Patent ID: 7087759
Filing Date: 2006-08-08
Classification: A61P,C07D,C07K

Abstract:
1. A compound, including all enatiomeric and diasteriomeric forms and pharmaceutically acceptable salts thereof, said compound having the formula: wherein the carbon atoms marked with an asterisk can have any stereochemical configuration; W has the formula: R is phenyl or substituted phenyl; wherein R a) rings consisting of: b) hydrogen; c) a unit selected from the group consisting of —CH d) two of R e) mixtures thereof; Y is a pendant unit containing at least one heteroatom having the formula: wherein R i) —C(O)OCH ii) —C(O)OCH iii) —C(O)OCH iv) —C(O)OCH v) —C(O)OCH(CH vi) —C(O)OCH vii) —C(O)OCH viii) —C(O)OCH ix) —C(O)OCH x) —OC(O)CH xi) —OC(O)CH xii) —OC(O)CH xiii) —OC(O)CH(CH xiv) —OC(O)CH xv) —OC(O)CH xvi) —OC(O)CH xvii) —OC(O)CH xviii) —OC(O)CH an amide selected from the group consisting of: i) —C(O)NHCH ii) —C(O)NHCH iii) —C(O)NHCH iv) —C(O)NHCH v) —C(O)NHCH(CH vi) —C(O)NHCH vii) —C(O)NHCH viii) —C(O)NHCH ix) —C(O)NHCH x) —NHC(O)CH xi) —NHC(O)CH xii) —NHC(O)CH xiii) —NHC(O)CH(CH xiv) —NHC(O)CH xv) —NHC(O)CH xvi) —NHC(O)CH xvii) —NHC(O)CH xviii) —NHC(O)CH a unit selected from the group consisting of: a) —C(X)N(R b) —C(X)NR c) —NR d) —NHN(R wherein X is ═O, ═S, or ═NR the index b is from 1 to 4; Z is a pendant unit, which contains an aromatic carbocyclic ring; said unit having the formula: wherein R