Patent ID: 8785431
Filing Date: 2014-07-22
Classification: A61K,A61P,C07D,C07K

Abstract:
1. A compound selected from the group consisting of: (1S,9S)-1-(ethoxycarbonyloxy)ethyl 9-[[(1S)-1-ethoxycarbonyl-3-phenylpropyl]amino]-10-oxooctahydro-1H-pyridazino[1,2-a][1,2]diazepine-1-carboxylate; (1S,9S)-1-(cyclohexyloxycarbonyloxy)ethyl 9-[[(1S)-1-ethoxycarbonyl-3-phenylpropyl]amino]-10-oxooctahydro-1H-pyridazino[1,2-a][1,2]diazepine-1-carboxylate; (1S,9S)-2-morpholinoethyl 9-[[(1S)-1-ethoxycarbonyl-3-phenylpropyl]amino]-10-oxooctahydro-1H-pyridazino[1,2-a][1,2]diazepine-1-carboxylate; (1S,9S)-1-(isopropyloxycarbonyloxy)ethyl 9-[[(1S)-1-ethoxycarbonyl-3-phenylpropyl]amino]-10-oxooctahydro-1H-pyridazino[1,2-a][1,2]diazepine-1-carboxylate; (1S,9S)-1-(acetoxy)ethyl 9-[[(1S)-1-ethoxycarbonyl-3-phenylpropyl]amino]-10-oxooctahydro-1H-pyridazino[1,2-a][1,2]diazepine-1-carboxylate; (1S,9S)-1-(2,2-dimethylpropanoyloxy)ethyl 9-[[(1S)-1-ethoxycarbonyl-3-phenylpropyl]amino]-10-oxooctahydro-1H-pyridazino[1,2-a][1,2]diazepine-1-carboxylate; and (1S,9S)-1-(2-morpholinoacetoxy)ethyl 9-[[(1S)-1-ethoxycarbonyl-3-phenylpropyl]amino]-10-oxooctahydro-1H-pyridazino[1,2-a][1,2]diazepine-1-carboxylate.