Patent ID: 6686318
Filing Date: 2004-02-03
Classification: A01N,C07D

Abstract:
An aromatic amino compound of the formula whereinR1 represents a moiety selected from the group consisting of hydrogen; hydroxyl; amino; alkyl, alkoxy, alkylamino, or dialkylamino, each of which has 1 to 6 carbon atoms in the alkyl groups; â€”CQ1â€”R5; and â€”CQ1â€”Q2â€”R6; R2 is selected from the group consisting of â€”CQ1â€”R5 and â€”CQ1â€”Q2â€”R6; R3 represents a moiety selected from the group consisting of hydrogen; hydroxyl; amino; carboxyl; cyano; carbamoyl; thiocarbamoyl; nitro; halogen; unsubstituted alkyl, alkoxy, alkoxycarbonyl, alkylthio, alkylsulphinyl, or alkylsulphonyl, each of which has 1 to 6 carbon atoms in the alkyl groups; cyano-, halogen-, or C1-C4-alkoxy-substituted alkyl, alkoxy, alkoxycarbonyl, alkylthio, alkylsulphinyl, or alkylsulphonyl, each of which has 1 to 6 carbon atoms in the alkyl groups; â€”SO2â€”NHâ€”R5; â€”NHâ€”SO2â€”R7; â€”N(SO2â€”R7)2; and â€”N(SO2â€”R7)(COâ€”R5); R4 represents a moiety selected from the group consisting of hydrogen; hydroxyl; amino; carboxyl; cyano; carbamoyl; thiocarbamoyl; nitro; halogen; unsubstituted alkyl, alkoxy, alkoxycarbonyl, alkylthio, alkylsulphinyl, or alkylsulphonyl, each of which has 1 to 6 carbon atoms in the alkyl groups; cyano-, halogen- or C1-C4-alkoxy-substituted alkyl, alkoxy, alkoxycarbonyl, alkylthio, alkylsulphinyl, or alkylsulphonyl, each of which has 1 to 6 carbon atoms in the alkyl groups; â€”SO2â€”NHâ€”R5; â€”NHâ€”SO2â€”R7; â€”N(SO2â€”R7)2; and â€”N(SO2â€”R7)(COâ€”R5); Q1 and Q2 each represent O; R5 represents a moiety selected from the group consisting of hydrogen; unsubstituted or cyano-, halogen-, or C1-C4-alkoxy-substituted alkyl which has 1 to 6 carbon atoms; cycloalkyl or cycloalkylalkyl, each of which has 3 to 6 carbon atoms in the cycloalkyl group and, where appropriate, 1 to 4 carbon atoms in the alkyl moiety and each of which is optionally substituted by cyano, halogen, or C1-C4-alkyl; and aryl or arylalkyl, each of which has 6 or 10 carbon atoms in the aryl group and, where appropriate, 1 to 4 carbon atoms in the alkyl moiety and each of which is optionally substituted by cyano, nitro, halogen, C1-C4-alkyl, C1-C4-halogenoalkyl, C1-C4-alkoxy, or C1-C4-halogenoalkoxy; R6 represents a moiety selected from the group consisting of alkyl which has 1 to 6 carbon atoms and which is optionally substituted by cyano, halogen, or C1-C4-alkoxy; alkenyl or alkynyl, each of which has 2 to 6 carbon atoms and each of which is optionally substituted by halogen; cycloalkyl or cycloalkylalkyl, each of which has 3 to 6 carbon atoms in the cycloalkyl group and, where appropriate, 1 to 4 carbon atoms in the alkyl moiety and each of which is optionally substituted by cyano, halogen, or C1-C4-alkyl; and aryl or arylalkyl, each of which has 6 or 10 carbon atoms in the aryl group and, where appropriate, 1 to 4 carbon atoms in the alkyl moiety and each of which is optionally substituted by cyano, nitro, halogen, C1-C4-alkyl, C1-C4-halogenoalkyl, C1-C4-alkoxy, or C1-C4-halogenoalkoxy; R7 represents a moiety selected from the group consisting of alkyl which has 1 to 6 carbon atoms and which is optionally substituted by halogen; cycloalkyl or cycloalkylalkyl, each of which has 3 to 6 carbon atoms in the cycloalkyl moiety and, where appropriate, 1 to 4 carbon atoms in the alkyl moiety and each of which is optionally substituted by halogen; and aryl or arylalkyl, each of which has 6 or 10 carbon atoms in the aryl group and, where appropriate, 1 to 4 carbon atoms in the alkyl moiety and each of which is optionally substituted by cyano, nitro, halogen, C1-C4-alkyl, C1-C4-halogenoalkyl, C1-C4-alkoxy, C1-C4-halogenoalkoxy, C1-C4-alkylthio, C1-C4-alkylsulphinyl, C1-C4-alkylsulphonyl, or C1-C4-alkoxy-carbonyl; Z represents whereinR8 represents a moiety selected from the group consisting of hydrogen; amino; nitro; cyano; carboxyl; carbamoyl; thiocarbamoyl; halogen; alkyl which has 1 to 6 carbon atoms and which is optionally substituted by cyano, halogen or C1-C4-alkoxy; alkenyl or alkynyl, each of which has 2 to 6 carbon atoms and each of which is optionally substituted by halogen; alkoxy or alkoxycarbonyl, each of which has 1 to 6 carbon atoms in the alkyl groups and each of which is optionally substituted by cyano, halogen or C1-C4-alkoxy; alkenyloxy, or alkynyloxy, each of which has 3 to 6 carbon atoms and each of which is optionally substituted by halogen; alkylthio which has 1 to 6 carbon atoms and which is optionally substituted by cyano, halogen, or C1-C4-alkoxy; alkenylthio or alkynylthio, each of which has 3 to 6 carbon atoms and each of which is optionally substituted by halogen; alkylamino or dialkylamino, each of which has 1 to 6 carbon atoms in the alkyl groups, each of which is optionally substituted by cyano, halogen, or C1-C4-alkoxy; and cycloalkyl or cycloalkylalkyl, each of which has 3 to 6 carbon atoms in the cycloalkyl groups and, where appropriate, 1 to 4 carbon atoms in the alkyl moiety and each of which is optionally substituted by cyano, halogen, or C1-C4-alkyl; and R9 represents a moiety selected from the group consisting of hydrogen; hydroxyl; amino; cyano; alkyl which has 1 to 6 carbon atoms and which is optionally substituted by cyano, halogen, or C1-C4-alkoxy; alkenyl or alkynyl, each of which has 2 to 6 carbon atoms and which is optionally substituted by halogen; alkoxycarbonyl, which is optionally substituted by cyano, halogen, or C1-C4-alkoxy; cycloalkyl or cycloalkylalkyl, each of which has 3 to 6 carbon atoms in the cycloalkyl groups and, where appropriate, 1 to 4 carbon atoms in the alkyl moiety and each of which is optionally substituted by cyano, halogen, or C1-C4-alkyl; and phenyl or phenyl-C1-C4-alkyl, each of which is optionally substituted by cyano, nitro, halogen, C1-C4-alkyl, C1-C4-halogenoalkyl, C1-C4-alkoxy and/or C1-C4-halogenoalkoxy, where the individual radicals R8 and R9 may have identical or different meanings.