Patent ID: 7368566
Filing Date: 2008-05-06
Classification: A61P,C07D

Abstract:
1. A process for preparing a compound of Formula (I): from a benzazepine-phenol of Formula (II): wherein the benzazepine-phenol of Formula (II) is prepared by a process comprising converting a compound of Formula (III): to a compound of Formula (IV): wherein: R R R A is H, C R each R R R R R W is —(CHR U is absent or CO, CR G is NR R R R R R R R Q R′ is H, C R″ is R′, —C(O)R′ or —C(O)OR′; R′″ is H, C R a is 0, 1 or 2; b is 0, 1 or 2; k is 0, 1 or 2; m is 1 or 2; r is 0, 1 or 2; s is 0, 1 or 2; u is 0 or 1; and v is 0 or 1; or a pharmaceutically acceptable salt thereof.