Patent ID: 6573266
Filing Date: 2003-06-03
Classification: A61P,C07D

Abstract:
A compound of the following formula (Id): wherein,R1b is one or more substituents independently selected from the group consisting of hydrogen, alkyl, haloalkyl, aralkyl, hydroxyalkenyl, alkoxyalkyl, dialkylaminoalkyl, alkoxycarbonyl, alkoxycarbonylalkyl, piperazinylalkyl, tetrazolylalkyl, and imidazolylalkyl; R3 is phenyl substituted by one or more substituents independently selected from the group consisting of hydrogen, halo, alkyl, alkoxy, formyl, nitro, cyano, aminoalkoxy, alkenyl, hydroxyalkyl, amino, alkylcarbonylamino, arylcarbonylamino, alkoxycarbonylalkylcarbonylamino, alkoxycarbonyl, alkylcarbonyl, aminocarbonyl, ureido, glycinamido, tetrazolylalkyl, piperidinylalkyl, and imidazolylalkyl; R4 is â€”Oâ€”; R5 is an alkylene chain or an alkylidene chain, R6 is â€”C(O)â€” or â€”C(S)â€”; and R10 is a heterocyclyl selected from the group consisting of furanyl and thienyl wherein the heterocyclyl is optionally substituted by one or more substituents selected from the group consisting of halo and nitro; as a single stereoisomer or a mixture thereof; or a pharmaceutically acceptable salt thereof.