Patent ID: 8569313
Filing Date: 2013-10-29
Classification: A61P,C07D

Abstract:
1. A compound according to the formula (I) or a salt thereof, wherein R (i) an aryl residue, which may be partially or wholly hydrogenated, (ii) a heteroaryl residue, which may be partially or wholly hydrogenated, (iii) a non-hydrogenated aryl residue, (iv) a non-hydrogenated heteroaryl residue, (v) a heteroaryl residue with one or two nitrogen atoms, (vi) a phenyl residue, (vii) a pyridyl residue, (viii) a pyrimidine residue, (ix) an indole residue, (x) a tetrahydropyridyl residue, (xi) a piperidinon residue, or (xii) a pyridazinone residue; and R (i) a ramified or straight chain alkyl residue having 1-6 carbon atoms, wherein one or more methylene groups may be replaced by oxygen or nitrogen, (ii) a ramified or straight chain amino alkyl residue having 1-6 carbon atoms, (iii) a ramified or straight chain guanidine alkyl residue having 1-6 carbon atoms, (iv) —(CH (v) R or R (i) a ramified or straight chain hydroxy alkyl residue having 1 to 6 carbon atoms, (ii) a straight chain aminoalkyl residue, (iii) a 3-azetidin-C(═O)—NH-residue, or (iv) an unramified n-amino butyl residue; and R (i) a ramified or straight chain aminoalkyl residue having 1-6 carbon atoms, (ii) a ramified or straight chain guanidino alkyl residue having 1-6 carbon atoms, (iii) a straight chain amino ethyl residue, or (iv) R or R (i) a H (ii) a HO—(CH (iii) a 3-azetidin-C(═O)—NH-residue; and R (i) each independently a non-basic residue, (ii) R (iii) R (iv) R and R