Patent ID: 6127364
Filing Date: 2000-10-03
Classification: A01N,B27K,C07C,C07D

Abstract:
An oxadiazine derivative of the formula ##STR81## in which R.sup.1 and R.sup.2 independently of one another each represent a residue selected from the group consisting of hydrogen, respectively optionally halogen-substituted alkyl, hydroxyalkyl, alkanoyloxyalkyl, alkoxyalkyl, arylalkoxyalkyl, mercaptoalkyl, alkylthioalkyl, alkylsulphinylalkyl, alkylsulphonylalkyl, carboxyalkyl, alkoxycarbonylalkyl, aryloxycarbonylalkyl, arylalkyloxycarbonylalkyl, carbamoylalkyl, aminoalkyl, alkylaminoalkyl, dialkylaminoalkyl, alkoxycarbonylaminoalkyl, alkylcarbonyl, cycloalkylcarbonyl, cycloalkyl, cycloalkylalkyl, aryl, arylalkyl, arylcarbonyl, and a 5- or 6-membered hetaryl substituent selected from the group consisting of thienyl, thiazolyl, or pyridyl, and 5- or 6-membered hetaryl, C.sub.1 -C.sub.4 -alkyl or indolyl-C.sub.1 -C.sub.4 -alkyl, each of which is optionally substituted by a residue selected from the group consisting of fluorine-, chlorine-, bromine-, iodine-, hydroxyl-, nitro-, cyano-,amino-, C.sub.1 -C.sub.4 -alkylamino, di-(C.sub.1 -C.sub.4) alkylamino, benzylamino, dibenzylamino, and protected amino selected from the group consisting of acetyl-, t-butoxycarbonyl-, benzyloxycarbonyl- or FMOC-amino, C.sub.1 -C.sub.4 -alkoxy and C.sub.1 -C.sub.2 -halogenoalkoxy, orR.sup.1, R.sup.2 and the two linking nitrogen atoms represent a 5 to 8 membered saturated or unsaturated heterocyclic ring optionally substituted by a substituent selected from the group consisting of fluorine-, chlorine-, bromine-, hydroxyl-, nitro-, cyano-, C.sub.1 -C.sub.4 -alkyl-, C.sub.1 -C.sub.4 -halogenoalkyl-, C.sub.1 -C.sub.4 -alkoxy-, and C.sub.1 -C.sub.2 -halogenoalkoxy,R.sup.3 and R.sup.4 independently of one another each represent a residue selected from the group consisting of hydrogen, respectively optionally halogen-substituted alkyl, alkenyl, hydroxyalkyl, alkanoyloxyalkyl, alkoxyalkyl, arylalkoxyalkyl, mercaptoalkyl, alkylthioalkyl, alkylsulphinylalkyl, alkylsulphonylalkyl, alkoxycarbonylalkyl, aryloxycarbonylalkyl, arylalkyloxycarbonylalkyl, carbamoylalkyl, aminoalkyl, alkylaminoalkyl, dialkylaminoalkyl, alkylcarbonyl, cycloalkylcarbonyl, cycloalkyl, cycloalkylalkyl, aryl, arylalkyl, and a 5- or 6- membered hetaryl, selected from the group consisting of thienyl, thiazolyl, pyridyl, indolyi, benzo-1,3-dioxolyl, and 5- or 6-membered hetaryl-C.sub.1 -C.sub.4 -alkyl selected from the group consisting of thienylmethyl, thiazolylmethyl, imidazolylmethyl, pyridylmethyl, indolyl-C.sub.1 -C.sub.4 -alkyl, each of which is optionally substituted by fluorine, chlorine, bromine, iodine, hydroxyl, cyano, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.4 -halogenoalkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -halogenoalkoxy, benzyloxy and silyloxy which is trisubstituted bv C.sub.1 -C.sub.4 -alkyl and/or phenyl orR.sup.3 and R.sup.4 together represent alkylene or the radical (a) ##STR82## wherein R.sup.5 and R.sup.6 independently of one another each represent a residue selected from the group consisting of hydrogen, respectively optionally halogen substituted alkyl, alkenyl, hydroxyalkyl, alkanoyloxyalkyl, alkoxyalkyl, arylalkoxyalkyl, mercaptoalkyl, alkylthioalkyl, alkylsulphinylalkyl, alkylsulphonylalkyl, alkoxycarbonylalkyl, aryloxycarbonylalkyl, aminoalkyl, alkylaminoalkyl, dialkylaminoalkyl, alkylcarbonyl, cycloalkyl, cycloalkylalkyl, aryl, arylalkyl, and 5- or 6-membered hetaryl,Q.sup.1 and Q.sup.2 independently of one another each represent oxygen or sulphur, except for 6,6-diphenyl-(1,3,4)-oxadiazinane-2,5-dione.