Patent ID: 6638940
Filing Date: 2003-10-28
Classification: A01N,C07D

Abstract:
Compound of formula whereinR1 and R2, independently of one another, are halogen, C1-C6-alkyl, C3-C6-cycloalkyl, halogen-C1-C6-alkyl, halogen-C3-C6-cycloalkyl, C2-C4-alkenyl, C2-C4-alkinyl, halogen-C2-C4-alkenyl, halogen-C2-C4-alkinyl, C1-C6-alkoxy, halogen-C1-C6-alkoxy, C2-C6-alkenyloxy, C2-C6-alkinyloxy, halogen-C2-C6-alkenyloxy, halogen-C2-C6-alkinyloxy, â€”SF5, â€”C(&boxH;O)N(R5)2, â€”Oâ€”C(&boxH;O)N(R5)2, â€”CN, â€”NO2, â€”S(&boxH;O)2N(R5)2, â€”S(&boxH;O)pâ€”C1-C6-alkyl, â€”S(&boxH;O)p-halogen-C1-C6-alkyl, â€”Oâ€”S(&boxH;O)pâ€”C1-C6-alkyl, â€”Oâ€”S(&boxH;O)p-halogen-C1-C6-alkyl, phenyl, benzyl, phenoxy or benzyloxy, wherein each of the phenyl, benzyl, phenoxy or benzyloxy radicals is either unsubstituted or mono- to penta-substituted in the aromatic ring, independently of each other, by substituents selected from the group consisting of halogen, cyano, NO2, C1-C6-alkyl, halogen-C1-C6-alkyl, C1-C6-alkoxy and halogen-C1-C6-alkoxy; R3 is hydrogen, OH, halogen, C1-C6-alkoxy, or â€”Oâ€”C(&boxH;O)â€”C1-C6-alkyl; R4 is phenyl, which is mono- to penta-substituted, independently of each other, by substituents selected from the group consisting of halogen, cyano, NO2, C1-C6-alkyl, C3-C8-cycloalkyl, C3-C8-cycloalkyl-C1-C6-alkyl, halogen-C1-C6-alkyl, C1-C6-alkoxy, C3-C8-cycloalkoxy, C3-C8-cycloalkoxy-C1-C6-alkyl, C3-C8-cycloalkyl-C1-C6-alkoxy, halogen-C1-C6-alkoxy, C2-C4-alkenyl, C2-C4-alkinyl, C2-C6-alkenyloxy, C2-C6-alkinyloxy, â€”NR6â€”C(&boxH;O)â€”Oâ€”C1-C6-alkyl, â€”NR6â€”C(&boxH;O)â€”O-halogen-C1-C6-alkyl, â€”C(R7)&boxH;Nâ€”Wâ€”R8, the two R5 independently of one another, are hydrogen or C1-C6-alkyl; R6 is hydrogen, C1-C6-alkyl or benzyl; R7 is halogen, C1-C6-alkyl, C3-C8-cycloalkyl, C3-C8-cycloalkyl-C1-C6-alkyl, halogen-C1-C6-alkyl, C1-C6-alkoxy, C3-C8-cycloalkoxy, C3-C8-cycloalkoxy-C1-C6-alkyl, halogen-C1-C6-alkoxy, â€”NH(C1-C6-alkyl) or â€”N(C1-C6-alkyl)2; R8 is hydrogen, C1-C6-alkyl, C3-C8-cycloalkyl, C3-C8-cycloalkyl-C1-C6-alkyl, halogen-C1-C6-alkyl or â€”C(&boxH;O)â€”C1-C6-alkyl; m is 0, 1, 2, 3, 4 or 5; n is 0, 1, 2, 3, 4 or 5; p is 0, 1 or 2; q is 0 or 1 W is O or NH or Nâ€”C1-C6-alkyl; and, the E/Z isomers, E/Z isomeric mixtures and/or tautomers thereof, each in free form or in salt form.