Patent ID: 6297374
Filing Date: 2001-10-02
Classification: A01N,C07D,C07F

Abstract:
A compound of the formula ##STR701##in whichn represents 0 or 1,R.sup.1, R.sup.2, R.sup.5 and R.sup.6 independently represent a hydrogen atom or an alkyl group, R.sup.3 and R.sup.4 independently represent a hydrogen atom, a hydroxy group or an alkyl group,where n represents 1, then R.sup.2 may form a single bond, together with R.sup.5,X represents a sulfur atom, an oxygen atom,##STR702##or ##STR703##R.sup.7 represents a hydrogen atom, a halogen atom,a hydroxy group, an alkoxy group,a benzyloxy group, an alkyl group which may be substituted by at least one member selected from the class consisting of alkoxy groups, alkylthio groups, a cyano group, halogen atoms, dialkylamino groups and trialkylsilyl,an alkenyl group which may be substituted by a halogen atom, an alkynyl group which may be substituted by a halogen atom, a phenyl group which may be substituted by an alkyl group and/or a halogen atom,a benzyl group which may be substituted by at least one member selected from the class consisting of a methyl group, a methoxy group, halogen atoms, halomethyl groups, halomethoxy groups and a nitro group, a formyl group,an alkenylcarbonyl group, an alkylcarbonyl group which may be substituted by at least one member selected from the class consisting of alkoxy groups, a phenoxy group, alkylthio groups, and halogen atoms, a benzoyl group which may be substituted by at least one member selected from the class consisting of halogen atoms, alkyl groups, halomethyl groups, alkoxy groups, haloalkoxy groups and a nitro group, a benzylcarbonyl group which may be substituted by an alkyl group and/or a halogen atom, an alkoxycarbonyl group which may be substituted by a halogen atom, an alkylthiocarbonyl group,a phenoxycarbonyl group which may be substituted by at least one member selected from the class consisting of methyl group, a methoxy group, halomethyl group, halomethoxy groups, halogen atoms anda nitro group, a phenylthiocarbonyl group which may be substituted by a halogen atom and/or an alkyl group,a benzyloxycarbonyl group,a monoalkyl- or dialkyl-aminocarbonyl group,a phenylaminocarbonyl group which may be substituted by at least one member selected from the class consisting of alkyl groups, haloalkyl groups and halogen atoms, a benzoylaminocarbonyl group which may be substituted by an alkyl group and/or a halogen atom,a phenylsulfonylaminocarbonyl group which may be substituted by an alkyl group and/or a halogen atom, a phenylthio group which may be substituted by an alkyl group and/or a halogen atom,an alkylsulfonyl group which may be substituted by a halogen atom, a phenylsulfonyl group which may be substituted by at least one member selected from the class consisting of alkyl groups, halogen atoms and a nitro group, an alkylcarbonylmethyl group,a phenacyl group which may be substituted by a halogen atom and/or an alkyl groups,an organophosphono group, an organothionophosphono group,--CH.sub.2 W or --CO--W,W represents a 5 to 6 membered heterocyclic group, containing at least one hetero atom selected from the class consisting of an oxygen atom, a sulfur atom and a nitrogen atom, which may be substituted by at least one member selected from the class consisting of halogen atoms, alkyl groups and haloalkyl groups,R.sup.8 represents a hydrogen atom, an alkyl group, an aryl group or a benzyl group,Y represents a nitrogen atom or ##STR704##R.sup.9 represents a hydrogen atom, a halogen atom, a hydroxy group, an alkoxy group, a benzyloxy group, an alkyl group which may be substituted by at least one member selected from the class consisting of halogen atoms, a hydroxy group, alkoxy groups, alkylthio groups, a cyano group, mono- or di-alkylamino groups, alkylcarbonyl groups, alkoxycarbonyl groups and phenoxycarbonyl groups,an alkenyl group which may be substituted by a halogen atom, an alkynyl group, a phenyl group which may be substituted by an alkyl group and/or a halogen atom, an alkylcarbonyl group which may be substituted by a halogen atom, an alkenylcarbonyl group, a benzoyl group which may be substituted by at least one member selected from the class consisting of halogen atoms, alkyl groups and alkoxy groups,an alkoxycarbonyl group which may be substituted by a halogen atom,an alkkylthiocarbonyl group,a phenoxycarbonyl group which may be substituted by at least one member selected from the class consisting of halogen atoms, alkyl groups, alkoxy groups and a nitro group,a phenylthiocarbonyl group which may be substituted by an alkyl group and/or a halogen atom, a phenylthiocarbonyl group which may be substituted by an alkyl group and/or a halogen atom, a benzyloxycarbonyl group,a benzoylaminocarbonyl group which may be substituted by an alkyl group and/or a halogen atom,a phenylsulfonylaminocarbonyl group which may be substituted by an alkyl group and/or a halogen atom, an alkylsulfonylaminocarbonyl group,an alkylthio group,an alkylsulfonyl group which may be substituted by a halogen atom,a phenylthio group which may be substituted by an alkyl group and/or a halogen atom,a phenylsulfonyl group which may be substituted by an alkyl group and/or a halogen atom, in addition, R.sup.9 may form a bis-form of the formula (I), via a methylene group,R represents a hydrogen atom or an alkyl group, andz represents a 5 to 6 membered heterocyclic group containing at least one hetero atom selected from the class consisting of an oxygen atom, a sulfur atom and a nitrogen atom, which may be subsituted by at least one member selected from the class consisting of halogen atoms, alkyl groups, haloalkyl groups, a nitro group, a cyano group, alkoxy groups, alkylthio groups, alkylsulfinyl groups, alkylsulfonyl groups, alkenyl groups, haloalkoxy group, haloalkylthio groups, haloalkenyl groups, acylamino groups, haloacylamino groups, alkoxycarbonyl groups,a thiocyanato group, alkynyl groups, an amino group, alkylamino groups, dialkylamino groups,a carboxy group, a hydroxy group, a mercapto group, cycloalkyl groups, an oxo group,a thioxo group, haloalkenylthio groups, alkoxyalkyl groups, alkoxycarbonylamino groups,a carbamoyl group, acyl groups, alkylaminocarbonyl groups, dialklaminocarbonyl groups, a formyl group, aryl groups optionally substituted by a substituent selected from the class consisting of halogen atoms, alkyl groups, halogenoalkyl groups, alkoxy groups, a nitro group and a cyano group, aryloxy groups optionally substituted by a substituent as shown for the above aryl groups, andaralkyl groups optionally substituted by the same substituent as that shown for the aryl groups, provided that where R.sup.1, R.sup.2, R.sup.3, R.sup.4, R.sup.5 and R.sup.6 represent hydrogen atoms simultaneouly,X represents ##STR705##and Y represents ##STR706##then Z does not stand for a pyridyl group.