Patent ID: 6359136
Filing Date: 2002-03-19
Classification: A61P,C07D

Abstract:
An azaindole of formula II whereinone of X and Y is N, and the other of X and Y is CH; R2 is â€”X2â€”(CH2)mâ€”NRaRb in which X2 is a direct bond, methylene, O or S; m is 1, 2, 3, 4 or 5; provided that when m is 1, then X2 is a direct bond; and Ra and Rb are independently hydrogen or (1-3C)alkyl or the group NRaRb is pyrrolidino, piperidino, or morpholino; or R2 is â€”X2â€”(CH2)n-Rf in which X2 is a direct bond, methylene or O; n is 1, 2 or 3; and Rf is 5-tetrazolyl, carboxy, (1-4C) alkoxy )carbonyl or hydroxymethyl.