Patent ID: 8815893
Filing Date: 2014-08-26
Classification: A61P,C07D

Abstract:
1. A compound of formula (I) wherein W W W under the proviso that at least one of W X denotes NR1, Alk, O, or S; R1 denotes H, A or Cyc; R5 denotes H, A, Hal, OY, CN, -Alk-OY, COOY, —CO—NYY, SA, SO or R1, R5 together denote —CH═CH—, —C(Y)═N—, —N═C(Y)—, —C(COY)═N—, —C(CO—R2)=N—, —CO—NH—, —NH—CO—, —SO R6 denotes H, A, Hal, OY, CN, -Alk-OY, COOY, —CO—NYY, NYY, —NY—COOY, —NH-Alk-NYY, —NH—COA, —NH—CO-Alk-NYY, —NH-Het R2 denotes a monocyclic carboaryl having 5-8 C atoms or a monocyclic heteroaryl having 2-7 C atoms and 1-4 N, O and/or S atoms, each of which is unsubstituted or substituted by at least one substituent selected from A, Hal, CN, NYY, OY, and ═O; R3, R4 each denote, independently from one another, H, A, Hal, CN, NYY, OY, —OAlk-NYY, or —OAlk-OY; Y denotes H or A; A denotes unbranched or branched alkyl having 1-10 C atoms, in which 1-7 H atoms are each optionally replaced by Hal; Cyc denotes cycloalkyl having 3-7 C atoms, in which 1-4 H atoms are each optionally replaced independently from one another by A, Hal or OY; Alk denotes alkylene having 1-6 C atoms, in which 1-4 H atoms are each optionally replaced independently of one another by Hal or CN; Ar denotes a saturated, unsaturated or aromatic, mono- or bicyclic carbocycle having 6-10 C atoms, which is unsubstituted or substituted by at least one substituent selected from Het Het Het Het Hal denotes F, Cl, Br or I; or a physiologically acceptable salt thereof.