Patent ID: 7939467
Filing Date: 2011-05-10
Classification: A01N,A61P,C07D,Y02P

Abstract:
1. A 4-(3-aminobenzoyl)-1-ethylpyrazole of the formula (I), or a salt thereof in which R R Y is hydrogen, (C m is 0, 1, 2 or 3, with the proviso that (1-ethyl-5-hydroxy-1H-pyrazol-4-yl)[2-methyl-3-(methylamino)-4-(methylsulfonyl) phenyl]methanone, [3-(ethylamino)-2-methyl-4-(methylsulfonyl)phenyl](1-ethyl-5 -hydroxy-1H-pyrazol-4-yl) methanone, (1-ethyl-5-hydroxy-1H-pyrazol-4-yl)[2-methyl-4-(methylsulfonyl)-3-(propylamino) phenyl]methanone, (1-ethyl-5-hydroxy-1H-pyrazol-4-yl){2-methyl-3-[(1-methylethyl)amino]-4-(methyl-sulfonyl) phenyl}methanone, [3-(butylamino)-2-methyl-4-(methylsulfonyl)phenyl](1-ethyl-5-hydroxy-1H-pyrazol-4-yl) methanone, (1-ethyl-5-hydroxy-1H-pyrazol-4-yl){3-[(2-methoxyethyl)amino]-2-methyl-4- (methylsulfonyl)phenyl}methanone, [3-(cyclopropylamino)-2-methyl-4-(methylsulfonyl)phenyl](1-ethyl-5-hydroxy-1H-pyrazol-4-yl) methanone, (1-ethyl-5-hydroxy-1H-pyrazol-4-yl)[2-methyl-4-(methylsulfonyl)-3-(prop-2-en-1-ylamino) phenyl]methanone and [3-(dimethylamino)-2-methyl-4-(methylsulfonyl)phenyl](1-ethyl-5-hydroxy-1H-pyrazol-4-yl) methanone are excluded.