Plenary, Award, and Intivited Lectures

updated on Aug. 24

Plenary Lectures
Sep 2, 2PL-A-1
9:30

Scott J.

MillerYale University

USA

Sep 2, 2PL-A-2
10:30

StefanMatileUniversity of Geneva

Switzerland

Aida

The University of Tokyo Japan

Sep 3, 3PL-A-1
9:20

TakuzoSep 4, 4PL-A-1
9:20

HiroakiSuga

Sep 4, 4PL-A-2
10:20

HerbertWaldmann Max-Planck-Institut für

Sep 5, 5PL-A-1
11:45

The University of Tokyo Japan

Chair: Hidetoshi Tokuyama (Tohoku University, Japan)
Selective Catalytic Reactions in Complex Heterocyclic Scaffolds

Chiar: Michinori Suginome (Kyoto University, Japan)
Functional Supramolecular Chemistry

Chair: Albert Padwa (Emory University, USA)
Noncovalent Design of Advanced Porous Materials

Chair: Christopher Vanderwal (University of California, Irvine, USA)
Revolutionizing the discovery processes of de novo bioactive peptides
and biologics

Germany

Chair: Satoshi Shuto (Hokkaido University, Japan)
Pseudo Natural Products

China

Chair: Frederick A. Luzzio (University of Louisville, USA)
Total Synthesis of ent -Kauranes and Et-743

Chair: Shun-ichi Hashimoto (Hokkaido University, Japan)
Polyfunctional Heterocyclic Organometallics in Synthesis

Molekulare Physiologie

Dawei

Ma

Chinese Academy of
Sciences

Sep 6, 6PL-A-1
9:30

Paul

KnochelUniversity Munich

Germany

Sep 6, 6PL-A-3
10:30

Masakatsu

Shibasaki

Institute of Microbial
Chemistry (BIKAKEN)

Japan

Boger

The Scripps ResearchInstitute

USA

Chair: Masayuki Inoue (The University of Tokyo, Japan)
Vinblastine: Synthetic and Mechanistic Studies

Sarpong

University of California– USA
Berkeley

Chair: Oliver Reiser (University of Regensburg, Germany)
Strategies and Methods for Synthesis Inspired by Complex Natural
Products

Chair: David R. Williams (Indiana University, USA)
Catalytic Asymmetric Synthesis of Heterocyclic Compounds throughCooperation Asymmetric Catalysis

Award Lectures
Sep 5, 5AL-A-1
9:20

Sep 5, 5AL-A-2
10:25

Sep 5, 5AL-A-3
14:00

Dale L.

Richmond

Guy

Humphrey Merck Sharp and

USA

Dohme

Chair: Walter Huebsch (Bayer AG, Germany)
Innovation: Key Enabler for the Development of Sustainable Commercial
Manufacturing Processes at MSD

Intivited Lectures
Sep 2, 2IL-A-1
11:50

SeijiroMatsubara Kyoto University

Sep 2, 2IL-A-2
12:20

Ying-Yeung

Yeung

Chinese University ofHong Kong

Hong
Kong

Sep 2, 2IL-A-3
14:00

Brigitte

Bibal

University of BordeauxFranceSep 2, 2IL-A-4
14:30

SensukeOgoshi

Osaka University

Japan

Sep 2, 2IL-B-1
11:50

Hideaki

KakeyaKyoto University

Japan

Sep 2, 2IL-B-2
12:20

Junko

OhkandaShinshu University

Japan

Japan

Chair: Toshiaki Murai (Gifu University, Japan)
Preparation of Chiral Molecules for Pharmacophores
Recent Advances in Halocyclizations

Chair: Bo Liu (Sichuan University, China)
9,10-diphenylanthracenes as scaffolds for metal coinage catalysts
Nickel-catalyzed Synthesis of Benzoxasiloles: Ligand-Controlled
Switching from Inter- to Intramolecular Aryl-Transfer Process
Chair: Corinne Fruit (Rouen Normandy University, France)
Frontier Research on Chemical Communications Unveils the Mystery ofLife Science
A Synthetic Molecule-based Approach Toward Controlling of Transient
Protein Interactions

Sep 2, 2IL-B-3
14:00

ChunyanSep 2, 2IL-B-4
14:30

Thomas J. J. Müller

Chi

National University ofSingapore

Chair: Jie Han (Nankai University, China)
Singapore Heterocyclic Acenes and Quinodimethanes

Heinrich-Heine-Universit Germanyät Düsseldorf

Dithieno-anellated [1,4]Thiazines – Redox Activity, Luminescence
Characteristics and Antiaromaticity of Novel Congeners of Phenothiazine

Sep 3, 3IL-A-1
10:40

Norio

Shibata

Nagoya Institute ofTechnology

Japan

Chair: Darren J. Dixon (University of Oxford, UK)
Synthesis of Trifluoromethylated Heterocycles under Palladium Catalysis

Sep 3, 3IL-A-2
11:10

Debabrata

Maiti

IIT Bombay

India

Designing of templates to reach the distal C‒H bondSep 3, 3IL-A-3
11:40

Aaron

Aponick

University of Florida

USA

Chair: Satoshi Minakata (Osaka University, Japan)
Making Chiral Heterocycles Using Chiral Heterocycles as Ligands

Sep 3, 3IL-A-4
12:10

MasatoKitamura

Nagoya University

Japan

Sep 3, 3IL-B-1
10:40

TomokiOgoshi

Kyoto University

Japan

Chair: Takashi Kubo (Osaka University, Japan)
Pillar-Shaped Macrocyclic Compounds “Pillar[n]arenes”:
from Simple Molecular Receptors to Bulk Supramolecular Assemblies

Sep 3, 3IL-B-2
11:10

Ma Angeles

Herranz

Complutense University Spainof Madrid

p-Extended Tetrathiafulvalenes (exTTFs): Versatile Heterocyclic Partnersof Carbon Nanostructures in Donor-Acceptor Systems

Sep 3, 3IL-B-3
11:40

Andrei K.

Yudin

University of Toronto

CanadaChair: Yoshito Tobe (National Chiao Tung University, Taiwan)
Dominant Rotors as a Tool to Control Macrocycles

Sep 3, 3IL-B-4
12:10

Toshikazu

TakataTokyo Institute ofTechnologyJapan

Sep 3, 3IL-C-1
10:40

Masayuki

Wasa

Boston CollegeUSA

Sep 3, 3IL-C-2
11:10

Sayuri

HiranoSPERA PHARMA, Inc.

Japan

Asymmetric route to chiral heterocyclic compounds toward efficientmanufacturing process

Sep 3, 3IL-C-3
11:40

Bo

Liu

Sichuan University

China

Total Synthesis of Natural Dimeric Terpenoids: Inspired but Not Limited
by Biohypothesis

CpRu-catalyzed Enantioselective Dehydrative Cyclization of Protic
Nucleophile tethered Allylic Alcohols

Synthesis of Rotaxane Catalysts for Asymmetric and Processive
Reactions
Chair: Michael S. Sherburn (Australian National University, Australia)
Enantioselective Cooperative Catalysis with Frustrated Acid/BaseComplexes

Sep 4, 4IL-A-1
11:40

Koichi

FukaseOsaka University

Japan

Chair: Jeffrey Aubé (University of North Carolina at Chapel Hill, USA)
Synthesis and biofunctional studies of immunomodulating
glycoconjugatesSep 4, 4IL-A-2
12:10

Dan

Yang

The University of Hong
Kong

Hong
Kong

Novel Fluorescent Probes for Selective Detection and Imaging of Superoxide,
Hydrogen Peroxide, Hypochlorous Acid, Hydroxyl Radical, and Peroxynitrite

Chair: Aaron Aponick (University of Florida, USA)
Step Economic Total Synthesis of Heterocyclic Natural Products

Sep 4, 4IL-B-1
11:40

Michael S.

Sherburn

Australian National
University

Australia

Sep 4, 4IL-B-2
12:10

Sanghee

Kim

Seoul National
University

Korea

Asymmetric Total Synthesis of Heterocyclic Alkaloids with Chirality
EconomySep 4, 4IL-C-1
11:40

Yoshiharu

IwabuchiTohoku University

Japan

Chair: Alan Aitken (University St Andrews, Scotland)
Exploration and Exploitation of AZADO for Highly Selective Catalytic
Oxidative Transformations

Sep 4, 4IL-C-2
12:10

Rong-Jie

Chein

Academia Sinica

TaiwanChiral Tetrahydrothiophene Ligands in Asymmetric Catalysis

Sep 5, 5IL-A-1
14:35

MakotoMichidaDaiichi Sankyo Co., Ltd. Japan

Chair: Walter Huebsch (Bayer AG, Germany)
Development of an Efficient Synthetic Method for a Key Intermediate of
Edoxaban
Chair: Takeo Kawabata (Kyoto University, Japan)
Aerobic Oxygen-Driven Functionalizations of ProteinsSep 5, 5IL-B-1
14:00

MotomuKanai

The University of Tokyo Japan

Sep 5, 5IL-B-2
14:30

TobiasRitterMax-Planck-Institut fürKohlenforschung

GermanyLate-Stage Functionalizations

University of Oxford

UK

Chair: Sanghee Kim (Seoul National University, Korea)
Catalytic Approaches for Simplifying Complex Molecule Synthesis

Japan

Asymmetric Total Syntheses of Gelsemium Alkaloids

Sep 5, 5IL-C-1
14:00

Darren J.

Dixon

Sep 5, 5IL-C-2
14:30

Hiromitsu

Takayama Chiba University

Oral Presentations

updated on Aug. 26
Chair: Adrian Dobbs (University of Greenwich, UK)
Total Synthesis of (–)–Dehydrobatzalladine C via Construction of Pyrrolopyrimidine
Skeleton by Gold-Catalyzed Tandem Cyclization

Sep. 2nd

2O-A-1

Hidetoshi

Tokuyama

Tohoku University

Sep. 2nd

2O-A-2

YoshioAndoTokyo Institute of Technology Japan

Stereochemical Dichotomy in Two Competing Cascade Reactions: Enantio-divergent Total
Synthesis of Spiroxin A

Sep. 2nd

2O-A-3

Mingji

Dai

Purdue University

USA

Total Synthesis for Better and New Function: From Enabling Synthetic Methodology andStrategy to Novel Disease Target

Sep. 2nd

2O-A-4

Fumihiko

Yoshimura

University of Shizuoka

Japan

Chair: Yoshio Ando (Tokyo Institute of Technology, Japan)
Total Synthesis of (+)-Laurallene

Sep. 2nd

2O-A-5Adrian

Dobbs

University of Greenwich

UK

Heterocycles and Neglected Diseases: Still a role for total synthesis

Sep. 2nd

2O-B-1YouheiTakedaOsaka University

Japan

Chair: Sachie Arae (Kumamoto University, Japan)
Dibenzo[a,j]phenazine-Cored Twisted Donor-Acceptor-Donor Triads: Promising Platform
for Multi-Photofunctional Organic Materials

Sep. 2nd

2O-B-2

Katsuhiko

Tomooka

Kyushu University

Japan

Chemistry of Planar Chiral Heterocycles

Sep. 2nd

2O-B-3

DanielWerz

TU Braunschweig

Germany

Chair: Youhei Takeda (Osaka University, Japan)
BOIMPYs and Oligomerized BODIPYs: A Key to Superfluorophors

Sep. 2nd

2O-B-4

SachieArae

Kumamoto University

Japan

Regio- and Stereoselective Intramolecular Cyclization Reactions of Benzoheteroles andAlkynes through the Formation of Vinylidene ortho-Quinone Methide Intermediates

Sep. 2nd

2O-B-5

Jie

Han

Nankai University

China

Photoluminescent 1,3,4-Thiadiazole-based Liquid Crystals with Wide Mesomorphic
Temperature Ranges and Excellent Thermal Stability

Sep. 2nd

2O-C-1

Atsuhiko

Taniguchi

Tokyo University of Pharmacy Japanand Life Sciences

Sep. 2nd

2O-C-2Shin

Aoki

Tokyo University of ScienceJapan

Selective Substitution and Decomposition Reactions of Cyclometalated Iridium Complexes
and Their Applications to Biomedical and Material Sciences

Sep. 2nd

2O-C-3

Luhan

Zhai

The University of TokyoJapan

Application of 7-azabicyclo[2.2.1]heptane derivatives to stabilize β-strand-like extended
conformation of neighboring α-amino acids

Sep. 2nd

2O-C-4

LennartBrewitz

University of Oxford

UK

Chair: Atsuhiko Taniguchi (Tokyo University of Pharmacy and Life Sciences, Japan)
Synthesis of 3- and 5-Substituted 2,4-Pyridinedicarboxylates which are Novel Potent andSelective Inhibitors of the Human Enzyme ‘Aspartate/Asparagine-β-Hydroxylase’

Sep. 2nd

2O-C-5

R. T.

Pardasani

Central University ofRajasthan

India

Transition-metal mediated synthesis of complex N-heterocycles

Sep. 2nd

2O-D-1

NorbertKrauseDortmund University ofTechnology

Germany

Chair: Yusuke Kobayashi (Kyoto University, Japan)
Gold-catalyzed Synthesis of [N,N]-, [N,O]-, and [N,S]-Spiroacetals

Sep. 2nd

2O-D-2

Li

Liu

Institute of Chemistry, Chinese China
Academy of Sciences

Asymmetric transformations of Morita-Baylis-Hillman adducts for construction of chiralaromatic heterocycles

Sep. 2nd

2O-D-3

Nagatoshi

Nishiwaki

Kochi University of Technology Japan

Direct Synthesis of Nitroaziridines and the Subsequent Lewis Acid Mediated Isomerization
to Nitroenamines

Sep. 2nd

2O-D-4

Yoshihiro

Sohtome

RIKEN

Japan

Sep. 2nd

2O-D-5

YusukeKobayashi

Kyoto University

Japan

Sep. 3rd

3O-A-1

Boris

Nachtsheim

University of Bremen

Germany

Sep. 3rd

3O-A-2

ShinobuTakizawa

ISIR, Osaka University

Japan

Enantioselective Synthesis of Highly Functionalized Heterocycles via Organocatalyzed
Domino Reactions

Sep. 3rd

3O-A-3Yu

Zhao

National University ofSingapore

Singapore

Medium-Sized Heterocycles: Stereoselective Synthesis and Functionalization

Sep. 3rd

3O-A-4

Fumitoshi

Kakiuchi

Keio University

Japan

Chair: Boris Nachtsheim (University of Bremen, Germany)
Rhodium-catalyzed Deallylative Alkenylation via C-C Bond Cleavage

Sep. 3rd

3O-A-5

Toshimichi

OhmuraKyoto University

Japan

New Route to Indoles through Iridium-Catalyzed C(sp3)–H Activation

Sep. 3rd

3O-A-6

Chikara

Dohno

Osaka University

Japan

Chair: Yu Zhao (National University of Singapore, Singapore)
Modulation of ribozyme activity by conformational changes induced by a synthetic RNA
binding molecule

Sep. 3rd

3O-A-7

Kei

Goto

Tokyo Institute of Technology Japan

Sep. 3rd

3O-A-8

CorinneFruit

Rouen Normandy University

Sep. 3rd

3O-A-9Jeffrey

Aubé

University of North Carolina at USA
Chapel Hill

P.

B.

J.

Japan

FranceChair: R. T. Pardasani (Central University of Rajasthan, India)
Inactivation of Myostatin using Photooxygenation Catalyst-Peptide Conjugate

Chair: Norbert Krause (Dortmund University of Technology, Germany)
Catalytic Asymmetric [3+2] Cycloadditions With alpha-Keto Ester Enolates
Direct addition of Amides to Glycals Enabled by Solvation-insusceptible 2-Haloazolium
Salt Catalysis
Chair: Toshimichi Ohmura (Kyoto University, Japan)
N-Heterocycle-Stabilized Hypervalent Iodine Compounds - Highly Modular Oxidation
Catalysts with Unique Reactivities

Model Study on the Formation of Cyclic N-Selenoamide Intermediates in Selenocysteine
Oxidation in Glutathione Peroxidase Catalysis
Chair: Fumitoshi Kakiuchi (Keio University, Japan)
Promising DYRK1A inhibitor synthesized by late-stage C-H Arylation
Synthesis and applications of the MR1 ligand precursor 5-amino-6-Dribitylaminouracil (5A-RU)

Nakayama

Tokushima University

Japan

Chair: Hong Ren (Merck Sharp & Dohme, USA)
Synthetic Studies on Chippiine-type alkaloids

Till

Opatz

Johannes Gutenberg
University

Germany

Xylochemistry and Photochemistry with Heterocycles – Towards a Greener Synthesis

3O-B-3HiroshiTakikawa

Kyoto University

Japan

Synthetic Study on Helisorin, an Antiviral Neolignan Natural ProductSep. 3rd

3O-B-4Jin

Qu

Nankai University

China

Chair: Atsushi Nakayama (Tokushima University, Japan)
Three Two-step Enantioselective Total Syntheses of (–)-Glabrescol Implicate Alternative
Biosynthetic Pathways Starting from Squalene

Sep. 3rd

3O-B-5Hong

Ren

Merck Sharp & Dohme

USA

Development of a Commercial Manufacturing Process for Gefapixant

Sep. 3rd

3O-B-6

AndreasSchmidt

Clausthal University ofTechnology

Germany

Chair: Yuko Otani (The University of Tokyo, Japan)
N-Heterocyclic carbenes derived from sydnones in heterocycle synthesis and catalysis

Sep. 3rd

3O-B-7

Sunna

Jung

Kwansei Gakuin University

Japan

Syntheses of Isoanthracenoheteroles by Cycloaddition of Didehydroisobenzofuran

Sep. 3rd

3O-B-8R. AlanAitkenUniversity of St Andrews

UK

1,4-Thiazine

Sep. 3rd

3O-B-9

Yuko

Otani

The University of Tokyo

Japan

Chain Length-dependent Acceleration of Rotation of Lactams with Nitrogen-pyramidal
Tertiary Amide

Sep. 3rd

3O-C-1

Qiu

Wang

Duke University

USA

Chair: Chao Wang (The University of Tokyo, Japan)
Alkene Amino Difunctionalization as a Rapid Approach to Diverse Heterocycles

Sep. 3rd

3O-C-2

Xinfang

Xu

Soochow University

China

Catalytic Alkyne Functionalization via Metal Carbene Intermediate

Sep. 3rd

3O-C-3

Itaru

Nakamura

Tohoku University

Japan

Au-Catalyzed Skeletal Rearrangement of O-Propargylic Oximes via N-O Bond Cleavage
with the Aid of a Brønsted Base Cocatalyst

Sep. 3rd

3O-C-4

Takayoshi

Arai

Chiba University

Japan

Chair: Qiu Wang (Duke University, USA)
Catalytic Asymmetric Synthesis of Thiochromanes

Sep. 3rd

3O-C-5Chao

Wang

The University of TokyoJapan

Cross-Coupling via Ammonium or Pyridinium C–N Bond Cleavage

Sep. 3rd

3O-C-6

Jia-Rong

Chen

Central China Normal
University

China

Chair: Yoshihiro Nishimoto (Osaka University, Japan)
Visible Light-driven Generation of N-Radicals and Application to N-Heterocycle Synthesis

Sep. 3rd

3O-C-7

Keisuke

Asano

Kyoto University

Japan

Sep. 3rd

3O-C-8

Seiji

Shirakawa

Nagasaki University

Japan

Sep. 3rd

3O-C-9

Yoshihiro

Nishimoto

Osaka University

Japan

Sep. 3rd

3O-D-1

Jiří

Pospíšil

Czech
Republic

Sep. 3rd

3O-D-2

Koji

HiranoThe Czech Academy of
Sciences, Institute ofExperimental Botany

Osaka University

Japan

Synthesis of Benzophospholes with Phosphenium Cations of Unique Reactivity

Sep. 3rd

3O-D-3

Kentaro

Okano

Kobe University

Japan

Termination of Halogen Dance by in situ Transmetalation

Sep. 3rd

3O-D-4

Mario

Waser

University of Linz

Sep. 3rd

3O-D-5

NorbertHoffmann

CNRS, Université de Reims

FrancePhotochemically induced electron and hydrogen transfer in heterocyclic chemistry

Sep. 3rd

3O-D-6

MamoruIto

Waseda University

Japan

Chair: Kanako Nozawa-Kumada (Tohoku University, Japan)
Construction of Nitrogen-Containing Medium-Sized Ring by Gold-Catalyzed
Cycloisomerization

Sep. 3rd

3O-D-7

Yoshihiro

Ueda

Kyoto University

Japan

Sep. 3rd

3O-D-8Simon

BlakeyEmory University

USA

Chair: Mamoru Ito (Waseda University, Japan)
Development and Application of Allylic C-H Amidation Chemistry

Sep. 3rd

3O-D-9KanakoNozawaKumada

Tohoku University

Japan

Copper-Catalyzed Oxidative C(sp3)-H Functionalization for the Synthesis of Heterocycles

Sep. 5th

5O-A-1

Gavin ChitTsui

The Chinese University ofHong Kong

Sep. 5th

5O-A-2

De-Xian

Wang

Institute of Chemistry, Chinese China
Academy of Sciences

Sep. 3rd

3O-B-1

AtsushiSep. 3rd

3O-B-2

Sep. 3rd

Chair: Andreas Schmidt (Clausthal University of Technology, Germany)

B.

Organocatalytic Enantio- and Diastereoselective Construction of syn-1,3-Diol Motifs via
Dynamic Kinetic Resolution of In Situ Generated Chiral Cyanohydrins
Chair: Jia-Rong Chen (Central China Normal University, China)
Design of Chiral Bifunctional Sulfide Catalysts for Asymmetric Bromolactonizations
Synthesis of Highly Coordinated Organoaluminum Complexes Bearing a Lewis Basic
Substituent and Their Application to Catalytic Cycloaddition Reaction
Chair: Norbert Hoffmann (CNRS, Université de Reims, France)
Benzo[d]thiazol-2-yl Sulfonyl Group – A new look for an old synthetic tool

Chair: Jiří Pospíšil (The Czech Academy of Sciences, Institute of Experimental Botany, Czech Republic)
Austria
Syntheses of Chiral Heterocycles Using Ammonium Ylides

β-Silicon Effect in Intermolecular Site-Selective C(sp3)-H Amination Promoted by
Dirhodium Nitrenes

Chair: Makoto Michida (Daiichi Sankyo Co.,Ltd., Japan)
Hong Kong A Three-Pronged Approach to the Synthesis of Trifluoromethylated Heterocycles
Diversity-Oriented Construction of Multicavity-Containing Supermacrocycles

Sep. 5th

5O-B-1

Jen-Chieh

Sep. 5th

5O-B-2

OliverSep. 5th

5O-C-1

Sep. 5th

5O-C-2

Sep. 5th

5O-D-1

Sep. 5th

5O-D-2Chair: Motomu Kanai (The University of Tokyo, Japan)
Synthesis of Heterocyclic Compounds through the Transition-Metal-Catalyzed Coupling
Reactions of Benzoimine

Hsieh

Tamkang University

TaiwanReiserUniversity of Regensburg

Germany

Shigeru

Arai

Chiba University

Japan

TomoyaMiura

Kyoto University

Japan

Naoki

Kanoh

Hoshi University

Japan

Chair: Tobias Ritter (Max Planck Institute for Coal Research, Germany)
Second-Generation Synthesis and Biological Evaluation of Heronamides, Naturally
Occurring Polyene Macrolactams

ToshioNishikawa

Nagoya University

Japan

Synthesis of Aplysiatoxin/Oscillatoxin Family of Marine Natural Products

Regio- and Stereoselective Synthesis of Functionalized Dihydropyridines, Pyridines, and
2H-Pyrans: Heck Coupling of Monocyclopropanated Heterocycles
Chair: Hiromitsu Takayama (Chiba University, Japan)
Synthesis of nitrogen heterocycles under nickel catalysis: reaction development and its
application
Enantioselective Denitrogenative Annulation of 1H-Tetrazoles with Styrenes Catalyzed by
Rhodium

Flash Presentations
Pagire

BIKAKENJapan

Chair: Mingji Dai (Purdue University, USA)
Enantioselective Photocatalysis utilizing 7-Azaindolines as an Auxiliary: Challenges andOpportunities

Kenta

Rakumitsu

Kumamoto University

Japan

Total Syntheses of (–)-Secologanin, (–)-5-Carboxystrictosidine, and (–)-Rubenine

2F-A-3

TakuyaIshii

Kanazawa University

Japan

N-Heterocyclic Carbene-Catalyzed Decarboxylative Alkylation of Aldehydes

Sep. 2nd

2F-A-4

ShinobuArikawa

Osaka University

Japan

The First Synthesis and Characterization of a Polycyclic Zwitterion with Open-Shell
Character

Sep. 2nd

2F-B-1

KeitaroYamamoto

Osaka University

Japan

Sep. 2nd

2F-B-2

UpendraSharmaUniversity of Leuven (KU
Leuven)Belgium

Synthesis of Diversely Functionalized Heterocycles via Trapping of Transient σAlkyl/Vinyl-Palladium (II) Intermediates

Sep. 2nd

2F-B-3

MuhammadSohailJapan

Dynamic Stereoselective Annulation to Afford Spirooxindole Pyran Polycycles

Sep. 2nd

2F-B-4

FlorianOstlerOkinawa Institute of Scienceand Technology Graduate
University
University of Muenster

Germany

Design & Synthesis of Novel Halogen-Bond-Donor Catalysts

Sep. 2nd

2F-C-1

Taka

Sawazaki

The University of Tokyo

Japan

Chair: Shin Aoki (Tokyo University of Science, Japan)
Catalytic photo-oxygenation enables inhibition of tau amyloid formation

Sep. 2nd

2F-C-2Ruofang

Hu

Osaka University

Japan

Chemical synthesis and function of Helicobacter pylori peptidoglycan fragments

Sep. 2nd

2F-C-3

AkitomoKasahara

The University of TokyoJapan

Conformational Analysis and cis-trans Control of Cyclized Tryptophan Tertiary Amides

Sep. 2nd

2F-C-4

KazusaAoki

Sophia University

Japan(Di-(2-picolyl)amino)quinazolines as Fluorescent Probes for ATP

Sep. 2nd

2F-D-1

Philipp

KramerTu Kaiserslautern

Germany

Chair: Li Liu (Institute of Chemistry, Chinese Academy of Sciences, China)
Enamides as versatile tools for the stereoselective construction of heterocycles

Sep. 2nd

2F-D-2

Shibo

Xu

Osaka University

Japan

Synthesis of Six- and Seven-Membered Benzolactones by Nickel-Catalyzed C-H Couplingof Benzamides with Small-Sized Cyclic Ethers

Sep. 2nd

2F-D-3Matthieu

Daniel

CEA - Le Ripault, Orleans
University - ICOAFranceHypervalent Iodine (III) in Direct Intramolecular N-N Bond Formation with HeteroaromaticAmines: Synthesis of Triazapentalene Derivatives

Sep. 2nd

2F-D-4

Amol

Sonawane

Gifu University

Japan

Fe (III) Promoted Intramolecular Cascade Cyclization for the Synthesis of Quinoline fused
Selenophene-based Heteroacene Scaffolds

Sep. 3rd

3F-A-1

ZonidisUniversity of Huddersfield

UK

Sep. 3rd

3F-A-2

Dimitrios
Christodoul
Quan-Qing

Zhao

Central China Normal
University

China

Visible Light-driven Generation of Hydrazone Radicals for the Synthesis of
Dihydropyrazoles and Tetrahydropyridazines

Sep. 3rd

3F-A-3

Tagui

NaganoKyoto University

Japan

Optically Active trans-Cyclooctene-pyridine Ligands in Rhodium-catalyzed Asymmetric
1,4-Addition

Sep. 3rd

3F-A-4

Piotr

DrelichLodz University of Technology Poland

Sep. 3rd

3F-B-1

MartinPetzold

TU Braunschweig

Germany

Sep. 3rd

3F-B-2

Dong-Mei

Yan

Central China Normal
University

China

Dual Copper and Photoredox-Catalyzed Cross-Coupling of Alkenes, OBenzoylhydroxylamines, and Sulfur Ylides

Sep. 3rd

3F-B-3

Christopher R.

Opie

Institute of Microbial
Chemistry, BIKAKEN

Japan

Systematic examination of catalytic amide bond formation by the readily accessible
B3NO2 heterocycle-containing molecule Pym-DATB

Sep. 3rd

3F-B-4

TakuyaMurai

Institute for Chemical
Research, Kyoto University

Japan

Chalcogen-Bond Assisted Dirhodium Complex –Total Syntheses of Naturally Occurring γLactones–

Sep. 3rd

3F-C-1

AnkitaBal

National Institute of Scence
Education and Research

India

Nitrenium Ion from λ3-Iodanes

Sep. 3rd

3F-C-2

KosukeOkada

Tohoku University

Japan

Total Synthesis of (–)-Deoxoapodine

Sep. 3rd

3F-C-3

Takahiro

Asada

Osaka University

Japan

Complexation between Al(C6F5)3 and N-Phoshpnine Oxide-Substituted Imidazolidenes

Sep. 3rd

3F-C-4

KirstyAnderson

University of Auckland

New
Zealand

A new indole to benzoxazole rearrangement enabled by C-H borylation

Sep. 3rd

3F-D-1

KhokanChoudhuri

India

Sep. 3rd

3F-D-2

Yuya

KakiuchiNational Institute of Science
Education and Research(NISER),
Bhubaneswar
Osaka UniversityJapan[2+2+1] Pyrrole Synthesis from Alkynes and Azobenzene via N=N Bond Cleavage
Catalyzed by Vanadium Complexes

Sep. 3rd

3F-D-3MiguelParajaUniversity of Geneva

Spain

Anion-π Catalysis for Epoxide-Opening Ether Cyclizations, from Monomers to Oligomers,
Challenging Baldwin Rules

Sep. 3rd

3F-D-4Masaki

Fujie

Osaka University

Japan

Synthesis of Hypervalent Iodine Reagents Bearing Cationic Heterocycles and Application
to Oxidative Cyclization

Sep. 2nd

2F-A-1

SantoshSep. 2nd

2F-A-2

Sep. 2nd

K.

K.

D.

Chair: Katsuhiko Tomooka (Kyushu University, Japan)
Development of Quinoidal Oligothiophenes Having Fluorine Atoms

Chair: Kei Goto (Tokyo Institute of Technology, Japan)
Synthesis and Photochromism of Bis(Thienyl) Substituted 1,2-Oxathiine 2,2-dioxides

Synthesis of γ,γ‐Disubstituted Butenolides through a Doubly Vinylogous Organocatalytic
Cycloaddition
Chair: Sunna Jung (Kwansei Gakuin University, Japan)(3+3)‐Annulation of Carbonyl Ylides with Donor–Acceptor Cyclopropanes: Synergistic
Dirhodium(II) and Lewis Acid Catalysis

Chair: Keisuke Asano (Kyoto University, Japan)

Chair: Yoshihiro Ueda (Kyoto University, Japan)
Advanced method for the construction of C-S bond via C-H functionalization

Matsumura

Osaka City University

Japan

Chair: Gavin Chit Tsui (The Chinese University of Hong Kong, Hong Kong)
Total Synthesis of Histrionicotoxin 235A

Takahiro

Watanabe

The University of Tokyo

Japan

Synthetic Study of TPI 287

5F-A-3

Lucie

Cechova

IOCB Prague

Czech
Republic

5-Phenylazopyrimidines: A new class of orthogonal photoswitches?

Sep. 5th

5F-A-4

EisakuOhashiTokushima university

Japan

Studies on the Second Generation Synthesis of Palau’amine

Sep. 5th

5F-B-1Yuan

Jin

Nagoya University

Japan

Synthetic Studies on Haliclonin A

Sep. 5th

5F-B-2

Shinsuke

Shimizu

The University of TokyoJapan

Total Syntheses of Bufadienolides

Sep. 5th

5F-B-3Jun

ShimuraTokyo Institute of Technology Japan

Total Synthesis of Saptomycin H

Sep. 5th

5F-B-4

Naoki

Matsuyama

Osaka University

Facile Synthesis of Chiral Spirooxindoles via Pictet-Spengler/Oxidative Rearrangement

Sep. 5th

5F-C-1

DanielPayne

National Institute for Materials Japan
Science (NIMS)

Sep. 5th

5F-C-2

Ryuichi

MurataKyoto University

Japan

Desymmetrization of gem-Diols via Enantio- and Diastereoselective Cycloetherification
Using Bifunctional Organocatalysts

Sep. 5th

5F-C-3

Keigo

Higashida

Osaka University

Japan

Chiral Vanadium Complex-catalyzed Enantioselective Oxidative Hetero-coupling
Reactions of Arenols

Sep. 5th

5F-C-4

Gabriella

Stockholm University

SwedenRegiospecific N-Arylation of Aliphatic Amines under Mild and Metal-Free Reaction
Conditions

Sep. 5th

5F-D-1

Ryo

TanifujiTokyo University of Agriculture Japanand Technology

Chair: Naoki Kanoh (Hoshi University, Japan)
Chemo–enzymatic total synthesis of tetrahydroisoquinoline alkaloids exhibiting potent DNA
alkylating ability

Sep. 5th

5F-D-2

FabianHogenkamp

Heinrich Heine University

Germany

Heterocyclic Photocages for Carbohydrates

Sep. 5th

5F-D-3

Bimolendu

Das

Osaka University

Japan

ANP77: A Three-carbon Atom Linked 2-Amino-1,8-naphthyridine Dimer that Recognizes
Cytosine Rich Bulge-mismatched Sequences of Duplex DNA and RNA

Sep. 5th

5F-D-4

JeremyConradDobrowolski The University of New South

Australia

Biologically Active Novel Nitrogen Heterocycles Containing The Benzoazepine Moiety

Sep. 5th

5F-A-1

Kunihiro

Sep. 5th

5F-A-2

Sep. 5th

Chair: Jen-Chieh Hsieh (Tamkang University, Taiwan)

T.

M. Kervefors

Wales

Japan

Chair: Shigeru Arai (Chiba University, Japan)
Non-planar Porphyrinoids as Asymmetric Bifunctional Hydrogen-Bond Donor Catalysts

Poster Presentations
Note: The presentation numbers having an 's' at their end are candidates for Poster Prizes.
Sep. 2nd

2P-001

Yen-KuWu

National Chiao Tung
University

TaiwanSep. 2nd

2P-002

AlexeyZazybinKazakhstan Synthesis and plant growth stimulating activity of morpholine and piperidine ioniccompounds

Sep. 2nd

2P-003s Beatričė

Razmienė

Kazakh-British Technical
University, Satbayev
University
Kaunas University of

PagirePalladium-catalyzed N1-selective allylation of indoles with allylic alcohols promoted bytitanium tetraisopropoxide

Lithuania

Synthesis of novel 2H-pyrazolo[4,3-c]pyridines and investigation of their anti-mitotic activity

BIKAKENJapan

Enantioselective Photocatalysis utilizing 7-Azaindolines as an Auxiliary: Challenges andOpportunities

Technology

Sep. 2nd

2P-004s Santosh

Sep. 2nd

2P-005s Philipp

KramerTu Kaiserslautern

Germany

Enamides as versatile tools for the stereoselective construction of heterocycles

Sep. 2nd

2P-006

Osamu

OnomuraNagasaki University

Japan

Regioselective Addition of Quinoline Derivatives to Carbonyl Compounds via Pd-catalyzed
Umpolung with Diethyl Zinc

Sep. 2nd

2P-007

Ionel

Mangalagiu

Alexandru Ioan Cuza
University of Iasi

Romania

Anticancer and antimicrobial activity of six member ring azaheterocycles

Sep. 2nd

2P-008s Yohei

Ueda

Osaka University

Japan

N,N’-Bis(trimethylsilyl)dihydropyrazine as a Salt-free Reductant for Ni-catalyzed Reductive
C-C Bond Formation of Aryl Halides

Sep. 2nd

2P-009Fung-E

Hong

National Chung Hsing
University

TaiwanPyrrole Ring Formation from the Amido-substituted Benzoquinone Derivatives via
Palladium Catalyzed Carbon-hydrogen Bond Functionalization

Sep. 2nd

2P-010

Muhammet

UyanikNagoya University

Japan

Hypoiodite-catalyzed Chemoselective Oxidative Generation of ortho-Quinone Methides
and Tandem Reactions

Sep. 2nd

2P-011

Shinji

Tanimori

Osaka Prefecture University

Japan

A Rapid Synthesis of Substituted Oxazoles via PIFA-Mediated Oxidative Cyclization of
EnamidesSep. 2nd

2P-012s Mayo

Ishibashi

University of Toyama

Japan

Trialkylborane-Mediated Propargylation of Aldehydes and New Synthetic Approach to
2,3,5-Trisubstituted Furans by Brønsted Catalysis

Sep. 2nd

2P-013s Taka

Sawazaki

The University of TokyoJapan

Development of BODIPY-based photo-oxygenation catalyst that inhibits tau amyloid
formation

Sep. 2nd

2P-014

Suga

Shinshu University

Japan

Lewis Acid-Catalyzed Alcohol Addition Reactions to Cyclic Carbonyl Ylides Generated
from Diazoacyloxazolidinones

Sep. 2nd

2P-015s Kenta

Rakumitsu

Kumamoto University

Japan

Total Syntheses of (–)-Secologanin, (–)-5-Carboxystrictosidine, and (–)-Rubenine

Sep. 2nd

2P-016

Gary Jing

ChuangChung Yuan Christian
University

TaiwanFormal Synthesis of (±)-Pentalenolactone A Methyl Ester

Sep. 2nd

2P-017

HidetoMiyabeHyogo University of Health
SciencesJapan

Tricyclic Oxygen Heterocycles for Aqueous-Medium Thiol-Selective Modification

Sep. 2nd

2P-018UpendraSharmaUniversity of Leuven (KU
Leuven)Belgium

Synthesis of Diversely Functionalized Heterocycles via Trapping of Transient σAlkyl/Vinyl-Palladium (II) Intermediates

Sep. 2nd

2P-019cancelled

Sep. 2nd

2P-020s Shibo

Xu

Osaka University

Japan

Synthesis of Six- and Seven-Membered Benzolactones by Nickel-Catalyzed C-H Couplingof Benzamides with Small-Sized Cyclic Ethers

Sep. 2nd

2P-021

Tzeng

Kaohsiung Medical University Taiwan

Discovery of hydrazide derivatives as glycine N-methyltransferase (GNMT) inducers forthe treatment of hepatocellular carcinoma

Sep. 2nd

2P-022s Ravindra

Aher

Japan

Enantioselective Synthesis of Functionalized Decalins via Desymmetrization of Substituted
Dihydropyrans and 1,3-Diketones

Sep. 2nd

2P-023s Bishoy

El-Aarag

Okinawa Institute of Scienceand Technology Graduate
University
Menoufia University

Egypt

Hepatoprotective activities of 3,5-dihydroxy-7-methoxy-2-(4-methoxyphenyl)-4benzopyrone against CCl4-induced liver fibrosis in mice

Sep. 2nd

2P-024s Mayuki

Goto

Gifu Pharmaceutical University Japan

Development of Carboiodination Reaction of Unsaturated Bonds Using Cationic Iodine

Sep. 2nd

2P-025s Muhammad

SohailJapan

Dynamic Stereoselective Annulation to Afford Spirooxindole Pyran Polycycles

Sep. 2nd

2P-026

Kamimura

Okinawa Institute of Scienceand Technology Graduate
University
Yamaguchi University

Japan

A Novel Higher-order Radical Cascade Provides Efficient Synthesis of a Variety ofHeterocycles

Sep. 2nd

2P-027s Rebecca

WilsonUniversity of HuddersfieldUK

Cyclisations of 3-(o-Substituted-phenyl)penta-1,4-diyn-3-ols: Construction of Bicyclic,
Tricyclic and Tetracyclic Rings Containing N, S and/or O

Sep. 2nd

2P-028s Matthieu

Daniel

CEA - Le Ripault, Orleans
University - ICOAFranceHypervalent Iodine (III) in Direct Intramolecular N-N Bond Formation with HeteroaromaticAmines: Synthesis of Triazapentalene Derivatives

Sep. 2nd

2P-029Burtoloso

University of São Paulo

BrazilTotal Synthesis of Brussonol via Cross-Electrophile Coupling from Epoxides

Clausen

University of Münster

Germany

Formal Anti-Markovnikov Hydromethylation of Olefins

Quadrelli

University of Pavia

Italy

Nitrile Oxide Chemistry in a Renovate Use of Isoxazoles

K.

I.

Hiroyuki

CherngK.

C.

Dattatray

Akio

Sep. 2nd

Antonio
Carlos
2P-030s FlorianB.

Sep. 2nd

2P-031

Sep. 2nd

2P-032s Keitaro

Matsuoka

Hokkaido University

Japan

Synthesis of Functionalized Monoaryl Iodanes(III) via ipso-Substitution Reactions

Sep. 2nd

2P-033

He

Nankai University

China

Cyclization of Spiro(Nitrocyclopropane)-oxindoles with Huisgen Zwitterions and Synthesisof Fused Pyrazole Derivatives

Sep. 2nd

2P-034s Saki

Maejima

Gifu Pharmaceutical University Japan

Development of Lactamization Reaction Through Three-Components Reaction Using
Iodine and Visible Light

Sep. 2nd

2P-035

Zhou

Nankai University

China

Asymmetric Synthesis of Novel Fused Polycyclic 3,4-Dihydropyrano[4,3-b]pyran-5(2H)ones via an Organocatalyzed Formal [3 + 3] Annulation

Sep. 2nd

2P-036s Nikolai

Li-Zhulanov

Novosibirsk State University

RussiaSynthesis of 4-acetamido-octahydrochromene derivatives based on (-)-isopulegol via
Prins-Ritter tandem reaction

Sep. 2nd

2P-037s Toshimasa

Okita

Waseda University

Japan

Pd-Catalyzed Intramolecular C–H Arylation of Aromatic Esters and Nitroarenes

Sep. 2nd

2P-038s Shinobu

Arikawa

Osaka University

Japan

The First Synthesis and Characterization of a Polycyclic Zwitterion with Open-Shell
Character

Sep. 2nd

2P-039s Kazuki

FukushiTohoku University

Japan

Synthesis and Biological Evaluation of 3D Structure-Mimicked Apratoxin A Analogues

Sep. 2nd

2P-040s Ruofang

Hu

Osaka University

Japan

Chemical synthesis and function of <I>Helicobacter pylori</I> peptidoglycan fragments

Sep. 2nd

2P-041

Takashi

Nishikata

Yamaguchi University

Japan

Electron-assisted tert-Alkylative Macrocylization

Sep. 2nd

2P-042

RyukichiTakagi

Hiroshima University

Japan

Intramolecular [2+2] Photocycloaddition using Chiral Phosphoric Acid as a Template

Paolo

Zhengjie

ZhenghongS.

Sep. 2nd

2P-043

Sep. 2nd

InamotoMukogawa Women's
University

Japan

Synthesis of Benzo[b]thiophene-3-Carboxamides via Rhodium-Catalyzed Cyclization of(ortho-Alkynyl)phenyl Sulfides in the Presence of Isocyanates

2P-044s Seitaro

KoshinoTohoku University

Japan

A new methodology to constructing axially chiral biaryls using organocatalyst

Sep. 2nd

2P-045s Florian

OstlerUniversity of Muenster

Germany

Design & Synthesis of Novel Halogen-Bond-Donor Catalysts

Sep. 2nd

2P-046s AMOL

India

Fe (III) Promoted Intramolecular Cascade Cyclization for the Synthesis of Quinoline fused
Selenophene-based Heteroacene Scaffolds

Sep. 2nd

2P-047

Hiroshi

NishinoKumamoto University

Japan

Synthesis of Tripodand- and Dicryptand-Type Compounds Using Mn(III)-Based
Dihydrofuran-Clipping Reaction

Sep. 2nd

2P-048

ToshikiNokami

Tottori University

Japan

Electrochemical Synthesis of Cyclic Oligosaccharides

Sep. 2nd

2P-049Kenji

Sugimoto

University of Toyama

Japan

Novel approaches toward de novo syntheses of N-heterocycles triggered by gold(I)catalyzed aza-enyne metathesis

Sep. 2nd

2P-050Shohei

HamadaKyoto Pharmaceutical
University

Japan

Oxidation of p-Methoxybenzyl Ethers by Electronically Tuned Nitroxyl Radical Catalysts

Sep. 2nd

2P-051

Tun-Cheng

Chien

National Taiwan Normal
University

TaiwanTotal Synthesis of Pseudouridine

Sep. 2nd

2P-052s Tetsuji

Yata

Osaka University

Japan

Regioselective Synthesis of Metalated 2-Pyrones by Intramolecular Oxymetalation Using
Indium Trihalide

Sep. 2nd

2P-053s Iliya

Dragutinovic University of New South

Australia

Accessing Pyrrolodiazine Scaffolds for Kinase Inhibition

Sep. 2nd

2P-054

Fumie

Sakurai

Takeda Pharmaceutical
Company LimitedJapan

Development of Direct and Regioselective Monofluorination of 1-Isoquinolones and 2Pyridones with N-fluorobenzenesulfonimide (NFSI)

Sep. 2nd

2P-055

Tohru

Oishi

Kyushu University

Japan

Structure-Activity Relationship Studies of Maitotoxin Based on the Chemical Synthesis ofPartial Structures

Sep. 2nd

2P-056s Yuki

MORITAKyushu University

Japan

Synthesis of Biologically Active Molecules Based on Unique Right-Side Structure of
Physalins

Sep. 2nd

2P-057

Sengoku

Shizuoka University

Japan

Divergent synthesis of methylene lactone- and methylene lactam-based spiro compounds

Sep. 2nd

2P-058s Tobias

WilckeHeinrich-Heine-University,
Duesseldorf

Germany

Alkynoyl o-Iodo Anilides as Versatile Substrates for the Synthesis of Heterocyclic
Luminophores

Sep. 2nd

2P-059s Mariko

Inoue

Osaka University

Japan

Synthesis of ortho-Aminoalkylated Pyridine Derivatives via Direct C–H Bond
Aminoalkylation Catalyzed by Group 3 Metal Complexes

Sep. 2nd

2P-060s Hideaki

Ikeda

Osaka University

Japan

Metathesis Cleavage of N=N Bond in Benzo[c]cinnolines and Azobenzenes by Ditungsten
Complexes bearing a Metal-metal Triple Bond

Sep. 2nd

2P-061

Motoki

Ito

Meiji Pharmaceuticaluniversity

Japan

Development of Catalytic ortho-Selective C–H Amination of N,N-Dialkylanilines with Rh(II)Nitrene

Sep. 2nd

2P-062

Yuichiro

Kawamoto

Tokyo University of Pharmacy Japanand Life Sciences

Enantioselective Total Synthesis of Diocollettines A

Sep. 2nd

2P-063s Kyohei

UchidaTokyo University of Pharmacy Japanand Life Sciences

Total Synthesis of Applanatumol B

Sep. 2nd

2P-064s Akane

EnomotoKyoto University

Japan

Synthesis of 2-Methylquinoxaline Derivatives from Glycerol and Diamines Catalyzed by
Iridium Complex

Sep. 2nd

2P-065

YazakiKyushu University

Japan

Acylpyrazole as Carboxylic Acid Equivalent Platform for Chemoselective Catalysis

Sep. 2nd

2P-066s Ayuta

Yamaguchi

Kyoto University

Japan

Gold-Catalyzed Cascade Cyclization of Anilines with Diynes: Controllable Formation ofEight-Membered Ring Fused Indoles and Propellane-Type Indolines

Sep. 2nd

2P-067

YamazakiNara University of Education

Japan

Fused pyrrolidine and piperidine formation via intramolecular cycloadditions of styrenederived ethenetricarboxylate amides

Sep. 2nd

2P-068s Takuya

Matsumoto

Kyoto Pharmaceutical
University

Japan

Convergent Synthesis and Growth Inhibitory Activity Evaluation of Stereoisomers around
THF Ring of Acetogenin Thiophene Analogues

Sep. 2nd

2P-069s Chisako

Kanzaki

Kyoto Prefectural University

Japan

Controlled Self-assembly of Porphyrins in Microflow Space

Sep. 2nd

2P-070s Tatsuya

Takahashi

Ritsumeikan University

Japan

Synthesis and Photophysical and Electrochemical Properties of Cationic PyridiniumChlorophyll Conjugates

Sep. 2nd

2P-071s Yusuke

WashinoMeijo University

Japan

Asymmetric [3+2] Annulations of Allenes with Alkylideneoxindoles Catalyzed by Planar
Chiral [2.2]Paracyclophanol-based Phosphines

Sep. 2nd

2P-072

Kato

Toho University

Japan

Pd(II) catalyzed ligand controlled synthesis of bis(3-furanyl)methanones and methyl 3furancarboxylates

Sep. 2nd

2P-073s Karolína

Straková

University of Geneva

Switzerland Fluorescent Probes to Image Physical Forces in Biology

Sep. 2nd

2P-074s Hiromu

HosoyaOsaka University

Japan

Reduction of Nitroarenes for Generating Arylnitrenes by 1,1'-Bis(trimethylsilyl)-1H,1'H-4,4'bipyridinylidene

Sep. 2nd

2P-075s Shinje

MiñozaMindanao State UniversityIligan Institute of Technology

Philippines

A One-Pot, Tandem-Sequential Approach for a Facile and Rapid Synthetic Access to 3Hydroxyflavone Scaffolds

Sep. 2nd

2P-076s Dmitri

Trubitsõn

Tallinn University ofTechnology

Estonia

Enantioselective N-alkylation of Nitroindoles

Sep. 2nd

2P-077

Shigehisa

Musashino University

Japan

Co-catalyzed deprotective cyclization affording cyclic carbamates, ureas, and isoureas

Sep. 2nd

2P-078s Aleksandra

Murre

Tallinn University ofTechnology

Estonia

Diastereoselective α-alkylation of Ammonium Salts

Sep. 2nd

2P-079s Akihiro

SakamaKeio University

Japan

Synthetic Studies of (–)-Callophycoic Acid A

Sep. 2nd

2P-080

Yuichiro

Kadonaga

Osaka University

Japan

Total Synthesis of Peroxide-bridged Jungermatrobrunin A

Sep. 2nd

2P-081

Atsuo

Nakazaki

Nagoya University

Japan

Concise Synthesis of Oxy-Functionalized Steroids through Intramolecular Diels-Alder
Reaction of 2-Pyrone

Sep. 2nd

2P-082s Xue-Song

Zhou

Central China Normal
University

China

Copper-Catalyzed Radical Cross-Coupling of Cycloketone Oxime Esters and Sulfinate
Salts

Sep. 2nd

2P-083

Jiann-Jyh

Huang

National Chiayi University

TaiwanA New Cascade Reaction for the Synthesis of 5,11-Dihydro-6H-indolo[3,2-c]quinolin-6ones as Topoisomerase-I Inhibitors

Sep. 2nd

2P-084Masahiro

Ikejiri

Osaka Ohtani University

Japan

Synthesis and Fluorescence Properties of the Diarylmethylene Analogs of the Green
Fluorescent Protein Chromophore

Sep. 2nd

2P-085s Kazuki

Tojo

Nara institute of science andtechnology

Japan

Synthetic study of suaveolindole and related indolosesquiterpenes

Kiyofumi

Tetsuya

Ryo

Shoko

Keisuke

HirokiD.

SONAWANE Gifu University

WalesSep. 2nd

2P-086s Supriya

RejOsaka University

Japan

Rhodium-Catalyzed Selective C‒H Alkylation of Benzenesulfonamide Derivatives with
Alkenes and Investigation of Its Mechanistic Study

Sep. 2nd

2P-087s Aymen

Skhiri

Osaka University

Japan

Nickel(II)–Catalyzed Reaction of Aromatic Amides with Bicyclic Alkenes through Carbon–
Hydrogen and Carbon–Nitrogen Bond Cleavage

Sep. 2nd

2P-088Masahiro

Noji

Meiji Pharmaceutical
University

Japan

An Immobilized Vanadium-Binaphthylbishydroxamic Acid Complex as a Reusable Catalyst
for the Asymmetric Epoxidation of Allylic Alcohols

Sep. 2nd

2P-089Takahiro

Suzuki

Hokkaido University

Japan

An Intermolecular [4+3] Cycloaddition Reaction Using 3-Hydroxy-2-Pyrone Derivatives withan Oxyallyl Cation

Sep. 2nd

2P-090s Asahi

TakakiWaseda University

Japan

Synthesis of Nitrogen-Containing Seven-and Eight-Membered Compounds via Gold(I)Catalyzed Cycloisomerization

Sep. 2nd

2P-091s Marina

Tane

Waseda University

Japan

Iodine-Catalyzed Asymmetric Synthesis of 4-Imidazolidinones
via Dehydrogenative N-H/C(sp3)-H Coupling Using α-Amino Acids and Amines

Sep. 2nd

2P-092Kazuaki

Katakawa

Musashino University

Japan

Synthesis of Polycyclic Chromene Natural Products Based on Benzyne Cycloaddition
Strategy

Sep. 2nd

2P-093

MakotoSako

Osaka University

Japan

Asymmetric Reactions Using Chiral Vanadium Complex as Acid Catalyst

Sep. 2nd

2P-094s Sari

Urata

Kitasato University

Japan

2,6-Bis(trifluoromethyl)phenylboronic Esters as Protective Groups for Diols: A
Protection/Deprotection Protocol for Use under Mild Conditions

Sep. 2nd

2P-095

OkitsuKobe Pharmaceutical
University

Japan

Iodocyclization of Ynamides for the Construction of Medium-Sized Oxacycles

Sep. 2nd

2P-096s Yuta

Goto

Aichi University of Education

Japan

Chemical synthesis of 4-azido-β-galactosamine derivatives for generation of compound
library with inhibitory activity against GalNAc4S-6ST

Sep. 2nd

2P-097

Masakazu

Nambo

Nagoya University

Japan

Pd-Catalyzed Suzuki–Miyaura Cross-Coupling of a-Fluorinated Benzylic Triflones

Sep. 2nd

2P-098

TakuyaKumamoto

Hiroshima University

Japan

Total synthesis of 6-deoxydehydrokarafungin

Sep. 2nd

2P-099s Tsubasa

NakaueHiroshima University

Japan

Synthetic studies towards natural xanthones blennolides via spiro intermediates

Sep. 2nd

2P-100s Joshua

Nillama

Mindanao State UniversityIligan Institute of Technology

Philippines

A Simple Protocol for the Synthesis of 4-Hydroxyquinolin-2(1H)-one and its Derivatization
with Substituted Benzaldehydes

TakashiTapales

Mindanao State UniversityIligan Institute of Technology

Philippines

Synthesis and Photophysical Properties of Flavylium Salts as Potential Bioinspired Dye
Sensitizer

Khake

Osaka University

Japan

Rhodium(III)-Catalyzed Direct C-H Bond Amidation of Aniline Derivatives Using a
Pyrimidinyl Directing Group

MahatoOsaka University

Japan

Iridium (III)- Catalyzed Direct C-H Alkynylation of Aromatic Acid Derivatives Using an
Imidazole Directing Group

Sep. 2ndP.
Andrew
2P-101s RadynP.
Vanessa
2P-102s Shrikant
Manmathappa
2P-103s Sanjit
Kumar
2P-104s Shiori

TakedaMeiji Pharmaceutical
University

Japan

Determining Nonempirical Absolute Configuration of Chiral Alkyl-substituted Epoxides
Using Bis(zinc porphyrin) as a CD-Sensitive Bidentate Host Molecule

Sep. 2nd

2P-105

TetsuroOsaka City University

Osaka

First Total Synthesis of Antrimycin A and D

Sep. 2nd

2P-106s Shota

Kawai

Kyoto university

Japan

Synthetic Study of Sigillin A, Polychlorinated Polyketide

Sep. 2nd

2P-107s Ruri

KozonoShowa Pharmaceutical
University

Japan

Spontaneous resolution of the chiral crystal and metal complex of N,N'-dimethylpyridine2,6-dicarboxamides bearing pyrimidine

Sep. 2nd

2P-108s Akitomo

Kasahara

The University of TokyoJapan

Conformational Analysis and cis-trans Control of Cyclized Tryptophan Tertiary Amides

Sep. 2nd

2P-109s Haruo

Matsuzaki

Kobe Pharmaceutical
University

Japan

Synthesis of pyrazoles from conjugated hydrazone through acid-promoted βprotonation/nucleophilic addition/cyclization/aromatization sequence

Sep. 2nd

2P-110s Keiji

Konishi

Kobe Pharmaceutical
University

Japan

Copper-Catalyzed Synthesis of Multisubstituted Pyrroles by Cycloisomerization of
Cyclopropenyl Oxime Ether

Sep. 2nd

2P-111s Hiroki

Yamagishi

Kyoto University

Japan

Four-component Coupling Strategy for 2,3,4-Trisubstituted 3,4-Dihydroquinoline

Sep. 2nd

2P-112s Sayuri

Saito

Nagoya City University

Japan

Studies on the Synthesis of Kadcoccilactone A

Sep. 2nd

2P-113MagataOsaka Ohtani University

Japan

Stereoselective Synthesis of Regioisomeric 2,5-Disubstituted Thiazole Amino Acid Units
for Dendroamide A Analogues

Sep. 2nd

2P-114s Takuro

Yamakawa

Kyoto University

Japan

Total Synthesis of Tylophorine and Cryptopleurine

Sep. 2nd

2P-115

Fujisaka

Osaka Ohtani University

Japan

Facile Synthesis of 3-Substituted 2-Trifluoromethylindoles from Trifluoroacetoanilides
Bearing a Vinylogous Electron-withdrawing group

Sep. 2nd

2P-116s Kento

Yokoi

Hokkaido University

Japan

Synthetic Study of 4″α-Substituted cyclic ADP Carbocyclic-ribose as a Target
Identification Probe

Sep. 2nd

2P-117

NemotoChiba University

Japan

Catalytic Asymmetric Dearomatization of Phenols Using Chiral Silver(I) Phosphate forSynthesizing Chiral Spirolactams

Sep. 2nd

2P-118s Haruki

YamauraOsaka University

Japan

Synthesis and function of Alcaligenes faecalis lipid A and its derivative

Sep. 2nd

2P-119s Shunya

SatakeHokkaido University

Japan

Synthetic study of 2”-fluoro analogues of cyclic ADP-ribose (cADPR), a Ca2+ mobilizing
second messenger, as a stable equivalents of cADPR

Sep. 2nd

2P-120s Kenta

DemuraOsaka University

Japan

Diversity-oriented synthesis of multi-antennary N-glycans containing sialic acid

Sep. 2nd

2P-121

Takashi

Otani

National Institute ofTechnology, Anan College

Japan

Synthesis of Highly Fluorescent Polyaza[7]helicenes

Sep. 2nd

2P-122

Hirofumi

NakanoAichi University of Education

Japan

Investigation of reaction conditions to synthesize sulfated GalN3 derivatives with various
phenyls having methoxy groups at O-1 position using closed-vessel reactor

Sep. 2nd

2P-123s Reo

Kondo

Aichi University of Education

Japan

Synthesis of Japanese encephalitis virus infection inhibitor with unsaturated bondintroduced to glucuronic acid having hydroxy or acetamido group at C-2 position

Sep. 2nd

2P-124s Matthias

Krumb

Johannes GutenbergUniversity

Germany

Total Synthesis of a Pentasaccharide Fragment from Arabinogalactan and its Application
for Allergy Prevention

Sep. 2nd

2P-125s Kazusa

Aoki

Sophia University

Japan(Di-(2-picolyl)amino)quinazolines as Fluorescent Probes for ATP

Sep. 2nd

2P-126s Kuo Yuan

Chiu

Institute of Chemistry,
Academia Sinia

TaiwanOrganic Dyes Containing non-Substituted Aryl Amino Moiety and Azobenzene Unit for
Dye-Sensitized Solar Cell

Sep. 2nd

2P-127s Kuo Yuan

Chiu

Institute of Chemistry,
Academia Sinia

TaiwanElectrochemical Study of the imidazole-based star-shaped oligo(benzonitrile)s andapplication for inverted-type MAPbI3 solar cells

Sep. 2nd

2P-128

TanabeKindai University

Japan

Facile Synthesis of Neokotalanol, a Potent α-Glycosidase Inhibitor Isolated from the
Ayurvedic Traditional Medicine “Salacia”

Sep. 2nd
Sep. 2nd
Sep. 2nd

ShinadaTakujiAki

Tetsuhiro

GenzohSep. 2nd

2P-129s Michitaka

Kurimoto

Nagoya University

Japan

Efficient Construction of Quaternary Carbon via Tandem Dibromocyclopropane Ring
Opening/Wagner-Meerwein Rearrangement

Sep. 2nd

2P-130s Toshihiro

MasudaKyoto university, ICR

Japan

Peptide modulating tension in cell membranes: the regulation of cell movement andmorphology via actin remodelingSep. 2nd

2P-131s Sorachi

Miwa

Kyoto University

Japan

Synthesis and structure–ATPase activity relationship of rhodamine derivatives against Pglycoprotein CmABCB1

Sep. 2nd

2P-132Miki

Kyoto University

Japan

Molecular Imaging Utilizing Stimuli-Responsive Dyes Bearing Nucleophilic Substituents

Sep. 2nd

2P-133s Jin

Sakai

Hokkaido University

Japan

Synthesis of Enantiomerically Pure 1,2,3-trisubstituted Cyclopropane Nucleosides

Sep. 2nd

2P-134s Yota

Sakurai

Osaka University

Japan

Facile Synthesis of 5-Hydroxycytidine Analogues: 2'-O-Me-RNA and scpBNA Bearing a 5Hydroxycytosine Nucleobase

Sep. 2nd

2P-135s Mikako

Higa

University of the Ryukyus

Japan

Theoretical Analysis of Absolute Configurations of Natural Organic Compounds

Sep. 2nd

2P-136

Watanabe

RIKEN

Japan

Development of On-Demand Bioconjugation/Deconjugation Platforms

Sep. 2nd

2P-137s Kento

Seki

Muroran Institute oftechnology

Japan

Asymmetric Aldol Reaction of Isatins with Carbonyl Compounds Using Diamino Alcohol
Organocatalyst and Its Application to The Total Synthesis of Indoloquinazoline Alkaloids

Sep. 2nd

2P-138s Midori

KawasakiDoshisha Women's College of Japan
Liberal Arts

Enantioselective Oxidation and Kinetic Optical Resolution of Carboxylic Acids by Chiral
Lithium Amides

Sep. 2nd

2P-139s Manmath

BhusseMuroran Institute oftechnology

Japan

New Amino Amide Alcohol Organocatalysts for Asymmetric Michael Addition of β-Keto
Esters with Nitroolefins

Sep. 2nd

2P-140s Makoto

MiyoshiOsaka University

Japan

Oxidative Rearrangement of Secondary Amines Using Hypervalent Iodine(III) Reagent

Sep. 2nd

2P-141

SakataTohoku University

Japan

Total Synthesis of (+)-CC-1065 via Two Directional Double Ring Expansion of Benzo-bisCyclobutenone Oxime Sulfonate

Sep. 2nd

2P-142s Takuya

Ishii

Kanazawa University

Japan

N-Heterocyclic Carbene-Catalyzed Decarboxylative Alkylation of Aldehydes

Sep. 2nd

2P-143

Iwao

HachiyaMie University

Japan

Sep. 2nd

2P-144

Midori

Arai

Chiba University

Japan

Synthetic Study of (–)-A58365B via a Chiral 2-Pyridone Synthesis Using Conjugate
Additionof
β-Keto Ester
to Chiral Alkynyl
Imine
as a Key Reaction
Synthesis
and Evaluationof Chiral
Spirooxindoles
for Notch Signal Inhibitors

Sep. 2nd

2P-145s Keitaro

Yamamoto

Osaka University

Japan

Development of Quinoidal Oligothiophenes Having Fluorine Atoms

Sep. 3rd

3P-001

ZonidisUniversity of Huddersfield

UK

Synthesis and Photochromism of Bis(Thienyl) Substituted 1,2-Oxathiine 2,2-dioxides

Sep. 3rd

3P-002Maegawa

Kindai University

Japan

Benzofuran synthesis from 2-hydroxychalcones via chloromethoxylation using hypervalentiodine reagent

Sep. 3rd

3P-003s Martin

Petzold

TU Braunschweig

Germany(3+3)‐Annulation of Carbonyl Ylides with Donor–Acceptor Cyclopropanes: Synergistic
Dirhodium(II) and Lewis Acid Catalysis

Sep. 3rd

3P-004s Ankita

Bal

National Institute of Scence
Education and Research

India

Nitrenium Ion from λ3-Iodanes

Sep. 3rd

3P-005s Khokan

Choudhuri

India

Advanced method for the construction of C-S bond via C-H functionalization

Sep. 3rd

3P-006s Quanqing

Zhao

National Institute of Science
Education and Research(NISER),
Bhubaneswar
Central China
NormalChina

Visible-Light-Driven Neutral Nitrogen Radical Mediated Intermolecular Styrene
Difunctionalization

Sep. 3rd

3P-007s Dong-Mei

Yan

Central China Normal
University

China

Dual Copper and Photoredox-Catalyzed Cross-Coupling of Alkenes, OBenzoylhydroxylamines, and Sulfur Ylides

Sep. 3rd

3P-008s Kosuke

Okada

Tohoku University

Japan

Total Synthesis of (–)-Deoxoapodine

Sep. 3rd

3P-009s Yuya

KakiuchiOsaka UniversityJapan[2+2+1] Pyrrole Synthesis from Alkynes and Azobenzene via N=N Bond Cleavage
Catalyzed by Vanadium Complexes

Sep. 3rd

3P-010s Tagui

NaganoKyoto University

Japan

Optically Active trans-Cyclooctene-pyridine Ligands in Rhodium-catalyzed Asymmetric 1,4Addition

Sep. 3rd

3P-011s Christopher R.

Opie

Institute of Microbial
Chemistry, BIKAKEN

Japan

Systematic examination of catalytic amide bond formation by the readily accessible
B3NO2 heterocycle-containing molecule Pym-DATB

Sep. 3rd

3P-012s Takahiro

Asada

Osaka University

Japan

Complexation between Al(C6F5)3 and N-Phoshpnine Oxide-Substituted Imidazolidenes

Sep. 3rd

3P-013s MiguelParajaUniversity of Geneva

Spain

Anion-π Catalysis for Epoxide-Opening Ether Cyclizations, from Monomers to Oligomers,
Challenging Baldwin Rules

Sep. 3rd

3P-014s Piotr

DrelichLodz University of Technology Poland

Synthesis of γ,γ‐Disubstituted Butenolides through a Doubly Vinylogous Organocatalytic
Cycloaddition

Sep. 3rd

3P-015s Takuya

Murai

Institute for Chemical
Research, Kyoto University

Japan

Chalcogen-Bond Assisted Dirhodium Complex –Total Syntheses of Naturally Occurring γLactones–

Sep. 3rd

3P-016s Onnicha

Khaikate

Mahidol Univesity

ThailandIntramolecular cyclization of o-alkynylisocyanobenzenes: synthesis of 3-substituted
quinolin-2(1H)-ones and 2-sulfonyl- and 2-thiocyanato-3-substituted quinolines

Sep. 3rd

3P-017

Shinobu

Honzawa

Niigata University of Pharmacy Japanand Applied Life Sciences

Synthesis and Fluorescence Spectra of 5- or 6-Substituted 2-(4-Aminophenyl)-1,3benzothiazole Derivatives

Sep. 3rd

3P-018Hisanori

Nambu

University of Toyama

Japan

Concise Synthesis of Aspidospermidine from Spirocyclopropane through Ring-Opening
Cyclization–Regioselective Alkylation Sequence

Sep. 3rd

3P-019s Koushi

Sugiyama

University of Toyama

Japan

Stereoselective Synthesis of Actinoallolide A Furanone Fragment Using Rh(II)-Catalyzed
O-Ylide Formation-Rearrangement Followed by C-H Amination

Sep. 3rd

3P-020

Giomi

Florence University

Italy

Pyridyl and quinolyl methanols as valuable reagents for metal-free reductions ofaromatic/heteroaromatic nitro compounds and imines

Sep. 3rd

3P-021s Young-In

Jo

Korea University

Republic of Concise Total Synthesis of Phenanthroindolizidine and Phenanthroquinolizidine Alkaloids
Korea

Sep. 3rd

3P-022s Lisa Marie

KammerJohannes Gutenberg
University Mainz

Germany

Visible Light-Induced Sulfonylation/Arylation of Styrenes in a Double Radical ThreeComponent Photoredox Reaction

Sep. 3rd

3P-023s Jonas

Kühlborn

Johannes GutenbergUniversity Mainz

Germany

Xylochemical Synthesis of Natural Products

Sep. 3rd

3P-024s Kirsty

Anderson

University of Auckland

New
Zealand

A new indole to benzoxazole rearrangement enabled by C-H borylation

Sep. 3rd

3P-025

Mase

Shizuoka University

Japan

CSTR Synthesis of Fairy Chemicals Using Fine Bubble and Flow Optimization Method

Sep. 3rd

3P-026s Ryo

NozawaYamaguchi University

Japan

Preparation of Bicyclic Stannolanelactam via Radical Cascade Reaction

Koji

Kenji

Juri

A.

Dimitrios
Christodoulos
Tomohiro

Donatella

Nobuyuki

UniversitySep. 3rd

3P-027s Masaki

Fujie

Osaka University

Japan

Synthesis of Hypervalent Iodine Reagents Bearing Cationic Heterocycles and Application
to Oxidative Cyclization

Sep. 3rd

3P-028

HikawaToho University

Japan

Gold(III)-Catalyzed Decarboxylative C3-Benzylation of Indole-3-carboxylic Acids with
Benzylic Alcohols in Water

Sep. 3rd

3P-029s Hayate

IshizukaTokyo University of Agliculture Japanand Technology

Intramolecular Hydroamination of N-Alkoxyamides under Blue LEDs mediated a
Photoredox Catalyst conditions

Sep. 3rd

3P-030

Qiu

Hunan University

China

Synthesis, Application and Coordinatiion Chemistry Study of Water-Tolerant
Oganoantimony Complexes

Sep. 3rd

3P-031s Yusuke

HaradaKobe University

Japan

Computational Study for the Selective Aromatic Nucleophilic Substitution on 4Dimethylamino-2-methoxy-3-trifluoroacetylquinoline

Sep. 3rd

3P-032

Sato

Setsunan University

Japan

Fluorinated isoxazoles and isoxazolines: Synthesis, reaction and bioactive evaluation

Sep. 3rd

3P-033s Keitaro

Umeno

Kyushu University

Japan

Synthetic Study of the C30–C63 Section of Karlotoxin 2

Sep. 3rd

3P-034s Tsubasa

Hironaka

Okayama University

Japan

Acylative Desymmetrization of meso-1,3-Diols by Chiral DMAP Derivatives

Sep. 3rd

3P-035s Rikako

Nagai

Waseda University

Japan

Synthesis of Silicon-Containing Fused Polycyclic Compounds by Consecutive
Intramolecular Dehydro-Diels-Alder Reactions of Silicon-Tethered Tetraynes

Sep. 3rd

3P-036

Kitajima

Chiba University

Japan

Isolation and Asymmetric Total Synthesis of New Biphenyl Quinolizidine Lactone Alkaloids
from Heimia salicifolia

Sep. 3rd

3P-037s Kohei

Takemoto

Meijo University

Japan

Site-Selective Esterification of α- Hydroxyamides in Polyols by Metal Template Strategy

Sep. 3rd

3P-038s Yuko

Ikeda

Kwansei Gakuin University

Japan

Direct α-Heteroarylation of Heteroatom-Containing Aliphatic Compounds through a
Radical Chain Mechanism

Sep. 3rd

3P-039s Yundong

Chung

Seoul National University

Republic of Formal Synthesis of (−)-cephalotaxine via Proline Ester Enolate Claisen Rearrangement
Korea

Sep. 3rd

3P-040s Yeonji

Kim

Seoul National University

Republic of Asymmetric synthesis of Cα-Quaternary Proline via Chirality Transfers: Application to the
Korea
Total Synthesis of (–)-Amathaspiramide F.

Sep. 3rd

3P-041s Ryoya

Imaizumi

Meiji University

Japan

Synthesis of Toxoflavin derivatives and Uracil derivatives

Sep. 3rd

3P-042s Takumi

FukudaThe University of TokyoJapan

Total Synthesis of Diospyrodin

Sep. 3rd

3P-043s Sitanan

Sartyoungkul

Osaka University

Japan

Synthesis and Properties of Cup- and Bowl-shaped Cyclic Trilactams and Its Derivatives

Sep. 3rd

3P-044

TsubogoTokyo University of ScienceJapan

Total Synthesis of Antibiotic CJ-16,264

Sep. 3rd

3P-045s Kohei

Aoki

Kwanseigakuin University

Japan

Direct α-Heteroarylation of Alcohols with Heteroaryl Chlorides through a Radical Chain
Mechanism

Sep. 3rd

3P-046s Shohei

Yoshioka

Osaka University

Japan

Metathesis reaction of Aryldimethylpropenylsilane

Sep. 3rd

3P-047s Yosuke

Ashikari

Kyoto University

Japan

Functionalization of Organic Azides via Generation and Reactions of Organolithiums
bearing Masked Azides using Flow Microreactors

Sep. 3rd

3P-048s JYOTICHAUHANSHIV NADAR UNIVERSITY,
GREATER NOIDA,

INDIA

Sep. 3rd

3P-049Nagasawa

Tohoku University

Japan

Design, synthesis and biological evaluation of a novel library of antimitotic C2aroyl/arylimino tryptamine derivatives that are also potent inhibitors of indoleamine-2,3dioxygenase(IDO).
Oxidative
Transformationsof Alkenes Employing Azaadamantane-type Oxoammonium

Hidemasa

RenhuaKazuyukiMariko

Tetsu

Shota

Salts

Sep. 3rd

3P-050s Yuki

Wada

Osaka University

Japan

Synthesis of Metal-Free NIR Dyes by One-Pot Ring-Closing
Metathesis(RCM)/Oxidation/1,3-Dipolar Cycloaddition Reaction

Sep. 3rd

3P-051s Kei

Soeda

Osaka University

Japan

Design and Synthesis Conformationally Restricted of Acetogenin Derivatives with Fusedbis THF Skeleton

Sep. 3rd

3P-052s Ferdinand

H.

LutterLMU Munich

Deutschlan Cobalt-Catalyzed Acylation-Reactions of (Hetero)arylzinc Pivalates with OrganicdThiopyridylester Derivatives

Sep. 3rd

3P-053s Maximilian

S.

Hofmayer

LMU Munich

Germany

Stereoselective Cobalt-Catalyzed Cross-Couplings of α-Bromocarbonyl Compounds

Sep. 3rd

3P-054s Toshitaka

OkamuraTohoku University

Japan

Novel Difluoropropargylation of Alcohols and Ketones with Difluoropropargyl Dicobalt
Complexes; Access to Various Cyclic a-Fluoroethers

Sep. 3rd

3P-055s Juri

Skotnitzki

Ludwig-Maximilians-University Germany
MunichPalladium-catalyzed Stereoselective Csp3-Csp2 Cross-Couplings of Chiral Secondary
Alkylzinc Reagents with Alkenyl and Heteroaryl Halides

Sep. 3rd

3P-056s Takumi

MaesatoOsaka University

Japan

Selective Synthesis of Benzonaphthosilines by Rhodium-Catalyzed [2 + 2 + 2]
Cycloaddition

Sep. 3rd

3P-057s Taiki

Ogawa

Kyoto University

Japan

Synthetic study of tubingensin B, a hexacyclic indole diterpenoid natural productSep. 3rd

3P-058s Kyoungmin

Kang

Osaka University

Japan

Synthesis of 2-Substituted Indoles and Benzofurans Using Carbozincation of Alkynyl
EthersSep. 3rd

3P-059

Kondo

Japan

Room-Temperature, Metal-Free and One-Pot Preparation of 2H-indazoles via a Mills
Reaction and Cyclization Sequence

Sep. 3rd

3P-060s Tomohiro

KimuraThe Institute of Scientific andIndustrial Research (ISIR),
Osaka
University
Kyoto University

Japan

Catalyst-Free Aromatic C-H Amidation Using Newly Designed N-Acyliminoiodinanes

Sep. 3rd

3P-061

InagakiKobe Gakuin University

Japan

Coinage Metal Catalyzed 7-Endo-Trig Cyclization of Ene-Dios: Construction of 2,2Dimethyloxepane Frameworks

Sep. 3rd

3P-062s Daiki

KuwanaThe University of Tokyo

Japan

Installation of O-Heterocycles to N-Heteroarenes via an Et3B/O2- Mediated Radical
Reaction of α-Alkoxy and α-Alkoxyacyl Tellurides

Sep. 3rd

3P-063s Asumi

Iida

Shibaura Institute ofTechnology

Japan

N-C Axially Chiral Quinazolinones with ortho-Fluorophenyl Group and the Application to
Enolate Chemistry

Sep. 3rd

3P-064s Tomomi

Imai

Shibaura Institute ofTechnology

Japan

Synthesis of Optically Pure Bioactive N-C Axially Chiral Quinazolinone Derivatives

Sep. 3rd

3P-065s Tomohiro

Tsuda

Osaka University

Japan

Selective Synthesis of 8H-Benzo[e]phenanthro[1,10-bc]silines under Palladium Catalysis

Sep. 3rd

3P-066s Fei

Rao

Kindai University

Japan

A Convenient Synthesis of Hemithioindigo by the Cyclization of 2'-Mercaptochalcone with
NBS under Mild Conditions

Sep. 3rd

3P-067Hiromichi

Egami

University of Shizuoka

Japan

Asymmetric Dearomatizing Fluorination of Indole Derivatives under Phase-Transfer
Catalysis

Sep. 3rd

3P-068

ChihiroTsukanoKyoto University

Japan

Asymmetric Synthesis of γ-alkoxybutenolides by the Thiourea-Ammonium salt-catalyzed
Acetalization and Its Application

Sep. 3rd

3P-069s Lingaiah

MaramOIST, OKINAWA

JAPAN

Synthesis of Ployoxy-Functionalized Piperidines via Mannich and Micheal Reactions ofCarbohydrate Derivatives

MasaruFuyuhikoSep. 3rd

3P-070s Waku

Shimizu

Chiba University

Japan

Absolute Asymmetric Flavanone Synthesis involving Dynamic Enantioselective
Crystallization Process

Sep. 3rd

3P-071s Naoyoshi

IshidaOsaka University

Japan

Cu(I)-Catalyzed Pentafluoroethylation of Aryl Iodides Using Tetrafluoroethylene and CsF

Sep. 3rd

3P-072s Keita

AshidaOsaka University

Japan

Enantioselective Synthesis of Chiral γ-Lactams by Ni(0)-Catalyzed Asymmetric
Carbonylative Cycloaddition

Sep. 3rd

3P-073s Shohei

OhnoOsaka University

Japan

Ni-Catalyzed Cleavage and Formation of C-O Bond to give Disubstituted Benzofurans

Sep. 3rd

3P-074s Jiawei

Qiu

Osaka University

Japan

Ir-catalyzed Cycloisomerization between Aryl Enol Ether and Silylalkyne to Give 2,3Disubstituted Benzofurans

Sep. 3rd

3P-075s Kohei

Teratani

Kyushu Institute of Technology Japan

Novel synthesis method of γ-lactam from Vinylketenimine-iron complexes

Sep. 3rd

3P-076s Yusuke

Tokuhiro

Kyoto University

Japan

Organocatalyzed Enantioselective Addition of Glyoxylate Cyanohydrin to Imines for
Divergent and Scalable Synthesis of α-Keto-β-Amino Acid Analogues

Sep. 3rd

3P-077

Ishihara

Meijo university

Japan

Various Tetrazoles Synthesis from Ketoximes Using DPPA : Substrate Scope andLimitations

Sep. 3rd

3P-078s Yu

Nakamura

Tokyo Medical and Dental
University

Japan

Facile Synthesis of Diverse Heterocyclic Compounds via Au-Catalyzed Cyclization andGeneration of Arynes

Sep. 3rd

3P-079

Fumitoshi

Shibahara

Gifu University

Japan

Imidazo[1,5-a]pyridine-derived NHC-type Carbenes as a Ligand for Catalysts:
Characterization and Reactivity in Catalyses

Sep. 3rd

3P-080

KotaroKikushima

Ritsumeikan University

Japan

Synthesis of Aryl Esters through Accelerated Ligand Coupling of Diaryliodonium(III) Salts

Sep. 3rd

3P-081s Sota

Uno

Toho University

Japan

Suppressing Decarbonylation with Silanes during Stille Coupling Reaction of Aromatic Acid
Chlorides with Heterocyclic Stannane

Sep. 3rd

3P-082s Chika

Nishimura

Osaka University

Japan

Catalytic Synthesis of Isoquinolines from 1,5-Yne-Imines through Migration of N-Aryl
Sulfonyl Groups

Sep. 3rd

3P-083s Kazuma

Ban

Chiba University

Japan

Dynamic Enantioselective Crystallization of Axially Chiral Nicotinamides

Sep. 3rd

3P-084s Tomohiro

KuroseKyoto University

Japan

Synthetic Studies of Lyconesidines Based on Domino Ring-Transformation Strategy

Sep. 3rd

3P-085s Natsuki

Kato

Kyoto University

Japan

Chemoselective, Decarboxylative Acylation of Amines.

Sep. 3rd

3P-086s Sanae

Izumi

Kyoto University

Japan

Borinic Acid Catalyzed Anomeric O-Alkylation for the Synthesis of 1,2-cis-Glycosides

Sep. 3rd

3P-087s Marvin

MantelHeinrich-Heine-Universität
Düsseldorf

Germany

Bio- and Organocatalysts in Highly Enantioselective One-Pot-Cascades

Sep. 3rd

3P-088s Tsubasa

Matsuzawa

Tokyo Medical and Dental
University

Japan

Facile Synthesis of N-Arylphenothiazines by Rearrangement of o-Sulfanylanilines

Sep. 3rd

3P-089s Mahiro

Sakuraba

Osaka University

Japan

Complexation between Lewis Acids and N-Phosphine Oxide-substituted Imidazolylidenes(PoxIms)

Sep. 3rd

3P-090s Yusuke

Yoshikawa

Osaka University

Japan

Total Synthesis of (-)-Aplysiallene and it’s Biological Active Study

Sep. 3rd

3P-091s Hikari

KashouYamaguchi University

Japan

Structural Properties and Antifungal Activities of Heterocyclic Compounds Bearing a
Heavier Pnictogen(III) Center

Sep. 3rd

3P-092

Daisuke

Yamamoto

Kitasato University

Japan

Development of Catalytic Oxidative Difunctionalization Reactions of Carbon-Carbon
Double Bond Using Molecular Oxygens in the Air

Sep. 3rd

3P-093s Ryotaro

Yoshizaki

Kyoto University

Japan

Asymmetric Cyanation of Acylsilanes with Chiral Lewis Base Catalysts

Sep. 3rd

3P-094s Priscilla Mei

Yoong

Osaka City University

Japan

Studies on Total Synthesis of Polycitorol A Utilizing Hg(OTf)2-Catalyzed
Cycloisomerization Reaction

Sep. 3rdYen
3P-095s HIroki

Murakami

Kyoto University

Japan

Development of a New Asymmetric α-Protonation in Aza-Michael Addition of α,βUnsaturated Carboxylic Acids Catalyzed by Chiral Multifunctional Thiourea-Boronic Acid

Sep. 3rd

3P-096s Kento

Nishikibe

Osaka City University

Japan

Asymmetric Total Synthesis and Structural Elucidation of Marine Triterpene Polyethers(−)-Aplysiol B and (+)-Saiyacenol A with Potent Antitumor Activity

Sep. 3rd

3P-097s Ikumi

Kobayashi

Waseda University

Japan

Highly Enantio- and Stereoselective Construction of ent-Atisane Scaffold via
Organocatalytic Asymmetric Intramolecular Michael Reaction and [4+2] Cycloaddition

Sep. 3rd

3P-098s Ramon

Avena

Osaka University

Japan

Sep. 3rd

3P-099s Shintaro

MatsumotoKwansei Gakuin University

Japan

Synthesis and Fluorescent Properties of 5Phenylisoindolo[2,1-a]quinoline
and Isoindolo[1,2-a]isoquinoline Dyes via One-pot Ring-closing Metathesis/
Oxidation/1,3-Dipolar
Cycloaddition
Reaction
Constructionof 4,6-O-(R)-HHDP
Group
by Intramolecular Oxidative Coupling

Sep. 3rd

3P-100s Kazuki

MurataTokyo Institute of Technology Japan

Studies on stereoselective synthesis of lactonamycin

Sep. 3rd

3P-101s Yuki

Yamamoto

Osaka Prefecture University

Japan

Metal-Free and One-pot Synthesis of β-Lactam Derivatives via 4,6-Dihydroxysalicylic AcidCatalyzed Oxidative Coupling of Amines to Imines under Mild Conditions

Sep. 3rd

3P-102

Sato

Kyoto University

Japan

Theoretical Study on Self-assembly process of Octahedron-shaped Molecular Capsule

Sep. 3rd

3P-103s Minami

KimuraKyoto University

Japan

Theoretical study on the isomerization mechanism of α-acids

Sep. 3rd

3P-104s Ryo

Fujimura

Kyusyu Institute of Technology Japan

Pd(II)-Catalyzed Acetalization with Diazoquinone

Sep. 3rd

3P-105s Tatsuro

Yoshinaga

Kyushu University

Japan

Synthesis of Distorted 1,8,13-Trisilyltriptycenes and its Transformation into Heterocyclic
Cage Molecules

Sep. 3rd

3P-106s Junyi

HanOsaka University

China

Synthesis and Properties of Sumanene-Ruthenium Complex

Sep. 3rd

3P-107

SawanoAoyama Gakuin University

Japan

Efficient Synthesis of Azatriphenylenes by Iridium-Catalyzed [2+2+2] Cycloaddition of
Biaryl-Linked Diynes with Nitriles

Sep. 3rd

3P-108s Akito

TomidaTohoku University

Japan

Concise total synthesis of haouamine A·B and their derivatives

Sep. 3rd

3P-109s Koichi

Higashio

Osaka University

Japan

Enantiodivergent and Quantitative Conversion of Racemic Propargyl Alcohols into Their
Both Enantiomers Using Lipase-Catalyzed Dynamic Kinetic Resolution

Sep. 3rd

3P-110s Hiroki

Ishikawa

Chiba University

Japan

Chiral Symmetry Breaking of Spiropyrans and Spirooxazines

Sep. 3rd

3P-111s Woohyeong

Lee

Pusan National University

Korea

Regio- and Stereoselective Hydroarylation of Alkynes with Azoles

Sep. 3rd

3P-112s Birakishore

Padhi

Pusan National University

Korea

Synthesis of Polycyclic Heterocycles by Annulation with Alkenes

KotaroB.

Francisco

Hirofumi

TakahiroSep. 3rd

3P-113

Sep. 3rd

ShiraiResearch Foundation ITSUU
Laboratory

Japan

Nickel-Catalyzed Regioselective Olefin Migration Reaction

3P-114s Naoki

KimuraKeio University

Japan

Fe(PMe3)4-Catalyzed C–H Alkylation of Aromatic Ketones with N-Alkenylindoles andPartial Indolylation via 1,4-Iron Migration

Sep. 3rd

3P-115s Yuya

Tatsui

Osaka University of
Pharmaceutical Sciences

Japan

C4-Functionalization of Pyrazoles by Buchwald-Hartwig Coupling Reaction

Sep. 3rd

3P-116s Takashi

Eto

Kyushu Institute of Technology Japan

Diazotization of phenol using azido imidazolinium salt

Sep. 3rd

3P-117

Sumii

Nagoya Institute ofTechnology

Japan

Synthesis of Pyrazole-3-triflones via [3+2] Cycloaddition Reaction

Sep. 3rd

3P-118s Mizushi

Yanagihara

Osaka University

Japan

Reaction of Aromatic Methoxymethyl Ethers with Trialkylsilyl Triflate and 2,2’-Bipyridyl:
Deprotection and Direct Conversion to Aromatic Triethylsilyl Ethers

Sep. 3rd

3P-119s Shu

Sakurai

Osaka University

Japan

Synthetic Study of Bryostatin

Sep. 3rd

3P-120s Tatsuhiko

Sakaguchi

Kyoto University

Japan

gem-Diboronic Acid-Catalyzed Dehydrative Peptide Synthesis

Sep. 3rd

3P-121s Ryuta

Wada

Gifu University

Japan

Synthesis of Sulfur-Containing Fused Ring Compounds Using Thionyl Chloride as a Sulfer
SourceSep. 3rd

3P-122

Ohrui

Research Foundation ITSUU
Laboratory

Japan

Essential structure of orexin 1 receptor antagonist YNT-707

Sep. 3rd

3P-123s Yasunori

Shio

Osaka University

Japan

Nickel Nanoparticle-catalyzed Ligand-free C(sp2)-C(sp3) Kumada Coupling

Sep. 3rd

3P-124s Makito

YamadaOsaka university

Japan

Ligand-free Suzuki-Miyaura Coupling of Chlorinated Heterocycles using Continuously
Irradiating Microwave and Glass-Supported Palladium Nanoparticle Catalyst

Sep. 3rd

3P-125s Kousuke

OhyamaTohoku university

Japan

Total Synthesis of JBIR-126 toward Elucidation of Structure Activity Relationships

Sep. 3rd

3P-126s Yuichi

Kuboki

Osaka University

Japan

Efficient synthesis of N-trifluoromethylthiomethyl indoles: Physical property, metabolism
and IDO inhibitory activity evaluation of substituted indoles

Sep. 3rd

3P-127

KurouchiResearch Foundation ITSUU
Laboratory

Japan

Strong acid-promoted C-N bond cleavage of tetrahydroisoquinoline derivatives

Sep. 3rd

3P-128s Naoko

Oyobe

Osaka University

Japan

Synthesis of cis-3,4-disubstituted piperidines

Sep. 3rd

3P-129IshidaShowa Pharmaceutical
University

Japan

Design and synthesis of the vitamin D receptor ligand containing three-memberedheterocyclic ring

Sep. 3rd

3P-130s Chisato

YoshikawaShowa Pharmaceutical
University

Japan

A facile synthesis of coumarin conjugated PPARγ Ligand

Sep. 3rd

3P-131

Hirao

Osaka University

Japan

Synthesis and Aggregation Properties of Deazahypoxanthine Derivatives Bearing Multiple
Hydrogen-Bonding Sites

Sep. 3rd

3P-132s Kyoka

KagawaKyoto Prefectural University

Japan

Synthetic Study of Blespirol Using a Novel Rearrangement Reaction

Sep. 3rd

3P-133

Nakamura

Kindai University

Japan

Selective Synthesis of Disubstituted Isoxazole Isomers by the Rearrangement ofChalcones Mediated by Hypervalent Iodine Reagents

Sep. 3rd

3P-134s Nikolay

Zimnitskiy

Ural Federal University

Russia(2Z,4E)-3-Hydroxy-1,5-diarylpenta-2,4-dien-1-ones in the reaction of [3+2] cycloaddition
with stabilized azomethine ylides

Sep. 3rd

3P-135s Hayato

Saito

Osaka University

Japan

An Efficient Method for the Construction of cis-1,2-oxazadecaline Skeleton and its
Application to Formal Enantioselective Synthesis of Trichodermamide B and C

Sep. 3rd

3P-136

KomineNagasaki University

Japan

Formal Synthesis of Haliclonin A Using Tandem Radical Reaction

Sep. 3rd

3P-137s Toshiki

AkiyamaOsaka University

Japan

Iron(0) Nanoparticle-catalyzed Ligand-free C-C/C-N Bond Forming Tandem Reaction

Sep. 3rd

3P-138s Landmark

MSU-IIT

Philippines

A Pot-Economical Approach for Accessing Pyrimidines via a Chalcone Intermediate

Sep. 3rd

3P-139s Ryo

Ninomiya

Kyoto University

Japan

Asymmetric Desymmetrization of 1,3-Alkane Bisphenols via Organocatalytic Aromatic
Bromination

Sep. 3rd

3P-140s Kenta

MoritaOsaka University

Japan

One-pot synthesis of THF rings using phosphonium salts : Formal synthesis ofAmphidinolide F

Sep. 3rd

3P-141s Satoru

Hirabayashi

Osaka University

Japan

Pd-Catalyzed Migratory Cycloisomerization of N-Allyl-o-allenylaniline Derivatives

Sep. 3rd

3P-142AndreaPenoniUniversità degli Studidell'Insubria

ItaliaRegioselective Synthesis of 3-Aroylindoles by Cycloaddition of C-Nitrosoaromatics with
Alkynones

Sep. 3rd

3P-143

Karanjit

Sangita

Tokushima University

Japan

Development of Active and Stable Hydrotalcite‒supported Pd and Pd/Ag Bimetallic
Nanocluster Catalysts for Reactions under Mild Conditions

Sep. 3rd

3P-144

Yasufumi

Fuchi

Showa Pharmaceutical
University

Japan

Fluorescence properties of push-pull type benzoquinoline derivatives

Sep. 3rd

3P-145Masanari

KimuraNagasaki University

Japan

Cu-Catalyzed Stereoselective Formation of 2,5-Dihydro-1,2-oxaborole from Alkyne,
Aldehyde, and Organoborane

Sep. 5th

5P-001s Jeremy

Dobrowolski

The University of New South
Wales

Australia

Biologically Active Novel Nitrogen Heterocycles Containing The Benzoazepine Moiety

Okuda

Okayama Univesity of Science Japan

Regio-divergent Syntheses of Heteroatom-Substituted 1,2,3-Triazoles via CopperCatalyzed Click Reaction of Phosphorylethynes

Takahiro

Yuji

SayakaHiroaki

HiroakiYasukazu

Akira

Keita

ConradYasuhiroS.

M. Estopa

Sep. 5th

5P-002

Sep. 5th

5P-003s Hikaru

Watanabe

Okayama University of
ScienceJapan

Perylene Photocatalyst-Promoted Desulfonylation of Ethenyl Sulfones

Sep. 5th

5P-004

Osamu

TamuraShowa Pharmaceutical
University

Japan

Inverse-Electron-Demand Diels–Alder Reactionsof α,β-Unsaturated Hydrazones withα-Pyrones Having Electron-Withdrawing Group

Sep. 5th

5P-005

Kosho

MakinoTokyo University of ScienceJapan

Chemoselective demethylation of methoxypyridine

Sep. 5th

5P-006

Kazuhiro

HiguchiMeiji Pharmaceutical
University

Japan

Palladium-Catalyzed Oxidative Cyclization: Application to the Synthesis of Lapidilectine B

Sep. 5th

5P-007s Kohei

YasudaOsaka City University

Japan

Synthetic Study of Phomopsin A : Catalytic Asymmetric Synthesis of β-OH-DOPA

Sep. 5th

5P-008

Nakajima

Kumamoto University

Japan

Dramatic Enantioselectivity Reversal in the Propargylation of Aldehyde with Alkynyllithium
Catalyzed by Dilithium Binaphtholate Derivatives

Sep. 5th

5P-009s Keigo

Sato

Chiba University

Japan

Total Syntheses of Pleiocarpamine, Normavacurine, and C-Mavacurine

Sep. 5th

5P-010s Kasumi

Miyoshi

Mukogawa Women's
University

Japan

Synthesis of pemetrexed medoxomil ester prodrugs aiming for the oral administration

MakotoSep. 5th

5P-011s Takuma

Sasayama

Waseda University

Japan

New Polyazahelicenes: Facile Synthesis by Consecutive N-H/C-H Coupling with
Hypervalent Iodine and Evaluation of Their Photophysical Properties

Sep. 5th

5P-012s Hanbi

Kim

Kangwon University

Korea

Partial reduction of isopropyl esters to aldehydes using MeLi catalyzed hydroboration

Sep. 5th

5P-013

Hidetsugu

TabataTeikyo University

Japan

Conformational properties based on the axis of 6N-benzoyl- and 6N-p-tosyl-1,6benzodiazocines: Comparison with those of 1,5-benzodiazepines

Sep. 5th

5P-014ASHOKDONGAMANTIOSMANIA UNIVERSITY,

India

Synthesis of diverse heterocyclic library consisting macrocyclic moieties

HYDERABAD

Sep. 5th

5P-015Masanori

Kitamura

Kanazawa University

Japan

Triazine-Based Dehydrative Condensing Reagents Bearing Carbon-Substituents

Sep. 5th

5P-016

Nobuyoshi

MoritaShowa Pharmaceutical
University

Japan

Gold-catalyzed One-Pot Synthesis of Oxazoles from 3-Trimethylsilyl Propargylic Alcohols
and Amides

Sep. 5th

5P-017

Eiji

Yamaguchi

Gifu Pharmaceutical University Japan

Development of visible light/iodine mediated inter/intramolecular CDC type reaction ofheteroarenes.

Sep. 5th

5P-018s Naoki

Yasukawa

Gifu Pharmaceutical University Japan

Highly-Functionalized Pyrrole Synthesis via 3,6-Dihydro-1,2-oxazines using
Heterogeneous Copper Catalyst

Sep. 5th

5P-019

TanakaNagasaki International
University

Japan

Synthesis of aggregation inductive luminous organic fluorescence dyes, and evaluation of
their fluorescence properties

Sep. 5th

5P-020s Jiye

Jeon

Korea University

Republic of Total Synthesis of Hinckdentine A
Korea

Sep. 5th

5P-021s Jooyeon

Yoon

Korea University

Republic of Development of Novel Protocols for Synthesis of 2-Arylquinolines from 2-Aminochalcones
Korea
via Nucleophile-catalyzed Dehydrative Cyclization

Sep. 5th

5P-022

Takamura

Okayama University

Japan

Unified Total Synthesis, Stereochemical Elucidation, and Antifouling Activity ofSarcophytonolides

Sep. 5th

5P-023s Asaki

Miyairi

Hokkaido University

Japan

Au(I)-Catalyzed Sequential Reaction of Ynamide for Synthesis of γ,δ-Unsaturated Amides
and Polysubstituted Furans

Sep. 5th

5P-024s Masatoshi

Takabatake

Okayama University

Japan

Synthesis and Properties of Ethene-Bridged Terthiophene Multi-Oxides

Sep. 5th

5P-025s Simon

GrasslLMU Munich

Germany

Transition Metal-Catalyzed Electrophilic Amination of Organozinc Reagents

Sep. 5th

5P-026s Ho Jea

Kim

Kangwon University

republic ofkorea

Simple magnesium catalyzed hydroboration of various carbonyl compounds

Sep. 5th

5P-027s Whee

Hong

Kangwon University

republic ofkorea

A new one pot synthesis of ester to α,β-unsaturated esters from esters

Sep. 5th

5P-028s Seong

Choi

Kangwon University

republic of
korea

Catalyst and solvent-free hydroboration of alkynes

Sep. 5th

5P-029s Jaeeun

Yi

Kangwon University

republic of
korea

Partial reduction of isopropyl esters to aldehydes using MeLi catalyzed hydroboration

Sep. 5th

5P-030

Hyeon
Hiroyuki

Yamakoshi

Nagoya City University

Japan

Formal Synthesis of (±)-Morphine via Tandem Oxidation/Cycloaddition Sequence

Sep. 5th

5P-031s Eunjoon

Park

Korea University

South
Korea

Total syntheses of (±)- and (+)-Goniomitine

Sep. 5th

5P-032

Sugai

Keio University

Japan

The Utilization of Enzyme-mediated Acylation and De-acylation in the Transformation of
Heterocycles

Sep. 5th

5P-033s Hao

Hu

RIKEN, CSRSJapan

A Self-Assembled Polymeric Pyridine Copper Catalyst for the Huisgen Cycloaddition of
Alkynes and Acetylene Gas: Application in Synthesis of Tazobactam

Sep. 5th

5P-034

YoshidaMeijo University

Japan

Development of oxidative N-N coupling reaction of carbazole alkaloids by using NaOCl・
5H2O

Sep. 5th

5P-035s Mayu

Hirashima

Mukogawa Women's
University

Japan

Synthesis of optically active pharmaceuticals by using recyclable catalytic asymmetrictransfer hydrogenation in ionic liquid

Sep. 5th

5P-036s Ryo

Sekizawa

Kanazawa University

Japan

Synthesis of 15E-anti Phytochrome Chromophore Derivatives

Sep. 5th

5P-037s Shohei

KasanoChiba University

Japan

Synthesis of 3-Allylindole Derivatives Using Palladium Catalyst with P,Olefin Type Ligand

Sep. 5th

5P-038s Hiroto

Uno

Nagoya Institute ofTechnology

Japan

Synthesis of Trifluoromethyl Nine-Membered Heterocycles via a Double Decarboxylative
Ring-Expansion under Palladium Catalysis

Sep. 5th

5P-039s Yuta

Onuki

University of Toyama

Japan

Ring-Opening Cyclization of Spirocyclopropanes with Sulfonium Ylides for theConstruction of a Chromane Skeleton

Sep. 5th

5P-040s Kunihiro

Matsumura

Osaka City University

Japan

Total Synthesis of Histrionicotoxin 235A

Sep. 5th

5P-041s Ryo

TanifujiTokyo University of Agriculture Japanand Technology

Chemo–enzymatic total synthesis of tetrahydroisoquinoline alkaloids exhibiting potent DNA
alkylating ability

Sep. 5th

5P-042s Yuan

Jin

Nagoya University

Synthetic Studies on Haliclonin A

Sep. 5th

5P-043s Daniel

Payne

National Institute for Materials Japan
Science (NIMS)

Non-planar Porphyrinoids as Asymmetric Bifunctional Hydrogen-Bond Donor Catalysts

Sep. 5th

5P-044s Takahiro

Watanabe

The University of Tokyo

Japan

Synthetic Study of TPI 287

Sep. 5th

5P-045s Shinsuke

Shimizu

The University of TokyoJapan

Total Syntheses of Bufadienolides

Sep. 5th

5P-046s Ryuichi

MurataKyoto University

Japan

Desymmetrization of gem-Diols via Enantio- and Diastereoselective Cycloetherification
Using Bifunctional Organocatalysts

Sep. 5th

5P-047s Fabian

Hogenkamp

Heinrich Heine University

Germany

Heterocyclic Photocages for Carbohydrates

Sep. 5th

5P-048s Mako

TamuraToho University

Japan

Synthetic Study on Zinc(II) Complexes of 3-Hydroxy-5-(p-substituted)phenylthiazole-2(3H)thiones toward the Development of New Antidiabetic Agents

Sep. 5th

5P-049s Lucie

Cechova

IOCB Prague

Czech
Republic

5Phenylazopyrimidines: A new class of orthogonal photoswitches?

Sep. 5th

5P-050s Jun

ShimuraTokyo Institute of Technology Japan

Total Synthesis of Saptomycin H

Sep. 5th

5P-051s Keigo

Higashida

Osaka University

Japan

Chiral Vanadium Complex-catalyzed Enantioselective Oxidative Hetero-coupling
Reactions of Arenols

Sep. 5th

5P-052s Takuya

Jinnouchi

Okayama University

Japan

Studies on the Total Synthesis of Hamigeran B

Sep. 5th

5P-053

MiyakeOsaka University

Japan

In situ click reaction activated by a metal ion in targeted proteins: Identification of a triazole
compound as a lysine demethylase 5C inhibitor

KeitaroHiroyoshi

Chang

Takeshi

Keisuke

Yuka

T.

Japan

Sep. 5th

5P-054s Naoki

Matsuyama

Osaka University

Japan

Facile Synthesis of Chiral Spirooxindoles via Pictet-Spengler/Oxidative Rearrangement

Sep. 5th

5P-055s Hibiki

KomineOsaka University

Japan

Synthesis and evaluation of novel artificial nucleic acid having an oxanorbornane skeleton

Stockholm University

SwedenRegiospecific N-Arylation of Aliphatic Amines under Mild and Metal-Free Reaction
Conditions

Sep. 5thcancelled

Sep. 5th

5P-057s Gabriella

M. Kervefors

Sep. 5th

5P-058s Takayuki

Sakai

Kyoto University

Japan

Promoting accumulation of curvature-inducing peptides on cell membranes

Sep. 5th

5P-059s Saki

WatanabeRitsumeikan University

Japan

Synthetic Study of Pyridone-embedded Analogs of Cortistatin A

Sep. 5th

5P-060s Koki

Fujimoto

Ritsumeikan University

Japan

Synthesis and Evaluation of Novel Analogs of Arenastain A

Sep. 5th

5P-061s Perumalsamy

Parasuraman

Muroran Institute ofTechnology

Japanβ-Amino Alcohol Organocatalyst for Asymmetric Hetero Diels-Alder Reaction of Isatinswith Enones

Sep. 5th

5P-062s Divakar

GanesanMuroran Institute ofTechnology

Japan

Xylofuranose Based γ-Amino Alcohol Organocatalysts for Asymmetric Michael Addition of
β-Keto Esters with Nitro Olefins

Sep. 5th

5P-063s Ryota

Nakahashi

Kwansei Gakuin University

Japan

Synthesis and Property of Propeller-Shaped Isoacenoheteroles

Sep. 5th

5P-064

Higashi

Kyoto University

Japan

Theoretical Analysis of Water Effect on a Stereoselective Fluorination Reaction

Sep. 5th

5P-065s Yusuke

Miyashita

Waseda University

Japan

Asymmetric Catalysis of Racemization-Free Planar-Chiral Pyridinophanes Including
Hemiacetal and Acetal SkeletonsSep. 5th

5P-066s Tsuyoshi

MasudaWaseda University

Japan

Highly Efficient Asymmetric Total Synthesis of (–)-Dehydro-exo-Brevicomin via
Photoisomerization-Acetalization Strategy

Sep. 5th

5P-067s Kotaro

Nishiyama

Sophia University

Japan

Synthesis and Structure-Activity Relationship Study of 1-(4-Methoxyphenyl)-1-(quinazolin4-yl)ethanols as Anticancer Agent

Sep. 5th

5P-068

Vorob'ev

RussianFederation

Cycloaddition of alkynes and nitriles to heterocyclic N-imines as a tool for functionalized
pyrazolo[1,5-a]pyridines and 1,2,4-triazolo[1,5-a]pyridines synthesis

Sep. 5th

5P-069s Kiyoteru

Niina

Novosibirsk State University,
Novosibirsk Institute ofOrganic
Chemistry
Nagoya Institute
of

Japan

Reaction of (Hetero)aryl Tetrafluoro-λ6-Sulfanyl Chlorides with Alkynes and Alkenes under
Visible Light

Sep. 5th

5P-070

Shigeki

SasakiKyushu University

Japan

Simultaneous binding of Chromomycin A3 to the CGG repeat of DNA

Sep. 5th

5P-071

Takumichi

Sugihara

Niigata University of Pharmacy Japanand Applied Life Sciences

Reaction of 2-Phenylbenzo[1,3,2]dioxaboridines with Various Oxidants

Sep. 5th

5P-072s Ryutaro

Kondo

Nagoya University

Japan

IBS-catalyzed Highly Efficient and Selective Oxidation of Alcohols with Oxone

Sep. 5th

5P-073

Yoshimatsu

Gifu University

Japan

Synthesis of Azepino[1,2-a]indoles by the [6+1] Annulation Reaction of Ynenitriles

Sep. 5th

5P-074s Hirotaka

Sasa

Ritsumeikan University

Japanµ-Oxo Hypevalent Iodine(III)-Catalyzed Oxidative Aryl Amination for Synthesis of NHeterocycles

Sep. 5th

5P-075s Junichi

Taguchi

Kyoto University

Japan

Synthetic Study of Aspidophylline A Based on Gold(I)-Catalyzed Cascade Cyclization

Sep. 5th

5P-076s Takahiro

Kawajiri

Gifu Pharmaceutical University Japan

Chemoselective Nucleophilic Functionalizations of Aromatic Aldehydes / Acetals via
Pyridinium Salt Intermediates

Sep. 5th

5P-077s Haruka

TakeuchiKyoto University

Japan

Approach to Spirocyclohexadiene through Visible Light-Mediated ipso Cyclization of
Biaryls

Sep. 5th

5P-078s Junpei

Matsuoka

Kyoto University

Japan

Total Synthesis of Dictyodendrins by the Gold-Catalyzed Cascade Cyclization of
Conjugated Diynes with Pyrroles

Sep. 5th

5P-079

Ouchi

University of Shizuoka

Japan

Synthetic Study of Fairy Chemicals

Sep. 5th

5P-080s Kengo

KasamaOsaka University

Japan

A Biocatalytic Highly Enantioselective Synthesis of Axially Chiral Bihydroxycarbazoles

Sep. 5th

5P-081

Kamikawa

Osaka Prefecture University

Japan

Planar-Chiral Phosphine-Olefin Ligands Exploiting a (Cyclopentadienyl)manganese(I)Scaffold: Application in Asymmetric Catalysis

Sep. 5th

5P-082s Keina

Komiyama

Ritsumeikan University

Japan

Benzylic Oxidation and C-H Functionalization of Xanthenes using Hypervalent Iodine(III)Reagents

Sep. 5th

5P-083s Yukiya

Sato

Kanazawa University

Japan

Tertiary Alkylations of Aldehydes, Ketones, or Imines Using Organoboronates and Base
Catalyst

Sep. 5th

5P-084s Yoshito

Takahashi

Keio University

Japan

An Iridium-Catalyzed Reductive Nucleophilic Addition to Amidea

Sep. 5th

5P-085s Yuki

KanekoOsaka University

Japan

N2-Selective Alkylation of Benzotriazoles via Cobalt Catalyzed Hydroamination Reaction of
Non-Activated Olefins

Sep. 5th

5P-086s Daisuke

SatoTokyo University of Agriculture Japanand Technology

Nonmetal-Catalyzed Skeletal Reorganization of 7-En-2-ynones into 3Alkylidenecyclohexenes

Sep. 5th

5P-087

Takashi

Nishiyama

Fukuyama University

Japan

Synthesis of 4-Aroyl-5-arylpyrazoles and 4-Aroyl-3-arylpyrazoles via the Reaction of
Enaminodiketones with Substituted Hydradines

Sep. 5th

5P-088Tohru

Kamitanaka

Ritsumeikan University

Japan

Synthetic Strategy for Highly Substituted Indoles based on Regioselective Coupling ofIminoquinone Monoacetals

Sep. 5th

5P-089s Hiroto

SagaraUniversity of Shizuoka

Japan

Synthetic study of silybins

Sep. 5th

5P-090MORIMOTO

Ritsumeikan University

Japan

Hypervalent Iodine(III) Induced Oxidative Cross-Coupling of Phenols

Sep. 5th

5P-091s Toshitaka

Shoji

Ritsumeikan university

Japan

Efficient N-Arylation of Azole Compounds utilizing Designer TMP-Iodonium(III) Salts

Sep. 5th

5P-092s Takumi

Ikeda

Ritsumeikan University

Japan

N-Glycosylation Reaction of Thioglycoside using Hypervalent Iodine(III) Reagent

Sep. 5th

5P-093s Ibuki

Odaka

Ritsumeikan University

Japan

Glucuronidation Reaction Using Odorless Thio-glycoside and Hypervalent Iodine Reagent

Sep. 5th

5P-094s Joan

Ondevilla

Osaka University

Japan

Membrane and Cholesterol Interactions of the Diosgenyl Saponins

Morikawa

Kindai University

Japan

Limonoids from Andiroba (Carapa guianensis) Improve Glucose and Lipid Metabolism in
Hepatocytes

HoriOsaka University

Japan

Synthetic study of the furanosteroid, viridin

Masahiro

Aleksey

Mitsuhiro

HitoshiKen

KOJI

CandiceToshioSep. 5th

5P-095

Sep. 5th

5P-096s Shuhei

V.

Technology

Sep. 5th

5P-097

Masakazu

Kobayashi

Kobayashi PharmaceuticalCo., Ltd.

Japan

Neokotalanol, a Principal Thiosugar Sulfonium Constituent in Salacia chinensis,
Suppresses HbA1c Levels in Genetically Obese-hyperglycemic ob/ob Mice

Sep. 5th

5P-098

Shinsuke

Mizumoto

The University of TokyoJapan

Development of novel acyl-transfer catalysts for protein modification

Sep. 5th

5P-099

Yoshiaki

Manse

Kaminomoto co., ltd.

Japan

Ent-Kaurane Type Diterpenoids from the Aerial Part of Isodon trichocarpus
as Proproliferative Agents on Human Follicle Dermal Papilla Cells

Sep. 5th

5P-100

Akira

Otaka

Tokushima Unmiversity

Japan

Copper-mediated Ring Opening of Thiazolidine Derivative for Protein Chemical Synthesis

Sep. 5th

5P-101s Ahmed

Osaka University

Japan

Regioselective Dienone-phenol Rearrangement of 4,4-Disubstituted 2-Hydroxycyclohexa2,5-dienones into 3,4-Disubstituted Catechols

Sep. 5th

5P-102s Ryoya

Sep. 5th

5P-103s Yamato

Sep. 5th

AbuBakr

M. Ibrahim
S.
Takakura

Gifu Pharmaceutical University Japan

Platinum on carbon-catalyzed aqueous oxidative lactonization of diols using molecularoxygenKanzaki

The University of TokyoJapan

One-Pot Incorporation of Nucleophiles to Cyclic Hemiacetal Aldols: Ring Opening Strategy
Prompted by Amine Pendant Boronic Acid

5P-104s Kentarou

Sakamoto

Institute for Chemical
Research, Kyoto University

Japan

Improvement of Peptide-Mediated Cytosolic Delivery of Macromolecules

Sep. 5th

5P-105s Kota

Koike

Gifu Pharmaceutical University Japan

Structural Modification and Biological Evaluation of Quinomycin Antibiotics Focusing on
Cross-bridge Structures of Bicyclic Depsipeptide

Sep. 5th

5P-106s Yoshinori

MakitaChiba University

Japan

Synthesis and Evaluation of Heterocyclic Rocaglamide Derivatives with Wnt Signaling
Inhibition

Sep. 5th

5P-107AsaharaOsaka University

Japan

Photooxygenation of Aromatic Substrates using Azafluorenone Derivatives as
Photocatalysts

Sep. 5th

5P-108s Kishin

InuiToyama University

Japan

Design and synthesis of novel transthyretin amyloidogenesis inhibitors

Sep. 5th

5P-109s Tomohiro

Tsutsumi

Tokushima University

Japan

A Concise Asymmetric Total Synthesis of (+)-Epilupinine

Sep. 5th

5P-110s Katsuki

Takashima

Toyama university

Japan

Stereodivergent asymmetric synthesis of DHQ-type poison-frog alkaloids for SAR study toinhibitory effect of nicotinic acetylcholine receptors

Sep. 5th

5P-111s Amaechi

Odoh

Tohoku University

Japan

Access to trisubstituted piperidines using an organocatalyst-mediated asymmetricconjugate addition of aldehydes and β-substituted-α-cyano ethyl acrylates as a key step

Sep. 5th

5P-112s Tomoki

Niwa

University of Shizuoka

Japan

Dianionic phase transfer catalyst for asymmetric fluorofunctionalizations

Sep. 5th

5P-113s Ryuji

Kouda

Hokkaido University

Japan

Synthetic Studies on Iridoids: Construction of a cis-Fused Cyclopenta[c]pyran Ring via
Pauson-Khand Reaction

Sep. 5th

5P-114

Creencia

MSU-Iligan Institute ofTechnology

Philippines

Synthesis of Quinolines via Friedlander Reaction under One-pot-one-step, Solvent-free,
Microwave-assisted Conditions

Sep. 5th

5P-115s Yusuke

TsunodaRitsumeikan University

Japan

Dihydrobenzofuran Synthesis by [3+2] Coupling of Quinone Monoacetals with Vinyl Ethers

Sep. 5th

5P-116s Riho

Korogi

Nagasaki University

Japan

Pd-Catalyzed Asymmetric Allylic Alkylation of Tryptamine for Construction of Pyrroloindole
Alkaloids

Sep. 5th

5P-117

HuebschBayer AG, Medicinal
Chemistry, Wuppertal

Germany

The Specific Reactivity of Pyrrolo[2,1-f][1,2,4]triazines
and the Synthesis of Rogaratinib (BAY 1163877)

Sep. 5th

5P-118s Madoka

Waku

Okayama University

Japan

The Tandem Cyclization Reaction to Form Heteroatoms-Containing Tetracyclic
Compounds

Sep. 5th

5P-119s Yusuke

Ueda

Tohoku University

Japan

Total Synthesis of (–)-Emestrin H and (–)-Asteroxepin.

Sep. 5th

5P-120s Eisaku

OhashiTokushima university

Japan

Studies on the Second Generation Synthesis of Palau’amine

Sep. 5th

5P-121s Ryuji

Kyan

Shizuoka University

Japan

N-Aryl Effect on the Enhanced Catalytic Activity of Imidazolium-Salt Derived NHCs

Sep. 5th

5P-122s Shu

Takahashi

Kitasato University

Japan

Asymmetric Total Synthesis of Diatretol, A Potent Antimalarial Agent

Sep. 5th

5P-123s Keisuke

Aoki

Kyoto University

Japan

Synthetic Study of TIGIT Protein for Mirror-Image Screening

Sep. 5th

5P-124s Bimolendu

DasOsaka University

Japan

ANP77: A Three-carbon Atom Linked 2-Amino-1,8-naphthyridine Dimer that Recognizes
Cytosine Rich Bulge-mismatched Sequences of Duplex DNA and RNA

Sep. 5th

5P-125s Akito

Heguri

Osaka University

Japan

Synthesis of Helicenes Using Diels–Alder Reactions of Fused Benzynes with Furans

Sep. 5th

5P-126s Seiya

Hiranaka

Kansai University

Japan

Drug discovery of pyrilamine derivatives as blood-brain-barrier permeable histone
deacetylase inhibitors.

Sep. 5th

5P-127

Asakawa

Tokai university

Japan

Total Synthesis of Sophoraflavanone H

Sep. 5th

5P-128s Saki

Imai

Shizuoka University

Japan

Sep. 5th

5P-129

YamadaGifu Pharmaceutical University Japan

One-Pot Synthesis of Highly Functionalized 2-Chloroaziridines for Stereoselective
Synthesis of (Z)-Chloroalkene Dipeptide Isosteres Containing alpha,alpha-Disubstituted
Amino
Acids
Gold-Catalyzed
Indenone Synthesis from 2-Alkynylaldehyde Cyclic Acetal

Sep. 5th

5P-130s Satoko

Akiyama

Hokkaido University

Japan

Genome mining of hydrazine-forming machinery identified novel natural productswith unique dihydropyridazinone rings

Sep. 5th

5P-131s Jan

SkácelIOCB PragueČeskoDesign and Synthesis of Inhibitors of Enzymes of Purine Metabolism – Application of
Direct Metalation of Heterocycles

Sep. 5th

5P-132s Hideyasu

China

Ritsumeikan University

Japan

Functionalized Lactone Formations on the Basis of Halogen-Controlled Rapid Cyclizationof Haloketo Acids under Mild Conditions

Sep. 5th

5P-133

TakuyaOkada

University of Toyama

Japan

Synthetic Studies Towards Broussonetine N

Sep. 5th

5P-134s Hirotaka

SuzukiTohoku University

Japan

Development of an efficient synthetic method for α-methylene γ-butyrolactone skeleton
and its application to total synthesis of arglabin and ludartin

Sep. 5th

5P-135s Ryo

Hirokawa

University of Shizuoka

Japan

Parallel Kinetic Resolution of Various rac-Allylic Amides via Asymmetric Bromocyclization

Sep. 5th

5P-136s Takuto

Koide

Kogakuin University

Japan

Synthetic studies on GPR35 agonist without species-specificity

Sep. 5th

5P-137Masahiro

Yamanaka

Rikkyo University

Japan

Rational design of bis-2-aminothiazoline as a new chiral scaffold beyond bisoxazoline

Sep. 5th

5P-138

Nobuhiro

Kanomata

Waseda University

Japan

Parapyrazinophane - An Intrinsically Chiral Diazine-cyclophane and the Kinetics of Its
Racemization

Sep. 5th

5P-139s Yuto

Emi

Osaka University

Japan

Synthetic Study of Aloin through Regioselective Diels-Alder Reactions of Benzaines

Haruyasu

EvelynWalterTomohiro

TsuyoshiS.

C.

Sep. 5th

5P-140Sep. 5th

YamadaTokushima University

Japan

The Enhancement of Enantio-recognition in Kinetic Resolution of Chiral Secondary
Alcohols with Chiral Acyltriazolium by Formation of Alcohol–Carboxylate Complexes

5P-141s Masaki

Kawabata

Osaka University

Japan

Regioslective Synthesis of Fused Heterocycles Using 2-Silyl-3,4-Pyridyne

Sep. 5th

5P-142

Akira

TakagiKobe Pharmaceutical
University

Japan

Development of Drugs for Modulating Endoplasmic Reticulum Stress Response

Sep. 5th

5P-143

AlexeyFesta

Peoples' Friendship University Russia
of Russia

Transformations of N-(allenyl)indoles: syntheses of pyrazino[1,2-a]indoles andvinylsulfones

Sep. 5th

5P-144

FrederickLuzzioUniversity of Louisville

Nucleoside Antibiotic Support Studies: Uridine-Based Homologation Strategies Using the
Nitroaldol ApproachKen-ichiA.

USA