Patent ID: 6407041
Filing Date: 2002-06-18
Classification: A01N,C07D

Abstract:
A compound of the formula (I) whereinQ represents O, S, SO, SO2, NH or N(C1-C4-alkyl), R1 represents hydrogen or represents unsubstituted or hydroxyl-, cyano-, halogen- or C1-C4-alkoxy-substituted alkyl having 1 to 6 carbon atoms, R2 represents hydrogen, represents formyl or represents in each case unsubstituted or cyano-, halogen- or C1-C4-alkoxy-substituted alkyl, alkylcarbonyl, alkoxycarbonyl or alkylaminocarbonyl having in each case 1 to 6 carbon atoms in the alkyl groups, R3 represents unsubstituted or hydroxyl-, cyano-, halogen- or C1-C4-alkoxy-substituted alkyl having 1 to 6 carbon atoms or represents unsubstituted or cyano-, halogen- or C1-C4-alkyl-substituted cycloalkyl having 3 to 6 carbon atoms, R4 represents hydrogen or alkyl having 1 to 4 carbon atoms, R5 represents hydrogen or alkyl having 1 to 4 carbon atoms, Ar represents in each case unsubstituted or substituted phenyl, naphthyl, tetralinyl or heteroaryl, wherein the heteroaryl is selected from the group consisting of: furyl, benzofuryl, thienyl, benzothienyl, thiazolyl, benzothiazolyl, oxazolyl, benzoxazolyl, isoxazolyl, thiadiazolyl, oxadiazolyl, pyrazolyl, imidazolyl, pyrrolyl, pyridinyl, and pyrimidinyl, and wherein the substituent are in each case selected from the group consisting of: hydroxyl, cyano, carbamoyl, thiocarbamoyl, nitro, halogen; unsubstituted or hydroxyl-, cyano- or halogen-substituted alkyl or alkoxy having in each case 1 to 6 carbon atoms; unsubstituted or halogen-substituted alkylcarbonyl, alkoxycarbonyl, alkylthio, alkylsulphinyl, alkylsulphonyl, dialkylamino, alkylcarbonylamino, alkylsulphonyl-amino, bis-alkylcarbonyl-amino, bis-alkylsulphonyl-amino, N-alkyl-N-alkylcarbonyl-amino or N-alkyl-N-alkylsulphonyl-amino having in each case 1 to 6 carbon atoms in the alkyl groups; unsubstituted or hydroxyl-, cyano-, nitro-, halogen-, C1-C4-alkyl-, C1-C4-halogenoalkyl-, C1-C4-alkoxy- or C1-C4-halogenoalkoxy-substituted phenyl or phenoxy; and unsubstituted or halogen-substituted methylenedioxy or ethylenedioxy, and Z is selected from the group consisting of hydrogen, cyano, halogen; unsubstituted or hydroxyl-, cyano-, halogen-, C1-C4-alkoxy-, C1-C4-alkyl-carbonyl-, C1-C4-alkoxy-carbonyl-, C1-C4-alkylthio-, C1-C4-alkylsulphinyl- or C1-C4-alkylsulphonyl-substituted alkyl, alkoxy, alkylcarbonyl, alkoxycarbonyl, alkylthio, alkylsulphinyl or alkylsulphonyl having in each case 1 to 6 carbon atoms in the alkyl groups: unsubstituted or cyano-, halogen- or C1-C4-alkoxy-substituted alkenyl or alkynyl having in each case 2 to 4 carbon atoms in the alkenyl or alkynyl group; and unsubstituted or cyano-, halogen- or C1-C4-alkyl-substituted cycloalkyl having 3 to 6 carbon atoms.