RU-57073

RU-57073

Section Title:
Table Section Text: None

Compound	AR	ER	PR	GR	MR

Metribolone	290	< 0.1	190	4	38

Dihydrotestosterone	180	ND	ND	ND	ND

Testosterone	100	ND	ND	ND	ND

Cyproterone acetate	10	ND	ND	ND	ND

Bicalutamide	1.8	ND	ND	ND	ND

Nilutamide	0.8	ND	ND	ND	ND

Hydroxyflutamide	0.8	ND	ND	ND	ND

RU-59063	300	<0.1	<0.1	<0.1	<0.1

RU-58841	150	ND	ND	ND	ND

RU-58642	46	<0.1	<0.1	<0.1	<0.1

RU-57073	163	<0.1	<0.1	<0.1	<0.1

RU-56187	92	<0.1	<0.1	<0.1	<0.1

Notes: Values are RBAs (%). Reference ligands (100%) were testosterone for the AR, estradiol for the ERα and ERβ, progesterone for the PR, dexamethasone for the GR, and aldosterone for the MR.

Sentence(s)

RU-57073 shows 163 for the androgen receptor and negligible for other receptors.

final_sentence: RU-57073 shows 163 for the androgen receptor and negligible for other receptors.