RESTRICTED  
  
G/MA/TAR/RS/457  
23 mars 2017 
(17-1617) Page: 1/31 
Comité de l'accès aux marchés  Original:  anglais  
 
  RECTIFICATIONS ET MO DIFICATIONS DES LIST ES 
LISTE XIV – NORVÈGE  
La communication ci -après, datée du  13 mars 2017, est distribuée à la demande de la délégation 
de la Norvège.  
 
_______________  
 
 
Conformément au quatrième réexamen de l'Accord sur le commerce d es produits pharmaceutiques 
(G/MA/W/102) et à la Décision du 2 6 mars 1980 ( IBDD S27/26) , la Norvège communique  son 
projet de modifications de la Liste XIV . Ces modifications sont entrées en vigueur le 
1er janvier  2011. Les documents1 communiqués sont les s uivants:  
− Annexe I  Liste des dénominations communes internationales;  
− Annexe II  Liste des préfixes et suffixes des sels, esters et hydrates de la DCI ; 
− Annexe II I  Liste consolidée de s produits intermédiaires ; 
− Annexe IV  Liste des produits  pharmaceutiques inte rmédiaires . 
 
_______________  
 
 
Si aucune objection n'est notifiée au Secrétariat dans un délai de trois mois à compter de la date 
du présent document, les rectifications et modifications apportées à la Liste  XIV – Norvège seront 
considérées comme approuvée s et seront officiellement certifiées.  
                                                
1 En anglais seulement.  G/MA/TAR/RS/457  
- 2 - 
  ANNEX I  
List of international non -proprietary names (INNs) to be added to the list of products 
receiving duty -free treatment included in Annex 3 to Annex I to Regulation (EEC) 
No 2658/87  
 
 
CN code  CAS RN  Name  
2842 9 0 80 119175 -48-3 fermagate  
2843 90 90  759457 -82-4 padeliporfin  
2844 40 30  123748 -56-1 iodofiltic acid (123I)  
2904 10 00  21668 -77-9 eprodisate  
2906 19 00  199798 -84-0 elocalcitol  
2909 30 90  24150 -24-1 terameprocol  
2916 19 95  81485 -25-8 peretinoin   
2916 39 00  51543 -40-9 tarenflurbil  
2918 19 98  174022 -42-5 bevirimat  
2919 90 00  258516 -89-1 fospropofol  
2920 90 85  163133 -43-5 naproxcinod  
2921 19 99  3687-18-1 tramiprosate  
2922 19 85  68392 -35-8 afimoxifene  
2922 19 85  753449 -67-1 ronacaleret  
2922 29 00  433265 -65-7 faxeladol  
2922 50 00  121524 -08-1 amibegron  
2922 50 00  329773 -35-5 cinaciguat  
2922 50 00  643094 -49-9 fasobegron  
2923 10 00  856676 -23-8 choline fenofibrate  
2924 29 98  847353 -30-4 arbaclofen placarbil  
2924 29 98  194785 -19-8 bedoradrine  
2924 29 98  194085 -75-1 carisbamate  
2924 29 98  254750 -02-2 emricasan  
2924 29 98  355129 -15-6 eprotirome  
2924 29 98  402567 -16-2 firategrast  
2924 29 98  478296 -72-9 gabapentin enacarbil  
2924 29 98  15866 -90-7 incyclinide  
2924 29 98  202844-10-8 indantadol  
2924 29 98  96847 -55-1 levomilnacipran  
2924 29 98  608137 -32-2 lisdexamfetamine  
2924 29 98  652990 -07-3 milveterol  
2924 29 98  181816 -48-8 ombrabulin  
2924 29 98  289656 -45-7 senicapoc  
2925 19 95  19171 -19-8 pomalidomide  
2928 00 90 22033 -87-0 olesoxime  
2928 00 90  2675-35-6 sivifene  
2928 00 90  816458 -31-8 tecovirimat  
2928 00 90  238750 -77-1 tosedostat  G/MA/TAR/RS/457  
- 3 - 
  CN code  CAS RN  Name  
2928 00 90  149647 -78-9 vorinostat  
2929 90 00  31645 -39-3 palifosfamide  
2930 90 99  608141 -41-9 apremilast  
2930 90 99  216167-92-9 camobucol  
2930 90 99  211513 -37-0 dalcetrapib  
2930 90 99  69819 -86-9 darinaparsin  
2930 90 99  488832 -69-5 elesclomol  
2930 90 99  216167 -95-2 elsibucol  
2930 90 99  168682 -53-9 ezatiostat  
2930 90 99  58569 -55-4 metenkefalin  
2930 90 99  887148 -69-8 monepantel  
2930 90 99  603139 -19-1 odanacatib  
2930 90 99  162520 -00-5 salirasib  
2930 90 99  216167 -82-7 succinobucol  
2930 90 99  125961 -82-2 tipelukast  
2931 00 99  125973 -56-0 amsilarotene  
2932 19 00  253128 -41-5 eribulin  
2932 19 00  186953 -56-0 pafuramidine  
2932 29 85  195883 -06-8 omtriptolide  
2932 99 00  664338 -39-0 arterolane  
2932 99 00  183133 -96-2 cabazitaxel  
2932 99 00  401925 -43-7 celivarone  
2932 99 00  461432 -26-8 dapagliflozin  
2932 99 00  118457 -15-1 dexnebivolol  
2932 99 00  156294-36-9 larotaxel  
2932 99 00  118457 -16-2 levonebivolol  
2932 99 00  83461 -56-7 mifamurtide  
2932 99 00  117570 -53-3 vadimezan  
2933 19 90  496775 -61-2 eltrombopag  
2933 19 90  206884 -98-2 niraxostat  
2933 19 90  410528 -02-8 palovarotene  
2933 19 90  376592-42-6 totrombopag  
2933 29 90  183659 -72-5 catramilast  
2933 29 90  944263 -65-4 demiditraz  
2933 29 90  867153 -61-5 dulanermin  
2933 29 90  320367 -13-3 lixisenatide  
2933 29 90  698389 -00-3 rolipoltide  
2933 29 90  697766 -75-9 velafermin  
2933 39 99  147084-10-4 alcaftadine  
2933 39 99  54-96-6 amifampridine  
2933 39 99  249921 -19-5 anamorelin  
2933 39 99  319460 -85-0 axitinib  
2933 39 99  208110 -64-9 befiradol  
2933 39 99  330942 -05-7 betrixaban  G/MA/TAR/RS/457  
- 4 - 
  CN code  CAS RN  Name  
2933 39 99  201034 -75-5 daporinad  
2933 39 99  209783 -80-2 entinostat  
2933 39 99  412950 -27-7 goxalapladib  
2933 39 99  218791 -21-0 imisopasem manganese  
2933 39 99  103129 -82-4 levamlodipine  
2933 39 99  154357 -42-3 levonadifloxacin  
2933 39 99  108147 -54-2 migalastat  
2933 39 99  453562 -69-1 motesanib  
2933 39 99  139145 -27-0 parogrelil  
2933 39 99  459856 -18-9 pexacerfont  
2933 39 99  706779 -91-1 pimavanserin  
2933 39 99  362665 -56-3 pitolisant  
2933 39 99  861151 -12-4 rosonabant  
2933 39 99  701977 -09-5 taranabant  
2933 39 99  189950 -11-6 tropantiol  
2933 39  99 793655 -64-8 vapitadine  
2933 39 99  139290 -65-6 volinaserin  
2933 49 90  141388 -76-3 besifloxacin  
2933 49 90  697761 -98-1 elvitegravir  
2933 49 90  185055 -67-8 ferroquine  
2933 49 90  445041 -75-8 intiquinatine  
2933 49 90  378746 -64-6 nemonoxacin  
 2933 49 90  245765 -41-7 ozenoxacin  
2933 49 90  412950 -08-4 rilapladib  
2933 49 90  871224 -64-5 almorexant  
2933 49 90  863029 -99-6 balamapimod  
2933 49 90  698387 -09-6 neratinib  
2933 49 90  154652 -83-2 tezampanel  
2933 49 90  128253 -31-6 veliflapon  
2933 59 95  791828 -58-5 aderbasib  
2933 59 95  840486 -93-3 adipiplon  
2933 59 95  850649 -61-5 alogliptin  
2933 59 95  859212 -16-1 bafetinib  
2933 59 95  380843 -75-4 bosutinib  
2933 59 95  839712 -12-8 cariprazine  
2933 59 95  414910 -27-3 casopitant  
2933 59 95  288383-20-0 cediranib  
2933 59 95  849550 -05-6 cevipabulin  
2933 59 95  827318 -97-8 danusertib  
2933 59 95  356057 -34-6 darapladib  
2933 59 95  501000 -36-8 dutacatib  
2933 59 95  247257 -48-3 fimasartan  
2933 59 95  3432-99-3 folitixorin  
2933 59 95  668270 -12-0 linagliptin  G/MA/TAR/RS/457  
- 5 - 
  CN code  CAS RN  Name  
2933 59 95  441798 -33-0 macitentan  
2933 59 95  641571 -10-0 nilotinib  
2933 59 95  763113 -22-0 olaparib  
2933 59 95  686344 -29-6 otenabant  
2933 59 95  625115 -55-1 riociguat  
2933 59 95  486460 -32-6 sitagliptin  
2933 59 95  425637 -18-9 sotrastaurin  
2933 59 95  309913 -83-5 talmapimod  
2933 59 95  113857 -87-7 talotrexin  
2933 59 95  274693 -27-5 ticagrelor  
2933 59 95  306296 -47-9 vicriviroc  
2933 69 80  775351 -65-0 imeglimin  
2933 79 00  461443 -59-4 aplaviroc  
2933 79 00  189691 -06-3 bremela notide  
2933 79 00  813452 -18-5 carmegliptin  
2933 79 00  405169 -16-6 dovitinib  
2933 79 00  536748 -46-6 eribaxaban  
2933 79 00  473289 -62-2 ilepatril  
2933 79 00  180694 -97-7 mimopezil  
2933 79 00  579475 -18-6 orvepitant  
2933 79 00  449811 -01-2 pamapimod   
2933 79 00  248282 -01-1 paquinimod  
2933 79 00  380917 -97-5 perampanel  
2933 79 00  552292 -08-7 rolapitant  
2933 79 00  425386 -60-3 semagacestat  
2933 79 00  515814 -01-4 voclosporin  
2933 99 80  481629 -87-2 aleplasinin  
2933 99 80  394730 -60-0 boceprevir   
2933 99 80  649735 -63-7 brivanib alaninate  
2933 99 80  483369 -58-0 denagliptin  
2933 99 80  284019 -34-7 denibulin  
2933 99 80  481631 -45-2 diaplasinin  
2933 99 80  272105 -42-7 disitertide  
2933 99 80  227318 -71-0 epetirimod  
2933 99 80  259793 -96-9 favipiravir  
2933 99 80  871576 -03-3 flovagatran  
2933 99 80  229305 -39-9 golotimod  
2933 99 80  258818 -34-7 larazotide  
2933 99 80  571170 -77-9 laropiprant  
2933 99 80  616202 -92-7 lorcaserin  
2933 99 80  868771 -57-7 melogliptin  
2933 99 80  803712 -67-6 obato clax  
2933 99 80  404950 -80-7 panobinostat  
2933 99 80  625114 -41-2 piragliatin  G/MA/TAR/RS/457  
- 6 - 
  CN code  CAS RN  Name  
2933 99 80  74847 -35-1 pyronaridine  
2933 99 80  872178 -65-9 rabeximod  
2933 99 80  355151 -12-1 rotigaptide  
2933 99 80  497221 -38-2 rusalatide  
2933 99 80  187602 -11-5 sofiga tran  
2933 99 80  227318 -75-4 sotirimod  
2933 99 80  402957 -28-2 telaprevir  
2933 99 80  848084 -83-3 tigapotide  
2933 99 80  393105 -53-8 tiplasinin  
2933 99 80  620948 -93-8 vabicaserin  
2933 99 80  794466 -70-9 vernakalant  
2934 10 00  544417 -40-5 capadenos on 
2934 10 00  302962 -49-8 dasatinib  
2934 10 00  223132 -37-4 inolitazone  
2934 10 00  241479 -67-4 isavuconazole  
2934 10 00  338990 -84-4 isavuconazonium chloride  
2934 10 00  607723 -33-1 lobeglitazone  
2934 10 00  280782 -97-0 managlinat dialanetil  
2934 1 0 00 790299 -79-5 masitinib  
2934 10 00  223673 -61-8 mirabegron  
2934 10 00  501948 -05-6 rosabulin  
2934 10 00  447406 -78-2 sodelglitazar  
2934 10 00  760937 -92-6 teneligliptin  
2934 20 80  848344 -36-5 bentamapimod  
2934 20 80  870093 -23-5 talarozole  
2934 99 90  320345 -99-1 aclidinium bromide  
2934 99 90  222551 -17-9 adoprazine  
2934 99 90  207623 -20-9 agatolimod  
2934 99 90  475479 -34-6 aleglitazar  
2934 99 90  870524 -46-2 amolimogene bepiplasmid  
2934 99 90  875446 -37-0 anacetrapib  
2934 99 90  250386 -15-3 apadenoson  
2934 99 90  541550 -19-0 apilimod  
2934 99 90  160707 -69-7 apricitabine  
2934 99 90  147403 -03-0 azilsartan  
2934 99 90  863031 -21-4 azilsartan medoxomil  
2934 99 90  757942 -43-1 bederocin  
2934 99 90  627861 -07-8 beperminogene perplasmid  
2934 99 90  959961 -96-7 bevasiranib  
2934 99 90  769901 -96-4 capeserod  
2934 99 90  868540 -17-4 carfilzomib  
2934 99 90  872847 -66-0 cenersen  
2934 99 90  80295 -38-1 conestat alfa  
2934 99 90  903916 -27-8 custirsen  G/MA/TAR/RS/457  
- 7 - 
  CN code  CAS RN  Name  
2934 99 90  187865 -22-1 derquantel  
2934 9 9 90 134379 -77-4 dexelvucitabine  
2934 99 90  247046 -52-2 dilopetine  
2934 99 90  480449 -70-5 edoxaban  
2934 99 90  188181 -42-2 elacytarabine  
2934 99 90  98819 -76-2 esreboxetine  
2934 99 90  763903 -67-9 fosalvudine tidoxil  
2934 99 90  172673 -20-0 fosapre pitant  
2934 99 90  522664 -63-7 ibodutant  
2934 99 90  405159 -59-3 idrabiotaparinux sodium  
2934 99 90  188116 -07-6 imepitoin  
2934 99 90  335619 -18-6 inakalant  
2934 99 90  1391-36-2 lancovutide  
2934 99 90  189059 -71-0 lapaquistat  
2934 99 90  327026 -93-7 lensiprazine  
2934 99 90  170632 -47-0 lificiguat  
2934 99 90  852313 -25-8 litenimod  
2934 99 90  1000120 -98-8 mipomersen  
2934 99 90  62253 -63-8 nepidermin  
2934 99 90  26833 -87-4 omacetaxine mepesuccinate  
2934 99 90  269718 -84-5 pardoprunox  
2934 99 90  219923 -85-0 pramiconazole  
2934 99 90  377727 -87-2 preladenant  
2934 99 90  524684 -52-4 prinaberel  
2934 99 90  865311 -47-3 quarfloxin  
2934 99 90  869884 -78-6 radezolid  
2934 99 90  496054 -87-6 radiprodil  
2934 99 90  518048 -05-0 raltegravir  
2934 99 90  787548 -03-2 regrelor  
2934 99 90  820957 -38-8 retosiban  
2934 99 90  572924 -54-0 ridaforolimus  
2934 99 90  128517 -07-7 romidepsin  
2934 99 90  93265 -81-7 ropidoxuridine  
2934 99 90  151823 -14-2 sapacitabine  
2934 99 90  379231 -04-6 saracatinib  
2934 99 90  791635 -59-1 simotaxel  
2934 99 90  119567 -79-2 taribavirin  
2934 99 90  332012 -40-5 telatinib  
2934 99 90  925681 -61-4 trabedersen  
2934 99 90  189003 -92-7 trelanserin  
2934 99 90  296251 -72-4 velimogene aliplasmid  
2934 99 90  904302 -98-3 viquidacin  
2934 99 90  872525 -61-6 votucalis  
2934 99 90  221877 -54-9 zotarolimus  G/MA/TAR/RS/457  
- 8 - 
  CN code  CAS RN  Name  
2935 00 90  197904 -84-0 apricoxib  
2935 00 90  769169 -27-9 begacestat  
2935 00 90  414864 -00-9 belinostat  
2935 00 90  313682 -08-5 brecanavir  
2935 00 90  839673 -52-8 cevoglitazar  
2935 00  90 358970 -97-5 drinabant  
2935 00 90  865200 -20-0 giripladib  
2935 00 90  464213 -10-3 ibipinabant  
2935 00 90  173424 -77-6 laromustine  
2935 00 90  398507 -55-6 lodenafil carbonate  
2935 00 90  136564 -68-6 masilukast  
2935 00 90  170569 -88-7 mavacoxib  
2935 00 90  862189 -95-5 mirodenafil  
2935 00 90  439687 -69-1 nelivaptan  
2935 00 90  691852 -58-1 nesbuvir  
2935 00 90  778576 -62-8 oglemilast  
2935 00 90  444731 -52-6 pazopanib  
2935 00 90  362505 -84-8 relacatib  
2935 00 90  243984 -11-4 resatorvid  
2935 00 9 0 519055 -62-0 tasisulam  
2935 00 90  186497 -07-4 zibotentan  
2936 29 00  104121 -92-8 eldecalcitol  
2936 29 00  31690 -09-2 levomefolic acid  
2937 19 00  782500 -75-8 albiglutide  
2937 19 00  348119 -84-6 obinepitide  
2937 19 00  295350 -45-7 ozarelix  
2937 19 00 275371 -94-3 taspoglutide  
2937 19 00  218949 -48-5 tesamorelin  
2937 19 00  22006 -64-0 tridecactide  
2937 22 00  132245 -57-9 dexamethasone cipecilate  
2937 22 00  397864 -44-7 fluticasone furoate  
2937 29 00  211254 -73-8 lonaprisan  
2937 50 00  333963 -42-1 cobiprostone  
2937 50 00  172740 -14-6 posaraprost  
2937 90 00  834153 -87-6 elagolix  
2937 90 00  609799 -22-6 tasimelteon  
2937 90 00  342577 -38-2 velneperit  
2939 19 00  73232 -52-7 methylnaltrexone bromide  
2939 59 00  136199 -02-5 rolofylline  
2939 99 00  850607 -58-8 darotropium bromide  
2939 99 00  187852 -63-7 delimotecan  
2940 00 00  9007-72-1 ferric carboxymaltose  
2940 00 00  442201 -24-3 remogliflozin etabonate  
2940 00 00  408504 -26-7 sergliflozin etabonate  G/MA/TAR/RS/457  
- 9 - 
  CN code  CAS RN  Name  
2941 90 00  467214 -20-6 alvespimycin  
2941 90 00  677017 -23-1 berubicin  
2941 90 00  229016 -73-3 ceftaroline fosamil  
2941 90 00  318498 -76-9 flopristin  
2941 90 00  145435 -72-9 gamithromycin  
2941 90 00  325965 -23-9 linopristin  
2941 90 00  857402 -23-4 retaspimycin  
2941 90 00  305841 -29-6 sagopilone  
2941 90 00  75747 -14-7 tanespimycin  
2941 90 00  328898 -40-4 tildipirosin  
2941 90 00  222400 -20-6 tomopenem  
2941 90 00  63409 -12-1 tylvalosin  
3001 90 91  9041-08-1 semuloparin sodium  
3002 10 91  792921 -10-9 abagovomab  
3002 10 91  910649 -32-0 anrukinzum ab  
3002 10 91  648904 -28-3 bavituximab  
3002 10 91  402710 -27-4 
(light chain)  
402710 -25-2 
(heavy chain)  canakinumab  
3002 10 99  945228 -49-9 citatuzumab bogatox  
3002 10 91  880486 -59-9 dacetuzumab  
3002 10 91  615258 -40-7 denosumab  
3002 10 91  762260 -74-2 efungumab  
3002 10 91  89957 -37-9 gantenerumab  
3002 10 91  680188 -33-4 ibalizumab  
3002 10 91  477202 -00-9 ipilimumab  
3002 10 91  640735 -09-7 iratumumab  
3002 10 91  845816 -02-6 lexatumumab  
3002 10 91  903512 -50-5 lucatumumab  
3002 10 91  899796 -83-9 milatuzumab  
3002 10 91  677010 -34-3 motavizumab  
3002 10 91  676258 -98-3 naptumomab estafenatox  
3002 10 91  828933 -51-3 nimotuzumab  
3002 10 91  949142 -50-1 obinutuzumab  
3002 10 91  637334 -45-3 ocrelizumab  
3002 10 91  881191 -44-2 otelixizumab  
3002 10 91 372075 -37-1 sontuzumab  
3002 10 91  705287 -60-1 stamulumab  
3002 10 91  339086 -80-5 tadocizumab  
3002 10 91  592557 -43-2 
(light chain)  
592557 -41-0 
 (heavy chain)  tenatumomab  
3002 10 91  876387 -05-2 teplizumab  
3002 10 91  918127 -53-4 tigatuzumab  G/MA/TAR/RS/457  
- 10 - 
  CN code  CAS RN  Name  
3002 10 91  745013 -59-6 tremelimumab  
3002 10 91  339986 -90-2 tucotuzumab celmoleukin  
3002 10 91  728917 -18-8 veltuzumab  
3002 10 91  896731 -82-1 conatumumab  
3002 10 91  892553 -42-3 etaracizumab  
3002 10 91  944548 -38-3 foravirumab  
3002 10 91  944548 -37-2 rafivirumab  
3002 10 91  880266 -57-9 tanezumab  
3002 10 91  815610 -63-0 ustekinumab  
3002 10 95  862111 -32-8 aflibercept  
3002 10 95  845264 -92-8 atacicept  
3002 10 95  909110 -25-4 baminercept  
3002 10 95  9001-27-8 beroctocog alfa  
3002 10 95  879555 -13-2 epoetin kappa  
3002 10 95  762263 -14-9 epoetin theta  
3002 10 95  501081 -76-1 rilonacept  
3002 10 95  267639 -76-9 romiplostim  
3002 10 95  869858 -13-9 thrombin alfa  
3002 10 95  897936 -89-9 vatreptacog alfa (activated)  
3002 10 95  472960 -22-8 albinterf eron alfa -2b  
3002 10 95  869881 -54-9 briobacept  
3002 10 95  606138 -08-3 catridecacog  
3002 10 95  716840 -32-3 denenicokin  
3002 10 95  931101 -84-7 troplasminogen alfa  
3002 10 99  934216 -54-3 alacizumab pegol  
3002 20 00  181477 -43-0 disomotide  
3002 20 00  181477 -91-8 ovemotide  
3002 20 00  915019 -08-8 tertomotide  
3002 20 00  295371 -00-5 verpasep caltespen  
3002 90 90  473553 -86-5 alferminogene tadenovec  
3002 90 90  929881 -05-0 alipogene tiparvovec  
3002 90 90  600735 -73-7 contusugene ladenovec  
3002 90 90  851199 -59-2 linaclotide  
3002 90 90  898830 -54-1 sitimagene ceradenovec  
3002 90 90  721946 -42-5 transferrin aldifitox  
3507 90 90  9026-00-0 bucelipase alfa  
3507 90 90  885051 -90-1 pegloticase  
3507 90 90  884604 -91-5 velaglucerase alfa  
3911 90 99  892497 -01-7 azoximer bromide  
 
 G/MA/TAR/RS/457  
- 11 - 
  ANNEX II  
List of prefixes and suffixes which, in combination with the INNs of Annex 3 to Annex I 
to Regulation (EEC) No 2658/87, describe the salts, esters or hydrates of INNs; these 
salts, esters and hydrates are free of duty, on condition that they are classifiable in the 
same six -digit HS subheading as the corresponding INN  
 
The references to "International Nonproprietary Names (INN) for pharmaceutical substances, 
Names for radicals & groups, comprehensive list 2004" are  replaced by "International 
Nonproprietary Names (INN) for pharmaceutical substances, Names for radicals, groups & others, 
comprehensive list 2007".  
 
The following prefixes or suffixes are added:  
 
 
Preferred prefix  
or suffix  Synonym  Systematic name  
when d ifferent  
alanetil (INNRG)   [(S)-1-ethoxy -1-oxo-propan -2-
yl]amino (INNCN)  
alaninate (INNRG)   L-alaninate (INNCN)  
alapivoxil (INNRG)   L-alanyl, [(2,2 -
dimethylpropanoyl)oxy]methyl 
(INNCN)  
aldifitox (INNRG)   (4-iminobutane -1,4-
diyl)sulfanediyl[(3RS) -2,5-
dioxopyrrolidine -1,3-diyl]-1,3-
phenylenecarbonyl and forming 
an N-benzoyl derivative of a 
primary amine group of 
diphtheria [550 -L-
phenylalanine]toxin from 
Corynebacterium diphtheriae -
(26-560)-peptide (INNCN)  
besudotox (INNRG)   L-lysyl-L-alanyl -L-
serylglyc ylglycine (linker) fusion 
protein with des -(365-380)-
[Asn364,Val407,Ser515,Gln590,Gln6
06,Arg613]exotoxin A 
(Pseudomonas aeruginosa )-
(251-613)-peptide (toxin with 
region IA and first 16 residues 
of region IB deleted) (INNCN)  
ceribate (INNRG)   rac-2,3-dihyd roxypropyl 
carbonate (ester) (INNCN)  
cipecilate (INNRG)   cyclohexanecarboxylate (ester), 
cyclopropanecarboxylate 
(ester) (INNCN)  
dalanated (INNRG)   des-B30-alanine (INNCN)  
enacarbil (INNRG)   {rac-1-[(2-
methylpropanoyl)oxy]ethoxy}c
arbonyl (INNCN)  G/MA/TAR/RS/457  
- 12 - 
  Preferred prefix  
or suffix  Synonym  Systematic name  
when d ifferent  
estafe natox (INNRG)   glycylglycyl -L-proline (linker) 
fusion protein with enterotoxin 
type A ( Staphylococcus 
aureus )-(1-33)-peptidyl -L-
seryl[Ser36,Ser37,Glu38,Lys39,Ala
41,Thr46,Thr71,Ala72,Ser75,Glu76,
Glu78,Ser80,Ser81,Thr214,Ser217,T
hr219,Ser220,Ser222,Ser224]entero
toxin type E ( Staphylococcus 
aureus )-(32-230)-peptide 
(synthetic superantigen SEA/E -
120) (INNCN)  
etexilate (INNRG)   ethyl, (hexyloxy)carbonyl  
fosamil (INNRG)   phosphono (INNCN)  
glucuronide (INNRG)   β-D-glucopyranosiduronic acid 
[oside] (INNCN)  
medocaril (INNRG)   [(5-methyl -2-oxo-1,3-dioxol -4-
yl)methoxy]carbonyl (INNCN)  
paptox (INNRG)   protein PAP ( Phytolacca 
americana  antiviral) (INNCN)  
placarbil (INNRG)   (R)-2-methyl -1-[(2-
methylpropanoyl)oxy]pro poxy}
carbonyl) (INNCN)  
 G/MA/TAR/RS/457  
- 13 - 
  ANNEX III  
List of pharmaceutical intermediates, i.e. compounds used for the manufacture of 
finished pharmaceutical products, to be added to the list of products receiving duty -free 
treatment included in Annex 6 to Annex I to Regul ation (EEC) No 2658/87  
 
ID CN code  CAS RN  Name  
95 2843 29 00  22199 -08-2 [4-amino -N-(pyrimidin -2(1H) -ylidene -
κN1)benzenesulfonamidato -κO]silver  
428 2905 39 95  281214 -27-5 (2R,3R) -2,3-dimethylbutane -1,4-diyl bis(4 -
methylbenzenesulfonate)  
76 2905 59 98  441002 -17-1 4-chlorobutyl 2 -nitrobenzenesulfonate  
538 2909 30 90  92878 -95-0 2-(3-chloropropoxy) -1-methoxy -4-nitrobenzene  
168 2909 30  503070 -57-3 2-({2-[(6-bromohexyl)oxy]ethoxy}methyl) -1,3-
dichlorobenzene  
386 2909 30  461432 -23-5 4-(5-bromo -2-chlorobenzyl)phenyl ethyl ether  
51 2909 49 80  185954 -75-0 (3R)-3-methoxydecan -1-ol 
167 2909 49 80  85309 -91-7 2-[(2,6-dichlorobenzyl)oxy]ethanol  
64 2909 49 80  160969 -03-9 2-[2-(2,2,2 -trifluoroethoxy)phenoxy]ethyl 
methanesulfonate  
98 2909 50 00  167145 -13-3 2-[2-(3-methoxyphenyl)ethyl]phenol  
377 2910 20 00  15448 -47-2 (2R)-2-methyloxirane  
177 2910 90 00  62600 -71-9 (2R)-2-(3-chlorophenyl)oxirane  
184 2910 90 00  702687 -42-1 (2R)-2-[(5-bromo -2,3-difluorophenoxy)methyl]oxirane  
88 2910 90 00  683276 -64-4 [(2R) -2-methyloxiran -2-yl]methyl 4 -
nitrobenzenesulfonate  
191 2913 00 00  90035 -34-0 4'-(trifluoromethyl)biphenyl -4-carbaldehyd e 
38 2914 40 90  17752 -16-8 (3β)-3-hydroxycholest -5-en-24-one 
244 2914 50 00  974-23-2 (3β,16α)-3-hydroxy -16,17 -epoxypregn -5-en-20-one 
586 2914 70 00  13054 -81-4 4-chloro -heptane -3,5-dione  
236 2914 70 00  10226 -30-9 6-chlorohexan -2-one 
122 2915 60 90  53064 -79-2 iodomethyl pivalate  
426 2915 90 00  22328 -90-1 (3R)-3-methylhexanoic acid  
266 2915 90 00  1069-66-5 sodium 2 -propylpentanoate  
19 2916 20 00  211515 -46-7 1-(2-ethylbutyl)cyclohexanecarbonyl chloride  
32 2916 20 00  381209 -09-2 1-(2-ethylbutyl)cyclohexanecarboxylic acid  
37 2916 20 00  7077-05-6 trans-4-(propan -2-yl)cyclohexanecarboxylic acid  
531 2916 39 00  21900 -39-0 5-fluoro -2-methylbenzoyl chloride  
250 2916 39 00  17625 -03-5 sodium hydrogen 3 -sulfonatobenzoate  
561 2917 19 90  76-72-2 diethyl ethyl(pentan -2-yl)propanedioate  
193 2918 29 00  376592 -58-4 5'-chloro -2'-hydroxy -3'-nitrobiphenyl -3-carboxylic acid  
369 2918 99 90  709031 -28-7 (3-hydroxytricyclo[3.3.1.1(3,7)]dec -1-yl)(oxo)acetic 
acid 
552 2918 99 90  35480 -52-5 2,5-bis(2,2,2 -trifluoroethoxy)benzoic acid  
559 2918 99 90  4651-67-6 (3α,5β) -3-hydroxy -7-oxocholan -24-oic acid  
264 2918 99 90  52179 -28-9 ethyl 2 -[4-(2,2-dichlorocyclopropyl)phenoxy] -2-
methylpropanoate  
143 2918 99 90  530141 -60-7 methyl 3 -(5-{[4-(cyclopentyloxy) -2-G/MA/TAR/RS/457  
- 14 - 
  ID CN code  CAS RN  Name  
hydroxyphenyl]carbonyl} -2-hydroxyphenyl)propanoate  
114 2920 90 10  91526 -18-0 4-(hydroxymethyl) -5-methyl -1,3-dioxol -2-one 
161 2921 49 00  334477 -60-0 (1R)-1-[3,5-bis(trifluoromethyl)phenyl] -N-
methylethanamine  
287 2921 49 00  376608 -71-8 (1R,2S) -2-(3,4-difluorophenyl)cyclopropanaminium 
(2R)-hydroxy(phenyl)ethanoate  
342 2921 49 00  1034457 -07-2 2-(2,3-dihydro -1H-inden -2-yl)propan -2-amine 
hydrochloride  
27 2921 49 00  945717 -05-5 2-(4-chloro -3-ethylphenyl)ethanamine hydrochloride  
221 2921 49 00  89-97-4 2-chlorobenzylamine  
26 2921 49 00  945717 -43-1 N-(4-tert-butylbenzy l)-2-(4-chloro -3-
ethylphenyl)ethanamine  
518 2921 51 90  150812 -21-8 N4-[(4-fluorophenyl)methyl] -2-nitro-1,4-
benzenediamine  
343 2922 19 80  1035455 -90-3 (2R)-1-(5-bromo -2,3-difluorophenoxy) -3-{[1-(2,3-
dihydro -1H-inden -2-yl)-2-methylpropan -2- 
yl]amino}propan -2-ol hydrochloride  
397 2922 19 80  0-00-0 [2-(chloromethyl) -4-(dibenzylamino)phenyl]methanol 
hydrochloride  
248 2922 19 80  133-51-7 antimonic acid -- 1-deoxy -1-(methylamino) -D-glucitol 
(1:1) 
344 2922 19 80  1035455 -87-8 ethyl (2E) -3-(3-{[(2R) -3-{[1-(2,3-dihydro -1H-inden -2-
yl)-2-methylpropan -2-yl]amino} -2-hydroxypropyl]oxy} -
4,5-difluorophenyl)prop -2-enoate hydrochloride  
185 2922 19 80  702686 -97-3 ethyl 3 -(3-{[(2R) -3-{[1-(2,3-dihydro -1H-inden -2-yl)-2-
methylpropan -2-yl]amino} -2-hydroxypropyl]oxy} -4,5-
difluor ophenyl)propanoate hydrochloride  
36 2922 29 00  20059 -73-8 2-[4-(aminomethyl)phenoxy] -N,N-dimethylethanamine  
536 2922 49 85  848133 -35-7 (2E)-4-(dimethylamino)but -2-enoic acid hydrochloride  
425 2922 49 85  610300 -07-7 (3S,5R) -3-amino -5-methyloctanoic acid  
424 2922 49 85  610300 -00-0 (3S,5R) -3-amino -5-methyloctanoic acid hydrochloride  
433 2922 49 85  143785 -86-8 4-(1-aminocyclopropyl) -2,3,5-trifluorobenzoic acid  
398 2922 49 85  848949 -85-9 4-fluoro -L-leucine -- ethyl hydrogen sulfate (1:1)  
475 2922 49 85  39068-93-4 methyl 2 -(dimethylamino) -2-phenylbutanoate  
174 2922 49 85  168619 -25-8 methyl 3' -aminobiphenyl -3-carboxylate  
565 2922 49 85  82834 -12-6 N-[(2S) -1-ethoxy -1-oxopentan -2-yl]-L-alanine  
474 2922 49 85  94133 -84-3 sodium 2 -amino -2-phenylbutanoate  
171 2922 50 00  503070 -58-4 triphenylacetic acid -- 4-{(1R) -2-[(6-{2-[(2,6-
dichlorobenzyl)oxy]ethoxy}hexyl)amino] -1-
hydroxyethyl} -2-(hydroxymethyl)phenol (1:1)  
149 2924 19 00  62009 -47-6 2-aminomalonamide  
175 2924 19 00  7355-58-0 N-(2-chloroethyl)acetamide  
367 2924 29 98  361442 -00-4 {2-[(tert -butoxycarbonyl)amino] -3-
hydroxytricyclo[3.3.1.1(3,7)]dec -1-yl}acetic acid  
521 2924 29 98  266993 -72-0 2,3-diaminobenzamide dihydrochloride  
532 2924 29 98  168080 -49-7 2-chloro -4-{[(5-fluoro -2-
methylphenyl)carbonyl]amino}be nzoic acid  
81 2924 29 98  317374 -08-6 2-methyl -4-{[(2-methylphenyl)carbonyl]amino}benzoic 
acid 
125 2924 29 98  143785 -84-6 4-(1-carbamoylcyclopropyl) -2,3,5-trifluorobenzoic acid  
434 2924 29 98  143785 -87-9 4-[1-(acetylamino)cyclopropyl] -2,3,5 -trifluorobenz oic 
acid G/MA/TAR/RS/457  
- 15 - 
  ID CN code  CAS RN  Name  
80 2924 29 98  108166 -22-9 4-{[(2-methylphenyl)carbonyl]amino}benzoic acid  
519 2924 29 98  150812 -23-0 ethyl {4 -[(4-fluorobenzyl)amino] -2-
nitrophenyl}carbamate  
237 2924 29 98  22316 -45-6 ethyl 3 -[(5-chloro -2-nitrophenyl)(phenyl)amino] -3-
oxopropano ate 
3 2924 29 98  316173 -29-2 methyl (1S,2S,3S,4R) -3-[(1S) -1-amino -2-ethylbutyl] -4-
[(tert -butoxycarbonyl)amino] -2-
hydroxycyclopentanecarboxylate  
378 2924 29 98  1142-20-7 N-benzyloxycarbonyl -L-alanine  
102 2924 29 98  84996 -93-0 N-cyclohexyl -5-hydroxypentan amide  
270 2924 29 98  579494 -66-9 propyl {4 -[2-(diethylamino) -2-oxoethoxy] -3-
ethoxyphenyl}acetate  
533 2925 19 95  265136 -65-0 ethyl 3 -amino -4-[2-(1,3-dioxo -1,3-dihydro -2H-isoindol -
2-yl)ethoxy]but -2-enoate  
33 2926 90 95  855425 -38-6 1-(2-ethylbutyl)cyclohex anecarbonitrile  
537 2926 90 95  846023 -24-3 2-cyano -N-(2,4-dichloro -5-methoxyphenyl)acetamide  
417 2926 90 95  591769 -05-0 3-cyclopentylprop -2-enenitrile  
50 2926 90 95  20099 -89-2 4-(bromoacetyl)benzonitrile  
54 2926 90 95  474554 -45-5 4,5-diethoxy -3-fluorob enzene -1,2-dicarbonitrile  
587 2926 90 95  79370 -78-8 5-hydroxybenzene -1,3-dicarbonitrile  
118 2926 90 95  139481 -28-0 methyl 2 -{[(2'-cyanobiphenyl -4-yl)methyl]amino} -3-
nitrobenzoate  
182 2928 00 90  860035 -10-5 1-({[(2,5 -dioxopyrrolidin -1-yl)oxy]carbonyl}oxy )ethyl 
2-methylpropanoate  
403 2928 00 90  910656 -45-0 2-hydroxy -2-(trifluoromethyl)butanehydrazide  
104 2928 00 90  95759 -10-7 4-chloro -2-[(2-methoxy -2-oxoethoxy)imino] -3-
oxobutanoic acid  
383 2928 00 90  473927 -63-8 ethyl (2Z) -chloro[2 -(4-
methoxyphenyl)hydr azinylidene]ethanoate  
144 2928 00 90  158671 -29-5 N,2-dihydroxy -4-methylbenzamide  
106 2928 00 90  84080 -68-2 tert-butyl (2Z) -2-[(2-methoxy -2-oxoethoxy)imino] -3-
oxobutanoate  
105 2928 00 90  268544 -50-9 tert-butyl-2-[(2-methoxy -2-oxoethoxy)imino] -3-
oxobutano ate 
101 2930 90 85  13459 -62-6 {2-[(4-chlorophenyl)sulfanyl]phenyl}acetic acid  
20 2930 90 85  211513 -21-2 1-(2-ethylbutyl) -N-(2-
sulfanylphenyl)cyclohexanecarboxamide  
181 2930 90 85  860035 -07-0 1-{[(methylsulfanyl)carbonyl]oxy}ethyl 2 -
methylpropanoate  
396 2930 90 85  893407 -18-6 2,2,2-trifluoro -1-[4'-(methylsulfonyl)biphenyl -4-
yl]ethanone  
86 2930 90 85  60759 -00-4 3,4-diethoxybenzenecarbothioamide  
180 2930 90 85  21048 -05-5 N-methylbenzenecarbothiohydrazide  
47 2931 00 95  13682 -94-5 (2-bromoethenyl)(trimeth yl)silane  
46 2931 00 95  914922 -89-7 (2R,4R) -4-[[(1,1 -dimethylethyl)dimethylsilyl]oxy] -N-
methoxy -N,2-dimethyl -7-oxoheptanamide  G/MA/TAR/RS/457  
- 16 - 
  ID CN code  CAS RN  Name  
44 2931 00 95  914922 -88-6 (2R,4R) -4-{[tert -butyl(dimethyl)silyl]oxy} -N-methoxy -
N,2-dimethyloct -7-enamide  
45 2931 00 95  871355 -80-5 (4R)-2-bromo -7-{[tert -butyl(diphenyl)silyl]oxy}hept -1-
en-4-yl 4-methylbenzenesulfonate  
192 2931 00 95  89694 -48-4 (5-chloro -2-methoxyphenyl)boronic acid  
359 2931 00 95  701278 -08-2 [(1R,5S) -5-[dimethyl(phenyl)silyl] -2-{[(2-
methoxypropan -2-yl)oxy]methyl }cyclopent -2-en-1-
yl]methanol  
360 2931 00 95  701278 -09-3 {(4S,5R) -5-[(benzyloxy)methyl] -4-
[dimethyl(phenyl)silyl]cyclopent -1-en-1-yl}methanol  
318 2931 00 95  796967 -18-5 1-(2-fluoro -5-methylphenyl) -3-[4-(4,4,5,5 -tetramethyl -
1,3,2-dioxaborolan -2-yl)phenyl] urea 
52 2931 00 95  172732 -52-4 2-(1,3,2 -dioxaborinan -2-yl)benzonitrile  
48 2931 00 95  185411 -12-5 methyl 3 -(trimethylsilyl)pent -4-enoate  
43 2932 19 00  253128 -10-8 (1S)-1,5:7,10 -dianhydro -12,13 -bis-O-[tert-
butyl(dimethyl)silyl] -2,3,4,6,8,11 -hexadeoxy -1-{2-
[(2S,5S) -5-(3-hydroxypropyl) -3-
methylidenetetrahydrofuran -2-yl]ethyl} -3-methyl -9-O-
methyl -4-methylidene -8-[(phenylsulfonyl)methyl] -D-
arabino -D-altro-tridecitol  
571 2932 19 00  441045 -17-6 (1S,3S,6S,9S,12S,14R,16R,18S,20R,21R,22S,26R,29S,
31R,32S,33R,35R,36 S)-20-[(2S) -3-amino -2-
hydroxypropyl] -21-methoxy -14-methyl -8,15-
bis(methylene) -2,19,30,34,37,39,40,41 -
octaoxanonacyclo[24.9.2.13,32.13,33.16,9.112,16.018,
22.029,36.031,35]hentetracontan -24-one 
methanesulfonate  
35 2932 29 85  916069 -80-2 (4S)-4-(fluoromethy l)dihydrofuran -2(3H) -one 
554 2932 29 85  63106 -93-4 1-phenyl -3-oxabicyclo[3.1.0]hexan -2-one 
140 2932 29 85  7734-80-7 2-oxo-2H-chromene -6-carboxylic acid  
399 2932 29 85  0-00-0 4-(4-fluorophenyl) -7-(isothiocyanatomethyl) -2H-
chromen -2-one 
142 2932 29 85  947408-91-5 6-[(2,4-dihydroxyphenyl)carbonyl] -2H-chromen -2-one 
141 2932 29 85  947408 -90-4 6-[(2,4-dimethoxyphenyl)carbonyl] -2H-chromen -2-one 
165 2932 99 00  452342 -08-4 (1R)-2-(benzylamino) -1-(2,2-dimethyl -4H-1,3-
benzodioxin -6-yl)ethanol  
206 2932 99 00  99541-23-8 (1R,2S,3R,4R,5R) -4-azido-2-{[(4aR,6S,7R,8S,8aR) -7,8-
bis(benzyloxy) -2-phenylhexahydropyrano[3,2 -
d][1,3]dioxin -6-yl]oxy} -6,8-dioxabicyclo[3.2.1]oct -3-yl 
acetate  
389 2932 99 00  461432 -25-7 (1S)-2,3,4,6 -tetra-O-acetyl -1,5-anhydro -1-[4-chloro -3-
(4-ethoxybenzyl)phenyl] -D-glucitol  
116 2932 99 00  196597 -79-2 (2E)-1,2,6,7 -tetrahydro -8H-indeno[5,4 -b]furan -8-
ylideneethanenitrile  
550 2932 99 00  
 3308-94-9 2-(3-chloropropyl) -2-(4-fluorophenyl) -1,3-dioxolane  G/MA/TAR/RS/457  
- 17 - 
  ID CN code  CAS RN  Name  
568 2932 99 00  274693 -53-7 [(3aS,4R,6S,6aR) -6-hydro xy-2,2-dimethyltetrahydro -
3aH-cyclopenta[d][1,3]dioxol -4-yl]carbamate  
61 2932 99 00  185954 -98-7 [6(2Z,3R)] -3-O-decyl-2-deoxy -6-O-[2-deoxy -3-O-(3-
metoxydecyl) -6-methyl -2-[(1-oxo-11-
octadecenyl)amino] -4-O-phosphono -β-D-
glucopyranosyl] -2-[(1,3-dioxotetradecy l)amino] -α-D-
glucopyranose 1 -(dihydrogen phosphate) tetrasodium 
salt 
203 2932 99 00  136172 -58-2 1,6-di-O-acetyl -2-azido-3,4-di-O-benzyl -2-deoxy -D-
glucopyranose  
115 2932 99 00  196597 -80-5 2-[(8S) -1,6,7,8 -tetrahydro -2H-indeno[5,4 -b]furan -8-
yl]ethanamine hy drochloride  
354 2932 99 00  666860 -59-9 2-amino -2-oxoethyl{3 -[trans -5-(6-methoxynaphthalen -
1-yl)-1,3-dioxan -2-yl]propyl}carbamate  
576 2932 99 00  117661 -72-0 5-(chloromethyl) -6-methyl -1,3-benzodioxole  
405 2932 99 00  959624 -24-9 6-(hydroxymethyl) -4-phenyl -3,4-dihydro -2H-chromen -
2-ol 
388 2932 99 00  960404 -59-5 but-2-yne-1,4-diol -- methyl 1 -C-[4-chloro -3-(4-
ethoxybenzyl)phenyl] -α-D-glucopyranoside (1:1)  
13 2932 99 00  15826 -37-6 disodium 5,5' -[(2-hydroxypropane -1,3-
diyl)bis(oxy)]bis(4 -oxo-4H-chromene -2-carboxylate)  
28 2932 99 00  204254 -84-2 ethyl (3aR,7R,7aR) -2,2-dimethyl -7-
[(methylsulfonyl)oxy] -3a,6,7,7a -tetrahydro -1,3-
benzodioxole -5-carboxylate  
205 2932 99 00  99541 -26-1 methyl (2S,3S,4S,5S,6S) -6-{[(1S,2S,3S,4R,5R) -3-
(acetyloxy) -4-azido-6,8-dioxabicyclo[3.2.1]oct -2-
yl]methyl} -4,5-bis(benzyloxy) -3-hydroxytetrahydro -2H-
pyran -2-carboxylate  
204 2932 99 00  114869 -97-5 methyl 6-O-acetyl -4-O-(2-O-acetyl -3-O-benzyl -6-
methyl -α-L-idopyranuronosyl) -3-O-benzyl -2-
{[(benzyloxy)carbonyl]amino} -2-deoxy -α-D-
glucopyranoside  
478 2933 19 90  1035677 -60-1 (4S)-3-(4-chlorophenyl) -N-methyl -4-phenyl -4,5-
dihydro -1H-pyrazole -1-carboximidamide 2,3 -
dihydroxybutanedioate  
194 2933 19 90  18048 -64-1 2-(3,4-dimethylphenyl) -5-methyl -2,4-dihydro -3H-
pyrazol -3-one 
477 2933 19 90  1035675 -24-1 3-(4-chlorophenyl) -N-methyl -4-phenyl -4,5-dihydro -1H-
pyrazole -1-carboximidamide  
310 2933 19 90  1028026 -83-6 5-methyl -1-(propan -2-yl)-4-[4-(propan -2-
yloxy)benzyl] -1,2-dihydro -3H-pyrazol -3-one 
585 2933 19 90  473921 -12-9 5-{[3,5 -diethyl -1-(2-hydroxyethyl) -1H-pyrazol -4-
yl]oxy}benzene -1,3-dicarbonitrile  
89 2933 29 90  65902 -59-2 2-bromo -4-nitro-1H-imidazole  G/MA/TAR/RS/457  
- 18 - 
  ID CN code  CAS RN  Name  
90 2933 29 90  57531-37-0 2-chloro -4-nitro-1H-imidazole  
24 2933 29 90  1000164 -35-1 3-(1,1-dimethylethyl) -N-[(9H-fluoren -9-
ylmethoxy)carbonyl] -1-(triphenylmethyl) -L-histidyl -2-
methylalanyl -L-α-glutamylglycine  
488 2933 29 90  152074 -97-0 L-α-aspartyl -L-α-glutamyl -L-asparagi nyl-L-prolyl -L-
valyl-L-valyl-L-histidyl -L-phenylalanyl -L-phenylalanyl -L-
lysyl-L-asparaginyl -L-isoleucyl -L-valyl-L-threonyl -L-
prolyl -L-arginyl -L-threonine  
489 2933 29 90  781666 -30-6 L-α-aspartyl -L-α-glutamyl -L-asparaginyl -L-prolyl -L-
valyl-L-valyl-L-histidy l-L-phenylalanyl -L-phenylalanyl -L-
lysyl-L-asparaginyl -L-isoleucyl -L-valyl-L-threonyl -L-
prolyl -L-arginyl -L-threonine tetraacetate  
176 2933 29 90  451470 -33-0 methyl 3' -(2-methyl -4,5-dihydro -1H-imidazol -1-
yl)biphenyl -3-carboxylate  
348 2933 39 99  925978 -49-0 (+)-5-[6-(1-methyl -1H-pyrazol -4-yl)pyridin -3-yl]-1-
azabicyclo[3.2.1]octane  
325 2933 39 99  876170 -44-4 (1S,5S) -3-(5,6-dichloropyridin -3-yl)-3,6-
diazabicyclo[3.2.0]heptane benzenesulfonate  
1 2933 39 99  741705 -70-4 (2R)-phenyl[(2R) -piperidin -2-yl]ethanoic acid 
hydrochloride  
162 2933 39 99  414910 -13-7 (2S)-hydroxy(phenyl)ethanoic acid -- (2R)-2-(4-fluoro -
2-methylphenyl)piperidin -4-one (1:1)  
314 2933 39 99  0-00-0 (3aR,6aR) -1-(pyridin -3-yl)octahydropyrrolo[3,4 -
b]pyrrole 4 -methylbenzenesulfonate  
315 2933 39 99 370882 -57-8 (3aR,6aR) -1-(pyridin -3-yl)octahydropyrrolo[3,4 -
b]pyrrole dihydrochloride  
121 2933 39 99  334618 -23-4 (3R)-piperidin -3-amine dihydrochloride  
579 2933 39 99  1062580 -52-2 (3R,4R) -1-benzyl -N,4-dimethylpiperidin -3-amine 
dihydrochloride  
578 2933 39 99  27262 -47-1 (S)-1-butyl-N-(2,6-dimethylphenyl)piperidine -2-
carboxamide  
183 2933 39 99  105812 -81-5 [(3S,4R) -4-(4-fluorophenyl) -1-methylpiperidin -3-
yl]methanol  
324 2933 39 99  876068 -51-8 [(3S,4S) -4-amino -1-(5,6-dichloropyridin -3-yl)pyrrolidin -
3-yl]me thanol  
408 2933 39 99  871022 -14-9 1-({4-[({[2-oxo-3-(propan -2-yl)-2,3-dihydro -1H-
benzimidazol -1-yl]carbonyl}amino)methyl]piperidin -1-
yl}methyl)cyclobutanecarboxylic acid  
549 2933 39 99  5421-92-1 1-(pyridin -4-yl)pyridinium chloride hydrochloride  
541 2933 39 99  272776 -12-2  1,1'-binaphthalene -2,2'-diol -- 
5-methoxy -2-{(S)-[(4-methoxy -3,5-dimethylpyridin -2-
yl)methyl]sulfinyl} -1H-benzimidazole  
(1:1) G/MA/TAR/RS/457  
- 19 - 
  ID CN code  CAS RN  Name  
409 2933 39 99  871022 -19-4 1-[(4-{[(tert -butoxycarbonyl)amino]methyl}piperidin -1-
yl)methyl]cyclobutanecarboxy lic acid  
414 2933 39 99  3613-73-8 2,8-dimethyl -5-[2-(6-methylpyridin -3-yl)ethyl] -2,3,4,5 -
tetrahydro -1H-pyrido[4,3 -b]indole  
535 2933 39 99  179687 -79-7 2-[(2-chloro -4-nitrophenoxy)methyl]pyridine  
201 2933 39 99  122321 -04-4 2-[methyl(pyridin -2-yl)amino]eth anol 
311 2933 39 99  945405 -37-8 2-methyl -3-[(2S) -pyrrolidin -2-ylmethoxy]pyridine 2,3 -
dihydroxybutanedioate  
155 2933 39 99  936637 -40-0 3,3'-piperidine -1,4-diyldipropan -1-ol 4-
methylbenzenesulfonate  
40 2933 39 99  88150 -62-3 3-ethyl-5-methyl -4-(2-chlorophe nyl)-2-{[2-(1,3-dioxo -
1,3-dihydro -2H-isoindol -2-yl)ethoxy]methyl} -6-methyl -
1,4-dihydropyridine -3,5-dicarboxylate  
404 2933 39 99  84100 -54-9 4-(ethylamino)piperidine -4-carboxamide  
157 2933 39 99  873546 -30-6 4,4'-[piperidine -1,4-diylbis(propane -3,1-diyloxy) ]bis(N' -
hydroxybenzenecarboximidamide)  
158 2933 39 99  873546 -74-8 4,4'-[piperidine -1,4-diylbis(propane -3,1-diyloxy)]bis[N' -
(acetyloxy)benzenecarboximidamide]  
159 2933 39 99  873546 -38-4 4,4'-[piperidine -1,4-diylbis(propane -3,1-
diyloxy)]dibenzenecarboximid amide trihydrochloride 
pentahydrate  
156 2933 39 99  873546 -80-6 4,4'-[piperidine -1,4-diylbis(propane -3,1-
diyloxy)]dibenzonitrile  
316 2933 39 99  78750 -61-5 4-[(3-nitropyridin -2-yl)amino]phenol  
87 2933 39 99  866109 -93-5 4-{4-[4-(trifluoromethoxy)phenoxy]pi peridin -1-
yl}phenol 4 -methylbenzenesulfonate  
472 2933 39 99  927889 -51-8 4-bromo -2,6-diethylpyridine 4 -methylbenzenesulfonate  
272 2933 39 99  691882 -47-0 4-hydroxybenzoic acid -- (2S,4E) -N-methyl -5-[5-
(propan -2-yloxy)pyridin -3-yl]pent -4-en-2-amine (1:1)  
323 2933 39 99  876068 -46-1 5,6-dichloro -N-(2,2-dimethoxyethyl)pyridin -3-amine  
220 2933 39 99  1072-98-6 5-chloropyridin -2-amine  
85 2933 39 99  298692 -34-9 6-(chloroacetyl)pyridine -2-carboxylic acid  
349 2933 39 99  550349 -58-1 7-chloro -3-(6-methoxypyridin -3-yl)-N,N,5 -trimethyl -4-
oxo-4,5-dihydro -3H-pyridazino[4,5 -b]indole -1-
carboxamide  
160 2933 39 99  414909 -98-1 benzyl 2 -(4-fluoro -2-methylphenyl) -4-oxo-3,4-
dihydropyridine -1(2H) -carboxylate  
164 2933 39 99  56880 -11-6 ethyl [(3 -endo) -8-methyl -8-azabicyclo[3.2. 1]oct-3-
yl)acetate  
273 2933 39 99  548797 -97-3 N-(2-{[(2S) -3-{[1-(4-chlorobenzyl)piperidin -4-
yl]amino} -2-hydroxy -2-methylpropyl]oxy} -4-
hydroxyphenyl)acetamide  
352 2933 39 99  0-00-0 N-[(S)-1-azabicyclo[2.2.2]oct -2-yl(phenyl)methyl] -2,6-
dichloro -3-(trifluor omethyl)benzamide hydrochloride  G/MA/TAR/RS/457  
- 20 - 
  ID CN code  CAS RN  Name  
289 2933 39 99  329003 -65-8 sodium hydrogen [1 -hydroxy -1-phosphono -2-(pyridin -
3-yl)ethyl]phosphonate hemipentahydrate  
58 2933 49 10  417716 -92-8 4-{3-chloro -4-[(cyclopropylcarbamoyl)amino]phenoxy} -
7-methoxyquinoline -6-carbox amide methanesulfonate  
584 2933 49 90  503291 -53-0 2-ethylbutyl (3S,4aS,6S,8aR) -6-[3-chloro -2-(1H-
tetrazol -5-yl)phenoxy]decahydro -3-
isoquinolinecarboxylate 4 -methylbenzenesulfonate  
539 2933 49 90  103733 -32-0  benzyl (3S) -6,7-dimethoxy -1,2,3,4 -
tetrahydrois oquinoline -3-carboxylate hydrochloride  
581 2933 49 90  503293 -98-9 (3S,4aS,6S,8aR) -6-hydroxy -2-
(methoxycarbonyl)decahydroisoquinoline -3-carboxylic 
acid 
583 2933 49 90  503290 -66-2 (3S,4aS,6S,8aR) -6-[3-chloro -2-(2H-tetrazol -5-
yl)phenoxy]decahydro -3-isoquino linecarboxylic acid 
hydrochloride  
580 2933 49 90  134388 -95-7 (3S,4aS,8aR) -2-(methoxycarbonyl) -6-
oxodecahydroisoquinoline -3-carboxylic acid -- 
(1R)-1-phenylethanamine (1:1)  
328 2933 49 90  868210 -14-4 4-(4-{[(2S,4R) -4-[acetyl(4 -chlorophenyl)amino] -2-
methyl -3,4-dihydroquinolin -1(2H) -
yl]carbonyl}phenoxy) -2,2-dimethylbutanoic acid  
545 2933 49 90  00-00-0 methyl 2 -[(3R) -3-{3-[(E)-2-(7-chloroquinolin -2-
yl)ethenyl]phenyl} -3-({[1-
(hydroxymethyl)cyclopropyl]methyl}sulfanyl)propyl]ben
zoate hydrochloride  
534 2933 49  90  848133 -76-6 N-(4-chloro -3-cyano -7-ethoxyquinolin -6-yl)acetamide  
479 2933 59 95  869490 -23-3 (3,3-difluoropyrrolidin -1-yl){(2S,4S) -4-[4-(pyrimidin -2-
yl)piperazin -1-yl]pyrrolidin -2-yl}methanone  
421 2933 59 95  941685 -40-1 (3R)-3-cyclopentyl -3-[4-(7-{[2-
(trimethylsilyl)ethoxy]methyl} -7H-pyrrolo[2,3 -
d]pyrimidin -4-yl)-1H-pyrazol -1-yl]propanenitrile  
416 2933 59 95  941678 -49-5 (3R)-3-cyclopentyl -3-[4-(7H-pyrrolo[2,3 -d]pyrimidin -4-
yl)-1H-pyrazol -1-yl]propanenitrile  
420 2933 59 95  941685 -41-2 (3S)-3-cyclopent yl-3-[4-(7-{[2-
(trimethylsilyl)ethoxy]methyl} -7H-pyrrolo[2,3 -
d]pyrimidin -4-yl)-1H-pyrazol -1-yl]propanenitrile  
394 2933 59 95  957187 -34-7 [(8R) -8-(3,5-difluorophenyl) -10-oxo-6,9-
diazaspiro[4.5]dec -9-yl]acetic acid  
190 2933 59 95  356058 -42-9 {2-[(4-fluorob enzyl)sulfanyl] -4-oxo-4,5,6,7 -tetrahydro -
1H-cyclopenta[d]pyrimidin -1-yl}acetic acid  
395 2933 59 95  0-00-0 2,3-dihydroxy -2,3-bis(phenylcarbonyl)butanedioic acid -
- ethyl [(8R) -8-(3,5-difluorophenyl) -10-oxo-6,9-
diazaspiro[4.5]dec -9-yl]acetate (1:1)  
407 2933 59 95  90213 -66-4 2,4-dichloro -7H-pyrrolo[2,3 -d]pyrimidine  
197 2933 59 95  3934-20-1 2,4-dichloropyrimidine  G/MA/TAR/RS/457  
- 21 - 
  ID CN code  CAS RN  Name  
189 2933 59 95  451487 -18-6 2-[(4-fluorobenzyl)sulfanyl] -1,5,6,7 -tetrahydro -4H-
cyclopenta[d]pyrimidin -4-one 
120 2933 59 95  865758 -96-9 2-[(6-chloro-3-methyl -2,4-dioxo -3,4-dihydropyrimidin -
1(2H) -yl)methyl]benzonitrile  
340 2933 59 95  934815 -71-1 2-[3-(6-{[2-(2,4-dichlorophenyl)ethyl]amino} -2-
methoxypyrimidin -4-yl)phenyl] -2-methylpropanoic acid 
phosphate  
278 2933 59 95  722543 -31-9 2-{ethyl[3 -({4-[(5-{2-[(3-fluorophenyl)amino] -2-
oxoethyl} -1H-pyrazol -3-yl)amino]quinazolin -7-
yl}oxy)propyl]amino}ethyl dihydrogen phosphate  
361 2933 59 95  1032066 -96-8 2-amino -9-{(1S,3R,4S) -3-[(benzyloxy)methyl] -4-
[dimethyl(phenyl)silyl] -2-methylidenecyclopentyl} -1,9-
dihydr o-6H-purin-6-one -- methanesulfonate (2:1)  
406 2933 59 95  540737 -29-9 3-{(3R,4R) -4-methyl -3-[methyl(7H -pyrrolo[2,3 -
d]pyrimidin -4-yl)amino]piperidin -1-yl}-3-
oxopropanenitrile 2 -hydroxypropane -1,2,3 -
tricarboxylate  
400 2933 59 95  1137917 -12-4 3-{[6-(ethylsu lfonyl)pyridin -3-yl]oxy} -5-{[(2S) -1-
hydroxypropan -2-yl]oxy}benzoic acid -- 1,4-
diazabicyclo[2.2.2]octane (2:1)  
422 2933 59 95  941685 -39-8 3-cyclopentyl -3-[4-(7-{[2-
(trimethylsilyl)ethoxy]methyl} -7H-pyrrolo[2,3 -
d]pyrimidin -4-yl)-1H-pyrazol -1-yl]propanenitr ile 
419 2933 59 95  941685 -27-4 4-(1H-pyrazol -4-yl)-7-{[2-
(trimethylsilyl)ethoxy]methyl} -7H-pyrrolo[2,3 -
d]pyrimidine  
365 2933 59 95  1780-26-3 4,6-dichloro -2-methylpyrimidine  
567 2933 59 95  145783 -14-8 4,6-dichloro -5-nitro-2-(propylsulfanyl)pyrimidine  
423 2933 59 95  3680-69-1 4-chloro -7H-pyrrolo[2,3 -d]pyrimidine  
215 2933 59 95  61379 -64-4 4-cyclopentylpiperazin -1-amine  
219 2933 59 95  55112 -42-0 4-methylpiperazine -1-carbonyl chloride hydrochloride  
338 2933 59 95  0-00-0 5-(benzylamino) -2-(3-methoxyphenyl) -7-(4-
methylpiperazin -1-yl)[1,2,4]triazolo[1,5 -a]quinoline -4-
carbonitrile -- (2E)-but-2-enedioate (2:1) hydrate  
471 2933 59 95  55293 -96-4 5,7-dimethyl[1,2,4]triazolo[1,5 -a]pyrimidine -2-
carbaldehyde  
288 2933 59 95  179688 -01-8 7-(benzyloxy) -6-methoxyquinaz olin-4(3H) -one 
198 2933 59 95  444731 -74-2 N-(2-chloropyrimidin -4-yl)-2,3-dimethyl -2H-indazol -6-
amine  
355 2933 59 95  0-00-0 N-(5-fluoro -3-methyl -1H-indol-1-yl)-4-methyl -2-
(pyridin -2-yl)pyrimidine -5-carboxamide  
484 2933 79 00  586414 -48-4 (-)-3-{3-bromo -4-[(2,4-difluorobenzyl)oxy] -6-methyl -
2-oxopyridin -1(2H) -yl}-N,4-dimethylbenzamide  
486 2933 79 00  425663 -71-4 (1S)-1-amino -3-methyl -1,3,4,5 -tetrahydro -2H-3-
benzazepin -2-one hydrochloride  G/MA/TAR/RS/457  
- 22 - 
  ID CN code  CAS RN  Name  
34 2933 79 00  813452 -14-1 (4S)-1-[(2S,3S,11bS) -2-amino -9,10-dimethoxy -
1,3,4,6,7,11b -hexahydro -2H-pyrido[2,1 -a]isoquinolin -3-
yl]-4-(fluoromethyl)pyrrolidin -2-one dihydrochloride  
77 2933 79 00  5162-90-3 3-(2-oxo-1,2-dihydroquinolin -4-yl)alanine  
384 2933 79 00  536760 -29-9 3-chloro -1-(4-nitrophenyl) -5,6-dihydropyridin -2(1H) -
one 
78 2933 79 00  4876-10-2 4-(bromomethyl)quinolin -2(1H) -one 
69 2933 79 00  5057-12-5 4,6,7,8 -tetrahydroquinoline -2,5(1H,3H) -dione  
72 2933 79 00  54197 -66-9 6-hydroxy -3,4-dihydroquinolin -2(1H) -one 
75 2933 79 00  22246 -18-0 7-hydroxy -3,4-dihydroquinolin -2(1H)-one 
380 2933 79 00  536759 -91-8 ethyl 1 -(4-methoxyphenyl) -6-(4-nitrophenyl) -7-oxo-
4,5,6,7 -tetrahydro -1H-pyrazolo[3,4 -c]pyridine -3-
carboxylate  
382 2933 79 00  503614 -91-3 ethyl 1 -(4-methoxyphenyl) -7-oxo-6-[4-(2-oxopiperidin -
1-yl)phenyl] -4,5,6,7 -tetrahydr o-1H-pyrazolo[3,4 -
c]pyridine -3-carboxylate  
485 2933 79 00  586379 -61-5 methyl 3 -(4-hydroxy -6-methyl -2-oxopyridin -1(2H) -yl)-
4-methylbenzoate  
368 2933 99 80  709031 -45-8 (1S,3S,5S) -2-azabicyclo[3.1.0]hexane -3-carboxamide 
methanesulfonate  
376 2933 99 80  649735-46-6 (2R)-1-({4-[(4-fluoro -2-methyl -1H-indol-5-yl)oxy] -5-
methylpyrrolo[2,1 -f][1,2,4]triazin -6-yl}oxy)propan -2-ol 
276 2933 99 80  51077 -14-6 (2S)-1-(tert-butoxycarbonyl)azetidine -2-carboxylic acid  
277 2933 99 80  631916 -97-7 (2S)-N-{4-[(Z)-amino(methoxyi mino)methyl]benzyl} -1-
{(2R) -2-[3-chloro -5-(difluoromethoxy)phenyl] -2-
hydroxyethanoyl}azetidine -2-carboxamide -- 
benzenesulphonic acid (1:1)  
564 2933 99 80  80875 -98-5 (2S,3aS,7aS) -octahydro -1H-indole -2-carboxylic acid  
313 2933 99 80  948846 -40-0 (2S,3S) -2,3-bis[(phenylcarbonyl)oxy]butanedioic acid -- 
ethyl (3aR,6aR) -hexahydropyrrolo[3,4 -b]pyrrole -5(1H) -
carboxylate (1:1)  
302 2933 99 80  1000164 -36-2 (5S,8S,11S,14S,17S,20S,23S,26S,29S,32S,35S,38S) -
5-(3-amino -3-oxopropyl) -20-benzyl -23-[(2S) -butan -2-
yl]-14,38 -bis{4-[(tert -butoxycarbonyl)amino]butyl} -29-
{[1-(tert-butoxycarbonyl) -1H-indol-3-yl]methyl} -17-(3-
tert-butoxy -3-oxopropyl) -1-(1H-fluoren -9-yl)-
8,11,26,41,41 -pentamethyl -32-(2-methylpropyl) -
3,6,9,12,15,18,21,24,27,30,33,36,39 -tridecaoxo -35-
(propan -2-yl)-2-oxa-
4,7,10,13,16,19,22,25,28,31,34,37,40 -
tridecaazadotetracontan -42-oic acid  
529 2933 99 80  22162 -51-2 1-(2-nitrobenzyl) -1H-pyrrole -2-carbaldehyde  
410 2933 99 80  35681 -40-4 1-(propan -2-yl)-1,3-dihydro -2H-benzimidazol -2-one 
522 2933 99 80  166170 -15-6 1-(tert-butoxycarbonyl) -2-methyl -D-proline  G/MA/TAR/RS/457  
- 23 - 
  ID CN code  CAS RN  Name  
322 2933 99 80  796967 -16-3 1-[4-(3-amino -1H-indazol -4-yl)phenyl] -3-(2-fluoro -5-
methylphenyl)urea  
321 2933 99 80  0-00-0 1-[4-(3-amino -1H-indazol -4-yl)phenyl] -3-(2-fluoro -5-
methylphenyl)urea hydrochloride  
196 2933 99 80 444731 -72-0 2,3-dimethyl -2H-indazol -6-amine  
415 2933 99 80  19686 -05-6 2,8-dimethyl -2,3,4,5 -tetrahydro -1H-pyrido[4,3 -b]indole  
524 2933 99 80  912444 -00-9 2-[(2R) -2-methylpyrrolidin -2-yl]-1H-benzimidazole -4-
carboxamide  
523 2933 99 80  912445 -36-4 2-[(2S) -2-methylpyrrolidin -2-yl]-1H-benzimidazole -4-
carboxamide dihydrochloride  
481 2933 99 80  163457 -23-6 3,3-difluoropyrrolidine hydrochloride  
65 2933 99 80  239463 -85-5 3-{5-[(2R) -2-aminopropyl] -7-cyano -2,3-dihydro -1H-
indol-1-yl}propyl benzoate (2R,3R) -2,3-
dihydroxybutanedioate  
150 2933 99 80  55321 -99-8 3-oxo-3,4-dihydropyrazine -2-carboxamide  
375 2933 99 80  952490 -01-6 4-[(4-fluoro -2-methyl -1H-indol-5-yl)oxy] -5-
methylpyrrolo[2,1 -f][1,2,4]triazin -6-yl 2,2 -
dimethylpropanoate  
274 2933 99 80  942436 -93-3 4-amino -8-(2,5-dimethoxyphenyl) -N-propylcinnoline -3-
carboxamide  
275 2933 99 80  942437 -37-8 4-amino -8-(2-fluoro -6-methoxyphenyl) -N-
propylcinnoline -3-carboxamide  
285 2933 99 80  288385 -88-6 4-fluoro -2-methyl -1H-indol-5-ol 
582 2933 99 80  503293 -47-8 5-(2-chloro -6-fluorophenyl) -2H-tetrazole  
71 2933 99 80  73963 -42-5 5-(4-chlorobutyl) -1-cyclohexyl -1H-tetrazole  
271 2933 99 80  606143 -52-6 5-[(4-bromo -2-chlorophenyl)amino] -4-fluoro -N-(2-
hydroxyethoxy) -1-methyl -1H-benzimidazole -6-
carboxamide  
347 2933 99 80  0-00-0 5-fluoro-1-(3-fluorobenzyl) -N-(1H-indol-5-yl)-1H-
indole -2-carboxamide  
373 2933 99 80  872206 -47-8 5-methyl -4-oxo-1,4-dihydropyrrolo[2,1 -f][1,2,4]triazin -
6-yl 2,2 -dimethylpropanoate  
151 2933 99 80  259793 -88-9 6-bromo -3-oxo-3,4-dihydropyrazine -2-carboxamide  
562 2933 99 80  1137606 -74-6 6-fluoro -3-oxo-3,4-dihydropyrazine -2-carbonitrile -- N-
cyclohexylcyclohexanamine (1:1)  
482 2933 99 80  261953 -36-0 6-iodo-1H-indazole  
73 2933 99 80  80076 -47-7 8,9-difluoro -5-methyl -1-oxo-6,7-dihydro -1H,5H -
pyrido[3,2,1 -ij]quinoline -2-carboxylic acid  
188 2933 99 80  52602 -39-8 9H-carbazol -4-ol 
235 2933 99 80  145641 -35-6 benzyl (2S,3aR,7aS) -octahydro -1H-indole -2-carboxylate 
hydrochloride  
540 2933 99 80  87269 -87-2 benzyl (2S,3aS,6aS) -octahydrocyclopenta[b]pyrrole -2-
carboxylate hydroc hloride  
21 2933 99 80  1012065 -72-3 ethyl 2 -amino -9,10-dimethoxy -1,6,7,11b -tetrahydro -
4H-pyrido[2,1 -a]isoquinoline -3-carboxylate  G/MA/TAR/RS/457  
- 24 - 
  ID CN code  CAS RN  Name  
563 2933 99 80  131707 -24-9 ethyl 6 -bromo -5-hydroxy -1-methyl -2-
[(phenylsulfanyl)methyl] -1H-indole -3-carboxylate  
124 2933 99 8 0 105152 -95-2 ethyl 7 -(3-aminopyrrolidin -1-yl)-1-(2,4-difluorophenyl) -
6-fluoro -4-oxo-1,4-dihydro -1,8-naphthyridine -3-
carboxylate  
117 2933 99 80  139481 -44-0 methyl 1 -[(2'-cyanobiphenyl -4-yl)methyl] -2-ethoxy -1H-
benzimidazole -7-carboxylate  
393 2933 99 80  0-00-0 methyl 1 -tert-butyl-2-hydroxy -1H-pyrrolo[2,3 -
b]pyridine -3-carboxylate  
555 2933 99 80  21688 -11-9 N2-[(benzyloxy)carbonyl] -L-glutaminyl -L-asparaginyl -S-
benzyl -L-cysteinyl -L-prolyl -L-leucylglycinamide  
370 2933 99 80  361440 -67-7 tert-butyl (1S,3S,5S) -3-carbamoyl -2-
azabicyclo[3.1.0]hexane -2-carboxylate  
371 2933 99 80  709031 -38-9 tert-butyl (2S) -2-carbamoyl -2,3-dihydro -1H-pyrrole -1-
carboxylate  
366 2933 99 80  709031 -43-6 tert-butyl [(1S) -2-[(1S,3S,5S) -3-cyano -2-
azabicyclo[3.1.0]hex -2-yl]-1-(3-
hydroxytricy clo[3.3.1.1(3,7)]dec -1-yl)-2-
oxoethyl]carbamate  
588 2933 49 90  936359 -25-0 methyl 2 -((R)-3-(3-((E)-2-(7-chloroquinolin -2-
yl)vinyl)phenyl) -3-(((1-
(hydroxymethyl)cyclopropyl)methyl)sulfanyl)propyl)ben
zoate  
341 2934 10 00  110130 -88-6 (2Z)-[(acetyloxy)imino ](2-amino -1,3-thiazol -4-
yl)ethanoic acid  
547 2934 10 00  68672 -66-2 (2Z)-{[(1-tert-butoxy -2-methyl -1-oxopropan -2-
yl)oxy]imino}[2 -(tritylamino) -1,3-thiazol -4-yl]ethanoic 
acid 
202 2934 10 00  291536 -35-1 (5Z)-5-(4-fluorobenzylidene) -1,3-thiazolidine -2,4-dione 
362 2934 10 00  302964 -24-5 2-amino -N-(2-chloro -6-methylphenyl) -1,3-thiazole -5-
carboxamide  
339 2934 10 00  866920 -24-3 3-[2-chloro -4-({4-methyl -2-[4-(trifluoromethyl)phenyl] -
1,3-thiazol -5-yl}methoxy)phenyl] -1,2,4 -oxadiazol -
5(4H) -one 
353 2934 10 00  75225 3-39-7 4-(2-chloro -4-methoxy -5-methylphenyl) -N-[(1S) -2-
cyclopropyl -1-(3-fluoro -4-methylphenyl)ethyl] -5-
methyl -N-(prop -2-yn-1-yl)-1,3-thiazol -2-amine  
57 2934 10 00  914361 -45-8 L-lysine -- {[(2R,3R) -3-[4-(4-cyanophenyl) -1,3-thiazol -
2-yl]-2-(2,4-difluorophen yl)-1-(1H-1,2,4 -triazol -1- 
yl)butan -2-yl]oxy}methyl dihydrogen phosphate -- 
ethanol (1:1:1)  
363 2934 10 00  302964 -08-5 N-(2-chloro -6-methylphenyl) -2-[(6-chloro -2-
methylpyrimidin -4-yl)amino] -1,3-thiazole -5-
carboxamide  G/MA/TAR/RS/457  
- 25 - 
  ID CN code  CAS RN  Name  
107 2934 10 00  127660 -04-2 sodium (2Z )-(2-amino -1,3-thiazol -4-
yl)(hydroxyimino)ethanoate  
135 2934 99 90  17381 -54-3 (1-benzothiophen -5-yl)acetic acid  
60 2934 99 90  630100 -90-2 (1R)-1,2-anhydro -4-C-{(1E,3E) -4-
[(1S,2S,3E,5R,6R,9R) -5-(1-carboxylato -4-
cycloheptylpiperazin -2-yl)-6,9-dihydroxy -2,6-dimethyl -
11-oxooxacyclododec -3-en-1-yl]penta -1,3-dien-1-yl}-
3,5-dideoxy -1-[(2R,3S) -3-hydroxypentan -2-yl]-D-
erythropentitol  
283 2934 99 90  220099 -91-2 (2R)-3'H-spiro[4 -azabicyclo[2.2.2]octane -2,2'-furo[2,3 -
b]pyridine]  
282 2934 99 90  220100 -81-2 (2R)-3'H-spiro[4 -azabicyclo[2.2.2]octane -2,2'-furo[2,3 -
b]pyridine] (S,S) -2,3-dihydroxybutanedioate  
29 2934 99 90  161599 -46-8 (2R,3R,4R,5R) -2-(4-amino -5-fluoro -2-oxopyrimidin -
1(2H) -yl)-2-fluoro -5-methyltetrahydrofuran -3,4-diyl 
diacetate  
30 2934 99 90  690270 -65-6 (2R,3S,4R) -5-(4-amino -2-oxopyrimidin -1(2H) -yl)-2-
azido-2-{[(2-
methylpropanoyl)oxy]methyl}tetrahydrofuran -3,4-diyl 
bis(2-methylpropanoate) hydrochloride  
392 2934 99 90  265121 -04-8 (3-{[(2R,3S) -2-{(1R) -1-[3,5-
bis(trifluoromethyl)phenyl]ethoxy} -3-(2-
fluorophe nyl)morpholin -4-yl]methyl} -5-oxo-2,5-
dihydro -1H-1,2,4-triazol -1-yl)phosphonic acid -- 1-
deoxy -1-(methylamino) -D-glucitol (1:2)  
126 2934 99 90  163680 -80-6 (3S)-10-[1-(acetylamino)cyclopropyl] -9-fluoro -3-
methyl -7-oxo-2,3-dihydro -7H-[1,4]oxazino[2,3,4 -
ij]quinoline -6-carboxylic acid  
544 2934 99 90  132335 -46-7 (3S)-N,N-dimethyl -3-(naphthalen -1-yloxy) -3-(thiophen -
2-yl)propan -1-amine  
345 2934 99 90  133413 -70-4 (3S,6R,9S,12R,15S,18R,21S,24R) -6,18-dibenzyl -
4,10,12,16,22,24 -hexamethyl -3,9,15,21 -tetrakis(2 -
methylpr opyl)-1,7,13,19 -tetraoxa -4,10,16,22 -
tetraazacyclotetracosane -2,5,8,11,14,17,20,23 -octone  
169 2934 99 90  503068 -36-8 (5R)-3-(6-{2-[(2,6-dichlorobenzyl)oxy]ethoxy}hexyl) -
5-(2,2-dimethyl -4H-1,3-benzodioxin -6-yl)-1,3-
oxazolidin -2-one 
166 2934 99 90  452339 -73-0 (5R)-5-(2,2-dimethyl -4H-1,3-benzodioxin -6-yl)-1,3-
oxazolidin -2-one 
470 2934 99 90  877130 -28-4 (6R)-6-cyclopentyl -6-[2-(2,6-diethylpyridin -4-yl)ethyl] -
3-[(5,7-dimethyl[1,2,4]triazolo[1,5 -a]pyrimidin -2-
yl)methyl] -4-hydroxy -5,6-dihydro -2H-pyran -2-one 
543 2934 99 90  132335 -44-5 (S)-3-(dimethylamino) -1-(thiophen -2-yl)propan -1-ol  G/MA/TAR/RS/457  
- 26 - 
  ID CN code  CAS RN  Name  
31 2934 99 90  812647 -80-6 {(2R,3S,4R,5R) -2-azido-5-(2,4-dioxo -3,4-
dihydropyrimidin -1(2H) -yl)-3,4-
bis[(phenylcarbonyl)oxy]tetrahydrofuran -2-yl}methyl 3 -
chlorobenzoate  
551 2934 99 90 00-00-0 1-(1-{4-[2-(4-fluorophenyl) -1,3-dioxolan -2-yl]butyl} -
1,2,3,6 -tetrahydropyridin -4-yl)-1,3-dihydro -2H-
benzimidazol -2-one 
418 2934 99 90  1029716 -44-6 1-(1-ethoxyethyl) -4-(4,4,5,5 -tetramethyl -1,3,2-
dioxaborolan -2-yl)-1H-pyrazole  
358 2934 99 90  165172-60-1 1-[(2R,5S) -5-(hydroxymethyl) -2,5-dihydrofuran -2-yl]-
5-methylpyrimidine -2,4(1H,3H) -dione -- 1-
methylpyrrolidin -2-one (1:1)  
139 2934 99 90  519187 -97-4 1-[3-(2-benzo[b]thien -5-ylethoxy)propyl] -3-azetidinol -
- (2Z)-2-butenedioate (1:1)  
49 2934 99 90  127000 -90-2 1-{[(2R,3S) -2-(2,4-difluorophenyl) -3-methyloxiran -2-
yl]methyl} -1H-1,2,4-triazole  
332 2934 99 90  710281 -33-7 2-({[(1R,3S) -3-{[2-(3-methoxyphenyl) -5-methyl -1,3-
oxazol -4-yl]methoxy}cyclohexyl]oxy}methyl) -6-
methylbenzoic acid  
136 2934 99 90  96803-30-4 2-(1-benzothiophen -5-yl)ethanol  
59 2934 99 90  913695 -00-8 2-[({4-[(2,2-dimethyl -1,3-dioxan -5-yl)methoxy] -3,5-
dimethylpyridin -2-yl}methyl)sulfinyl] -1Hbenzimidazole, 
sodium salt (1:1)  
286 2934 99 90  376608 -74-1 2-{[(3aR,4S,6R,6aS) -6-{[5-amino -6-chloro-2-
(propylsulfanyl)pyrimidin -4-yl]amino} -2,2-
dimethyltetrahydro -3aH-cyclopenta[d][1,3]dioxol -4-
yl]oxy}ethanol  
55 2934 99 90  474554 -48-8 2-bromo -1-[3-tert-butyl-4-methoxy -5-(morpholin -4-
yl)phenyl]ethanone  
148 2934 99 90  530141 -72-1 3-(5-{[4-(cyclopentyl oxy)-2-hydroxyphenyl]carbonyl} -
2-[(3-hydroxy -1,2-benzoxazol -6-
yl)methoxy]phenyl)propanoic acid  
138 2934 99 90  519188 -55-7 3-[2-(1-benzothiophen -5-yl)ethoxy] -1-(3-
hydroxyazetidin -1-yl)propan -1-one 
137 2934 99 90  519188 -42-2 3-[2-(1-benzothiophen -5-yl)etho xy]propionic acid  
566 2934 99 90  753015 -42-8 3-{(E)-2-[(3R) -pyrrolidin -3-yl]ethenyl} -5-(tetrahydro -
2H-pyran -4-yloxy)pyridine  
557 2934 99 90  26638 -53-9 3-chloro -6-methyldibenzo[c,f][1,2]thiazepin -11(6H) -one 
5,5-dioxide  
153 2934 99 90  499785 -81-8 3-oxo-4-(2,3,5 -tri-O-acetyl -β-D-ribofuranosyl) -3,4-
dihydropyrazine -2-carboxamide  
154 2934 99 90  356782 -84-8 3-oxo-4-(β-D-ribofuranosyl) -3,4-dihydropyrazine -2-
carboxamide  G/MA/TAR/RS/457  
- 27 - 
  ID CN code  CAS RN  Name  
211 2934 99 90  6504-57-0 4-[3-hydroxy -3-phenyl -3-(thiophen -2-yl)propyl] -4-
methylmorpholin -4-ium methyl sulfate  
329 2934 99 90  871484 -32-1 4-[4-({3-[(4-deoxy -4-fluoro -b-D-glucopyranosyl)oxy] -
5-(propan -2-yl)-1H-pyrazol -4-yl}methyl)phenyl] -N-
[1,3-dihydroxy -2-(hydroxymethyl)propan -2-
yl]butanamide  
575 2934 99 90  166964 -09-6 4-chloro -3-methyl -1,2-oxazol-5-amine  
93 2934 99 90  655233 -39-3 4-nitrobenzyl(6R,7R) -7-amino -8-oxo-3-[(2S) -
tetrahydrofuran -2-yl]-5-thia-1-azabicyclo[4.2.0]oct -2-
ene-2-carboxylate hydrochloride  
542 2920 90 85  89729 -09-9 5,7-dioxa -6-thiaspiro[2.5]octane -6-oxide  
172 2934 99 90  388082-75-5 5-[4-[[3-chloro -4-[(3-
fluorophenyl)methoxy]phenyl]amino] -6-quinazolinyl] -2-
furancarboxaldehyde -- 4-methylbenzenesulfonate (1:1)  
134 2934 99 90  4923-87-9 5-bromo -1-benzothiophene  
146 2934 99 90  947408 -95-9 6-(bromomethyl) -2-triphenylmethyl -1,2-benzisoxazol -
3(2H) -one 
145 2934 99 90  947408 -94-8 6-methyl -2-trityl-1,2-benzoxazol -3(2H) -one 
110 2934 99 90  67978 -05-6 diphenylmethyl(2R) -3-methyl -2-[(1R,5S) -3-(4-
methylphenyl) -7-oxo-4-oxa-2,6-
diazabicyclo[3.2.0]hept -2-en-6-yl]but -3-enoate  
357 2934 99 9 0 1001859 -46-6 DNA (synthetic plasmid vector pCOR human interferon 
beta signal peptide fusion protein with 21 -154-human 
acidic fibroblast growth factor -specifying)  
326 2934 99 90  665058 -78-6 DNA, d(T -sp-C-G-sp-T-sp-C-G-sp-T-sp-T-sp-T-sp-T-sp-
G-sp-A-sp-C-G-sp-T-sp-T-sp-T-sp-T-sp-Gsp- 
T-sp-C-G-sp-T-sp-T) 
401 2934 99 90  923591 -06-4 methyl (5R,7S,10S) -10-tert-butyl-15,15 -dimethyl -
3,9,12 -trioxo -6,7,9,10,11,12,14,15,16,17,18,19 -
dodecahydro -1H,5H -2,23:5,8 -dimethano -4,13,2,8,11 -
benzodioxatriazacyclohenicosine -7(3H)-carboxylate  
577 2934 99 90  59337 -92-7 methyl 3 -(chlorosulfonyl)thiophene -2-carboxylate  
147 2934 99 90  947409 -01-0 methyl 3 -[5-[4-(cyclopentyloxy) -2-hydroxybenzoyl] -2-
[(2-triphenylmethyl -1,2-benzisoxazol -3(2H) -on- 
6-yl)methoxy]phenyl]propionate  
212 2934 99 90  85006 -31-1 methyl 3 -amino -4-methylthiophene -2-carboxylate  
280 2934 99 90  893428 -72-3 N-(5-chloro -1,3-benzodioxol -4-yl)-7-[2-(4-methyl -1-
piperazinyl)ethoxy] -5-[(tetrahydro -2H-pyran -4-yl)oxy] -
4-quinazolinamine -- (2E)-2-butenedioate (1:2)  
18 2934 99 90  390800 -88-1 N,N',N'' -(boroxin -2,4,6-triyltris{[(1S) -3-methylbutane -
1,1-diyl]imino[(2S) -1-oxo-3-phenylpropane -1,2-
diyl]})tripyrazine -2-carboxamide  
99 2934 99 90  112913 -94-7 N-{[4-(4-fluorobenzyl)morpholin -2-
yl]methyl}acetamide  G/MA/TAR/RS/457  
- 28 - 
  ID CN code  CAS RN  Name  
412 2934 99 90  120788 -03-6 S-[(1R,3S) -1-oxidotetrahydrothiophen -3-yl] 
ethanethioate  
402 2935 00 90  1198178 -65-2 (1R,2R) -1-[(cyclopropylsulfonyl)carbamoyl] -2-
ethylcyclopropanaminium 4 -methylbenzenesulfonate  
556 2935 00 90  39570 -96-2 (2R)-3-(benzylsulfanyl) -N-[(2S) -1-{[(2S,3S) -1-
hydrazinyl -3-methyl -1-oxopentan -2-yl]amino} - 
3-(4-hydroxyphenyl) -1-oxopropan -2-yl]-2-{[(4-
methylphenyl)sulfonyl]amino}propanamide  
79 2935 00 90  24310 -36-9 1-[(4-methylphenyl)sulfonyl] -1,2,3,4 -tetrahydro -5H-1-
benzazepin -5-one 
346 2935 00 90  0-00-0 2-(cyclohexylmethyl) -N-{2-[(2S) -1-methylpyrrolidin -2-
yl]ethyl} -1,2,3,4 -tetrahydroisoquinoline -7-sulfonamide 
di[(2E) -but-2-enedioate] hydrate  
281 2935 00 90  941690 -55-7 3-[(methylsulfonyl)amino] -2-phenyl -N-[(1S) -1-
phenylpropyl]quinoline -4-carboxamide  
199 2935 00 90  6973-09-7 5-amino -2-methylbenzenesulfonamide  
82 2935 00 90  193686 -76-9 7-chloro -1-[(4-methylphenyl)sulfonyl] -1,2,3,4 -
tetrahydro -5H-1-benzazepin -5-one 
130 2935 00 90  123664 -84-6 N-(5-methoxy -2-phenoxyphenyl)methanesulfonamide  
133 2935 00 90  149457 -03-4 N-[4-(N-formylglycyl) -5-hydroxy -2-
phenoxyphenyl]methanesulfonamide  
132 2935 00 90  149456 -98-4 N-[4-(N-formylglycyl) -5-methoxy -2-
phenoxyphenyl]methanesulfonamide  
319 2935 00 90  141450 -48-8 N-{2-[(4-hydroxyphenyl)amino]pyridin -3-yl}-4-
methoxybenzenesu lfonamide hydrochloride  
391 2935 00 90  289042 -10-0 N-{5-[(diphenylphosphoryl)methyl] -4-(4-fluorophenyl) -
6-(propan -2-yl)pyrimidin -2-yl}-N-
methylmethanesulfonamide  
187 2939 99 00  7689-03-4 (4S)-4-ethyl-4-hydroxy -1H-
pyrano[3',4':6,7]indolizino[1,2 -b]quinoli ne-
3,14(4H,12H) -dione  
239 2939 99 00  477-29-2 colchicoside  
173 2940 00 00  604-69-3 1,2,3,4,6 -penta -O-acetyl -β-D-glucopyranose  
333 2940 00 00  647834 -15-9 2-(4-methoxybenzyl)thiophen -3-yl β-D-glucopyranoside  
127 2941 90 00  76610 -92-9 (6R,7R) -7-({N-[(4-ethyl-2,3-dioxopiperazin -1-
yl)carbonyl] -D-threonyl}amino) -3-{[(1-methyl -1H-
tetrazol -5-yl)sulfanyl]methyl} -8-oxo-5-thia-1-
azabicyclo[4.2.0]oct -2-ene-2-carboxylic acid  G/MA/TAR/RS/457  
- 29 - 
  ID CN code  CAS RN  Name  
570 3907 20 99  913976 -27-9 poly(oxy -1,2-ethanediyl), α -hydro -ω-methoxy, diester 
with 21N6, 21’N6 -[[(N2, N6 -dicarboxy -L-lysyl-β-
alanyl)imino]bis(1 -oxo-2, 1-ethanediyl)]bis[N -
acetylglycyl -L-leucyl -L-tyrosyl-L-alanyl -L-cysteinyl -L-
histidyl -L-methionylglycyl -L-prolyl -L-isoleucyl -L-
threonyl -3-(1-naphthalenyl) -L-alanyl -L-valyl-L-
cysteinyl -L-glutaminyl -L-prolyl -L-leucyl -L-arginyl -N-
methylglycyl -L-lysinamide] cyclic (6 →15), (6 ’→15’) 
bis(disulfide)  
 G/MA/TAR/RS/457  
- 30 - 
  ANNEX IV  
List of pharmaceutical intermediates, i.e. compounds used for the manufacture of 
finished pharmaceutical products, to be withdrawn from the list of products receiving 
duty-free treatment included in Annex 6 to Annex I to Regulation (EEC) No 2658/87 due 
to their transfer to the list of products receiving duty -free treatment included in Annex 3  
to Annex I to Regulation (EEC) No 2658/87  
 
CN code  CAS RN  Name  
2915 39 00  
 
 
2937 29 00  7753-60-8 17-alpha -hydroxy -3,20-dioxopregna -4,9(11) -diene -21-yl acetate  
 
see a necortave (INN)  
2920 90 85  163133 -43-5 4-(nitrooxy)butyl (2S) -2-(6-methoxy -2-naphthyl)propanoate  
 
see naproxcinod (INN)  
2924 29 98  194085 -75-1 2-(2-chlorophenyl) -2-hydroxyethyl carbamate  
 
see carisbamate (INN)  
2933 39 99  103129 -82-4 3-ethyl 5 -methyl 2 -[(2-aminoethoxy)methyl] -4-(2-chlorophenyl) -
6-methyl -1,4-dihydropyridine -3,5-dicarboxylate  
 
see levamlodipine (INN)  
2933 39 99  319460 -85-0 N-methyl -2-{[3-((E)-2-pyridin -2-ylvinyl) -1H-indazol -6-
yl]sulfanyl}benzamide  
 
see axitinib (INN)  
2934 10 00  302962 -49-8 N-(2-chloro -6-methylphenyl) -2-({6-[4-(2-
hydroxyethyl)piperazin -1-yl]-2-methylpyrimidin -4-
yl}amino)thiazole -5-carboxamide  
 
see dasatinib (INN)  
2934 99 90  143491 -57-0 (2R,5S) -4-amino -5-fluoro -1-[2-(hydroxymethyl) -1,3-oxathiolan -
5-yl]pyrimidin -2(1H) -one 
 
see emtricitabine(INN)  
2934 99 90  98819 -76-2 (2S)-2-[(S)-(2-ethoxyphenoxy)phenylmethyl]morpholine  
 
see esreboxetine (INN)  
2934 99 90  475479 -34-6 (2S)-2-methoxy -3-{4-[2-(5-methyl -2-phenyl -1,3-oxazol -4-
yl)ethoxy] -1-benzothiophen -7-yl}propanoic acid  
 
see ale glitazar (INN)  
2934 99 90  377727 -87-2 2-(2-furyl) -7-(2-{4-[4-(2-methoxyethoxy)phenyl]piperazin -1-
yl}ethyl) -7H-pyrazolo[4,3 -e][1,2,4]triazolo[2,3 -c]pyrimidin -5-
amine  
 
see preladenant (INN)  
2934 99 90  189003 -92-7 2-{7-fluoro -2-oxo-4-[2-(4-thieno[3,2 -c]pyri din-4-ylpiperazin -1-
yl)ethyl]quinolin -1(2H) -yl}acetamide  
 
see trelanserin (INN)  
2934 99 90  134379 -77-4 4-amino -5-fluoro -1-[(2R,5S) -5-(hydroxymethyl) -2,5-
dihydrofuran -2-yl]pyrimidin -2(1H) -one 
 
see dexelvucitabine (INN)  
 
 
2934 99 90  518048 -05-0 potassium 4 -[N-(2-fluorobenzyl)carbamoyl] -1-methyl -2-[1-G/MA/TAR/RS/457  
- 31 - 
  CN code  CAS RN  Name  
methyl -1-(5-methyl -1,3,4 -oxadiazole -2-carboxamido)ethyl] -6-
oxo-1,6-dihydropyrimidine -5-olate 
 
see raltegravir (INN)  
2935 00 90  170569 -88-7 4-[5-(4-fluorophenyl) -3-(trifluoromethyl)pyrazol -1-yl]benzene -1-
sulfona mide 
 
see mavacoxib (INN)  
2935 00 90  186497 -07-4 N-(3-methoxy -5-methylpyrazin -2-yl)-2-[4-(1,3,4 -oxadiazol -2-
yl)phenyl]pyridine -3-sulfonamide  
 
see zibotentan (INN)  
 
 
__________