Patent ID: 6498253
Filing Date: 2002-12-24
Classification: A01N,C07C,C07D

Abstract:
A compound of the formula (II) or a salt thereof, in which W1 is an oxygen or sulfur atom, R1 is H, C1-C24-alkyl, C2-C24-alkenyl, C2-C24-alkynyl, C1-C24-alkoxy, C2-C24-alkenyloxy C2-C24-alkynyloxy, C3-C8-cycloalkyl or C5-C8-cycloalkenyl, where each of the eight last-mentioned radicals is unsubstituted or substituted by one or more radicals from the group consisting of halogen, cyano, azido, COâ€”R5, OR6, NR7R8, SR9, SOâ€”R10 and SO2â€”R11, or unsubstituted or substituted phenyl, and has a total of up to 24 carbon atoms, R2 is H, C1-C24-alkyl, C2-C24-alkenyl and C2-C24-alkynyl, where each of the three last-mentioned radicals is unsubstituted or substituted by one or more radicals from the group consisting of halogen, cyano, azido, COâ€”R12, OR13, NR14R15, SR16, SOâ€”R17 and SO2â€”R18 and has a total of up to 24 carbon atoms, or the group NR1R2 is a saturated heterocyclic ring of three to eight ring atoms, which can have up to one further hetero atom in the ring from the group consisting of N, O and S and is unsubstituted or substituted by one or more radicals from the group consisting of C1-C6-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy, C1-C4-haloalkoxy, C1-C4-alkylthio, halogen, NO2, N3, CN and oxo, and has a total of up to 18 carbon atoms, R3 is an acyl radical of the formula COâ€”R19, CSâ€”R20, SO2â€”R21, SOâ€”R21 or C(&boxH;NR21)â€”R19, and has a total of up to 24 carbon atoms, R5 is H, C1-C5-alkyl, C2-C5-alkenyl, C2-C5-alkynyl, C1-C5-alkoxy, C2-C5-alkenoxy, C2-C5-alkynoxy, NR22R23 or OH, R6 is H, C1-C5-alkyl, C1-C5-haloalkyl, C2-C5-alkenyl, C2-C5-haloalkenyl, C2-C5-alkynyl or C2-C5-haloalkynyl, R7 is H, C1-C5-alkyl, C2-C5-alkenyl, C2-C5-alkynyl, C1-C5-alkoxy, COâ€”CH3, COâ€”H or COOCH3, R8 is H, C1-C5-alkyl, C2-C5-alkenyl or C2-C5-alkynyl or the group NR7R8 is a heterocyclic ring selected from the group consisting of the heteroaromatic or non-heteroaromatic rings pyridyl, pyrimidinyl, pyridazinyl, pyrazinyl, thiazolyl, oxazolyl, pyrrolyl, pyrazolyl, imidazolyl, pyrrolidyl, piperidyl, piperazinyl and morpholinyl, where each of the heterocyclic rings is unsubstituted or substituted by one or more radicals selected from the group consisting of halogen, C1-C6-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy, C1-C4-haloalkoxy, C1-C4-alkythio, NO2, N3, CN and oxo, R9 is H, C1-C5-alkyl, C2-C5-alkenyl, C2-C5-alkynyl, C1-C5-haloalkyl, C2-C5-haloalkenyl or C2-C5-haloalkynyl, R10 is C1-C5-alkyl, C2-C5-alkenyl, C2-C5-alkynyl, C1-C5-haloalkyl, C2-C5-haloalkenyl or C2-C5-haloalkynyl, R11 is C1-C5-alkyl, C2-C5-alkenyl, C2-C5-alkynyl, C1-C5-haloalkyl, C2-C5-haloalkenyl, C2-C5-haloalkynyl, C1-C5-alkoxyalkyl, C3-C8-cycloalkyl or C5-C8-cycloalkenyl, R12 is a radical as defined for R5, R13 is a radical as defined for R6, R14 is a radical as defined for R7, R15 is a radical as defined for R8, or the group NR14R15 is a group as defined for NR7R8, R16 is a radical as defined for R9, R17 is a radical as defined for R10, R18 is a radical as defined for R11, R19 is H, C1-C12-alkyl, C2-C12-alkenyl, C2-C12-alkynyl, C1-C12-alkoxy, C1-C12-alkylthio, C2-C12-alkenoxy, C2-C12-alkynoxy, C3-C8-cycloalkyl, C5-C8-cycloalkenyl, C1-C12-alkylamino, di(C1-C6-alkyl)amino, Nâ€”C1-C4-alkoxy-Nâ€”C1-C4-alkylamino, where each of the thirteen last-mentioned radicals are unsubstituted or substituted by one or more radicals from the group consisting of halogen, cyano, azido, COâ€”R24, OR25, NR26R27, SR28, SOR29 and SO2R30, or an unsubstituted or substituted phenyl, phenoxy or phenylamino radical, R20 is a radical as defined for R19, R21 is a radical as defined for R11, R22 is H, C1-C5-alkyl, C2-C5-alkenyl, C2-C5-alkynyl, C1-C5-alkoxy, C2-C5-alkenoxy or C2-C5-alkynoxy, where each of the six last-mentioned radicals are unsubstituted or substituted by one or more radicals from the group consisting of halogen, cyano, azido, amino, mono- and disubstituted amino, C1-C3-alkyl, C1-C3-alkoxy, C1-C3-alkylsulfonyl, C1-C3-alkylsulfinyl and C1-C3-alkylthio, R23 is H, C1-C5-alkyl, C2-C5-alkenyl, C2-C5-alkynyl, C1-C5-alkoxy or C2-C5-alkenoxy, where each of the five last-mentioned radicals is unsubstituted or substituted by one or more radicals from the group consisting of halogen, cyano, azido, amino, mono- and disubstituted amino, C1-C3-alkoxy, C1-C3-alkylthio, C1-C3-alkylsulfonyl and C1-C3-alkylsulfinyl, or the group N22R23 is a heterocyclic ring as defined for NR7R8, R24 is H, C1-C3-alkyl, C1-C3-alkoxy, NH2 or mono- or disubstituted amino, R25 is H, C1-C5-alkyl, C2-C5-alkenyl, C2-C5-alkynyl, C1-C5-haloalkyl, C2-C5-haloalkenyl or C2-C5-haloalkynyl, R26 is H, C1-C3-alkyl, C1-C3-alkoxy, COâ€”CH3 or COâ€”H, R27 is H or C1-C3-alkyl, or the group NR26R27 is a group as defined for NR22R23, R28 is H, C1-C3-alkyl, C1-C3-haloalkyl, C2-C5-alkenyl, C2-C5-haloalkenyl, C2-C5-alkynyl or C2-C5-haloalkynyl, R29 is C1-C5-alkyl, C1-C5-haloalkyl, C2-C5-alkenyl, C2-C5-haloalkyl, C2-C5-alkynyl or C2-C5-haloalkynyl, and R30 is a radical as defined for R29.