Patent ID: 9487529
Filing Date: 2016-11-08
CPC Classification: A61K,C07D

Claim Text:
1. A compound of Formula I wherein: A is H, cyano, F, Cl, Br, CH R1 is H, heterocyclyl, heteroaryl, carbocyclyl, aryl, C where, when R1 is a nitrogen containing heterocyclyl, the nitrogen may be substituted with C and where, when R1 is heterocyclyl, heteroaryl, carbocyclyl, or aryl, such heterocyclyl, heteroaryl, carbocyclyl, or aryl may be unsubstituted, or substituted with one or two substituents independently selected from the group consisting of C and where, when R1 is C R2 is H, heterocyclyl, heteroaryl, carbocyclyl, aryl, C where, when R2 is a nitrogen containing heterocyclyl, the nitrogen may be substituted with H, C and where, when R2 is heterocyclyl, heteroaryl, carbocyclyl, or aryl, such heterocyclyl, heteroaryl, carbocyclyl, or aryl may be unsubstituted, or substituted with one or two substituents independently selected from the group consisting of C and where, when R2 is C R1 and R2, together with the phenyl ring to which they are attached, form a five- to eight-membered monocarbocyclic or monoheterocyclic ring, where the ring so formed by R1 and R2, may be unsubstituted, or substituted with one to three substituents independently selected from the group consisting of C R3 is H, C where at least one of R1 and R3 is other than H; R4 and R5, independently, are H, C and where, when R4 or R5 is N-(C R4 and R5, together with the phenyl ring to which the are attached, form a five- to eight-membered monoheterocyclic ring, where the ring so-formed by R4 and R5 may be unsubstituted, or substituted with one or two substituents independently selected from the group consisting of C —X— is —CH═CH—, —CH a pharmaceutically acceptable salt thereof.