Patent ID: 7241775
Filing Date: 2007-07-10
Classification: C07D

Abstract:
1. A compound of formula I, a pharmaceutically acceptable salt or a trifluoroacetate thereof wherein: R1, R2, R3 and R4 are each independently selected from the group consisting of H, F, Cl, Br, I, CN, NO R14 and R15 are each independently selected from the group consisting of H, or alkyl having 1, 2, 3, 4, 5, 6, 7 or 8 carbon atoms with none, some or all of the carbon atoms fluorinated and further having one or more CH R5 is selected from the group consisting of H, alkyl having 1, 2, 3, 4, 5, 6, 7 or 8 carbon atoms with none, some or all of the carbon atoms being fluorinated, cycloalkyl having 3, 4, 5, 6, 7 or 8 carbon atoms with none, some or all of the carbon atoms being fluorinated, COR20 and SO R6 is selected from the group consisting of H, OH, F, Cl, Br, alkyl having 1, 2, 3, 4, 5, 6, 7 or 8 carbon atoms with none, some or all of the carbon atoms being fluorinated, cycloalkyl having 3, 4, 5, 6, 7 or 8 carbon atoms with none, some or all of the carbon atoms being fluorinated, O-alkyl having 1, 2, 3, 4, 5, 6, 7 or 8 carbon atoms with none, some or all of the carbon atoms being fluorinated, and O-acyl having 1, 2, 3, 4, 5, 6, 7 or 8 carbon atoms with none, some or all of the carbon atoms being fluorinated; R7, R8 and R9 are each independently selected from the group consisting of H, F, Cl, Br, I, OH, alkyl having 1, 2, 3, 4, 5, 6, 7 or 8 carbon atoms with none, some or all of the carbon atoms being fluorinated, cycloalkyl having 3, 4, 5, 6, 7 or 8 carbon atoms with none, some or all of the carbon atoms being fluorinated, O-alkyl having 1, 2, 3, 4, 5, 6, 7 or 8 carbon atoms with none, some or all of the carbon atoms being fluorinated, O provided that at least one of the R7, R8 or R9 radicals in formula I is a -L-G group.