Patent ID: 8691990
Filing Date: 2014-04-08
Classification: A61P,C07D,C07F

Abstract:
1. A compound selected from the group consisting of: 6-Bromo-N-phenylimidazo[1,2-a]pyridine-2-carboxamide; 6-Iodo-N-phenylimidazo[1,2-a]pyridine-2-carboxamide; N-Phenyl-6-cyanoimidazo[1,2-a]pyridine-2-carboxamide; 6-Trimethylstannyl-N-phenylimidazo[1,2-a]pyridine-2-carboxamide; N-Phenyl-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)imidazo[1,2-a]pyridine-2-carboxamide and the hydrobromide (1:1) thereof; 2-Phenylcarbamoylimidazo[1,2-a]pyridine-6-boronic acid hydrochloride (1:1); N-Phenyl-6-vinylimidazo[1,2-a]pyridine-2-carboxamide; 6-Formyl-N-phenylimidazo[1,2-a]pyridine-2-carboxamide; 6-(2-Bromoacetyl)-N-phenylimidazo[1,2-a]pyridine-2-carboxamide; 6-(1-Ethoxyvinyl)-N-phenylimidazo[1,2-a]pyridine-2-carboxamide; N-(3,5-Difluorophenyl)-6-iodoimidazo[1,2-a]pyridine-2-carboxamide; 6-(6-{[(1,1-Dimethylethoxy)carbonyl]amino}pyrid-2-yl)imidazo[1,2-a]pyridine-2-carboxylic acid; Ethyl 6-(6-aminopyrid-2-yl)imidazo[1,2-a]pyridine-2-carboxylate; Ethyl 6-(6-{[(1,1-dimethylethoxy)carbonyl]amino}pyrid-2-yl)imidazo[1,2-a]pyridine-2-carboxylate; Ethyl 6-(6-{bis[(1,1-dimethylethoxy)carbonyl]amino}pyrid-2-yl)imidazo[1,2-a]pyridine-2-carboxylate; 6-(Pyrid-2-yl)imidazo[1,2-a]pyridine-2-carboxylic acid; Ethyl (6-pyrid-2-yl)imidazo[1,2-a]pyridine-2-carboxylate; 6-(1-Triphenylmethyl-1H-imidazol-4-yl)imidazo[1,2-a]pyridine-2-carboxylic acid; Ethyl 6-(1-triphenylmethyl-1H-imidazol-4-yl)imidazo[1,2-a]pyridine-2-carboxylate; 6-(2-{[(1,1-Dimethylethoxy)carbonyl]amino}thiazol-4-yl)imidazo[1,2-a]pyridine-2-carboxylic acid; Ethyl 6-(2-{[(1,1-dimethylethoxy)carbonyl]amino}thiazol-4-yl)imidazo[1,2-a]pyridine-2-carboxylate; 6-(1H-Pyrrol-3-yl)imidazo[1,2-a]pyridine-2-carboxylic acid and the hydrochloride (1:1) thereof; Ethyl 6-[1-(triisopropylsilyl)-1H-pyrrol-3-yl]imidazo[1,2-a]pyridine-2-carboxylate; 6-(1H-Pyrazol-3-yl)imidazo[1,2-a]pyridine-2-carboxylic acid; Ethyl 6-(1H-pyrazol-3-yl)imidazo[1,2-a]pyridine-2-carboxylate; 6-(1H-Pyrazol-4-yl)imidazo[1,2-a]pyridine-2-carboxylic acid; Ethyl 6-(1H-pyrazol-4-yl)imidazo[1,2-a]pyridine-2-carboxylate; 6-(Furan-2-yl)imidazo[1,2-a]pyridine-2-carboxylic acid; Ethyl 6-(furan-2-yl)imidazo[1,2-a]pyridine-2-carboxylate; 6-(Furan-3-yl)imidazo[1,2-a]pyridine-2-carboxylic acid; Ethyl 6-(furan-3-yl)imidazo[1,2-a]pyridine-2-carboxylate; 6-[5-(Hydroxymethyl)furan-2-yl]imidazo[1,2-a]pyridine-2-carboxylic acid; Ethyl 6-(5-formylfuran-2-yl)imidazo[1,2-a]pyridine-2-carboxylate; Ethyl 6-[5-(hydroxymethyl)furan-2-yl]imidazo[1,2-a]pyridine-2-carboxylate; 6-(Thiophen-3-yl)imidazo[1,2-a]pyridine-2-carboxylic acid; Ethyl 6-(thiophen-3-yl)imidazo[1,2-a]pyridine-2-carboxylate; 6-(Oxazol-2-yl)imidazo[1,2-a]pyridine-2-carboxylic acid; Ethyl 6-(oxazol-2-yl)imidazo[1,2-a]pyridine-2-carboxylate; 6-(1H-1,2,4-Triazol-3-yl)imidazo[1,2-a]pyridine-2-carboxylic acid; Ethyl 6-[ethoxy(imino)methyl]imidazo[1,2-a]pyridine-2-carboxylate; Ethyl 6-[hydrazino(imino)methyl]imidazo[1,2-a]pyridine-2-carboxylate; Ethyl 6-(1H-1,2,4-triazol-3-yl)imidazo[1,2-a]pyridine-2-carboxylate; 6-(1H-1,2,3-Triazol-4-yl)imidazo[1,2-a]pyridine-2-carboxylic acid; Ethyl 6-(1H-1,2,3-triazol-4-yl)imidazo[1,2-a]pyridine-2-carboxylate; 6-(1H-1,2,3-Triazol-4-yl)imidazo[1,2-a]pyridine-2-carboxylic acid; Ethyl 6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)imidazo[1,2-a]pyridine-2-carboxylate hydrobromide (1:1); and 2-Ethoxycarbonylimidazo[1,2-a]pyridine-6-boronic acid.