Patent ID: 6815443
Filing Date: 2004-11-09
Classification: A61P,C07C,C07D

Abstract:
A compound of formula I, whereinR1 and R2 independently of one another are C1-6 alkyl, branched or unbranched, saturated or unsaturated, unsubstituted or singly or multiply substituted, or R1 and R2 together form a (CH2)2-9 ring that may optionally be substituted by C1-8 alkyl, which is branched or unbranched, saturated or unsaturated, unsubstituted or singly or multiply substituted; or by aryl, unsubstituted or singly or multiply substituted, R3 and R4 independently of one another are C1-6 alkyl, branched or unbranched, saturated or unsaturated, unsubstituted or singly or multiply substituted; C3-6 cycloalkyl, saturated or unsaturated, unsubstituted or singly or multiply substituted; or phenyl, benzyl or phenethyl, unsubstituted or singly or multiply substituted, orR3 and R4 together form a ring and denote CH2CH2OCH2CH2, CH2CH2NR22CH2CH2 or (CH2)3-6, wherein R22 is H; C1-10 alkyl or C3-10 cycloalkyl that is saturated or unsaturated, branched or unbranched, singly or multiply substituted or unsubstituted; aryl or heteroaryl, singly or multiply substituted or unsubstituted; or aryl bound via C1-3 alkyl that is saturated or unsaturated, via C3-10 cycloalkyl or via heteroaryl, singly or multiply substituted or unsubstituted, R5 is C1-10 alkyl, saturated or unsaturated, branched or unbranched, singly or multiply substituted or unsubstituted; C3-9 cycloalkyl, saturated or unsaturated, aryl, heteroaryl, aryl bound via saturated or unsaturated C1-3 alkyl; C3-10 cycloalkyl bound via saturated or unsaturated C1-3 alkyl; or heteroalkyl bound via saturated or unsaturated C1-3 alkyl, wherein all aryl, heteroaryl and cycloalkyl may independently of one another be unsubstituted or may be independently singly or multiply substituted with F, Cl, Br, I, OR18, SR18, SO2R18, SO2OR18, CN, COOR18, NR19R20; C1-C10 alkyl, saturated or unsaturated, branched or unbranched, singly or multiply substituted or unsubstituted; C3-9 cycloalkyl, saturated or unsaturated, unsubstituted or singly or multiply substituted; aryl or heteroaryl, in each case unsubstituted or singly or multiply substituted; or aryl, C3-9 cycloalkyl or heteroaryl bound via saturated or unsaturated C1-3 alkyl, which may be unsubstituted or singly or multiply substituted, wherein R18 is H; C1-10 alkyl, saturated or unsaturated, branched or unbranched, unsubstituted or singly or multiply substituted; C3-9 cycloalkyl, saturated or unsaturated, unsubstituted or singly or multiply substituted; aryl or heteroaryl, unsubstituted or singly or multiply substituted; or aryl, C3-9 cycloalkyl or heteroaryl bound via saturated or unsaturated C1-3 alkyl which may be unsubstituted or singly or multiply substituted; and wherein R19 and R20 independently of one another are H; C1-10 alkyl, saturated or unsaturated, branched or unbranched, unsubstituted or singly or multiply substituted; C3-9 cycloalkyl, saturated or unsaturated, unsubstituted or singly or multiply substituted; aryl or heteroaryl, unsubstituted or singly or multiply substituted; or aryl, C3-9 cycloalkyl or heteroaryl bound via saturated or unsaturated C1-3 alkyl which may be unsubstituted or singly or multiply substituted; or R19 and R20 together form CH2CH2OCH2CH2, CH2CH2NR21CH2CH2 or (CH2)3-6, where R21 is H; substituted or unsubstituted phenyl; C1-10 alkyl, saturated or unsaturated, branched or unbranched, unsubstituted or singly or multiply substituted; R6 is C1-10 alkyl, saturated or unsaturated, branched or unbranched, singly or multiply substituted or unsubstituted; or C5-7 cycloalkyl, aryl or heteroaryl, unsubstituted or singly or multiply substituted; R7 is H; aryl or heteroaryl; unsubstituted or singly or multiply substituted, or a derivative thereof in the form of an acid, a base, a salt, or a solvate.