Patent ID: 7517995
Filing Date: 2009-04-14
Classification: A61P,C07D

Abstract:
1. A compound of the formula (I), wherein R R or an optionally substituted group selected from among C R or R or R or R or R wherein X and Y may be linked to the same or different atoms of G, and X denotes a bond or an optionally substituted group selected from among C or X together with R Y denotes a bond or optionally substituted C Q denotes an optionally substituted group selected from among C Q together with R R or in each case two of the substituents R G denotes a saturated, partially saturated or unsaturated ring system consisting of 3-10 C atoms, wherein optionally up to 6 C atoms are replaced by heteroatoms selected from among nitrogen, oxygen and sulphur; R or a group selected from among ═O, NR n denotes 1, 2 or 3; R or in each case two of the substituents R with the proviso that the following compounds are excluded: a) 1,1-dimethyl-3-(4-phenyl-4,7-dihydro-3-thia-1,4,5-triaza-cyclopenta[a]pentalen-2-yl) -urea b) (4-phenyl-4,7-dihydro-3 -thia- 1 ,4,5-triaza-cyclopenta[a]pentalen-2-yl)-urea c) 1-(2-dimethylamino-ethyl)-3-(4-phenyl-4,7-dihydro-3-thia-1,4,5-triaza -cyclopenta[a]pentalen-2-yl)-urea d) 1-(2-dimethylamino-ethyl)-1-methyl-3-(4-phenyl-4,7-dihydro-3-thia-1,4,5-triaza -cyclopenta[a]pentalen-2-yl)-urea e) 4-methyl-piperazine-1-carboxylic acid (4-phenyl-4,7-dihydro-3-thia-1,4,5-triaza -cyclopenta[a]pentalen-2-yl)-amide f) 1-[4-(2-chloro-phenyl)-4,7-dihydro-3-thia-1,4,5-triaza-cyclopenta[a]pentalen-2-yl]-3-(2-dimethylamino-ethyl)-urea g) 3-[4-(2-chloro-phenyl)-4,7-dihydro-3-thia-1,4,5 -triaza-cyclopenta[a]pentalen-2-yl]-1-(2-dimethylamino-ethyl)- 1-methyl-urea h) 1-[4-(2-chloro-phenyl)-4,7-dihydro-3-thia-1,4,5-triaza-cyclopenta[a]pentalen-2-yl]-3-methyl-urea i) 1-[4-(2-chloro-phenyl)-4,7-dihydro-3-thia-1,4,5-triaza-cyclopenta[a]pentalen-2-yl]-3-(2-imidazol-1-yl-ethyl)-urea j) 3-4-(2-chloro-phenyl)-4,7-dihydro-3-thia-1,4,5-triaza-cyclopenta[a]pentalen-2-yl]-1,1-dimethyl-urea, and k) piperidine-1-carboxylic acid (4-phenyl-4,7-dihydro-3-thia-1,4,5-triaza -cyclopenta[a]pentalen-2-yl)-amide.