Patent ID: 6197963
Filing Date: 2001-03-06
Classification: C07H

Abstract:
A compound having the structure: ##STR29##wherein;R.sub.1, R.sub.2, R.sub.3, R.sub.4, and R.sub.5 are, independently, H, OH, OCH.sub.3, O--(CH.sub.2).sub.n NH.sub.2, O--(CH.sub.2).sub.n OH, O--(CH.sub.2).sub.n NHC(O)CH.sub.3, O--(CH.sub.2).sub.n -indole, O-(benzyl), O--(CH.sub.2).sub.n (imidazole), pyridine, p-fluoro-benzyl, CH.sub.2 -.beta.-naphthyl, CH.sub.2 -.alpha.-naphthyl, --(CH.sub.2).sub.n -indole, --CH.sub.2 Ph-OH,--CH.sub.2 -picolyl, --NH(CH.sub.2).sub.5 NH.sub.2, --NH(CH.sub.2).sub.3 NH(CO)CH.sub.3, or --NH(CH.sub.2).sub.5 OH, --NH(CH.sub.2).sub.6 OH,at least one of R.sub.2, R.sub.3, and R.sub.4, is OCH.sub.3, O--(CH.sub.2).sub.n NH.sub.2, O--(CH.sub.2).sub.n OH, O--(CH.sub.2).sub.n NHC(O)CH.sub.3, O--(CH.sub.2).sub.n -indole, O--(CH.sub.2)(imidazole), pyridine, p-fluoro-benzyl, CH.sub.2 -.beta.-naphthvl, CH.sub.2 -.alpha.-naphthyl, --(CH.sub.2).sub.n -indole, --CH.sub.2 Ph-OH,--CH.sub.2 -picolyl, --NH(CH.sub.2).sub.5 NH.sub.2, --NH(CH.sub.2).sub.3 NH(CO)CH.sub.3, or --NH(CH.sub.2).sub.5 OH, --NH(CH.sub.2).sub.6 OH, andn is 1, 2, 3, 4, 5, or 6.