Patent ID: 8962846
Filing Date: 2015-02-24
Classification: A61P,C07D

Abstract:
1. A compound of formula (I): in which: R1 represents a hydrogen atom, an aryl, a substituted aryl, an alkyl, a cycloalkyl or a cycloalkylalkyl, R2 represents a hydrogen atom, a hydroxyl or a lower alkyl, a substituted lower alkyl, a higher alkyl, a substituted higher alkyl, a cycloalkyl, a cycloalkylalkyl, a lower alkoxy, a substituted lower alkoxy, a higher alkoxy, a substituted higher alkoxy, a cycloalkylalkoxy, an acyloxy, an acyl, an alkoxycarbonyl, a carboxamide, a carboxylic acid, a cyano or an amino disubstituted with an acyl and an aryl or alkyl, R3 represents an aralkyl or a substituted aralkyl, R4 represents a heteroaralkyl or a substituted heteroaralkyl, R5 represents a hydrogen atom or an alkyl, X represents an oxygen atom or a sulfur atom, n, m may be equal to 1 or 2; or a corresponding salt or enantiomer, having antagonist activity with respect to the MC4R receptor.