Patent ID: 6548449
Filing Date: 2003-04-15
Classification: C07D

Abstract:
A phenyluracil of the formula (I) in whichm represents the numbers 0, 1 or 2, n represents the numbers 0, 1, 2 or 3, Q represents O, S, SO, SO2, NH or N(C1-C4-alkyl), R1 represents hydrogen, amino or optionally cyano-, halogen- or C1-C4-alkoxy-substituted alkyl having 1 to 6 carbon atoms, R2 represents carboxyl, cyano, carbamoyl, thiocarbamoyl, or represents in each case optionally cyano-, halogen- or C1-C4-alkoxy-substituted alkyl or alkoxy-carbonyl having in each case up to 6 carbon atoms, R3 represents hydrogen, halogen or optionally cyano-, halogen- or C1-C4-alkoxy-substituted alkyl having 1 to 6 carbon atoms, R4 represents hydrogen, cyano or halogen, R5 represents nitro, amino, hydroxyl, carboxyl, cyano, carbamoyl, thiocarbamoyl, sulpho, chlorosulphonyl, aminosulphonyl, halogen, or represents in each case optionally cyano-, halogen- or C1-C4-alkoxy-substituted alkyl, alkoxy, alkyl-thio, alkylsulphinyl, alkylsulphonyl, alkylamino, alkylcarbonyl, alkoxycarbonyl, alkylaminocarbonyl, alkylcarbonylamino, alkoxycarbonylamino or alkyl-sulphonylamino having in each case up to 6 carbon atoms, and R6 represents amino or one of the groupings below â€”NHâ€”R8, â€”N(R8)2, â€”NHâ€”SO2â€”R8, â€”N(R8)(SO2â€”R8), â€”N(SO2â€”R8)2, â€”NHâ€”COâ€”R9, â€”N(R8)(COâ€”R9), â€”N(COâ€”R9)2, â€”N(SO2â€”R8)(COâ€”R9), R7 represents nitro, amino, hydroxyl, mercapto, carboxyl, cyano, carbamoyl, thio-carbamoyl, sulpho, chlorosulphonyl, aminosulphonyl, halogen, or represents in each case optionally cyano-, halogen- or C1-C4-alkoxy-substituted alkyl, alkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl, alkylamino, alkylcarbonyl, alkoxycarbonyl, alkylaminocarbonyl, alkylcarbonylamino, alkoxycarbonyl-amino, alkylsulphonylamino or bis-alkylsulphonyl-amino having in each case up to 6 carbon atoms, R8 represents optionally halogen-substituted alkyl having 1 to 6 carbon atoms, represents optionally halogen-substituted alkenyl having 2 to 6 carbon atoms, represents optionally cyano-, halogen- or C1-C4-alkyl-substituted cycloalkyl having 3 to 6 carbon atoms, represents in each case optionally nitro-, cyano-, thiocarbamoyl-, halogen-, C1-C4-alkyl, C1-C4-halogenoalkyl-, C1-C4-alkoxy-, C1-C4-halogenoalkoxy-, C1-C4-alkylthio-, C1-C4-halogenoalkylthio-, C1-C4-alkylsulphinyl-, C1-C4-halogenoalkylsulphinyl-, C1-C4-alkylsulphonyl-, C1-C4-halogenoalkylsulphonyl- or C1-C4-alkoxy-carbonyl-substituted aryl or arylalkyl having in each case 6 or 10 carbon atoms in the aryl group and optionally 1 to 4 carbon atoms in the alkyl moiety, or represents optionally cyano-, halogen-, C1-C4-alkyl-, C1-C4-halogenoalkyl-, C1-C4-alkoxy-, C1-C4-halogenoalkoxy-, C1-C4-alkylthio-, C1-C4-halogenoalkylthio-, C1-C4-alkylsulphinyl-, C1-C4-halogenoalkylsulphinyl-, C1-C4-alkylsulphonyl- or C1-C4-halogenoalkyl-sulphonyl-substituted heterocyclyl selected from the group consisting of furyl, thienyl, oxazolyl, isoxazolyl, pyrazolyl, pyridyl and pyrimidyl, and R9 represents hydrogen, represents in each case optionally cyano-, halogen- or C1-C4-alkoxy-substituted alkyl, alkoxy, alkylamino or dialkylamino having in each case 1 to 6 carbon atoms, represents in each case optionally cyano- or halogen-substituted alkenyl or alkinyl having in each case 2 to 6 carbon atoms, represents in each case optionally cyano-, halogen- or C1-C4-alkyl-substituted cycloalkyl or cycloalkylalkyl having in each case 3 to 6 carbon atoms in the cycloalkyl group and optionally 1 to 4 carbon atoms in the alkyl moiety, represents in each case optionally nitro-, cyano-, thiocarbamoyl-, halogen-, C1-C4-alkyl-, C1-C4-halogenoalkyl-, C1-C4-alkoxy-, C1-C4-halogenoalkoxy-, C1-C4-alkylthio-, C1-C4-halogenoalkylthio-, C1-C4-alkylsulphinyl-, C1-C4-halogenoalkylsulphinyl-, C1-C4-alkylsulphonyl-, C1-C4-halogenoalkylsulphonyl- or C1-C4-alkoxy-carbonyl-substituted aryl or arylalkyl having in each case 6 or 10 carbon atoms in the aryl group and optionally 1 to 4 carbon atoms in the alkyl moiety, or represents optionally cyano-, halogen-, C1-C4-alkyl-, C1-C4-halogenoalkyl-, C1-C4-alkoxy-, C1-C4-halogenoalkoxy-, C1-C4-alkylthio-, C1-C4-halogenoalkylthio-, C1-C4-alkylsulphinyl-, C1-C4-halogenoalkylsulphinyl-, C1-C4-alkylsulphonyl- or C1-C4-halogenoalkyl-sulphonylsubstituted heterocyclyl selected from the group consisting of furyl, thienyl, oxazolyl, isoxazolyl, pyrazolyl, pyridyl and pyrimidyl.