Patent ID: 8816086
Filing Date: 2014-08-26
Classification: A61P,C07D

Abstract:
1. A process for preparing a compound of formula (Ib) or (IIIa) or salt thereof, wherein R R R R A G R G R R R G R wherein the monocyclic cycloalkyl, as a substituent or part of a substituent, of R q, q1, and q2, at each occurrence, are each independently 1, 2, 3, or 4; R q3, at each occurrence, is independently 1, 2 or, 3; q4, at each occurrence, is independently 2, 3, 4, or 5; q5, at each occurrence, is independently 1, 2, 3, 4, 5, or 6; z is 0, 1, 2, 3, or 4; one of X u is 0, 1, 2, or 3; and each R (1a) treating a compound of formula (IV) wherein R (1b) reacting a compound of formula (V) with a compound of formula (VI) wherein R (2a) treating a compound of formula (II) or a salt thereof with a compound of formula HO—(CR R (2b) deprotect a compound of formula (IIIb) or a salt thereof wherein R