Patent ID: 8119795
Filing Date: 2012-02-21
Classification: A61P,C07D

Abstract:
1. A compound of the formula I in which R R R R R Y denotes OH or SH, A, A′ each, independently of one another, denote unbranched or branched alkyl having 1-10 C atoms, in which one, two or three CH A and A′ together also denote an alkylene chain having 2, 3, 4, 5 or 6 C atoms, in which a CH Alk denotes alkenyl having 2-6 C atoms, R R cycloalkylalkylene having 4-10 C atoms, Alk or R R Ar denotes phenyl, naphthyl or biphenyl, each of which is unsubstituted or mono-, di- or trisubstituted by Hal, A, XR Ar′ denotes phenyl, naphthyl or biphenyl, each of which is mono-, di- or trisubstituted by Hal, A, XR Het denotes a mono- or bicyclic saturated, unsaturated or aromatic heterocycle having 1 to 4 N, O and/or S atoms, which may be unsubstituted or mono-, di- or trisubstituted by Hal, A, XR Het′ denotes a mono- or bicyclic saturated, unsaturated or aromatic heterocycle having 1 to 4 N, O and/or S atoms, which may be unsubstituted or mono-, di- or trisubstituted by Hal, A, XR and/or in which a ring nitrogen may be substituted by —O Het″ denotes a monocyclic aromatic heterocycle having 1 to 3 N, O and/or S atoms, Het′″ denotes a monocyclic saturated heterocycle having 1 to 3 N, O and/or S atoms, X denotes unbranched or branched alkylene having 1-10 C atoms, in which one, two or three CH R Hal denotes F, Cl, Br or I, m denotes 0, 1 or 2, n denotes 0, 1, 2, 3 or 4, o denotes 1, 2 or 3, or pharmaceutically usable salts, tautomers or stereoisomers thereof, including mixtures thereof in all ratios.