Patent ID: 6262065
Filing Date: 2001-07-17
Classification: C07D,Y02P

Abstract:
A compound having the formula (II) ##STR35##wherein:each R.sup.1, independently of the other, is H, acetyl, benzyl, methoxymethyl, tosyl, mesyl, trifluoromesyl, .sub.tri (C.sub.1-4 alkyl)silyl, di(C.sub.1-4 alkyl)phenylsilyl, diphenyl(C.sub.1-4 alkyl)silyl, triphenylsilyl, or together both R' form a C.sub.3-6 alkylidene protecting group;each R"", independently of the other, is H, acetyl, benzyl, methoxymethyl, tosyl, mesyl, trifluoromesyl, tri(C.sub.1-4 alkyl)silyl, di(C.sub.1-4 alkyl)phenylsilyl, diphenyl(C.sub.1-4 alkyl)silyl, or triphenylsilyl; andR* isH;straight chain C.sub.1-22 -alkyl;branched C.sub.3-22 -alkyl;C.sub.3-8 -cycloalkyl;C.sub.3-8 -cycloalkyl substituted with straight chain C.sub.1-22 -alkyl;C.sub.3-8 -cycloalkyl substituted with branched C.sub.3-22 -alkyl;a group of the formula ##STR36##wherein:X'=O, S, NH, NR.sup.1 (R.sup.1 is C.sub.1-22 -alkyl), or NAr,m=0-5;n=0-5; andm+n.gtoreq.2;--(CH.sub.2).sub.n' Ar (n'=1 to 22);--(CH.sub.2).sub.n' G (n'=1 to 22);--Ar; and--G;wherein Ar is: ##STR37##wheren""=2 to 5;X'=NH, NR.sup.1 (R.sup.1 is C.sub.1-22 -alkyl), NAr, O, or Sand each carbon atom may be substituted with halogen, C.sub.1-22 -alkyl, C.sub.6-10 -aryl or G;wherein G is:F, Cl, Br, I,--CN, --CHO, --COR.sup.1, --CHNOH, --CHNOR.sup.1, --CR.sup.1 NOH, --CR.sup.1 NHOR.sup.2, --CN, --CO.sub.2 H, --CO.sub.2 R.sup.1, --CONH.sub.2, --CONHR.sup.1, --CONR.sup.1 R.sup.2, --CSNH.sub.2, --CSNHR.sup.1, --CSNR.sup.1 R.sup.2, --C(NH)OR.sup.1, --C(NR)OR.sup.1, --C(NH)SR.sup.1, --C(NR)SR.sup.1, --C(NH)NH.sub.2, --C(NR.sup.1)NH.sub.2, --C(NH)NR.sup.1 R.sup.2, --C(NR)R.sup.1 R.sup.2, --C(NR.sup.1)NHR.sup.2, --CONHOH, --CONR.sup.1 OH, --CONHOR.sup.1, --CONR.sup.1 OR.sup.2, --CONHNH.sub.2, --CONR.sup.1 NH.sub.2, --CONHNR.sup.1 R.sup.2, --CONR.sup.1 NHR.sup.2, -or CONR.sup.1 NR.sup.2 R.sup.3,(wherein R.sup.1, R.sup.2, and R.sup.3 are each independently C.sub.1-22 -alkyl).