Patent ID: 6392043
Filing Date: 2002-05-21
Classification: C07D,C08G,G02B

Abstract:
Compounds of formula (I): in which:R1 and R2, identical or different, independently represent: hydrogen, a linear or branched alkyl group having 1 to 12 carbon atoms, a cycloalkyl group having 3 to 12 carbon atoms, an aryl or heteroaryl group having 6 to 24 carbon atoms or 4 to 24 carbon atoms respectively in its basic structure and at least one heteroatom selected from sulfur, oxygen and nitrogen; said basic structure optionally being substituted with at least one substituent selected from: a halogen, a linear or branched alkyl group having 1 to 12 carbon atoms, a linear or branched alkoxy group having 1 to 12 carbon atoms, a linear or branched haloalkyl or haloalkoxy group corresponding respectively to the (C1-C12)alkyl and (C1-C12)alkoxy groups above substituted with at least one halogen atom, a linear or branched alkenyl group having 2 to 12 carbon atoms, an NH2 group, an NHR group, R representing a linear or branched alkyl group having 1 to 6 carbon atoms, a â€ƒRâ€² and Râ€³, identical or different, representing independently a linear or branched alkyl group having 1 to 6 carbon atoms or representing, together with the nitrogen atom to which they are bound, a 5- to 7-membered ring which can comprise at least one other heteroatom selected from oxygen, sulfur and nitrogen, said nitrogen optionally being substituted with an Râ€²â€³ group, wherein the Râ€²â€³ group is a linear or branched alkyl group having 1 to 6 carbon atoms, an epoxy group of formula: an aralkyl or heteroaralkyl group, the linear or branched alkyl group having 1 to 4 carbon atoms and the aryl and heteroaryl groups having the definitions given above, or said two substituents R1 and R2 together form an adamantyl, a norbornyl, a fluorenylidene, a di(C1-C6)alkylanthracenylidene or a spiro(C5-C6)cycloalkylanthracenylidene group; said group optionally being substituted with at least one of the substituents listed above for R1, R2: aryl or heteroaryl group; R3 represents: hydrogen, a linear or branched alkyl group having 1 to 12 carbon atoms, a cycloalkyl group having 3 to 12 carbon atoms, an linear or branched alkoxy group, having 1 to 12 carbon atoms, a haloalkyl, a halocycloalkyl or a haloalkoxy group corresponding respectively to the alkyl, cycloalkyl, or alkoxy groups above, substituted with at least one halogen atom, an aryl or heteroaryl group having the same definition as that given above for R1, R2, an aralkyl or heteroaralkyl group, the linear or branched alkyl group having 1 to 4 carbon atoms and the aryl and heteroaryl groups having the same definitions as those given above for R1, R2, an â€”OCOR6 or â€”COOR6 group, R6 representing a straight or branched alkyl group having 1 to 6 carbon atoms or a cycloalkyl group having 3 to 6 carbon atoms or a phenyl group optionally substituted with at least one of the substituents listed above for the R1, R2 values: aryl or heteroaryl; R4 represents: hydrogen, a halogen, a linear or branched alkyl group having 1 to 12 carbon atoms, a cycloalkyl group having 3 to 12 carbon atoms, an linear or branched alkoxy group having 1 to 12 carbon atoms, a haloalkyl, a halocycloalkyl or a haloalkoxy group corresponding respectively to the alkyl, cycloalkyl, or alkoxy groups above, substituted with at least one halogen atom, an aryl or heteroaryl group having the same definition as that given above for R1, R2, an aralkyl or heteroaralkyl group, the linear or branched alkyl group having 1 to 4 carbon atoms and the aryl and heteroaryl groups having the same definitions as those given above for R1, R2, an amine or amide group: â€”NH2, â€”NHR, â€”CONH2, â€”CONHR, â€ƒR, Râ€², Râ€³ having their respective definitions given above for the amine substituents of the R1, R2 values: aryl or heteroaryl, an â€”OCOR6 or â€”COOR6 group, R6 representing a straight or branched alkyl group having 1 to 6 carbon atoms or a cycloalkyl group having 3 to 6 carbon atoms or a phenyl group optionally substituted with at least one of the substituents listed above for the R1, R2 values: aryl or heteroaryl; m and n are, independently, integers of 0 to 4; R5 represents: hydrogen, a linear or branched alkyl group having 1 to 12 carbon atoms, a cycloalkyl group having 3 to 12 carbon atoms, a linear or branched alkenyl group having 2 to 12 carbon atoms, a phenyl or benzyl group, optionally substituted with at least one of the substituents listed above for the R1, R2 values: aryl or heteroaryl, a â€”COR7, â€”COOR7 or â€”CONHR7 group, R7 representing a straight or branched alkyl group having 1 to 6 carbon atoms or a cycloalkyl group having 3 to 6 carbon atoms or a linear or branched alkenyl group having 2 to 12 carbon atoms or a phenyl or benzyl group optionally substituted with at least one of the substituents listed above for the R1, R2 values: aryl or heteroaryl, a methacryloyl group or an acryloyl group, an epoxy group of formula: