Patent ID: 7244741
Filing Date: 2007-07-17
Classification: A61P,C07D

Abstract:
1. A compound according to the general formula Ia or Ib: wherein in each, R1 is H, C R2 is C  —CH═N—NHSO wherein, m is 1 to 6, o is 1, p is 1 to 2m+o; m is 2 to 6, o is −1, p is 1 to 2m+o; or m is 4 to 6, o is −2, p is 1 to 2m+o; and Y independently from each other is selected from the group consisting of halogen, OH, OR21, NH wherein X′ is NR215, O, or S; and R211, R212, R213, R214, and R215 are independently from each other H or C R21, R22 are independently from each other C R23 independently of R21, is R21, CH R24 independently of R21, is R21, H, CN, COCH R25 independently of R21, is R21, H, CN, COCH R24, R25 together are C R3 is H, F, Cl, Br, I, OH, OR31, NO R31, 32 independently from each other are C R5, R6 Independently from each other are H, C wherein, m is 1 to 6, o is 1, p is 1 to 2m+o; m is 2 to 6, o is −1, p is 1 to 2m+o; or m is 4 to 6, o is −2, p is 1 to 2m+o; and Y independently from each other is selected from the group consisting of halogen, OH, OR21, NH R4, R7, R8 independently from each other are H, C R41 independently from R21 is R21; X1 is O, S, NH, N—C X2 is O, S, NH, N—C Y1 is O, or N—R9, wherein R9, independently from R5, is R5; Y2 is O, or N—R10, wherein R10, independently from R5, is R5; and, if Y1 or Y2 are N—R9 or N—R10, X2—R6 may be H; Y3 is O, S, or NH; or a stereoisomer, tautomer or physiologically tolerable salt thereof.