Patent ID: 8008304
Filing Date: 2011-08-30
Classification: A61P,C07D

Abstract:
1. A substituted propiolic acid amide of the formula I, in which a, b and c, mutually independently, in each case denote 0 or 1, wherein the sum of a, b and c is equal to 1, 2 or 3; A denotes one of the following residues Q and U respectively denote CR R and V respectively denote CR K and W respectively denote CR P and T respectively denote O, S or NR with the proviso that compounds are excluded in which P denotes S, Q denotes N, R denotes CR R R or R or R wherein d denotes 1, 2 or 3 and b denotes 0 or 1 and c denotes 0 or 1; or R wherein e denotes 1, 2, 3 or 4 and, in this case, b denotes 0 or 1 and c denotes 0; or R wherein f denotes 1, 2, 3 or 4, and, in this case, c denotes 0; or R wherein g denotes 1, 2 or 3; or R wherein h denotes 1, 2, 3 or 4 and, in this case, b denotes 0 or 1 and a denotes 0; or R wherein k denotes 1, 2, 3 or 4, and, in this case, a denotes 0; or R wherein m denotes 1, 2 or 3; R R R and R in each case optionally in the form of one of the pure stereoisomers thereof, in the form of one of the racemates thereof or in the form of a mixture of stereoisomers in any mixing ratio, or in each case in the form of a corresponding salt.