Patent ID: 7812041
Filing Date: 2010-10-12
Classification: A61P,C07D

Abstract:
1. A compound of the general formula (III) or a salt, or a stereoisomer thereof, wherein R R R R R wherein R R R R R A is CO or SO X is NR Z is N or CR R p is 1 to 6; q is 1 to 6; r is 0, or 1; R R wherein an alkyl group, if not stated otherwise, denotes a linear or branched C a heterocycle denotes a heterocycloalkyl group or a heteroaryl group; a cycloalkyl group denotes a non-aromatic ring system containing three to eight carbon atoms, one or more of the carbon atoms in the ring can be substituted by a group R a heterocycloalkyl group denotes a non-aromatic ring system containing two to ten carbon atoms and at least one heteroatom O, N, or S, wherein one or more of the carbon atoms in the ring can be substituted by R an alkoxy group denotes an O-alkyl group, the alkyl group being as defined above; an alkylthio group denotes an S-alkyl group, the alkyl group being as defined above; a haloalkyl group denotes an alkyl group which is substituted by one to five halogen atoms, the alkyl group being as defined above; a hydroxyalkyl group denotes an HO-alkyl group, the alkyl group being as defined above; a haloalkyloxy group denotes an alkoxy group which is substituted by one to five halogen atoms, the alkyl group being as defined above; a hydroxyalkylamino group denotes an (HO-alkyl) an alkylamino group denotes an HN-alkyl or N-dialkyl group, the alkyl group being as defined above; a halogen group is fluorine, chlorine, bromine, or iodine; an aryl group denotes an aromatic group having five to fifteen carbon atoms, which can be substituted by one or more substituents R a heteroaryl group denotes a 5- to 10-membered aromatic heterocyclic group which contains at least one heteroatom O, N, S, wherein the heterocyclic group may be fused to another ring, and the heterocyclic group or the fused ring can both be substituted independently by one or more substituents R an alkylaryl or arylalkyl group denotes an alkyl group as defined above, which is bound to an aryl fragment as defined above via a single bond, wherein the linkage to the central moiety occurs through the alkyl part or the aryl part.