Design, green synthesis, X-ray characterization, in silico, and in vitro evaluation of novel sulfonylimine derivatives as acetyltransferase inhibitors
Year: 2025
Type: article
Language: en
Topic: Enzyme function and inhibition
Authors and affiliations:
raw_author_name: Meriem Boussaker
raw_affiliation_strings: Laboratory of Applied Organic Chemistry, Synthesis of Biomolecules and Molecular Modelling Group, Department of Chemistry, Faculty of Sciences, Badji-Mokhtar - Annaba University, Box 12, 23000 Annaba, Algeria
raw_author_name: Radia Bouasla
raw_affiliation_strings: Laboratory of Applied Organic Chemistry, Synthesis of Biomolecules and Molecular Modelling Group, Department of Chemistry, Faculty of Sciences, Badji-Mokhtar - Annaba University, Box 12, 23000 Annaba, Algeria
National Higher School of Technology and Engineering-Annaba, Box 218, 23000 Annaba Algeria
raw_author_name: Malika Berredjem
raw_affiliation_strings: Laboratory of Applied Organic Chemistry, Synthesis of Biomolecules and Molecular Modelling Group, Department of Chemistry, Faculty of Sciences, Badji-Mokhtar - Annaba University, Box 12, 23000 Annaba, Algeria
raw_author_name: Vipin Kumar Mishra
raw_affiliation_strings: Chemistry division, School of advanced sciences and languages, Bhopal, 440033, India
raw_author_name: Malika Ouali Ibrahim
raw_affiliation_strings: Aix Marseille Univ, CNRS, Centrale Marseille, iSm2, Marseille, France
raw_author_name: Khadidja Otmane Rachedi
raw_affiliation_strings: El-Tarf University, Faculty of Science and Technology, BP 73, El-Tarf, Algeria
Laboratory of Applied Organic Chemistry, Synthesis of Biomolecules and Molecular Modelling Group, Department of Chemistry, Faculty of Sciences, Badji-Mokhtar - Annaba University, Box 12, 23000 Annaba, Algeria
raw_author_name: Noureddine Dadda
raw_affiliation_strings: Laboratory of Synthesis and organic Biocatalysis, chemistry department, Sciences faculty, Badji Mokhtar Annaba University, Annaba, Box 12, 23000, Algeria
raw_author_name: Lina Manel Djendi
raw_affiliation_strings: Laboratory of Microbiology and Molecular Biology, Badji-Mokhtar- Annaba University, Box 12, 23000, Algeria
raw_author_name: Sara Grine
raw_affiliation_strings: Laboratory of Applied Organic Chemistry, Synthesis of Biomolecules and Molecular Modelling Group, Department of Chemistry, Faculty of Sciences, Badji-Mokhtar - Annaba University, Box 12, 23000 Annaba, Algeria
raw_author_name: Chahrazed Benzaid
raw_affiliation_strings: Laboratory of Microbiology and Molecular Biology, Badji-Mokhtar- Annaba University, Box 12, 23000, Algeria
raw_author_name: Yacine Laichi
raw_affiliation_strings: Centre de Recherche Scientifique et Technique en Analyses Physico-chimiques (CRAPC), BP384, Bou-Ismail, RP 42004, Tipasa, Algeria
raw_author_name: Khaldoune Bachari
raw_affiliation_strings: Centre de Recherche Scientifique et Technique en Analyses Physico-chimiques (CRAPC), BP384, Bou-Ismail, RP 42004, Tipasa, Algeria
raw_author_name: Christelle Marminon
raw_affiliation_strings: Small Molecules for Biological Targets Team, Centre de Recherche en Cancérologie de Lyon, Centre Léon Bérard, Institut National de la Santé et de la Recherche Médicale (INSERM) 1052, Centre National de la Recherche Scientifique (CNRS) 5286, Université Claude Bernard Lyon 1, 69373 Lyon, France
raw_author_name: Ismahene Grib
raw_affiliation_strings: Laboratory of Applied Organic Chemistry, Synthesis of Biomolecules and Molecular Modelling Group, Department of Chemistry, Faculty of Sciences, Badji-Mokhtar - Annaba University, Box 12, 23000 Annaba, Algeria