Patent ID: 6951855
Filing Date: 2005-10-04
Classification: A61P,C07D

Abstract:
1. A compound of Formula (II) or a salt, pro-drug or solvate thereof, wherein: X is selected from: —O—, —S—, —S(O)—, —S(O R R R R n is 0, 1 or 2; and p is 0, 1, 2 or 3; with the proviso that the following compounds are excluded: 6-benzyloxy-2H-1,4-benzoxazin-3(4H)-one; 7-benzyloxy-2H-1,4-benzoxazin-3(4H)-one; 2-methyl-7-benzyloxy-2H-1,4-benzoxazin-3(4H)-one; 2,4-dimethyl-7-benzyloxy-2H-1,4-benzoxazin-3(4H)-one; 2-methyl-7-(3,5-dichlorobenzyloxy)-2H-1,4-benzoxazin-3(4H)-one; 2,4-dimethyl-7-(3,5-dichlorobenzyloxy)-2H-1,4-benzoxazin-3(4H)-one; 7-phenylthio-2H-1,4-benzoxazin-3(4H)-one; 4-methyl-7-phenylthio-2H-1,4-benzoxazin-3(4H)-one; 4-methyl-7-phenylsulfinyl-2H-1,4-benzoxazin-3(4H)-one; and 6-phenylsulfonyl-2H-1,4-benzoxazin-3(4H)-one.