Patent ID: 7893049
Filing Date: 2011-02-22
Classification: A61P,C07D

Abstract:
1. A compound of formula (1), wherein R R R R R R two R n is equal to 0, 1 or 2, or R R each R each R each R each R or a pharmacologically acceptable salt thereof, with the proviso that following compounds are not included: N-[1-(4-morpholin-4-ylmethyl-phenyl)-3-pyridin-2-yl-4,5-dihydro-1H-pyrazolo[4,3-g]benzothiazol-7-yl]-acetamide, N-[1-(4-dimethylaminomethyl-phenyl)-3-pyridin-3-yl-4,5-dihydro-1H-pyrazolo[4,3-g]benzothiazol-7-yl]-acetamide, N-{1-[4-(benzylamino-methyl)-2-chloro-phenyl]-3-pyrazin-2-yl-4,5-dihydro-1H-pyrazolo[4,3-g]benzothiazol-7-yl}-acetamide and N-(1-{2-chloro-4-[(1-cyclopentyl-piperidin-4-ylamino)-methyl]-phenyl}-3-pyrazin-2-yl-4,5-dihydro-1H-pyrazolo[4,3-g]benzothiazol-7-yl)-acetamide.