Patent ID: 9243010
Filing Date: 2016-01-26
CPC Classification: C07C,C07D,C07F

Claim Text:
1. A process for the preparation of the compound which comprises: (a) reacting the compound 1 with the acid chloride compound to form the compound 2 and then (b) contacting the compound 2 with a di-substituted amine (R and thereafter (c) reacting the compound 3 with the dihydroxy compound HO—C and (d) reacting the compound 4 with the compound in acid to produce the compound 5 (e) contacting the compound 5 with Me-X and then (f) performing an oxidation reaction on compound 6 to yield the compound 7 and (g) performing an activation reaction to yield the resultant compound 10 and then (h) adding the triazolyl group 9  to compound 10 in the presence of Cu and a ligand to yield the compound of Formula (I) above wherein: and also wherein said ligand is selected from the group consisting of 1,2-diaminocyclohexane, trans-1,2-diaminocyclohexane, cis-/trans-diaminocyclohexane, cis-N,N′-dimethyl-1,2-diaminocyclohexane, trans-N,N′-dimethyl-1,2-diaminocyclohexane, cis-/trans-N,N′-dimethyl-1,2-diaminocyclohexane, 1,2-diaminoethane, N,N′-dimethyl-1,2-diaminoethane, 1,10-phenanthroline, 4,7-diphenyl-1,10-phenantroline, 5-methyl-1,10-phenanthroline, 5-chloro-1,10-phenantroline, and 5-nitro-1,10-phenanthroline.