Patent ID: 6379591
Filing Date: 2002-04-30
Classification: C07D,G02B

Abstract:
A compound of the following formula (I): in which:R1 and R2, which are identical or different, independently represent: hydrogen, a linear or branched alkyl group comprising 1 to 12 carbon atoms, a cycloalkyl group comprising 3 to 12 carbon atoms, an aryl group comprising, in its basic structure, 6 to 24 carbon atoms or a heteroaryl group comprising, in its basic structure, 4 to 24 carbon atoms and at least one heteroatom selected from sulphur, oxygen, and nitrogen; said basic structure being optionally substituted with at least one substituent selected from: a halogen, a hydroxy group, a linear or branched alkyl group comprising 1 to 12 carbon atoms, a linear or branched alkoxy group comprising 1 to 12 carbon atoms, a haloalkyl or haloalkoxy group corresponding to the (C1-C12) alkyl or alkoxy groups above, respectively, which are substituted with at least one halogen atom, a linear or branched alkenyl group comprising 2 to 12 carbon atoms, an â€”NH2 group, an â€”NHR group, wherein R represents a linear or branched alkyl group comprising 1 to 6 carbon atoms, a â€ƒgroup, wherein Râ€² and Râ€³, which are identical or different, represent, independently, a linear or branched alkyl group comprising 1 to 6 carbon atoms or Râ€² and Râ€³, together with the nitrogen atom to which they are bound, represent a 5- to 7-membered ring which optionally comprises at least one other heteroatom selected from oxygen, sulphur, and nitrogen, said nitrogen being optionally substituted with an Râ€²â€³ group, which is a linear or branched alkyl group comprising 1 to 6 carbon atoms, and a methacryloyl group or an acryloyl group, or an aralkyl or heteroaralkyl group, the alkyl part of which is linear or branched and comprises 1 to 4 carbon atoms and the aryl part of which has the same definition as that given above for the aryl and heteroaryl group; or said two substituents R1 and R2 together form an adamantyl, norbornyl, fluorenylidene, di(C1-C6)alkylanthracenylidene, or spiro (C5-C6)cycloalkylanthracenylidene group; said group being optionally substituted with at least one substituent selected from the group consisting of: a halogen, a hydroxy group, a linear or branched alkyl group comprising 1 to 12 carbon atoms, a linear or branched alkoxy group comprising 1 to 12 carbon atoms, a haloalkyl or haloalkoxy group corresponding to the (C1-C12) alkyl or alkoxy groups above, respectively, which are substituted with at least one halogen atom, a linear or branched alkenyl group comprising 2 to 12 carbon atoms, an â€”NH2 group, an â€”NHR group, wherein R represents a linear or branched alkyl group comprising 1 to 6 carbon atoms, a â€ƒgroup, wherein Râ€² and Râ€³, which are identical or different, represent, independently, a linear or branched alkyl group comprising 1 to 6 carbon atoms or Râ€² and Râ€³, together with the nitrogen atom to which they are bound, represent a 5- to 7-membered ring which optionally comprises at least one other heteroatom selected from oxygen, sulphur, and nitrogen, said nitrogen being optionally substituted with an Râ€²â€³ group, which is a linear or branched alkyl group comprising 1 to 6 carbon atoms, and a methacryloyl group or an acryloyl group; R3 represents: a hydrogen, a linear or branched alkyl group comprising 1 to 12 carbon atoms, a cycloalkyl group comprising 3 to 12 carbon atoms, a haloalkyl, halocycloalkyl, or haloalkoxy group corresponding to the alkyl, cycloalkyl, and alkoxy groups above, respectively, which are substituted with at least one halogen atom, an aralkyl or heteroaralkyl group, the alkyl part of which is linear or branched and comprises 1 to 4 carbon atoms and the aryl part of which has the same definition as that given above for R1, R2, a â€”COR6, â€”COOR6, or â€”CONHR6 group, wherein R6 represents a straight or branched alkyl group comprising 1 to 6 carbon atoms, a cycloalkyl group comprising 3 to 6 carbon atoms, or a linear or branched alkenyl group comprising 2 to 12 carbon atoms, optionally substituted with at least one substituent selected from the group consisting of: a halogen, a hydroxy group, a linear or branched alkyl group comprising 1 to 12 carbon atoms, a linear or branched alkoxy group comprising 1 to 12 carbon atoms, a haloalkyl or haloalkoxy group corresponding to the (C1-C12) alkyl or alkoxy groups above, respectively, which are substituted with at least one halogen atom, a linear or branched alkenyl group comprising 2 to 12 carbon atoms, an â€”NH2 group, an â€”NHR group, wherein R represents a linear or branched alkyl group comprising 1 to 6 carbon atoms, a â€ƒgroup, wherein Râ€² and R â€³, which are identical or different, represent, independently, a linear or branched alkyl group comprising 1 to 6 carbon atoms or Râ€² and Râ€³, together with the nitrogen atom to which they are bound, represent a 5- to 7-membered ring which optionally comprises at least one other heteroatom selected from oxygen, sulphur, and nitrogen, said nitrogen being optionally substituted with an Râ€²â€³ group, which is a linear or branched alkyl group comprising 1 to 6 carbon atoms, and a methacryloyl group or an acryloyl group; R4 and R5, which are identical or different, represent, independently: a halogen, a linear or branched alkyl group comprising 1 to 12 carbon atoms, a cycloalkyl group comprising 3 to 12 carbon atoms, a linear or branched alkoxy group comprising 1 to 12 carbon atoms, a haloalkyl, halocycloalkyl, or haloalkoxy group corresponding to the alkyl, cycloalkyl, and alkoxy groups above, respectively, which are substituted with at least one halogen atom, an aryl or heteroaryl group having the same definition as that given above for R1, R2, an aralkyl or heteroaralkyl group, the alkyl part of which is linear or branched and comprises 1 to 4 carbon atoms and the aryl part of which has the same definition as that given above for R1, R2, an amine or amide group: â€”NH2, â€”NHR, â€”CONH2, â€”CONHR, â€ƒwherein R represents a linear or branched alkyl group comprising 1 to 6 carbon atoms and wherein Râ€² and Râ€³, which are identical or different, represent, independently, a linear or branched alkyl group comprising 1 to 6 carbon atoms or Râ€² and Râ€³, together with the nitrogen atom to which they are bound, represent a 5- to 7-membered ring which optionally comprises at least one other heteroatom selected from oxygen, sulphur, and nitrogen, said nitrogen being optionally substituted with an Râ€²â€³ group, which is a linear or branched alkyl group comprising 1 to 6 carbon atoms, or an â€”OCOR7 or â€”COOR7 group, wherein R7 represents a straight or branched alkyl group comprising 1 to 6 carbon atoms, or a cycloalkyl group comprising 3 to 6 carbon atoms, or a phenyl group, optionally substituted with at least one substituent selected from the group consisting of: a halogen, a hydroxy group, a linear or branched alkyl group comprising 1 to 12 carbon atoms, a linear or branched alkoxy group comprising 1 to 12 carbon atoms, a haloalkyl or haloalkoxy group corresponding to the (C1-C12) alkyl or alkoxy groups above, respectively, which are substituted with at least one halogen atom, a linear or branched alkenyl group comprising 2 to 12 carbon atoms, an â€”NH2 group, an â€”NHR group, wherein R represents a linear or branched alkyl group comprising 1 to 6 carbon atoms, a â€ƒgroup, wherein Râ€² and Râ€³, which are identical or different, represent, independently, a linear or branched alkyl group comprising 1 to 6 carbon atoms or Râ€² and Râ€³, together with the nitrogen atom to which they are bound, represent a 5- to 7-membered ring which optionally comprises at least one other heteroatom selected from oxygen, sulphur, and nitrogen, said nitrogen being optionally substituted with an Râ€²â€³ group, which is a linear or branched alkyl group comprising 1 to 6 carbon atoms, and a methacryloyl group or an acryloyl group; and m and n are integers of 0 to 4.