabuchi
Selective Synthesis of 1,3-Substituted Cuneanes and Its Application to Bioisosteresof m-Substituted Benzenes
Momona Eguchi, Hiroaki Matoba, Makoto Yoritate, Go Hirai
Synthetic Studies of Cyclic Peptides Consisting of Sugar Amino Acid
Rintaro Nakahashi, Takahiro Moriyama, Hiroaki Matoba, Makoto Yoritate,
Go Hirai
Synthesis of C-linked Neotrehalose Analogues
Nanako Kawate, Koetsu Minamide, Kodai Sueyoshi, Risa Nozawa,
Takanori Matsumaru, Yukari Fujimoto
Synthetic Study of Phospholipids for Lipid-Dependent Immunological Evaluation
Yuki Takatori, Haruhiko Fuwa
Total Synthesis of (−)-Fasicularin
Huiying Mu, Shuai Shao, Koji Miki, Kouichi OheSelective Tumor Imaging in Living Mice Using Near-Infrared pH-Activatable
Cyanine Dyes
Yaseen A. Almehmadi, Pablo Gabriel, Darren J. Dixon
A General Iridium-Catalyzed Reductive Dienamine Synthesis Allows a Five-Step
Synthesis of Catharanthine via the Elusive Dehydrosecodine
Shunya Kikuchi, Nanako Kawate, Juri Takayama, Takanori Matsumaru,
Yukari Fujimoto
Synthetic Studies of Peptide-Lipid Antigen Complexes for Analysis of Antigen
Presentation
Koichi Deyama, Kohei Kamatani, Keisuke Suzuki, Ken Ohmori
Synthetic Studies on Quartromicins, Spirotetronate Antibiotics
Kumpei Yano, Yoshiyuki Manabe, Koichi Fukase
Synthetic Study of Sialyl N-Glycans
Ju Young Ko, Ji-Yoon Jeon, Jae Hyun Kim
A Practical and Scalable Synthesis of Cynandione A
Tomoki Tsuruta, Yukika Yoshino, Keisuke Nishikawa, Yoshiki Morimoto
Studies on Total Synthesis of the Dolastane-Type Diterpene Possessing Inhibition
Activity against Byssal Threads of the Mussel

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Takuya Okada, Atsushi Kato, Izumi Nakagome, Maki Kise,
Kousuke Yoshimura, Nobutada Tanaka, Robert J. Nash, George W. J. Fleet,
Yota Kobayashi, Hayato Ikeda, Naoki Toyooka
Design and Pharmacological Chaperone Effects of DAB Derivatives Targeting the
Lipophilic Pocket of Lysosomal Acid α-Glucosidase
Soichiro Sato, Kenta Noda, Hiroyuki Hakamata, Eunsang Kwon,
Nagao Kobayashi, Hirofumi Ueda, Hidetoshi Tokuyama
Iron-catalyzed Aerobic Dimerization of Tryptophane-Containing Peptides
Yuusei Tokunaga, Kazuki Doi, Takahiro Ikazaki, Hiroaki Matoba,
Makoto Yoritate, Go Hirai
Synthesis of Maltose Analogue with a Novel Type of Inhibition Mechanism
Jiann-Jyh Huang
New Synthesis of Benzofuro[3,2-c]quinolinones as G-quadruplex DNA Stabilizers
Jian Zhang, Keisuke Suzuki, Ken OhmoriTotal Syntheses of Pyrimidinylpropenamide Antibiotics Sparsomycin andSparoxomycins
Hinata Odaira, Naoki Mori, Yujiro Hayashi
Organocatalyst-Mediated Total Synthesis of (−)-Kainic Acid
Yuichiro Uchida, Takuto Oe, Yuki Shimizu, Hirosato Takikawa,
Bubwoong Kang
Convergent and Divergent Synthesis of Isoflavonoid Natural Products throughClaisen Rearrangement-Cyclyzation Cascade
Takayuki Shioda, Hironori Okamura, Yusuke Ogura, Hirosato Takikawa
Synthetic Studies on Artemisidiyne A
Yoshiaki Manse, Fenglin Luo, Kazuhiro Kato, Akane Okazaki,
Eriko Okada, Mitsuhiro Yanagida, Sho Nakamura, Toshio Morikawa
Effect of Enmein from Isodonis Herba on Proliferation-promoting Activity in
Human Hair Follicle Dermal Papilla Cells: Structural Requirements and Mode of Action
Kenji Nemoto, Kento Miura, Hirosato Takikawa, Yusuke Ogura
Syntheses of (+)-Costic Acid and Structurally Related Eudesmane Sesquiterpenoids
and Their Biological Evaluations as Acaricidal Agents Against Varroa destructor
Yusuke Nakagawa, Kishin Inui, Wakana Katayama, Ayaka Shimane,Ryota Kitakamid, Takuya Okada, Yuko Nabeshima, Takeshi Yokoyama,
Mineyuki Mizuguchi, Naoki Toyooka
Creation of Chlorinated Naringenin Derivatives as Potential Inhibitors ofTransthyretin Amyloidogenesis
Tadachika Miyasaka, Masaatsu Adachi, Yuta Kudo, Keita Sugimoto,
Mari Yotsu-Yamashita, Toshio Nishikawa
Synthetic Studies on the Proposed Biosynthetic Intermediates of Tetrodotoxin
S. Luo, J. Wang
Enantioselective Construction and Bioactivities Evaluation of Flavonoid Derivatives

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Yuki Nakatani, Risa Kimura, Hitoshi Takatsu, Naoyuki Kotoku
Total Synthesis of 3-(Phenethylamino)demethyl(oxy)aaptamine
Atsushi Yoshimura, Kyoya Ohyama, Taisei Masuda, Haruhiko Fuwa
Total Synthesis of (−)-Enigmazole A by the Macrocyclization/Transannular Pyran
Cyclization Strategy
Syarifatul Mufidah, Ahmed Salahelden Aboelhamd Atito, Yusaku Miyamae
A Screening for Identification of a Fragment Compound to Synthesize a New
Covalent PPARγ Agonists
Bubwoong Kang, Akari Yamada, Yuika Jotatsu
Four-Step Total Syntheses of Amorfrutins A and B by Final-Stage Meroterpenic
Phenol Carboxylation Strategy

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Ryota Ozawa, Kouhei Inoue, Tetsuya Ishikawa, Tetsuya Yamamoto
Synthesis of Isoindolinones using Optically Active Amines as Chiral AuxiliaryGroupsYoshihiro Nishimoto, Ryota Takahashi, Takuma Miyamura,Yasuko Osakada, Mamoru Fujitsuka, Manabu Abe, Makoto Yasuda
Visible-Light-Mediated Hydrodechlorination and Borodechlorination of Aryl
Chlorides Catalyzed by Aluminum Complex
Taichi Yumura, Takeshi Nanjo, Yoshiji Takemoto
Radical Cyclization of α,β-Unsaturated Carboxylic Acids Catalyzed by
Benzophenothiazine/Boronic Acid Hybrid Photocatalyst
Kenji Muroi, Shohei Furuya, Shin-ichi Fukuzawa
Copper-catalyzed endo’-Selective Asymmetric [3+2] Cycloaddition of
Iminolactone with Alkylidene Pyrazolone
Maho Uchida, Akira Fujimoto, Naoko Nippashi, Tetsuya Yamamoto
Synthesis of Multi-substituted α-Naphthols via Diels-Alder Reaction with Furans
and Aryne
Yuta Sato, Momoko Nagafuchi, Makoto Sako, Kenichi Murai, Mitsuhiro Arisawa
Long-Range Isomerization / Cycloisomerization / Hydroboration of 1,n-Dienes toGive 2,3-Disubstituted Dihydrobenzofurans Using a Multitasking Single Rhodium
Catalyst
Tomoya Nishio, Kyohei Kanomata, Shuji Akai
Racemization of Chiral Sulfoxides Using Immobilized Oxovanadium Catalysts
Amit K Jaiswal, Dennis Chung-Yang Huang
Selective Mono-Hydrodefluorination of Trifluoromethyl Arenes with NHC-Boranes
via Organophotoredox Catalysis
Jihoon Moon, Takusho Kin, Karin Mizuno, Shuji Akai, Kyohei Kanomata
Lipase/H2SO4 Co-Catalyzed Dynamic Kinetic Resolution of Alcohols in Pickering
Emulsions
Kenichi Michigami, Yoshiki Otawa, Yosuke Kanda, Mitsuhiro Ueda,
Masato Ohashi
Pd-Catalyzed Atom-Economical Synthesis of 1,3-Diketone and Its Derivatives
through Cacyl–O Bond Cleavage of O-Acyl Enolates
Ryota Yabe, Takahiro NishimuraIr-Catalyzed Asymmetric [3+2] Annulation of ortho-Keto Arylboron Reagents with
1,3-Dienes
Midori Kawasaki, Kenji Yatsuzuka, Ryuichi Shirai
Hydrolytic Dynamic Kinetic Resolution of Racemic 3-Phenyl-2-oxetanone by
Chiral Phase-Transfer Catalyst
Yusuke Miyazaki, Kenichi Michigami, Mitsuhiro Ueda, Masato Ohashi
Synthesis of Highly-Active Allenylnickel Complexes in Ni-Catalyzed Propargylic
Substitution Reactions

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Hirotaka Okamoto, Yoshihiro Nishimoto, Makoto Yasuda
Synthesis of Al Complexes with Phosphino Group-Substituted Carbon Ligand andTheir Application to Organic Synthesis
Tatsuhiro Uchikura, Fua Akutsu, Haruna Tani, Takahiko Akiyama
Lithium Assisted Fluoride-Coupled Electron Transfer Driven Photoreduction of
Trifluoromethyl Group via EDA complex
Honoka Kasahara, Yuna Nishiguchi, Katsuhiko Moriyama
Enantioselective Oxidative Aryl Rearrangement Reaction of α-Styryl Esters Using
Lewis Acid–Hypervalent Iodine (III)
Hiroko Wasaki, Katsuhiko Moriyama
Remote Csp2–Csp3 Dual Functionalization of 2-Methylindoles with Iodine Reagents
Yuna Yamaguchi, Takumi Yagihashi, Tetsuya Yamamoto
Palladium Catalyzed Synthesis of α-Aryl-α-difluoromethylalcohols using
Arylboronates and Difluoroacetaldehyde Bis(triethylsilyl)acetals
Shunsuke Kataoka, Hiroyuki Morimoto, Takashi Ohshima
Mild and Practical Direct Catalytic Synthesis of Primary Allylic Amines from
Allylic Alcohols Using Ammonium Acetate as the Amine Source
Ryunosuke Akazawa, Mohamed A.B. Ahmed, Masaki Togami, Kohei Miyagaki,
Kenzo Yahata, Kyohei Kanomata, Shuji Akai
Reagent Control for Divergent Rearrangement of 4,4-Disubstituted
2-Hydroxycyclohexa-2,5-dienones
Moena Hirao, Futa Koyama, Toyonobu Usuki, Yumiko Suzuki
NHC-catalyzed Benzoylation of Chromones and Its Application to Synthesis of
Wrightiadione
Miyu Mae, Riku Ogasahara, Keisuke Matsuura, Hyoga Shimizu, Shuji Akai,
Yoshinari Sawama
Photocatalytic and α-Position-Selective H/D Exchange Reactions of
Sulfur-Containing Organic Compounds
Hibiki Okabe, Masamichi Ogasawara
Design, Synthesis, and Application of Planar-Chiral Skewed DPPF Derivatives
Kakeru Masaoka, Haruka Taue, Tatsuya Higaki, Yasuhiro Ohki,
Masamichi Ogasawara
Competitive Double Friedel-Crafts 2,5- and 1',2-Diacylation of Monophosphaferrocenes
Yuuki Mori, Tsukasa Hitomi, Masamichi Ogasawara
Palladium-Catalyzed Synthesis of Alkoxyallenes and Their Application in
Regioselective Hydroelementation Reactions
Yasuhiro Nishikawa, Daiki Mori, Mayuko Toyoda, Yukiho Amano,
Midori Hosoi, Momoka Ando, Osamu Hara
Chelating Picolinaldehyde Hydrazone Amides as Protecting Groups for Carboxylic
Acids
Daisuke Yamamoto, Kazuishi Makino
Manganese-Catalyzed Oxygenative Transformations Using Molecular Oxygen in Air

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Kota Hashimoto, Daiki Higuchi1, Satoshi Matsubara, Kei Murakami
Copper-Catalyzed Reaction of Aziridine for the Synthesis of Substituted
Imidazolidine and Imidazolidinone
Nobuya Tsuji, Pavel Sidorov, Chendan Zhu, Yuuya Nagata, Timur Gimadiev,
Alexandre Varnek, Benjamin List
Predicting Highly Enantioselective Catalysts Using Tunable Fragment Descriptors
Seiya Kikukawa, Kazuki Kobayashi, Nozomi Kasakura, Takeshi Hata
Facile Preparation of 5-Halo-1,2,3-triazole-fused Benzotricyclic Compounds from1-(ω-azidoalkyl)-2-(2,2-dihalovinyl)arenes and Their Conversion into Polycyclic
Triazoles
Teruki Takahashi, Shintaro Okumura, Kaoru Torii, Yasuhiro Uozumi
Photocatalytic Cross-Pinacol Coupling and Carbonyl 1,4-Addition via Umpoled
Carbinol Anions
Hugo Ohki, Masaaki Komatsuda, Hiroki Jr. Kondo, Junichiro Yamaguchi
Ring-opening Functionalization of Heteroaromatics
Hikaru Nakahara, Ryota Isshiki, Junichiro Yamaguchi
A Functional Group Metathesis between Ketones and Esters via Sequential Claisen/
Retro-Claisen Condensation
Yuki Fujimaki, Nobuharu Iwasawa, Jun Takaya
Borylation of Carbon–Carbon σ-Bonds of Aryl Ketones
Yuto Morita, Tatsuyoshi Ito, Nobuharu Iwasawa, Jun Takaya
Synthesis and Reactivity of Cp Rhenium Hydride Complexes Bearing Multidentate
Silyl Ligands
Kazuya Inagaki, Kei Muto, Junichiro Yamaguchi
Synthesis of Polycyclic Compounds through Pd-catalyzed Generation ofo-Quinodimethane from Bromoarenes
Weiwei Guo, Masahiro Hori, Yoshihiro Ogura, Kazuki Nishimura,Kazuaki Ishihara
Tandem Isomerization/α,β-Site- and Enantioselective Addition Reactions of N-(3Butynoyl)-3,5-dimethylpyrazole Induced by Chiral π–Cu(II) Catalysts
Bubwoong Kang, Tatsuro Imamura, Tetsuya SatohRapid and Safer Wurtz Coupling Reaction by Sodium Dispersion
Masaharu Takatsuki, Hiroshi Aoyama, Kenichi Murai, Mitsuhiro Arisawa,
Makoto Sako
Synthesis of Spiro-heterocyclic Cyclobutanes: Heteroannulation of Bicyclobutane
Derivatives via Gold-catalyzed Hydration/Intramolecular Cyclization Sequence
Shohei Yoshioka, Tsunayoshi Takehara, Takeyuki Suzuki, Makoto Sako,
Kenichi Murai, Mitsuhiro Arisawa
Reagent-Controlled Regioselective Intramolecular [2+2] Cycloaddition between
Vinylsilanes and Allenes
Kohei Yamada, Narumi Umekawa, Kokono Tanaka, Kotaro Kikushima,
Yasuyuki Kita, Toshifumi DohiIntroduction of Difluromethyl Group into (Herero)arenes via Decarboxylative
Arylation Using Iodonium(III) Salt
10

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PA(D)-43

PA(D)-44

PA(D)-45
PA(D)-46

Bubwoong Kang, Yuta Nakamura, Rei Nishioka, Vy M. Dong
Catalyst-Free Regioselective Sugar Alkylation by Alkaline-Metal ChelationAssistance
Kotaro Kikushima, Narumi Umekawa, Keina Komiyama, Yasuyuki Kita,
Toshifumi Dohi
Silver-Catalyzed Direct O-Arylation of α-Fluorinated Carboxylic Acid withDiaryliodonium(III) Salt
Taiichi Takeuchi, Kurumi Orihara, Yujiro Sato, Shizuno Otaki,
Tsukasa Aoyama, Ryosuke Masuda, Kento Ishida, Hiroyuki Kusama
Visible Light Induced In-situ Generation of Copper-Siloxycarbene Complex and Its
Application to Catalytic Transformations
Takaya Fujie, Yamato Hirota, Takuya Kochi, Fumitoshi Kakiuchi
Off/on/off Two-Times Switching of Electric Current as a Strategy for One-Pot
Synthesis of Teraryl by Cross-Coupling/ C−H Bromination/ Cross-Coupling
Rin Seki, Hikaru Takaya, Yoshiaki Nakao
Reductive C–O Silylation by Rhodium/Lanthanum Cooperative Catalysis

11

Room E
PA(E)-01

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PA(E)-07

PA(E)-08
PA(E)-09
PA(E)-10

PA(E)-11
PA(E)-12

Katsuhiro Isozaki, Kenta Iseri, Masaharu Nakamura
Dual Catalysis of Gold Nanocluster Functionalized by Peptide Dendron Thiolate
toward Photocatalytic Cross-Dehydrogenative Coupling between Amines andAlkynesTsuyuka Sugiishi, Ryohei Motegi, Hideki Amii
Synthesis of Fluoroalkylated Oxazoles from N-propargylic Amides by
Intramolecular Cyclization
Abhijit Sen, Takuma Sato, Aya Ohno, Heeyoel Baek, Yoichi M. A. Yamada
Convoluted Polymer Supported Cobalt-Catalyzed Regioselective Cyclotrimerizationof Aryl Alkynes
Huihui Zhang, Jesus Rodrigalvarez, Ruben MartinC(sp2)–H Hydroxylation via Catalytic 1,4-Ni Migration with N2O
Nemrud Demirel, Eric Meggers
Chiral-At-Iron Complexes: A Journey Between Reactivity And Stability
Hiroki Nakata, Atsushi Shoji, Izumi Shirakawa, Tatsuo Saito, Ryo Katsuta,
Ken Ishigami, Arata Yajima
Synthesis of Several Bioactive Natural Products Using Asymmetric Allyl Alcohol
Synthesis by AD-Julia-Type Reaction as a Key Reaction
Yuta Chikashige, Tsunayoshi Takehara, Tsuyoshi Matsuzaki, Takeyuki Suzuki,
Kenichi Murai, Mitsuhiro Arisawa, Makoto Sako
Design and Synthesis of Axially Chiral Borinic Acid Catalysts and its Application
to Alkylative Desymmetrization of 1,2-Diols
Daigo Hayashi, Tomohiro Tsuda, Ryo Shintani
Palladium-Catalyzed Skeletal Rearrangement of Substituted 2-Silylaryl Triflates via
1,5-C–Pd/C–Si Bond Exchange
Yusuke Oyamada, Miku Fujii, Shuichi Nakamura
Hydrogen-Bonding-Donor Catalyzed Enantioselective Construction of Unknown
α-Aminonitriles with Tetrasubstituted Stereogenic Carbon Center
Elghareeb E. Elboray, Ahmed G. Taha, Mohammed F. Radwan,
Hemat M. Dardeer, Yusuke Kobayashi, Takumi Furuta, Shohei Hamada,Toshifumi Dohi, Moustafa F. Aly[3+2] Cycloaddition of Azomethine Ylides with Arylidenes and in situ
Diastereodivergent via Retrocycloaddition
Kentaro Yamakawa, Takahiro Nishimura
Iridium-Catalyzed Branch-Selective and Enantioselective Alkylation of
N-Benzimidazolyl Indoles
Kazuhiro Morisaki, Kohei Miyamoto, Emiko Kawaguchi, Yoshihiro Sato
Zn/F carbenoids: Preparation, Stability, Structures, and Application to Nucleophilic
Monofluoroalkylation

12

PA(E)-13

PA(E)-14
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PA(E)-16
PA(E)-17
PA(E)-18
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PA(E)-20
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PA(E)-25
PA(E)-26

Shuhei Ohmura, Kei Katagiri, Haruna Kato, Takahiro Horibe, Sho Miyakawa,
Jun-ya Hasegawa, Kazuaki Ishihara
Highly Enantioselective Radical Cation [2+2] and [4+2] Cycloadditions of
Chalcone Derivatives by Chiral Iron(Ⅲ) Photoredox Catalysis
Mirei Takashima, Makoto Miyoshi, Makoto Sako, Mitsuhiro Arisawa,
Kenichi Murai
Oxidative Rearrangement Approach to Ring Contraction of Piperidines
Tomohiro Ishizaka, Yuji Nakayama, Taichiro Touge, Yamato Yuki,
Kazuhiko Matsumura, Taiga Yurino, Takeshi Ohkuma
Ruthenabicyclic Borohydride Complexes for Asymmetric Hydrogenation of
Ketones and Asymmetric Formal Hydroamination of Allylic Alcohols under BaseFree Conditions
Tsukasa Tawatari, Riku Kudo, Takaya Sakaue, Kiyosei Takasu,
Hiroshi Takikawa
Intramolecular (3+2) Cycloadditions of Benzyne with Nitrogen-substituted Alkynes
Aniket Mishra, Xuefeng Cong, Masayoshi Nishiura, Zhaomin HouEnantioselective Synthesis of 1-Aminoindanes via [3 + 2] Annulation of Aldimines
with Alkenes by Scandium-Catalyzed C−H Activation
Hiroto Shigematsu, Matsutani Takanari, Toshiyuki Moriuchi
Synthesis of Ureas through Carbon Dioxide Activation under Atmospheric Pressure
Using Phosphorus Organic Catalyst
Takuya Kobayakawa, Chika Azuma, Kenichi Yamamoto, Kohei Tsuji,
Hirokazu Tamamura
Development of Synthetic Strategies for Peptidomimetic Based on a Chloroalkene
Dipeptide Isostere and its Application to a Cyclic Peptide
Hasil Aman, Yu-Hao Liu, Jia-Luo Li, Jen-Chieh Hsieh, Gary Jing Chuang
Denitrogenative Cyclization of Benzothiatriazines to Seven-Membered Sultams.
Sei Murayama, Zhurong Li, Huatai Liang, Yan Liu, Hiroshi Naka,
Keiji Maruoka
Impact of Catalyst Deuteration on The Stability and Reactivity of Organocatalyst
Shousuke Miki, Tairin Kawasaki, Masahiro Murakami, Naoki Ishida
Photoinduced Dehydrogenative Coupling of Thiols with Aldehydes Forming
Thioesters
Yamato Ezo, Takashi Niwa, Takamitsu Hosoya
Photoinduced ipso-Azidation of 1-Aryltriazenes
Yuki Hirata, Daichi Sekine, Yoshimi Kato, Lin Luqing, Masahiro Kojima,
Tatsuhiko Yoshino, Shigeki Matsunaga
Enantioselective Synthesis of Thiadiazine-1-oxides Catalyzed by Cp*Co(III)/Chiral
Carboxylic Acid via Asymmetric C–H Amidation
Yixiao Zhang, Zhongxing Huang
Zinc-Catalyzed Desymmetric Hydrosilylation of Monosubstituted Malonic Esters
Masaki Hosaka, Shota Nagasawa, Yoshiharu Iwabuchi
C-H Alkylation of Cubane via Catalytic Generation of Cubyl Radical

13

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PA(E)-29
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PA(E)-31
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PA(E)-35
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PA(E)-38
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Tasuku Ito, Falk William Seidel, Jin Xiongjie, Kyoko Nozaki
TEMPO as a Hydrogen Atom Transfer Catalyst for Aerobic Dehydrogenation of
Activated Alkanes to Alkenes
Natsuho Harada, Toshifumi Asano, Masaharu Sugiura, Shunsuke Kotani,
Makoto Nakajima
Development of Asymmetric Michael Reaction of Acrylamides and Its Mechanistic
Study
Mizuki Kuwajima, Yasushi Shimoda, Sachie Arae, Shunsuke Kotani,
Makoto Nakajima
Chiral Tropone-catalyzed Asymmetric Ring-opening Reaction of Epoxide
Xiaodong Gu, Kexin Liu, Limin Yang, Chengyi Xie, Mingliang Li,
Jun (Joelle) Wang
Nickel-Catalyzed Enantioselective α-Heteroarylation of Ketones via C–F Bond
Activation to Construct All-Carbon Quaternary Stereocenters
Naoki Sugihara, Masayuki Abe, Yoshihiro Nishimoto, Makoto Yasuda
Defluoroarylation of Trifluoromethylarenes with Heteroarenes by Photoredox
Catalysis
Shunsuke Sueki, Azumi Watanabe, Minori Nakamura, Naoyuki Machida,
Asuka Shuto, Kosho Makino, Masahiro Anada
Synthesis of Phosphine Chalcogenides Using Thiocyanate or Selenocyanate Salts
Takahiro Doba, Yu Harabuchi, Yuuya Nagata, Satoshi Maeda
Prediction of Reaction Yields Enabled by Global Reaction Route Mapping andMachine Learning
Kaushalendra Patel, Veeranjaneyulu Lanke, Xu Chen, Ilan MarekStereospecific Nucleophilic Substitution at Quaternary Carbon Stereocenters
Yuki Izumiya, Tetsuya Yamamoto
Palladium-Catalyzed Synthesis of 2,3-Diaryl-1,1-difluoropropenes via
Defluoroarylation of α-(Trifluoromethyl)styrenes with Arylboronic Acids
Takuma Sugimura, Hiroki Shigehisao
MHAT/RPC Promoted [n + 2] Annulation: Access to Cyclic AcetalMichiko Sasaki, Kei Takeda
Abnormal Michael Reaction: Conditions-Dependent Product Distributions in the
Michael Reaction of Monoalkylmalonates
Hayato Nakagawa, Akane Yamaji, Ryohei Hanzawa, Atsushi Yoshimura,
Haruhiko Fuwa
Stereodivergent Tandem Synthesis of Pyrrolidine Derivatives from Amino Alkynes
Kota Sato, Kotaro Yamashita, Yutaka Tanji, Jun-ya Hasegawa, Tetsuaki Fujihara
Synthesis of Dirhodium Complexes Bearing Bulky Carboxylate Ligands and Their
Use in Catalytic Carbene Insertion Reactions
Yiliang Zhang, Yanxin Jiang, Mingliang Li, Jun (Joelle) Wang
Palladium-Catalyzed Diastereo- and Enantioselective DesymmetricHydrophosphination of Cyclopropenes

14

PA(E)-41
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PA(E)-45
PA(E)-46
PA(E)-47
PA(E)-48
PA(E)-49

PA(E)-50
PA(E)-51
PA(E)-52
PA(E)-53
PA(E)-54
PA(E)-55

Ryosuke Isogai, Kosuke Yasui, Aiko Fukazawa
Regioselective Transformation of Weiss Diketone by Introducing Phenylsulfanyl
Groups
Che-Ming Hsu, Hsuan-Hung Liao
Azetidines with All-Carbon Quaternary Centers: Merging Relay Catalysis with
Strain Release Functionalization
Butsaratip Suwattananuruk, Yuta Uetake, Hidehiro Sakurai
Dehydrogenative Coupling of Hydrosilanes Using Gold Nanoparticles Deposited on
Fibrillated Citric Acid-modified Cellulose
Junki Nitta, Takako Yamazaki, Ren Tomita, Katsuhiro Akiyama, Tsubasa Hirata,
Manabu Hatano
Chemoselective Triflation of Phenols Using N-Trifluoromethanesulfonylimidazole
Bo-Wei Huang, Jeng-Liang Han
A Regioselectivity Switch between Enantioselective 1,2- and 1,4-Addition of Allyl
Aryl Ketones with 2,3-Dioxopyrrolidines
Jiangtao Cheng, Jun (Joelle) Wang
Palladium-Catalyzed Asymmetric Hydrophosphination of gem-Difluoroallenes
Shogo Nakamura, Koji Hirano
Copper-Catalyzed Electrophilic Etherification with Acetal-Based Peroxides
Wu Di, Zhongxing Huang
Kinetic Resolution of Malonic Ester Half Amides by Zinc-Catalyzed Reduction
Kazuhiro Aida, Marina Hirao, Aiko Funabashi, Natsuhiko Sugimura,
Eisuke Ota, Junichiro Yamaguchi
Reverse Regioselectivity in Reductive Ring Opening of Epoxides and Oxetanes
Enabled by Zirconocene and Photoredox Catalysis
Duona Fan, Ganesh T. Kamble, Hiroaki Sasai, Shinobu Takizawa
Vanadium(V) Complex-catalyzed Oxidative Hetero-coupling of Arenols and/or
Aryl Amines
Kohei Hatakeyama, Yuya Kogure, Satoshi Ueno
Ruthenium-Catalyzed Cross-Coupling of Pyridylketones as an Alkenyl
Electrophiles with Organoboronates
Dattatraya H. Dethe, Amar D. Uike, Nagabhushana C. B.
Ruthenium-Catalyzed Oxidative Cross-Coupling Reaction of Activated Olefins withVinyl Boronates for the Synthesis of (E,E)-1,3-Dienes
Kenji Yatsuzuka, Midori Kawasaki, Ryuichi Shirai
Tetracoordinated Chiral Lithium Amide Mediated Enantioselective [2,3]-Wittig
Rearrangement of α-Allyloxycarboxylic Acids
Yoichi Dokai, Kodai Saito, Tohru Yamada
Lewis Acid-Catalyzed C-C Bond Formation Based on Decarboxylation of Cyclic
Carbonates
Mohamed S. H. Salem, Masaru Kondo, H. D. P. Wathsala, Akimasa Sugizaki,
Md. Imrul Khalid, Hiroaki Sasai, Takashi Washio, Shinobu Takizawa
Bayesian Optimization (BO)-driven Screening of Multiple Parameters: Towards
Efficient Electrochemical and Flow Synthesis  
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PA(E)-57

Emanuele Silvi, Aitor Bermejo López, Sarko Jabbari, Magnus J Johansson,
Belén Martín-MatuteCyclodehydration and Selective Amination of 1,4-Diols Catalyzed by an NHCiridium(III) Complex
Ting Zhi Yao, Yi Cheng Tseng, Gary Jing Chuang
Research on the Reactivity of Bicyclo[2,2,2]octenoxime16