Patent ID: 6617281
Filing Date: 2003-09-09
Classification: A01N,A61P,C07D

Abstract:
An acylaminophenyl-uracil of the formula (I) whereinn represents the numbers 0 or 1, A represents unsubstituted or halogen-substituted alkanediyl(alkylene) having 1 to 6 carbon atoms or cycloalkanediyl having 3 to 6 carbon atoms, or A represents a single bond or an unsubstituted or halogen-substituted alkanediyl(alkylene) having 1 to 6 carbon atoms or cycloalkanediyl having 3 to 6 carbon atoms attached to Ar via an alkanediyl grouping having 1 to 3 carbon atoms where n represents 1; Ar represents substituted aryl or arylalkyl having 6 or 10 carbon atoms in the aryl group and optionally 1 to 4 carbon atoms in the alkyl moiety, or represents unsubstituted or substituted heterocyclyl or heterocyclylalkyl selected from the group consisting of oxiranyl, oxiranylmethyl, oxetanyl, oxetanylmethyl, furyl, furylmethyl, tetrahydrofuryl, tetrahydrofurylmethyl, thienyl, thienylmethyl, tetrahydrothienyl, tetrahydrothienylmethyl, benzofuryl, benzofurylmethyl, dihydrobenzofuryl, dihydrobenzofurylmethyl, benzothienyl, benzothienylmethyl, pyrrolyl, pyrrolylmethyl, pyrazolyl, pyrazolylmethyl, pyranyl, pyranylmethyl, benzopyranyl, benzopyranylmethyl, dihydrobenzopyranyl, dihydrobenzopyranylmethyl, tetrahydrobenzopyranyl, tetrahydrobenzopyranylmethyl, pyridinyl, pyridinylmethyl, pyrimidinyl, and pyrimidinylmethyl, wherein the substituent(s) for Ar is/are selected from the group consisting of nitro, cyano, carboxyl, carbamoyl, thiocarbamoyl, halogen, C1-C4-alkyl, C1-C4-halogenoalkyl, C1-C4-alkoxy, C1-C4-halogenoalkoxy, C1-C4-alkylthio, C1-C4-halogenoalkylthio, C1-C4-alkylsulphinyl, C1-C4-halogenoalkylsulphinyl, C1-C4-alkylsulphonyl, C1-C4-halogenoalkylsulphonyl, C1-C4-alkylamino, di-(C1-C4-alkyl)amino, C1-C4-alkyl-carbonyl, C1-C4-alkoxy-carbonyl, C1-C4-alkylamino-carbonyl, di-(C1-C4-alkyl)-amino-carbonyl, and di-(C1-C4-alkyl)-amino-sulphonyl, Q represents O (oxygen), S (sulphur), SO, SO2, NH or N(C1-C4-alkyl), R1 represents hydrogen, amino or unsubstituted or cyano-, carboxyl-, halogen-, C1-C4-alkoxy- or â€”C1-C4-alkoxycarbonyl-substituted alkyl having 1 to 6 carbon atoms, R2 represents carboxyl, cyano, carbamoyl, thiocarbamoyl or represents unsubstituted or cyano-, halogen- or C1-C4-alkoxy-substituted alkyl or alkoxycarbonyl having 1 to 6 carbon atoms in the alkyl groups, R3 represents hydrogen, halogen or unsubstituted or halogen-substituted alkyl having 1 to 6 carbon atoms, R4 represents hydrogen, cyano, carbamoyl, thiocarbamoyl, or halogen, R5 represents cyano, carbamoyl, thiocarbamoyl, halogen, or represents unsubstituted or halogen-substituted alkyl or alkoxy having 1 to 4 carbon atoms, and R6 represents hydrogen, represents unsubstituted or cyano-, halogen- or C1-C4-alkoxy-substituted alkyl, alkylcarbonyl or alkoxycarbonyl having 1 to 6 carbon atoms in the alkyl groups, represents unsubstituted or halogen-substituted alkylsulphonyl having 1 to 6 carbon atoms, represents unsubstituted or halogen-substituted alkenyl, alkenylcarbonyl, alkenylsulphonyl or alkynyl having up to 6 carbon atoms, represents unsubstituted or halogen-substituted cycloalkylcarbonyl or cycloalkylsulphonyl having 3 to 6 carbon atoms in the cycloalkyl groups, represents unsubstituted or nitro-, cyano-, halogen-, C1-C4-alkyl-, C1-C4-halogenoalkyl-, C1-C4-alkoxy-, C1-C4-halogenoalkoxy-, C1-C4-alkylthio-, C1-C4- halogenoalkylthio-, C1-C4-alkylsulphinyl-, C1-C4- halogenoalkylsulphinyl-, C1-C4-alkylsulphonyl-, C1-C4- halogenoalkylsulphonyl, C1-C4-alkyl-carbonyl-, C1-C4-alkoxy-carbonyl- or di-(C1-C4- alkyl-amino)-sulphonyl-substituted arylcarbonyl, arylsulphonyl, arylalkylcarbonyl or arylalkylsulphonyl having 6 or 10 carbon atoms in the aryl groups and 1 to 4 carbon atoms in the alkyl moiety, or represents unsubstituted or nitro-, cyano-, halogen-, C1-C4-alkyl-, C1-C4-halogenoalkyl-, C1-C4-alkoxy-, C1-C4-halogenoalkoxy-, C1-C4-alkylthio-, C1-C4-halogenoalkylthio-, C1-C4-alkylsulphinyl, C1-C4-halogenoalkylsulphinyl-, C1-C4-alkylsulphonyl-, C1-C4-halogenoalkylsulphonyl-, C1-C4-alkyl-carbonyl-, C1-C4-alkoxy-carbonyl- or di-(C1-C4- alkyl-aminoysulphonyl-substituted heterocyclylcarbonyl or heterocyclylsulphonyl selected from the group consisting of furylcarbonyl, furylsulphonyl, thienylcarbonyl, thienylsulphonyl, pyrazolylcarbonyl, pyrazolylsulphonyl, pyridinylcarbonyl, pyridinylsulphonyl, quinolinylcarbonyl, quinolinylsulphonyl, pyrimidinylcarbonyl, and pyrimidinylsulphonyl.