Patent ID: 8987465
Filing Date: 2015-03-24
Classification: A01N,A61K,C07D

Abstract:
1. A compound of the formula (I) wherein wherein R1 is hydrogen; R2 is hydrogen; R3 is hydrogen; R4 is hydrogen; R5 is pyridyl, which has one or more substituents, provided at least one of which is an unsubstituted or substituted aromatic heterocycle (HET); R6 is hydrogen or C1-C4-alkyl; R7 is hydrogen, cyano, hydroxyl, formyl, C1-C4-alkyl, C1-C4-alkoxy, C2-C4-alkenyl, C2-C4-alkynyl, C1-C4-alkoxy- C1-C4-alkyl, C1-C4-cyanoalkyl, C1-C4-alkylcarbonyl, C1-C4-alkoxycarbonyl, benzyl, C3-C6-cycloalkylcarbonyl or C3-C6-cycloalkoxycarbonyl; A1 is N, C—H or C—X; A2 is N, C—H or C—X; A3 is N, C—H or C—X; A4 is N, C—H or C—X; A5 is N, C—H or C—X; X is a halogen, OH, cyano, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy or C1-C4-haloalkoxy; with the proviso that at most three of A1 to A5 are N; as well as its acceptable salts, enantiomers, diastereomers, tautomers, and N-oxides.