Patent ID: 6057270
Filing Date: 2000-05-02
Classification: C07D

Abstract:
Substituted pyrazol derivatives of the general formula (I) ##STR113## in which R.sup.1 =C.sub.1 -C.sub.4 alkyl,R.sup.2 =C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 - alkylthio, C.sub.1 -C.sub.4 alkoxy; or C.sub.1-C.sub.4 alkyl, C.sub.1 -C.sub.4 alkylthio, C.sub.1 -C.sub.4 alkoxy all substituted one or more times with halogen,R.sup.1 and R.sup.2 together form the group --(CH.sub.2).sub.m --,R.sup.3 =hydrogen or halogen,R.sup.4 =hydrogen or C.sub.1 -C.sub.4 alkyl,R.sup.5 =hydrogen, nitro, cyano or the groups --COOR.sup.7, ##STR114## R.sup.6 = ##STR115## R.sup.7, R.sup.8 and R.sup.9, independent of one another, are hydrogen or C.sub.1 -C.sub.4 alkyl,R.sup.8 and R.sup.9, together with the adjacent nitrogen atom, form a 5-membered or 6-membered saturated heterocyclic ring,R.sup.10 =hydrogen, C.sub.1 -C.sub.4 alkyl, or a C.sub.1 -C.sub.4 alkyl substituted one ore more times by halogen,R.sup.11 =hydrogen, C.sub.1 -C.sub.6 alkyl, C.sub.3 -C.sub.6 cycloalkyl, C.sub.2 -C.sub.6 alkenyl, C.sub.3 -C.sub.6 alkynyl; or C.sub.1 -C.sub.6 alkyl, C.sub.3 -C.sub.6 cycloalkyl, C.sub.2 -C.sub.6 alkenyl, C.sub.3 -C.sub.6 alkynyl all substituted similarly or differently one or more times by halogen, hydroxy or C.sub.1 -C.sub.4 alkoxy; or C.sub.2 -C.sub.8 alkyl, C.sub.3 -C.sub.6 cycloalkyl, C.sub.3 -C.sub.8 alkenyl, C.sub.3 -C.sub.6 alkynyl all interrupted times by oxygen; or the group OR.sup.12,R.sup.12 =C.sub.1 -C.sub.6 alkyl, C.sub.3 -C.sub.6 cycloalkyl, C.sub.2 -C.sub.6 alkenyl, C.sub.3 -C.sub.6 alkynyl; C.sub.1 -C.sub.6 alkyl substituted similarly or differently one or more times by halogen, hydroxy or by C.sub.1 -C.sub.4 alkoxyY=oxygen, sulphur, --N--OR.sup.13 and ##STR116## R.sup.13 =hydrogen, C.sub.1 -C.sub.6 alkyl, C.sub.3 -C.sub.6 cycloalkyl, C.sub.2 -C.sub.6 alkenyl, C.sub.3 -C.sub.6 alkynyl; C.sub.1 -C.sub.6 alkyl, C.sub.3 -C.sub.6 cycloalkyl, C.sub.2 -C.sub.6 alkenyl, C.sub.3 -C.sub.6 alkynyl all substituted similarly differently one or more times by halogen, cyano, hydroxy or C.sub.1 -C.sub.4 alkoxy; C.sub.2 -C.sub.8 alkyl, C.sub.3 -C.sub.8 cycloalkyl, C.sub.3 -C.sub.8 alkenyl, C.sub.3 -C.sub.8 alkynyl all interrupted one or more times by oxygen; C.sub.1 -C.sub.4 alkoxycarbonyl-C.sub.1 -C.sub.4 alkyl, which can optionally be substituted by halogen atoms; C.sub.1 -C.sub.4 alkoxycarbonyl-C.sub.2 -C.sub.4 alkenyl, which can optionally be substituted by halogen atoms; C.sub.1 -C.sub.4 alkoxycarbonyl,R.sup.14 and R.sup.15, independent of one another, are hydrogen, halogen, cyano, carboxyl, formyl, C.sub.1 -C.sub.6 alkyl, C.sub.3 -C.sub.6 cycloalkyl, C.sub.2 -C.sub.6 alkenyl, C.sub.3 -C.sub.6 alkynyl; C.sub.1 -C.sub.6 alkyl, C.sub.3 C.sub.6 cycloalkyl, C.sub.2 -C.sub.6 alkenyl, C.sub.3 -C.sub.6 alkynyl all substituted similarly differently one or more times by halogen, cyano, hydroxy or C.sub.1 -C.sub.4 alkoxy; C.sub.2 -C.sub.8 alkyl, C.sub.3 -C.sub.8 cycloalkyl, C.sub.3 -C.sub.8 alkenyl, C.sub.3 -C.sub.8 alkynyl all interrupted one times by oxygen; C.sub.1 -C.sub.4 alkoxycarbonyl-C.sub.1 -C.sub.4 alkyl, which can optionally be substituted by halogen atoms; C.sub.1 -C.sub.4 alkoxycarbonyl-C.sub.2 -C.sub.4 alkenyl, which can optionally be substituted by halogen atoms; C.sub.1 -C.sub.4 alkoxycarbonyl, C.sub.1 -C.sub.4 alkoxy or C.sub.1 -C.sub.4 alkylthio,R.sup.14 and R.sup.15 together with the carbon atom form a saturated carbocyclic C.sub.3 -C.sub.6 ring which can be interrupted one or more times by oxygen or sulphur,X=oxygen or sulphur.