Desymmetrization of <i>meso</i> -Anhydride Enabled Enantioselective Synthesis of (−)-7-(Bromomethylene)-3-amidobicyclo[2.2.1]heptane-2-carboxamide, a Scaffold for Divergent Drug Discovery Synthesis
Year: 2025
Type: article
Language: en
Topic: Advanced Synthetic Organic Chemistry
Authors and affiliations:
raw_author_name: Jianqing Li
raw_affiliation_strings: Bristol Myers Squibb Research and Early Development
Small Molecule Drug Discovery
Small Molecule Drug Discovery, Bristol Myers Squibb Research and Early Development, Cambridge, Massachusetts 02142, United States
raw_author_name: Subramaniam Krishnananthan
raw_affiliation_strings: Small Molecule Drug Discovery, Bristol Myers Squibb Research and Early Development, P.O. Box 4000, Princeton, New Jersey 08543-4000, United States
raw_author_name: Daniel Smith
raw_affiliation_strings: Small Molecule Drug Discovery, Bristol Myers Squibb Research and Early Development, P.O. Box 4000, Princeton, New Jersey 08543-4000, United States
raw_author_name: Chetan Padmakar Darne
raw_affiliation_strings: Bristol Myers Squibb Research and Early Development
Small Molecule Drug Discovery
Small Molecule Drug Discovery, Bristol Myers Squibb Research and Early Development, Cambridge, Massachusetts 02142, United States
raw_author_name: Ning Li
raw_affiliation_strings: Bristol Myers Squibb Research and Early Development
Small Molecule Drug Discovery
Small Molecule Drug Discovery, Bristol Myers Squibb Research and Early Development, Cambridge, Massachusetts 02142, United States
raw_author_name: Lyndon Cornelius
raw_affiliation_strings: Small Molecule Drug Discovery, Bristol Myers Squibb Research and Early Development, P.O. Box 4000, Princeton, New Jersey 08543-4000, United States
raw_author_name: Bei Wang
raw_affiliation_strings: Small Molecule Drug Discovery, Bristol Myers Squibb Research and Early Development, P.O. Box 4000, Princeton, New Jersey 08543-4000, United States
raw_author_name: Rulin Zhao
raw_affiliation_strings: Small Molecule Drug Discovery, Bristol Myers Squibb Research and Early Development, P.O. Box 4000, Princeton, New Jersey 08543-4000, United States
raw_author_name: Peng Li
raw_affiliation_strings: Small Molecule Drug Discovery, Bristol Myers Squibb Research and Early Development, P.O. Box 4000, Princeton, New Jersey 08543-4000, United States
raw_author_name: Dauh-Rurng Wu
raw_affiliation_strings: Small Molecule Drug Discovery, Bristol Myers Squibb Research and Early Development, P.O. Box 4000, Princeton, New Jersey 08543-4000, United States
raw_author_name: James Kempson
raw_affiliation_strings: Small Molecule Drug Discovery, Bristol Myers Squibb Research and Early Development, P.O. Box 4000, Princeton, New Jersey 08543-4000, United States
raw_author_name: Sarah C. Traeger
raw_affiliation_strings: Small Molecule Drug Discovery, Bristol Myers Squibb Research and Early Development, P.O. Box 4000, Princeton, New Jersey 08543-4000, United States
raw_author_name: Michael A. Galella
raw_affiliation_strings: Analytical Strategy & Operations
Bristol Myers Squibb Product Development
Analytical Strategy & Operations, Bristol Myers Squibb Product Development, New Brunswick, New Jersey 08901, United States
raw_author_name: Amy Sarjeant
raw_affiliation_strings: Bristol Myers Squibb
Drug Product Development
Drug Product Development, Bristol Myers Squibb, New Brunswick, New Jersey 08903, United States
raw_author_name: Shun Su
raw_affiliation_strings: Small Molecule Drug Discovery, Bristol Myers Squibb Research and Early Development, P.O. Box 4000, Princeton, New Jersey 08543-4000, United States
raw_author_name: Roshan Y. Nimje
raw_affiliation_strings: Biocon Bristol Myers Squibb R&D Center
Department of Chemical Synthesis
Department of Chemical Synthesis, Biocon Bristol Myers Squibb R&D Center, Bangalore 560099, India
raw_author_name: Yoganand Shanmugam
raw_affiliation_strings: Biocon Bristol Myers Squibb R&D Center
Department of Chemical Synthesis
Department of Chemical Synthesis, Biocon Bristol Myers Squibb R&D Center, Bangalore 560099, India
raw_author_name: Dyamanna Doddalingappa
raw_affiliation_strings: Biocon Bristol Myers Squibb R&D Center
Department of Chemical Synthesis
Department of Chemical Synthesis, Biocon Bristol Myers Squibb R&D Center, Bangalore 560099, India
raw_author_name: Rajesh Krishnan
raw_affiliation_strings: Biocon Bristol Myers Squibb R&D Center
Department of Chemical Synthesis
Department of Chemical Synthesis, Biocon Bristol Myers Squibb R&D Center, Bangalore 560099, India
raw_author_name: Anuradha Gupta
raw_affiliation_strings: Biocon Bristol Myers Squibb R&D Center
Department of Chemical Synthesis
Department of Chemical Synthesis, Biocon Bristol Myers Squibb R&D Center, Bangalore 560099, India
raw_author_name: Arvind Mathur
raw_affiliation_strings: Small Molecule Drug Discovery, Bristol Myers Squibb Research and Early Development, P.O. Box 4000, Princeton, New Jersey 08543-4000, United States