Patent ID: 6239306
Filing Date: 2001-05-29
Classification: A01N,C07C,C07D

Abstract:
A compound of the formula (I) or salts thereof, ##STR26##in whichR.sup.1 is CO--Q--R.sup.8,R.sup.2 and R.sup.3 independently of one another are H or (C.sub.1 -C.sub.4)alkyl,R.sup.4 is H, (C.sub.1 -C.sub.8)alkyl which is unsubstituted or is substituted by one or more radicals from the group consisting of halogen, (C.sub.1 -C.sub.4)alkoxy, (C.sub.1 -C.sub.4)alkylthio, (C.sub.1 -C.sub.4)alkylsulfinyl, (C.sub.1 -C.sub.4)alkylsulfonyl, ((C.sub.1 -C.sub.4)alkoxy)carbonyl and CN, or is (C.sub.3 -C.sub.6)alkenyl which is unsubstituted or is substituted by one or more halogen atoms, or is (C.sub.3 -C.sub.6)alkynyl which is unsubstituted or is substituted by one or more halogen atoms, or is hydroxyl, (C.sub.1 -C.sub.4)alkoxy, (C.sub.1 -C.sub.4)alkyl)carbonyl or (C.sub.1 -C.sub.4)alkylsulfonyl, each of the three latter radicals being unsubstituted or substituted in the alkyl moiety by one or more halogen atoms or by (C.sub.1 -C.sub.4)alkoxy or (C.sub.1 -C.sub.4)alkylthio, or is phenylsulfonyl in which the phenyl radical is unsubstituted or substituted, andR.sup.5 is (C.sub.1 -C.sub.4)alkylsulfonyl or (C.sub.3 -C.sub.6)alkenylsulfonyl, each of the two latter radicals being unsubstituted or substituted by one or more halogen atoms or by (C.sub.1 -C.sub.4)alkoxy or (C.sub.1 -C.sub.4)alkylthio, or is phenylsulfonyl or phenylcarbonyl, the phenyl radical in each of the two latter radicals being unsubstituted or substituted, or is mono- or di-((C.sub.1 -C.sub.4)alkyl)aminosulfonyl or ((C.sub.1 -C.sub.6)alkyl)carbonyl, each of the three latter radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen, (C.sub.1 -C.sub.4)alkoxy, (C.sub.1 -C.sub.4)alkylthio, (C.sub.1 -C.sub.4)alkylsulfinyl, (C.sub.1 -C.sub.4)alkylsulfonyl, ((C.sub.1 -C.sub.4)alkyl)carbonyl, ((C.sub.1 -C.sub.4)alkoxy)carbonyl and CN, or is formyl, a group of the formula --CO--CO--R' in which R'=H, OH, (C.sub.1 -C.sub.4)alkoxy or (C.sub.1 -C.sub.4)alkyl, or is ((C.sub.3 -C.sub.6)cycloalkyl)carbonyl, ((C.sub.2 -C.sub.6)alkenyl)carbonyl or ((C.sub.2 -C.sub.6)alkynyl)carbonyl, each of the three latter radicals being unsubstituted or substituted by one or more halogen atoms, or is a group of the formula ##STR27##orR.sup.4 and R.sup.5 together are a chain of the formula (--CH.sub.2).sub.m B-- or --B.sup.1 --(CH.sub.2).sub.m1 --B--, the chain being unsubstituted or substituted by one or more (C.sub.1 -C.sub.3)alkyl radicals and m being 3 or 4 or m.sup.1 being 2 or 3, andW is an oxygen or sulfur atom,B and B.sup.1 independently of one another are SO.sub.2 or CO,Q is O, S or --NR.sup.13 --,T is O or S,R.sup.6 is H, (C.sub.1 -C.sub.4)alkyl, (C.sub.1 -C.sub.4)alkoxy, [(C.sub.1 -C.sub.4)alkyl]carbonyl or ((C.sub.1 -C.sub.4)alkoxy)carbonyl, each of the 4 latter radicals being unsubstituted or substituted in the alkyl moiety by one or more halogen atoms, or is halogen, NO.sub.2 or CN,R.sup.8 is H, (C.sub.1 -C.sub.4)alkyl, (C.sub.3 -C.sub.4)alkenyl or (C.sub.3 -C.sub.4)alkynyl, each of the three latter radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen, (C.sub.1 -C.sub.4)alkoxy, (C.sub.1 -C.sub.4)alkylthio, ((C.sub.1 -C.sub.4)alkyl)carbonyl and ((C.sub.1 -C.sub.4)alkoxy)carbonyl,R.sup.9 is (C.sub.1 -C.sub.4)alkyl, (C.sub.3 -C.sub.4)alkenyl or (C.sub.3 -C.sub.4)alkynyl, each of the three latter radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen, (C.sub.1 -C.sub.4)alkoxy, (C.sub.1 -C.sub.4)alkylthio, ((C.sub.1 -C.sub.4)alkyl)carbonyl and ((C.sub.1 -C.sub.4)alkoxy)carbonyl,R.sup.10 and R.sup.11 independently of one another are H, (C.sub.1 -C.sub.4)alkyl, (C.sub.3 -C.sub.4)alkenyl or (C.sub.3 -C.sub.4)alkynyl, each of the three latter radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen, (C.sub.1 -C.sub.4)alkoxy, (C.sub.1 -C.sub.4)alkylthio, ((C.sub.1 -C.sub.4)alkyl)carbonyl and ((C.sub.1 -C.sub.4)alkoxy)carbonyl,the radicals R.sup.12 together with the nitrogen atom are a heterocyclic ring having 5 or 6 ring members, which may contain further heteroatoms from the group consisting of N, O and S in the possible oxidation states and is unsubstituted or is substituted by (C.sub.1 -C.sub.4)alkyl or the oxo group, or is benzo-fused,R.sup.13 is H, (C.sub.1 -C.sub.4)alkyl, (C.sub.3 -C.sub.4)alkenyl or (C.sub.3 -C.sub.4)alkynyl, each of the three latter radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen, (C.sub.1 -C.sub.4)alkoxy, (C.sub.1 -C.sub.4)alkylthio.