Patent ID: 8895741
Filing Date: 2014-11-25
Classification: C07D

Abstract:
1. A process for preparing a compound having the formula: the process comprising the steps of: combining a compound of formula (I): with a compound of formula (II): in a solvent in the presence of a base and a palladium catalyst, wherein A is selected from the group consisting of: B is selected from the group consisting of: Het-CH M-L is selected from the group consisting of: alternatively, L in M-L is a bond; M is selected from the group consisting of: Q is a borane having the formula —BY alternatively, Q is a BF Z is selected from the group consisting of: R R R R R R R R R m is 0, 1, 2, 3, or 4; n is 0, 1, 2, 3, or 4; and p, at each occurrence, independently is 0, 1, or 2.