Patent ID: 7019143
Filing Date: 2006-03-28
Classification: C07D

Abstract:
1. A process for preparing a compound according to the steps shown in Scheme I: wherein the resulting compound is a compound according to Formula I: wherein, for Formula I: (a) X is selected from the group consisting of (b) R1 is selected from the group consisting of C (c) R8 is selected from the group consisting of fluoro, and chloro; (d) R7 is amino which is attached to a ring carbon of X which is not adjacent to the ring nitrogen, the amino being unsubstituted or substituted with one or two C (e) each R9 is independently selected from the group consisting of hydrogen, C (f) a R7 moiety described in (d) and a R9 moiety described in (e) may optionally be connected thus forming a fused or spirocycle ring with the N-containing ring shown in (a), the fused or spirocycle ring comprising from 2 to about 5 ring carbons and 0 or 1 ring nitrogen; or an optical isomer, diastereomer or enantiomer thereof; a pharmaceutically-acceptable salt, hydrate, or biohydrolyzable ester, amide or imide thereof.