Patent ID: 7781613
Filing Date: 2010-08-24
Classification: A61P,C07C,C07D

Abstract:
1. A compound of formula (I) wherein: R1 is hydrogen, halogen or —CF R2 is hydrogen, —NH R3 is unsubstituted or monosubstituted C R4 and R5 are, independently of one another, hydrogen, unsubstituted or substituted C R6 is hydrogen, —SO R7 is C A is CO or CH X is NR6 or O; and wherein heteroaryl is a 5 to 10-membered, aromatic, mono-r bicyclic heterocycle which comprises one or more heteroatoms selected from N, O and S; aryl is a 5 to 10-membered aromatic mono- or bicyclic system; and heterocyclyl is a 5 to 10-membered, nonaromatic, mono- or bicyclic heterocycle which comprises one or more heteroatoms selected from N, O and S; or a physiologically tolerated salt thereof; with the proviso that when R2 is hydrogen and R1 is halogen, then —A—X—R3 is not i) —C(O) —O—CH