Patent ID: 11958839
Assignee: GOLGI NEUROSCIENCES, S.R.L.
Field: Organic fine chemistry (Chemistry)
Classification: CPC C | IPC C

Claim 23:
24. The method as recited in claim 1, wherein:
n is a number between 1 and 4, forming a 6-10-membered cycloalkyl;
A is 3-methylthiophene;
R1 is chosen from hydrogen and methyl;
R2 and R3 are independently hydrogen, methyl, ethyl, and phenyl; or R2 and R3 are joined together via a group Y, wherein R2—Y—R3, together with the carbon to which R2 and R3 attach, forms C3-C6 cycloalkyl or C3-C6 heterocycloalkyl chosen from cyclopropyl, cyclobutyl, cyclopentyl, cyclohexyl, furan-3-yl, pyran-3-yl, and pyran-4-yl, any of which is optionally substituted with one or more substituents chosen from hydroxyl, fluorine, and methyl; or the C3-C6 cycloalkyl or C3-C6 heterocycloalkyl is fused with a phenyl ring which is optionally substituted with one or more substituents chosen from hydroxyl, halogen, and C1-C6 alkyl;
Y is chosen from C and O;
R4 is chosen from, R5 and R6 are independently C1-C3 alkyl;
R7, R8, R9, and R10 are independently chosen from hydrogen, hydroxyl, methyl, and C1-C3 alkyloxy, optionally substituted with methoxy;
p is 1 or 2; and
X is chosen from C, O, and NR11; and
R11 is C1-C3 alkyl.