Patent ID: 6242647
Filing Date: 2001-06-05
Classification: A01N,C07C

Abstract:
A compound of formula I ##STR23##whereinR is hydrogen,C.sub.1 -C.sub.10 alkyl optionally substituted with one or more halogen,C.sub.3 -C.sub.6 cycloalkyl,C.sub.1 -C.sub.4 alkoxy,C.sub.1 -C.sub.4 haloalkoxy,(C.sub.1 -C.sub.4 -alkyl)SO.sub.x,(C.sub.1 -C.sub.4 haloalkyl)SO.sub.y,phenyl optionally substituted with one to three halogen,C.sub.1 -C.sub.4 alkyl,C.sub.1 -C.sub.4 haloalkyl,C.sub.1 -C.sub.4 alkoxy,C.sub.1 -C.sub.4 haloalkoxy,(C.sub.1 -C.sub.4 alkyl)SO.sub.x,(C.sub.1 -C.sub.4 haloalkyl)SO.sub.y,NO.sub.2 or CN groups, orphenoxy optionally substituted with one to three halogen,C.sub.1 -C.sub.4 alkyl,C.sub.1 -C.sub.4 haloalkyl,C.sub.1 -C.sub.4 alkoxy,C.sub.1 -C.sub.4 haloalkoxy,(C.sub.1 -C.sub.4 alkyl)SO.sub.x,(C.sub.1 -C.sub.4 haloalkyl)SO.sub.y,NO.sub.2 or CN groups;C.sub.3 -C.sub.12 cycloalkyl optionally substituted with one or more halogens,C.sub.1 -C.sub.6 alkyl,C.sub.1 -C.sub.4 haloalkyl,C.sub.1 -C.sub.4 alkoxy,C.sub.1 -C.sub.4 haloalkoxy,(C.sub.1 -C.sub.4 alkyl)SO.sub.x,(C.sub.1 -C.sub.4 haloalkyl)SO.sub.x,phenyl optionally substituted with one to three halogen,C.sub.1 -C.sub.4 alkylC.sub.1 -C.sub.4 haloalkyl,C.sub.1 -C.sub.4 alkoxy,C.sub.1 -C.sub.4 haloalkoxy,NO.sub.2 or CN groups, orphenoxy optionally substituted with one to three halogen,C.sub.1 -C.sub.4 alkyl,C.sub.1 -C.sub.4 haloalkyl,C.sub.1 -C.sub.4 alkoxy,C.sub.1 -C.sub.4 haloalkoxy,NO.sub.2 or CN groups; orphenyl optionally substituted with one or more halogen,C.sub.1 -C.sub.4 alkyl,C.sub.1 -C.sub.4 haloalkyl,C.sub.1 -C.sub.4 alkoxy,C.sub.1 -C.sub.4 haloalkoxy,NO.sub.2 or CN groups;with the proviso that when R is an optionally substituted phenyl, then m must be 1 or 2;R.sub.1 is R.sub.12 ;C.sub.1 -C.sub.10 alkyl optionally substituted with one or more halogen,hydroxy,phenyl optionally substituted with one or more halogen,C.sub.1 -C.sub.4 alkyl,C.sub.1 -C.sub.4 haloalkyl,C.sub.1 -C.sub.4 alkoxy,C.sub.1 -C.sub.4 haloalkoxy,NO.sub.2 or CN groups,C.sub.1 -C.sub.4 alkoxy,C.sub.1 -C.sub.4 haloalkoxy,(C.sub.1 -C.sub.4 alkyl)SO.sub.x,CONR.sub.8 R.sub.9,CO.sub.2 R.sub.10,R.sub.11,R.sub.12,C.sub.3 -C.sub.6 cycloalkyl optionally substituted with one to three halogen,C.sub.1 -C.sub.4 alkyl,C.sub.1 -C.sub.4 haloalkyl,C.sub.1 -C.sub.4 alkoxy,C.sub.1 -C.sub.4 haloalkoxy,NO.sub.2 or CN groups,phenyl optionally substituted with one or more halogen,C.sub.1 -C.sub.4 alkyl,C.sub.1 -C.sub.4 haloalkyl,C.sub.1 -C.sub.4 alkoxy,C.sub.1 -C.sub.4 haloalkoxy,NO.sub.2 or CN groups, orpyridyl optionally substituted with one or more halogen,C.sub.1 -C.sub.4 alkyl,C.sub.1 -C.sub.4 haloalkyl,C.sub.1 -C.sub.4 alkoxy,C.sub.1 -C.sub.4 haloalkoxy,NO.sub.2 or CN groups;C.sub.2 -C.sub.10 alkenyl optionally substituted with one or more halogen,hydroxy,C.sub.1 -C.sub.4 alkoxy,(C.sub.1 -C.sub.4 alkyl)SO.sub.x,CONR.sub.8 R.sub.9,CO.sub.2 R.sub.10,R.sub.11,R.sub.12,C.sub.3 -C.sub.6 cycloalkyl optionally substituted with one to three halogen,C.sub.1 -C.sub.4 alkyl,C.sub.1 -C.sub.4 halo-alkyl,C.sub.1 -C.sub.4 alkoxy,C.sub.1 -C.sub.4 haloalkoxy,NO.sub.2 or CN groups,phenyl optionally substituted with one or more halogen,C.sub.1 -C.sub.4 alkyl,C.sub.1 -C.sub.4 haloalkyl,C.sub.1 -C.sub.4 alkoxy,C.sub.1 -C.sub.4 haloalkoxy,NO.sub.2 or CN groups, orpyridyl optionally substituted with one or more halogen,C.sub.1 -C.sub.4 alkyl,C.sub.1 -C.sub.4 haloalkyl,C.sub.1 -C.sub.4 alkoxy,C.sub.1 -C.sub.4 haloalkoxy,NO.sub.2 or CN groups;C.sub.2 -C.sub.10 alkynyl optionally substituted with one or more halogen,hydroxy,C.sub.1 -C.sub.4 alkoxy,(C.sub.1 -C.sub.4 alkyl)SO.sub.x,CONR.sub.8 R.sub.9,CO.sub.2 R.sub.10,R.sub.11,R.sub.12,C.sub.3 -C.sub.6 cycloalkyl optionally substituted with one to three halogen,C.sub.1 -C.sub.4 alkyl,C.sub.1 -C.sub.4 halo-alkyl,C.sub.1 -C.sub.4 alkoxy,C.sub.1 -C.sub.4 haloalkoxy,NO.sub.2 or CN groups,phenyl optionally substituted with one or more halogen,C.sub.1 -C.sub.4 alkyl,C.sub.1 -C.sub.4 haloalkyl,C.sub.1 -C.sub.4 alkoxy,C.sub.1 -C.sub.4 haloalkoxy,NO.sub.2 or CN groups, orpyridyl optionally substituted with one or more halogen,C.sub.1 -C.sub.4 alkyl,C.sub.1 -C.sub.4 haloalkyl,C.sub.1 -C.sub.4 alkoxy,C.sub.1 -C.sub.4 haloalkoxy,NO.sub.2 or CN groups; orC.sub.3 -C.sub.12 cycloalkyl optionally substituted with one or more halogen,hydroxy,C.sub.1 -C.sub.4 alkoxy,(C.sub.1 -C.sub.4 alkyl)SO.sub.x,CONR.sub.8 R.sub.9,CO.sub.2 R.sub.10,R.sub.11,R.sub.12,C.sub.3 -C.sub.6 cycloalkyl optionally substituted with one to three halogen,C.sub.1 -C.sub.4 alkyl,C.sub.1 -C.sub.4 halo-alkyl,C.sub.1 -C.sub.4 alkoxy,C.sub.1 -C.sub.4 haloalkoxy,NO.sub.2 or CN groups,phenyl optionally substituted with one or more halogen,C.sub.1 -C.sub.4 alkyl,C.sub.1 -C.sub.4 haloalkyl,C.sub.1 -C.sub.4 alkoxy,C.sub.1 -C.sub.4 haloalkoxy,NO.sub.2 or CN groups, orpyridyl optionally substituted with one or more halogen,C.sub.1 -C.sub.4 alkyl,C.sub.1 -C.sub.4 haloalkyl,C.sub.1 -C.sub.4 alkoxy,C.sub.1 -C.sub.4 haloalkoxy,NO.sub.2 or CN groups;phenyl optionally substituted with one or more halogen,C.sub.1 -C.sub.4 alkyl,C.sub.1 -C.sub.4 haloalkyl,C.sub.1 -C.sub.4 alkoxy,C.sub.1 -C.sub.4 haloalkoxy,NO.sub.2 or CN groups, orpyridyl optionally substituted with one or more halogen,C.sub.1 -C.sub.4 alkyl,C.sub.1 -C.sub.4 haloalkyl,C.sub.1 -C.sub.4 alkoxy,C.sub.1 -C.sub.4 haloalkoxy,NO.sub.2 or CN groups;R.sub.2 is hydrogen or C.sub.1 -C.sub.4 alkyl;R.sub.3, R.sub.4, R.sub.5, R.sub.6, and R.sub.7 are each independently hydrogen, halogen, CN, NO.sub.2, C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 alkoxy, C.sub.1 -C.sub.6 haloalkoxy, or phenyl optionally substituted with one to three halogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy, (C.sub.1 -C.sub.4 alkyl)SO.sub.x, (C.sub.1 -C.sub.4 haloalkyl)SO.sub.y, NO.sub.2 or CN groups,with the proviso that at least one of R.sub.3, R.sub.4, R.sub.5, R.sub.6 or R.sub.7 must be phenyl optionally substituted with one to three halogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy, (C.sub.1 -C.sub.4 alkyl)SO.sub.x, (C.sub.1 -C.sub.4 haloalkyl)SO.sub.x, NO.sub.2 or CN groups;x and y are each independently 0, 1 or 2;m is an integer of 0, 1 or 2;R.sub.8, R.sub.9 and R.sub.10 are each independently hydrogen or C.sub.1 -C.sub.4 alkyl;R.sub.11 is NR.sub.13 R.sub.14, ##STR24##R.sub.12 is ##STR25##R.sub.13, R.sub.14, and R.sub.15 are each independently hydrogen or C.sub.1 -C.sub.4 alkyl;R.sub.16 is hydrogen, halogen or C.sub.1 -C.sub.4 alkyl;X is O, S or NR.sub.15 ;r is an integer of 0 or 1;p and q are each independently an integer of 0, 1, 2, or 3 with the proviso that only one of p, q, or r can be 0 and with the further proviso that the sum of p+q+r must be 4, 5 or 6; andx is an integer of 0, 1 or 2; orthe acid addition salts thereof.