Patent ID: 9216992
Filing Date: 2015-12-22
Classification: C07D

Abstract:
1. A compound of the formula: wherein: R1 is unsubstituted or substituted aryl, wherein the substituents are selected from the group consisting of cyano, halogen, nitro, trifluoromethyl, unsubstituted alkyl, alkylthio, alkoxy, NR9R10, CO R2 is H or unsubstituted or substituted alkyl, wherein the substituents are selected from the group consisting of halogen, cyano, nitro, NR9R10, alkoxy, hydroxyl, unsubstituted aryl, unsubstituted heteroaryl, aryloxy, heteroaryloxy, CO R3 is unsubstituted or substituted alkyl, wherein the substituents are selected from the group consisting of halogen, cyano, nitro, NR9R10, alkoxy, hydroxyl, unsubstituted aryl, unsubstituted heteroaryl, aryloxy, heteroaryloxy, CO R4 is H; unsubstituted or substituted alkyl, wherein the substituents are selected from the group consisting of halogen, cyano, nitro, NR9R10, alkoxy, hydroxyl, unsubstituted aryl, unsubstituted heteroaryl, aryloxy, heteroaryloxy, CO R5 and R6 may be the same or different, and may be H; unsubstituted or substituted alkyl, wherein the substituents are selected from the group consisting of halogen, cyano, nitro, alkoxy, hydroxyl, unsubstituted aryl, unsubstituted heteroaryl, aryloxy, and heteroaryloxy; unsubstituted or substituted aryl, wherein the substituents are selected from the group consisting of cyano, halogen, nitro, trifluoromethyl, unsubstituted alkyl, alkylthio, alkoxy, NR9R10, CO R7 is H; unsubstituted or substituted alkyl, wherein the substituents are selected from the group consisting of halogen, cyano, nitro, alkoxy, hydroxyl, unsubstituted aryl, unsubstituted heteroaryl, aryloxy, and heteroaryloxy; unsubstituted or substituted aryl, wherein the substituents are selected from the group consisting of cyano, halogen, nitro, trifluoromethyl, unsubstituted alkyl, alkylthio, and alkoxy; unsubstituted or substituted heteroaryl, wherein the substituents are selected from the group consisting of cyano, nitro, halogen, unsubstituted alkyl, alkylthio, and alkoxy; or unsubstituted cycloalkyl; X is NR8; R8 is H; L is (CH Y is unsubstituted or substituted aryl, wherein the substituents are selected from the group consisting of cyano, halogen, nitro, trifluoromethyl, unsubstituted alkyl, alkylthio, alkoxy, NR9R10, CO R9 and R10 can be the same or different, and may be H, unsubstituted alkyl, unsubstituted aryl, unsubstituted heteroaryl, unsubstituted cycloalkyl, aminoethyl, methylaminoethyl, dimethylaminoethyl, hydroxyethyl, or alkoxyethyl, or R9 and R10 may together form a saturated or partially saturated 4 to 7 membered ring; or the products of oxidation of sulphur and/or nitrogen moieties on these molecules, or a pharmaceutically acceptable salt thereof.