Patent ID: 7812031
Filing Date: 2010-10-12
Classification: A61P,C07D

Abstract:
1. A compound of formula (I) wherein X is Ar is phenyl, a 5- or 6-membered heterocyclic ring containing 1, 2 or 3 heteroatoms independently selected from N, O or S, or a methylenedioxyphenyl group R is hydrogen or C Y is hydrogen or C W is hydrogen or C Z is hydroxyl, halogen, C or R and Y taken together with the nitrogen and carbon atoms to which they are attached form the following group or R and Z taken together form —(CH or Z and W taken together form an oxo group; Q is a 5- or 6-membered heterocyclic ring containing 1, 2 or 3 heteroatoms independently selected from N, O or S, or Q is the following group with the proviso that, if Q is a 5- or 6-membered heterocyclic ring containing 1, 2 or 3 heteroatoms as hereinbefore defined and said heterocyclic ring is optionally substituted with one or more groups independently selected from C W is hydrogen, and Z is hydroxyl, and R and Y together with the nitrogen and carbon atoms to which they are attached form the following group Ar is as defined above, then X cannot be C and pharmaceutically acceptable salts thereof.