Patent ID: 9242933
Filing Date: 2016-01-26
CPC Classification: A61P,C07D

Claim Text:
1. A compound of formula I wherein X is selected from the group consisting of O, S, S(O), S(O) R C phenyl, 5- or 6-membered hetaryl having 1, 2 or 3 heteroatoms as ring members, the heteroatoms being selected from the group consisting of O, S, and N, wherein hetaryl and phenyl are unsubstituted or carry 1, 2, 3, 4 or 5 identical or different radicals R C(═O)—R R C phenyl, and 5- or 6-membered hetaryl having 1, 2 or 3 heteroatoms as ring members, the heteroatoms being selected from the group consisting of O, S, and N, wherein phenyl and hetaryl are unsubstituted or may carry a fused benzene ring and/or 1, 2, 3, 4 or 5 identical or different radicals R R R R C R C R R R Y is a chemical bond; A is CR Ar is phenyl; R R C R C 3 -C 8 -cycloalkyl, which is unsubstituted or carries 1, 2, 3 or 4 radicals selected from the group consisting of halogen, C 1 -C 4 -alkyl, and C 1 -C 4 -alkoxy; R C C C C C phenyl, which is unsubstituted or carries 1, 2, 3, 4 or 5 identical or different radicals R 5- or 6-membered hetaryl having 1, 2 or 3 heteroatoms as ring members, the heteroatoms being selected from the group consisting of O, S, and N, wherein hetaryl is unsubstituted or carries 1, 2, 3 or 4 identical or different radicals R R R R R C phenyl or benzyl, wherein the phenyl ring in the last two radicals itself is unsubstituted or carries 1, 2, 3, 4 or 5 identical or different radicals selected from the group consisting of halogen, CN, OH, C C Het is pyrazolyl, wherein Het is unsubstituted or may carry a first substituent R R C C C C C C C C C(═O)—R phenyl, O-phenyl, CH 5- or 6-membered heteroaryl, having 1, 2, or 3 heteroatoms as ring members, the heteroatoms being selected from the group consisting of O, S, and N, which is unsubstituted or may carry 1, 2, 3, 4 or 5 substituents selected from the group consisting of halogen, CN, OH, C R R R R C C C phenyl, and 5- or 6-membered hetaryl having 1, 2 or 3 heteroatoms as ring members, the heteroatoms being selected from the group consisting of O, S, and N, wherein phenyl and hetaryl are unsubstituted or carry 1, 2, 3, 4 or 5 identical or different radicals R R R R R R R R C C phenyl, and 5- or 6-membered hetaryl having 1, 2 or 3 heteroatoms as ring members, the heteroatoms being selected from the group consisting of O, S, and N, wherein phenyl and hetaryl are unsubstituted or carry 1, 2, 3, 4, or 5 identical or different radicals R