Patent ID: 6753429
Filing Date: 2004-06-22
Classification: C07C,C07D

Abstract:
A compound of formula I: wherein:A is selected from the group consisting of hydrogen; aryl; alkylheterocyclyl; alkenylaminopolycyclyl; alkenylaminoheterocyclyl; alkylaminopolycyclyl; carbonylaminopolycyclyl; where the aryl, heterocyclyl and polycyclyl moieties are optionally substituted with one or more of the following: halogen, cyano, nitro, amino, carboxyl, alkyl, haloalkyl, alkoxy, haloalkoxy, carbonyl, alkylcarbonyl, haloalkylcarbonyl, alkoxycarbonyl, haloalkoxycarbonyl, or aryl; and Formula III, where Formula III is â€”(CH2)nâ€”Uâ€”R2â€ƒâ€ƒIII wherein n is 0 or 1; U is selected from the group consisting of â€”CH2â€”, â€”Oâ€”CH2â€”, oxygen, sulfur, sulfonyl, alkyl, oxyalkyloxy, alkenylamino, cabonylamino and â€”NR5, where R5 is selected from the group consisting of hydrogen, hydroxy, alkyl, haloalkyl, sulfonylalkyl, cabonylamino, and carbonylalkyl; R2 is selected from aryl; alkylpolycyclyl; heterocyclyl; polycyclyl; where the aryl, heterocyclyl and polycyclyl moieties are optionally substituted with one or more of the following: halogen, cyano, nitro, amino, carboxyl, alkyl, haloalkyl, alkoxy, haloalkoxy, carbonyl, alkylcarbonyl, haloalkylcarbonyl, alkoxycarbonyl, haloalkoxycarbonyl, or aryl; 1-R3; 1-R4; and 2-R4, wherein: R3 is â€ƒwhere J, L, and W are independently selected from the group consisting of hydrogen, halogen, cyano, nitro, amino, carboxyl, alkyl, haloalkyl, alkenyl, alkoxy, haloalkoxy, aminoalkoxy, nitrilyl, carbonyl, alkylcarbonyl, haloalkylcarbonyl, alkoxycarbonyl, haloalkoxycarbonyl, aryl, aryloxy, and heterocyclyl, where the aryl and heterocyclyl moieties may be optionally substituted with halogen, alkyl, haloalkyl, alkoxy, or haloalkoxy; R4 is â€ƒwhere X, Y, and Z are independently selected from the group consisting of hydrogen, halogen, cyano, nitro, amino, azido, carboxyl, alkyl, alkynyl, haloalkyl, haloalkylthio, nitrilyl, alkenyl, alkoxy, haloalkoxy, carbonyl, alkylcarbonyl, haloalkylcarbonyl, alkoxycarbonyl, haloalkoxycarbonyl, phenyl, aryl, aryloxy, and heterocyclyl, where the phenyl, aryl, and heterocyclyl moieties may be optionally substituted with halogen, haloalkyl, haloalkyl, alkoxy, or haloalkoxy; with the proviso that X, Y and Z cannot all be hydrogen; B and D are independently selected from hydrogen, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, alkoxyaminoalkyl, 2-(Formula III), 3-(Formula III), 5-(Formula III), and 6-(Formula III), wherein Formula III, n, U, R2, R3, R4, R5, J, L, W, X, Y, and Z are as defined above; R is â€”Tâ€”(CH2)mâ€”R1, â€”N(R6)(R7) or heterocyclyl, where the heterocyclyl moiety may be optionally substituted with halogen, hydroxy, alkyl, haloalkyl, alkoxy, haloalkoxy, alkoxycarbonyl, aryl, alkylaza, arylcarbonyl, benzyl, allyl, propargyl, alkylamino; where the aryl moiety may be optionally substituted with halogen, hydroxy, alkyl, haloalkyl, alkoxy, haloalkoxy, alkoxycarbonyl, aryl, arylcarbonyl; T is selected from the group consisting of â€”CH2â€”, carbonyl, oxygen, nitrogen, and sulfur; m is 0, 1, 2, 3, or 4; R1 is selected from the group consisting of â€”N(R8)(R9); aryl; â€”C(O)N(R12)(R13); oxyalkyl; haloalkyl; heterocyclyl; cycloalkyl; â€”N(O)(R14)(R15); â€”P(O)(R14)(R15); â€”P(S)(R14)(R15); alkylamino, where the cycloalkyl, aryl and heterocyclyl moieties may be optionally substituted with halogen, hydroxy, alkyl, haloalkyl, alkoxy, haloalkoxy, alkoxycarbonyl, aryl, arylcarbonyl, alkylamino; where R6, R7, R8, R9, R12, R13, R14, and R15 are independently selected from the group consisting of hydrogen, alkyl, alkoxy, alkylthio, acetyl, alkoxycarbonyl, alkoxyalkyl, aminoalkyl, carbonylamino, and â€”(CH2)pâ€”N(R16)(R17), where p is 1 or 2; R16 and R17 are independently selected from the group consisting of hydrogen, alkyl, alkoxy, alkoxyalkyl, and aminoalkyl; with the provisos that (i) when A, B and D are hydrogen, R is other than heterocyclyl; (ii) when A, B, and D are hydrogen, R is â€”Tâ€”(CH2)mâ€”R1, T is oxygen, m is 2, R1 is â€”N(R8)(R9), and R8 is hydrogen, R9 is other than hydrogen; and (iii) when B and D are hydrogen, A is â€”(CH2)nâ€”Uâ€”R2, R is â€”Tâ€”(CH2)mâ€”R1, T is oxygen, U is oxygen, m is 2, n is 1, R1 is â€”N(R8)(R9), R2 is 1-R3, J, L, W, are hydrogen; and R8 is alkyl, R9 is other than the same alkyl;and the corresponding agriculturally acceptable salts thereof.