Patent ID: 8912329
Filing Date: 2014-12-16
Classification: A61K,A61P,C07D

Abstract:
1. A pharmaceutical composition comprising a compound of formula wherein R unsubstituted phenyl or phenyl substituted by one, two or three substituents selected from C unsubstituted 2-, 3- or 4-pyridyl or 2-, 3- or 4-pyridyl substituted by one or two substituents selected from C unsubstituted indolyl or indolyl substituted by one or two substituents selected from C R R R unsubstituted 2- or 3-furanyl or 2- or 3-furanyl substituted by one or two substituents selected from C unsubstituted 2- or 3-thienyl or 2- or 3-thienyl substituted by one or two substituents selected from C R A is selected from wherein—represents the bond to C(═X or A together with —C(═X wherein → represents the bond to R X X and a compound of formula wherein R R R R R R wherein the sugar residue in R L- or D-hexofuranosyl selected from aldohexoses allose, altrose, glucose, mannose, gulose, idose, galactose and talose of formula 4 below; L- or D-hexofuranosyl selected from ketohexoses fructose, psicose, sorbose and tagatose of formula 5 below; L- or D-pyranosyl selected from aldohexoses allose, altrose, glucose, mannose, gulose, idose, galctose and talose of formula 6 below; or L- or D-pyranosyl selected from ketohexoses fructose, psicose, sorbose and tagatose of formula 7 below; in which one, two, three or four hydroxy groups can be methylated, benzylated or acetylated, or one hydroxy group can be replaced by hydrogen, halogen, methylamino, ethylamino, or acetamido.