Patent ID: 6759407
Filing Date: 2004-07-06
Classification: A01N,A61P,C07D

Abstract:
A compound of formula (I); whereinR1 is hydrogen or a radical from the group C1-C4alkyl, formyl, C1-C6alkylcarbonyl, C1-C4alkylsulfonyl, aryl, arylsulfonyl, arylcarbonyl, heterocyclyl whereby said heterocyclyl is selected from the group consisting of dioxolanyl, pyrrolidinyl, piperidinyl, morpholinyl, pyrrolyl, furyl, thienyl, imidazolyl, tetrahydrofuryl, tetrahydropyranyl, dihydrofuryl, dihydropyranyl, isoxazolyl, oxazolyl, thiazolyl, oxazolinyl, oxazolidinyl, imidazolinyl, imidazolidinyl and dioxanyl, and C1-C6alkyl substituted with said heterocyclyl, whereby the heterocyclyl moiety is unsubstituted or mono- or poly-substituted by identical or different substituents; the said substituents being C1-C4alkyl, C1-C4alkoxy, C1-C4alkylthio, C1-C4haloalkyl, halogen, hydroxy, cyano, nitro, amino, C1-C4alkylamino, C1-C4alkyl)2amino, alkoxycarbonyl, C1-C4alkylsulfonyl and arylsulfonyl; X is CH or N; Y is an electron-withdrawing radical, selected from the group consisting of cyano, nitro and C1-C6haloalkyl-carbonyl; T and U together form a C1-C4alkylene bridge which is unsubstituted or substituted by a radical R1, or T and U together with the group â€”Nâ€”Câ€”Nâ€” form a saturated or unsaturated 5- or 6-membered heterocyclic ring which may in addition contain as further hetero atom O or S or the hetero group â€”N(C1-C6alkyl)-; R2 is hydrogen or C1-C6alkyl; R2â€² is hydrogen or C1-C6alkyl; and R is C1-C20alkyl, C2-C20alkenyl, C2-C6alkynyl or heterocyclyl, each of those radicals being unsubstituted or substituted by one or more identical or different substituents, the said substituents being selected from the group halogen, cyano, nitro, hydroxy, C1-C6alkoxy, C1-C6alkylthio, C1-C6haloalkyl, C1-C6haloalkoxy and phenyl; whereby heterocyclyl is selected from the group consisting of dioxolanyl, pyrrolidinyl, piperidinyl, morpholinyl, pyrrolyl, furyl, thienyl, imidazolyl, tetrahydrofuryl, tetrahydropyranyl, dihydrofuryl, dihydropyranyl, isoxazolyl, oxazolyl, thiazolyl, oxazolinyl, oxazolidinyl, imidazolinyl, imidazolidinyl and dioxanyl; or is C3-C7cycloalkyl that is unsubstituted or mono- or poly-substituted by identical or different substituents selected from halogen, cyano, nitro, hydroxy, C1-C6alkyl, C2-C6alkenyl, C2-C6alkynyl, C1-C6alkoxy, C1-C6alkylthio, C1-C6haloalkyl, C1-C20haloalkoxy and phenyl; wherein each phenyl moiety is itself unsubstituted or mono- or poly-substituted by identical or different substituents selected from halogen, cyano, nitro, hydroxy, C1-C6alkyl, C1-C6alkoxy, C1-C6alkylthio, C1-C6haloalkyl and C1-C20haloalkoxy; oris phenyl phenoxyphenyl each of which is unsubstituted or mono- or poly-substituted by identical or different substituents selected from halogen, cyano, nitro, hydroxy, C1-C6alkyl, C1-C6alkoxy, C1-C6alkylthio, C1-C6haloalkyl and C1-C20haloalkoxy.