Patent ID: 6384225
Filing Date: 2002-05-07
Classification: A61P,C07D

Abstract:
A compound of the formula whereinX is N or CH; R1 is C1-C6 alkyl or C3-C6 cycloalkyl; R2 is hydrogen or C1-C6 alkyl; and R9 is C1-C6 alkyl, C3-C6 cycloalkyl, OCF3, OCHF2, OCH2F, halogen, CN, CF3, OH, C1-C6 alkoxy, C1-C6 alkoxy-C1-C6 alkyl, NR6R7, SO3CH3, SO3CF3, SO2NR6R7, an unsubstituted or substituted heterocyclic or heteroaromatic ring containing one or two heteroatoms selected from N and O, wherein the substituent(s) is(are) C1-C6 alkyl; or COR8; wherein R6 is H, C1-C6 alkyl or C3-C6 cycloalkyl; R7 is H, C1-C6 alkyl or C3-C6 cycloalkyl; and R8 is C1-C6 alkyl, C3-C6 cycloalkyl, CF3, NR6R7, phenyl, a heteroaromatic ring containing one or two heteroatoms selected from the group consisting of N, O and S or a heterocyclic ring containing one or two heteroatoms selected from the group consisting of N, O, S, SO and SO2 wherein R6 and R7 are as defined above.