Patent ID: 6011032
Filing Date: 2000-01-04
Classification: A61P,C07D

Abstract:
N-heterocyclyl-1-aryloxyalkyl-4-piperidinamines selected from those of formula I ##STR100## in which the substituents are defined as follows: R.sub.1 to R.sub.4, which may be identical or different, represent:hydrogenbranched or unbranched alkyl containing 1 to 4 carbon atomsbranched or unbranched alkyloxy containing 1 to 4 carbon atomshalogennitrohydroxyltrifluoromethyl or trifluoromethoxy,R.sub.5 represents:hydrogenbranched or unbranched alkyl containing 1 to 6 carbon atomsbranched or unbranched phenylalkyl containing 7 to 12 carbons, which can be substituted on the phenyl with one or two radicals defined as R.sub.1,W and X represent:oxygen or sulfur,Y represents:polymethylene group containing 2 to 6 carbon atoms, or--CH.sub.2 --CH(OH)--CH.sub.2 --n is 0, when the compounds contain an asymmetric carbon, in the form of their racemic mixtures or the pure enantiomers or mixtures thereof, and in any case therapeutically-acceptable inorganic or organic salts and hydrates thereof.