Patent ID: 6432879
Filing Date: 2002-08-13
Classification: A01N,C07D

Abstract:
A phenyluracil compound of the formula (I), in whichn represents the number 0, 1, 2 or 3, Q represents O, S, SO, SO2, NH or N(C1-C4-alkyl), R1 represents hydrogen, amino or optionally cyano-, halogen- or C1-C4alkoxy-substituted alkyl having 1 to 4 carbon atoms, R2 represents carboxyl, cyano, carbamoyl, thiocarbamoyl or represents in each case optionally cyano-, halogen- or C1-C4-alkoxy-substituted alkyl or alkoxycarbonyl having in each case 1 to 4 carbon atoms, R3 represents hydrogen, halogen or optionally halogen-substituted alkyl having 1 to 4 carbon atoms, R4 represents amino or represents one of the groupings below â€”NHâ€”COâ€”R7 or â€”N(COâ€”R7)2, R5 represents nitro, amino, hydroxyl, mercapto, carboxyl, cyano, carbamoyl, thiocarbamoyl, sulfo, chlorosulfonyl, aminosulfonyl, halogen, or represents in each case optionally cyano-, halogen- or C1-C4-alkoxy-substituted alkyl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, alkylamino, alkylcarbonyl, alkoxycarbonyl, alkylaminocarbonyl, alkylcarbonylamino, alkoxycarbonylamino, alkylsulfonylamino or bis-alkylsulfonyl-amino having in each case 1 to 6 carbon atoms in the alkyl groups, R6 represents in each case optionally nitro-, cyano-, carboxyl-, carbamoyl-, thiocarbamoyl-, sulfo-, chlorosulfonyl-, aminosulfonyl-, halogen-, C1-C4-alkyl-, C1-C4-halogenoalkyl-, C1-C4-alkoxy-, C1-C4halogenoalkoxy-, C1-C4-alkylthio-, C1-C4-halogenoalkylthio-, C1-C4alkylsulfinyl-, C1-C4-halogenoalkylsulfinyl-, C1-C4-alkylsulfonyl-, C1-C4-halogenoalkylsulfonyl- or C1-C4-alkoxy-carbonyl-substituted phenyl, naphthyl or heterocyclyl selected from the group consisting of furyl, tetrahydrofuryl, benzofuryl, dihydrobenzofuryl, dioxolanyl, dioxanyl, benzodioxanyl, pyrrolyl, pyrazolyl, imidazolyl, benzimidazolyl, triazolyl, oxazolyl, isoxazolyl, benzoxazolyl, thiazolyl, isothiazolyl, benzothiazolyl, pyridinyl, quinolinyl, isoquinolinyl, pyrimidinyl, pyrazinyl, pyridazinyl, quinazolinyl, quinoxalinyl, and R7 represents hydrogen, represents in each case optionally cyano-, halogen- or C1-C4-alkoxy-substituted alkyl, alkoxy, alkylthio, alkylamino or dialkylamino having in each case 1 to 6 carbon atoms in the alkyl groups, represents in each case optionally cyano- or halogen-substituted alkenyl or alkinyl having in each case 2 to 6 carbon atoms, represents in each case optionally cyano-, halogen- or C1-C4-alkyl-substituted cycloalkyl or cycloalkylalkyl having in each case 3 to 6 carbon atoms in the cycloalkyl groups and optionally 1 to 4 carbon atoms in the alkyl moiety, or represents in each case optionally nitro-, cyano-, carboxyl-, carbamoyl-, thiocarbamoyl-, sulfo-, chlorosulfonyl-, aminosulfonyl-, halogen-, C1-C4-alkyl-, C1-C4-halogenoalkyl-, C1-C4-alkoxy-, C1-C4-halogenoalkoxy-, C1-C4-alkylthio-, C1-C4-halogenoalkylthio-, C1-C4-alkylsulfinyl-, C1-C4-halogenoalkylsulfinyl-, C1-C4alkylsulfonyl-, C1-C4-halogenoalkylsulfonyl- or C1-C4-alkoxy-carbonyl-substituted phenyl, naphthyl or heterocyclyl selected from the group consisting of furyl, tetrahydrofuryl, benzofuryl, dihydrobenzofuryl, benzodioxanyl, pyrrolyl, pyrazolyl, imidazolyl, benzimidazolyl, oxazolyl, isoxazolyl, benzoxazolyl, benzothiazolyl, pyridinyl, quinolinyl, isoquinolinyl, pyrimidinyl, pyrazinyl, pyridazinyl, quinazolinyl, quinoxalinyl.