Patent ID: 8703720
Filing Date: 2014-04-22
Classification: A61P,C07H

Abstract:
1. A compound of the general formula (I): wherein the configuration of the pyranose ring is D-galacto; X is selected from the group consisting of O, S, and SO; Y and Z are independently selected from being CONH or a 1 H- 1,2,3-triazole ring; R 1 and R 2 are independently selected from the group consisting of: a) an alkyl group of at least 4 carbons, an alkenyl group of at least 4 carbons, an alkynyl group of at least 4 carbons; b) a carbamoyl group, a carbamoyi group substituted with an alkyl group, a carbamoyi group substituted with an aikenyl group, a carbamoyl group substituted with an alkynyl group, a carbamoyl group substituted with an aryl group, a carbamoyl group substituted with an substituted alkyl group, and a carbamoyl group substituted with an substituted aryl group; c) a phenyl group substituted with at least one carboxy group, a phenyl group substituted with at least one halogen, a phenyl group substituted with at least one alkyl group, a phenyl group substituted with at least one alkoxy group, a phenyl group substituted with at least one trifluoromethyl group, a phenyl group substituted with at least one trifluoromethoxy group, a phenyl group substituted with at least one sulfo group, a phenyl group substituted with at least one hydroxy group, a phenyl group substituted with at least one carbonyl group, and a phenyl group substituted with at least one substituted carbonyi group; d) a naphthyl group, a naphthyl group substituted with at least one carboxy group, a naphthyl group substituted with at least one halogen, a naphthyl group substituted with at least one alkyl group, a naphthyl group substituted with at least one alkoxy group, a naphthyl group substituted with at least one sulfo group, a naphthyl group substituted with at least one hydroxyl group, a naphthyl group substituted with at least one carbonyl group, and a naphthyi group substituted with at least one substituted carbonyl group; e) a heteroaryl group comprising 4 to 18 carbon atoms, and at least one heteroatom selected from N, O and S, wherein the heteroaryl group may be substituted with at least one group selected from a carboxy group, a halogen, an alkoxy group, a sulfo group, an arylamino group, a hydroxyl group, a carbonyl group, and a substituted carbonyl group; and f) a thienyl group, a thienyl group substituted with at least one carboxy group, a thienyl group substituted with at least one halogen, a thienyl thienyl group substituted with at least one alkoxy group, a thienyl group substituted with at least one sulfo group, a thienyl group substituted with at least one arylamino group, a thienyl group substituted with at least one hydroxy group, a thienyl group substituted with at least one halogen, a thienyl group substituted with at least one carbonyl group, and a thienyl group substituted with at least one substituted carbonyl group.