Patent ID: 6130225
Filing Date: 2000-10-10
Classification: A01N,C07D

Abstract:
A substituted p-trifluoromethylphenyluracil of the formula (I) ##STR45## wherein R.sup.1 represents hydrogen, cyano or halogen,R.sup.2 represents a grouping A.sup.1 -A.sup.2 -A.sup.3 whereinA.sup.1 represents --SO.sub.2 --, --CO-- or a grouping --N-A.sup.4 - wherein A.sup.4 represents hydrogen, hydroxyl, alkyl, alkenyl, alkynyl, alkoxy, aryl, alkylsulphonyl or arylsulphonyl,A.sup.2 represents a single bond, represents O, S, --SO--, --SO.sub.2 --, --CO-- or the grouping --N-A.sup.4 - wherein A.sup.4 represents hydrogen, hydroxyl, alkyl, alkoxy, aryl, alkylsulphonyl or arylsulphonyl, orA.sup.2 represents alkanediyl, alkenediyl, azaalkenediyl, alkynediyl, cycloalkanediyl, cycloalkenediyl or phenylene, each of which is unsubstituted or substituted by halogen,A.sup.3 represents hydrogen, hydroxyl, mercapto, amino, cyano, isocyanato, thiocyanato, nitro, carboxyl, carbamoyl, thiocarbamoyl, sulpho, chlorosulphonyl, halogen, represents alkyl, alkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl, alkylamino, dialkylamino, alkoxycarbonyl or dialkoxy(thio)phosphoryl, each of which is unsubstituted or substituted by halogen or alkoxy, represents alkenyl, alkenyloxy, alkenylamino, alkylideneamino, alkenyloxycarbonyl, alkynyl, alkynyloxy, alkynylamino or alkynyloxycarbonyl, each of which is unsubstituted or substituted by halogen, represents cycloalkyl, cycloalkyloxy, cycloalkylalkyl, cycloalkylalkoxy, cycloalkylideneamino, cycloalkyloxycarbonyl or cycloalkylalkoxycarbonyl, each of which is unsubstituted or substituted by a compound selected from the group consisting of halogen, cyano, carboxyl, alkyl and alkoxycarbonyl, or represents aryl, aryloxy, aralkyl, arylalkoxy, aryloxycarbonyl or arylalkoxycarbonyl, each of which is unsubstituted or substituted by one or more compounds selected from the group consisting of nitro, cyano, carboxyl, halogen, alkyl, halogenoalkyl, alkyloxy, halogenoalkyloxy and alkoxycarbonyl, orA.sup.3 represents in each case fully or partially hydrogenated pyrrolyl, pyrazolyl, imidazolyl, triazolyl, furyl, oxiranyl, oxetanyl, dioxolanyl, thienyl, oxazolyl, isoxazolyl, thiazolyl, isothiazolyl, oxadiazolyl, thiadiazolyl, pyridinyl, pyrimidinyl, triazinyl, pyrazolylalkyl, furylalkyl, thienylalkyl, oxazolylalkyl, isoxazolalkyl, thiazolalkyl, pyridinylalkyl, pyrimidinylalkyl, pyrazolylalkoxy, furylalkoxy, represents perhydropyranylalkoxy or pyridylalkoxy,R.sup.3 represents hydrogen, halogen or unsubstituted or halogen-substituted alkyl,R.sup.4 represents unsubstituted or halogen-substituted alkyl, andR.sup.5 represents hydrogen, amino or unsubstituted or hydroxyl-, cyano-, halogen- or alkoxy-substituted alkyl.