Patent ID: 8476194
Filing Date: 2013-07-02
Classification: A01N,A61P,C07C

Abstract:
1. A compound of Formula 1: wherein at least one X3-X6 is not H; X3, X4, X5, and X6 are independently H, halogen, nitro, CN, C1-C4 alkyl, C1-C4 alkoxy, or C1-C4 haloalkoxy; R is C1-C4 alkyl, C2-C4 alkenyl, C2-C4 alkynyl, C3-C6 cycloalkyl, C1-C4 haloalkyl, C2-C4 haloalkenyl, C2-C4 haloalkynyl, or C3-C6 halocycloalkyl; and Y2, Y3, Y4, Y5, and Y6 are independently selected from the group consisting of H, halogen, nitro, hydroxyl, cyano, C1-C4 alkyl, C1-C4 alkoxy, C2-C4 alkenyl, C2-C4 alkynyl, C1-C4 alkylthio, C1-C4 haloalkyl, C1-C4 haloalkoxy, C2-C4 haloalkenyl, C2-C4 haloalkynyl, C1-C4 haloalkylthio, —SO R1 is H, C1-C4 alkyl, C2-C4 alkenyl, C2-C4 alkynyl, C1-C4 haloalkyl, C2-C4 haloalkenyl, C2-C4 haloalkynyl,; with the proviso that: if R is CH3 and X4 is CH3, then X3, X5, and X6 are not all H; if R is CH3, and X3, X4 and X6 are H then X5 is not CH3; if R and X4 are CH3, and if X3, X5, and X6 are H, then Y2, Y3 and Y4 are not CH3; if R is CH3CH2 and if X5 is F and X3, X4, X5, X6, Y2, Y3, Y5, and Y6 are H, then Y4 is not F; if X3 and X5 are Br, Y2, Y3, Y4, Y5, Y6 are not all H; if X3 and X5 are Br and X4, X6, Y2, Y3, Y5, and Y6 are H, Y4 is not —NO2, or H; if X3 and X5 are Br, R is CH3, X4, X6, Y2, Y5, and Y6 are H, Y3 and Y4 are not OCH3; if X5 is Br, CI, CH3, or MeO, R is CH3, and X3, X4, X6, Y2, Y3, Y5, and Y6 are H, Y4 is not CI, H, CH3, NO2, MeO, or OH; if X4 is F or MeO, R is CH3, X3, X5, X6, Y2, Y3, Y5, Y6, are H, Y4 is not —NO2, CH3, MeO, or H; if X3 is Br, R, X4 and X5 are CH3, and X6, Y3, Y4, Y5, and Y6 are not H, Y2 is not —OH; if X5 is CI, R is CF3 or CH3, X3, X4, X6, Y3, Y4, Y5, and Y6 are H, Y2 is not —OH; if X4, X5, and R are CH3, and X3, X6, Y3, Y4, Y5, and Y6 are H, Y2 is not hydroxyl; if X3 is Br, R, X4, and X5 are CH3, and X6, Y3, Y4, Y5, and Y6 are H, Y2 is not hydroxyl; if X3 and X5 are CI, and X4, X6, Y2, Y3, Y4, Y5, and Y6 are not all H, R is not CH3 or CH2CH3; if X3 and R are CH3, and X4, X5, X6, Y5, Y6 are H, then independently of one another Y2, Y3 and Y4 are not NO2; if X5 is CI, and X4 and R are CH3 and X3, X6, Y2, Y3, and Y5 are H, then Y4 is not NO2; if X5 is CI and X3, X4, X6, Y2, Y3, Y4, Y5, and Y6 are H, R is not CH3; if X5 and R are CH3, X2, X3, X4, X6, Y2, Y4, Y5, Y6 are H, then Y3 is not NO2, CH3, or —OH; if X5 and R are CH3, X2, X3, X4, X6, Y3, Y4, Y5, Y6 are H, then Y2 is not NO2, CH3, or —OH; if X5 is CH3, R is isopropyl, X2, X3, X4, X6, Y3, Y4, Y5, Y6 are H, then Y2 is not —OH; if X3 and R are CH3, X2, X3, X4, X6, Y3, Y4, Y5, Y6 are H, then Y2 is not —OH and if X5 is F, and X3, X4, X6, Y2, Y3, Y4, Y5, and Y6 are not H, R is not CH3, CH2CH3, or CH2CH2CH3.