Patent ID: 6537989
Filing Date: 2003-03-25
Classification: A01N,A61P,C07D

Abstract:
An azadioxacycloalkene of the formula I, in which the substituents R1 to R5 and X, the index n and the bridge member W have the following meanings:R1 is C1-C4-alkyl, halogen, cyano, C1-C4-haloalkyl or C3-C6-cycloalkyl; R2 is C1-C4-alkyl, C1-C4-haloalkyl, C3-C4-alkenyl, C3-C4-haloalkenyl, C3-C4-alkynyl or C3-C4-haloalkynyl; R3 is hydrogen, C1-C4-alkyl, C1-C4-haloalkyl or unsubstituted or substituted phenyl; R4 is &boxH;CRaRb, CRd&boxH;CRaRb or &boxH;Nâ€”ORc, where Ra, Rb, Rd independently of one another are each hydrogen, halogen, C1-C6-alkyl, C1-C4-haloalkyl or unsubstituted or substituted phenyl and Rc is one of the radicals mentioned under R2; R5 is nitro, cyano, halogen, C1-C6-alkyl or in the case that n is greater than 1, is additionally a bridge which is attached to two adjacent ring atoms and which contains three or four members selected from the group: 3 or 4 carbon atoms, 2 or 3 carbon atoms and 1 or 2 nitrogen atoms, oxygen atoms and/or sulfur atoms, where this bridge, together with the ring to which it is attached, may form a partially unsaturated or aromatic radical and where furthermore the carbon atoms of the bridge may be partly or fully substituted by halogen atoms or methyl groups; n is 0, 1, 2, 3 or 4, where the substituents R5 may be different if n is greater than 1; X is C1-C4-alkoxy-N&boxH;, C1-C4-alkoxy-CH&boxH; or R6â€”CH&boxH;, where R6 is halogen, C1-C4-alkyl, C1-C4-alkylthio, C1-C4-alkylamino or di-C1-C4-alkylamino and W is C1-C3-alkylene which is unsubstituted or mono- or disubstituted by R7, where R7 is halogen, cyano, C1-C4-alkyl, C1-C4-haloalkyl, C2-C4-alkenyl, C2-C4-haloalkenyl, C2-C4-alkynyl, C2-C4-haloalkynyl, C1-C4-alkoxy, C1-C4-haloalkoxy, C2-C4-alkenoxy, C2-C4-haloalkenoxy, C2-C4-alkynoxy, C2-C4-haloalkynoxy or C1-C4-alkylcarbonyloxy.