Patent ID: 6200970
Filing Date: 2001-03-13
Classification: A61P,C07D

Abstract:
A compound of formula I ##STR5##in whichX means hydrogen or halogen,Y means --NR.sup.3 -- or --N.dbd.,R.sup.1 and R.sup.2 are the same or different and mean hydrogen, C.sub.1 -C.sub.6 alkyl, nitro, halogen, the group --NR.sup.8 R.sup.9, --O--C.sub.1-4 alkyl, --CF.sub.3, OH or C.sub.1-6 alkanoyloxy,R.sup.3 means hydrogen, the group --CO--R.sup.10, C.sub.1-6 alkyl or C.sub.3-7 cycloalkyl,R.sup.4 means optionally substituted C.sub.1 -C.sub.6 alkyl,R.sup.5 means hydrogen orR.sup.4 and R.sup.5 together mean oxygen,R.sup.6 means C.sub.1-4 alkyl,R.sup.8 and R.sup.9 are the same or different and mean hydrogen, C.sub.1 -C.sub.6 alkyl or --CO--C.sub.1-6 alkylR.sup.10 means hydrogen, optionally substituted C.sub.1 -C.sub.6 alkyl, optionally substituted C.sub.6-10 aryl, the group --NR.sup.11 R.sup.12, --O--C.sub.1-6 alkyl, C.sub.3-7 cycloalkyl, C.sub.2-6 alkenyl or --O--C.sub.3-7 cycloalkyl,R.sup.11 and R.sup.12 are the same or different and mean hydrogen, optionally substituted C.sub.1 -C.sub.6 alkyl or optionally substituted C.sub.6-10 aryl and--C.sub.... C.sub.... means a double bond or single bondsor an isomer or physiologically compatible salt thereofwith the proviso that the compound is not 1-(3-chlorophenyl)-4-methyl-8-methoxy, 5H-2,3-benzodiazepine.