Patent ID: 6936614
Filing Date: 2005-08-30
Classification: C07D

Abstract:
1. A compound represented by A: wherein X represents (C(R)2)n; Z represents 0 or H2; R represents independently for each occurrence H, alkyl, cycloalkyl, aryl, heteroaryl, aralkyl, or heteroaralkyl; or any two geminal instances of R taken together represent O; R1 represents optionally substituted aryl or heteroaryl; wherein any optional substituent is selected from the group consisting of alkyl, cycloalkyl, fluoro, chloro, bromo, iodo, hydroxy, alkoxy, acyloxy, acyl, nitro, nitroso, amino, acylamino, sulfonyl, and sulfonylamino; R2 represents optionally substituted aryl, heteroaryl, arylalkyl, heteroarylalkyl, di(aryl)alkyl, or di(heteroaryl)alkyl; wherein any optional substituent is selected from the group consisting of alkyl, cycloalkyl, fluoro, chloro, bromo, iodo, hydroxy, alkoxy, acyloxy, acyl, nitro, nitroso, amino, acylamino, sulfonyl, and sulfonylamino; m is 0, 1, 2, or 3; n is 1, 2, or 3; and the stereochemical configuration at any stereocenter of compound represented by A is R, S, or a mixture of these configurations.