Patent ID: 6114286
Filing Date: 2000-09-05
Classification: A01N,C07D

Abstract:
A pyrimidinone compound encompassed by the following formula: ##STR36## wherein, R.sup.1 represents hydrogen, halogen, C.sub.1 -C.sub.3 alkyl or C.sub.1 -C.sub.3 haloalkyl;R.sup.2 represents hydrogen, halogen, C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 haloalkyl, OR.sup.8, SR.sup.9, NHR.sup.10, COOR.sup.11, COR.sup.12, SO.sub.2 R.sup.13, NO.sub.2 or CN;R.sup.3 represents hydrogen, halogen, C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.3 alkoxy C.sub.1 -C.sub.3 alkyl, OR.sup.8, SR.sup.9, NHR.sup.10, COOR.sup.11, COR.sup.12, SO.sub.2 R.sup.13, C(R.sup.12).dbd.C(R.sup.14)(R.sup.15), NO.sub.2 or CN;R.sup.4 represents hydrogen, halogen, C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.3 alkoxy C.sub.1 -C.sub.3 alkyl, OR.sup.8, SR.sup.9, NHR.sup.10, COOR.sup.11, COR.sup.12, SO.sub.2 R.sup.13, CH.dbd.C(R.sup.14)(R.sup.15), C(R.sup.16).dbd.NOR.sup.17, NO.sub.2 or CN;R.sup.5 represents hydrogen, halogen or C.sub.1 -C.sub.3 alkyl;R.sup.6 represents C.sub.1 -C.sub.3 alkyl or C.sub.1 -C.sub.3 haloalkyl;R.sup.7 represents nitrogen or CH;in whichR.sup.8 represents hydrogen, C.sub.1 -C.sub.10 alkyl, C.sub.1 -C.sub.10 haloalkyl, C.sub.3 -C.sub.8 alkenyl, C.sub.3 -C.sub.8 haloalkenyl, C.sub.3 -C.sub.8 alkynyl, C.sub.3 -C.sub.8 haloalkynyl, C.sub.3 -C.sub.10 cycloalkyl, C.sub.3 -C.sub.10 halocycloalkyl, C.sub.3 -C.sub.10 cycloalkenyl, C.sub.3 -C.sub.10 halocycloalkenyl, C.sub.1 -C.sub.5 alkylcarbonyl, C.sub.1 -C.sub.5 haloalkylcarbonyl, C.sub.3 -C.sub.6 cycloalkylcarbonyl, C.sub.3 -C.sub.6 halocycloalkylcarbonyl, C.sub.1 -C.sub.6 alkylcarbonyl C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 haloalkylcarbonyl C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 alkylcabonyl C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 haloalkylcarbonyl C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 alkoxycarbonyl, C.sub.1 -C.sub.6 haloalkoxycarbonyl, C.sub.3 -C.sub.10 cycloalkoxycarbonyl, carboxy C.sub.1 -C.sub.5 alkyl, C.sub.1 -C.sub.10 alkoxycarbonyl C.sub.1 -C.sub.5 alkyl, C.sub.1 -C.sub.10 haloalkoxycarbonyl C.sub.1 -C.sub.5 alkyl, C.sub.1 -C.sub.10 alkoxycarbonyl C.sub.1 -C.sub.5 haloalkyl, C.sub.1 -C.sub.10 haloalkoxycarbonyl C.sub.1 -C.sub.5 haloalkyl, C.sub.3 -C.sub.10 cycloalkoxycarbonyl C.sub.1 -C.sub.5 alkyl, C.sub.3 -C.sub.10 halocycloalkoxycarbonyl C.sub.1 -C.sub.5 alkyl, C.sub.3 -C.sub.10 halocycloalkoxycarbonyl C.sub.1 -C.sub.5 haloalkyl, C.sub.3 -C.sub.10 cycloalkoxycarbonyl C.sub.1 -C.sub.5 haloalkyl, C.sub.1 -C.sub.6 alkoxy C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 alkoxy C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 haloalkoxy C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 haloalkoxy C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 alkylthio C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 alkylthio C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 haloalkylthio C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 haloalkylthio C.sub.1 -C.sub.6 haloalkyl, cyano C.sub.1 -C.sub.4 alkyl, aryl that may have substituent(s), aryl C.sub.1 -C.sub.3 alkyl that may have substituent(s) or arylcarbonyl that may have substituent(s);R.sup.9 represents hydrogen, C.sub.1 -C.sub.10 alkyl, C.sub.1 -C.sub.10 haloalkyl, C.sub.3 -C.sub.8 alkenyl, C.sub.3 -C.sub.8 haloalkenyl, C.sub.3 -C.sub.8 alkynyl, C.sub.3 -C.sub.8 haloalkynyl, C.sub.3 -C.sub.10 cycloalkyl, C.sub.3 -C.sub.10 halocycloalkyl, C.sub.3 -C.sub.10 cycloalkenyl, C.sub.3 -C.sub.10 halocycloalkenyl, C.sub.1 -C.sub.5 alkylcarbonyl, C.sub.1 -C.sub.5 haloalkylcarbonyl, C.sub.3 -C.sub.6 cycloalkylcarbonyl, C.sub.3 -C.sub.6 halocycloalkylcarbonyl, C.sub.1 -C.sub.6 alkylcarbonyl C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 haloalkylcarbonyl C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 alkylcarbonyl C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 haloalkylcarbonyl C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 alkoxycarbonyl, C.sub.1 -C.sub.6 haloalkoxycarbonyl, C.sub.3 -C.sub.10 cycloalkoxycarbonyl, carboxy C.sub.1 -C.sub.5 alkyl, C.sub.1 -C.sub.10 alkoxycarbonyl C.sub.1 -C.sub.5 alkyl, C.sub.1 -C.sub.10 haloalkoxycarbonyl C.sub.1 -C.sub.5 alkyl, C.sub.1 -C.sub.10 alkoxycarbonyl C.sub.1 -C.sub.5 haloalkyl, C.sub.1 -C.sub.10 haloalkoxycarbonyl C.sub.1 -C.sub.5 haloalkyl, C.sub.3 -C.sub.10 cycloalkoxycarbonyl C.sub.1 -C.sub.5 alkyl, C.sub.3 -C.sub.10 halocycloalkoxycarbonyl C.sub.1 -C.sub.5 alkyl, C.sub.3 -C.sub.10 halocycloalkoxycarbonyl C.sub.1 -C.sub.5 haloalkyl, C.sub.3 -C.sub.10 cycloalkoxycarbonyl C.sub.1 -C.sub.5 haloalkyl, C.sub.1 -C.sub.6 alkoxy C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 alkoxy C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 haloalkoxy C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 haloalkoxy C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 alkylthio C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 alkylthio C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 haloalkylthio C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 haloalkylthio C.sub.1 -C.sub.6 haloalkyl, cyano C.sub.1 -C.sub.4 alkyl, aryl that may have substituent(s), aryl C.sub.1 -C.sub.3 alkyl that may have substituent(s), arylcarbonyl that may have substituent(s) or SR.sup.18 ;R.sup.10 represents hydrogen, C.sub.1 -C.sub.10 alkyl, C.sub.1 -C.sub.10 haloalkyl, C.sub.3 -C.sub.8 alkenyl, C.sub.3 -C.sub.8 haloalkenyl, C.sub.3 -C.sub.8 alkynyl, C.sub.3 -C.sub.8 haloalkynyl, C.sub.3 -C.sub.10 cycloalkyl, C.sub.3 -C.sub.10 halocycloalkyl, C.sub.3 -C.sub.10 cycloalkenyl, C.sub.3 -C.sub.10 halocycloalkenyl, C.sub.1 -C.sub.5 alkylcarbonyl, C.sub.1 -C.sub.5 haloalkylcarbonyl, C.sub.3 -C.sub.6 cycloalkylcarbonyl, C.sub.3 -C.sub.6 halocycloalkylcarbonyl, C.sub.1 -C.sub.6 alkylcabonyl C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 haloalkylcarbonyl C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 alkylcabonyl C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 haloalkylcarbonyl C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 alkoxycarbonyl, C.sub.1 -C.sub.6 haloalkoxycarbonyl, C.sub.3 -C.sub.10 cycloalkoxycarbonyl, carboxy C.sub.1 -C.sub.5 alkyl, C.sub.1 -C.sub.10 alkyoxycarbonyl C.sub.1 -C.sub.5 alkyl, C.sub.1 -C.sub.10 haloalkoxycarbonyl C.sub.1 -C.sub.5 alkyl, C.sub.1 -C.sub.10 alkoxycarbonyl C.sub.1 -C.sub.5 haloalkyl, C.sub.1 -C.sub.10 haloalkoxycarbonyl C.sub.1 -C.sub.5 haloalkyl, C.sub.3 -C.sub.10 cycloalkoxycarbonyl C.sub.1 -C.sub.5 alkyl, C.sub.3 -C.sub.10 halocycloalkoxycarbonyl C.sub.1 -C.sub.5 alkyl, C.sub.3 -C.sub.10 halocycloalkoxycarbonyl C.sub.1 -C.sub.5 haloalkyl, C.sub.3 -C.sub.10 cycloalkoxycarbonyl C.sub.1 -C.sub.5 haloalkyl, C.sub.1 -C.sub.6 alkoxy C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 alkoxy C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 haloalkoxy C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 haloalkoxy C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 alkylthio C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 alkylthio C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 haloalkylthio C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 haloalkylthio C.sub.1 -C.sub.6 haloalkyl, cyano C.sub.1 -C.sub.4 alkyl, aryl that may have substituent(s), aryl C.sub.1 -C.sub.3 alkyl that may have substituent(s), arylcarbonyl that may have substituent(s), SR.sup.18, SOR.sup.19 or SO.sub.2 R.sup.20 ;R.sup.11 represents hydrogen, C.sub.1 -C.sub.10 alkyl, C.sub.1 -C.sub.10 haloalkyl, C.sub.3 -C.sub.8 cycloalkyl, C.sub.3 -C.sub.8 halocycloalkyl, N(R.sup.21)(R.sup.22), N.dbd.C(R.sup.21)(R.sup.22), carboxy C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.5 alkoxycarbonyl C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.5 haloalkoxycarbonyl C.sub.1 -C.sub.3 alkyl, C.sub.3 -C.sub.6 cycloalkoxycarbonyl C.sub.1 -C.sub.3 alkyl or C.sub.3 -C.sub.8 alkenyloxycarbonyl C.sub.1 -C.sub.3 alkyl;R.sup.12 represents hydrogen, chlorine, C.sub.1 -C.sub.5 alkyl, C.sub.1 -C.sub.5 haloalkyl, C.sub.3 -C.sub.6 cycloalkyl, C.sub.3 -C.sub.6 halocycloalkyl or N(R.sup.23)(R.sup.24);R.sup.13 represents chlorine, C.sub.1 -C.sub.10 alkyl, C.sub.1 -C.sub.10 haloalkyl, N(R.sup.25)(R.sup.26) or OR.sup.27 ;R.sup.14 represents hydrogen, halogen or C.sub.1 -C.sub.3 alkyl;R.sup.15 represents hydrogen, COOR.sup.28 or CN;R.sup.16 represents hydrogen, halogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.3 -C.sub.5 cycloalkyl or C.sub.3 -C.sub.5 halocycloalkyl;R.sup.17 represents hydrogen, C.sub.1 -C.sub.10 alkyl, C.sub.1 -C.sub.10 haloalkyl, C.sub.3 -C.sub.6 cycloalkyl, C.sub.3 -C.sub.6 halocycloalkyl, C.sub.3 -C.sub.5 alkenyl, C.sub.3 -C.sub.5 haloalkenyl, C.sub.3 -C.sub.5 alkynyl, C.sub.3 -C.sub.5 haloalkynyl, carboxy C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.5 alkoxycarbonyl C.sub.1 -C.sub.3 alkyl, aryl that may have substituent(s) or aryl C.sub.1 -C.sub.3 alkyl that may have substituent(s);R.sup.18 represents C.sub.1 -C.sub.10 alkyl, C.sub.1 -C.sub.10 haloalkyl or aryl that may have substituent(s);R.sup.19 represents C.sub.1 -C.sub.10 alkyl, C.sub.1 -C.sub.10 haloalkyl, C.sub.3 -C.sub.8 cycloalkyl, C.sub.3 -C.sub.8 halocycloalkyl or aryl that may have substituent(s);R.sup.20 represents C.sub.1 -C.sub.10 alkyl, C.sub.1 -C.sub.10 haloalkyl, C.sub.3 -C.sub.8 cycloalkyl, C.sub.3 -C.sub.8 halocycloalkyl or aryl that may have substituent(s);R.sup.21 represents hydrogen or C.sub.1 -C.sub.5 alkyl;R.sup.22 represents hydrogen, C.sub.1 -C.sub.5 alkyl, C.sub.1 -C.sub.5 haloalkyl or aryl that may have substituent(s);R.sup.23 represents hydrogen, C.sub.1 -C.sub.10 alkyl, C.sub.1 -C.sub.10 haloalkyl, C.sub.3 -C.sub.10 cycloalkyl, C.sub.3 -C.sub.10 halocycloalkyl or aryl that may have substituent(s);R.sup.24 represents hydrogen, C.sub.1 -C.sub.10 alkyl, or C.sub.1 -C.sub.10 haloalkyl;R.sup.25 represents hydrogen, C.sub.1 -C.sub.5 alkyl or C.sub.1 -C.sub.5 haloalkyl;R.sup.26 represents hydrogen, C.sub.1 -C.sub.10 alkyl, or C.sub.1 -C.sub.10 haloalkyl;R.sup.27 represents C.sub.1 -C.sub.10 alkyl;R.sup.28 represents hydrogen, C.sub.1 -C.sub.10 alkyl, C.sub.1 -C.sub.10 haloalkyl, C.sub.3 -C.sub.10 cycloalkyl, C.sub.3 -C.sub.10 halocycloalkyl or aryl that may have substituent(s); andG represents G-1, or G-3 given in the formula: ##STR37## wherein E.sup.1, E.sup.2, E.sup.3, E.sup.4, E.sup.5, E.sup.6, E.sup.7, E.sup.8, E.sup.9, E.sup.10, E.sup.11, E.sup.12, E.sup.13 or E.sup.14 each represent hydrogen, halogen or C.sub.1 -C.sub.3 alkyl.